| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 2 | 1 | 0 | 0 |
| Binding ≤ 1μM | 0 | 0 | 0 | 0 |
| Functional ≤ 10μM | 2 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_75770 | Voltage gated Potassium channels | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| KCAB1_HUMAN | Q14722 | CHEMBL5884 | Voltage-gated Potassium Channel Subunit Beta-1, Human | 1 |
| KCNA1_HUMAN | Q09470 | CHEMBL2309 | Voltage-gated Potassium Channel Subunit Kv1.1, Human | 4 |
| KCNA2_HUMAN | P16389 | CHEMBL2086 | Voltage-gated Potassium Channel Subunit Kv1.2, Human | 2 |
| KCNA5_HUMAN | P22460 | CHEMBL4306 | Voltage-gated Potassium Channel Subunit Kv1.5, Human | 2 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 2 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| KCNA1_HUMAN | Q09470 | CHEMBL2309 | Voltage-gated Potassium Channel Subunit Kv1.1, Human | 13 | 2 | 0 | 0 |
| KCNA2_HUMAN | P16389 | CHEMBL2086 | Voltage-gated Potassium Channel Subunit Kv1.2, Human | 7 | 0 | 0 | 0 |
| KCNA3_HUMAN | P22001 | CHEMBL4633 | Voltage-gated Potassium Channel Subunit Kv1.3, Human | 232 | 11 | 7 | 1 |
| KCNA5_HUMAN | P22460 | CHEMBL4306 | Voltage-gated Potassium Channel Subunit Kv1.5, Human | 537 | 11 | 5 | 5 |
| KCNA7_HUMAN | Q96RP8 | CHEMBL2773 | Voltage-gated Potassium Channel Subunit Kv1.7, Human | 1 | 1 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| KCNA1_HUMAN | Q09470 | CHEMBL2309 | Voltage-gated Potassium Channel Subunit Kv1.1, Human | 4 |
| KCNA2_HUMAN | P16389 | CHEMBL2086 | Voltage-gated Potassium Channel Subunit Kv1.2, Human | 2 |
| KCNA3_MOUSE | P16390 | CHEMBL4818 | Voltage-gated Potassium Channel Subunit Kv1.3, Mouse | 2 |
| KCNA5_HUMAN | P22460 | CHEMBL4306 | Voltage-gated Potassium Channel Subunit Kv1.5, Human | 2 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 2 |
| Z100759 | Z100759 | CHEMBL614167 | T-lymphocytes | 2 |
| KCAB1_HUMAN | Q14722 | CHEMBL5884 | Voltage-gated Potassium Channel Subunit Beta-1, Human | 1 |