| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 66 | 9 | 1 | 0 |
| Binding ≤ 1μM | 53 | 3 | 0 | 0 |
| Functional ≤ 10μM | 1 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_13639 | Astrocytic Glutamate-Glutamine Uptake And Metabolism | Homo sapiens |
| REACT_19397 | Transport of inorganic cations/anions and amino acids/oligopeptides | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| EAA1_HUMAN | P43003 | CHEMBL3085 | Excitatory Amino Acid Transporter 1, Human | 51 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| EAA1_HUMAN | P43003 | CHEMBL3085 | Excitatory Amino Acid Transporter 1, Human | 51 |
| EAA3_HUMAN | P43005 | CHEMBL2721 | Excitatory Amino Acid Transporter 3, Human | 60 |
| EAA4_HUMAN | P48664 | CHEMBL3173 | Excitatory Amino Acid Transporter 4, Human | 2 |
| EAA5_HUMAN | O00341 | CHEMBL4390 | Excitatory Amino Acid Transporter 5, Human | 2 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| EAA2_RAT | P31596 | CHEMBL2900 | Excitatory Amino Acid Transporter 2, Rat | 10 | 2 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| EAA1_HUMAN | P43003 | CHEMBL3085 | Excitatory Amino Acid Transporter 1, Human | 129 | 66 | 0 | 0 |
| EAA3_HUMAN | P43005 | CHEMBL2721 | Excitatory Amino Acid Transporter 3, Human | 70 | 8 | 1 | 1 |
| EAA4_HUMAN | P48664 | CHEMBL3173 | Excitatory Amino Acid Transporter 4, Human | 2 | 1 | 0 | 0 |
| EAA5_HUMAN | O00341 | CHEMBL4390 | Excitatory Amino Acid Transporter 5, Human | 2 | 1 | 0 | 0 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| EAA2-1-E | Excitatory Amino Acid Transporter 2 (cluster #1 Of 2), Eukaryotic | 53 | 8 | 0 | 0 |
| EAA2-2-E | Excitatory Amino Acid Transporter 2 (cluster #2 Of 2), Eukaryotic | 22 | 2 | 1 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| EAA3_HUMAN | P43005 | CHEMBL2721 | Excitatory Amino Acid Transporter 3, Human | 60 |
| EAA1_HUMAN | P43003 | CHEMBL3085 | Excitatory Amino Acid Transporter 1, Human | 51 |
| EAA1_RAT | P24942 | CHEMBL4190 | Excitatory Amino Acid Transporter 1, Rat | 2 |
| EAA2_RAT | P31596 | CHEMBL2900 | Excitatory Amino Acid Transporter 2, Rat | 2 |
| EAA3_RAT | P51907 | CHEMBL3113 | Excitatory Amino Acid Transporter 3, Rat | 2 |
| EAA4_HUMAN | P48664 | CHEMBL3173 | Excitatory Amino Acid Transporter 4, Human | 2 |
| EAA5_HUMAN | O00341 | CHEMBL4390 | Excitatory Amino Acid Transporter 5, Human | 2 |
| SATT_HUMAN | P43007 | CHEMBL2315 | Neutral Amino Acid Transporter A, Human | 2 |
| Z104302 | Z104302 | CHEMBL1907608 | Glutamate NMDA Receptor | 1 |