c1ccc(c(c1)c2nnco2)O 10A-002 CC(=O)c1ccc(cc1)n2ccnc2 10A-004 Cc1ccc(cc1)S(=O)(=O)Oc2ccccc2c3nnco3 10A-008 c1ccc(c(c1)c2nnco2)OS(=O)(=O)c3ccc(cc3)Cl 10A-009 COc1ccc(cc1)S(=O)(=O)Oc2ccccc2c3nnco3 10A-010 CN(C)/C=C/[N+](=O)[O-] 10A-011 c1ccc(cc1)S(=O)(=O)Oc2ccccc2c3nnco3 10A-013 c1cc(ccc1Cn2c(nnn2)N)Cl 10A-024 c1ccc(cc1)C(=O)Oc2ccccc2c3nnco3 10A-026 Cc1cccc(c1)C(=O)Oc2ccccc2c3nnco3 10A-027 c1ccc(c(c1)c2nnco2)OC(=O)c3ccc(cc3)Cl 10A-028 c1ccc(c(c1)c2nnc3n2CCCC3)O 10A-031 CN1CCN(CC1)c2ccc(cc2)c3ccno3 10B-001 CCSC(C(=O)NC)SCC 10B-003 c1ccc(cc1)/C=C/c2ncnn2c3ccccc3F 10B-004 c1ccnc(c1)c2ccnc(n2)N 10B-006 c1ccc(cc1)NC(=O)Nc2nccc(n2)c3ccccn3 10B-007 CN(C)/C=C/C(=O)c1ccc(c(c1)[N+](=O)[O-])Cl 10B-008 c1cc(c(cc1c2ccn[nH]2)[N+](=O)[O-])Cl 10B-010 Cc1c(c(on1)/C=C/Nc2ccccc2)[N+](=O)[O-] 10B-011 CCOC(CC(=O)NN)OCC 10B-013 COC(CC(=O)NNC(=S)Nc1ccccc1)OC 10B-015 c1c(cnc(c1C(F)(F)F)NN)C(F)(F)F 10B-018 c1c(cc(nc1C(F)(F)F)NN)C(F)(F)F 10B-019 c1c(cc(nc1C(F)(F)F)C(F)(F)F)NN 10B-020 c1c(c(cnc1NN)C(F)(F)F)C(F)(F)F 10B-021 COC(Cc1nnc(n1c2ccccc2)S)OC 10B-022 c1ccnc(c1)c2c[nH]nc2N3CCOCC3 10B-023 c1cc(c(c(c1)Cl)C(=O)NNc2cc(nc(c2)C(F)(F)F)C(F)(F)F)Cl 10B-029 c1ccnc(c1)CNC=C2C(=NNC2=O)C(F)(F)F 10B-031 c1cc(cnc1)CNC=C2C(=NNC2=O)C(F)(F)F 10B-032 C1COCCN1NC=C2C(=NNC2=O)C(F)(F)F 10B-033 CC1=NNC(=O)C1=CNN2CCOCC2 10B-035 CC1=NNC(=O)C1=CNCc2cccs2 10B-036 c1cc(sc1)CNC=C2C(=NNC2=O)C(F)(F)F 10B-037 CCOC(CNC(=O)NC(=O)c1cccnc1)OCC 10B-040 c1ccc2c(c1)c(c[nH]c2=O)C(=O)O 10B-046 c1ccc(cc1)C\2=NNC(=O)/C2=C/NCc3cccs3 10B-048 c1ccc(cc1)C2=NNC(=O)C2=CNN3CCOCC3 10B-049 Cc1c(c(no1)c2ccccc2)C(=O)N 10B-051 CCOC(CNC(=O)NC(=O)c1ccncc1)OCC 10B-052 Cn1ccc2c(c1=O)cc3c(=O)c4ccccc4oc3n2 10B-055 c1ccc(cc1)Cn2ccc3c(c2=O)cc4c(=O)c5ccccc5oc4n3 10B-057 Cc1c(c(no1)c2ccccc2)C#N 10B-058 Cc1cccc(c1)N/C=C/c2c(c(no2)C)[N+](=O)[O-] 10B-059 Cc1c(c(on1)/C=C/Nc2cccc(c2)OC)[N+](=O)[O-] 10B-060 CCOC(CNC(=O)NC(=O)c1ccc(nc1)OC)OCC 10B-061 Cc1c(c(on1)/C=C/Nc2ccc(cc2)Cl)[N+](=O)[O-] 10B-062 Cc1c(c(on1)/C=C/Nc2ccc(cc2)C(=O)O)[N+](=O)[O-] 10B-063 Cc1c(c(on1)/C=C/Nc2ccc(cc2F)F)[N+](=O)[O-] 10B-064 CCOC(CNC(=O)NC(=O)c1cnccn1)OCC 10B-065 Cc1c(c(on1)/C=C/Nc2ccsc2C(=O)OC)[N+](=O)[O-] 10B-066 COC(Cc1nnc(n1c2ccccc2)SCc3ccccc3)OC 10B-067 Cc1c(cccc1[N+](=O)[O-])C(=O)OC 10B-068 CCOC(CNC(=O)NC(=O)c1cccnc1OC)OCC 10B-069 CNC(=S)NNC(=O)CC(OC)OC 10B-070 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3c(onc3c4ccccc4)C 10B-073 Cn1c(c2c(n1)CCCC2)N(C)C(=O)Nc3ccc(cc3)Cl 10B-074 Cn1c(c2c(n1)CCCC2)N(C)S(=O)(=O)c3ccccc3 10B-075 CN(C)C=C1C(=NNC1=O)COC 10B-079 c1ccc2c(c1)c(cnc2Cl)C(=O)Nc3ccc(cc3)Cl 10B-083 Cn1c(c2c(n1)CCCC2)N(C)S(=O)(=O)C 10B-086 CN(c1ccc(cc1)Cl)C(=O)c2cnc(c3c2cccc3)Cl 10B-088 CN(C)C(=O)c1cnc(c2c1cccc2)Cl 10B-089 COCC1=NNC(=O)C1=CNc2ccccc2 10B-090 COCC1=NNC(=O)C1=CNc2ccc(cc2)Cl 10B-091 COCC1=NNC(=O)C1=CNc2cc(cc(c2)Cl)Cl 10B-092 COCC1=NNC(=O)C1=CNc2ccc(cc2F)F 10B-093 Cc1c(c(on1)/C=C/Nc2cc(ccc2O)Cl)[N+](=O)[O-] 10B-095 Cc1c(c(on1)/C=C/Nc2cc(cc(c2)Cl)Cl)[N+](=O)[O-] 10B-096 Cc1cccc(c1N/C=C/c2c(c(no2)C)[N+](=O)[O-])C 10B-097 c1cc2c(cc[nH]c2=O)c(c1)[N+](=O)[O-] 10B-099 COCC1=NNC(=O)C1=CNCc2cccs2 10B-100 COCC1=NNC(=O)C1=CNN2CCOCC2 10B-101 Cn1c(nnc1S)CC(OC)OC 10B-102 Cc1ccc(cc1)N/C=C/c2c(c(no2)C)[N+](=O)[O-] 10B-104 Cc1c(c(on1)/C=C/Nc2ccccc2OC)[N+](=O)[O-] 10B-105 CN(C)/C=C/c1c(c(no1)c2ccccc2)C#N 10B-107 COCC1=NNC(=O)C1=CNCc2ccccn2 10B-108 COCC1=NNC(=O)C1=CNCc2ccc(cc2)Cl 10B-109 COCC1=NNC(=O)C1=CNCc2cccnc2 10B-110 Cn1c(nnc1SCc2ccccc2)CC(OC)OC 10B-111 CN(C)/C=C(/C#N)\c1cccs1 10B-112 CN(C)/C=C(/C#N)\c1ccsc1 10B-113 COCC1=NNC(=O)C1=CNCC(=O)OC 10B-115 CCOC(=O)c1cc2c(=O)c3ccccc3oc2nc1/C=C/Nc4cc(cc(c4)Cl)Cl 10B-116 Cc1ccc(cc1C)N/C=C/c2c(c(no2)C)[N+](=O)[O-] 10B-118 Cc1c(c(on1)/C=C/Nc2ccc(cc2)Oc3ccccc3)[N+](=O)[O-] 10B-119 Cc1c(c(on1)/C=C/Nc2cccc(c2)SC)[N+](=O)[O-] 10B-120 Cc1cc(ccc1N/C=C/c2c(c(no2)C)[N+](=O)[O-])O 10B-121 Cc1c(c(on1)/C=C/Nc2ccc(cc2OC)OC)[N+](=O)[O-] 10B-122 c1cc(cnc1)C(=N)NNC(=O)CC#N 10B-124 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)NCc4ccc(cc4)Cl 10B-125 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)NCc4ccccn4 10B-126 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)NCc4cccnc4 10B-127 CNC(=O)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F 10B-128 CC(C)NC(=O)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F 10B-129 Cc1c(c(on1)/C=C/Nc2ccccc2c3ccccc3)[N+](=O)[O-] 10B-131 C=CCNC(=O)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F 10B-133 Cc1cccc(c1NC(=O)c2cc3c(=O)c4ccccc4oc3nc2C(F)(F)F)C 10B-134 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)NCc4cccc(c4)C(F)(F)F 10B-135 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)Nc4ccc(cc4F)F 10B-136 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)Nc4cccc(c4)C(F)(F)F 10B-137 CN(C)/C=C(/c1ccccc1C(=O)OC)\C(=O)OC 10B-138 CC(c1ccnn1S(=O)(=O)c2ccccc2)Oc3cccc(c3)C(F)(F)F 10C-001 CC(c1ccnn1C(=O)C)Oc2ccccc2 10C-002 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)Br)/C#N 10C-003 CCNC(=O)n1c(ccn1)C(C)Oc2ccccc2 10C-004 CC(c1ccnn1S(=O)(=O)C)Oc2ccccc2 10C-007 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)C#N)/C#N 10C-010 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)[N+](=O)[O-])/C#N 10C-011 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccccc1F)/C#N 10C-012 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)C(=O)OC)/C#N 10C-013 CCNC(=O)n1c(ccn1)C(C)Oc2ccc(cc2)Cl 10C-014 CC(C)(C)S(=O)(=O)/C(=N\Nc1ccc(cc1)OC)/C#N 10C-015 CC(C)(C)S(=O)(=O)/C(=N/Nc1cccc(c1)OC)/C#N 10C-020 Cc1cccc(c1)N/N=C(\C#N)/S(=O)(=O)C(C)(C)C 10C-021 CC(C)(C)c1ccc(cc1)N/N=C(\C#N)/S(=O)(=O)C(C)(C)C 10C-022 CC(C)(C)S(=O)(=O)/C(=N\Nc1ccc(cc1)SC)/C#N 10C-023 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(c(c1)Cl)Cl)/C#N 10C-024 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)S(=O)(=O)N)/C#N 10C-026 CCNC(=O)n1c(ccn1)C(C)Oc2cccc(c2)C(F)(F)F 10C-027 CC(c1ccnn1S(=O)(=O)C)Oc2ccc(cc2)Cl 10C-030 CC(C)(C)S(=O)(=O)/C(=N\Nc1ccc2c(c1)OCO2)/C#N 10C-031 CC(c1ccnn1S(=O)(=O)C)Oc2cccc(c2)C(F)(F)F 10C-035 C[N+](C)(CC(=O)c1ccc(cc1)Cl)CC(=O)c2ccc(cc2)Cl.[Br-] 10C-036 CC(c1ccnn1C(=O)C)Oc2cccc(c2)C(F)(F)F 10C-041 CC(c1ccnn1C(=O)C)Oc2ccc(cc2)Cl 10C-044 CCOC(=O)/C(=C\N(C)C)/C#N 10C-046 CS/C(=N\C#N)/N1CCN(CC1)c2ccccc2 10C-047 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)F)C(=O)N 10C-052 c1ccc2c(c1)c(nn(c2=O)c3cccc(c3)C(F)(F)F)C(=O)N 10C-053 c1ccc(cc1)N2CCN(CC2)c3[nH]nc(n3)N 10C-054 c1cc(ccc1N2CCN(CC2)c3[nH]nc(n3)N)F 10C-055 Cc1cc(nc2c1c(=O)[nH]cn2)C 10C-056 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)N 10C-057 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)N 10C-058 Cn1c(nc(n1)N)N2CCN(CC2)c3ccc(cc3)F 10C-060 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)N 10C-061 CN(C)/C=C/C(=O)c1ccccc1O 10C-065 CO/N=C/CC(=O)c1ccccc1O 10C-066 CN(C)/C=C/C(=O)c1ccc(cc1)F 10C-067 CO/N=C/CC(=O)c1ccc(cc1)F 10C-068 Cn1c(nc(n1)N)N2CCN(CC2)c3cccc(c3)C(F)(F)F 10C-070 CN(C)/C=C/C(=O)c1ccc(cc1)Oc2ccccc2 10C-072 CO/N=C/CC(=O)c1ccc(cc1)Oc2ccccc2 10C-075 CO/N=C/C1C(=O)CCCC1=O 10C-077 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/OCc3c(cccc3Cl)Cl 10D-002 COC(=O)c1c(ccs1)c2ccc(o2)C(=O)O 10D-003 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)Cl 10D-005 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/OCc3ccc(c(c3)Cl)Cl 10D-009 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/OC 10D-010 CN(C)/C=C/C(=O)c1ccc(cc1)n2ccc(=O)cc2 10D-011 C[N+](=C/N=C(\Nc1ccccc1)/SCc2c(cccc2Cl)Cl)C.[Cl-] 10D-013 COC(=O)c1c(ccs1)c2ccc(o2)C(=O)Nc3ccccc3 10D-014 COC(=O)c1c(ccs1)c2ccc(o2)C=C(C#N)C#N 10D-015 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)NN 10D-016 c1cc(ccc1c2ccn[nH]2)n3ccc(=O)cc3 10D-017 c1ccc(cc1)N2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 10D-018 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)N3CCOCC3 10D-019 Cc1cc(n(n1)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)C 10D-020 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/OC(=O)c3ccccc3 10D-021 CCOC(=O)/C(=C/c1ccc(o1)c2ccsc2C(=O)OC)/C#N 10D-022 COC(=O)c1c(ccs1)c2ccc(o2)/C=C(/C#N)\c3ccccc3 10D-023 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/OCc3ccc(cc3Cl)Cl 10D-024 c1ccc(cc1)Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10D-025 c1cc(ccc1Sc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 10D-026 COc1ccc(cc1)Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10D-027 c1cc(ccc1Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 10D-028 c1cc(cc(c1)Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)C(F)(F)F 10D-029 c1ccc(cc1)Oc2ccc(cc2)Nc3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 10D-030 c1cc(c(cc1Cl)Cl)Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10D-031 c1cc(ccc1Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 10D-032 c1cc(ccc1C#N)Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10D-033 CC(=O)c1ccccc1Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10D-034 COC(=O)c1c(ccs1)c2ccc(o2)/C=C/[N+](=O)[O-] 10D-035 CCOC(=O)C(=Cc1ccc(o1)c2ccsc2C(=O)OC)C(=O)OCC 10D-036 c1cc(ccc1CNc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 10D-037 c1ccc(cc1)Sc2ccc(nn2)Cc3ccc(cc3Cl)Cl 10D-038 c1ccc(cc1)Sc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10D-039 Cc1ccc(cc1)Sc2ccc(nn2)Cc3ccc(cc3Cl)Cl 10D-041 c1cc(ccc1Sc2ccc(nn2)Cc3ccc(cc3Cl)Cl)Cl 10D-042 Cc1c(c(ns1)S(=O)(=O)/C(=N\Nc2ccccc2)/C#N)C#N 10D-044 CCOC(=O)/C(=C/c1ccc(o1)c2ccsc2C(=O)OC)/C(=O)C 10D-045 CC(=O)C(=Cc1ccc(o1)c2ccsc2C(=O)OC)C(=O)C 10D-046 c1ccc(cc1)NC(=O)CC(=O)c2cnc(s2)Nc3ccccc3Cl 10D-048 c1cc(cc(c1)Cl)Sc2ccc(nn2)Cc3ccc(cc3Cl)Cl 10D-049 CC(=O)CC(=O)Nc1ccc(cc1Cl)Cl 10D-050 c1ccc(cc1)CSc2ccc(nn2)Cc3ccc(cc3Cl)Cl 10D-051 c1cc(ccc1c2ccnc(n2)N)n3ccc(=O)cc3 10D-052 c1cc(ccc1N/C=C/C(=O)Nc2ccc(cc2Cl)Cl)Cl 10D-053 c1cc(ccc1/N=C/c2c(nc3n2ccs3)Cl)Cl 10D-054 c1ccc(cc1)/N=C/c2c(nc3n2ccs3)Cl 10D-055 c1cc(ccc1/N=C/c2c(nc3n2ccs3)Cl)OC(F)(F)F 10D-056 c1ccc(c(c1)/N=C/c2c(nc3n2ccs3)Cl)O 10D-057 c1ccc(cc1)Oc2ccc(cc2)/N=C/c3c(nc4n3ccs4)Cl 10D-058 CNc1ncc(s1)C(=O)CC(=O)Nc2ccccc2 10D-060 c1cc(ccc1NC(=O)CC(=O)O)Cl 10D-061 c1cc(cc(c1)/N=C/c2c(nc3n2ccs3)Cl)C(F)(F)F 10D-062 c1cc(c(cc1Cl)/N=C/c2c(nc3n2ccs3)Cl)O 10D-063 c1cc(cc(c1)Cl)/N=C/c2c(nc3n2ccs3)Cl 10D-064 COC(=O)c1c(c2ccncc2s1)N 10D-065 CC(=O)CC(=O)Nc1ccc(cc1)Cl 10D-066 CC(=O)CC(=O)Nc1cccc(c1)C(F)(F)F 10D-067 CC(=O)CC(=O)Nc1ccc(cc1)OC 10D-068 Cc1ccc(cc1)NC(=O)CC(=O)C 10D-069 CN(C)/C=C/C(=O)Nc1ccc(cc1)Cl 10D-070 c1ccc2c(c1)NC(S2)c3c(nc4n3ccs4)Cl 10D-071 c1ccc(cc1)NC(=O)CC(=O)c2cnc(s2)Nc3ccc(c(c3)Cl)Cl 10D-073 COC(=O)c1c(ccs1)c2ccc(o2)COC(=O)Nc3ccc(cc3)Cl 10D-075 COc1ccc(cc1)C/N=C/c2c(nc3n2ccs3)Cl 10D-076S Cc1ccc(cc1)C/N=C/c2c(nc3n2ccs3)Cl 10D-077S c1ccc(cc1)C/N=C/c2c(nc3n2ccs3)Cl 10D-078S c1cc(ccc1C/N=C/c2c(nc3n2ccs3)Cl)Cl 10D-079S c1ccc(c(c1)C/N=C/c2c(nc3n2ccs3)Cl)Cl 10D-080S C=CCSc1ccc(nn1)Cc2ccc(cc2Cl)Cl 10D-081 c1cc(c(cc1Cl)Cl)Cc2ccc(nn2)S 10D-082 Cc1c(c(ns1)S(=O)(=O)/C(=N\Nc2ccc(cc2)OC)/C#N)C#N 10D-083 c1cc(ccc1CSc2ccc(nn2)Cc3ccc(cc3Cl)Cl)Br 10D-084 CO/N=C\CC(=O)Nc1ccc(cc1)Cl 10D-085 c1cc(ccc1NC(=O)C/C=N\O)Cl 10D-086 Cc1c(c(ns1)S(=O)(=O)/C(=N/Nc2cccc(c2)C(F)(F)F)/C#N)C#N 10D-087 c1cc(ccc1NC(=O)C/C=N\OCc2ccc(c(c2)Cl)Cl)Cl 10D-088 c1cc(ccc1NC(=O)C/C=N\OCc2ccc(cc2Cl)Cl)Cl 10D-089 c1cc(ccc1NC(=O)CC(=O)O)OC(F)(F)F 10D-090 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CC(=O)O 10D-091 CN(C)/C=C/C(=O)Nc1ccc(cc1)Oc2ccccc2 10D-092 Cc1c(c(ns1)S(=O)(=O)/C(=N\Nc2ccc(cc2)OC(F)(F)F)/C#N)C#N 10D-093 Cc1c(c(ns1)S(=O)(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/C#N)C#N 10D-094 c1ccc(cc1)Oc2ccc(cc2)NC(=O)C/C=N\O 10D-095 c1cc(cc(c1)Cl)C/N=C/c2c(nc3n2ccs3)Cl 10D-096S c1cc(cnc1)C/N=C/c2c(nc3n2ccs3)Cl 10D-097S CSc1ccc(nn1)Cc2ccc(cc2Cl)Cl 10D-098 CC1(OC(=O)C(=C2C3CC4CC(C3)CC2C4)C(=O)O1)C 10D-500 C(CSSCCC(=O)N)C(=O)N 10D-504 CC1(OC(=O)C(C(=O)O1)C2(C3CC4CC(C3)CC2C4)c5ccccc5)C 10D-505 C1CCN2C(C1)CC(O2)CO 10D-506 c1ccc(c(c1)C2(C3CC4CC(C3)CC2C4)O)NC=O 10D-509 CCOC(=O)c1c(nc2n1cccc2)C 10D-518 CNC(=O)CCSSCCC(=O)NC 10D-526 c1ccc(cc1)CNC(=O)CCSSCCC(=O)NCc2ccccc2 10D-527 c1ccc(c(c1)NC(=O)CCSSCCC(=O)Nc2ccccc2Cl)Cl 10D-528 c1ccc(cc1)NC(=O)CCSSCCC(=O)Nc2ccccc2 10D-529 Cc1c(n2ccccc2n1)C(=O)O 10D-545 CCOC(=O)c1c(nc2n1ccc(c2)C)C 10D-547 CCOC(=O)c1c(nc2n1cccc2C)C 10D-548 c1ccc2c(c1)C3(C4CC5CC(C4)CC3C5)OC(=N2)C(F)(F)F 10D-552 CCOC(=O)c1c(nc2n1cc(cc2)C)C 10D-574 Cc1ccn2c(c1)nc(c2C(=O)O)C 10D-582 c1ccc(c(c1)C2(C3CC4CC(C3)CC2C4)O)NC(=O)C5CC5 10D-587 Cc1ccc(cc1)NC(=O)c2c(nc3n2cccc3)C 10D-591 Cc1cccn2c1nc(c2C(=O)Nc3ccc(cc3)Cl)C 10D-593 c1cc([nH]c1)C(=O)C(F)(F)F 10E-001 c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4cccc(c4)Cl 10E-002 c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4ccc(cc4)Cl 10E-003 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)C(F)(F)F 10E-004 CC1(CC(=CC(=O)C1)/C=C/N(C)C)C 10E-005 CC1(C/C(=N\O)/CC2(C1)CC=NO2)C 10E-007 CN(C)C(=O)c1cc(c[nH]1)C(c2ccc(cc2Cl)Cl)O 10E-008 COc1ccc(cc1)N2CCN(CC2)c3cnc4ccccc4n3 10E-009 c1ccc2c(c1)ncc(n2)N3CCN(CC3)Cc4ccc5c(c4)OCO5 10E-010 c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4ccc(cc4)[N+](=O)[O-] 10E-011 c1ccc(cc1)C(=O)Cn2cncn2 10E-013 CCOC(=O)Cn1cncn1 10E-014 CN(C)/C=C(/C(=O)c1ccccc1)\n2cncn2 10E-015 CC1(CC(=CC(=O)C1)/C=C/Nc2ccc(cc2)C(=O)O)C 10E-016 c1ccc(cc1)c2c(c[nH]n2)n3cncn3 10E-017 CC1(CC(=CC(=O)C1)/C=C/Nc2ccc(cc2Cl)Cl)C 10E-018 CC1(CC(=CC(=O)C1)/C=C/Nc2ccc(cc2)Oc3ccccc3)C 10E-020 CO/N=C\NC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)Cl 10E-023 COc1ccc(cc1)c2cnc3nc(nn3c2N)N4CCN(CC4)C(c5ccccc5)c6ccccc6 10E-024 c1ncn(n1)CC(=O)N 10E-025 c1ccc(cc1)c2c(cnc(n2)N)n3cncn3 10E-026 c1cc(c(cc1Cl)Cl)CO/N=C/NC(=O)Cn2cncn2 10E-028 c1cc(c(cc1C(F)(F)F)F)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 10E-029 c1cc(c(cc1CO/N=C/NC(=O)Cn2cncn2)Cl)Cl 10E-034 c1cc(c(c(c1)Cl)CO/N=C/NC(=O)Cn2cncn2)Cl 10E-035 c1cc(ccc1CO/N=C/NC(=O)Cn2cncn2)Cl 10E-036 CNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2F)C(F)(F)F 10E-037 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4cnc5ccccc5n4 10E-038 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)c3[nH]ncn3 10E-040 CN(C)C(=O)Cn1cncn1 10E-041 c1ccc(cc1)c2cnc3nc(nn3c2N)N4CCN(CC4)C(c5ccccc5)c6ccccc6 10E-042 c1ccc2c(c1)ncc(n2)N3CCOCC3 10E-043 CN(C)/C=C(\C#N)/C(=C(C#N)C#N)N 10E-044 c1ccc2c(c1)-c3c(cccn3)C2=O 10E-045 c1ccc\2c(c1)-c3c(cccn3)/C2=N/O 10E-046 CO/N=C\NC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 10E-047 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4nc5ncc(c(n5n4)N)c6ccsc6 10E-049 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)C(F)(F)F 10E-053 CNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)C(F)(F)F 10E-055 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)C(F)(F)F 10E-056 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)C(F)(F)F 10E-057 CCOC(=O)C(C)(C)n1cncn1 10E-058 c1ncn(n1)CC#N 10E-060 c1ccc2c(c1)/C(=C/Nc3cccc(c3)Oc4c(cc(cn4)C(F)(F)F)Cl)/OC2=O 10E-061 c1ccc2c(c1)c(n[nH]c2=O)CNc3cccc(c3)Oc4c(cc(cn4)C(F)(F)F)Cl 10E-062 c1cnccc1c2nnc(o2)S 10E-063 Cc1cccc(c1)c2cnn(c2N)c3ccccc3 10E-301S Cc1cccc(c1)c2cnn(c2N)c3cccc(c3)[N+](=O)[O-] 10E-302S Cc1cccc(c1)c2cnn(c2N)c3cccc(c3)Cl 10E-303S COC(=O)c1ccc(=O)n(c1)Cc2ccc(c(c2)F)F 10E-304S Cc1ccc(cc1)c2cnn(c2N)c3ccccc3 10E-305S Cc1ccc(cc1)c2cnn(c2N)c3cccc(c3)[N+](=O)[O-] 10E-306S Cc1ccc(cc1)c2cnn(c2N)c3cccc(c3)Cl 10E-307S c1cc(ccc1Cn2cc(cc(c2=O)C(=O)N)Cl)C(F)(F)F 10E-308S COC(=O)c1ccccc1NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)C(F)(F)F)Cl 10E-309S c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3ccc(cc3)Cl 10E-310S Cc1cccc(c1)c2cnn(c2N)c3cccc(c3)C(F)(F)F 10E-311S Cc1ccc(cc1)c2cnn(c2N)c3cccc(c3)C(F)(F)F 10E-312S c1cc(ccc1NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3Cl)Cl)Cl)Cl 10E-313S c1cc(c(cc1Cl)Cl)Cn2cc(cc(c2=O)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl 10E-314S c1cc(ccc1C(F)(F)F)NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3Cl)Cl)Cl 10E-315S c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3ccc(cc3Cl)Cl 10E-316S COC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2Cl)Cl 10E-317S c1cc(c(cc1Cl)Cl)Cn2cc(ccc2=O)C(=O)O 10E-318S c1cc(c(cc1Cn2cc(ccc2=O)C(=O)O)F)F 10E-320S c1cc(cc(c1)Cl)c2cnn(c2N)c3cccc(c3)C(F)(F)F 10E-321S COC(=O)c1ccccc1NC(=O)c2cc(cn(c2=O)Cc3cccc(c3)Cl)Cl 10E-323S COC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)Cl 10E-326S c1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)F)F 10E-327S CNC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2Cl)Cl 10E-328S CCNC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2Cl)Cl 10E-329S CN(C)C(=O)c1ccc(=O)n(c1)Cc2ccc(cc2Cl)Cl 10E-330S c1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3Cl)Cl 10E-331S COc1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3Cl)Cl 10E-332S c1cc(cc(c1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3Cl)Cl)C(F)(F)F 10E-333S c1cc(c(cc1Cl)Cl)Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F 10E-334S Cc1c(cccc1Cl)NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)F)F 10E-335S c1cc(c(cc1Cn2cc(ccc2=O)C(=O)Nc3cc(cc(c3)Cl)Cl)F)F 10E-336S c1cc(ccc1NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)F)F)Cl 10E-337S Cc1ccc(cc1C)NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)F)F 10E-338S COC(=O)c1ccccc1NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)F)F 10E-339S c1cc(c(cc1Cn2cc(ccc2=O)C(=O)N)F)F 10E-340S c1cc(c(cc1Cl)Cl)Cn2cc(cc(c2=O)Cl)C(=O)O 10E-341S c1cc(c(cc1Cl)Cl)Cn2cc(ccc2=O)C(=O)N 10E-342S COC(=O)c1ccccc1NC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3Cl)Cl 10E-343S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)NN 10E-344S c1cc(cc(c1)C(F)(F)F)Cn2cccc(c2=O)C(=O)NN 10E-345S CNC(=S)NNC(=O)c1cccn(c1=O)Cc2cccc(c2)C(F)(F)F 10E-347S CNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 10E-348S Cn1c(nnc1S)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 10E-349S Cn1c(nnc1S)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 10E-350S CN(C)S(=O)(=O)N1CCN(CC1)C(c2ccccc2)c3ccccc3 10E-352S c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)C(=O)NN 10E-354S c1ccc(cc1)NC(=S)NNC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 10E-355S CNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccc(cc2Cl)Cl 10E-357S CCNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccc(cc2Cl)Cl 10E-358S c1ccc(cc1)n2c(nnc2S)c3cccn(c3=O)Cc4cccc(c4)C(F)(F)F 10E-359S Cn1c(nnc1S)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 10E-360S CCn1c(nnc1S)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 10E-361S C=CCNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccc(cc2Cl)Cl 10E-362S C=CCn1c(nnc1S)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 10E-364S c1cc(cc(c1)C(F)(F)F)Cn2cccc(c2=O)c3nnc(o3)S 10E-365S CC(C)OC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)Cl 10E-367S CCCCOC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)Cl 10E-368S C#CCOC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)Cl 10E-369S CCOCCOC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)Cl 10E-370S c1cc(ccc1CNC(=O)c2cc(c(=O)n(c2)Cc3ccc(cc3Cl)Cl)Cl)Cl 10E-371S CC(C)OC(=O)c1ccc(=O)n(c1)Cc2ccc(c(c2)Cl)Cl 10E-375S c1ccc(cc1)N2CCN(CC2)C(=O)c3ccc(=O)n(c3)Cc4ccc(c(c4)Cl)Cl 10E-376S c1ccc(cc1)CNC(=O)c2cc(c(=O)n(c2)Cc3ccc(cc3Cl)Cl)Cl 10E-377S c1ccc(c(c1)CCN2CCN(CC2)C(=O)c3ccc(=O)n(c3)Cc4ccc(c(c4)Cl)Cl)C(F)(F)F 10E-379S c1cc(ccc1N2CCN(CC2)C(=O)c3ccc(=O)n(c3)Cc4ccc(c(c4)Cl)Cl)Cl 10E-382S c1cc(cc(c1)Cl)N2CCN(CC2)C(=O)c3ccc(=O)n(c3)Cc4ccc(c(c4)Cl)Cl 10E-383S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)NN 10E-384S CNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2ccccc2 10E-385S C=CCNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2ccccc2 10E-386S CCNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2ccccc2 10E-387S Cn1c(nnc1S)c2ccc(=O)n(c2)Cc3ccccc3 10E-388S CCn1c(nnc1S)c2ccc(=O)n(c2)Cc3ccccc3 10E-390S C=CCn1c(nnc1S)c2ccc(=O)n(c2)Cc3ccccc3 10E-391S c1ccc(cc1)Cn2cc(ccc2=O)c3nnc(o3)S 10E-392S c1ccc(cc1)Cn2cccc(c2=O)C(=O)NN 10E-393S c1ccc(cc1)Cn2cccc(c2=O)c3nnc(o3)S 10E-394S CNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccccc2 10E-395S