| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 1 | 0 | 0 | 0 |
| Binding ≤ 1μM | 0 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_15344 | Chemokine receptors bind chemokines | Homo sapiens |
| REACT_19231 | G alpha (i) signalling events | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| CCR4_HUMAN | P51679 | CHEMBL2414 | C-C Chemokine Receptor Type 4, Human | 1 |
| CCR5_HUMAN | P51681 | CHEMBL274 | C-C Chemokine Receptor Type 5, Human | 1 |
| CCR7_HUMAN | P32248 | CHEMBL4594 | C-C Chemokine Receptor Type 7, Human | 1 |
| CXCR2_HUMAN | P25025 | CHEMBL2434 | Interleukin-8 Receptor B, Human | 1 |
| CXCR4_HUMAN | P61073 | CHEMBL2107 | C-X-C Chemokine Receptor Type 4, Human | 1 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| CCR4_HUMAN | P51679 | CHEMBL2414 | C-C Chemokine Receptor Type 4, Human | 1 |
| CCR5_HUMAN | P51681 | CHEMBL274 | C-C Chemokine Receptor Type 5, Human | 1 |
| CCR7_HUMAN | P32248 | CHEMBL4594 | C-C Chemokine Receptor Type 7, Human | 1 |
| CXCR2_HUMAN | P25025 | CHEMBL2434 | Interleukin-8 Receptor B, Human | 1 |
| CXCR4_HUMAN | P61073 | CHEMBL2107 | C-X-C Chemokine Receptor Type 4, Human | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| CCR1_HUMAN | P32246 | CHEMBL2413 | C-C Chemokine Receptor Type 1, Human | 383 | 10 | 0 | 0 |
| CCR2_HUMAN | P41597 | CHEMBL4015 | C-C Chemokine Receptor Type 2, Human | 1,214 | 6 | 1 | 2 |
| CCR3_HUMAN | P51677 | CHEMBL3473 | C-C Chemokine Receptor Type 3, Human | 908 | 15 | 2 | 1 |
| CCR4_HUMAN | P51679 | CHEMBL2414 | C-C Chemokine Receptor Type 4, Human | 238 | 6 | 1 | 1 |
| CCR5_HUMAN | P51681 | CHEMBL274 | C-C Chemokine Receptor Type 5, Human | 1,843 | 7 | 2 | 4 |
| CCR7_HUMAN | P32248 | CHEMBL4594 | C-C Chemokine Receptor Type 7, Human | 1 | 0 | 0 | 0 |
| CCR8_HUMAN | P51685 | CHEMBL4596 | C-C Chemokine Receptor Type 8, Human | 68 | 3 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| CCR4_HUMAN | P51679 | CHEMBL2414 | C-C Chemokine Receptor Type 4, Human | 1 |
| CCR5_HUMAN | P51681 | CHEMBL274 | C-C Chemokine Receptor Type 5, Human | 1 |
| CCR7_HUMAN | P32248 | CHEMBL4594 | C-C Chemokine Receptor Type 7, Human | 1 |
| CXCR2_HUMAN | P25025 | CHEMBL2434 | Interleukin-8 Receptor B, Human | 1 |
| CXCR4_HUMAN | P61073 | CHEMBL2107 | C-X-C Chemokine Receptor Type 4, Human | 1 |
| CXCR4_RAT | O08565 | CHEMBL5556 | C-X-C Chemokine Receptor Type 4, Rat | 1 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 1 |