| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 1 | 1 | 0 | 1 |
| Binding ≤ 1μM | 1 | 1 | 0 | 1 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_247448 | ERK1 activation | Mus musculus |
| REACT_224208 | Interleukin-1 signaling | Mus musculus |
| REACT_247566 | MEK activation | Mus musculus |
| REACT_257146 | RAF phosphorylates MEK | Mus musculus |
| REACT_215461 | Signal transduction by L1 | Mus musculus |
| REACT_242456 | Signaling by FGFR | Mus musculus |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| MP2K1_HUMAN | Q02750 | CHEMBL3587 | Dual Specificity Mitogen-activated Protein Kinase Kinase 1, Human | 463 | 35 | 15 | 12 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| MP2K1-1-E | Dual Specificity Mitogen-activated Protein Kinase Kinase 1 (cluster #1 Of 4), Eukaryotic | 212 | 20 | 4 | 10 |
| MP2K1-2-E | Dual Specificity Mitogen-activated Protein Kinase Kinase 1 (cluster #2 Of 4), Eukaryotic | 114 | 2 | 0 | 0 |
| MP2K1-3-E | Dual Specificity Mitogen-activated Protein Kinase Kinase 1 (cluster #3 Of 4), Eukaryotic | 131 | 9 | 5 | 2 |
| MP2K1-4-E | Dual Specificity Mitogen-activated Protein Kinase Kinase 1 (cluster #4 Of 4), Eukaryotic | 9 | 7 | 7 | 1 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| AA3R_HUMAN | P33765 | CHEMBL256 | Adenosine A3 Receptor, Human | 1 |