C=CCNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccccc2 10E-396S Cn1c(nnc1S)c2cccn(c2=O)Cc3ccccc3 10E-397S C=CCn1c(nnc1S)c2cccn(c2=O)Cc3ccccc3 10E-398S CSc1nnc(o1)c2cccn(c2=O)Cc3ccccc3 10E-399S c1ccc(cc1)Cn2cccc(c2=O)c3nnc(o3)SCc4ccc(c(c4)Cl)Cl 10E-400S c1ccc(cc1)Cn2cccc(c2=O)c3nnc(o3)SCc4ccc(cc4Cl)Cl 10E-401S c1ccc(cc1)Cn2cccc(c2=O)c3nnc(o3)SCc4ccc(cc4)Cl 10E-402S CNC(=S)NNC(=O)c1cccn(c1=O)Cc2cccc(c2)Cl 10E-405S C=CCNC(=S)NNC(=O)c1cccn(c1=O)Cc2cccc(c2)Cl 10E-406S c1ccc(cc1)COC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 10E-407S c1cc(cc(c1)Cl)Cn2cccc(c2=O)c3nnc(o3)S 10E-408S c1ccc(cc1)n2c(nnc2S)c3cccn(c3=O)Cc4cccc(c4)Cl 10E-409S Cn1c(nc(n1)c2cccn(c2=O)Cc3cccc(c3)Cl)S 10E-410S C=CCn1c(nnc1S)c2cccn(c2=O)Cc3cccc(c3)Cl 10E-411S COC(=O)/C(=C\Nc1ccccc1)/NC(=O)c2ccccc2 10E-900 COC(=O)/C(=C\Nc1ccc(cc1Cl)Cl)/NC(=O)c2ccccc2 10E-901 c1cc(cc(c1)NC(=O)CC(=O)Nc2cccc(c2)C(F)(F)F)C(F)(F)F 10E-902 COc1ccc(cc1)N/C=C(\C(=O)OC)/NC(=O)c2ccc(cc2Cl)Cl 10E-903 COC(=O)/C(=C\Nc1ccccc1)/NC(=O)c2ccc(cc2Cl)Cl 10E-904 c1ccc(cc1)N2C(=O)NC3(N2)CCCCC3 10E-905 CN(C)C=C(C(=O)Nc1cccc(c1)C(F)(F)F)C(=O)Nc2cccc(c2)C(F)(F)F 10E-907 CN(C)C=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 10E-908 Cc1c(c(n(n1)c2nc(cs2)c3ccc(cc3Cl)Cl)O)C(=O)/C=C(/C)\O 10E-909 Cc1ccc(cc1)c2csc(n2)n3c(c(c(n3)C)C(=O)/C=C(/C)\O)O 10E-910 COC(=O)/C(=C\Nc1ccc(cc1Cl)Cl)/NC(=O)c2ccc(cc2Cl)Cl 10E-911 c1ccc(cc1)Nc2c3nncn3c4ccccc4n2 10E-912 c1ccc2c(c1)nc(c3n2cnn3)N4CCCCC4 10E-913 Cc1cc(n(n1)c2ccccc2)c3c(nn(c3O)c4nc(cs4)c5ccc(cc5Cl)Cl)C 10E-914 COc1ccc(cc1)C(=O)N/C(=C/Nc2ccc(cc2)OC)/C(=O)OC 10E-915 c1ccc(cc1)NC(=O)C(/C=N/O)C(=O)Nc2ccccc2 10E-916 COc1ccc(cc1)C(=O)N/C(=C/Nc2ccccc2)/C(=O)OC 10E-917 Cc1cc(n(n1)c2ccc(cc2)Cl)c3c(nn(c3O)c4ccccc4)C 10E-918 Cc1cc(n(n1)c2ccccc2)c3c(nn(c3O)c4nc(cs4)c5ccccc5)C 10E-919 COc1ccc(cc1)C(=O)N/C(=C/Nc2ccc(cc2Cl)Cl)/C(=O)OC 10E-920 Cc1cc(n(n1)c2ccc(cc2)OC)c3c(nn(c3O)c4nc(cs4)c5ccccc5)C 10E-921 CO/N=C/C(C(=O)Nc1ccccc1)C(=O)Nc2ccccc2 10E-922 Cc1cc(c(c(=O)o1)/C(=N/Nc2ccc(cc2)Cl)/C)O 10E-923 CC1(NC(=O)N(N1)c2ccccc2)c3ccc(cc3)N 10E-924 Cc1c(c(n(n1)c2ccc(cc2)Cl)O)C(=O)/C=C(/C)\O 10E-925 CC1(NC(=O)N(N1)c2ccccc2)c3ccc(cc3)O 10E-926 Cc1cc(n(n1)c2ccccc2)c3c(nn(c3O)c4ccc(cc4)Cl)C 10E-927 c1cc(c(cc1Cl)Cl)CO/N=C/C(C(=O)Nc2ccc(cc2Cl)Cl)C(=O)Nc3ccc(cc3Cl)Cl 10E-929 Cc1cc(c(c(=O)o1)/C(=N/Nc2nc(cs2)c3cccc(c3)C(F)(F)F)/C)O 10E-930 c1ccc2c(c1)nc(c3n2cnn3)NOCc4ccc(cc4)Cl 10E-932 c1ccc(cc1)N2CCN(CC2)c3c4nncn4c5ccccc5n3 10E-933 Cc1cc(n(n1)c2c(nc3ccccc3n2)Cl)C 10E-934 Cc1c(c(n(n1)c2nc(cs2)c3ccc(cc3)OC)O)C(=O)/C=C(/C)\O 10E-935 Cc1c(c(n(n1)c2nc(cs2)c3cccc(c3)C(F)(F)F)O)C(=O)/C=C(/C)\O 10E-936 Cc1cc(n(n1)c2ccccc2)c3c(nn(c3O)c4nc(cs4)c5ccc(cc5)OC)C 10E-937 c1ccc(cc1)N2C(=O)NC3(N2)C4CC5CC(C4)CC3C5 10E-938 c1cc2c(cc1Cl)[nH]c(=O)c(=O)[nH]2 10E-939 c1ccc(cc1)CNc2c3nncn3c4ccccc4n2 10E-940 Cc1cc(n(n1)c2ccc(cc2)Cl)c3c(nn(c3O)c4ccc(cc4)Cl)C 10E-941 CO/N=C/C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 10E-943 Cc1cc(n(n1)CCO)c2c(nn(c2O)c3ccccc3)C 10E-944 c1cc(cc(c1)NC(=O)C(/C=N/OCc2ccc(cc2Cl)Cl)C(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F 10E-945 Cc1cc2c(o1)CC(CC2=O)(C)C 10E-946 c1cc2c(cc1Cl)nc(c(n2)Cl)Cl 10E-949 c1cc2c(cc1Cl)nc(c(n2)Cl)NN 10E-953 c1ccc2c(c1)n3cnnc3c4n2cnn4 10E-954 c1cc(c(nc1)I)OC(=O)c2ccc(cc2Cl)Cl 10E-955 c1ccc2c(c1)nc(c3n2cnn3)Sc4ccc(cc4)Cl 10E-957 COc1ccc(cc1)C(=O)Oc2cccnc2I 10E-961 CO/N=C/C(C(=O)Nc1cccc(c1)C(F)(F)F)C(=O)Nc2cccc(c2)C(F)(F)F 10E-962 c1ccc(cc1)C(=O)Oc2cccnc2I 10E-963 c1ccc(cc1)C(=O)C[n+]2ccccc2.[I-] 10E-964 c1cc[n+](cc1)CC(=O)c2ccc(cc2)Cl.[I-] 10E-965 c1cc(c(nc1)I)OC(=O)Nc2ccc(cc2)[N+](=O)[O-] 10E-967 CCNC(=O)Oc1cccnc1I 10E-968 Cc1cc(n(n1)C(C)(C)C)c2c(nn(c2O)c3nc(cs3)c4ccccc4)C 10E-969 COc1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccccc5F 10E-970 c1cc[n+](cc1)CC(=O)c2ccco2.[I-] 10E-971 Cc1cc(n(n1)c2ccc(cc2Cl)Cl)c3c(nn(c3O)c4nc(cs4)c5ccccc5)C 10E-973 Cc1cc(n(n1)C(C)(C)C)c2c(nn(c2O)c3nc(cs3)c4ccc(cc4)Cl)C 10E-974 Cc1cc([nH]n1)c2c(nn(c2O)c3ccc(cc3)Cl)C 10E-975 c1cc(cc(c1)C(F)(F)F)C(=O)Oc2cccnc2I 10E-976 CC(=O)Oc1cccnc1I 10E-977 c1ccc2c(c1)[nH]c(=O)c(n2)NN 10E-979 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3ccccc3 10E-980 c1ccc(cc1)/C=N/Nc2c(=O)[nH]c3ccccc3n2 10E-981 c1cc[n+](cc1)CC(=O)c2ccc(cc2Cl)Cl.[I-] 10E-982 CC(=O)CC1C(=O)CC(CC1=O)(C)C 10E-984 c1cc[n+](cc1)CC(=O)c2ccc(cc2)[N+](=O)[O-].[I-] 10E-985 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3ccco3 10E-986 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3ccc(cc3)Cl 10E-987 CN(C)c1nc(c(c(=O)o1)C#N)Cl 10E-988 C/C(=N\Oc1c(cc(cn1)C(F)(F)F)Cl)/c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F 10F-004 c1ccc(cc1)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl 10F-005 c1c(cnc(c1Cl)CC(C#N)c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 10F-008 CO/N=C/C(c1ncc(cc1Cl)C(F)(F)F)/C=N/OC 10F-009 Cc1c(c(n(n1)C)C)Br 10F-010 Cc1c(c(n(n1)C)C)C=O 10F-011 Cn1cc(cc1/C=C(\C#N)/c2cccc(c2)C(F)(F)F)C(=O)c3ccc(cc3Cl)Cl 10F-012 Cn1cc(cc1/C=C(\C#N)/c2ccccn2)C(=O)c3ccc(cc3Cl)Cl 10F-013 c1c(cnc(c1Cl)c2cnoc2)C(F)(F)F 10F-014 CO/N=C/C(=C\Nc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)Cl 10F-015 Cc1c(c(n(n1)C)C)/C=N/O 10F-016 Cc1c(c(n(n1)C)C)C#N 10F-017 c1ccc(cc1)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10F-018 c1c(cnc(c1Cl)/C=N/O)C(F)(F)F 10F-019 c1cc(c(cc1Cl)Cl)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10F-022 Cc1c(c(n(n1)C)C/C=N/OC)[N+](=O)[O-] 10F-024 c1c(cnc(c1Cl)c2c[nH]nc2)C(F)(F)F 10F-025 Cc1c(c(n(n1)C)/C(=C/N(C)C)/C=N/OC)[N+](=O)[O-] 10F-026 c1c(cnc(c1Cl)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 10F-027 CC1(OC(=O)C(=Cc2c(cc(cn2)C(F)(F)F)Cl)C(=O)O1)C 10F-028 Cn1c(ccc1C(=O)C(Cl)(Cl)Cl)/C(=C/c2ccc(cc2)Cl)/C#N 10F-029 c1ccc(c(c1)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 10F-030 CCOC(=O)c1cnn(c1N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 10F-031 c1cc(cc(c1)C(F)(F)F)Cn2cc(ccc2=O)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 10F-032 c1cc(ccc1Cn2cc(ccc2=O)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl)Cl 10F-036 CN(C)/C=N\C(=O)c1cc2c(s1)cc(cn2)C(F)(F)F 10F-040 CNC(=O)c1cc2c(s1)cc(cn2)C(F)(F)F 10F-042 CCOC(=O)CNc1c(cc(cn1)C(F)(F)F)Cl 10F-043 c1c(cnc(c1Cl)C#N)C(F)(F)F 10F-048 c1cc(ccc1NC(=O)/C=C/c2c(cc(cn2)C(F)(F)F)Cl)Oc3ccc(cn3)C(F)(F)F 10F-049 c1cc(ccc1OC(=O)/C=C/c2c(cc(cn2)C(F)(F)F)Cl)Cl 10F-054 c1ccc(cc1)OCC(=N)NNC(=O)c2cccnc2Oc3ccccc3 10F-055 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=N)COc3ccc(cc3)F 10F-056 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=N)COc3cccc(c3)C(F)(F)F 10F-057 c1c(cnc(c1Cl)NCC(=O)N)C(F)(F)F 10F-058 c1cc(ccc1NC(=O)/C=C/c2c(cc(cn2)C(F)(F)F)Cl)Cl 10F-059 Cc1c(snn1)S(=O)c2ccccc2C(=O)OC 10F-302S c1cc(ccc1CNc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])Cl 10F-304S c1cc(ccc1c2nc3ccc(cc3n2O)[N+](=O)[O-])Cl 10F-305S c1ccc(cc1)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-] 10F-306S CCOC(=O)C(C)On1c2cc(ccc2nc1c3ccc(cc3)OC)Cl 10F-307S CC(C(=O)O)On1c2cc(ccc2nc1c3ccc(cc3)OC)Cl 10F-308S CN(C)C(=O)On1c2cc(ccc2nc1c3ccc(cc3)OC)Cl 10F-309S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4ccccc4Cl)Cl 10F-310S CC1=CC(NC(=N1)SC)(C)C 10F-312S COc1ccc(cc1)c2nc3ccccc3n2OCC(=O)O 10F-313S CC(C(=O)O)On1c2ccccc2nc1c3ccc(cc3)OC 10F-314S CC1(C=C(N=C(N1)SC)/C=C/c2cccc(c2)Cl)C 10F-316S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4cccc(c4)Cl)Cl 10F-317S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4)Cl)Cl 10F-318S CCSC1=NC(=CC(N1)(C)C)C 10F-319S CC1(C=C(N=C(N1)SC)/C=C/c2ccc(cc2Cl)Cl)C 10F-320S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4cccc(c4)C(F)(F)F)Cl 10F-321S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4)C(F)(F)F)Cl 10F-322S CCn1c(nnc1S)c2cccn(c2=O)Cc3ccccc3 10F-323S Cc1ccc(cc1)COn2c3cc(ccc3nc2c4ccc(cc4)OC)Cl 10F-324S Cc1cc(cc(c1)COn2c3cc(ccc3nc2c4ccc(cc4)OC)Cl)C 10F-325S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4)Br)Cl 10F-326S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4Cl)Cl)Cl 10F-327S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)F)Cl 10F-330S Cc1c(snn1)S(=O)c2ccc(cc2)Br 10F-331S Cc1c(snn1)S(=O)c2ccc(cc2)C(F)(F)F 10F-332S Cc1c(snn1)S(=O)c2ccc(cc2)Cl 10F-333S Cc1c(snn1)S(=O)c2ccc(cc2)F 10F-334S CCOC(=O)COn1c2cc(ccc2nc1c3ccc(cc3)Cl)[N+](=O)[O-] 10F-335S CN(C)C(=O)On1c2cc(ccc2nc1c3ccc(cc3)Cl)[N+](=O)[O-] 10F-336S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(c(c4)Cl)Cl)Cl 10F-337S COc1ccc(cc1)c2nc3ccc(cc3n2OCc4c(cccc4Cl)Cl)Cl 10F-338S Cn1c(c(c(n1)C(F)(F)F)CO)Cl 10F-341S Cc1ccc(cc1)S(=O)c2c(nns2)C 10F-342S CCSC1=NC(=CC(N1)(C)C)/C=C/c2ccc(cc2)Cl 10F-343S CC1=CC(N(C(=S)N1)C)(C)C 10F-344S Cc1ccc(cc1)CNc2ccc(cc2[N+](=O)[O-])Cl 10F-345S Cc1ccc(cc1)c2nc3ccc(cc3n2O)Cl 10F-346S Cc1ccc(cc1)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-] 10F-347S Cn1c(nnc1SCC=C)c2cccn(c2=O)Cc3ccccc3 10F-348S Cn1c(nnc1SCC#C)c2cccn(c2=O)Cc3ccccc3 10F-349S COc1ccc(cc1)COn2c3cc(ccc3nc2c4ccc(cc4)OC)Cl 10F-350S Cc1c(snn1)S(=O)c2ccc(c(c2)Cl)Cl 10F-351S Cn1c(nnc1SCC(=O)O)c2cccn(c2=O)Cc3ccccc3 10F-352S CC(C(=O)O)Sc1nnc(n1C)c2cccn(c2=O)Cc3ccccc3 10F-353S CC(=O)Sc1nnc(n1C)c2cccn(c2=O)Cc3ccccc3 10F-354S Cn1c(nnc1SC(=O)c2ccccc2)c3cccn(c3=O)Cc4ccccc4 10F-355S Cn1c(c(c(n1)C(F)(F)F)C=O)Oc2cccc(c2)C(F)(F)F 10F-356S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Cl 10F-357S CC1(C=C(N=C(N1)SC)/C=C/c2c(cccc2Cl)Cl)C 10F-358S Cc1cc(cc(c1)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-])C 10F-359S c1cc(cc(c1)C(F)(F)F)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-] 10F-360S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2ccc(cc2)Cl)Cl 10F-362S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)F)Oc3cccc(c3)C(F)(F)F 10F-364S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Oc3cccc(c3)C(F)(F)F 10F-365S Cn1c(c(c(n1)C(F)(F)F)C=O)Oc2cccc(c2)Cl 10F-366S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2cccc(c2)Cl)Cl 10F-367S c1ccc(cc1)CNc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] 10F-368S c1ccc(cc1)c2nc3ccc(cc3n2O)[N+](=O)[O-] 10F-369S CC1(C=C(N=C(N1)SC)/C=C/c2ccccc2Cl)C 10F-370S CCOC(=O)C(C)On1c2cc(ccc2nc1c3ccccc3)Cl 10F-371S CC(C(=O)O)On1c2cc(ccc2nc1c3ccccc3)Cl 10F-372S CCOC(=O)C(C)On1c2cc(ccc2nc1c3ccc(cc3)Cl)[N+](=O)[O-] 10F-373S CC(C(=O)O)On1c2cc(ccc2nc1c3ccc(cc3)Cl)[N+](=O)[O-] 10F-374S c1cc(ccc1COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-])Cl 10F-375S Cn1c(nnc1SC)c2cccn(c2=O)Cc3ccccc3 10F-376S c1cc(cc(c1)Cl)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-] 10F-377S c1ccc(c(c1)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-])Cl 10F-378S c1cc(c(c(c1)Cl)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-])Cl 10F-379S c1cc(ccc1c2nc3ccc(cc3n2OCc4ccc(c(c4)Cl)Cl)[N+](=O)[O-])Cl 10F-380S c1cc(ccc1c2nc3ccc(cc3n2OCc4ccc(cc4Cl)Cl)[N+](=O)[O-])Cl 10F-381S Cn1c(c(c(n1)C(F)(F)F)C(=O)O)Oc2cccc(c2)Cl 10F-382S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)F)Oc3cccc(c3)Cl 10F-384S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Oc3cccc(c3)Cl 10F-385S c1cc(ccc1COn2c3cc(ccc3nc2c4ccc(cc4)Cl)[N+](=O)[O-])C(F)(F)F 10F-386S Cc1ccc(cc1)c2nc3ccc(cc3n2OCc4cccc(c4)C(F)(F)F)Cl 10F-388S Cc1ccc(cc1)c2nc3ccc(cc3n2OC(=O)N(C)C)Cl 10F-389S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccccc2Cl)Cl 10F-390S Cc1ccc(cc1)S(=O)(=O)NC(=O)OCc2c(nn(c2Cl)C)C(F)(F)F 10F-392S CCOC(=O)C(C)On1c2cc(ccc2nc1c3ccc(cc3)C)Cl 10F-393S CCOC(=O)COn1c2cc(ccc2nc1c3ccc(cc3)C)Cl 10F-394S c1cc(ccc1c2[nH]c3cc(ccc3n2)[N+](=O)[O-])Cl 10F-395S c1ccc(cc1)COn2c3cc(ccc3nc2c4ccccc4)[N+](=O)[O-] 10F-397S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4)Cl)[N+](=O)[O-] 10F-398S c1ccc(cc1)c2nc3ccc(cc3n2OCc4cccc(c4)Cl)[N+](=O)[O-] 10F-399S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccccc4Cl)[N+](=O)[O-] 10F-400S C=CCN(Cc1cccc(c1)C(F)(F)F)C(=O)c2cc(cc(c2)Cl)Cl 10F-401S Cn1c(c(c(n1)C(F)(F)F)COC(=O)C2CC2)Cl 10F-403S c1ccc(cc1)c2nc3ccc(cc3n2OCc4cccc(c4)C(F)(F)F)[N+](=O)[O-] 10F-405S CN(C)C(=O)On1c2cc(ccc2nc1c3ccccc3)[N+](=O)[O-] 10F-406S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2cccc(c2)Cl)Cl 10F-407S CCOC(=O)c1ccccc1c2csc(n2)Nc3ccc(c(c3)Cl)Cl 10F-901 CN(C)/C=C/C(=O)c1ccc(cc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 10F-902 c1ccc(cc1)n2cc3c(n2)CCN(C3)c4c(cc(cn4)C(F)(F)F)Cl 10F-904 CCOC(=O)CC(=N)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 10F-905 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)O)C(F)(F)F 10F-906 C/C(=N\OCc1ccc(cc1)Cl)/c2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 10F-907 c1cc(ccc1NC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 10F-909 COc1ccc(cc1)N2CCN(CC2)C(=O)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 10F-910 c1cc(ccc1CON/C=N\C(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 10F-911 c1cc(ccc1c2ccnc(n2)N)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 10F-912 c1ccc(cc1)n2c(ncn2)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 10F-914 CN(C)/C=C(\C#N)/C(=O)/N=C/NOCc1c(cccc1Cl)Cl 10F-916 CN(CCOc1c(cc(cn1)C(F)(F)F)Cl)C(=O)Cc2ccccc2 10F-917 Cc1cc(n2cc(c(c2n1)C(=O)N)c3ccc(cc3)Cl)C 10F-919 CN(CCOc1c(cc(cn1)C(F)(F)F)Cl)C(=O)/C(=C\Nc2ccc(cc2)OC)/c3ccccc3 10F-920 c1cc(ccc1c2c[nH]c(c2C#N)N)Cl 10F-921 c1c(cnc(c1Cl)N2CCC(CC2)c3[nH]cnn3)C(F)(F)F 10F-922 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)N 10F-923 c1ccc2c(c1)C(=O)N(C2=O)OCc3cccc(c3)Cl 10F-924 c1ccc(cc1)/C=N/c2c(c(c[nH]2)c3ccc(cc3)Cl)C#N 10F-925 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)O 10F-926 CCOC(=O)c1c(c[nH]c1NC(=O)Nc2ccc(cc2)Cl)c3ccccc3 10F-927 CCOC(=O)c1ccccc1c2csc(n2)NC(=O)c3ccc(cc3)F 10F-928 CCOC(=O)c1ccccc1c2csc(n2)NC(=O)c3cccc(c3)C(F)(F)F 10F-929 c1cc(cc(c1)Cl)CON.Cl 10F-930 CCOC(=O)c1ccccc1c2csc(n2)NS(=O)(=O)c3ccc(cc3)Cl 10F-931 Cc1ccc(cc1)n2c3c(c(n2)N)c(=O)oc(n3)N(C)C 10F-932 CN(C)c1nc2c(c(nn2c3ccc(cc3)F)N)c(=O)o1 10F-933 CN(C)c1nc2c(c(nn2c3ccc(cc3)Cl)N)c(=O)o1 10F-934 CCOC(=O)c1ccccc1c2csc(n2)N/C=N/OCc3cccc(c3)Cl 10F-936 CCOC(=O)c1ccccc1c2csc(n2)N/C=N/OCc3c(cccc3Cl)F 10F-937 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)N3CCN(CC3)c4ccc(cc4)OC 10F-938 CCOC(=O)c1ccccc1c2csc(n2)NC(=O)Nc3cccc(c3)C(F)(F)F 10F-940 CCOC(=O)c1ccccc1c2csc(n2)NC(=O)c3c(onc3c4c(cccc4Cl)F)C 10F-942 c1ccc(cc1)/C=N/c2c(c(cn2Cc3ccc(cc3)F)c4ccc(cc4)Cl)C#N 10F-944 CCOC(=O)c1ccccc1c2csc(n2)NC(=O)c3cccs3 10F-945 CCOC(=O)c1ccccc1c2csc(n2)NC(=O)c3ccco3 10F-947 C/C(=N\OC)/c1ccc(cc1)NC(=O)CC2(C3CC4CC(C3)CC2C4)c5ccccc5 10F-949 C/C(=N\O)/c1ccc(cc1)NC(=O)CC2(C3CC4CC(C3)CC2C4)c5ccccc5 10F-950 c1ccc(cc1)N2C(=O)NC3(N2)CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 10F-951 c1c(cnc(c1Cl)N2CCC3(CC2)NC(=O)N(N3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 10F-952 CCOC(=O)C=C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 10F-953 c1ccc(cc1)C(=O)CN2CCN(CC2)c3ccc(cc3)Cl 10F-954 c1ccc(cc1)C(=O)CN2CCN(CC2)c3cccc(c3)Cl 10F-955 c1ccc(cc1)CN2CCN(CC2)CC(=O)c3ccccc3 10F-956 c1ccc(cc1)C(=O)CN2CCN(CC2)c3ccccc3 10F-957 c1cc(ccc1NC(=O)ON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 10F-958 c1ccc(cc1)/C(=N/OCc2ccc(cc2)Cl)/CN3CCN(CC3)c4ccc(cc4)Cl 10F-960 c1ccc(cc1)/C(=N/OCc2ccc(cc2)Cl)/CN3CCN(CC3)c4ccccc4 10F-961 c1cc(ccc1CON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 10F-962 c1c(cnc(c1Cl)N2CCC(=CC(=O)O)CC2)C(F)(F)F 10F-963 c1ccc(cc1)CN2CCN(CC2)C/C(=N\OCc3ccc(cc3)Cl)/c4ccccc4 10F-964 Cc1ccc(cc1)CON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 10F-965 c1ccc(cc1)/C(=N/OCc2ccc(cc2)Cl)/CN3CCN(CC3)c4cccc(c4)Cl 10F-966 c1cc(c(cc1CON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl 10F-967 c1cc(cc(c1)C(F)(F)F)CON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 10F-968 c1cn(c(=O)[nH]c1=O)c2c(cc(cn2)C(F)(F)F)Cl 10F-969 CON=C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 10F-970 Cc1ccc(cc1)n2cc3c(n2)CCN(C3)c4c(cc(cn4)C(F)(F)F)Cl 10F-980 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)C 10G-001 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)/C=C/N(C)C 10G-002 c1c(cnc(c1Cl)Sc2nc([nH]n2)N)C(F)(F)F 10G-003 C/C(=N\OC)/c1cccs1 10G-004 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)/C(=N\OC)/C 10G-005 CSc1cccc(n1)Cl 10G-006 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 10G-007 CN(C)/C=N/C(=N\C=[N+](C)C)/SC.[I-] 10G-008 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)/C(=N\O)/C 10G-010 Cc1[nH]c(cn1)C(=O)/C=C/N(C)C 10G-012 Cn1ccc2c1c(c3ccccc3c2N)C#N 10G-014 c1c(cn(n1)C2CCS(=O)(=O)C2)C(=O)N 10G-016 CON/C=N/OC 10G-018 COC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3ccccc3 10G-020 CN(C)/C=N/C(=O)c1cnn(c1)C2CCS(=O)(=O)C2 10G-022 CO/N=C/N(C(=O)Nc1ccc(cc1)Cl)OC 10G-024 Cn1cccc1C(C#N)N(C)C 10G-025 c1cc(ccc1c2cnc3nc(nn3c2N)Sc4c(cc(cn4)C(F)(F)F)Cl)Cl 10G-026 c1ccc(cc1)/C=C\c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 10G-028 c1cc(ccc1c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl)Cl 10G-033 c1ccc(cc1)NC(=O)NC(=O)c2cnn(c2)C3CCS(=O)(=O)C3 10G-036 c1ccc(cc1)/C(=N\O)/c2c(cc(cn2)C(F)(F)F)Cl 10G-038 CCCCCCCCCCC(=O)c1cc([nH]c1)C(=O)C(Cl)(Cl)Cl 10G-043 CCOC(=O)c1cc(cc(c1O)C(=O)OCC)c2c(cc(cn2)C(F)(F)F)Cl 10G-044 CCCCCCCCCCC(=O)c1cc([nH]c1)C(=O)N 10G-045 c1cc(cc(c1)S(=O)(=O)Oc2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 10G-047 Cc1ccc(cc1)S(=O)(=O)Oc2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl 10G-048 c1cc(cc(c1)NC(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 10G-049 c1cc(cc(c1)C(F)(F)F)C(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 10G-050 c1cc(c(cc1Cl)Cl)C(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 10G-051 COc1ccc(cc1)C(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 10G-052 CC(=O)n1cc(cn1)c2c(cc(cn2)C(F)(F)F)Cl 10G-053 c1ccc(c(c1)Sc2ccc(cc2)NC(=O)c3cccnc3Cl)Cl 10G-301S Cc1cccc(c1)C(=O)Nc2ccc(cc2)Sc3ccccc3Cl 10G-302S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccccc3Cl 10G-303S c1csc(c1S)C(=O)O 10G-306S c1cc(ccc1N)N2CCOCC2 10G-307S c1cc(ccc1N2CCCC2)[N+](=O)[O-] 10G-310S c1cc(ccc1NC(=O)C(Oc2ccc(cc2)Cl)(F)F)Cl 10G-312S c1cc(ccc1OC(C(=O)Nc2cc(cc(c2)Cl)Cl)(F)F)Cl 10G-313S c1cc(ccc1N)N2CCCC2 10G-314S c1cc(ccc1C(=O)Nc2ccc(cc2)N3CCOCC3)F 10G-315S c1cc(ccc1C(=O)Nc2ccc(cc2)N3CCCCC3)F 10G-316S CC(=O)Nc1ccc(cc1)N2CCOCC2 10G-318S c1cc(ccc1NC(=O)CCl)N2CCOCC2 10G-319S c1cc(cc(c1)C(F)(F)F)CSc2ccsc2C(=O)O 10G-320S c1ccc(cc1)C(C(=O)O)NS(=O)(=O)c2ccc(cc2)Cl 10G-322S c1cc(ccc1NC(=O)C(Cl)Cl)N2CCOCC2 10G-324S c1cc(ccc1NC(=O)C(Cl)(Cl)Cl)N2CCOCC2 10G-325S Cc1ccc(cc1)S(=O)(=O)NC(c2ccccc2)C(=O)OC 10G-326S COc1ccc(cc1)S(=O)(=O)NC(c2ccccc2)C(=O)OC 10G-327S CC(C)CC(C(=O)OC)NS(=O)(=O)c1ccc(cc1)Cl 10G-328S Cc1ccc(cc1)S(=O)(=O)NC(CC(C)C)C(=O)OC 10G-329S c1cc(c(cc1CSc2ccsc2C(=O)O)Cl)Cl 10G-330S c1cc(c(cc1CSc2ccsc2C(=O)Nc3ccc(cc3F)F)Cl)Cl 10G-332S c1cc(ccc1OC(C(=O)Nc2ccc(cc2F)F)(F)F)Cl 10G-333S c1cc(c(cc1CSc2ccsc2C(=O)Nc3cc(cc(c3)Cl)Cl)Cl)Cl 10G-334S c1cc(c(cc1CSc2ccsc2C(=O)Nc3ccc(c(c3)Cl)Cl)Cl)Cl 10G-335S COc1ccc(cc1)S(=O)(=O)NC(c2ccccc2)C(=O)O 10G-336S c1ccc(cc1)C(C(=O)O)NS(=O)(=O)c2cccc(c2)C(F)(F)F 10G-337S c1ccc(cc1)C(C(=O)O)NS(=O)(=O)c2ccccc2Cl 10G-338S c1cc(cc(c1)C(F)(F)F)CSc2ccsc2C(=O)Nc3ccc(cc3)F 10G-339S C#CCSc1nnc(n1N)c2ccccc2 10G-340S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)N3CCOCC3 10G-341S c1cc(cc(c1)Cl)C(=O)Nc2ccc(cc2)N3CCOCC3 10G-342S c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)N3CCOCC3 10G-343S c1cc(cc(c1)C(F)(F)F)CSc2ccsc2C(=O)Nc3ccc(cc3F)F 10G-344S Cc1ccc(cc1)NC(=O)c2c(ccs2)SCc3cccc(c3)C(F)(F)F 10G-345S COc1ccc(cc1)NC(=O)c2c(ccs2)SCc3cccc(c3)C(F)(F)F 10G-346S Cc1cccc(c1NC(=O)c2c(ccs2)SCc3cccc(c3)C(F)(F)F)C 10G-347S Cc1ccc(cc1)S(=O)(=O)NC(c2ccccc2)C(=O)O 10G-348S CC(C(=O)O)NS(=O)(=O)c1cccc(c1)C(F)(F)F 10G-349S c1cc(ccc1C(=O)Nc2ccc(cc2)N3CCOCC3)Cl 10G-350S CC(C)(C)C(=O)Nc1ccc(cc1)N2CCOCC2 10G-351S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)N3CCOCC3 10G-352S CC(C(=O)O)NS(=O)(=O)c1ccc(cc1)OC 10G-353S c1ccc(cc1)CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)Cl 10G-354S c1cc(ccc1NC(=O)C(Oc2ccc(cc2)Cl)(F)F)F 10G-355S c1ccc(cc1)c2nnc3n2nc(n3c4ccccc4)S 10G-357S c1cc(ccc1NC(=O)c2c(ccs2)SCc3ccc(c(c3)Cl)Cl)F 10G-360S