| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 3,485 | 332 | 79 | 95 |
| Functional ≤ 10μM | 48 | 5 | 3 | 3 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| SGMR1_CAVPO | Q60492 | CHEMBL4153 | Sigma-1 Receptor, Guinea Pig | 823 | 43 | 14 | 13 |
| SGMR1_HUMAN | Q99720 | CHEMBL287 | Sigma Opioid Receptor, Human | 1,873 | 230 | 56 | 56 |
| SGMR1_MOUSE | O55242 | CHEMBL3465 | Sigma Opioid Receptor, Mouse | 205 | 11 | 8 | 7 |
| SGMR1_RAT | Q9R0C9 | CHEMBL3602 | Sigma Opioid Receptor, Rat | 1,157 | 146 | 42 | 57 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| SGMR1-2-E | Sigma Opioid Receptor (cluster #2 Of 6), Eukaryotic | 15 | 6 | 3 | 3 |
| SGMR1-3-E | Sigma Opioid Receptor (cluster #3 Of 6), Eukaryotic | 135 | 9 | 7 | 4 |
| SGMR1-4-E | Sigma Opioid Receptor (cluster #4 Of 6), Eukaryotic | 193 | 26 | 3 | 3 |
| SGMR1-5-E | Sigma Opioid Receptor (cluster #5 Of 6), Eukaryotic | 1 | 1 | 1 | 0 |
| SGMR1-6-E | Sigma Opioid Receptor (cluster #6 Of 6), Eukaryotic | 42 | 5 | 1 | 1 |
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