| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 232 | 13 | 10 | 8 |
| Functional ≤ 10μM | 1 | 1 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GBRP_HUMAN | O00591 | CHEMBL3506 | GABA Receptor Pi Subunit, Human | 240 | 19 | 11 | 9 |
| GBRP_MOUSE | Q8QZW7 | CHEMBL2746 | GABA Receptor Pi Subunit, Mouse | 37 | 3 | 2 | 2 |
| GBRP_RAT | O09028 | CHEMBL294 | GABA Receptor Pi Subunit, Rat | 37 | 7 | 7 | 3 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| GBRP-2-E | GABA Receptor Pi Subunit (cluster #2 Of 6), Eukaryotic | 3 | 3 | 1 | 1 |
| GBRP-3-E | GABA Receptor Pi Subunit (cluster #3 Of 6), Eukaryotic | 26 | 8 | 5 | 4 |
| GBRP-4-E | GABA Receptor Pi Subunit (cluster #4 Of 6), Eukaryotic | 22 | 0 | 0 | 0 |
| GBRP-5-E | GABA Receptor Pi Subunit (cluster #5 Of 6), Eukaryotic | 26 | 3 | 3 | 0 |
| GBRP-6-E | GABA Receptor Pi Subunit (cluster #6 Of 6), Eukaryotic | 3 | 0 | 0 | 0 |