c1cc(ccc1NC(=O)c2c(ccs2)SCc3ccc(c(c3)Cl)Cl)Br 10G-361S c1cc(ccc1NC(=O)c2c(ccs2)SCc3ccc(c(c3)Cl)Cl)Cl 10G-362S c1cc(ccc1NC(=O)c2c(ccs2)SCc3ccc(c(c3)Cl)Cl)OC(F)(F)F 10G-363S CCCC(=O)Nc1ccc(cc1)N2CCOCC2 10G-365S CC(C)C(=O)Nc1ccc(cc1)N2CCOCC2 10G-366S c1ccc(cc1)CC(C(=O)O)NS(=O)(=O)c2ccccc2Cl 10G-367S c1ccc(cc1)CC(C(=O)O)NS(=O)(=O)c2cccc(c2)C(F)(F)F 10G-368S CC(C(=O)O)NS(=O)(=O)c1ccc(cc1)Br 10G-370S CCCCC(=O)Nc1ccc(cc1)N2CCOCC2 10G-371S c1cc(ccc1OC(C(=O)Nc2ccc(cc2Cl)Cl)(F)F)Cl 10G-372S c1cc(ccc1C(F)(F)F)NC(=O)C(Oc2ccc(cc2)Cl)(F)F 10G-373S c1ccc(c(c1)NC(=O)C(Oc2ccc(cc2)Cl)(F)F)F 10G-374S c1cc(ccc1OC(C(=O)N2CCCC2)(F)F)Cl 10G-375S c1ccc(cc1)C(C(=O)O)NS(=O)(=O)c2ccc(cc2)F 10G-376S CC(C(=O)O)NS(=O)(=O)c1ccccc1Cl 10G-377S CC(C)CC(=O)Nc1ccc(cc1)N2CCOCC2 10G-378S COc1cccc(c1)C(=O)Nc2ccc(cc2)N3CCOCC3 10G-379S CC(C)(CCl)C(=O)Nc1ccc(cc1)N2CCOCC2 10G-380S CC(C(=O)Nc1ccc(cc1)N2CCOCC2)Cl 10G-381S c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3)F 10G-382S CC(C)C(C(=O)O)NS(=O)(=O)c1ccc(cc1)F 10G-383S CC(C)C(C(=O)O)NS(=O)(=O)c1ccc(cc1)Cl 10G-384S CC(C)C(C(=O)O)NS(=O)(=O)c1ccc(cc1)Br 10G-385S CC(C)C(C(=O)O)NS(=O)(=O)c1ccccc1Cl 10G-386S c1cc(ccc1NC(=O)CCCl)N2CCOCC2 10G-387S c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)N3CCOCC3)F 10G-388S C=CCSc1nnc(n1N)c2ccccc2 10G-389S CC(C)CSc1nnc(n1N)c2ccccc2 10G-390S c1ccc(cc1)c2nnc(n2N)SCc3cccc(c3)C(F)(F)F 10G-391S c1ccc(cc1)c2nnc(n2N)SCc3ccc(cc3)Cl 10G-394S c1cc(ccc1NC(=O)CCl)N2CCCCC2 10G-395S c1cc(ccc1NC(=O)C(Cl)Cl)N2CCCCC2 10G-396S CC(C)C(C(=O)O)NS(=O)(=O)c1cccc(c1)C(F)(F)F 10G-397S c1cc(ccc1NC(=O)C(Cl)(Cl)Cl)N2CCCCC2 10G-398S CC(C)Sc1nnc(n1N)c2ccccc2 10G-399S CCOC(=O)CSc1nnc(n1N)c2ccccc2 10G-400S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)N3CCCCC3 10G-401S c1cc(cc(c1)Cl)C(=O)Nc2ccc(cc2)N3CCCCC3 10G-402S c1ccc(cc1)CSc2nnc(n2N)c3ccccc3 10G-404S c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)N3CCCCC3 10G-405S CC(C)(C)C(=O)Nc1ccc(cc1)N2CCCCC2 10G-406S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)N3CCCCC3 10G-407S c1cc(c(c(c1)Cl)CSc2ccsc2C(=O)O)Cl 10G-408S c1cc(c(c(c1)Cl)CSc2ccsc2C(=O)Nc3ccc(cc3F)F)Cl 10G-410S c1cc(c(c(c1)Cl)CSc2ccsc2C(=O)Nc3ccc(cc3)F)Cl 10G-411S Cc1ccc(cc1)NC(=O)c2c(ccs2)SCc3c(cccc3Cl)Cl 10G-412S c1cc(c(c(c1)Cl)CSc2ccsc2C(=O)Nc3ccc(cc3)Cl)Cl 10G-413S c1cc(c(c(c1)Cl)CSc2ccsc2C(=O)Nc3ccc(cc3)C(F)(F)F)Cl 10G-414S CCCC(=O)Nc1ccc(cc1)N2CCCCC2 10G-415S CC(C)C(=O)Nc1ccc(cc1)N2CCCCC2 10G-416S CCCCC(=O)Nc1ccc(cc1)N2CCCCC2 10G-417S CC(C)CC(=O)Nc1ccc(cc1)N2CCCCC2 10G-418S CN1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 10G-419S CN1CCN(CC1)c2ccc(cc2)N 10G-420S c1ccc(cc1)CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)F 10G-421S c1ccc(cc1)CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)Br 10G-422S COc1ccc(cc1)S(=O)(=O)NC(Cc2ccccc2)C(=O)O 10G-423S COC(=O)CSc1ccsc1C(=O)O 10G-424S CCC(=O)Nc1ccc(cc1)N2CCCCC2 10G-425S c1cc(c(nc1)Cl)C(=O)Nc2ccc(cc2)N3CCCCC3 10G-427S c1cc(ccc1S(=O)(=O)N2CCCC2C(=O)O)Cl 10G-428S c1ccc(c(c1)S(=O)(=O)N2CCCC2C(=O)O)Cl 10G-429S c1cc(ccc1F)S(=O)(=O)N2CCCC2C(=O)O 10G-430S c1cc(cc(c1)S(=O)(=O)N2CCCC2C(=O)O)C(F)(F)F 10G-432S c1ccc(cc1)C(C(=O)Nc2ccc(cc2)N3CCCCC3)Cl 10G-435S c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2ccc(cc2)N3CCCCC3 10G-436S c1cc(ccc1NC(=O)c2cc(cc(c2)Cl)Cl)N3CCCCC3 10G-437S c1cc(c(c(c1)Cl)CSc2ccsc2C(=O)Nc3ccc(cc3)OC(F)(F)F)Cl 10G-438S c1cc(ccc1CSc2ccsc2C(=O)O)[N+](=O)[O-] 10G-439S c1cc(ccc1CSc2ccsc2C(=O)Nc3ccc(cc3)F)[N+](=O)[O-] 10G-441S c1cc(ccc1CSc2ccsc2C(=O)Nc3ccc(cc3)C(F)(F)F)[N+](=O)[O-] 10G-442S c1cc(ccc1CSc2ccsc2C(=O)O)Cl 10G-447S c1cc(ccc1CSc2ccsc2C(=O)Nc3ccc(cc3)Cl)Cl 10G-449S Cc1ccc(cc1)NC(=O)c2c(ccs2)SCc3ccc(cc3)Cl 10G-450S c1cc(c(c(c1)Cl)CS(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3F)F)Cl 10G-451S c1cc(c(c(c1)Cl)CS(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3)C(F)(F)F)Cl 10G-452S c1cc(ccc1CS(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3)Cl)Cl 10G-453S Cc1ccc(cc1)NC(=O)c2c(ccs2)S(=O)(=O)Cc3ccc(cc3)Cl 10G-454S c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCCC2C(=O)O 10G-456S COc1ccc(cc1)NC(=O)c2c(ccs2)SCC(=O)OC 10G-457S c1cc(ccc1C(=O)Nc2ccc(cc2)N3CCCC3)F 10G-458S CC(=O)Nc1ccc(cc1)N2CCCC2 10G-459S c1cc(ccc1NC(=O)CCl)N2CCCC2 10G-462S c1cc(ccc1S(=O)(=O)N2CCCC2C(=O)O)Br 10G-463S COC(=O)CS(=O)(=O)c1ccsc1C(=O)Nc2ccc(cc2)OC(F)(F)F 10G-465S c1cc(ccc1NC(=O)C(Cl)Cl)N2CCCC2 10G-466S c1cc(ccc1NC(=O)C(Cl)(Cl)Cl)N2CCCC2 10G-467S c1cc(cc(c1)Cl)C(=O)Nc2ccc(cc2)N3CCCC3 10G-468S c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 10G-470S COC(=O)CS(=O)(=O)c1ccsc1C(=O)Nc2ccc(cc2)F 10G-471S c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)N 10G-472S CC(C)Sc1nnc(n1N)c2ccc(cc2)Cl 10G-473S c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)N3CCCC3 10G-475S c1cc(ccc1C(=O)Nc2ccc(cc2)N3CCCC3)Cl 10G-476S CC(Cc1nnc(n1N)c2ccccc2)C(=O)O 10G-477S CC(C)(C)C(=O)Nc1ccc(cc1)N2CCCC2 10G-478S CC(C)CC(C(=O)O)NS(=O)(=O)c1ccc(cc1)Cl 10G-479S CC(C)CC(C(=O)O)NS(=O)(=O)c1ccc(cc1)F 10G-480S COC(=O)C(c1ccccc1)NS(=O)(=O)c2ccccc2Cl 10G-481S COC(=O)C(c1ccccc1)NS(=O)(=O)c2cccc(c2)C(F)(F)F 10G-482S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)N3CCCC3 10G-483S CC(C)C(=O)Nc1ccc(cc1)N2CCCC2 10G-484S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)N3CCCC3 10G-485S CCCCC(=O)Nc1ccc(cc1)N2CCCC2 10G-486S CC(C(=O)Nc1ccc(cc1)N2CCCC2)Cl 10G-487S CC(C)(CCl)C(=O)Nc1ccc(cc1)N2CCCC2 10G-488S CNC(=O)c1c(ccs1)SCc2c(cccc2Cl)Cl 10G-490S C=CCNC(=O)c1c(ccs1)SCc2c(cccc2Cl)Cl 10G-491S Cc1ccc(cc1C)NC(=O)c2c(ccs2)SCc3c(cccc3Cl)Cl 10G-494S c1cc(cc(c1)NC(=O)c2c(ccs2)SCc3c(cccc3Cl)Cl)C(F)(F)F 10G-495S c1ccc(cc1)NC(=O)c2c(ccs2)SCc3c(cccc3Cl)Cl 10G-496S c1cc(c(c(c1)Cl)CSc2ccsc2C(=O)Nc3ccc(cc3)Br)Cl 10G-497S Cc1cccc(c1)NC(=O)c2c(ccs2)SCc3c(cccc3Cl)Cl 10G-498S c1cc(c(cc1Cl)Cl)CSc2ccsc2C(=O)O 10G-499S c1cc(ccc1NC(=O)c2c(ccs2)SCc3ccc(cc3Cl)Cl)Cl 10G-500S c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)N3CCCC3)F 10G-501S c1ccc(cc1)C(C(=O)Nc2ccc(cc2)N3CCCC3)Cl 10G-502S Cc1ccc(cc1)C(=O)Nc2ccc(cc2)N3CCCC3 10G-503S Cc1nnc(n1N)S 10G-504S Cc1ccc(cc1)NC(=O)c2c(ccs2)SCc3ccc(cc3Cl)Cl 10G-505S c1cc(ccc1NC(=O)c2c(ccs2)SCc3ccc(cc3Cl)Cl)OC(F)(F)F 10G-506S c1cc(ccc1NC(=O)c2c(ccs2)SCc3ccc(cc3Cl)Cl)F 10G-507S c1cc(c(cc1CS(=O)(=O)c2ccsc2C(=O)Nc3cc(cc(c3)Cl)Cl)Cl)Cl 10G-509S c1cc(ccc1NC(=O)c2c(ccs2)S(=O)(=O)Cc3ccc(c(c3)Cl)Cl)OC(F)(F)F 10G-510S c1cc(c(c(c1)Cl)CS(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3)OC(F)(F)F)Cl 10G-511S CNC(=O)c1c(ccs1)S(=O)(=O)Cc2c(cccc2Cl)Cl 10G-512S Cc1ccc(cc1C)NC(=O)c2c(ccs2)S(=O)(=O)Cc3c(cccc3Cl)Cl 10G-513S c1cc(cc(c1)NC(=O)c2c(ccs2)S(=O)(=O)Cc3c(cccc3Cl)Cl)C(F)(F)F 10G-514S c1cc(c(c(c1)Cl)CS(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3)Br)Cl 10G-515S c1cc(ccc1NC(=O)c2c(ccs2)S(=O)(=O)Cc3ccc(cc3Cl)Cl)OC(F)(F)F 10G-516S c1cc(ccc1NC(=O)c2c(ccs2)S(=O)(=O)Cc3ccc(cc3Cl)Cl)F 10G-517S Cc1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)Cl)(F)F)C 10G-518S Cc1cc(cc(c1)OC(C(=O)Nc2cc(cc(c2)Cl)Cl)(F)F)C 10G-519S Cc1cc(cc(c1)OC(C(=O)Nc2ccc(c(c2)F)F)(F)F)C 10G-520S CC(C)CC(C(=O)O)NS(=O)(=O)c1ccc(cc1)Br 10G-521S CC(C)CC(C(=O)O)NS(=O)(=O)c1cccc(c1)C(F)(F)F 10G-522S CC(C)CC(C(=O)O)NS(=O)(=O)c1ccccc1Cl 10G-523S CC(C(=O)OC)NS(=O)(=O)c1ccc(cc1)Cl 10G-524S c1cc(ccc1N2CCN(CC2)c3ccc(cc3)F)[N+](=O)[O-] 10G-526S c1cc(ccc1N)N2CCN(CC2)c3ccc(cc3)F 10G-527S Cc1ccc(cc1)S(=O)(=O)C(CCC(=O)c2ccc(cc2)Cl)C(=O)N 10G-528S Cc1cc(cc(c1)OC(C(=O)Nc2cccc(c2)OC)(F)F)C 10G-529S Cc1cc(cc(c1)OC(C(=O)Nc2ccc(cc2F)F)(F)F)C 10G-530S Cc1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)NC(=O)C)(F)F)C 10G-531S Cc1ccc(cc1C)NC(=O)C(Oc2cc(cc(c2)C)C)(F)F 10G-532S Cc1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)OC(F)(F)F)(F)F)C 10G-533S c1cc(c(cc1CS(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3F)F)Cl)Cl 10G-534S c1cc(ccc1NC(=O)c2c(ccs2)S(=O)(=O)Cc3ccc(c(c3)Cl)Cl)F 10G-535S Cc1ccc(cc1)NC(=O)c2c(ccs2)S(=O)(=O)Cc3c(cccc3Cl)Cl 10G-536S Cc1ccc(cc1)S(=O)(=O)N2CC(CC2C(=O)OC)Cl 10G-900 C=CCON1C(=O)c2ccccc2C1=O 10G-906 COC(=O)C1CC(CN1c2c(cc(cn2)C(F)(F)F)Cl)O 10G-907 CCOC(=O)C1=NOC(C1)CON2C(=O)c3ccccc3C2=O 10G-909 c1c(cnc(c1Cl)NCC2CC(=NO2)C(=O)O)C(F)(F)F 10G-910 CN(C=C1C(=O)CCCC1=O)OC(=O)Nc2ccccc2 10G-912 c1ccc(cc1)n2c(cc3c2CCCC3=O)c4ccccc4Cl 10G-916 c1c(cc(cc1Cl)Cl)CO 10G-918 c1ccc(cc1)/C(=N/Nc2ccccc2)/C(=N\Nc3ccccc3)/c4ccccc4 10G-919 COc1ccc(cc1OC)S(=O)(=O)N2CC(CC2C(=O)O)O 10G-920 c1cc(cc(c1)Cl)C(=O)CC2C(=O)CCCC2=O 10G-921 c1c(cnc(c1Cl)NCC2CC(=NO2)C(=O)NN)C(F)(F)F 10G-922 c1c(cnc(c1Cl)NCC2CC(=NO2)C(=O)N)C(F)(F)F 10G-923 c1ccc2c(c1)C(=O)N(C2=O)OCc3cc(cc(c3)Cl)Cl 10G-925 COc1ccc(cc1OC)S(=O)(=O)N2CC(CC2C(=O)OC)O 10G-926 c1c(cc(cc1Cl)Cl)CO[NH3+].[Cl-] 10G-928 COc1ccc(cc1OC)S(=O)(=O)N2CC(CC2C(=O)OC)Cl 10G-930 COC(=O)C1CC(CN1C(=O)c2ccc(cc2Cl)Cl)Cl 10G-931 c1ccc2c(c1)CCC3=C2CCN(C3)C(=O)c4ccc(cc4)Cl 10G-932 CN(C1c2c3ccccc3ccc2OCC1CO)C(=O)c4ccccc4 10G-933 c1ccc(cc1)c2cc\3c(n2c4ccccc4)CCC/C3=N/OCc5cc(cc(c5)Cl)Cl 10G-934 COC(=O)C1CC(CN1c2c(cc(cn2)C(F)(F)F)Cl)Cl 10G-935 c1cc(sc1)S(=O)(=O)N2CC(CC2C(=O)O)O 10G-937 c1c(cnc(c1Cl)NCC2CC3CCCCN3O2)C(F)(F)F 10G-939 CC(C)(C)C(=O)N(C)C1c2c3ccccc3ccc2OCC1CO 10G-941 c1cc(oc1)C(=O)N2CC(CC2C(=O)O)O 10G-942 COC(=O)C1CC(CN1S(=O)(=O)c2cccs2)O 10G-944 COC(=O)C1CC(CN1S(=O)(=O)c2cccs2)Cl 10G-949 c1c(cnc(c1Cl)NCC2CC(=NO2)C(=O)N3CCOCC3)C(F)(F)F 10G-950 COC(=O)C1CC(CN1C(=O)c2ccco2)O 10G-951 c1ccc2c(c1)ccc3c2C4C(CO3)COC(N4)c5cccnc5 10G-952 COC(=O)C1CC(CN1C(=O)c2ccco2)Cl 10G-954 CCOC(=O)C=C1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 10G-956 c1ccc(cc1)CN2CCC3(CC2)C(=O)NC(=O)N3 10G-957 c1cc(ccc1N2CCC(=CC(=O)NN)CC2)[N+](=O)[O-] 10G-958 c1cc(ccc1NC(=O)NNC(=O)C=C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])Cl 10G-959 c1ccc(cc1)NC(=O)N2CCc3ccccc3C2CC(CNc4c(cc(cn4)C(F)(F)F)Cl)O 10G-960 c1ccc(cc1)OCCn2c(=O)ccn(c2=O)c3c(cc(cn3)C(F)(F)F)Cl 10G-962 c1ccc2c(c1)C(=O)N(C2=O)CCn3c(=O)ccn(c3=O)c4c(cc(cn4)C(F)(F)F)Cl 10G-964 c1ccc(cc1)CCn2c(=O)ccn(c2=O)c3c(cc(cn3)C(F)(F)F)Cl 10G-965 c1ccc(cc1)C2(OCCO2)CBr 10G-967 CN(/C=C/C(=O)c1ccc(cc1)c2ccccc2)OC(=O)NC3CCCCC3 10G-969 CN(/C=C/C(=O)c1ccc(cc1)Br)O 10G-970 COc1ccc(cc1)OCCBr 10G-971 c1c(cnc(c1Cl)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 10H-001 COc1cccc(c1)N/C=C(/C#N)\C(=O)CSc2c(cc(cn2)C(F)(F)F)Cl 10H-002 c1cc(ccc1N/C=C(\C#N)/C(=O)CCl)Oc2c(cc(cn2)C(F)(F)F)Cl 10H-003 c1ccc2c(c1)CCNC2C(C(=O)C(F)(F)F)C(=O)C(F)(F)F 10H-004 c1ccc(cc1)/C(=N\NC(=O)N)/c2c(cc(cn2)C(F)(F)F)Cl 10H-005 CC(=O)C(C1c2ccccc2CCN1)C(=O)C(F)(F)F 10H-007 CN(C)/C=C(/C#N)\C(=O)CSC 10H-008 CSCC(=O)/C(=C\Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl)/C#N 10H-009 CSCC(=O)/C(=C\Nc1ccc(cc1Cl)Cl)/C#N 10H-012 c1c(cnc(c1Cl)c2nnc3n2cc(cc3Cl)C(F)(F)F)C(F)(F)F 10H-015 Cn1cc(cc1C=O)C(=O)c2ccc(cc2)F 10H-017 Cn1cc(cc1/C=C(/C=N/OC)\C#N)C(=O)c2ccc(cc2)F 10H-019 Cn1cc(cc1C=O)C(=O)c2ccccc2 10H-020 Cn1cc(cc1/C=C(/C=N/OC)\C#N)C(=O)c2ccccc2 10H-021 Cn1cc(cc1C=O)C(=O)c2ccc(cc2)[N+](=O)[O-] 10H-022 Cn1cc(cc1/C=C(/C=N/OC)\C#N)C(=O)c2ccc(cc2)[N+](=O)[O-] 10H-023 CN(C)c1nc(n(n1)c2ccccc2)N(C)C 10H-024 CN(C)c1nc(n(n1)C2CCS(=O)(=O)C2)N(C)C 10H-025 CCOC(=O)C\1=C(NC(=O)/C1=C\Nc2ccc(cc2)Cl)C 10H-026 CCOC(=O)C\1=C(NC(=O)/C1=C\Nc2ccc(cc2)OC)C 10H-027 CCOC(=O)C\1=C(NC(=O)/C1=C\Nc2ccc(cc2)C(F)(F)F)C 10H-028 CO/N=C/C(=C\c1c(cc(cn1)C(F)(F)F)Cl)/C#N 10H-029 Cn1c2cc(cnc2c(n1)c3ccccc3)C(F)(F)F 10H-030 COC(=O)C1CC(=O)NN(C1)C(=O)CCl 10H-031 CO/N=C/C(=C/c1ccc(cc1)C(F)(F)F)/C#N 10H-036 COc1ccc(cc1)/C=C(\C=N\OC)/C#N 10H-037 COC(=O)C1CC(=O)NN(C1)C(=O)CSc2ccccn2 10H-038 c1ccc(cc1)c2c(c(on2)c3cnc(nc3C(F)(F)F)N)C#N 10H-039 c1ccc(cc1)c2c(sc3c2ncc(c3)C(F)(F)F)CO 10H-043 c1c(cnc(c1Cl)n2cnc(n2)Sc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 10H-044 CN(C)c1nc(n(n1)c2ccccc2F)N(C)C 10H-045 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)[nH]n2 10H-050 c1cc(c(nc1)n2cnc(n2)Sc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 10H-051 c1cc(c(nc1)Sc2nc[nH]n2)[N+](=O)[O-] 10H-052 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)n(n2)C(=O)Nc4ccc(cc4)Cl 10H-053 CN(C)c1nc(n(n1)c2cccc(c2)Cl)N(C)C 10H-054 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2c4nc[nH]n4 10H-055 COC(=O)CC(=NNc1c(cc(cn1)C(F)(F)F)Cl)CC(=O)OC 10H-056 c1cc(c(nc1)Sc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 10H-057 c1cc(c(nc1)n2cnc(n2)Sc3c(cccn3)[N+](=O)[O-])[N+](=O)[O-] 10H-058 COC(=O)C1CC(=O)NN(C1)C(=O)CSc2c(cc(cn2)C(F)(F)F)Cl 10H-059 CN(C)c1nc(n(n1)c2ccc(cc2F)F)N(C)C 10H-062 CN(C)c1nc(n(n1)c2ccc(cc2)F)N(C)C 10H-063 CN(C)c1nc(n(n1)c2ccccc2Cl)N(C)C 10H-064 Cc1c(c(=O)cco1)OCc2ccc(cc2)Cl 10H-065 c1ccc(cc1)C2(CO2)c3ccccc3 10H-304S c1ccc(cc1)C(CS(=O)(=O)c2ccc(cc2)Cl)(c3ccccc3)O 10H-305S c1ccc(cc1)C(CSc2ccc(cc2)Cl)(c3ccccc3)O 10H-306S CS(=O)(=O)c1cnc(nc1c2ccc(c(c2)Cl)Cl)c3ccccc3 10H-307S CN(C)/C=C(/C(=O)c1ccccc1Cl)\S(=O)(=O)C 10H-308S CN(C)c1ncc(c(n1)c2ccc(c(c2)Cl)Cl)S(=O)(=O)C 10H-309S Cc1ncc(c(n1)c2ccc(c(c2)Cl)Cl)S(=O)(=O)C 10H-310S CS(=O)(=O)c1cnc(nc1c2ccccc2Cl)c3ccccc3 10H-311S CS(=O)(=O)c1cnc(nc1c2ccccc2Cl)c3cccnc3 10H-312S c1ccc(cc1)C(CSc2ccc(cc2)F)(c3ccccc3)O 10H-313S c1ccc(cc1)C(CS(=O)(=O)c2ccc(cc2)F)(c3ccccc3)O 10H-314S c1ccc(cc1)C(CSc2ccc(cc2)Br)(c3ccccc3)O 10H-315S c1ccc(cc1)C(CS(=O)(=O)c2ccc(cc2)Br)(c3ccccc3)O 10H-316S c1ccc(cc1)C(CS(=O)c2ccc(cc2)Br)(c3ccccc3)O 10H-317S c1cc(c(c(c1)Cl)C(=O)Oc2c(ccc(n2)c3ccc(cc3)Cl)C#N)Cl 10H-321S c1ccc(cc1)C(CS(=O)c2ccc(cc2)F)(c3ccccc3)O 10H-322S c1ccc(cc1)C(CS(=O)c2ccc(cc2)Cl)(c3ccccc3)O 10H-323S c1cc(ccc1c2ccc(c(n2)OC(=O)c3ccc(cc3)F)C#N)F 10H-324S c1cc(cc(c1)C(F)(F)F)C(=O)Oc2c(ccc(n2)c3ccc(cc3)F)C#N 10H-325S c1ccc(cc1)CSCC(c2ccccc2)(c3ccccc3)O 10H-327S c1cc(c(c(c1)Cl)C(=O)Oc2c(ccc(n2)c3ccc(cc3)F)C#N)Cl 10H-328S c1ccc(cc1)CS(=O)(=O)CC(c2ccccc2)(c3ccccc3)O 10H-329S c1cc(ccc1C(F)(F)F)Sc2c(nns2)C(=O)O 10H-331S c1ccc(cc1)CS(=O)CC(c2ccccc2)(c3ccccc3)O 10H-335S c1ccc(cc1)C(CS(=O)(=O)c2ccccc2Cl)(c3ccccc3)O 10H-336S Cc1cccc(c1)S(=O)(=O)CC(c2ccccc2)(c3ccccc3)O 10H-337S c1ccc(cc1)C(CS(=O)(=O)c2cccc(c2)Cl)(c3ccccc3)O 10H-338S COC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F 10H-344S c1ccc(cc1)C(CS(=O)(=O)c2cccc(c2)C(F)(F)F)(c3ccccc3)O 10H-345S c1ccc(cc1)C(CSCc2ccc(cc2)Cl)(c3ccccc3)O 10H-346S c1ccc(cc1)C(CSc2c(cccc2Cl)Cl)(c3ccccc3)O 10H-347S c1ccc(cc1)C(CS(=O)c2c(cccc2Cl)Cl)(c3ccccc3)O 10H-348S COC(=O)c1c(ccs1)Oc2ccc(cc2F)[N+](=O)[O-] 10H-349S COc1ccc(cc1OC)c2ccc(c(n2)OC(=O)c3ccc(cc3)F)C#N 10H-350S c1ccc(cc1)C(CS(=O)Cc2ccc(cc2)Cl)(c3ccccc3)O 10H-351S c1ccc(c(c1)S(=O)(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-352S c1cc(ccc1C(CSc2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-356S c1cc(ccc1C(CS(=O)(=O)c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-357S c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2ccsc2C(=O)O 10H-358S Cc1ccc(cc1C)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F 10H-360S c1ccc(cc1)CSCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 10H-362S COC(=O)c1c(ccs1)Oc2ccc(cc2)[N+](=O)[O-] 10H-363S c1cc(ccc1[N+](=O)[O-])Oc2ccsc2C(=O)O 10H-364S c1cc(ccc1CSCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-365S c1cc(ccc1CS(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-366S c1ccc(c(c1)SCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-367S c1ccc(cc1)CS(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 10H-368S COC(=O)c1c(ccs1)Oc2ccccc2[N+](=O)[O-] 10H-369S c1ccc(c(c1)S(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-376S c1cc(cc(c1)Cl)S(=O)(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 10H-377S Cc1cccc(c1)S(=O)(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 10H-380S COC(=O)c1ccc(c(c1)Cl)Cl 10H-383S c1cc(ccc1CS(=O)(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-384S c1cc(ccc1NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-])F 10H-385S COC(=O)c1c(ccs1)NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-] 10H-386S c1cc(cc(c1)NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-])C(F)(F)F 10H-387S C=CCNC(=O)c1c(ccs1)Oc2ccc(cc2)[N+](=O)[O-] 10H-388S CC(=O)Nc1ccc(cc1)NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-] 10H-389S COC(=O)c1c(ccs1)Oc2c(cccn2)[N+](=O)[O-] 10H-390S COC(=O)c1c(ccs1)Oc2ccc(cc2C(F)(F)F)[N+](=O)[O-] 10H-391S c1ccc(c(c1)[N+](=O)[O-])Oc2ccsc2C(=O)O 10H-392S c1ccc(c(c1)[N+](=O)[O-])Oc2ccsc2C(=O)Nc3ccc(cc3F)F 10H-394S c1ccc(c(c1)[N+](=O)[O-])Oc2ccsc2C(=O)Nc3ccc(cc3)C(F)(F)F 10H-395S COc1ccc(c(c1)NC(=O)c2c(ccs2)Oc3ccccc3[N+](=O)[O-])OC 10H-396S c1ccc(c(c1)[N+](=O)[O-])Oc2ccsc2C(=O)Nc3ccc(cc3)Cl 10H-397S Cc1c(cccc1Cl)NC(=O)c2c(ccs2)Oc3ccccc3[N+](=O)[O-] 10H-398S CN(c1ccccc1)C(=O)c2c(ccs2)Oc3ccccc3[N+](=O)[O-] 10H-399S c1cc(c(cc1C(=O)CC#N)Cl)Cl 10H-401S c1cc(ccc1C(C(=O)Nc2ccc(cc2)Br)SCC(=O)O)Cl 10H-402S c1cc(ccc1C2C(=O)N(C(=O)CS2)c3ccc(cc3)Br)Cl 10H-403S c1cc(ccc1C2C(=O)N(C(=O)CS2=O)c3ccc(cc3)Cl)Cl 10H-404S c1cc(ccc1c2ccc(c(=O)[nH]2)C#N)F 10H-405S c1cc(ccc1Cn2c(ccc(c2=O)C#N)c3ccc(cc3)F)Cl 10H-406S c1cc(ccc1Cn2c(ccc(c2=O)C#N)c3ccc(cc3)F)F 10H-407S c1cc(cc(c1)C(F)(F)F)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)F 10H-408S c1ccc(cc1)C2C(=O)N(C(=O)CS2=O)c3ccc(c(c3)Cl)Cl 10H-412S c1cc(ccc1C2C(=O)N(C(=O)CS2=O)c3ccc(cc3)Br)Cl 10H-413S c1cc(ccc1c2ccc(c(=O)n2Cc3ccc(cc3Cl)Cl)C#N)F 10H-414S c1cc(c(c(c1)Cl)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)F)Cl 10H-415S c1cc(c(c(c1)Cl)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)F)F 10H-416S c1cc(ccc1c2ccc(c(=O)n2Cc3ccc(c(c3)Cl)Cl)C#N)F 10H-417S c1cc(cc(c1)F)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)F 10H-418S c1cc(ccc1C(C(=O)Nc2ccc(cc2)C(F)(F)F)SCC(=O)O)Cl 10H-420S c1cc(ccc1C2C(=O)N(C(=O)CS2)c3ccc(cc3)C(F)(F)F)Cl 10H-421S CCOC(=O)Cn1c(ccc(c1=O)C#N)c2ccc(cc2)F 10H-423S CCNC(=O)Nc1ccc(c(c1)Cl)OC 10H-427S c1ccc(cc1)c2ccc(c(n2)Cl)C#N 10H-428S c1ccc(cc1)c2ccc(c(n2)Sc3ccc(cc3)Cl)C#N 10H-431S c1ccc(cc1)c2ccc(c(n2)Sc3ccc(cc3)Br)C#N 10H-433S c1ccc(cc1)c2ccc(c(n2)Sc3ccc(cc3)F)C#N 10H-434S Cc1ccc(cc1)Sc2c(ccc(n2)c3ccccc3)C#N 10H-435S Cc1cccc(c1)Sc2c(ccc(n2)c3ccccc3)C#N 10H-436S CSc1c(ccc(n1)c2ccccc2)C#N 10H-437S CC(C)NC(=O)Nc1ccc(c(c1)Cl)OC 10H-439S C=CCNC(=O)Nc1ccccc1C#N 10H-440S c1ccc2c(c1)C3=NC(CN3C(=O)N2)CBr 10H-442S c1ccc(cc1)C2C(=O)N(C(=O)CS2(=O)=O)c3ccc(c(c3)Cl)Cl 10H-444S c1cc(ccc1C2C(=O)N(C(=O)CS2=O)c3ccc(cc3)C(F)(F)F)Cl 10H-445S CC(C)N1C(C(N(C1=O)c2ccc(c(c2)Cl)OC)O)O 10H-447 c1ccc(cc1)c2ccc(c(n2)Sc3cccc(c3)Cl)C#N 10H-453S c1ccc(cc1)c2ccc(c(n2)Sc3cccc(c3)C(F)(F)F)C#N 10H-454S c1ccc(cc1)c2ccc(c(n2)Oc3ccc(cc3)Cl)C#N 10H-455S c1ccc(cc1)c2ccc(c(n2)Oc3ccc(c(c3)Cl)Cl)C#N 10H-456S c1ccc(cc1)c2ccc(c(n2)Oc3cccc(c3)C(F)(F)F)C#N 10H-457S COc1ccc(cc1Cl)NC(=O)NCC=C 10H-460 c1cc(ccc1c2ccc(c(n2)Cl)C#N)Cl 10H-461S Cc1cccc(c1)Sc2c(ccc(n2)c3ccc(cc3)Cl)C#N 10H-462S c1cc(ccc1c2ccc(c(n2)Sc3ccc(cc3)F)C#N)Cl 10H-463S c1cc(cc(c1)Cl)Sc2c(ccc(n2)c3ccc(cc3)Cl)C#N 10H-467S c1cc(ccc1c2ccc(c(n2)Sc3ccc(cc3)Br)C#N)Cl 10H-468S c1cc(ccc1c2ccc(c(n2)Sc3ccc(cc3)Cl)C#N)Cl 10H-469S c1ccc(cc1)Sc2c(ccc(n2)c3ccc(cc3)Cl)C#N 10H-471S CSc1c(ccc(n1)c2ccc(cc2)Cl)C#N 10H-473S c1cc(ccc1CSc2c(ccc(n2)c3ccc(cc3)Cl)C#N)Cl 10H-474S c1ccc(c(c1)Oc2c(ccc(n2)c3ccc(cc3)Cl)C#N)Cl 10H-475S c1ccc(cc1)Oc2c(ccc(n2)c3ccc(cc3)Cl)C#N 10H-476S c1cc(cc(c1)Oc2c(ccc(n2)c3ccc(cc3)Cl)C#N)C(F)(F)F 10H-477S c1cc(ccc1c2ccc(c(n2)Oc3ccc(cc3)F)C#N)Cl 10H-478S c1cc(ccc1c2ccc(c(n2)Oc3ccc(cc3F)F)C#N)Cl 10H-479S c1cc(c(cc1c2ccc(c(=O)[nH]2)C#N)Cl)Cl 10H-482S c1ccc(c(c1)c2ccc(c(=O)n2Cc3c(cccc3Cl)Cl)C#N)Cl 10H-483S c1ccc(c(c1)c2ccc(c(=O)n2Cc3ccc(c(c3)Cl)Cl)C#N)Cl 10H-484S c1ccc(c(c1)c2ccc(c(=O)n2Cc3c(cccc3Cl)F)C#N)Cl 10H-485S c1ccc(c(c1)c2ccc(c(=O)n2Cc3ccc(cc3)[N+](=O)[O-])C#N)Cl 10H-486S c1ccc(c(c1)c2ccc(c(=O)n2Cc3ccc(cc3Cl)Cl)C#N)Cl 10H-487S c1ccc(c(c1)c2ccc(c(=O)n2Cc3ccc(cc3)Cl)C#N)Cl 10H-489S c1cc(c(c(c1)Cl)Cn2c(ccc(c2=O)C#N)c3ccc(c(c3)Cl)Cl)Cl 10H-495S c1cc(c(cc1Cn2c(ccc(c2=O)C#N)c3ccc(c(c3)Cl)Cl)Cl)Cl 10H-496S c1cc(c(cc1c2ccc(c(=O)n2Cc3ccc(cc3Cl)Cl)C#N)Cl)Cl 10H-497S c1cc(c(c(c1)Cl)Cn2c(ccc(c2=O)C#N)c3ccc(c(c3)Cl)Cl)F 10H-498S c1cc(ccc1Cn2c(ccc(c2=O)C#N)c3ccc(c(c3)Cl)Cl)Cl 10H-499S c1ccc(c(c1)Cn2c(ccc(c2=O)C#N)c3ccc(c(c3)Cl)Cl)Cl 10H-500S c1cc(cc(c1)C(F)(F)F)Cn2c(ccc(c2=O)C#N)c3ccc(c(c3)Cl)Cl 