| Annotation Type | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|
| Binding ≤ 10μM | 50 | 41 | 13 | 1 | 
| Binding ≤ 1μM | 43 | 34 | 9 | 1 | 
| Functional ≤ 10μM | 39 | 0 | 0 | 0 | 
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|---|---|---|
| EST1_HUMAN | P23141 | CHEMBL2265 | Acyl Coenzyme A:cholesterol Acyltransferase, Human | 254 | 88 | 22 | 5 | 
| EST1_PIG | Q29550 | CHEMBL3383 | Carboxylesterase, Pig | 31 | 2 | 2 | 2 | 
| Code | Description | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|---|
| EST1-1-E | Carboxylesterase (cluster #1 Of 7), Eukaryotic | 85 | 32 | 4 | 2 | 
| EST1-2-E | Carboxylesterase (cluster #2 Of 7), Eukaryotic | 23 | 8 | 1 | 0 | 
| EST1-3-E | Carboxylesterase (cluster #3 Of 7), Eukaryotic | 2 | 2 | 1 | 0 | 
| EST1-4-E | Carboxylesterase (cluster #4 Of 7), Eukaryotic | 3 | 3 | 1 | 0 | 
| EST1-5-E | Carboxylesterase (cluster #5 Of 7), Eukaryotic | 37 | 1 | 0 | 1 | 
| EST1-6-E | Carboxylesterase (cluster #6 Of 7), Eukaryotic | 126 | 48 | 16 | 3 | 
| EST1-7-E | Carboxylesterase (cluster #7 Of 7), Eukaryotic | 7 | 1 | 1 | 1 | 
| Uniprot | Swissprot | Chembl | Description | Number Shared | 
|---|---|---|---|---|
| EST2_HUMAN | O00748 | CHEMBL3180 | Carboxylesterase 2, Human | 45 | 
| EST1_HUMAN | P23141 | CHEMBL2265 | Acyl Coenzyme A:cholesterol Acyltransferase, Human | 42 | 
| ACES_HUMAN | P22303 | CHEMBL220 | Acetylcholinesterase, Human | 2 | 
| CHLE_HUMAN | P06276 | CHEMBL1914 | Butyrylcholinesterase, Human | 2 | 
| SOAT1_RAT | O70536 | CHEMBL285 | Acyl Coenzyme A:cholesterol Acyltransferase 1, Rat | 2 | 
| EST1_PIG | Q29550 | CHEMBL3383 | Carboxylesterase, Pig | 1 |