| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 35 | 1 | 0 | 0 |
| Binding ≤ 1μM | 34 | 1 | 0 | 0 |
| Functional ≤ 10μM | 1 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_207651 | G alpha (q) signalling events | Mus musculus |
| REACT_242871 | G alpha (s) signalling events | Mus musculus |
| REACT_210399 | Glucagon signaling in metabolic regulation | Mus musculus |
| REACT_231304 | Glucagon-type ligand receptors | Mus musculus |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GLR_HUMAN | P47871 | CHEMBL1985 | Glucagon Receptor, Human | 503 | 13 | 0 | 0 |
| GLR_RAT | P30082 | CHEMBL4720 | Glucagon Receptor, Rat | 15 | 0 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GLRA4_MOUSE | Q61603 | CHEMBL3500 | Glycine Receptor Alpha-4 Chain, Mouse | 3 | 1 | 1 | 1 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| GLR-1-E | Glucagon Receptor (cluster #1 Of 2), Eukaryotic | 183 | 3 | 0 | 0 |
| GLR-2-E | Glucagon Receptor (cluster #2 Of 2), Eukaryotic | 332 | 10 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| GLR_HUMAN | P47871 | CHEMBL1985 | Glucagon Receptor, Human | 36 |
| MK14_HUMAN | Q16539 | CHEMBL260 | MAP Kinase P38 Alpha, Human | 16 |
| GIPR_HUMAN | P48546 | CHEMBL4383 | Gastric Inhibitory Polypeptide Receptor, Human | 9 |
| GLR_RAT | P30082 | CHEMBL4720 | Glucagon Receptor, Rat | 9 |
| E2R517_CANFA | E2R517 | CHEMBL1649060 | Uncharacterized Protein, Canine | 1 |
| MK14_RAT | P70618 | CHEMBL4825 | MAP Kinase P38 Alpha, Rat | 1 |