10H-501S Cn1c(ccc(c1=O)C#N)c2ccc(c(c2)Cl)Cl 10H-502S c1cc(c(cc1c2ccc(c(n2)Cl)C#N)Cl)Cl 10H-503S c1cc(ccc1Sc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N)Cl 10H-505S c1cc(ccc1F)Sc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N 10H-506S c1cc(ccc1Sc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N)Br 10H-507S c1cc(cc(c1)Cl)Sc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N 10H-508S c1ccc(c(c1)Oc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N)Cl 10H-509S c1cc(cc(c1)Oc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N)C(F)(F)F 10H-510S c1cc(c(cc1c2ccc(c(n2)Oc3ccc(cc3Cl)Cl)C#N)Cl)Cl 10H-511S c1cc(c(cc1c2ccc(c(n2)Oc3ccc(c(c3)Cl)Cl)C#N)Cl)Cl 10H-512S c1cc(ccc1Oc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N)F 10H-513S c1cc(c(c(c1)Cl)Cl)Oc2c(ccc(n2)c3ccc(c(c3)Cl)Cl)C#N 10H-514S c1cc(c(cc1c2ccc(c(n2)Oc3cc(cc(c3)Cl)Cl)C#N)Cl)Cl 10H-515S c1cc(cc(c1)C(F)(F)F)c2ccc(c(=O)[nH]2)C#N 10H-516S c1cc(ccc1c2ccc(c(n2)Cl)C#N)F 10H-517S c1cc(cc(c1)C(F)(F)F)c2ccc(c(=O)n2Cc3c(cccc3Cl)F)C#N 10H-518S c1cc(cc(c1)C(F)(F)F)c2ccc(c(=O)n2Cc3c(cccc3Cl)Cl)C#N 10H-519S c1cc(cc(c1)C(F)(F)F)c2ccc(c(=O)n2Cc3ccc(cc3Cl)Cl)C#N 10H-520S c1cc(cc(c1)C(F)(F)F)c2ccc(c(=O)n2Cc3ccc(c(c3)Cl)Cl)C#N 10H-521S c1cc(cc(c1)C(F)(F)F)Cn2c(ccc(c2=O)C#N)c3cccc(c3)C(F)(F)F 10H-522S c1cc(cc(c1)Cl)Cn2c(ccc(c2=O)C#N)c3cccc(c3)C(F)(F)F 10H-523S c1cc(cc(c1)C(F)(F)F)c2ccc(c(=O)n2Cc3ccc(cc3)[N+](=O)[O-])C#N 10H-524S c1cc(cc(c1)Cl)Sc2c(ccc(n2)c3ccc(cc3)F)C#N 10H-527S c1cc(ccc1c2ccc(c(n2)Sc3ccc(cc3)Cl)C#N)F 10H-528S c1cc(ccc1c2ccc(c(n2)Sc3ccc(cc3)F)C#N)F 10H-529S c1cc(ccc1c2ccc(c(n2)Sc3ccc(c(c3)Cl)Cl)C#N)F 10H-530S c1cc(ccc1c2ccc(c(n2)Sc3ccc(cc3)Br)C#N)F 10H-531S c1cc(cc(c1)Sc2c(ccc(n2)c3ccc(cc3)F)C#N)C(F)(F)F 10H-532S c1ccc(cc1)CSc2c(ccc(n2)c3ccc(cc3)F)C#N 10H-534S c1ccc(cc1)Sc2c(ccc(n2)c3ccc(cc3)F)C#N 10H-535S COc1ccc(cc1)Sc2c(ccc(n2)c3ccc(cc3)F)C#N 10H-536S CSc1c(ccc(n1)c2ccc(cc2)F)C#N 10H-537S c1cc(ccc1c2ccc(c(n2)Oc3ccc(c(c3)Cl)Cl)C#N)F 10H-538S c1cc(c(c(c1)Cl)Cl)Oc2c(ccc(n2)c3ccc(cc3)F)C#N 10H-539S c1ccc(cc1)Oc2c(ccc(n2)c3ccc(cc3)F)C#N 10H-541S Cc1cc(ccc1Oc2c(ccc(n2)c3ccc(cc3)F)C#N)Cl 10H-542S Cc1cc(cc(c1)Oc2c(ccc(n2)c3ccc(cc3)F)C#N)C 10H-543S c1cc(ccc1c2ccc(c(n2)Oc3ccc(cc3)F)C#N)F 10H-544S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Cl)C#N 10H-545S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Sc3ccc(cc3)Br)C#N 10H-546S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Sc3ccc(cc3)Cl)C#N 10H-547S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Sc3cccc(c3)C(F)(F)F)C#N 10H-548S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Oc3cc(cc(c3)Cl)Cl)C#N 10H-549S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Oc3ccc(c(c3)Cl)Cl)C#N 10H-550S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Oc3ccc(cc3)F)C#N 10H-551S COc1ccc(cc1)c2ccc(c(=O)n2Cc3ccc(cc3)[N+](=O)[O-])C#N 10H-552S COc1ccc(cc1)c2ccc(c(=O)n2Cc3cccc(c3)Cl)C#N 10H-553S COc1ccc(cc1)c2ccc(c(=O)n2Cc3cccc(c3)C(F)(F)F)C#N 10H-554S COc1ccc(cc1)c2ccc(c(=O)n2Cc3ccc(cc3)F)C#N 10H-555S Cc1ccc(cc1)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)OC 10H-556S COc1ccc(cc1)c2ccc(c(=O)n2Cc3cccc(c3)OC)C#N 10H-557S COc1ccc(cc1)c2ccc(c(=O)n2Cc3ccc(c(c3)Cl)Cl)C#N 10H-558S COC(=O)c1c(ccs1)Oc2c(cccc2Cl)[N+](=O)[O-] 10H-601S c1cc(c(cc1[N+](=O)[O-])F)Oc2ccsc2C(=O)O 10H-602S CNC(=O)c1c(ccs1)Oc2ccccc2[N+](=O)[O-] 10H-603S C=CCNC(=O)c1c(ccs1)Oc2ccccc2[N+](=O)[O-] 10H-604S c1cc(c(c(c1)Cl)S(=O)(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-605S COc1ccc(cc1)S(=O)(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 10H-606S COc1ccc(cc1)SCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 10H-607S COc1ccc(cc1)S(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 10H-608S c1cc(ccc1C(CS(=O)c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 10H-609S COC(=O)CNC(=O)c1c(ccs1)Oc2ccccc2[N+](=O)[O-] 10H-610S c1cc(ccc1N2CCC3(CC2)OCC4C(CO3)ON=C4C(=O)NN)[N+](=O)[O-] 10H-900 c1ccnc(c1)N2CCN(CC2)c3c(cc(c(n3)N)C#N)C#N 10H-901 CN(C)/C=N/c1c(cc(c(n1)N2CCN(CC2)c3ccccn3)C#N)C#N 10H-904 c1cc(ccc1C2=NC=C3C(S2)C(=O)N(C3=O)CCNc4c(cc(cn4)C(F)(F)F)Cl)Cl 10H-907 c1cc(cc(c1)N2C(=O)C3C(=CN=C(S3)c4ccc(cc4)Cl)C2=O)C(F)(F)F 10H-908 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C(=CN=C(S3)c4ccc(cc4)Cl)C2=O 10H-909 CN(C)/C=N\C(=S)Nc1c(cc(cn1)C(F)(F)F)Cl 10H-910 CC(=O)C1=NOC2C1C(=O)N(C2=O)N(C)c3c(cc(cn3)C(F)(F)F)Cl 10H-911 CN(c1c(cc(cn1)C(F)(F)F)Cl)N/C(=C/C#N)/N 10H-912 CN(c1c(cc(cn1)C(F)(F)F)Cl)N/C(=C/C#N)/NC(=O)Nc2ccc(cc2)Cl 10H-913 CCOC(=O)c1c(con1)C(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 10H-914 Cc1c(c2ccccc2n1CCOc3ccc(cc3Cl)Cl)c4c(cc(cn4)C(F)(F)F)Cl 10H-915 Cc1c(c2ccccc2n1Cc3ccc(cc3)C(F)(F)F)c4c(cc(cn4)C(F)(F)F)Cl 10H-916 CCOC(=O)/C=C(\NC(=O)Nc1ccc(cc1Cl)Cl)/NN(C)c2c(cc(cn2)C(F)(F)F)Cl 10H-917 Cc1c(c2ccccc2n1Cc3ccc(cc3)Cl)c4c(cc(cn4)C(F)(F)F)Cl 10H-918 c1cc(ccc1C2=NC=C3C(S2)C(=O)N(C3=O)c4ccc(cc4)Cl)Cl 10H-920 Cc1ccc(cc1)NC(=O)N/C(=C\C#N)/N2CCN(CC2)c3ccc(cc3)OC 10H-921 CCCCOC1CC(N(O1)C)c2ccc(c(c2)OC)OCc3ccc(cc3)OC 10H-922 CN(c1c(cc(cn1)C(F)(F)F)Cl)N/C(=C/C#N)/NC(=O)Nc2cccc(c2)C(F)(F)F 10H-924 CC(C)(C)NC(=O)N/C(=C\C#N)/NN(C)c1c(cc(cn1)C(F)(F)F)Cl 10H-925 CC(=O)C1=NOC2C1C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 10H-926 CC1(OCCO1)c2ccc3c(c2)c(on3)c4ccc(cc4)Cl 10H-927 CC(=O)c1ccc2c(c1)c(on2)c3ccc(cc3)Cl 10H-928 CCOC(=O)/C=C(/NC(=O)NC1CCCCC1)\N2CCN(CC2)c3ccc(cc3)OC 10H-929 CCOC(=O)/C=C(\NC(=O)Nc1ccc(cc1)C)/N2CCN(CC2)c3ccc(cc3)OC 10H-930 c1ccc2c(c1)cc(n2c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)NNC(=S)Nc4cccc(c4)C(F)(F)F 10H-931 CCCCOC1CC(N(O1)C)c2ccc(c(c2)OC)OCc3ccc(cc3)F 10H-932 CCCCOC1CC(N(O1)C)c2ccc(c(c2)OC)OCc3ccc(cc3)Cl 10H-933 CC1(NC(=O)N(N1)c2ccccc2)C3=NOC4C3C(=O)N(C4=O)N(C)c5c(cc(cn5)C(F)(F)F)Cl 10H-935 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)Nc4ccc(cc4Cl)Cl 10H-936 CN(C)/C=C/C(=O)c1ccc2c(c1)c(on2)c3ccc(cc3)Cl 10H-937 CC1(NC(=O)N(N1)c2ccccc2)c3ccc4c(c3)c(on4)c5ccc(cc5)Cl 10H-940 CC(=O)C1=NOC2C1COC(OC2)c3ccccc3 10H-941 CCOC(=O)/C=C(\NC(=O)NC(C)(C)C)/NN(C)c1c(cc(cn1)C(F)(F)F)Cl 10H-942 c1ccc(cc1)n2c(ccn2)c3ccc4c(c3)c(on4)c5ccc(cc5)Cl 10H-943 CCOC(=O)c1c(con1)C(=O)c2ccc3c(c2)c(on3)c4ccc(cc4)Cl 10H-945 c1ccc(c(c1)C2OCC=CCO2)F 10H-946 CN(C)/C=C(/c1c[nH]c2c1cccc2)\C(=O)OC 10H-947 C/C(=N/Nc1c(cc(cn1)C(F)(F)F)Cl)/C2=NOC3C2C(=O)N(C3=O)N(C)c4c(cc(cn4)C(F)(F)F)Cl 10H-948 CCOC(=O)NC1Cc2ccccc2C1Cl 10H-949 c1ccc2c(c1)c(c(n2c3c(cc(cn3)C(F)(F)F)Cl)CSc4c(cc(cn4)C(F)(F)F)Cl)Br 10H-950 CCOC(=O)NC1Cc2ccccc2C1Sc3ccc(cc3)Cl 10H-951 c1ccc2c(c1)cc(n2c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)NCCNc4c(cc(cn4)C(F)(F)F)Cl 10H-952 c1cc(c(cc1Cl)Cl)C2OCC(C(CO2)Br)Br 10H-953 c1c(cnc(c1Cl)N2CCC3(CC2)OCC(C(CO3)Br)Br)C(F)(F)F 10H-954 CN(C)c1nc(c(c(=O)o1)C#N)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 10H-955 CCOC(=O)C(=CNCCNc1c(cc(cn1)C(F)(F)F)Cl)C(=O)OCC 10H-957 c1ccnc(c1)C(=O)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 10J-001 CCOC(=O)C(C(F)(F)F)(NNc1c(cc(cn1)C(F)(F)F)Cl)O 10J-002 c1ccc2c(c1)nc(c(n2)Cl)C(F)(F)F 10J-003 c1ccc(cc1)Sc2ccc(cc2)c3ccnc(n3)N 10J-004 c1ccc(cc1)Sc2ccc(cc2)c3ccn[nH]3 10J-009 c1ccc(cc1)Sc2ccc(cc2)c3ccnn3c4c(cc(cn4)C(F)(F)F)Cl 10J-010 CC(C)(CNC(=O)Nc1ccccc1)SCc2ccc(cc2)Cl 10J-011 c1ccc(cc1)NC(=O)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 10J-013 CN(C)CCCNC(=O)CCc1c(cc(cn1)C(F)(F)F)Cl 10J-014 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)Nc4ccc(cc4)OC(F)(F)F 10J-015 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)Nc4ccc(cc4)F 10J-016 COc1ccc(cc1)NC(=O)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 10J-017 c1ccc2c(c1)nc(c(n2)N3CCOCC3)C(F)(F)F 10J-018 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)Nc4ccc(cc4)C#N 10J-019 CC(C)(C)NC(=O)CCc1c(cc(cn1)C(F)(F)F)Cl 10J-022 CCC(=O)c1ccc2c(c1)ccc(c2Br)OC 10J-023 c1c(cnc(c1Cl)CCC(=O)N2CCOCC2)C(F)(F)F 10J-026 CN1CCN(CC1)C(=O)CCc2c(cc(cn2)C(F)(F)F)Cl 10J-028 CN1CCN(CC1)C(=O)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 10J-031 c1ccc(cc1)CNC(=O)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 10J-032 CN(C)/C=N\C(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3cccs3 10J-033 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2c4nc[nH]n4 10J-034 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)N4CCOCC4 10J-035 CC(=O)c1ccc(cc1)Oc2cccc(c2C#N)Cl 10J-036 CN(C)/C=C\C(=O)c1ccc(cc1)Oc2cccc(c2C#N)Cl 10J-037 c1ccc2c(c1)nc(s2)c3cccnc3Sc4ccc(cc4)Cl 10J-301S c1ccc2c(c1)nc(s2)c3cccnc3Sc4cccc(c4)C(F)(F)F 10J-302S CCCCCCn1c2ccc(cc2nc1c3ccc(nc3)Cl)C(F)(F)F 10J-303S c1ccc2c(c1)nc(s2)c3cccnc3Sc4ccc(cc4)F 10J-304S Cn1c2ccccc2nc1c3ccc(nc3)Cl 10J-308S COc1ccc(cc1)Cn2c3ccccc3nc2c4ccc(nc4)Cl 10J-309S c1ccc2c(c1)nc(n2Cc3cccc(c3)C(F)(F)F)c4ccc(nc4)Cl 10J-310S CC(C)n1c2ccc(cc2nc1c3ccc(nc3)Cl)C(F)(F)F 10J-311S c1cc(c(nc1)Cl)c2[nH]c3cc(c(cc3n2)Cl)Cl 10J-312S c1ccc2c(c1)nc(s2)c3cc(c[nH]c3=O)Cl 10J-315S c1ccc(cc1)Cn2cccc(c2=O)c3nc4ccccc4s3 10J-316S CCCCCCn1c2ccccc2nc1c3ccc(nc3)Cl 10J-317S Cc1cc2c(cc1C)n(c(n2)c3ccc(nc3)Cl)C 10J-318S CCCn1c(=O)cc(nc1SCc2ccc(cc2)C(C)(C)C)C(F)(F)F 10J-321S c1ccc2c(c1)nc(s2)c3cccn(c3=O)Cc4ccc(cc4Cl)Cl 10J-322S c1ccc2c(c1)nc(s2)c3cccn(c3=O)Cc4ccc(cc4)Cl 10J-323S Cc1ccc(cc1)Cn2cccc(c2=O)c3nc4ccccc4s3 10J-324S Cc1cc2c(cc1C)n(c(n2)c3ccc(nc3)Cl)Cc4ccc(cc4)Cl 10J-325S Cc1cc2c(cc1C)n(c(n2)c3ccc(nc3)Cl)Cc4ccccc4 10J-329S CC(C)c1c(snn1)C(=O)OC 10J-333S Cc1cc2c(cc1C)n(c(n2)c3ccc(nc3)Cl)Cc4ccc(cc4)OC 10J-334S Cc1ccc(cc1)Cn2c3cc(c(cc3nc2c4ccc(nc4)Cl)C)C 10J-335S c1ccc(cc1)Oc2c(cccn2)c3nc4ccccc4s3 10J-336S CCCCOc1c(cccn1)c2nc3ccccc3s2 10J-337S CC(C)c1c(snn1)C(=O)O 10J-338S c1ccc2c(c1)nc(s2)c3cccnc3Oc4ccc(cc4)Cl 10J-339S Cc1cc2c(cc1C)n(c(n2)c3ccc(nc3)Cl)Cc4ccc(c(c4)Cl)Cl 10J-344S COc1ccc(c[n+]1[O-])NC(=O)c2ccccc2 10J-345S CCOC(=O)Cn1c2cc(c(cc2nc1c3cccnc3Cl)Cl)Cl 10J-346S C=CCn1c2cc(c(cc2nc1c3cccnc3Cl)Cl)Cl 10J-347S c1ccc(c(c1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl)F 10J-348S c1cc(cc(c1)Cl)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 10J-349S c1ccc(c(c1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl)Cl 10J-350S c1cc(c(nc1)Cl)c2nc3cc(c(cc3n2Cc4ccc(cc4)Cl)Cl)Cl 10J-351S c1cc(c(nc1)Cl)c2nc3cc(c(cc3n2Cc4ccc(c(c4)Cl)Cl)Cl)Cl 10J-355S c1cc(cc(c1)C(F)(F)F)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 10J-356S c1cc2c(cc1Cl)nc([nH]2)c3ccc(nc3)Cl 10J-357S c1cc(ccc1/C(=N/O)/N)Cl 10J-360S c1cc(c(c(c1)Cl)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl)F 10J-362S Cn1c2cc(c(cc2nc1c3ccc(nc3)Cl)Cl)Cl 10J-363S COc1ccc(c[n+]1[O-])NC(=O)c2cccc(c2)Cl 10J-364S c1cc(cc(c1)Cl)c2nc(on2)c3ccc(nc3)Cl 10J-365S c1cc(ccc1c2nc(on2)c3ccc(nc3)Cl)Cl 10J-366S c1cc(cc(c1)C(F)(F)F)/C(=N/O)/N 10J-367S c1cc(cc(c1)C(F)(F)F)c2nc(on2)c3ccc(nc3)Cl 10J-369S c1cc(ccc1c2nc(on2)c3ccc(nc3)Cl)C(F)(F)F 10J-370S c1cc(cc(c1)Cl)c2c(cc(nc2Cl)O)O 10J-371S c1cc(c(=O)[nH]c1)c2nc3ccc(cc3s2)Cl 10J-374S Cc1ccc(cc1)c2c(c(c3n2CSC3)C(=O)OC)C(=O)OC 10J-502S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)Cl)CSC2 10J-504S Cc1ccc(cc1)c2c(c(c3n2CS(=O)C3)C(=O)OC)C(=O)OC 10J-505S Cc1ccc(cc1)c2c(c(c3n2CS(=O)(=O)C3)C(=O)OC)C(=O)OC 10J-506S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)Cl)CS(=O)C2 10J-507S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)Cl)CS(=O)(=O)C2 10J-508S CC(C)(C)c1ccc(cc1)c2c(c(c3n2CS(=O)C3)C(=O)OC)C(=O)OC 10J-509S CC(C)(C)c1ccc(cc1)c2c(c(c3n2CS(=O)(=O)C3)C(=O)OC)C(=O)OC 10J-510S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)F)CSC2 10J-511S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)Br)CSC2 10J-512S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)F)CS(=O)C2 10J-513S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)F)CS(=O)(=O)C2 10J-514S COC(=O)c1c2n(c(c1C(=O)OC)c3cc(cc(c3)Cl)Cl)CS(=O)C2 10J-516S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)Br)CS(=O)C2 10J-518S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)Br)CS(=O)(=O)C2 10J-519S CCOC(=O)c1c(nns1)C 10J-523S Cc1c(snn1)C(=O)O 10J-524S CCCn1c(=O)cc(nc1SCc2cccc(c2)Cl)C(F)(F)F 10J-527S CCCn1c(=O)cc(nc1SCc2ccccc2F)C(F)(F)F 10J-528S CCCn1c(=O)cc(nc1SCc2c(cccc2Cl)Cl)C(F)(F)F 10J-529S CCCn1c(=O)cc(nc1SCc2ccc(cc2)C)C(F)(F)F 10J-530S CCCn1c(=O)cc(nc1SCc2ccc(cc2)[N+](=O)[O-])C(F)(F)F 10J-531S CCCn1c(=O)cc(nc1SCc2cccc(c2)OC)C(F)(F)F 10J-533S CCCn1c(=O)cc(nc1SCc2cccc(c2)C#N)C(F)(F)F 10J-535S c1ccc(cc1)C(=O)c2cc3ccccc3o2 10J-537S COc1cccc(c1)C(=O)NCCSc2ccc(cc2)F 10J-538S COc1cc(cc(c1OC)OC)C(=O)NCCSc2ccc(cc2)F 10J-539S COc1cccc(c1)C(=O)NCCSc2ccc(cc2)Br 10J-541S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)C(F)(F)F)CSC2 10J-545S COc1cc(cc(c1OC)OC)C(=O)NCCSc2ccc(cc2)Br 10J-546S CCn1c(=O)cc([nH]c1=O)C(F)(F)F 10J-547S C=CCn1c(=O)cc([nH]c1=O)C(F)(F)F 10J-548S c1ccc(c(c1)n2c(=O)cc([nH]c2=O)C(F)(F)F)Cl 10J-550S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)C(F)(F)F)CS(=O)C2 10J-551S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)C(F)(F)F)CS(=O)(=O)C2 10J-552S CC(C)(C)c1ccc(cc1)c2c(c(c3n2CSC3)C(=O)O)C(=O)O 10J-554S c1cc(ccc1c2c(c(c3n2CSC3)C(=O)O)C(=O)O)Br 10J-555S Cc1ccc(cc1)c2c(c(c3n2CSC3)C(=O)O)C(=O)O 10J-556S c1cc(cc(c1)Cl)n2c(=O)cc([nH]c2=O)C(F)(F)F 10J-559S CCCn1c(=O)cc([nH]c1=O)C(F)(F)F 10J-561S c1c([nH]c(=O)n(c1=O)C2CCCCC2)C(F)(F)F 10J-562S CCOCCOc1ccc2ccccc2n1 10J-565S Cc1ccc2c(c1)nc(o2)c3cccnc3Cl 10J-567S CNc1c(cccn1)c2nc3cc(ccc3o2)Cl 10J-568S c1cc(cc(c1)n2c(=O)cc([nH]c2=O)C(F)(F)F)C(F)(F)F 10J-569S C=CCNc1c(cccn1)c2nc3cc(ccc3o2)Cl 10J-570S Cc1ccc2c(c1)nc(o2)c3cccnc3NC 10J-571S CCCNc1c(cccn1)c2nc3cc(ccc3o2)C 10J-574S c1cc(c(cc1c2c(c(c3n2CSC3)C(=O)O)C(=O)O)Cl)Cl 10J-576S CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3ccc(cc3)OC)c4c(ccs4)Cl 10J-900 c1cc2c(cc1C(F)(F)F)[nH]c(=O)c(=O)n2CCNc3c(cc(cn3)C(F)(F)F)Cl 10J-901 c1ccnc(c1)NC(=O)CC(=O)Nc2ccccn2 10J-902 CN(C)C=C(C(=O)Nc1ccccn1)C(=O)Nc2ccccn2 10J-903 c1cc(cnc1)NC(=O)CC(=O)Nc2cccnc2 10J-904 c1cc2c(cc1C(F)(F)F)nc(c(=O)n2CCNc3c(cc(cn3)C(F)(F)F)Cl)Cl 10J-905 c1cc2c(cc1C(F)(F)F)nc(c(=O)n2CCNc3c(cc(cn3)C(F)(F)F)Cl)NN 10J-906 c1cc2c(cc1C(F)(F)F)n3cnnc3c(=O)n2CCNc4c(cc(cn4)C(F)(F)F)Cl 10J-907 CCOC(=O)CSc1c(=O)n(c2ccc(cc2n1)C(F)(F)F)CCNc3c(cc(cn3)C(F)(F)F)Cl 10J-908 CO/N=C/C(C(=O)Nc1cccnc1)C(=O)Nc2cccnc2 10J-910 CN(C=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl)OC 10J-912 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)N3CCCCC3)Cl 10J-913 c1cc(ccc1N2CCN(CC2)C(=O)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-])Cl 10J-914 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)C(F)(F)F)Cl 10J-915 Cc1c(c(no1)C#N)C(=O)Nc2ccc(cc2)F 10J-916 CC(=O)CC(=O)Nc1ccc(cc1)C(F)(F)F 10J-917 CC(=O)CC(=O)Nc1ccccc1C(F)(F)F 10J-918 CC(=O)CC(=O)Nc1ccccn1 10J-919 CC(=O)O/C(=C(\C=N/OC)/C(=O)Nc1ccc(cc1)C(F)(F)F)/Nc2ccc(cc2)C(F)(F)F 10J-920 c1ccc(cc1)c2c3cc(ccc3[nH]c2C(F)(F)F)Cl 10J-921 c1ccc(cc1)c2c3cc(ccc3n(c2C(F)(F)F)Cc4ccc(cc4)[N+](=O)[O-])Cl 10J-922 C/C(=C\C(=O)Nc1ccc(cc1)C(F)(F)F)/N2CCCC2 10J-923 C/C(=C\C(=O)Nc1ccccc1C(F)(F)F)/N2CCCC2 10J-924 C/C(=C/C(=O)Nc1cccc(c1)Cl)/N2CCCC2 10J-925 C/C(=C\C(=O)Nc1ccccn1)/N2CCCC2 10J-927 C/C(=C\C(=O)N(C)c1ccccc1)/N2CCCC2 10J-928 CN(C=C(C(=O)Nc1ccc(cc1)C(F)(F)F)C(=O)Nc2ccc(cc2)C(F)(F)F)OC 10J-929 CC(=O)CC(=O)Nc1ccc(cc1)C(=O)OC 10J-930 Cc1c(c(no1)C(=O)N)C(=O)OC 10J-931 Cc1cc(c(c(=O)o1)/C(=N\Nc2nc(cs2)c3c(ccs3)Cl)/C)O 10J-932 Cc1c(c(n(n1)c2nc(cs2)c3c(ccs3)Cl)O)C(=O)CC(=O)C 10J-933 Cc1c(c(no1)C#N)C(=O)Nc2cccc(c2)Cl 10J-934 Cc1c(c(no1)C#N)C(=O)Nc2ccc(cc2)C(F)(F)F 10J-935 Cc1c(c(no1)C#N)C(=O)Nc2ccccc2C(F)(F)F 10J-936 C/C(=C\C(=O)Nc1ccc(cc1)C(=O)OC)/N2CCCC2 10J-937 C/C(=C\C(=O)Nc1ccc(cc1)OC)/N2CCCC2 10J-938 Cc1ccc(cc1)NC(=O)/C=C(\C)/N2CCCC2 10J-939 Cc1cc(n(n1)c2ccc(cc2)Cl)C(F)(F)Cl 10J-940 c1cc(ccc1N2CCN(CC2)c3c(cc([nH]3)c4c(ccs4)Cl)C#N)F 10J-941 c1csc(c1Cl)c2cc(c([nH]2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C#N 10J-942 Cc1cc([nH]n1)C(F)(F)Cl 10J-943 Cc1ccc(cc1)NC(=O)c2c(onc2C#N)C 10J-944 Cc1c(c(no1)C#N)C(=O)Nc2ccc(cc2)C(=O)OC 10J-945 c1ccc(cc1)C\2c3ccccc3C(=O)/C2=C\Nc4ccc(cc4)Cl 10K-001 Cc1ccc(cc1)/C=C\2/C(c3cccc(c3C2=O)F)c4ccccc4 10K-002 Cc1ccc(cc1)/C=C\2/C(c3cccc(c3C2=O)Oc4ccc(cc4)Cl)c5ccccc5 10K-003 COc1ccc(cc1)/C=C\2/C(c3cccc(c3C2=O)F)c4ccccc4 10K-004 Cc1ccsc1/C=C\2/C(c3cccc(c3C2=O)F)c4ccccc4 10K-006 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C\c4cccs4)F 10K-007 Cc1ccsc1/C=C\2/C(c3cccc(c3C2=O)Oc4ccc(cc4)Cl)c5ccccc5 10K-009 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C\c4cc(ccc4F)F)Oc5ccc(cc5)Cl 10K-010 COc1ccc(cc1)Oc2cccc3c2C(=O)/C(=C/c4ccc(cc4)Cl)/C3c5ccccc5 10K-011 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C\c4cccc(c4)Br)Oc5ccc(cc5)Cl 10K-012 Cc1ccc(cc1)/C=C\2/C(c3ccccc3C2=O)c4ccccc4 10K-013 Cc1ccc(c(c1)N/C=C/2\C(c3cccc(c3C2=O)Oc4ccc(cc4)Cl)c5ccccc5)C 10K-014 CO/N=C/C1C(c2cccc(c2C1=O)Oc3ccc(cc3)Cl)c4ccccc4 10K-015 CC(=O)C(/C=N/OCc1cccc(c1)C(F)(F)F)c2ccc(c(c2)OC)OC 10K-016 c1ccc(cc1)C(=O)c2ccc(cc2)C(C#N)c3ccc(cc3)F 10K-017 c1ccc(cc1)C(=O)c2ccc(cc2)C(c3ccc(cc3)F)C(=O)N 10K-018 COc1ccc(cc1)/C=C\2/C(c3cccc(c3C2=O)Oc4ccc(cc4)OC)c5ccccc5 10K-019 Cc1ccsc1/C=C\2/C(c3cccc(c3C2=O)Oc4ccc(cc4)OC)c5ccccc5 10K-020 COc1ccc(cc1)Oc2cccc3c2C(=O)/C(=C\c4ccco4)/C3c5ccccc5 10K-021 CN(C)c1ccc(cc1)/C=C/C=C/2\C(c3cccc(c3C2=O)Oc4ccc(cc4)OC)c5ccccc5 10K-022 COc1ccc(cc1)Oc2cccc3c2C(=O)/C(=C\c4ccc(cc4)F)/C3c5ccccc5 10K-023 COc1ccc(cc1)Oc2cccc3c2C(=O)C(=C3c4ccccc4)Cc5ccccn5 10K-024 Cc1ccc(cc1)/C=C\2/C(c3cccc(c3C2=O)Oc4ccc(cc4)OC)c5ccccc5 10K-025 COc1ccc(cc1)Oc2cccc3c2C(=O)/C(=C\c4cccs4)/C3c5ccccc5 10K-026 COc1ccc(cc1)Oc2cccc3c2C(=O)C(=C3c4ccccc4)Cc5ccncc5 10K-027 C/C(=N\Oc1cccc(n1)O/N=C(/C)\c2ccccc2)/c3ccccc3 10K-028 C/C(=N/Oc1nc(ccc1)O/N=C(\c2ccc(cc2)Oc3ccccc3)/C)/c4ccc(cc4)Oc5ccccc5 10K-029 CN(C)/C=N/C(=O)C(c1ccc(cc1)C(=O)c2ccccc2)c3ccc(cc3)F 10K-030 CO/N=C/NC(=O)C(c1ccc(cc1)C(=O)c2ccccc2)c3ccc(cc3)F 10K-031 c1ccc(cc1)C(=O)c2ccc(cc2)C(c3ccc(cc3)F)C(=O)/N=C/Nc4ccc(cc4)Cl 10K-032 C/C(=N\Oc1nc(ccc1)O/N=C(/c2ccc(cc2)F)\C)/c3ccc(cc3)F 10K-034 C/C(=N\Oc1nc(ccc1)O/N=C(/c2ccc(cc2)Cl)\C)/c3ccc(cc3)Cl 10K-035 Cc1nnc(n1N)n2c(ccn2)c3ccc(cc3Cl)Cl 10K-036 COc1ccc(cc1)Oc2cccc3c2C(CC3c4ccccc4)O 10K-037 CN(C)/C=C\1/C(c2cccc(c2C1=O)Oc3ccc(cc3)OC)c4ccccc4 10K-038 Cc1nnc(n1N)n2c(ccn2)c3ccc(cc3)OC 10K-039 c1ccc(cc1)C\2c3ccccc3C(=O)/C2=C\c4ccco4 10K-041 c1ccc(cc1)C2=C(C(=O)c3c2cccc3)Cc4ccccc4C(F)(F)F 10K-042 Cc1ccsc1/C=C\2/C(c3ccccc3C2=O)c4ccccc4 10K-043 c1ccc(cc1)C\2c3ccccc3C(=O)/C2=C\c4cc(ccc4F)F 10K-044 CN(C)c1ccc(cc1)/C=C\2/C(c3ccccc3C2=O)c4ccccc4 10K-045 CCOC(=O)C1CC(=NNC1=O)c2ccc(cc2)Cl 10K-046 CCOC(=O)C1CC(=NNC1=O)c2ccc(c(c2)Cl)Cl 10K-047 COC(=O)CSc1cccc2c1C(=O)CC2c3ccccc3 10K-048 c1ccc(cc1)C2CC(c3c2cccc3Oc4ccc(cc4)Cl)O 10K-049 c1ccc(cc1)C2CC(c3c2cccc3Oc4ccccc4)O 10K-050 COc1ccc(cc1)c2cc3c(nn2)-c4ccccc4C3=O 10K-051 c1ccc2c(c1)-c3c(cc(nn3)c4ccc(cc4)F)C2=O 10K-052 CN(C)c1ccc(cc1)/C=C/C=C\2/C(c3ccccc3C2=O)c4ccccc4 10K-053 COc1ccc(cc1OC)/C=C\2/C(c3ccccc3C2=O)c4ccccc4 10K-054 c1ccc(cc1)Oc2ccc(cc2)c3cc4c(nn3)-c5ccccc5C4=O 10K-055 c1ccc2c(c1)-c3c(cc(nn3)c4ccc(cc4)Cl)C2=O 10K-056 c1ccc(cc1)c2cc3c(nn2)-c4ccccc4C3=O 10K-057 COc1ccc(cc1OC)/C=C\2/C(c3cccc(c3C2=O)Oc4ccc(cc4)Cl)c5ccccc5 10K-058 COc1ccccc1/C=C\2/C(c3ccccc3C2=O)c4ccccc4 10K-059 COc1ccc(cc1OC)/C=C\2/C(c3cccc(c3C2=O)Oc4cccc(c4)C(F)(F)F)c5ccccc5 10K-060 c1ccc(cc1)C2CC(c3c2cccc3Oc4cccc(c4)C(F)(F)F)O 10k-062 c1ccc(cc1)C2CC(c3c2cccc3)O 10K-063 COc1ccc(cc1OC)c2cc3c(nn2)-c4ccccc4C3=O 10K-064 c1ccc2c(c1)-c3c(cc(nn3)c4cccs4)C2=O 10K-065 c1ccc(cc1)c2nnc(s2)N 10K-301S c1ccc(cc1)Oc2c(cc3ccccc3n2)c4cccc(c4)C(F)(F)F 10K-302S c1ccc2c(c1)cc(c(n2)Oc3ccc(cc3)Cl)c4cccc(c4)C(F)(F)F 10K-303S c1ccc2c(c1)cc(c(n2)Oc3ccc(cc3Cl)Cl)c4cccc(c4)C(F)(F)F 10K-304S c1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2ccccn2 10K-306S c1ccc(c(c1)N(CC(=O)O)S(=O)(=O)c2cc(ccc2Cl)Cl)Cl 10K-307S CCOC(=O)CN(c1ccccn1)S(=O)(=O)c2ccc(cc2)OC 10K-308S CCOC(=O)CN(c1ccccc1Cl)S(=O)(=O)c2ccc(cc2)F 10K-309S c1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2cccc(c2)C(F)(F)F 10K-310S c1ccc2c(c1)cc(c(n2)Oc3ccc(cc3)F)c4cccc(c4)C(F)(F)F 10K-311S c1ccc2c(c1)cc(c(n2)Oc3ccc(cc3)[N+](=O)[O-])c4cccc(c4)C(F)(F)F 10K-317S c1ccc2c(c1)cc(c(n2)Oc3cccc(c3)C(F)(F)F)c4cccc(c4)C(F)(F)F 