| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 12 | 3 | 1 | 0 |
| Binding ≤ 1μM | 12 | 3 | 1 | 0 |
| ADME/T ≤ 10μM | 6 | 2 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_198585 | Highly calcium permeable nicotinic acetylcholine receptors | Mus musculus |
| REACT_198583 | Highly calcium permeable postsynaptic nicotinic acetylcholine receptors | Mus musculus |
| REACT_198593 | Highly sodium permeable acetylcholine nicotinic receptors | Mus musculus |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| ACHA3_MOUSE | Q8R4G9 | CHEMBL1255158 | Neuronal Acetylcholine Receptor Subunit Alpha-3, Mouse | 6 |
| ACHA4_MOUSE | O70174 | CHEMBL4457 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Mouse | 8 |
| ACHA6_MOUSE | Q9R0W9 | CHEMBL6183 | Neuronal Acetylcholine Receptor Subunit Alpha-6, Mouse | 12 |
| ACHB3_MOUSE | Q8BMN3 | CHEMBL1781863 | Neuronal Acetylcholine Receptor Subunit Beta-3, Mouse | 8 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| ACHA3_MOUSE | Q8R4G9 | CHEMBL1255158 | Neuronal Acetylcholine Receptor Subunit Alpha-3, Mouse | 6 |
| ACHA4_MOUSE | O70174 | CHEMBL4457 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Mouse | 8 |
| ACHA6_MOUSE | Q9R0W9 | CHEMBL6183 | Neuronal Acetylcholine Receptor Subunit Alpha-6, Mouse | 12 |
| ACHA7_MOUSE | P49582 | CHEMBL3365 | Neuronal Acetylcholine Receptor Protein Alpha-7 Subunit, Mouse | 12 |
| ACHB3_MOUSE | Q8BMN3 | CHEMBL1781863 | Neuronal Acetylcholine Receptor Subunit Beta-3, Mouse | 8 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| ACHA3_MOUSE | Q8R4G9 | CHEMBL1255158 | Neuronal Acetylcholine Receptor Subunit Alpha-3, Mouse | 6 |
| ACHA4_MOUSE | O70174 | CHEMBL4457 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Mouse | 8 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| ACHB4_HUMAN | P30926 | CHEMBL3002 | Neuronal Acetylcholine Receptor Protein Beta-4 Subunit, Human | 43 | 8 | 6 | 5 |
| ACHB4_RAT | P12392 | CHEMBL2658 | Neuronal Acetylcholine Receptor Protein Beta-4 Subunit, Rat | 370 | 59 | 16 | 5 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| ACHB3_MOUSE | Q8BMN3 | CHEMBL1781863 | Neuronal Acetylcholine Receptor Subunit Beta-3, Mouse | 8 | 3 | 1 | 0 |
| ACHB_MOUSE | P09690 | CHEMBL2690 | Acetylcholine Receptor Protein Beta Chain, Mouse | 1 | 0 | 1 | 1 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| ACHB4-1-E | Neuronal Acetylcholine Receptor Subunit Beta-4 (cluster #1 Of 7), Eukaryotic | 98 | 14 | 1 | 0 |
| ACHB4-2-E | Neuronal Acetylcholine Receptor Subunit Beta-4 (cluster #2 Of 7), Eukaryotic | 51 | 7 | 8 | 2 |
| ACHB4-3-E | Neuronal Acetylcholine Receptor Subunit Beta-4 (cluster #3 Of 7), Eukaryotic | 84 | 6 | 0 | 1 |
| ACHB4-4-E | Neuronal Acetylcholine Receptor Subunit Beta-4 (cluster #4 Of 7), Eukaryotic | 2 | 2 | 2 | 2 |
| ACHB4-5-E | Neuronal Acetylcholine Receptor Subunit Beta-4 (cluster #5 Of 7), Eukaryotic | 153 | 30 | 6 | 3 |
| ACHB4-6-E | Neuronal Acetylcholine Receptor Subunit Beta-4 (cluster #6 Of 7), Eukaryotic | 21 | 8 | 3 | 0 |
| ACHB4-7-E | Neuronal Acetylcholine Receptor Subunit Beta-4 (cluster #7 Of 7), Eukaryotic | 1 | 1 | 1 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| ACHA6_MOUSE | Q9R0W9 | CHEMBL6183 | Neuronal Acetylcholine Receptor Subunit Alpha-6, Mouse | 12 |
| ACHA7_MOUSE | P49582 | CHEMBL3365 | Neuronal Acetylcholine Receptor Protein Alpha-7 Subunit, Mouse | 12 |
| Q8BGP7_MOUSE | Q8BGP7 | CHEMBL2235 | Neuronal Acetylcholine Receptor Protein Beta-2 Subunit, Mouse | 12 |
| ACHA4_MOUSE | O70174 | CHEMBL4457 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Mouse | 8 |
| ACHB3_MOUSE | Q8BMN3 | CHEMBL1781863 | Neuronal Acetylcholine Receptor Subunit Beta-3, Mouse | 8 |
| ACHA3_MOUSE | Q8R4G9 | CHEMBL1255158 | Neuronal Acetylcholine Receptor Subunit Alpha-3, Mouse | 6 |
| Z104283 | Z104283 | CHEMBL1907589 | Neuronal Acetylcholine Receptor; Alpha4/beta2 | 2 |
| Z104290 | Z104290 | CHEMBL1907596 | Neuronal Acetylcholine Receptor; Alpha4/beta2 | 1 |