10K-319S c1ccc2c(c1)cc(c(n2)Oc3ccc(cc3F)F)c4cccc(c4)C(F)(F)F 10K-320S Cc1cc(cc(c1)Oc2c(cc3ccccc3n2)c4cccc(c4)C(F)(F)F)C 10K-321S COc1ccc(cc1)Oc2c(cc3ccccc3n2)c4cccc(c4)C(F)(F)F 10K-322S c1ccc(cc1)/C=C/C(=O)CCC(=O)O 10K-323S c1ccc(cc1)/C=C/C2=NNC(=O)CC2 10K-324S c1ccc(cc1)CN2C(=O)CCC(=N2)/C=C/c3ccccc3 10K-325S CN1C(=O)CCC(=N1)/C=C/c2ccccc2 10K-326S C=CCN1C(=O)CCC(=N1)/C=C/c2ccccc2 10K-327S COc1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2ccccn2 10K-328S c1ccc(c(c1)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)F)Cl 10K-329S c1ccc(cc1)NC(=O)CN(c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 10K-330S CN(C)C(=O)CN(c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl 10K-331S C=CCNC(=O)CN(c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl 10K-332S COc1ccc(cn1)NC(=O)/C(=C(\SCc2ccc(cc2)Cl)/Cl)/Cl 10K-336S COc1ccc(cn1)NC(=O)/C(=C(\SCc2ccccc2Cl)/Cl)/Cl 10K-337S COc1ccc(cn1)NC(=O)/C(=C(\SCc2cccc(c2)C(F)(F)F)/Cl)/Cl 10K-338S Cc1ccc(cc1)CS/C(=C(\C(=O)Nc2ccc(nc2)OC)/Cl)/Cl 10K-339S COc1ccc(cc1)CS/C(=C(\C(=O)Nc2ccc(nc2)OC)/Cl)/Cl 10K-340S c1cc(ccc1N(CC(=O)N2CCCC2)S(=O)(=O)c3ccc(cc3)Cl)Cl 10K-341S c1ccc(cc1)CNC(=O)CN(c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 10K-342S c1ccnc(c1)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)Cl 10K-343S CCOC(=O)CN1C(=O)CCC(=N1)/C=C/c2ccccc2 10K-345S c1cc(cc(c1)N(CC(=O)O)S(=O)(=O)c2ccc(cc2Cl)Cl)C(F)(F)F 10K-346S CN(C)C(=O)CN(c1ccccc1Cl)S(=O)(=O)c2cc(ccc2Cl)Cl 10K-347S c1ccc(cc1)NC(=O)CN(c2ccccc2Cl)S(=O)(=O)c3cc(ccc3Cl)Cl 10K-348S COc1ccc(cc1)NC(=O)CN(c2ccccc2Cl)S(=O)(=O)c3cc(ccc3Cl)Cl 10K-349S COc1ccc(cc1)NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl 10K-350S CN(C)C(=O)CN(c1cccc(c1)C(F)(F)F)S(=O)(=O)c2ccc(cc2)Cl 10K-351S C=CCNC(=O)CN(c1cccc(c1)C(F)(F)F)S(=O)(=O)c2ccc(cc2)Cl 10K-352S c1ccc(cc1)NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl 10K-353S c1ccc(c(c1)NC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl)F 10K-354S COc1ccc(cn1)NC(=O)/C(=C(\S(=O)Cc2ccccc2)/Cl)/Cl 10K-356S COc1ccc(cn1)NC(=O)/C(=C(\S(=O)(=O)Cc2ccccc2)/Cl)/Cl 10K-357S COc1ccc(cn1)NC(=O)/C(=C(\S(=O)Cc2ccc(cc2)Cl)/Cl)/Cl 10K-359S COc1ccc(cc1)CS(=O)/C(=C(\C(=O)Nc2ccc(nc2)OC)/Cl)/Cl 10K-360S c1cc(cc(c1)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F 10K-361S Cc1ccc(cc1)CS(=O)/C(=C(\C(=O)Nc2ccc(nc2)OC)/Cl)/Cl 10K-362S c1ccc(cc1)/C=C/c2ccc(nn2)O 10K-364S c1ccc(cc1)Cn2c(=O)ccc(n2)/C=C/c3ccccc3 10K-365S c1ccc(cc1)CNC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccccc3 10K-366S c1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2cccc(c2)C(F)(F)F)c3cccc(c3)C(F)(F)F 10K-367S Cc1ccc(cc1)CS(=O)(=O)/C(=C(\C(=O)Nc2ccc(nc2)OC)/Cl)/Cl 10K-368S COc1ccc(cn1)NC(=O)/C(=C(\S(=O)(=O)Cc2ccc(cc2)Cl)/Cl)/Cl 10K-369S COc1cccc(n1)NC(=O)/C(=C(\S(=O)(=O)Cc2ccccc2Cl)/Cl)/Cl 10K-370S COc1ccc(cc1)CS(=O)(=O)/C(=C(\C(=O)Nc2ccc(nc2)OC)/Cl)/Cl 10K-371S COc1ccc(cn1)NC(=O)/C(=C(\S(=O)Cc2ccccc2Cl)/Cl)/Cl 10K-372S CN(C)C(=O)CN(c1cccc(c1)C(F)(F)F)S(=O)(=O)c2ccccc2 10K-373S c1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(cc2Cl)Cl)c3cccc(c3)C(F)(F)F 10K-374S c1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2ccc(cc2)Cl 10K-376S CN(C)C(=O)CN(c1ccc(cc1)Cl)S(=O)(=O)c2ccccc2 10K-378S C=CCNC(=O)CN(c1ccc(cc1)Cl)S(=O)(=O)c2ccccc2 10K-379S c1ccc(cc1)NC(=O)CN(c2ccc(cc2)Cl)S(=O)(=O)c3ccccc3 10K-383S c1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)c3ccc(cc3)Cl 10K-384S c1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(c(c2)F)F)c3ccc(cc3)Cl 10K-385S c1ccc(cc1)S(=O)(=O)N(CC(=O)N2CCOCC2)c3ccc(cc3)Cl 10K-386S Cc1ccc(cc1)/C=C/C(=O)CCC(=O)O 10K-387S Cc1ccc(cc1)/C=C/C2=NNC(=O)CC2 10K-388S Cc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)C 10K-389S CCOC(=O)C(C)N1C(=O)CCC(=N1)/C=C/c2ccc(cc2)C 10K-390S CCOC(=O)CN1C(=O)CCC(=N1)/C=C/c2ccc(cc2)C 10K-391S Cc1cccc(c1NC(=O)CN(c2ccccn2)S(=O)(=O)c3ccccc3)C 10K-392S Cc1cccc(c1NC(=O)CN(c2ccccn2)S(=O)(=O)c3ccc(cc3)F)C 10K-393S Cc1c(cc(c(n1)O)C#N)C(=O)C 10K-395S Cc1c(cc(c(n1)S)C#N)C(=O)C 10K-396S c1ccc(cc1)NC(=O)CN(c2ccccn2)S(=O)(=O)c3ccccc3 10K-397S Cc1c(cc2c(c(sc2n1)C(=O)OC)N)C(=O)C 10K-399S Cn1c(c(c(n1)C(F)(F)F)C#N)OC 10K-400S Cc1c(cc(c(n1)SCc2ccccc2)C#N)C(=O)C 10K-401S Cc1c(cc(c(n1)SCc2ccc(c(c2)Cl)Cl)C#N)C(=O)C 10K-402S Cc1c(cc(c(n1)SCC=C)C#N)C(=O)C 10K-403S Cc1c(cc(c(n1)SCc2cccc(c2)C(F)(F)F)C#N)C(=O)C 10K-404S Cc1c(cc(c(n1)SCc2ccc(cc2Cl)Cl)C#N)C(=O)C 10K-405S Cc1c(cc(c(n1)SC)C#N)C(=O)C 10K-406S c1ccc(cc1)NC(=O)CN(c2ccccn2)S(=O)(=O)c3ccc(cc3)F 10K-408S c1ccnc(c1)N(CC(=O)Nc2ccc(cc2F)F)S(=O)(=O)c3ccc(cc3)F 10K-409S Cc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)CC=C 10K-410S Cc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccccc3 10K-411S Cn1c(=O)ccc(n1)/C=C/c2ccccc2 10K-413S Cc1c(cc(c(n1)Cl)C#N)C(=O)C 10K-414S C=CCn1c(=O)ccc(n1)/C=C/c2ccccc2 10K-415S CCn1c(c(cc(c1=O)C#N)C(=O)C)C 10K-416S Cc1c(cc(c(n1)O)C#N)C(=O)OC 10K-419S CCOC(=O)C(C)n1c(=O)ccc(n1)/C=C/c2ccccc2 10K-420S CCOC(=O)Cn1c(=O)ccc(n1)/C=C/c2ccccc2 10K-421S COc1ccc(cc1)/C=C/C(=O)CCC(=O)O 10K-422S COc1ccc(cc1)/C=C/C2=NNC(=O)CC2 10K-423S CN1C(=O)CCC(=N1)/C=C/c2ccc(cc2)OC 10K-424S COc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)CC=C 10K-425S COc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccccc3 10K-426S CCOC(=O)CN1C(=O)CCC(=N1)/C=C/c2ccc(cc2)OC 10K-427S Cc1ccc(cc1)/C=C/c2ccc(=O)[nH]n2 10K-428S COc1ccc(cc1)/C=C/c2ccc(nn2)O 10K-429S CCOC(=O)CC(=O)CS(=O)c1ccc(cc1)Cl 10K-503S c1cc(ccc1SCc2cc(nc(n2)c3ccncc3)O)Cl 10K-504S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccccc3 10K-505S c1cc(ccc1SCCNC(=O)CSc2ccc(cc2)Cl)Cl 10K-509S c1cc(cc(c1)SCC(=O)NCCSc2ccc(cc2)Cl)C(F)(F)F 10K-510S c1cc(cc(c1)S(=O)(=O)CC(=O)NCCS(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F 10K-511S c1cc(ccc1S(=O)(=O)CCNC(=O)CS(=O)(=O)c2ccc(cc2)Cl)Cl 10K-519S CC(C(=O)NCCS(=O)(=O)c1ccc(cc1)Cl)S(=O)(=O)c2ccccc2 10K-520S c1ccnc(c1)c2nc(cc(n2)O)CSc3ccc(cc3)Cl 10K-522S c1ccc(cc1)SCc2cc(nc(n2)c3ccncc3)O 10K-523S c1cc(ccc1SCCNC(=O)CCCl)Cl 10K-524S c1ccc(cc1)Sc2cc(nc(n2)c3ccncc3)CSc4ccc(cc4)Cl 10K-525S Cc1ccc(cc1)SCCC(=O)NCCSc2ccc(cc2)Cl 10K-526S c1ccc(cc1)SCCC(=O)NCCSc2ccc(cc2)Cl 10K-527S COC(=O)c1ccccc1SCCC(=O)NCCSc2ccc(cc2)Cl 10K-528S c1ccc(cc1)SCc2cc(nc(n2)c3ccncc3)Cl 10K-532S Cc1ccc(cc1)S(=O)(=O)CCC(=O)NCCS(=O)(=O)c2ccc(cc2)Cl 10K-534S c1ccc(cc1)S(=O)(=O)CCC(=O)NCCS(=O)(=O)c2ccc(cc2)Cl 10K-535S Cc1ccc(cc1)S(=O)(=O)C(C)C(=O)NCCS(=O)(=O)c2ccc(cc2)Cl 10K-536S CC(C(=O)NCCS(=O)(=O)c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl 10K-537S c1ccc(cc1)SCCNC(=O)CCCl 10K-539S c1ccc(cc1)SCCNC(=O)CSc2ccc(cc2)F 10K-540S c1ccc(cc1)SCCNC(=O)CSc2ccc(cc2)Cl 10K-541S c1ccc(cc1)SCCNC(=O)CCSc2ccc(cc2)F 10K-542S c1ccc(cc1)SCCC(=O)NCCSc2ccccc2 10K-543S c1ccc(cc1)SCCNC(=O)CSc2c(cccc2Cl)Cl 10K-546S c1ccc(cc1)SCCNC(=O)CCSc2c(cccc2Cl)Cl 10K-547S CC(C(=O)NCCSc1ccc(cc1)Cl)Sc2ccccc2C(=O)OC 10K-550S c1ccc(cc1)S(=O)(=O)CCC(=O)NCCS(=O)(=O)c2ccccc2 10K-551S c1ccc(cc1)S(=O)(=O)CCNC(=O)CCS(=O)(=O)c2ccc(cc2)F 10K-552S c1ccc(cc1)S(=O)(=O)CCNC(=O)CS(=O)(=O)c2ccc(cc2)F 10K-553S c1ccc(cc1)S(=O)(=O)CCNC(=O)CS(=O)(=O)c2ccc(cc2)Cl 10K-554S CCOC(=O)CSc1cc(nc(n1)c2ccccn2)CSc3ccc(cc3)Cl 10K-555S c1cc(cnc1)c2nc(cc(n2)Sc3ccc(cc3)Cl)CSc4ccc(cc4)Cl 10K-559S c1cc(cnc1)c2nc(cc(n2)Oc3ccc(cc3)Cl)CSc4ccc(cc4)Cl 10K-560S CC(C(=O)NCCSc1ccccc1)Sc2c(cccc2Cl)Cl 10K-564S CC(C(=O)NCCSc1ccccc1)Sc2ccccc2C(=O)OC 10K-565S c1ccc(c(c1)SCC(=O)NCCSc2ccc(cc2)Br)Cl 10K-566S c1cc(c(c(c1)Cl)Cl)SCC(=O)NCCSc2ccc(cc2)Br 10K-567S CC(C(=O)NCCSc1ccc(cc1)Br)Sc2ccc(cc2)Cl 10K-568S CC(C(=O)NCCSc1ccc(cc1)Br)Sc2ccccc2C(=O)OC 10K-569S CC(C(=O)NCCS(=O)(=O)c1ccc(cc1)Br)S(=O)(=O)c2ccc(cc2)Cl 10K-570S CCOC(=O)CSc1cc(nc(n1)c2cccnc2)CSc3ccc(cc3)Cl 10K-572S c1ccnc(c1)c2nc(cc(n2)Sc3ccc(cc3)Cl)CSc4ccc(cc4)Cl 10K-573S CC(C(=O)NCCS(=O)(=O)c1ccc(cc1)Br)S(=O)(=O)c2ccccc2 10K-574S c1ccc(c(c1)CO)Sc2ccc(cc2)Cl 10K-578S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3ccncc3)O 10K-579S c1ccc(c(c1)CCl)Sc2ccc(cc2)Cl 10K-580S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C#N 10K-582S COC(=O)c1ccccc1SCc2ccccc2Sc3ccc(cc3)Cl 10K-583S CSCc1ccccc1Sc2ccc(cc2)Cl 10K-584S c1ccc(c(c1)CSCc2cccc(c2)C(F)(F)F)Sc3ccc(cc3)Cl 10K-585S c1ccc(c(c1)CSCc2ccc(cc2Cl)Cl)Sc3ccc(cc3)Cl 10K-586S c1ccc(c(c1)CSc2ccc(cc2)Cl)Sc3ccc(cc3)Cl 10K-587S c1ccc(c(c1)CSc2ccccc2Cl)Sc3ccc(cc3)Cl 10K-588S c1ccc(cc1)Sc2ccc(cc2N)C#N 10K-591S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3ccncc3)Cl 10K-592S c1ccc(cc1)c2nc(cc(n2)O)CSc3ccc(cc3)Cl 10K-593S c1ccc(cc1)Sc2cc(nc(n2)c3ccncc3)CS(=O)(=O)c4ccccc4 10K-594S c1ccc(c(c1)CSc2ccccc2Cl)S(=O)(=O)c3ccc(cc3)Cl 10K-597S COc1ccc(cc1)CSCc2ccccc2S(=O)(=O)c3ccc(cc3)Cl 10K-600S c1ccc(c(c1)CSCc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 10K-601S Cc1ccc(cc1)C(=O)Nc2cc(ccc2Sc3ccccc3)C#N 10K-602S c1ccnc(c1)c2nc(cc(n2)Cl)CS(=O)c3ccc(cc3)Cl 10K-603S c1ccc(cc1)Sc2ccc(cc2NC(=O)c3ccc(cc3)F)C#N 10K-604S c1ccc(cc1)c2nc(cc(n2)Cl)CSc3ccc(cc3)Cl 10K-608S Cc1ccc(cc1)Sc2ccc(cc2N)C#N 10K-614S c1ccc(cc1)COc2c(cc(c(c2Cl)OCc3ccccc3)Cl)Cl 10K-900 C[NH2+]C1c2c3ccccc3ccc2OCC1CO.[Cl-] 10K-904 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2)Cl)C#N 10K-905 CC1=C(C(C(=C(N1)C)C#N)c2c(cccc2Cl)Cl)C#N 10K-906 Cc1c(c(c(c(n1)C)C#N)c2ccc(cc2)Cl)C#N 10K-907 Cc1c(c(c(c(n1)/C=C/N(C)C)C#N)c2ccc(cc2)Cl)C#N 10K-908 Cc1c(c(c(c(n1)C)C#N)c2c(cccc2Cl)Cl)C#N 10K-909 Cc1c(c(c(c(n1)/C=C/Nc2ccc(cc2)OC)C#N)c3ccc(cc3)Cl)C#N 10K-910 c1ccc(cc1)CNS(=O)(=O)NCc2cccc(c2)C(F)(F)F 10L-001 c1ccc(cc1)CNS(=O)(=O)NCc2ccccc2F 10L-002 COc1ccc(cc1OC)CNS(=O)(=O)NCc2ccccc2 10L-003 COc1ccc(cc1)CNS(=O)(=O)NCc2ccccc2 10L-004 c1ccc(c(c1)CNS(=O)(=O)NCc2ccccc2F)F 10L-005 COc1ccc(cc1)CNS(=O)(=O)NCc2ccccc2F 10L-006 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccccc2F 10L-007 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccc(cc2Cl)Cl 10L-008 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccc(cc2)OC 10L-009 Cc1ccc(cc1)CNS(=O)(=O)NCc2cccc(c2)C(F)(F)F 10L-010 COc1ccc(cc1OC)CNS(=O)(=O)Oc2ccccc2O 10L-011 COc1ccc(cc1OC)CNS(=O)(=O)NCc2ccc(c(c2)OC)OC 10L-012 c1ccc(c(c1)CNS(=O)(=O)NCc2cccc(c2)C(F)(F)F)F 10L-013 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccc(c(c2)OC)OC 10L-014 c1ccc(c(c1)CNS(=O)(=O)NCc2ccc(cc2)Cl)F 10L-015 C/C(=N\NC(=O)OC)/c1ccc(cc1)O 10L-016 Cc1ccc(cc1)CNS(=O)(=O)NCc2cccs2 10L-017 c1cc(ccc1c2csnn2)O 10L-018 c1ccc2c(c1)c(nc(n2)C(F)(F)F)Cl 10L-019 COc1ccc(cc1)CNS(=O)(=O)NCc2ccc(c(c2)OC)OC 10L-020 COc1ccc(cc1OC)CNS(=O)(=O)NCc2ccc(cc2)Cl 10L-021 COc1ccc(cc1)Oc2c3ccccc3nc(n2)C(F)(F)F 10L-022 c1ccc(c(c1)CNS(=O)(=O)NCc2cccs2)F 10L-023 COc1ccc(cc1OC)CNS(=O)(=O)NCc2cccs2 10L-024 C/C(=N\OCc1cccc(c1Cl)Cl)/c2ccc(s2)CC#N 10L-025 C/C(=N\OCc1ccc(cc1Cl)F)/c2ccc(s2)CC#N 10L-026 c1ccc(cc1)NC(=O)Oc2ccc(cc2)c3csnn3 10L-027 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccncc2 10L-028 c1cc(ccc1c2csnn2)OC(=O)c3ccc(cc3)Cl 10L-030 COc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)c3csnn3 10L-031 c1cc(ccc1c2csnn2)OC(=O)Nc3ccc(cc3)Cl 10L-032 Cc1ccccc1NC(=O)Oc2ccc(cc2)c3csnn3 10L-033 COc1ccc(cc1)C(=O)Oc2ccc(cc2)c3csnn3 10L-034 c1cc(oc1)C(=O)Oc2ccc(cc2)c3csnn3 10L-035 CC(=O)Oc1ccc(cc1)c2csnn2 10L-036 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)OC 10L-037 c1cc(ccc1N2CCN(CC2)S(=O)(=O)c3ccc(s3)Cc4c(cc(cn4)C(F)(F)F)Cl)F 10L-039 CS(=O)(=O)Oc1ccc(cc1)c2csnn2 10L-040 CC(C)(C)c1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)c3csnn3 10L-041 C/C(=N\NC(=O)OC)/c1ccc(c(c1)Cl)Cl 10L-042 C/C(=N\NC(=O)OC)/c1ccc(cc1)Br 10L-043 C/C(=N\NC(=O)OC)/c1ccc(cc1)Cl 10L-044 C/C(=N\NC(=O)OC)/c1cccc(c1)OC 10L-045 C/C(=N\NC(=O)OC)/c1ccccc1O 10L-046 c1cc(c(cc1c2csnn2)Cl)Cl 10L-047 c1cc(ccc1c2csnn2)Br 10L-048 CCNC(=O)Oc1ccc(cc1)c2csnn2 10L-049 c1cc(ccc1c2csnn2)Cl 10L-050 c1ccc2c(c1)c(nc(n2)C(F)(F)F)Oc3ccc(cc3)Cl 10L-052 CC(C)(C)c1ccc(cc1)Oc2c3ccccc3nc(n2)C(F)(F)F 10L-053 c1ccc(cc1)Oc2c3ccccc3nc(n2)C(F)(F)F 10L-054 C/C(=N\NC(=O)OC)/c1ccc(c(c1)[N+](=O)[O-])Cl 10L-055 C/C(=N/NC(=O)OC)/c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 10L-056 C/C(=N\NC(=O)OC)/c1ccc2ccccc2c1 10L-057 C/C(=N\NC(=O)OC)/c1ccc(cc1)OC 10L-058 c1cc(c(cc1c2csnn2)[N+](=O)[O-])Cl 10L-059 c1cc(ccc1c2csnn2)Oc3c(cc(cn3)C(F)(F)F)Cl 10L-060 COc1cccc(c1)c2csnn2 10L-061 c1ccc2c(c1)c(nc(n2)C(F)(F)F)Oc3ccc(cc3F)F 10L-062 c1ccc2c(c1)c(nc(n2)C(F)(F)F)Oc3ccc(cc3Cl)[N+](=O)[O-] 10L-063 C/C(=N\NC(=O)OC)/c1ccco1 10L-064 Cc1cc(cc(c1)Oc2c3ccccc3nc(n2)C(F)(F)F)C 10L-065 Cc1ccc(cc1)Oc2c3ccccc3nc(n2)C(F)(F)F 10L-066 CC(=O)Nc1ccc(cc1)Oc2c3ccccc3nc(n2)C(F)(F)F 10L-067 c1ccc2cc(ccc2c1)c3csnn3 10L-068 C/C(=N\NC(=O)OC)/C=C/c1ccccc1 10L-069 c1ccc2c(c1)c(nc(n2)C(F)(F)F)NN 10L-070 C/C(=N\NC(=O)OC)/c1ccc(cc1)c2ccccc2 10L-071 COc1ccc(cc1)c2csnn2 10L-072 Cc1ccc(cc1)/C=N/Nc2c3ccccc3nc(n2)C(F)(F)F 10L-073 c1ccc(cc1)/C=C/c2csnn2 10L-074 c1ccc(cc1)c2ccc(cc2)c3csnn3 10L-075 c1cc(ccc1c2csnn2)OS(=O)(=O)c3ccc(cc3)Cl 10l-089 CC(C)CO/N=C/1\c2ccccc2N(C1=O)c3ccccc3 10L-301S CCCCO/N=C\1/c2ccccc2N(C1=O)c3ccccc3 10L-302S c1ccc(cc1)N2c3ccccc3/C(=N/OCc4ccc(cc4)Cl)/C2=O 10L-303S c1ccc(cc1)N2c3ccccc3/C(=N/OCc4ccc(c(c4)Cl)Cl)/C2=O 10L-304S c1ccc(cc1)N2c3ccccc3/C(=N/OCc4c(cccc4Cl)F)/C2=O 10L-305S CC(C)(C)c1ccc(cc1)CO/N=C\2/c3ccccc3N(C2=O)c4ccccc4 10L-306S c1ccc(cc1)N2c3ccccc3/C(=N/OCc4cccc(c4)C(F)(F)F)/C2=O 10L-307S c1ccc(cc1)N2c3ccccc3/C(=N\OCc4c(cccc4Cl)Cl)/C2=O 10L-308S c1cc(ccc1c2cc(c(c(n2)O)C#N)c3ccc(cc3Cl)Cl)Cl 10L-309S Cc1ccc(cc1)c2cc(c(c(n2)O)C#N)c3ccc(cc3Cl)Cl 10L-310S c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)O)C#N)c3ccc(cc3Cl)Cl 10L-311S Cc1ccc(cc1)c2cc(nc(c2C#N)O)c3ccccc3Cl 10L-312S Cc1ccc(cc1)c2cc(nc(c2C#N)O)c3ccc(c(c3)Cl)Cl 10L-314S COc1ccc(cc1)c2cc([nH]c(=O)c2C#N)c3ccc(c(c3)Cl)Cl 10L-315S COc1ccc(cc1)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)F 10L-316S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)NC 10L-317S Cc1c(n(c(c1C#N)N)Cc2ccccc2)C 10L-318S CC(C)(C)n1c(c(c(n1)c2ccc(cc2)Cl)C#N)N 10L-319S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CS(=O)CC(=O)NC 10L-321S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CS(=O)(=O)CC(=O)NC 10L-322S Cc1ccc(cc1)c2cc(c(c(n2)Cl)C#N)c3ccc(cc3Cl)Cl 10L-323S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)Nc2ccc(cc2)OC 10L-327S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CS(=O)(=O)CC(=O)N2CCOCC2 10L-328S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)Nc2ccc(cc2F)F 10L-329S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)N(C)C 10L-330S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CS(=O)CC(=O)N(C)C 10L-331S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CS(=O)(=O)CC(=O)N(C)C 10L-332S c1ccc(cc1)Cn2c(c(c3c2ncnc3Sc4ccc(cc4)Cl)c5ccccc5)c6ccccc6 10L-333S COc1ccc(cc1)Sc2c3c(c(n(c3ncn2)Cc4ccccc4)c5ccccc5)c6ccccc6 10L-334S Cc1c(n(c2c1c(ncn2)Cl)Cc3ccccc3)C 10L-335S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)Nc2cccc(c2)C(F)(F)F 10L-336S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CS(=O)CC(=O)Nc2cccc(c2)C(F)(F)F 10L-337S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CS(=O)(=O)CC(=O)Nc2cccc(c2)C(F)(F)F 10L-338S CNC(=O)CSCC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-340S CNC(=O)CS(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-341S CNC(=O)CS(=O)(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-342S CN(C)C(=O)CSCC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-343S Cc1ccc(cc1)c2cc(c(c(n2)Sc3ccc(cc3)OC)C#N)c4ccc(cc4Cl)Cl 10L-344S Cc1ccc(cc1)c2cc(c(c(n2)Sc3ccc(cc3)Br)C#N)c4ccc(cc4Cl)Cl 10L-345S Cc1ccc(cc1)c2cc(c(c(n2)N3CCCC3)C#N)c4ccc(cc4Cl)Cl 10L-346S CC(C)Nc1c(c(cc(n1)c2cccc(c2)C(F)(F)F)c3ccc(cc3Cl)Cl)C#N 10L-348S c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)N3CCOCC3)C#N)c4ccc(cc4Cl)Cl 10L-349S COc1ccc(cc1)Oc2c(c(cc(n2)c3cccc(c3)C(F)(F)F)c4ccc(cc4Cl)Cl)C#N 10L-350S CC(C)(C)n1c2c(c(n1)c3ccc(cc3)Cl)c(nc(n2)c4ccc(cc4)Cl)N 10L-351S CNc1nc(c(c(n1)Cl)SC)N2CCCC2 10L-352S CNc1nc(c(c(n1)Cl)SC)NCC=C 10L-353S CNc1nc(c(c(n1)Cl)SC)NCc2ccc(cc2)F 10L-354S c1cc(ccc1/C=N/O)Cl 10L-355S c1cc(ccc1/C(=N/O)/Cl)Cl 10L-356S CN(C)C(=O)CS(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-357S CN(C)C(=O)CS(=O)(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-358S CCN(CC)C(=O)CSCC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-359S CCN(CC)C(=O)CS(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-360S CCN(CC)C(=O)CS(=O)(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OCCOC 10L-361S CNc1nc(c(c(n1)Cl)SC)N2CCN(CC2)c3ccccc3 10L-362S CC(C)Nc1c(c(nc(n1)NC)Cl)SC 10L-363S CNc1nc(c(c(n1)Cl)SC)NCc2cccc(c2)OC 10L-364S c1cc(ccc1c2cc(on2)CO)Cl 10L-365S COc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)Nc2cccc(c2)C(F)(F)F 10L-367S CCN(CC)C(=O)CSCC(=O)Nc1cc(c(cc1Cl)Cl)OC 10L-368S CCN(CC)C(=O)CS(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OC 10L-369S CCN(CC)C(=O)CS(=O)(=O)CC(=O)Nc1cc(c(cc1Cl)Cl)OC 10L-370S CN(c1ccccc1)C(=O)CSCC(=O)Nc2cc(c(cc2Cl)Cl)OC 10L-371S CC(=O)Nc1c(c(nn1C(C)(C)C)c2ccc(cc2)Cl)C#N 10L-373S CCCCNc1c(c(nc(n1)NC)Cl)SC 10L-375S CNc1nc(c(c(n1)Cl)SC)NC2CCCCC2 10L-376S CNc1nc(c(c(n1)Cl)SC)NCc2ccc(c(c2)Cl)Cl 10L-377S CN(c1ccccc1)C(=O)CS(=O)CC(=O)Nc2cc(c(cc2Cl)Cl)OC 10L-378S CN(c1ccccc1)C(=O)CS(=O)(=O)CC(=O)Nc2cc(c(cc2Cl)Cl)OC 10L-379S CCOc1cc(nc(n1)SCc2cccc(c2)C(F)(F)F)CSc3c(cccc3Cl)Cl 10L-501S CNc1cc(nc(n1)SCc2cccc(c2)C(F)(F)F)CSc3c(cccc3Cl)Cl 10L-502S c1cc(ccc1C(F)(F)F)NC(=O)c2csnn2 10L-506S c1cc(c(cc1NC(=O)c2csnn2)F)F 10L-507S c1cc(c(cc1NC(=O)c2csnn2)Cl)Cl 10L-508S c1c(cc(cc1C(F)(F)F)NC(=O)c2csnn2)C(F)(F)F 10L-509S c1ccc(cc1)SCc2cc(nc(n2)SCc3c(cccc3Cl)Cl)Cl 10L-510S CSc1nc(c(c(n1)Cl)C#N)c2ccccc2 10L-512S c1ccc(cc1)NS(=O)(=O)N2CCOC2=O 10L-513S COc1ccc(cc1)Sc2c(c(nc(n2)SC)c3ccccc3)C#N 10L-515S COc1cc(nc(n1)SCc2c(cccc2Cl)Cl)CSc3ccccc3 10L-517S c1ccc(cc1)NC(=S)NC(=O)c2csnn2 10L-519S COc1ccc(cc1)NC(=S)NC(=O)c2csnn2 10L-520S CN(C)c1cc(nc(n1)SCc2c(cccc2Cl)Cl)CSc3ccccc3 10L-523S c1ccc(cc1)NS(=O)(=O)NC(=O)OCCCl 10L-524S CNc1cc(nc(n1)SCc2c(cccc2Cl)Cl)CSc3ccccc3 10L-525S c1cc(ccc1NC(=S)NC(=O)c2csnn2)Cl 10L-526S c1cc(cc(c1)NC(=S)NC(=O)c2csnn2)C(F)(F)F 10L-527S c1cc(ccc1C(F)(F)F)NC(=S)NC(=O)c2csnn2 10L-533S c1cc(c(cc1F)F)NC(=S)NC(=O)c2csnn2 10L-534S c1cc(c(cc1NC(=S)NC(=O)c2csnn2)Cl)Cl 10L-535S c1ccc(c(c1)NC(=S)NC(=O)c2csnn2)Cl 10L-536S COc1cc(c(cc1Cl)Cl)NC(=S)NC(=O)c2csnn2 10L-537S CN(c1ccccc1)C(=S)NC(=O)c2csnn2 10L-538S Cn1c(cnc1SCc2ccc(cc2)Cl)CO 10L-539S c1cc(ccc1CSc2nc(cc(n2)O)CSc3ccc(cc3)Cl)F 10L-543S c1ccc(cc1)SCc2cc(nc(n2)SCc3ccc(c(c3)Cl)Cl)O 10L-545S c1cc(ccc1CSc2nc(cc(n2)N3CCOCC3)CSc4ccc(cc4)Cl)F 10L-548S C=CCNc1cc(nc(n1)SCc2ccc(cc2)F)CSc3ccc(cc3)Cl 10L-549S Cn1c(c(c(n1)c2ccccc2)/C=N/O)Sc3ccccc3 10L-551S Cn1c(c(c(n1)c2ccccc2)/C=N/O)Sc3ccc(cc3)Cl 10L-552S CC(C)(C)c1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)C=O 10L-554S Cn1c(c(c(n1)c2ccccc2)C=O)Sc3ccc(cc3)OC 10L-555S CC(C)(C)c1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)/C=N/O 10L-556S Cn1c(c(c(n1)c2ccccc2)/C=N/O)Sc3ccc(cc3)OC 10L-557S Cn1c(c(c(n1)c2ccccc2)/C=N/O)Sc3ccccc3Cl 10L-558S Cn1c(c(c(n1)c2ccccc2)/C=N/O)Sc3cccc(c3)C(F)(F)F 10L-559S CNc1cc(nc(n1)SCc2ccc(cc2)F)CSc3ccc(cc3)Cl 10L-560S CN(C)c1cc(nc(n1)SCc2ccc(cc2)F)CSc3ccc(cc3)Cl 10L-561S c1cc(ccc1CSc2nc(cc(n2)Sc3ccc(cc3)Br)CSc4ccc(cc4)Cl)F 10L-562S c1cc(ccc1CSc2nc(cc(n2)Sc3ccc(cc3)Cl)CSc4ccc(cc4)Cl)F 10L-563S c1ccc(cc1)C(=O)ONC(=O)c2csnn2 10L-564S C=CCNc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)CSc3ccccc3 10L-565S CN(C)c1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)CSc3ccccc3 10L-566S CNc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)CSc3ccccc3 10L-567S c1ccc(cc1)SCc2cc(nc(n2)SCc3ccc(c(c3)Cl)Cl)N4CCOCC4 10L-568S Cn1c(c(c(n1)c2ccccc2)C#N)Sc3ccccc3 10L-569S Cn1c(c(c(n1)c2ccccc2)C#N)Sc3cccc(c3)C(F)(F)F 10L-570S Cn1c(c(c(n1)c2ccccc2)C#N)Sc3ccccc3Cl 10L-571S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3Cl)Cl)Sc4ccc(cc4)Cl 10L-573S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3cccc(c3Cl)Cl)Sc4ccc(cc4)Cl 10L-574S Cc1ccc(cc1)CO/N=C/c2c(nn(c2Sc3ccc(cc3)Cl)C)c4ccccc4 10L-575S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3cccc(c3Cl)Cl)Sc4ccccc4 10L-576S Cc1ccc(cc1)CO/N=C/c2c(nn(c2Sc3ccccc3)C)c4ccccc4 10L-577S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3cccc(c3)F)Sc4ccccc4 10L-578S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3)F)Sc4ccccc4 10L-579S CSCc1cc(nc(n1)S)O 10L-580S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)C#N 10L-581S Cc1ccccc1Sc2c(c(nn2C)c3ccccc3)C#N 10L-582S Cn1c(c(c(n1)c2ccccc2)C#N)Sc3cccc(c3)Cl 10L-583S Cn1c(c(c(n1)c2ccccc2)C#N)Sc3ccc(cc3)F 10L-584S CC(C)(C)c1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)C#N 10L-585S Cn1c(c(c(n1)c2ccccc2)/C=N/O)Sc3ccc(cc3)Br 10L-586S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3cccc(c3Cl)Cl)Sc4ccc(cc4)Br 10L-587S Cc1ccc(cc1)CO/N=C/c2c(nn(c2Sc3ccc(cc3)Br)C)c4ccccc4 10L-588S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3cccc(c3)F)Sc4ccc(cc4)Br 10L-589S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3)F)Sc4ccc(cc4)Br 10L-590S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3Cl)Cl)Sc4ccc(cc4)Br 10L-591S CSCc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)O 10L-592S CSCc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)O 10L-594S COc1ccc(cc1)CSc2nc(cc(n2)O)CSC 10L-595S c1cc(cc(c1)C(F)(F)F)C(=O)ONC(=O)c2csnn2 10L-598S c1cc(ccc1C(=O)ONC(=O)c2csnn2)Cl 10L-599S c1cc(c(cc1C(=O)ONC(=O)c2csnn2)Cl)Cl 10L-600S CN(C)c1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)CSC 10L-601S CNc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)CSC 10L-602S CSCc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)N3CCOCC3 10L-603S CSCc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)NCC=C 10L-604S Cn1c(c(c(n1)c2ccccc2)/C=N/OC)Sc3ccc(cc3)Cl 10L-605S c1ccc(c(c1)C(=O)ONC(=O)c2csnn2)Cl 10L-607S c1cc(c(cc1Cl)Cl)C(=O)ONC(=O)c2csnn2 10L-608S c1c(cc(cc1Cl)Cl)C(=O)ONC(=O)c2csnn2 10L-609S c1cc(c(c(c1)F)C(=O)ONC(=O)c2csnn2)F 10L-610S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3Cl)Cl)Sc4ccccc4C(=O)OC 10L-611S Cc1ccc(cc1)CO/N=C/c2c(nn(c2Sc3ccccc3C(=O)OC)C)c4ccccc4 10L-613S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3cccc(c3)F)Sc4ccccc4C(=O)OC 10L-614S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3)F)Sc4ccccc4C(=O)OC 10L-615S CSc1nc(c(c(n1)Sc2ccc(cc2)Cl)C#N)c3ccccc3 10L-616S CSc1nc(c(c(n1)Sc2cccc(c2)Cl)C#N)c3ccccc3 10L-617S CNc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)CSC 10L-618S CN(C)c1cc(nc(n1)SCc2ccc(cc2Cl)Cl)CSC 10L-619S CSCc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)N3CCOCC3 10L-620S CSCc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)NCC=C 10L-621S c1ccc(cc1)c2c(c(nc(n2)SCc3c(cccc3Cl)Cl)Cl)C#N 10L-622S CO/N=C(\CBr)/c1ccc(cc1)Cl 10L-628S Cc1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)c3ccccc3 10L-629S Cc1ccc(cc1)c2c(c(nc(n2)SC)Cl)C#N 10L-630S CO/N=C(/CSc1cccc(c1)Cl)\c2ccc(cc2)Cl 10L-631S CC1(CN(C1=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)C 10L-700 Cc1ccc(cc1)C(=O)Nc2nc(ns2)O 10L-700S CC(=C)C(=O)Nc1ccc(cc1)Cl 10L-701 CC(C)(CCl)C(=O)Nc1c(c(c(c(c1F)F)F)F)F 10L-703 CC1(CN(C1=O)c2c(c(c(c(c2F)F)F)F)F)C 10L-704 c1ccc(cc1)CN2C(=O)Cc3ccccc3C2=O 10L-705 CC(=C)C(=O)Nc1ccccc1 10L-706 CC(=C)C(=O)Nc1ccc(cc1)OC 10L-707 CC(=C)C(=O)Nc1ccc(cc1)C(F)(F)F 10L-708 CC(C)(CCl)C(=O)Nc1cccc(c1)C#N 10L-709 CC1(CN(C1=O)c2cccc(c2)C#N)C 10L-710 CCOC(=O)c1c(c(c(=O)n(c1N)NC2=CCCCC2=O)C#N)c3ccc(cc3)Cl 10L-711 CC1=C(C(NC(=S)N1)c2ccc(cc2)Cl)C(=O)Nc3ccccc3 10L-712 CC(C)(CCl)C(=O)Nc1ccc(cc1)OC(F)(F)F 10L-713 CC(C)(CCl)C(=O)Nc1ccc(cc1)NC(=O)C(C)(C)CCl 10L-714 CC1(CN(C1=O)c2ccc(cc2)N3CC(C3=O)(C)C)C 10L-715 COc1ccc(cc1)CN2C(=O)Cc3ccccc3C2=O 10L-716 CCOC(=O)c1ccc(cc1)NC(=O)C(C)(C)CCl 10L-718 CCOC(=O)c1ccc(cc1)N2CC(C2=O)(C)C 10L-719 CC1=C(C(NC(=S)N1)c2c(cccc2Cl)F)C(=O)Nc3ccccc3 10L-720 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3cc(n[nH]3)c4cccs4 10L-721 COc1ccc(cc1)/C=C/C(=O)c2ccccc2 10L-722 c1ccc(c(c1)/C=C\2/C(=O)C3CCN2CC3)C(F)(F)F 10L-723 CN(C)c1ccc(cc1)/C=C/2\C(=O)C3CCN2CC3 10L-724 c1cc(ccc1C(=O)/C=C/c2ccc(cc2Cl)Cl)Cl 10L-725 c1cc(ccc1C(=O)/C=C/c2ccc(cc2Cl)Cl)Br 10L-726 c1cc(sc1)c2cc(n[nH]2)C3CCN(CC3)C(=O)N 10L-727 CC(C)(CCl)C(=O)Nc1ccc(cn1)Cl 10L-728 CC1(CN(C1=O)c2ccc(cn2)Cl)C 10L-729 c1cc(ccc1/C=C/C(=O)c2cc(ccc2Cl)Cl)Cl 10L-730 Cc1c(cccc1Cl)NC(=O)C(C)(C)CCl 10L-731 Cc1c(cccc1Cl)N2CC(C2=O)(C)C 10L-732 CN1C(=O)Cc2ccccc2C1=O 10L-733 C=C(CS(=O)(=O)c1ccccc1)C(=O)Nc2ccc(cc2)Cl 10L-734 c1cc(sc1c2ccno2)S(=O)(=O)Cl 10L-736 CN(C)c1ccc(cc1)c2cc(n[nH]2)C3CCNCC3 10L-737 c1ccc2c(c1)C(=O)N(C2=O)N3C(=O)CSC3=S 10L-738 CO/N=C(\C=C\c1ccc(cc1Cl)Cl)/c2ccccc2 10L-739 CC1=C(C(NC(=S)N1)c2ccc(cc2)F)C(=O)Nc3ccccc3 10L-740 c1ccc2c(c1)CC(=O)N(C2=O)Cc3cccc(c3)Cl 10L-741 CC1=C(C(N2C(=O)CSC2=N1)c3ccc(cc3)Cl)C(=O)Nc4ccccc4 10L-743 C1CC(=O)N(C1=O)N2C(=O)CSC2=S 10L-744 CN(C)/C=C\1/C(=O)N(C(=S)S1)N2C(=O)c3ccccc3C2=O 10L-745 C1CC(=O)N(C(=O)C1)N2C(=O)CSC2=S 10L-746 Cc1cc(cc(c1)NC(=O)C(C)(C)CCl)C 10L-747 Cc1cc(cc(c1)N2CC(C2=O)(C)C)C 10L-748 c1cc(oc1c2ccno2)S(=O)(=O)Cl 10L-749 CC1=C(C(NC(=S)N1)c2ccc(cc2)OCc3ccccc3)C(=O)Nc4ccccc4 10L-750 c1ccc2c(c1)C(=O)N(C2=O)N3C(=O)/C(=C/c4ccc(cc4)Cl)/SC3=S 10L-751 CN(C)/C=C\1/C(=O)N(C(=S)S1)N2C(=O)CCC2=O 10L-752 CC(=C)C(=O)Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 10L-753 CC(=C)C(=O)Nc1ccc(cc1)C#N 10L-754 CC(=C)C(=O)Nc1ccc(cc1)N(C)C 10L-755 CC1=C(C(NC(=S)N1)c2ccco2)C(=O)Nc3ccccc3 10L-756 c1ccc2c(c1)/C(=N\Nc3ccc(cc3)C#N)/C(=O)OC2=O 10L-757 c1ccc2c(c1)C(=O)N(C2=O)N3C(=O)/C(=C/c4ccc(cc4)F)/SC3=S 10L-758 CC(C)(CCl)C(=O)Nc1ccc(cc1)N(C)C 10L-759 CC1(CN(C1=O)c2ccc(cc2)N(C)C)C 10L-760 CC(=C)C(=O)Nc1ccc(cn1)Cl 10L-761 CC(=C)C(=O)Nc1cccc(c1)[N+](=O)[O-] 10L-762 c1ccc(c(c1)C(=O)O)SCC(=O)O 10L-765 c1ccc(cc1)CN2C(=O)c3ccccc3C4(C2=O)CCCC4 10L-766 Cn1ccc(n1)c2cccs2 10L-767 CC(C)(CCl)C(=O)Nc1ccc(cc1)F 10L-768 CC1(CN(C1=O)c2ccc(cc2)F)C 10L-769 CN(C)/C=C/c1c(cc(c(=O)o1)NC(=O)c2cccc(c2)Cl)C(=O)OC 10L-900 Cc1cc(n(n1)c2ccnc3c2ccc(c3)Cl)C 10L-901 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C4CC(C3C2=O)C=C4 10L-902 Cc1cc(cc(c1)N/C=C/c2c(cc(c(=O)o2)NC(=O)c3cccc(c3)Cl)C(=O)OC)C 10L-904 Cc1cc(n(n1)c2ccccc2)c3c(nn(c3O)c4nc(cs4)c5c(ccs5)Cl)C 10L-905 Cc1c2cc(c(=O)oc2ccn1)NC(=O)c3ccc(cc3)Cl 10L-906 CCOC(=O)c1c(cn(c1N)c2c(cc(cn2)C(F)(F)F)Cl)c3c(ccs3)Cl 10L-907 CC(=O)c1cc(c(=O)oc1/C=C/C2=C(CC(CC2=O)(C)C)O)NC(=O)c3ccc(cc3)Cl 10L-908 Cc1cc(cc(c1)n2ccc3c(c2=O)cc(c(=O)o3)NC(=O)c4cccc(c4)Cl)C 10L-909 Cc1c(cc(c(=O)n1N)NC(=O)c2ccc(cc2)Cl)c3ccn[nH]3 10L-910 CN1C(C2C3CC(C2O1)C4C3C(=O)N(C4=O)CCNc5c(cc(cn5)C(F)(F)F)Cl)c6ccc(cc6)OC 10L-911 c1cc(ccc1Cn2c(=O)c(nn(c2=O)c3ccc(cc3)F)C#N)C(F)(F)F 10L-912 c1ccc2c(c1)C(=O)c3c(ccc(c3C2=O)NC(=O)C(F)(F)F)NC(=O)C(F)(F)F 10L-913 COc1ccc(cc1OC)CCN2C(=O)C3C4CC(C3C2=O)C=C4 10L-914 Cc1cc(cc(c1)n2c(=O)n(c(=O)c(n2)C(=O)/C=C/N(C)C)C)C 10L-915 Cc1cc(cc(c1)n2c(=O)n(c(=O)c(n2)C(=O)/C=C/Nc3ccc(cc3)Br)C)C 10L-916 Cc1cc(cc(c1)n2c(=O)n(c(=O)c(n2)C(=O)/C=C/Nc3ccc(cc3)OC(F)(F)F)C)C 10L-917 Cc1ccc(cc1)n2cc(cn2)c3c(=O)n(c(=O)n(n3)c4cc(cc(c4)C)C)C 10L-918 CC(=O)c1cc(c(=O)oc1C/C=N\OC)NC(=O)c2ccccc2 10L-920 COCCn1cc(c(=O)[nH]c1=O)C#N 10L-921 CN(C)/C=C/c1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(=O)OC 10L-922 Cc1ccc(cc1)C(=O)Nc2cc(c(oc2=O)/C=C/N(C)C)C(=O)C 10L-923 CN(C)/C=C/1\CCC(=O)c2c1oc(=O)c(c2)NC(=O)c3ccccc3 10L-924 CO/N=C\C1c2ccccc2C(=O)c3c1cccc3 10L-926 COCCN1CC(C(=O)NC1=O)C(=N)N 10L-927 COc1ccc(cc1)Cn2cc(c(=O)[nH]c2=O)C#N 10L-928 CN(C)/C=C/c1c(cc(c(=O)o1)NC(=O)c2cccc(c2)C(F)(F)F)C(=O)OC 10L-929 c1c(cnc(c1Cl)NCCN2CC(C(=O)NC2=O)C(=N)N)C(F)(F)F 10L-931 Cc1ccc(cc1)C(=O)Nc2cc(c(n(c2=O)N)C)c3ccn[nH]3 10L-932 c1cnccc1Cn2cc(c(=O)[nH]c2=O)C#N 10L-933 CCOC(=O)c1cc(on1)c2c(cc(c(=O)o2)NC(=O)c3ccccc3)C(=O)C 10L-934 COC(=O)c1cc(c(=O)oc1/C=C/Nc2ccc(cc2)Oc3ccccc3)NC(=O)c4ccccc4 10L-936 COC(=O)c1cc(c(=O)oc1C/C=N\OC)NC(=O)c2ccccc2 10L-937 Cc1ccc(cc1)C(=O)Nc2cc(c(n(c2=O)/N=C\c3ccc(cc3)F)C)c4ccn[nH]4 10L-938 c1ccc(cc1)C(=O)Nc2cc3c(ccn(c3=O)c4ccc(cc4)Oc5ccccc5)oc2=O 10L-939 CN(c1c(cc(cn1)C(F)(F)F)Cl)N/C=C/c2c(cc(c(=O)o2)NC(=O)c3cccc(c3)C(F)(F)F)C(=O)OC 10L-940 COC(=O)c1cc(c(=O)oc1/C=C/Nc2cccc(c2)Cl)NC(=O)c3cccc(c3)C(F)(F)F 10L-941 COC(=O)c1cc(c(=O)oc1/C=C/Nc2ccc(cc2)F)NC(=O)c3cccc(c3)C(F)(F)F 10L-942 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc3c(ccn(c3=O)c4cccc(c4)Cl)oc2=O 10L-943 COC(=O)c1cc(c(=O)oc1/C=C/Nc2nccs2)NC(=O)c3ccccc3 10L-944 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2ccc3c(c2=O)cc(c(=O)o3)NC(=O)c4cccc(c4)C(F)(F)F 10L-945 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc3c(ccn(c3=O)c4ccc(cc4)F)oc2=O 10L-946 c1ccc(cc1)C(=O)Nc2cc3c(ccn(c3=O)c4nccs4)oc2=O 10L-948 CCOC(=O)C1=NOC2C1C3CC2C4C3C(=O)N(C4=O)N(C)c5c(cc(cn5)C(F)(F)F)Cl 10L-949 COC(=O)c1cc(c(=O)oc1/C=C/c2c(nc(nc2O)O)O)NC(=O)c3ccccc3 10L-950 COn1ccc2c(c1=O)cc(c(=O)o2)NC(=O)c3ccccc3 10L-951 c1cc2c(nc1)n(c(=O)c(n2)N/N=C/c3ccc(cc3)F)CCNc4c(cc(cn4)C(F)(F)F)Cl 10L-952 COC(=O)c1ccc(cc1)n2ccc3c(c2=O)cc(c(=O)o3)NC(=O)c4ccccc4 10L-953 Cc1ccc(cc1)C(=O)Cn2cccn2 10L-955 c1cc(c(c(c1)Cl)NCCNc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 10L-956 c1cc(c(c(c1)Cl)NCCNc2c(cc(cn2)C(F)(F)F)Cl)N 10L-957 c1cc2c(c(c1)Cl)n(c(=O)c(=O)[nH]2)CCNc3c(cc(cn3)C(F)(F)F)Cl 10L-959 c1cnccc1CN2CC(C(=O)NC2=O)C(=N)N 10L-960 COC(=O)c1cc(c(=O)oc1C/C=N/OCc2cccc(c2Cl)Cl)NC(=O)c3cccc(c3)C(F)(F)F 10L-961 COC(=O)CN/C=C/c1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(=O)OC 10L-962 CCOC(=O)/C=C\1/CCCc2c1cco2 10L-963 CCOC(=O)Cc1c(cccn1)C(=O)NCc2ccc(cc2)OC 10L-964 c1cc(c(cc1Cl)[N+](=O)[O-])NCCNc2c(cc(cn2)C(F)(F)F)Cl 10L-965 c1cc(c(cc1Cl)N)NCCNc2c(cc(cn2)C(F)(F)F)Cl 10L-966 c1cc(c(cc1Cl)N)NCCNc2c(cc(cn2)C(F)(F)F)Cl.Cl 10L-967 CCOC(=O)Cc1cccc2c1cco2 10L-968 Cc1ccccc1CN2C(=O)C(=O)N(C2=O)Cc3cccc(c3)C(F)(F)F 10M-001 Cc1ccccc1CN2C(=O)C(=O)N(C2=O)Cc3ccc(c(c3)OC)OC 10M-002 c1cc(cc(c1)Cl)CN2C(=O)C(=O)NC2=O 10M-003 c1cc(ccc1CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3Cl)Cl)F 10M-004 Cc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3Cl)Cl 10M-005 c1cc(c(c(c1)Cl)CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)F)F 10M-006 CCOC(=O)c1c(c2c(ccnc2s1)OC)/N=C/N(C)C 10M-007 COc1ccnc(c1C(=O)N)Oc2ccc(cc2)F 10M-008 CC(=O)C1CC1c2ccc(cc2)Cl 10M-010 CCOC(=O)c1c(c2c(ccnc2s1)OC)/N=C/NOCc3ccc(cc3)Cl 10M-011 CN(C)/C=N\C(=O)c1c(ccnc1Oc2ccc(cc2)F)OC 10M-012 C/C(=N\OC(=O)c1ccc(cc1)F)/C2CC2c3ccc(cc3)OC 10M-013 C/C(=N\OC(=O)C1CC1)/C2CC2c3ccc(cc3)OC 10M-014 CCOC(=O)c1c(c2c(ccnc2s1)OC)N/C=N/OCc3c(cccc3Cl)Cl 10M-015 CCOC(=O)c1c(c2c(ccnc2s1)OC)N/C=N/OC 10M-016 CCOC(=O)c1c(c2c(ccnc2s1)OC)N/C=N/OCc3ccccc3 10M-017 COc1ccnc(c1C(=O)N/C=N/OC)Oc2ccc(cc2)F 10M-018 COc1ccnc(c1C(=O)N/C=N/OCc2c(cccc2Cl)Cl)Oc3ccc(cc3)F 10M-019 COc1ccnc(c1C(=O)N/C=N/OCc2ccccc2)Oc3ccc(cc3)F 10M-020 COc1ccnc(c1c2nc[nH]n2)Oc3ccc(cc3)F 10M-021 COc1ccnc(c1C(=O)N/C=N/OCc2ccc(cc2Cl)Cl)Oc3ccc(cc3)F 10M-022 COc1ccnc(c1C(=O)N/C=N/OCc2ccc(cc2Cl)F)Oc3ccc(cc3)F 10M-023 CCOC(=O)c1c(c2c(ccnc2s1)OC)N/C=N/OCc3ccc(cc3)F 10M-024 CCOC(=O)c1c(c2c(ccnc2s1)OC)N/C=N/OCc3ccc(cc3Cl)F 10M-025 CCOC(=O)c1c(c2c(ccnc2s1)OC)N/C=N/OCCOc3cccc(c3)C(F)(F)F 10M-026 CCOC(=O)c1c(c2c(ccnc2s1)OC)N/C=N/OCc3ccccc3OC 10M-027 COc1ccccc1CO/N=C/NC(=O)c2c(ccnc2Oc3ccc(cc3)F)OC 10M-028 COc1ccnc(c1C(=O)N/C=N/OCc2cccc(c2)F)Oc3ccc(cc3)F 10M-029 C/C(=N\OC(=O)c1cccs1)/C2CC2c3ccc(cc3)OC 10M-030 COC(=C(C#N)C#N)/C=C/Nc1ccc(cc1)Cl 10M-031 COc1ccnc(c1C#N)Nc2ccc(cc2)Cl 10M-032 C/C(=N\Oc1c(cc(cn1)C(F)(F)F)Cl)/C2CC2c3ccc(cc3)OC 10M-033 COc1ccnc(c1C(=O)N/C=N/OCc2ccc(cc2)F)Oc3ccc(cc3)F 10M-034 COc1ccnc(c1C#N)Nc2cc(cc(c2)Cl)Cl 10M-036 COC(=C(C#N)C#N)/C=C/Nc1ccc(cc1)Br 10M-038 COc1ccnc(c1C#N)Nc2ccc(cc2)Br 10M-039 COC(=C(C#N)C#N)/C=C/Nc1ccc(cc1)I 10M-040 COc1ccnc(c1C#N)Nc2ccc(cc2)I 10M-041 Cc1ccc(cc1)N/C=C/C(=C(C#N)C#N)OC 10M-042 Cc1ccc(cc1)Nc2c(c(ccn2)OC)C#N 10M-043 COc1ccnc(c1C(=O)N/C=N/OCCOc2cccc(c2)C(F)(F)F)Oc3ccc(cc3)F 10M-044 C/C(=N\OC(=O)c1ccccc1)/C2CC2c3ccc(cc3)OC 10M-045 C/C(=N\OC(=O)c1c(cccc1Cl)Cl)/C2CC2c3ccc(cc3)OC 10M-046 COc1ccccc1CN2C(=O)C(=O)N(C2=O)Cc3c(cccc3Cl)F 10M-047 COC(=C(C#N)C#N)/C=C/Nc1ccc(cc1)[N+](=O)[O-] 10M-048 COC(=C(C#N)C#N)/C=C/Nc1cccc(c1)[N+](=O)[O-] 10M-049 COc1ccnc(c1C#N)Nc2ccc(cc2)[N+](=O)[O-] 10M-050 COc1ccnc(c1C#N)Nc2cccc(c2)[N+](=O)[O-] 10M-051 Cc1cccc(c1)Nc2c(c(ccn2)OC)C#N 10M-052 COC(=C(C#N)C#N)/C=C/Nc1ccccc1 10M-053 COc1ccnc(c1C#N)Nc2ccccc2 10M-054 COc1ccccc1CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)Br 10M-055 C/C(=N\O)/C1CC1c2ccc(cc2)Cl 10M-056 COc1ccc(cc1)N/C=C/C(=C(C#N)C#N)OC 10M-057 COc1ccc(cc1)Nc2c(c(ccn2)OC)C#N 10M-058 CN(C)c1ccnc(c1C#N)Oc2ccccc2 10M-059 CC(=O)Nc1ccc(cc1)Oc2c(c(ccn2)N(C)C)C#N 10M-060 CN(C)c1ccnc(c1C#N)Oc2ccc(cc2)F 10M-061 CC(C)(C)c1ccc(cc1)Oc2c(c(ccn2)N(C)C)C#N 10M-062 COC(=C(C#N)C#N)/C=C/Nc1ccc(cc1)OCc2ccccc2 10M-063 COc1ccnc(c1C#N)Nc2ccc(cc2)OCc3ccccc3 10M-064 Cc1ccc(cc1C)N/C=C/C(=C(C#N)C#N)OC 10M-065 COC(=C(C#N)C#N)/C=C/Nc1ccc(c(c1)Cl)Cl 10M-066 COc1ccnc(c1C#N)Nc2ccc(c(c2)Cl)Cl 10M-067 Cc1ccc(cc1C)Nc2c(c(ccn2)OC)C#N 10M-068 CN(C)c1ccnc(c1C#N)Oc2cccc(c2)OC 10M-069 Cc1cc(ccc1Oc2c(c(ccn2)N(C)C)C#N)Cl 10M-070 Cc1cccc(c1)CN2C(=O)C(=O)N(C2=O)Cc3ccccc3OC 10M-071 c1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CCOc3ccccc3 10M-073 c1ccc(c(c1)CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)[N+](=O)[O-])Cl 10M-074 CN(C)c1ccnc(c1C#N)Sc2ccc(cc2)OC 10M-075 COc1ccccc1CN2C(=O)C(=O)N(C2=O)CC#N 10M-076 CCOC(=O)c1c(c2c(ccnc2s1)N(C)C)/N=C/N(C)C 10M-077 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2cccc(c2)C 10M-078 Cc1ccc(cc1)C(=O)CN2C(=O)C(=O)N(C2=O)Cc3ccccc3 10M-079 c1cc(cc(c1)Cl)CN2C(=O)C(=O)N(C2=O)Cc3c(cccc3Cl)Cl 10M-080 CCOC(=O)c1c(c2c(ccnc2s1)N(C)C)N/C=N/OCc3ccccc3 10M-081 CCOC(=O)c1c(c2c(ccnc2s1)N(C)C)N/C=N/OC 10M-082 CCOC(=O)c1c(c2c(ccnc2s1)N(C)C)N/C=N/OCc3c(cccc3Cl)F 10M-083 c1cc(cc(c1)Cl)CN2C(=O)C(=O)N(C2=O)Cc3cccc(c3)Cl 10M-084 c1ccc(c(c1)CN2C(=O)C(=O)N(C2=O)CC#N)Cl 10M-085 Cc1cc(c(c(c1)C)CN2C(=O)C(=O)N(C2=O)Cc3ccccc3)C 10M-086 CCOC(=O)c1c(c2c(ccnc2s1)N(C)C)n3cccc3 10M-087 c1ccc(cc1)c2ccc(cc2)C(=O)CN3C(=O)C(=O)N(C3=O)Cc4cccc(c4)C(F)(F)F 10M-088 Cc1cc(cc(c1)Oc2c(c(cc(n2)c3ccccc3)C)S(=O)(=O)C)C 10M-303S Cc1cccc(c1C)Oc2c(c(cc(n2)c3ccccc3)C)S(=O)(=O)C 10M-304S Cc1cc(nc(c1S(=O)(=O)C)Oc2ccc(cc2)OC)C 10M-305S Cc1ccccc1Oc2c(c(cc(n2)C)C)S(=O)(=O)C 10M-306S Cc1cc(nc(c1S(=O)(=O)C)Oc2cccc(c2)C(F)(F)F)C 10M-307S Cc1cc(nc(c1S(=O)(=O)C)Oc2ccc(cc2)F)C 10M-308S Cc1ccc(cc1)CN2CCn3c(cc(n3)C(=O)OC)C2=O 10M-311S Cc1cc(nc(c1S(=O)(=O)C)Oc2cccc(c2)Cl)C 10M-312S Cc1cc(nc(c1S(=O)(=O)C)Oc2ccc(cc2)C(C)(C)C)C 10M-313S COC(=O)c1cc2n(n1)CCN(C2=O)Cc3ccccc3F 10M-314S COC(=O)c1cc2n(n1)CCN(C2=O)Cc3ccc(cc3)F 10M-315S COc1ccc(cc1)CN2CCn3c(cc(n3)C(=O)OC)C2=O 10M-316S COC(=O)c1cc2n(n1)CCN(C2=O)Cc3ccccc3Cl 10M-317S Cc1cc(nc(c1S(=O)(=O)C)NN)C 10M-319S Cc1cc(nc(c1S(=O)(=O)C)N(C)N)C 10M-320S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2N(C)N)c3ccccc3)C 10M-321S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)c2cccc(c2)OC)C 10M-322S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)c2c(cccc2F)F)C 10M-323S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)c2ccc(c(c2)Cl)Cl)C 10M-324S Cc1cc(nc(c1S(=O)(=O)C)N(C)N)c2ccccc2 10M-325S COc1cccc(c1)CN2CCn3c(cc(n3)C(=O)OC)C2=O 10M-328S CC(=O)CCC(=O)c1ccc(cc1)SC 10M-332S CCSc1ncc(n1C)CO 10M-335S CC(=O)CCC(=O)c1ccc(cc1)S(=O)(=O)C 10M-336S CCSc1ncc(n1C)C=O 10M-337S Cc1ccc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C 10M-338S CCSc1ncc(n1C)/C=N/Nc2c(cc(cc2Cl)Cl)Cl 10M-339S CCSc1ncc(n1C)/C=N/Nc2ccccc2 10M-340S CCSc1ncc(n1C)/C=N/Nc2c(cc(cc2Cl)C(F)(F)F)Cl 10M-341S CCSc1ncc(n1C)/C=N/Nc2ccc(cc2)[N+](=O)[O-] 10M-342S C=CCSc1ncc(n1Cc2ccccc2)C=O 10M-344S CCOc1c(c(ccn1)c2ccc(cc2)F)C#N 10M-501S COC(=O)CSc1c(c(ccn1)c2ccc(cc2)F)C#N 10M-502S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)Cl)O 10M-511S Cc1cccn2c1nc(c2)c3cnoc3C 10M-515S c1cc2c(cc1F)nc(s2)CN3CCOCC3 10M-516S CSc1cc(n[nH]1)c2ccc(cc2)Cl 10M-517S c1cc(ccc1c2cc([nH]n2)N3CCOCC3)Cl 10M-518S c1cc(ccc1c2c[nH]c(n2)S)Cl 10M-521S CN(C)Cc1nc2cc(ccc2s1)F 10M-523S c1cc(ncc1C(F)(F)F)N2CCOCC2 10M-525S Cc1cc(nc(c1C#N)SCc2ccc(cc2)OC)c3ccccc3 10M-526S Cc1cc(nc(c1C#N)SCc2ccc(c(c2)Cl)Cl)c3ccccc3 10M-527S Cc1c2ccccc2nc(c1C(=O)C)Sc3ccc(cc3)Cl 10M-529S Cc1c2ccccc2nc(c1C(=O)/C=C/c3ccc(cc3)Br)Sc4ccc(cc4)Cl 10M-530S Cc1c2ccccc2nc(c1C(=O)C)Sc3ccc(cc3)Br 10M-533S Cc1ccc(cc1)Sc2c(c(c3ccccc3n2)C)C(=O)C 10M-534S Cn1c(c(c(n1)C(F)(F)F)/C=C/C(=O)c2ccc(cc2)Cl)Cl 10M-535S Cn1c(c(c(n1)C(F)(F)F)/C=C/C(=O)c2ccc(c(c2)Cl)Cl)Cl 10M-536S Cn1c(c(c(n1)C(F)(F)F)/C=C/C(=O)c2cccs2)Cl 10M-537S Cn1c(c(c(n1)C(F)(F)F)/C=C/C(=O)c2ccccn2)Cl 10M-538S Cc1c2ccccc2nc(c1C(=O)/C=C/c3c(nn(c3Cl)C)C(F)(F)F)Cl 10M-539S CCOC(=O)c1cnc([nH]c1=O)c2ccccc2 10M-541S COc1ccc(cc1)COC(=O)Nc2c(snn2)Sc3ccc(cc3)Cl 10M-542S c1cc(cc(c1)C(F)(F)F)COC(=O)Nc2c(snn2)Sc3ccc(cc3)Cl 10M-543S CC(C)(C)COC(=O)Nc1c(snn1)Sc2ccc(cc2)Cl 10M-544S c1cc(ccc1COC(=O)Nc2c(snn2)Sc3ccc(cc3)Cl)C(F)(F)F 10M-545S Cc1c2ccccc2nc(c1C(=O)/C=C/c3cccc(c3Cl)Cl)Sc4ccc(cc4)Br 10M-546S Cc1c2ccccc2nc(c1C(=O)/C=C/c3ccc(cc3)F)Sc4ccc(cc4)Br 10M-547S Cc1c2ccccc2nc(c1C(=O)C)SCc3ccc(cc3)Cl 10M-548S CCOC(=O)c1cnc(nc1Cl)c2ccccc2 10M-550S Cc1ccc(cc1)C/N=C/c2ccc(c(c2O)Cc3c(cccc3Cl)F)O 10M-701 Cc1c(c(=O)ccn1c2ccc(cc2)/C(=C/N(C)C)/C#N)Cc3c(cccc3Cl)Cl 10M-702 Cc1c(c(=O)ccn1n2cnnc2)Cc3c(cccc3Cl)Cl 10M-704 Cc1c(c(=O)ccn1CC(C)(C)SCc2cccc(c2)C(F)(F)F)Cc3c(cccc3Cl)Cl 10M-706 c1cc(c(c(c1)Cl)CO/N=C/CC(=O)c2cc(sc2Cl)Cl)F 10M-707 c1cc(c(c(c1)Cl)Cc2c(ccc(c2O)/C=N/Cc3ccncc3)O)F 10M-708 Cc1ccc(n1c2ccc(cc2)C#Cc3ccc(cc3)n4c(ccc4C)C)C 10M-709 C/C(=N\c1ccsc1C(=O)OC)/c2ccncc2 10M-710 CC(C)(CNC(=O)c1cccs1)SCc2ccc(cc2)F 10M-712 COc1ccc(cc1OC2CCCC2)C=O 10M-719 Cc1cc2c(cco2)c(=O)o1 10M-720 Cc1cc2c(c(=O)o1)C(CO2)O 10M-723 CC(=O)C(Cc1c(cccc1Cl)F)C(=O)c2ccccc2 10M-726 COc1cccc(c1)C/N=C/c2ccc(c(c2O)Cc3c(cccc3Cl)F)O 10M-728 c1cc(cc(c1)C(F)(F)F)C/N=C/c2ccc(c(c2O)Cc3c(cccc3Cl)F)O 10M-729 c1cc(c(c(c1)Cl)Cc2c(ccc(c2O)/C=N/Cc3ccco3)O)F 10M-730 CC(C)(CNC(=O)c1cccc(c1)OC)SCc2ccc(cc2)F 10M-731 Cc1ccc(cc1)C(=O)NCC(C)(C)Sc2c(cc(cn2)C(F)(F)F)Cl 10M-732 CC(=O)c1ccc(cc1)N2CC2c3ccncc3 10M-733 c1cc2c(nc1)n(nn2)CCNc3c(cc(cn3)C(F)(F)F)Cl 10M-903 CCOC(=O)C1C(C1C(=O)N/N=C/c2ccc(cc2)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 10M-907 CCOC(=O)C1C(C1C(=O)N/N=C\c2cccc(c2)[N+](=O)[O-])C(=O)Nc3cccc(c3)C(F)(F)F 10M-908 CCOC(=O)C1C(C1C(=O)N/N=C\c2c[nH]c3c2cccc3)C(=O)Nc4cccc(c4)C(F)(F)F 10M-909 CCOC(=O)C1C(C1C(=O)N/N=C/c2ccc(cc2)N(C)C)C(=O)Nc3cccc(c3)C(F)(F)F 10M-910 c1ccc(cc1)Oc2ccc(cc2)NC(=S)N 10N-001 c1ccc(cc1)Oc2ccccc2NC(=S)N 10N-002 CN(C)c1ccc(cc1)NC(=S)NC(=O)c2ccccc2 10N-003 COC(=O)c1ccc(cc1)Oc2ccc(cn2)C(F)(F)F 10N-004 COC(=O)c1ccc(cc1)Oc2c(cccn2)[N+](=O)[O-] 10N-005 Cc1ccc(cc1)NNC(=S)N 10N-006 COC(=O)c1ccc(cc1)OCc2c(cccc2Cl)F 10N-007 c1ccc(cc1)c2ccccc2NNC(=S)N 10N-008 CN(C)c1ccc(cc1)NC(=S)N 10N-009 c1cc(ccc1C(=O)C/C=N/OCc2cnc(s2)Cl)Br 10N-010 CC(C)(C)c1ccc(cc1)NC(=S)NC(=O)c2ccccc2 10N-011 c1ccc(cc1)NC(=O)OCc2cnc(s2)Cl 10N-012 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)C(c3ccccc3)(c4ccccc4)c5ccccc5 10N-013 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)OCCO3 10N-014 CC(C)(C)c1ccc(cc1)NC(=S)N 10N-015 c1ccc(cc1)C(=O)NC(=S)Nc2c(c(c(c(c2F)F)F)F)F 10N-016 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2cc4ccccc4c3 10N-017 c1cc(c(cc1NC(=O)OCc2cnc(s2)Cl)Cl)Cl 10N-018 c1cc2c(cc1NC(=S)N)OCCO2 10N-019 c1c(sc(n1)Cl)COC(=O)NC2CCCCC2 10N-020 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)c4ccc(cc4)NC(=S)N 10N-021 c1ccc(cc1)CN2CCN(CC2)Cc3cnc(s3)Cl 10N-022 COC(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 10N-023 COC(=O)c1ccc(cc1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 10N-024 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2CCCC3 10N-025 c1cc(cc(c1)Cl)NC(=O)OCc2cnc(s2)Cl 10N-026 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)NC4CC4)O 10N-027 Cc1cccc(c1)C(=O)OCc2cnc(s2)Cl 10N-029 c1ccc2cc3c(cccc3NC(=S)N)cc2c1 10N-030 c1cc2c(c(c1)NC(=S)N)CCCC2 10N-031 c1cc(cc(c1)C(F)(F)F)C(=O)OCc2cnc(s2)Cl 10N-035 c1ccc(cc1)C(=O)NC(=S)Nc2cc3ccccc3c4c2cccc4 10N-036 c1ccc(cc1)c2cc(c(c(c2)c3ccccc3)NC(=S)NC(=O)c4ccccc4)c5ccccc5 10N-037 c1cc(sc1)C(=O)OCc2cnc(s2)Cl 10N-038 CN1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(=O)O 10N-040 c1ccc(cc1)c2cc(c(c(c2)c3ccccc3)NC(=S)N)c4ccccc4 10N-042 c1ccc2c(c1)cc(c3c2cccc3)NC(=S)N 10N-043 c1cc(cc2c1cc[nH]2)NC(=S)N 10N-044 c1cc(ccc1C(=O)OCc2cnc(s2)Cl)I 10N-045 c1cc(c(cc1Cl)Cl)COCc2cnc(s2)Cl 10N-046 CCOC(=O)c1c(c2cccc3c2n(c1=O)CC3)O 10N-047 CN1CCN(CC1)Cc2cnc(s2)Cl 10N-048 c1cc(ccc1C(=O)NN)OCc2ccc(c(c2)Cl)Cl 10N-053 c1cc2c(c(c1)N[NH3+])CCCC2.[Cl-] 10N-054 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 10N-056 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)CC(=O)c3ccc(cc3)F 10N-057 c1cc(ccc1CN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)O)Cl 10N-058 c1ccc(cc1)c2ccc(cc2)C3Cc4ccccc4C(C3)O 10N-059 c1ccc(cc1)Oc2ccccc2NN 10N-062 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)CC(=O)c3cccc(c3)[N+](=O)[O-] 10N-063 Cc1ccc(cc1)C(=O)CN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 10N-064 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)NC4CCCCC4)O 10N-065 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3ccc(c(c3)Cl)Cl 10N-066 c1ccc(cc1)Oc2ccc(cc2)NNC(=S)N 10N-067 CC(C)(C)c1ccc(cc1)NNC(=S)N 10N-068 c1cc(ccc1/C(=N/O)/N)OCc2cnc(s2)Cl 10N-071 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)NCc4ccc(cc4)F)O 10N-072 c1ccc(cc1)Oc2ccccc2NNC(=S)N 10N-073 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)[N+](=O)[O-] 10N-074 c1c(sc(n1)Cl)C=O 10N-075 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)NCc4ccco4)O 10N-078 CC(c1ccccc1)NC(=O)c2c(c3cccc4c3n(c2=O)CC4)O 10N-079 c1c(sc(n1)Cl)C=C(C#N)C#N 10N-081 c1cncnc1C(=S)N 10N-082 c1(c(c(c(c(c1F)F)F)F)F)NNC(=S)N 10N-084 c1c(cc(c(c1[N+](=O)[O-])N2CCCNCC2)[N+](=O)[O-])C(F)(F)F 10N-086 c1cc(c(c(c1)Cl)Cl)C(=O)OCc2cnc(s2)Cl 10N-088 c1c(sc(n1)Cl)COC(=O)C2CC2 10N-089 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)Nc4ccc(cc4)C(F)(F)F)O 10N-091 c1c(sc(n1)N2CCOCC2)C=O 10N-092 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)Nc4cc(cc(c4)Cl)Cl)O 10N-093 c1c(sc(n1)N2CCOCC2)/C=N/NC(=S)N 10N-096 c1cc(ccc1C(=O)NC(=S)Nc2ccc(cc2)[N+](=O)[O-])[N+](=O)[O-] 10N-098 c1cc(cc(c1)[N+](=O)[O-])/C=N/OCc2cnc(s2)Cl 10N-101 c1cc(cc(c1)[N+](=O)[O-])/C=N/OC(=O)c2ccc(cc2)Cl 10N-104 c1c(sc(n1)N2CCCCC2)C=O 10N-105 c1cc2c(cc1Cl)NC(=O)CCS2 10N-301S CN1c2ccsc2/C(=N/Nc3ccccc3)/CS1(=O)=O 10N-303S CCN1CCSc2c(ccs2)C1=O 10N-308S CC(C)(C)OC(=O)N1CCC(CC1)C(=S)N 10N-311S CSc1nc2c(c(n1)Sc3ccccc3)CCCC2 10N-312S CC(C)Sc1nc2c(c(n1)O)CCCC2 10N-313S c1ccc(cc1)C(=O)N2CCSc3c(ccs3)C2=O 10N-317S C#CCN1CCSc2c(ccs2)C1=O 10N-318S CN1c2cc(ccc2SCCC1=O)Cl 10N-321S Cc1ccc(cc1)CN2c3cc(ccc3SCCC2=O)Cl 10N-322S Cc1ccc(cc1)N/N=C/2\CS(=O)(=O)N(c3c2scc3)C 10N-324S CN1c2ccsc2/C(=N/Nc3ccc(cc3)F)/CS1(=O)=O 10N-326S CN1c2ccsc2/C(=N/Nc3ccc(c(c3)Cl)Cl)/CS1(=O)=O 10N-329S c1ccc(cc1)CN2c3cc(ccc3SCCC2=O)Cl 10N-331S c1cc(ccc1CN2c3cc(ccc3SCCC2=O)Cl)F 10N-332S c1cc(cc(c1)F)CN2c3cc(ccc3SCCC2=O)Cl 10N-333S c1cc(ccc1CN2c3cc(ccc3SCCC2=O)Cl)Cl 10N-334S C=CCSc1[nH]c(=O)c2ccccc2n1 10N-335S CN1c2ccsc2/C(=N/N)/CS1(=O)=O 10N-336S c1ccc(cc1)C(=NNC(=O)COc2ccc(cc2Cl)Cl)c3ccccc3 10N-337S Cc1ccc(cc1)OCC(=O)NN=C(c2ccccc2)c3ccccc3 10N-338S COc1ccc(cc1)OCC(=O)NN=C(c2ccccc2)c3ccccc3 10N-339S Cc1ccc(c(c1)[N+](=O)[O-])OCC(=O)NN=C(c2ccccc2)c3ccccc3 10N-340S c1ccc(cc1)C(=NNC(=O)COc2ccc3ccccc3c2)c4ccccc4 10N-341S c1ccc(cc1)C(=NNC(=O)CSc2ccccc2)c3ccccc3 10N-342S c1ccc(cc1)C(=NNC(=O)CSc2ccc(cc2)Cl)c3ccccc3 10N-343S c1ccc(cc1)C(=NNC(=O)CSc2c(cccc2Cl)Cl)c3ccccc3 10N-344S Cc1ccc(cc1)SCC(=O)NN=C(c2ccccc2)c3ccccc3 10N-345S COc1cccc(c1)SCC(=O)NN=C(c2ccccc2)c3ccccc3 10N-346S COC(=O)c1ccccc1SCC(=O)NN=C(c2ccccc2)c3ccccc3 10N-347S CNCC(=O)NN=C(c1ccccc1)c2ccccc2 10N-348S C=CCNCC(=O)NN=C(c1ccccc1)c2ccccc2 10N-349S c1ccc(cc1)C(=NNC(=O)CNC2CCCCC2)c3ccccc3 10N-350S CC(=O)Cn1c(=O)c(c(cn1)Br)Br 10N-351S CC(=O)Cn1c(=O)c(c(cn1)N2CCOCC2)Br 10N-352S c1ccc2c(c1)c(=O)n3c(n2)SCC3CBr 10N-363S CC(=O)Cn1c(=O)cc(cn1)N2CCOCC2 10N-364S c1ccc(c(c1)CN2c3cc(ccc3SCCC2=O)Cl)Cl 10N-365S c1cc(cc(c1)Cl)CN2c3cc(ccc3SCCC2=O)Cl 10N-366S CN1c2ccsc2/C(=N/NC(=O)c3ccccc3)/CS1(=O)=O 10N-368S Cc1ccc(cc1)C(=O)N/N=C/2\CS(=O)(=O)N(c3c2scc3)C 10N-369S COc1ccc(cc1)CN2c3cc(ccc3SCCC2=O)Cl 10N-370S CC(C)(C)c1ccc(cc1)CN2c3cc(ccc3SCCC2=O)Cl 10N-371S c1cc(c(cc1CN2c3cc(ccc3SCCC2=O)Cl)Cl)Cl 10N-372S Cc1ccccc1CN2c3cc(ccc3SCCC2=O)Cl 10N-374S c1cc(c(cc1Cl)Cl)CN2c3cc(ccc3SCCC2=O)Cl 10N-375S C=C1CSc2n1c(=O)c3ccccc3n2 10N-376S C#CCSc1[nH]c(=O)c2ccccc2n1 10N-377S Cc1ccc(cc1)SCC2CSc3n2c(=O)c4ccccc4n3 10N-499S CC(=O)Cn1c(=O)c(c(cn1)N2CCCCC2)Cl 10N-501S CC(=O)Cn1c(=O)c(c(cn1)N(C)Cc2ccccc2)Cl 10N-502S CN(c1c2ccccc2nc(n1)SC)N 10N-503S CN(c1c2ccccc2nc(n1)SC)NC(=O)c3ccc(cc3)Cl 10N-504S CN(c1c2ccccc2nc(n1)SC)NC(=O)c3cccs3 10N-505S CN(c1c2ccccc2nc(n1)SC)NC(=O)c3ccccc3 10N-506S CN(c1c2ccccc2nc(n1)SC)NC(=O)c3ccc(cc3)F 10N-507S Cc1cccc(c1)C(=O)NN(C)c2c3ccccc3nc(n2)SC 10N-508S Cn1c2c(cn1)C(=O)CCC2 10N-510S C/C(=N\O)/Cn1c(=O)c(c(cn1)N2CCOCC2)Cl 10N-511S C/C(=N/OC(=O)c1ccc(cc1)Cl)/Cn2c(=O)cc(c(n2)Cl)N3CCOCC3 10N-512S Cn1c2c(cn1)C(=O)/C(=C/c3ccc(cc3Cl)Cl)/CC2 10N-514S c1cc(ccc1NC=C2C(=O)CCCC2=O)Cl 10N-519S c1c(cc(cc1Cl)Cl)NC=C2C(=O)CCCC2=O 10N-520S c1cc(c(cc1NC=C2C(=O)CCCC2=O)Cl)Cl 10N-521S c1cc(c(c(c1)Cl)Cl)NC=C2C(=O)CCCC2=O 10N-522S c1cc(c(cc1Cl)Cl)NC=C2C(=O)CCCC2=O 10N-523S c1cc(ccc1NC=C2C(=O)CCCC2=O)Br 10N-524S COc1ccc(cc1)NC=C2C(=O)CCCC2=O 10N-525S COC(=O)CSc1ncc(c(n1)O)S(=O)(=O)c2ccccc2 10N-561S c1ccc(cc1)CSc2ncc(c(n2)O)S(=O)(=O)c3ccccc3 10N-562S C#CCSc1ncc(c(n1)O)S(=O)(=O)c2ccccc2 10N-563S Cc1c(c(n(n1)c2ccccc2)/N=C/N(C)C)C=O 10N-564S CCC1CS/C(=N\c2ccccc2)/N1 10N-567S CCC1CS/C(=N\c2cccc(c2)C(F)(F)F)/N1 10N-568S c1ccc(cc1)CN2c3ccccc3CCCC2=O 10N-577S CC(C)(C)c1ccc(cc1)Oc2c3cnn(c3nc(n2)SC)c4ccccc4 10N-641S CSc1nc2c(cnn2c3ccccc3)c(n1)Oc4ccc(cc4)F 10N-642S CSc1nc2c(cnn2c3ccccc3)c(n1)Oc4cccc(c4)C(F)(F)F 10N-644S CSc1nc2c(cnn2c3ccccc3)c(n1)Oc4cc(c(cc4Cl)Cl)Cl 10N-645S CC(C)Nc1c2cnn(c2nc(n1)SC)c3ccccc3 10N-646S CSc1nc(c2cnn(c2n1)c3ccccc3)NCC=C 10N-647S CSc1nc2ccccc2c(n1)Oc3ccc(cc3)Cl 10N-650S COC(=O)c1c(ccs1)Oc2c3ccccc3nc(n2)SC 10N-652S CSc1nc2ccccc2c(n1)Oc3ccc(cc3)F 10N-653S CSc1nc2ccccc2c(n1)Oc3cccc(c3)C(F)(F)F 10N-654S COc1ccc(cc1)Oc2c3ccccc3nc(n2)SC 10N-655S CSc1nc2ccccc2c(n1)Oc3cc(ccc3Cl)Cl 10N-656S CSc1nc2ccccc2c(n1)Oc3ccc4ccccc4c3 10N-657S CSc1nc2ccccc2c(n1)Oc3ccc(cc3F)F 10N-658S CSc1nc2ccccc2c(n1)Sc3ccc(cc3)F 10N-663S CSc1nc2ccccc2c(n1)Sc3cc(ccc3Cl)Cl 10N-664S CSc1nc2ccccc2c(n1)Sc3ccc(cc3)Cl 10N-665S Cc1ccc(cc1)Sc2c3ccccc3nc(n2)SC 10N-666S CSc1nc2ccccc2c(n1)Sc3cccc(c3)Cl 10N-667S CSc1nc2ccccc2c(n1)Sc3ccccc3Cl 10N-668S COc1cccc(c1)Sc2c3ccccc3nc(n2)SC 10N-669S Cc1cccc(c1)Sc2c3ccccc3nc(n2)SC 10N-670S CSc1nc2ccccc2c(n1)Sc3ccc(cc3Cl)Cl 10N-671S CSc1nc2ccccc2c(n1)Sc3ccccc3 10N-672S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)Cl)Cl 10N-673S CSc1nc2ccccc2c(n1)Oc3cc(c(cc3Cl)Cl)Cl 10N-674S CC(C)(C)c1ccc(cc1)Oc2c3ccccc3nc(n2)SC 10N-675S COc1ccc(cc1OC)CCOC(=O)Nc2c(ccs2)OC 10N-676S COc1ccsc1NC(=O)OCc2ccc(cc2)Cl 10N-677S CSc1nc(cc(n1)Sc2ccc(cc2)Cl)C(F)(F)F 10N-678S CSc1nc(cc(n1)Oc2cc(c(cc2Cl)Cl)Cl)C(F)(F)F 10N-679S c1cc(cnc1)Cn2ccc(c(c2=O)Cc3ccc(cc3)F)O 10N-700 Cc1ccc(cc1)CO/N=C/c2cn(c(=O)c(c2O)Cc3ccc(cc3)F)Cc4ccc(cc4)OC 10N-703 c1ccc(c(c1)NC(=O)OCc2cncs2)F 10N-704 c1cc(ccc1NC(=O)OCc2cncs2)F 10N-705 CCOC(=O)C(Cc1ccc(cc1)F)c2ccnn2c3c(cc(cn3)C(F)(F)F)Cl 10N-710 c1ccc2c(c1)cccc2NC(=O)OCc3cncs3 10N-712 c1c(cnc(c1Cl)OCc2cncs2)C(F)(F)F 10N-713 c1ccc(cc1)COCc2cncs2 10N-714 CC(C)Oc1ccc(c(c1Cc2c(cccc2Cl)F)OC(C)C)C=O 10N-716 c1ccc2c(c1)Nc3c(cccn3)C(=O)N2CCCF 10N-721 c1cc(ccc1Cc2c(ccn(c2=O)CC3CCCO3)O)F 10N-722 c1cc(ccc1Cc2c(ccn(c2=O)NC(=O)c3ccc(cc3)Cl)O)F 10N-723 CC(=O)c1csc(n1)c2ccccc2 10N-724 c1c(cnc(c1Cl)Sc2nnc(s2)S)C(F)(F)F 10N-725 Cc1cc(cc(c1)n2ccc(c(c2=O)Cc3ccc(cc3)F)O)C 10N-727 CCOC(=O)CSc1nc2ccccc2s1 10N-728 C1CCC(C1)Sc2nnc(s2)S 10N-730 c1cc(c(nc1)Sc2nnc(s2)S)[N+](=O)[O-] 10N-731 c1cc(ccc1Cc2c(ccn(c2=O)CCCn3ccnc3)O)F 10N-732 c1cc(ccc1Cc2c(ccn(c2=O)CCCN3CCOCC3)O)F 10N-733 CCOC(=O)C(Cc1ccc(cc1)F)c2ccnn2c3c(cc(cc3Cl)Cl)Cl 10N-734 c1c(cc(c(c1[N+](=O)[O-])Sc2nnc(s2)SC3CCCC3)[N+](=O)[O-])C(F)(F)F 10N-737 c1ccc2c(c1)C(=O)N(C2=O)CCSc3nnc(s3)S 10N-738 c1c(cnc(c1Cl)n2cc(cc(c2=O)Cl)C(F)(F)F)C(F)(F)F 10N-740 c1ccc(cc1)CSc2nnc(s2)SC3CCCC3 10N-741 c1ccc(c(c1)CSc2nnc(s2)SC3CCCC3)F 10N-742 CCCCn1ccc(c(c1=O)Cc2ccc(cc2)F)O 10N-743 CCOC(=O)C(Cc1ccc(cc1)F)C(=O)C/C=N/OCc2ccc(cc2Cl)Cl 10N-744 c1cc(ccc1C(=O)CSc2nnc(s2)SC3CCCC3)Cl 10N-745 c1ccc(cc1)Cc2c(ccn(c2=O)c3cccc(c3)Oc4c(cc(cn4)C(F)(F)F)Cl)O 10N-747 CC1(C(=C(C(=C(C#N)C#N)N1)C#N)C(=O)c2ccccc2)O 10N-801 CCOC1=C(C(=C(C#N)C#N)NC1(C(F)(F)F)O)C#N 10N-803 CO/N=C/Nc1c2ccsc2ncn1 10N-805 c1cc(ccc1CO/N=C/Nc2c3ccsc3ncn2)Cl 10N-806 COc1ccc(cc1)CO/N=C/Nc2c3ccsc3ncn2 10N-807 c1cc(cc(c1)C(F)(F)F)CO/N=C/Nc2c3ccsc3ncn2 10N-808 Cc1c(c(c([nH]1)C(C#N)C#N)C#N)C(=O)c2ccccc2 10N-809 Cc1c(c(c([nH]1)C(=O)O)C#N)C(=O)c2ccccc2 10N-811 c1cc(c(c(c1)Cl)CO/N=C/Nc2c3ccsc3ncn2)F 10N-812 c1cc(cc(c1)OCCO/N=C/Nc2c3ccsc3ncn2)C(F)(F)F 10N-813 Cc1ccc(cc1)CO/N=C/Nc2c3ccsc3ncn2 10N-814 c1ccc(c(c1)CO/N=C/Nc2c3ccsc3ncn2)F 10N-815 c1cc(cc(c1)Cl)CO/N=C/Nc2c3ccsc3ncn2 10N-816 c1cc(c(c(c1)Cl)F)CO/N=C/Nc2c3ccsc3ncn2 10N-817 c1cc(c(cc1Cl)Cl)CO/N=C/Nc2c3ccsc3ncn2 10N-819 c1cc(c(c(c1)Cl)CO/N=C/Nc2c3ccsc3ncn2)Cl 10N-820 CCCn1ccc(c(c1=O)Cc2ccc(cc2)Cl)O 10N-821 c1ccc(cc1)Cn2ccc(c(c2=O)Cc3ccc(cc3)Cl)O 10N-823 COCCn1ccc(c(c1=O)Cc2ccc(cc2)Cl)O 10N-825 COc1cccc(c1)Cn2ccc(c(c2=O)Cc3ccc(cc3)Cl)O 10N-826 CCn1c(c(c(c1C(=O)O)C#N)C(=O)c2ccccc2)C 10N-827 c1cc(cc(c1)Cl)Cn2ccc(c(c2=O)Cc3ccc(cc3)Cl)O 10N-828 c1cc(ccc1Cc2c(ccn(c2=O)C3CCCCCC3)O)Cl 10N-829 CN(C)CCn1ccc(c(c1=O)Cc2ccc(cc2)Cl)O 10N-830 c1cc2c(cc1Cl)ncnc2O 10N-832 COc1ccc(cc1)n2ccc(c(c2=O)Cc3ccc(cc3)Cl)O 10N-833 COc1cc2c(cc1OC)nc[nH]c2=O 10N-834 COc1cccc(c1)CNc2c3ccc(cc3ncn2)Cl 10N-835 COC(=O)Cn1ccc(c(c1=O)Cc2ccc(cc2)Cl)O 10N-836 c1cc(ccc1c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N)N 10N-900 CCn1c2ccccc2c3c1ccc(c3)/C=C(/C#N)\C(=O)OCC 10N-901 CCOC(=O)/C(=C/c1ccc(cc1)C(C)(C)C)/C#N 10N-904 CC(C)(C)c1ccc(cc1)c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N 10N-906 CCOC(=O)/C(=C/c1ccc(cc1)C(F)(F)F)/C#N 10N-907 c1cc(ccc1c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N)C(F)(F)F 10N-909 CCOC(=O)C(=Cc1ccc(cc1)C(=O)OC)C#N 10N-910 CCOC(=O)C(=Cc1ccc2c(c1)OCCO2)C#N 10N-913 c1cc(ccc1c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N)OC(F)(F)F 10N-918 CCOC(=O)C(=Cc1cccc(c1)OC(F)(F)F)C#N 10N-919 c1cc(cc(c1)OC(F)(F)F)c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N 10N-921 COc1ccc(cc1F)c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N 10N-927 c1cc(c(cc1[N+](=O)[O-])Br)N2CCCCCC2 10P-001 CCOC(=O)C(CSCCCN1C(=O)c2ccccc2C1=O)[NH3+].C(=O)(C(F)(F)F)[O-] 10P-004 C/C(=N\N=C\1/NC(=O)CS1)/c2ccccc2 10P-007 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3nnc(o3)S 10P-011 CCOC(=O)C(=Cc1ccc(cc1)Cl)C(=O)OCC 10P-012 CN1CCN(CC1)c2ccc(cc2Br)[N+](=O)[O-] 10P-015 CCOC(=O)C(CSCc1ccccc1)NC(=O)OC(C)(C)C 10P-018 CN1CCN(CC1)c2ccc(cc2Br)N 10P-020 CCOC(=O)/C=C(/C)\N1CCCC1 10P-022 CC(C)(C)OC(=O)N1CCC(CC1)COS(=O)(=O)C 10P-023 c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)Cl 10P-024 CCOC(=O)C(CSCc1ccc(cc1)[N+](=O)[O-])NC(=O)OC(C)(C)C 10P-029 c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)F 10P-030 CCc1ccc(cc1)CSc2nnc(o2)c3ccccc3 10P-031 Cc1ccc(cc1)CSc2nnc(o2)c3ccccc3 10P-032 c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)[N+](=O)[O-] 10P-033 c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)Br 10P-034 CCOC(=O)C(CSCC=C)NC(=O)OC(C)(C)C 10P-036 CC(C(=O)OC)Oc1ccc(c(c1)F)c2ccccc2 10P-037 CCOC(=O)C1(CC1c2ccccc2)C(=O)OCC 10P-038 c1ccc(cc1)c2nnc(o2)SCC(=O)c3ccc(cc3)Br 10P-039 c1cc(ccc1C2=C(CCC(=O)N2)C#N)Oc3ccc(c(c3)F)Cl 10P-040 c1ccc(cc1)c2nnc(o2)SCc3ccccc3Cl 10P-041 CCOC(=O)CSCC(C(=O)OCC)NC(=O)OC(C)(C)C 10P-042 CCOC(=O)C(CSCCCC(=O)OC)NC(=O)OC(C)(C)C 10P-044 c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)C(F)(F)F 10P-048 c1cc(ccc1CSC(=[NH2+])N)F.[Cl-] 10P-049 c1ccc(cc1)c2nnc(o2)SCCCF 10P-050 c1ccc(cc1)c2ccc(cc2F)OCCCF 10P-053 CC(C(=O)C)Oc1ccc(c(c1)F)c2ccccc2 10P-054 c1ccc(cc1)c2nnc(o2)SCc3cc(cc(c3)C(F)(F)F)C(F)(F)F 10P-057 c1ccc(cc1)c2nnc(o2)SCCOc3ccccc3 10P-058 c1ccc(cc1)c2nnc(o2)SCC(=O)c3ccc(cc3Cl)Cl 10P-060 CCOC(=O)C(CSCCC(=O)O)NC(=O)OC(C)(C)C 10P-065 c1ccc(cc1)c2nnc3n2N=C(CS3)c4ccc(cc4Cl)Cl 10P-068 c1ccc(cc1)c2ccc(cc2F)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 10P-069 CCOC(=O)C(CSc1c(cc(cn1)C(F)(F)F)Cl)NC(=O)OC(C)(C)C 10P-070 CCOC(=O)C(CSCC(=O)O)NC(=O)OC(C)(C)C 10P-071 CCOC(=O)C(CSC(=O)CCC(=O)O)NC(=O)OC(C)(C)C 10P-072 CC(c1cc[nH]n1)Oc2ccc(c(c2)F)c3ccccc3 10P-073 c1ccc(cc1)c2nnc3n2N=C(CS3)c4ccc(cc4)Br 10P-074 c1ccc(cc1)c2ccc(cc2)C(=O)CSc3nnc(o3)c4ccccc4 10P-075 c1ccc(cc1)CSC(=[NH2+])N.[Cl-] 10P-076 c1cc(ccc1CSC(=[NH2+])N)C(F)(F)F.[Cl-] 10P-077 Cc1ccc(cc1)CSC(=[NH2+])N.[Cl-] 10P-079 c1cc(c(cc1CSC(=N)N)Cl)Cl.Cl 10P-080 c1cc(cc(c1)Cl)CSC(=[NH2+])N.[Cl-] 10P-081 c1ccc(cc1)c2ccc(cc2F)Oc3ncccn3 10P-082 c1cc(ccc1c2nccc(n2)c3ccc(cc3)F)O 10P-083 c1ccc(cc1)c2ccc(cc2F)Oc3c(cc(cn3)C(F)(F)F)Cl 10P-084 CCc1ccc(cc1)COc2ccc(c(c2)F)c3ccccc3 10P-086 c1cc(oc1)c2nnc(o2)S 10P-087 c1c(c(cc2c1OCO2)Br)/C=N/O 10P-088 c1cc(c(cc1Cl)Cl)CO/N=C/c2cc3c(cc2Br)OCO3 10P-089 c1ccc(c(c1)/C=C/2\C(=O)NC(=O)S2)Oc3cccc(c3)C(F)(F)F 10P-090 c1c(c(cc2c1OCO2)Br)/C=C\3/C(=O)NC(=O)S3 10P-091 c1ccc(c(c1)C#N)NC(=S)N 10P-0922 CC(C)(C)OC(=O)NC(CSCc1ccccc1)C(=O)O 10P-093 c1cc(ccc1c2cn(c(n2)SCc3ccc(c(c3)Cl)Cl)CC(=O)c4ccc(cc4)Cl)Cl 10P-097 Cc1ccc(cc1)CO/N=C/c2cc3c(cc2Br)OCO3 10P-098 c1cc(oc1)c2nnc(o2)SCc3ccc(cc3)Cl 10P-101 c1ccc(cc1)c2nnc(o2)S(=O)(=O)Cc3ccccc3Cl 10P-102 c1c(c(cc2c1OCO2)Br)CO 10P-113 c1ccc(cc1)c2nnc(o2)S(=O)(=O)CCOc3ccccc3 10P-114 c1cc(oc1)c2nnc(o2)SCC(=O)c3ccc(cc3)Cl 10P-115 c1cc(oc1)c2nnc3n2N=C(CS3)c4ccc(cc4)Cl 10P-116 CCOC(=O)C(=Cc1ccc(cc1)F)C(=O)OCC 10P-119 Cc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)O 10P-121 COC(=O)C1CCN(CC1)c2ccc(cc2Br)[N+](=O)[O-] 10P-122 CC(C(=O)O)Oc1ccc(c(c1)F)c2ccccc2 10P-123 CCOC(=O)C(CSCC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C 10P-124 CCOC(=O)C(CSCC(=O)OCC=C)NC(=O)OC(C)(C)C 10P-125 CCOC(=O)C(CSCC(=O)c1ccc(cc1Cl)Cl)NC(=O)OC(C)(C)C 10P-126 CN1CCN(CC1)c2ccc(cc2Br)NC(=O)c3cccc(c3)C(F)(F)F 10P-127 CCOC(=O)C(CSCC(=O)c1ccc(cc1)Cl)NC(=O)OC(C)(C)C 10P-128 CCOC(=O)C(CSCC(=O)c1ccc(cc1)Br)NC(=O)OC(C)(C)C 10P-129 CCOC(=O)C(CSC(=O)Cc1ccccc1)NC(=O)OC(C)(C)C 10P-130 CCOC(=O)C(CSC(=O)c1cccc(c1)Cl)NC(=O)OC(C)(C)C 10P-131 c1cc(ccc1CSC(=[NH2+])N)[N+](=O)[O-].[Cl-] 10P-132 CC(c1ccn(n1)C(=O)c2ccccc2)Oc3ccc(c(c3)F)c4ccccc4 10P-134 COc1ccc(cc1)c2c(c[nH]n2)C=O 10P-136 c1ccc2c(c1)c(c[nH]2)CCNc3ccc(cc3Br)[N+](=O)[O-] 10P-138 CCOC(=O)C(CSC(=O)c1ccc(cc1)F)NC(=O)OC(C)(C)C 10P-140 CCOC(=O)C(CSC(=O)c1ccc(cc1)[N+](=O)[O-])NC(=O)OC(C)(C)C 10P-141 c1cc(oc1)c2nnc(o2)SCC(=O)c3ccc(cc3)Br 10P-142 c1cc(c(c(c1)Cl)CSC(=[NH2+])N)F.[Cl-] 10P-143 CCOC(=O)C(CSC(=O)c1cc(cc(c1)Cl)Cl)NC(=O)OC(C)(C)C 10P-144 CCOC(=O)C(CSC(=O)/C=C(\C)/C(=O)O)NC(=O)OC(C)(C)C 10P-145 Cc1ccc(cc1)CSc2nnc(o2)c3ccco3 10P-147 Cc1cc(c(c(c1)C)CSc2nnc(o2)c3ccco3)C 10P-148 c1ccc(cc1)/C=C/CSc2nnc(o2)c3ccco3 10P-149 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)O 10P-150 Cc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OCc4ccc(c(c4)Cl)Cl 10P-151 CCOC(=O)C(CSCC(=O)c1ccc(c(c1)Cl)Cl)NC(=O)OC(C)(C)C 10P-152 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)O 10P-154 Cc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OCC#N 10P-155 c1cc(ccc1c2nccc(n2)c3ccc(cc3Cl)Cl)O 10P-156 c1cc(c(cc1[N+](=O)[O-])Br)N2CCOCC2 10P-162 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)c4ccc(cc4)O 10P-163 c1cc(ccc1c2nccc(n2)c3ccc(cc3)Br)O 10P-164 Cc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OCc4ccc(cc4)[N+](=O)[O-] 10P-165 CN(Cc1ccccc1)CC(C(F)(F)F)O 10P-200 c1c(cc(c(c1/C=N/C2CCCCCC2)O)Br)Br 10P-201 c1cc(c(c(c1)Cl)/C=C/2\CC(=O)C3CCN2CC3)F 10P-202 C1CN(CCN1CCO)CC(C(F)(F)F)O 10P-203 c1cc(c(cc1Cl)Cl)/C(=N\O)/c2cc3cc(cc(c3o2)Br)Br 10P-205 c1cc(ccc1/C(=N\O)/c2cc3cc(cc(c3o2)Br)Br)Br 10P-206 c1ccc(cc1)CC(C(=O)O)N2CCS(=O)(=O)CC2 10P-208 c1ccnc(c1)CCN2CCS(=O)(=O)CC2 10P-209 c1ccc(cc1)CCN2CCS(=O)(=O)CC2 10P-211 c1ccc2c(c1)c(n[nH]2)N 10P-212 c1ccc(c(c1)C(=O)O)N2CCS(=O)(=O)CC2 10P-213 c1ccc(cc1)C(=O)NC(=S)Nc2c3ccccc3[nH]n2 10P-216 COc1cccc2c1oc(c2)C(=O)c3ccccc3Cl 10P-217 C1CN(CCN(C1)CC(C(F)(F)F)O)CC(C(F)(F)F)O 10P-220 c1ccc2c(c1)c(n[nH]2)NC(=S)N 10P-221 CN1CCN(CC1)CC(C(F)(F)F)O 10P-225 CCOC(=O)c1cnc2ccc(cc2c1Nc3ccc(cc3)C)OC 10P-304S CCOC(=O)c1cnc2ccc(cc2c1Nc3ccc(cc3)C(F)(F)F)OC 10P-305S CCOC(=O)c1cnc2ccc(cc2c1Nc3ccccc3)OC 10P-306S CCOC(=O)c1cnc2ccc(cc2c1Nc3ccc(cc3)OC)OC 10P-307S CCOC(=O)c1cnc2ccc(cc2c1Sc3ccccc3)C 10P-311S CCOC(=O)c1cnc2ccc(cc2c1Sc3ccc(cc3)F)C 10P-312S CCOC(=O)c1cnc2ccc(cc2c1Sc3ccccc3C(=O)OC)C 10P-313S CCOC(=O)c1cnc2ccc(cc2c1Sc3cccc(c3)C(F)(F)F)C 10P-314S CCOC(=O)c1cnc2ccc(cc2c1Sc3ccc(cc3)C)C 10P-315S CCOC(=O)c1cnc2c(c1Sc3ccc(cc3C)C)cccc2C(F)(F)F 10P-316S c1cc2c(c(c1)C(F)(F)F)ncc(c2Sc3ccc(cc3)Cl)C(=O)O 10P-317S CCOC(=O)c1cnc2c(c1Oc3ccccc3)cccc2OC 10P-321S CCOC(=O)c1cnc2c(c1Oc3ccc(cc3)F)cccc2OC 10P-322S CCOC(=O)c1cnc2c(c1Oc3ccc4ccccc4c3)cccc2OC 10P-323S CCOC(=O)c1cnc2c(c1Oc3cccc(c3)C(F)(F)F)cccc2F 10P-324S CCOC(=O)c1cnc2c(c1Oc3ccccc3C(=O)OC)cccc2F 10P-325S CCN(CC)CC1(CCN(CC1)C(=O)c2ccc(c(c2)Cl)Cl)O 10P-337S c1ccc(cc1)c2c(c(sc2SCC#N)C#N)N 10P-339S Cc1ccc(cc1)c2nnc(n2N)S 10P-341S c1ccc(cc1)S(=O)(=O)N2CCC(=NOC(=O)c3ccc(cc3)Cl)CC2 10P-361S c1ccc(cc1)S(=O)(=O)N2CCC(=NOC(=O)c3ccc(cc3)F)CC2 10P-362S Cc1ccc(cc1)C(=O)ON=C2CCN(CC2)S(=O)(=O)c3ccccc3 10P-363S c1ccc(cc1)S(=O)(=O)N2CCC(=NOC(=O)c3cccc(c3)Cl)CC2 10P-365S c1ccc(cc1)S(=O)(=O)N2CCC(=NOC(=O)c3cccs3)CC2 10P-366S c1ccc(cc1)S(=O)(=O)N2CCC(=NOC(=O)C3CC3)CC2 10P-367S c1ccc(cc1)OCc2ccc(cc2)C(=O)O 10P-369S c1cc(c(cc1C(=O)N2CCC(CC2)(CO)F)Cl)Cl 10P-370S c1ccc(cc1)c2c(c(sc2SCC#N)C#N)NC(=O)c3ccccc3 10P-375S Cc1cccnc1NC(=O)OC(C)(C)C 10P-376S c1ccc(cc1)c2c(c(sc2SCC#N)C#N)NC(=O)c3ccc(cc3)F 10P-378S Cc1ccc(cc1)C(=O)Nc2c(sc(c2c3ccccc3)SCC#N)C#N 10P-379S CS(=O)(=O)ON=C1CCN(CC1)S(=O)(=O)c2ccccc2 10P-380S c1ccc(cc1)S(=O)(=O)N2CCC(=NOS(=O)(=O)c3ccccc3)CC2 10P-381S CCOC(=O)c1cnn(c1n2cccc2)c3ccccc3 10P-382S c1ccc(cc1)n2c(c(cn2)C(=O)O)n3cccc3 10P-383S c1ccc(cc1)S(=O)(=O)N2CCC(=NOS(=O)(=O)c3ccc(c(c3)Cl)Cl)CC2 10P-388S c1ccc(cc1)S(=O)(=O)N2CCC(=NOS(=O)(=O)c3ccccc3F)CC2 10P-389S c1ccc2c(c1)nnn2C(=O)n3c4ccccc4nn3 10P-392S c1ccc(cc1)S(=O)(=O)N2CCC(=NOS(=O)(=O)c3ccc(cc3)Br)CC2 10P-403S c1ccc(cc1)S(=O)(=O)N2CCC(=NOS(=O)(=O)c3ccc(cc3)Cl)CC2 10P-404S Cc1ccc(cc1)S(=O)(=O)ON=C2CCN(CC2)S(=O)(=O)c3ccccc3 10P-405S c1ccc(cc1)S(=O)(=O)N2CCC(=NOS(=O)(=O)c3ccc(cc3)F)CC2 10P-406S c1ccc(cc1)c2c(c(sc2SCC#N)C#N)NC(=O)C3CC3 10P-407S c1ccc(cc1)c2c(c(sc2SCC#N)C#N)NC(=O)c3ccc(cc3)Cl 10P-410S CC(C)C(=O)Nc1c(sc(c1c2ccccc2)SCC#N)C#N 10P-411S Cc1ccc(cc1)S(=O)(=O)n2ccc3c2nccc3 10P-414S c1ccc(cc1)CC(=O)Nc2c(sc(c2c3ccccc3)SCC#N)C#N 10P-415S c1cc(ccc1Sc2nc3ccsc3c(n2)N4CCOCC4)Br 10P-501S c1ccc(cc1)CNC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 10P-502S CCCNC(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 10P-503S CCN(CC)C(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 10P-504S c1cc2c(cc1[N+](=O)[O-])cc(s2)C(=O)NN3CCOCC3 10P-505S c1cc(cc(c1)n2c(cc(n2)C(=O)NN)c3ccc(cc3)Cl)C(F)(F)F 10P-507S c1ccc(cc1)C(=O)NNC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 10P-508S c1cc(sc1)C(=O)NNC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 10P-509S CC1CN(CC(O1)C)C(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 10P-510S c1ccc(cc1)NC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 10P-511S COC(=O)c1cc2cc(ccc2s1)NS(=O)(=O)c3ccc(cc3)Br 10P-512S COC(=O)c1cc2cc(ccc2s1)NS(=O)(=O)c3ccc(cc3)Cl 10P-513S Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)cc(s3)C(=O)OC 10P-514S COC(=O)c1cc2cc(ccc2s1)NS(=O)(=O)Cc3ccccc3 10P-516S COC(=O)c1cc2cc(ccc2s1)NS(=O)(=O)c3ccccc3 10P-517S COC(=O)c1cc2cc(ccc2s1)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl 10P-518S COC(=O)c1cc2cc(ccc2s1)NC(=O)c3ccc(cc3)Cl 10P-519S COC(=O)c1cc2cc(ccc2s1)NC(=O)c3ccc(cc3)F 10P-520S COC(=O)c1cc2cc(ccc2s1)NC(=O)c3cccc(c3)Cl 10P-521S COC(=O)c1cc2cc(ccc2s1)NC(=O)c3cccs3 10P-522S COC(=O)c1cc2cc(ccc2s1)NC(=O)c3ccccc3 10P-523S COC(=O)c1cc2cc(ccc2s1)NC(=O)c3cccc(c3)C(F)(F)F 10P-525S COC(=O)c1cc2cc(ccc2s1)NC(=O)c3ccccc3Cl 10P-526S c1cc2c(cc1[N+](=O)[O-])cc(s2)C(=O)NCCN3CCOCC3 10P-527S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)CSc4ccccc4Cl 10P-529S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)CSc4ccc(cc4Cl)Cl 10P-530S c1ccc(cc1)c2nnc(o2)c3cc4cc(ccc4s3)[N+](=O)[O-] 10P-531S c1cc(sc1)c2nnc(o2)c3cc4cc(ccc4s3)[N+](=O)[O-] 10P-532S c1ccc(cc1)c2c(snn2)C(=O)O 10P-535S C=CCNC(=O)c1c(nns1)c2ccccc2 10P-537S CC1CN(CC(O1)C)C(=O)c2c(nns2)c3ccccc3 10P-538S Cc1ccc2c(c1)c(=O)c3cc(ccc3s2)N 10P-569S CNC1=C(C(=O)C(O1)c2ccccc2)c3ccc(cc3)C(F)(F)F 10P-573S Cc1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4ccccc4Cl 10P-579S Cc1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4ccc(cc4)F 10P-580S Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)c(=O)c4cc(ccc4s3)C 10P-581S Cc1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4cccs4 10P-582S Cc1ccn2c(c1)nc(c2/C=C(\C#N)/c3cccc(c3)Cl)c4ccc(cc4)Cl 10P-641S Cc1ccn2c(c1)nc(c2/C=C(\C#N)/c3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl 10P-642S Cc1ccn2c(c1)nc(c2/C=C(\C#N)/c3ccccn3)c4ccc(cc4)Cl 10P-643S Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccc(cc3)OC 10P-646S Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3cccs3 10P-647S Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccc(cc3)Oc4ccccc4 10P-648S Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3c(cccc3Cl)F 10P-651S Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccco3 10P-652S Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccc(c(c3)OC)OC 10P-653S Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3cccc(c3)C(F)(F)F 10P-656S c1ccc(cc1)COC(=O)NCc2ccc(cc2)C(=O)O 10P-661S c1ccc(cc1)COC(=O)NCc2ccc(cc2)C(=O)NC3CCCCC3 10P-664S c1ccc(cc1)COC(=O)NCc2ccc(cc2)C(=O)Nc3ccc(cc3)Cl 10P-665S Cc1ccc(cc1)NC(=O)c2ccc(cc2)CNC(=O)OCc3ccccc3 10P-666S c1ccc(cc1)COC(=O)NCc2ccc(cc2)C(=O)Nc3cccc(c3)C(F)(F)F 10P-668S CNC(=O)c1ccc(cc1)CNC(=O)OCc2ccccc2 10P-669S c1cc(ccc1CNC(=O)OCC(F)(F)F)C(=O)O 10P-671S Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3ccc(cc3)Oc4ccccc4 10P-672S Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3cccs3 10P-673S Cc1c(sc(n1)c2ccccc2)c3cc[nH]n3 10P-700 Cc1c(sc(n1)c2ccccn2)C(=O)/C=C/c3ccccc3 10P-701 Cc1cccc(n1)n2cc(nc2)C(=O)O 10P-702 Cc1c(c(nc(n1)C)OCC(=O)N)I 10P-703 CC(=O)C(Cc1cccc(c1)C(F)(F)F)C(=O)C 10P-704 CC(=O)C(Cc1cccc(c1)C(F)(F)F)(Cc2cccc(c2)C(F)(F)F)C(=O)C 10P-705 CC(=O)C(Cc1cccc(c1)C(F)(F)F)Cc2cccc(c2)C(F)(F)F 10P-706 c1ccc(cc1)C2COC3N2C(CC3)n4c5ccccc5nn4 10P-707 Cc1c(sc(n1)c2ccccc2)c3ccnc(n3)N 10P-709 Cc1c(sc(n1)c2ccccn2)C(=O)CC(c3ccccc3)C(C#N)C#N 10P-711 c1ccc(c(c1)C(F)(F)F)n2cc(nn2)C(=O)c3ccc(cc3Cl)Cl 10P-713 c1ccc2c(c1)-c3ccccc3S(=O)(=O)N2 10P-714 CCOC(=O)c1ccc(cc1)n2cc(nn2)C(=O)c3cccs3 10P-715 Cc1ccc(cc1Cl)n2cc(nn2)C(=O)c3ccc(cc3)F 10P-716 CN(C)/C=C/c1c(nnn1c2ccc(cc2)OC(F)(F)F)C(=O)c3ccc(cc3)OC 10P-718 Cc1ccc(cc1Cl)n2cc(nn2)C(=O)C(C)Oc3ccc(cc3Cl)Cl 10P-720 Cc1ccc(cc1Cl)n2cc(nn2)C(=O)c3ccc(cc3)N4CCN(CC4)C 10P-721 Cc1c(c(nc(n1)C)OCc2ccc(cc2)C(F)(F)F)I 10P-722 CCOC(=O)COc1c(c(nc(n1)C)C)I 10P-723 C/C(=C\C(=O)c1ccncc1)/N(C)C 10P-724 CC(=O)C(Cc1cccc(c1)F)Cc2cccc(c2)F 10P-728 CC(=O)C(Cc1cccc(c1)F)(Cc2cccc(c2)F)C(=O)C 10P-729 Cc1c(sc(n1)c2ccncc2)c3ccnc(n3)N 10P-730 Cc1ccc(cc1Cl)n2c(c(nn2)C(=O)c3ccncc3)C 10P-731 c1cc(oc1)C(=O)c2cn(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F 10P-732 Cc1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccncc3 10P-733 CC(C(=O)c1cn(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Oc3cccc(c3)C(F)(F)F 10P-734 Cc1c(nnn1c2ccc(cc2)OC(F)(F)F)C(=O)c3ccncc3 10P-735 Cc1ccc(cc1Cl)n2cc(nn2)[N+](=O)[O-] 10P-737 Cc1c(sc(n1)c2cccnc2)c3ccnc(n3)N 10P-738 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccccc3 10P-739 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccccc3[N+](=O)[O-] 10P-740 Cc1ccc2cn[nH]c2c1[N+](=O)[O-] 10P-900 c1ccc2c(c1)c(cn2c3c(cccn3)C(F)(F)F)C=O 10P-904 Cc1cc2c(cc1[N+](=O)[O-])cn[nH]2 10P-906 c1cc(cc(c1)N2CCN(CC2)Cc3cnc(s3)Cl)C(F)(F)F 10P-909 CN(C)/C=C/C(=O)c1cc2cccc(c2o1)OC 10P-912 c1ccc(cc1)C(=O)NC(=S)Nc2ccccc2C#N 10P-913 COc1cc(c(c(c1)Br)O)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 10P-914 COc1cc(c(c(c1)Br)O)/C=N/NC(=O)c2ccco2 10P-915 Cc1ccc(cc1C)/N=C/c2cc(cc(c2O)Br)OC 10P-916 COc1cc(c(c(c1)Br)O)/C=N/NC(=O)c2cccnc2 10P-917 COc1cc(c(c(c1)Br)O)/C=N/c2ccc(cc2)C(=O)OC 10P-918 COc1cc(c(c(c1)Br)O)/C=N/NC(=O)c2ccc(cc2)Cl 10P-920 COc1cc(cc(c1O)C=O)Br 10P-921 COc1cccc2c1oc(c2)C(=O)c3ccc(cc3)Br 10P-923 c1ccc(cc1)C(=O)NC(=S)Nc2ccccc2OC(F)F 10P-924 Cc1cc(ccc1NC(=S)NC(=O)c2ccccc2)C(=O)OC 10P-926 Cc1ccc2c(c1NC(=S)NC(=O)c3ccccc3)C(=O)c4ccccc4C2=O 10P-927 Cc1cc(ccc1NC(=S)N)C(=O)O 10P-929 Cc1cccnc1NC(=S)N 10P-930 c1ccc(c(c1)NC(=S)N)OC(F)F 10P-931 c1ccc(c(c1)/C=C\2/C(=O)C3CCN2CC3)F 10P-932 c1ccc(c(c1)/C=C/2\CC(=O)C3CCN2CC3)C(F)(F)F 10P-933 c1ccc(c(c1)/C=C\2/C(C3CCN2CC3)O)C(F)(F)F 10P-934 COc1ccc(cc1)C(=O)c2cc3cccc(c3o2)OC 10P-935 COc1cccc2c1oc(c2)C(=O)c3ccc(cc3Cl)Cl 10P-936 C1CCC(CC1)OC(CN2CCCCC2)C(F)(F)F 10P-938 COc1cc(c(c(c1)Br)O)/C=N/Cc2ccc3c(c2)OCO3 10P-940 COc1cc(c(c(c1)Br)O)/C=N/c2ccc(cc2)C(F)(F)F 10P-941 COc1cc(c(c(c1)Br)O)/C=N/c2ccc(cc2)I 10P-942 COc1cc(c(c(c1)Br)O)/C=N/NC(=S)N 10P-943 CNC(=S)N/N=C/c1cc(cc(c1O)Br)Br 10P-944 COc1cc(cc(c1O)/C=N/NC(=O)c2ccc(cc2Cl)Cl)Br 10P-946 Cc1cccc(c1)/N=C/c2cc(cc(c2O)OC)Br 10P-947 COc1cc(cc(c1O)/C=N/c2cccc(c2)Br)Br 10P-948 COc1cc(cc(c1)OC)/N=C/c2cc(cc(c2O)OC)Br 10P-949 c1ccc(c(c1)CC2C(=O)C3CCN2CC3)C(F)(F)F 10P-950 c1ccc(c(c1)/C=C/2\CC(=O)C3CCN2CC3)F 10P-951 c1cc(ccc1NC(=O)OC(CN2CCCCC2)C(F)(F)F)Cl 10P-952 COc1ccc(cc1)NC(=O)OC(CN2CCCCC2)C(F)(F)F 10P-953 c1ccc(c(c1)/C=C\2/C(C3CCN2CC3)O)F 10P-954 c1ccc(cc1)NC(=O)OC(CN2CCCCC2)C(F)(F)F 10P-955 COc1cc(cc(c1O)/C=N/c2cccc(c2)C(=O)OC)Br 10P-956 COc1cc(cc(c1O)/C=N/c2ccc(cc2)F)Br 10P-957 c1cc(cc(c1)F)NC(=O)OC(CN2CCCCC2)C(F)(F)F 10P-959 COc1ccc(cc1OC)C/N=C/c2cc(cc(c2O)Br)OC 10P-960 c1cc(cc(c1)F)C(=O)OC(CN2CCCCC2)C(F)(F)F 10P-961 c1cc(cc(c1)Cl)C(=O)OC(CN2CCCCC2)C(F)(F)F 10P-963 COc1cccc(c1)C(=O)OC(CN2CCCCC2)C(F)(F)F 10P-964 c1cc(cc(c1)C(F)(F)F)C(=O)OC(CN2CCCCC2)C(F)(F)F 10P-965 c1cc(ccc1CC2C(=O)C3CCN2CC3)Cl 10P-966 c1cc(c(cc1Cl)Cl)C(=O)c2cc3cc(cc(c3o2)Br)Br 10P-967 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Br)Br)Br 10P-968 c1ccc(cc1)C(=O)c2cc3cc(cc(c3o2)Br)Br 10P-969 Cc1cc2c(cc1N)cn[nH]2 10P-970 c1ccc2c(c1)nnn2Cc3cnc(s3)Cl 10P-971 Cc1ccc2cn[nH]c2c1NC(=S)NC(=O)c3ccccc3 10P-972 c1ccc(cc1)NC(=O)OC\2C3CCN(/C2=C\c4ccccc4F)CC3 10P-973 COc1cc(c(c(c1)Br)O)/C=N/Cc2ccc(cc2)Cl 10P-975 COc1cccc2c1oc(c2)C(=O)O 10P-977 Cc1ccc2cn[nH]c2c1NC(=S)N 10P-978 C/C(=N\NC(=S)N)/c1cc2cccc(c2o1)OC 10P-980 c1cc(ccc1C/N=C/c2cc(cc(c2O)Br)Br)F 10P-981 Cc1cc2c(cc1NC(=S)NC(=O)c3ccccc3)cn[nH]2 10P-982 CN(Cc1ccccc1)Cc2cnc(s2)Cl 10P-983 c1cc(ccc1/C=C\2/C(=O)C3CCN2CC3)C(F)(F)F 10P-984 COc1cc(cc(c1O)/C=N/O)Br 10P-985 c1cc(ccc1/C=C\2/C(C3CCN2CC3)O)C(F)(F)F 10P-986 COc1cccc2c1oc(c2)/C(=N/O)/c3ccc(cc3)Br 10P-987 c1ccc(cc1)/C(=N/O)/c2cc3cc(cc(c3o2)Br)Br 10P-988 COc1cccc2c1oc(c2)/C(=N/O)/c3ccc(cc3Cl)Cl 10P-989 Cc1cc2c(cc1NC(=S)N)cn[nH]2 10P-990 c1cc(ccc1/C=C/2\CC(=O)C3CCN2CC3)C(F)(F)F 10P-991 COc1cc2cc(c(=O)oc2c(c1)Br)C(=O)O 10P-992 c1c2cc(c(=O)oc2c(cc1Br)Br)C(=O)O 10P-993 c1cc(c(c(c1)Cl)/C=C\2/C(=O)C3CCN2CC3)F 10P-995 c1cc(c(c(c1)Cl)C2=NOC(C2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 10P-996 c1ccc(c(c1)C/N=C/c2cc(cc(c2O)Br)Br)C(F)(F)F 10P-999 Cc1cc2nc(cc(n2n1)N)c3ccc(c(c3)Cl)Cl 10R-0002 Cc1c(c2nccc(n2n1)c3ccc(c(c3)[N+](=O)[O-])Cl)Br 10R-0006 Cc1c(c2nccc(n2n1)c3ccccn3)Br 10R-0008 Cc1cc(n(n1)c2nc(cs2)c3cccc(c3)C(F)(F)F)C 10R-0009 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(c(c3)Cl)Cl 10R-0010 c1cc(c(cc1c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F)Cl)Cl 10R-0011 CC(C)(C)OC(=O)N1CCC2(CCC(=O)O2)CC1 10R-0012 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)[N+](=O)[O-] 10R-0014 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)C 10R-0015 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc6ccccc6c5)C 10R-0024 c1cc(cc(c1)C(F)(F)F)C(C(=O)O)N 10R-0025 c1cc(ccc1S(=O)(=O)[O-])I.[K+] 10R-0026 Cc1cc2nccc(n2n1)c3ccc4ccccc4c3 10R-0027 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3cccc(c3)[N+](=O)[O-] 10R-0029 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3Cl)Cl 10R-0031 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)F 10R-0032 c1cc(oc1)c2cc(n3c(n2)cc(n3)c4ccc(c(c4)Cl)Cl)C(F)(F)F 10R-0033 c1cc(sc1)c2cc(n3c(n2)cc(n3)c4ccc(c(c4)Cl)Cl)C(F)(F)F 10R-0034 c1cc(cc(c1)Cl)c2cc(n3c(n2)cc(n3)c4ccc(c(c4)Cl)Cl)C(F)(F)F 10R-0035 c1ccc(cc1)c2cc(n3c(n2)cc(n3)c4ccc(c(c4)Cl)Cl)C(F)(F)F 10R-0036 Cc1cc(n2c(n1)cc(n2)c3ccc(c(c3)Cl)Cl)C(F)(F)Cl 10R-0037 COCc1cc(n2c(n1)cc(n2)c3ccc(c(c3)Cl)Cl)O 10R-0038 c1cc(ccc1C(C(=O)O)N)F 10R-0039 c1ccnc(c1)c2ccnc3n2nc(c3)c4ccc(c(c4)Cl)Cl 10R-0040 Cc1c(c2nccc(n2n1)c3ccc4ccccc4c3)Cl 10R-0042 c1cc(ccc1c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F)F 10R-0043 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F 10R-0044 Cc1cc(c(cc1F)[N+](=O)[O-])F 10R-0045 c1c(c(cc(c1F)[N+](=O)[O-])F)C(=O)O 10R-0046 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccccn5)C 10R-0050 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)c5ccc(cc5)F)C 10R-0051 CCc1c([nH]c(=O)n1CC)C(C)S(=O)(=O)c2ccccc2 10R-0200 CCn1cc(n(c1=O)Cc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)C 10R-0201 c1ccc(cc1)S(=O)(=O)C2C(N(C(=O)N2)c3ccc(cc3)OC(F)(F)F)O 10R-0202 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)C2CC2 10R-0204 c1cc(cnc1)CNC(=O)c2cc(c[nH]2)C(=O)C3CC3 10R-0205 c1cc(oc1)CNC(=O)c2cc(c[nH]2)C(=O)C3CC3 10R-0206 Cc1c([nH]c(=O)n1c2ccc(cc2)OC(F)(F)F)CS(=O)(=O)c3ccccc3 10R-0207 CCc1c([nH]c(=O)n1c2ccc(cc2)OC(F)(F)F)C(C)S(=O)(=O)c3ccccc3 10R-0213 Cc1ccccc1NC(=O)/C=C(\C)/N2CCN(CC2)c3ccccc3OC 10R-0214 CCc1c([nH]c(=O)n1c2ccc(cc2)OC(F)(F)F)C(C)S(=O)(=O)c3ccc(cc3)C 10R-0218 c1cc(ccc1CO/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])[N+](=O)[O-] 10R-0219 c1cc(cc(c1)F)CO/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 10R-0220 c1cc(ccc1CO/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl 10R-0221 Cc1ccc(cc1)S(=O)(=O)c2cn(c(=O)n2C)C 10R-0223 C#CCOc1ccc(cc1/C=C/C(=O)O)Cl 10R-0226 CC(=O)c1cc([nH]c1)C(=O)O 10R-0227 Cc1ccc(cc1)n2cc([nH]c2=O)S(=O)(=O)c3ccc(cc3)C 10R-0228 Cc1ccc(cc1)n2cc([nH]c2=O)S(=O)(=O)c3ccccc3 10R-0229 Cc1ccc(cc1)n2c(c([nH]c2=O)CS(=O)(=O)c3ccc(cc3)C)C 10R-0230 Cc1ccc(cc1)n2c(c([nH]c2=O)CS(=O)(=O)c3ccccc3)C 10R-0231 CCn1c(cn(c1=O)Cc2ccccc2)S(=O)(=O)c3ccc(cc3)C 10R-0232 C#CCOc1ccc(cc1CO)Cl 10R-0233 CCc1c([nH]c(=O)n1c2ccc(cc2)C)C(C)S(=O)(=O)c3ccc(cc3)C 10R-0236 CCc1c([nH]c(=O)n1c2ccc(cc2)C)C(C)S(=O)(=O)c3ccccc3 10R-0237 CCn1cc(n(c1=O)Cc2ccc(cc2)C(C)(C)C)S(=O)(=O)c3ccc(cc3)C 10R-0238 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)C2CC2 10R-0240 COC(=O)c1ccccc1OCC#C 10R-0241 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C4C=CC(C3C2=O)O4 10R-0244 CCc1c([nH]c(=O)n1Cc2ccc(c(c2)OC)OC)C(C)S(=O)(=O)c3ccccc3 10R-0245 CCc1c([nH]c(=O)n1Cc2cccc(c2)C(F)(F)F)C(C)S(=O)(=O)c3ccccc3 10R-0246 CCc1c([nH]c(=O)n1Cc2cccs2)C(C)S(=O)(=O)c3ccccc3 10R-0247 CCn1cc(n(c1=O)Cc2ccc(c(c2)Cl)Cl)S(=O)(=O)c3ccc(cc3)C 10R-0248 CC(C(=O)C)Oc1cccnc1 10R-0249 c1c(c[nH]c1C(=O)O)C(=O)C2CC2 10R-0250 c1c(c[nH]c1C(=O)NCC2CCCO2)C(=O)C3CC3 10R-0251 Cc1ccccc1CSc2nc3cc(c(cc3c(=N)n2Cc4ccco4)OC)OC 10R-0254 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccco3)SCc4c(cccc4Cl)F 10R-0255 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccco3)SCc4ccc(cc4)F 10R-0256 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccco3)SCc4c(cccc4Cl)Cl 10R-0257 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccco3)SCc4cnc(s4)Cl 10R-0258 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccco3)SCc4cccc(c4)C(F)(F)F 10R-0259 COCCCNC(=O)c1cc(c[nH]1)C(=O)C2CC2 10R-0260 Cc1ccc(c(c1)CSc2nc3cc(c(cc3c(=N)n2Cc4ccc(cc4)OC)OC)OC)C 10R-0263 COc1ccc(cc1Cl)Cn2c(=N)c3cc(c(cc3nc2SCc4ccccc4)OC)OC 10R-0264 Cc1ccccc1CSc2nc3cc(c(cc3c(=N)n2Cc4ccc(cc4)OC)OC)OC 10R-0265 CC(C)(C)c1ccc(cc1)CSc2nc3cc(c(cc3c(=N)n2Cc4ccc(cc4)OC)OC)OC 10R-0266 CCc1c([nH]c(=O)n1c2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(C)S(=O)(=O)c5ccc(cc5)C 10R-0267 CCc1c([nH]c(=O)n1CCNc2c(cc(cn2)C(F)(F)F)Cl)C(C)S(=O)(=O)c3ccccc3 10R-0268 COCCCn1c(=N)c2cc(c(cc2[nH]c1=S)OC)OC 10R-0270 COc1cc2c(cc1OC)nc(n(c2=N)C3CCCCCC3)SCCCC#N 10R-0271 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)CCc3ccccc3 10R-0272 COc1ccc(cc1)Cn2c(=N)c3cc(c(cc3nc2SCC4CO4)OC)OC 10R-0273 Cc1ccc(cc1)S(=O)(=O)c2cn(c(=S)n2C)C 10R-0274 c1ccc(cc1)c2c3c(c(c(n2)SCc4cccc(c4)C(F)(F)F)C#N)CCCC3 10R-0276 COCCn1c(=N)c2cc(c(cc2[nH]c1=S)OC)OC 10R-0278 Cc1cc2ncc(c(n2n1)N)c3ccc(cc3)OC 10R-0279 COCCCn1c(=N)c2cc(c(cc2nc1SCc3ccc(cc3)OC)OC)OC 10R-0280 COCCCn1c(=N)c2cc(c(cc2nc1SCCc3ccccc3)OC)OC 10R-0281 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NN 10R-0282 COCCCn1c(=N)c2cc(c(cc2nc1SCC(=O)O)OC)OC 10R-0283 COCCCn1c(=N)c2cc(c(cc2nc1SCc3cccc(c3)C(F)(F)F)OC)OC 10R-0284 COCCCn1c(=N)c2cc(c(cc2nc1SCc3ccccc3)OC)OC 10R-0286 CCCC(=O)c1cc([nH]c1)C(=O)NN 10R-0287 COCCCn1c(=N)c2cc(c(cc2nc1SCc3cccc(c3)OC)OC)OC 10R-0288 c1ccc(cc1)CSc2c(c3c(c(n2)c4ccccc4)CCCC3)C#N 10R-0289 c1ccc(cc1)c2c3c(c(c(n2)SCc4ccc(cc4)F)C#N)CCCC3 10R-0290 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NC2CCCCCC2 10R-0291 COc1cc2c(cc1OC)nc(n(c2=N)CCc3ccccc3)SCC#N 10R-0292 COc1cc2c(cc1OC)nc(n(c2=N)CCc3ccccc3)SCC(=O)N 10R-0293 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN=C(C=C3)C(F)(F)Cl 10R-0295 CC(=O)c1cc([nH]c1)C(=O)NC2CCCCCC2 10R-0296 COc1cc2c(cc1OC)nc(n(c2=N)CCc3ccccc3)SCc4ccc(cc4)C(F)(F)F 10R-0297 C#CCOc1ccc(cc1/C=N/O)Cl 10R-0299 c1ccc(cc1)c2c3c(c(c(n2)SCC(=O)N)C#N)CCCC3 10R-0300 c1cc(ccc1S(=O)(=O)N2CCN=C(C=C2)C(F)(F)Cl)Br 10R-0301 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN=C(C=C3)C(F)(F)Cl 10R-0302 Cc1ccc(cc1)C2C=C(NC(=O)N2)C(=O)O 10R-0303 c1ccc(cc1)/C(=N/C(=S)Nc2ccccc2)/N 10R-0304 COc1cc2c(cc1OC)nc(n(c2=N)CCc3ccccc3)SCc4ccncc4 10R-0305 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)Cl 10R-0306 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)Cl)C 10R-0307 c1cc(ccc1C(=O)N2CCN=C(C=C2)C(F)(F)Cl)Br 10R-0308 c1cc(ccc1S(=O)(=O)N2CCN=C(C=C2)C(F)(F)Cl)Cl 10R-0310 Cc1ccccc1C(=O)c2ccc([nH]2)C(=O)NC3CCCCCC3 10R-0311 c1c(c[nH]c1C(=O)NC2CCCCCC2)C(=O)C3CC3 10R-0312 CCOc1ccc(cc1)C2C=C(NC(=O)N2)C(=O)O 10R-0314 COc1ccc(c(c1)C2C=C(NC(=O)N2)C(=O)O)OC 10R-0315 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)Cc3cccs3 10R-0316 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)C3CCCCCC3 10R-0317 COc1cccc(c1)C2C(c3ccccc3C(=O)O2)C(=O)O 10R-0321 CC(C)(C)c1ccc(cc1)CSc2c(c3c(c(n2)c4ccccc4)CCCC3)C#N 10R-0322 COc1cc2c(cc1OC)nc(n(c2=N)C3CCCCCC3)SCc4cccnc4 10R-0324 COc1ccc(cc1)Cn2c(=N)c3cc(c(cc3[nH]c2=S)OC)OC 10R-0325 CCc1ccc(cc1)CSc2nc3cc(c(cc3c(=N)n2CCc4ccccc4)OC)OC 10R-0326 CCOC(=O)C1=C(NC(=O)NC1c2cc(ccc2OC)OC)C 10R-0327 c1cc(cc(c1)[N+](=O)[O-])C2C=C(NC(=O)N2)C(=O)O 10R-0328 c1c(c[nH]c1C(=O)C(Cl)(Cl)Cl)C(=O)C2CCCCC2 10R-0331 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccs3)SCCC(=O)c4ccccc4 10R-0333 COc1cc2c(cc1OC)nc(n(c2=N)C3CCCCCC3)SCCC(=O)c4ccccc4 10R-0334 COc1ccc(cc1)COC(=O)NC2=C(C(=O)c3ccccc3C2=O)Cl 10R-0335 COC(=O)c1cc(c[nH]1)C(=O)C2CCCCC2 10R-0336 COc1cc2c(cc1OC)nc(n(c2=N)C3CCCCCC3)SCC4CCCCO4 10R-0337 CCOC(=O)c1cn2c(n1)C=CC3C2N=C(C=C3C(F)(F)F)C(F)(F)F 10R-0339 CCOc1ccc(cc1)C2C(=C(NC(=S)N2)C)C(=O)OCC 10R-0340 c1ccc2c(c1)cccc2C3C=C(NC(=O)N3)C(=O)O 10R-0341 c1cc2c(cc1C3C=C(NC(=O)N3)C(=O)O)OCO2 10R-0342 COc1ccc(cc1)C2C=C(NC(=O)N2)C(=O)O 10R-0343 COc1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)C3CCCCC3 10R-0344 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)C2CCCCC2 10R-0345 c1c(c[nH]c1C(=O)NC2CCCCCC2)C(=O)C3CCCCC3 10R-0346 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2C4CCCCC4)C(=O)O 10R-0347 c1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)C3CCCCC3 10R-0349 c1cc(oc1)CNC(=O)c2cc(c[nH]2)C(=O)C3CCCCC3 10R-0350 c1c(c[nH]c1C(=O)NCC2CCCO2)C(=O)C3CCCCC3 10R-0354 c1cn(cn1)CCCNC(=O)c2cc(c[nH]2)C(=O)C3CCCCC3 10R-0355 c1c(c[nH]c1C(=O)NCCCN2CCOCC2)C(=O)C3CCCCC3 10R-0356 c1ccnc(c1)CCNC(=O)c2cc(c[nH]2)C(=O)C3CCCCC3 10R-0357 c1cnccc1CNC(=O)c2cc(c[nH]2)C(=O)C3CCCCC3 10R-0358 COc1ccc(cc1OC)COC(=O)NC2=C(C(=O)c3ccccc3C2=O)Cl 10R-0359 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cc(c[nH]3)C(=O)C4CCCCC4 10R-0360 c1c(c[nH]c1C(=O)O)C(=O)C2CCCCC2 10R-0361 c1cc(ccc1C(=O)N2CCNCC2)[N+](=O)[O-] 10R-0362 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccs3)SCc4ccc(cc4)C(F)(F)F 10R-0363 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccs3)SC/C=C/c4ccccc4 10R-0364 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccs3)SCc4ccc(cc4)F 10R-0365 Cc1ccc(cc1)C(=O)n2cc(c3c2cccc3)c4ccc(nn4)Cl 10R-0366 CCOC(=O)C1=C(NC(=O)NC1c2ccccc2)C 10R-0367 CCOC(=O)C1=C(NC(=S)NC1c2ccccc2)C 10R-0368 CCOC(=O)C1=C(N(C(=S)NC1c2ccccc2)C)C 10R-0369 COC(=O)/C=C/c1ccc(cc1)Br 10R-0601 COC(=O)/C=C\c1cccc2c1cccc2 10R-0602 COc1ccc(cc1)C(CC(=O)O)N2Cc3ccccc3C2=O 10R-0603 c1ccc2c(c1)cccc2C(CC(=O)O)N3Cc4ccccc4C3=O 10R-0604 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3cccc(c3)O 10R-0605 COC(=O)c1ccc(c(c1)NC(=O)c2cccs2)S(=O)(=O)c3ccccc3 10R-0607 COC(=O)c1ccc(c(c1)NC(=O)c2ccco2)S(=O)(=O)c3ccccc3 10R-0608 COc1ccc(cc1OC)/C=C/C(=O)OC 10R-0609 COc1ccc(cc1)C(CC(=O)O)N2CCS(=O)(=O)CC2 10R-0611 c1cc2c(cc1C(CC(=O)O)N3CCS(=O)(=O)CC3)OCO2 10R-0612 c1ccn(c1)c2ccc(cc2)Br 10R-0614 CCc1ccc(cc1)C(CC(=O)O)N 10R-0615 COc1ccc(cc1)C(CC(=O)O)NC(=O)C(F)(F)F 10R-0616 COC(=O)/C=C/c1cccc(c1)Br 10R-0617 CCc1ccc(cc1)/C=C/C(=O)O 10R-0618 c1cc(n(c1)c2ccc(cc2)Br)C=O 10R-0619 c1cc(ccc1C(CC(=O)O)N)C(F)(F)F 10R-0620 CC(C)(C)C(=O)NC(CC(=O)N1CCN(CC1)c2ccccc2)c3cccc4c3cccc4 10R-0623 CCOC(=O)C1CCN(CC1)Cc2cnc(s2)Oc3ccc(cc3)OC 10R-0624 Cc1cc(c(cc1Cl)NC(=O)C)[N+](=O)[O-] 10R-0625 Cc1cc(c(c(c1Cl)[N+](=O)[O-])NC(=O)C)[N+](=O)[O-] 10R-0626 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(cc3)C(F)(F)F 10R-0627 c1cc(n(c1)c2ccc(cc2)Br)C(=O)C(F)(F)F 10R-0628 c1cc(sc1)c2ccnc(n2)NC(=S)N 10R-0629 Cc1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)C=C(C#N)C#N 10R-0630 CCc1ccc(cc1)/C=C/C(=O)OC 10R-0631 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1)C(F)(F)F 10R-0632 c1ccc(cc1)COC(=O)NC(CC(=O)O)c2ccc(cc2)Br 10R-0633 CCc1ccc(cc1)C(CC(=O)O)N2Cc3ccccc3C2=O 10R-0634 c1ccc(cc1)COC(=O)NC(CC(=O)O)c2ccc3c(c2)OCO3 10R-0635 COC(=O)c1ccc(c(c1)NC(=O)c2ccco2)N3CCN(CC3)c4ccccc4 10R-0636 COC(=O)c1ccc(c(c1)NC(=O)C2CC2)N3CCN(CC3)c4ccccc4 10R-0637 COC(=O)c1ccc(cc1)C(C[N+](=O)[O-])O 10R-0638 CC(C)(C)OC(=O)N1CCC2(C1)CCNCC2 10R-0639 CC(C)(C)OC(=O)n1cc(c2c1cccc2)C=C(C#N)C#N 10R-0641 CC(C)(C)OC(=O)n1cc(c2c1cccc2)/C=N/NC(=O)c3ccco3 10R-0642 CCc1ccc(cc1)C(CC(=O)O)NC(=O)OC(C)(C)C 10R-0643 c1cc(n(c1)c2ccc(cc2)Br)C(=O)C(Cl)(Cl)Cl 10R-0644 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2N)C(=O)OC 10R-0645 CCOC(=O)C1CCN(CC1)Cc2cnc(s2)Oc3ccc(cc3)C(C)(C)C 10R-0646 COc1ccc(cc1)Oc2ncc(s2)CN3CCN(CC3)c4ccccc4 10R-0647 CC(C)(C)c1ccc(cc1)Oc2ncc(s2)CN3CCN(CC3)c4ccccc4 10R-0648 CC(C)(C)OC(=O)n1cc(c2c1cccc2)/C=C\3/c4ccccc4NC3=O 10R-0649 Cc1cc(ccc1Oc2ncc(s2)CN3CCN(CC3)c4ccccc4)Cl 10R-0650 Cc1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)/C=C\4/c5ccccc5NC4=O 10R-0651 c1cc(ccc1C(CC(=O)O)NC(=O)C(F)(F)F)Br 10R-0653 c1cc(ccc1n2ccc(c2)C=O)Br 10R-0654 c1ccc2c(c1)ccn2Cc3cnc(s3)Oc4ccc(cc4)Br 10R-0655 c1cc(ccc1N2CCN(CC2)Cc3cnc(s3)Oc4ccc(cc4)Br)F 10R-0656 c1cc(ccc1Oc2ncc(s2)CN3CCOCC3)Br 10R-0657 c1cc(n(c1)c2ccc(cc2)Br)C(=O)N3CCOCC3 10R-0659 CCOC(=O)C1CCN(CC1)Cc2cnc(s2)Oc3ccc(cc3C)Cl 10R-0660 CC(C)c1ccc(cc1)C(CC(=O)OC)n2cccc2 10R-0661 CCOC(=O)C1CCN(CC1)Cc2cnc(s2)Oc3ccc(cc3)N 10R-0663 c1ccc(cc1)N2CCN(CC2)c3ncc(s3)Cn4ccc5c4cccc5 10R-0664 c1cc(ccc1n2c(c(cn2)n3cncn3)O)OC(F)(F)F 10R-0800 CNc1nccc(n1)c2cnc(s2)c3ccncc3 10R-0802 c1cnccc1c2ncc(s2)c3ccncn3 10R-0803 Cc1c(sc(n1)c2cc[n+](cc2)C)c3ccncn3.[I-] 10R-0804 CCCCCCCc1ccc(cc1)/C=C\2/C(=C(N(C2=O)CCc3ccc(c(c3)OC)OC)C)C(=O)OC 10R-0806 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)CCCN3CCOCC3 10R-0808 CCc1cc(ccc1OCC#C)C=O 10R-0810 COc1cc(ccc1OCC#C)/C=N/O 10R-0811 COc1cc(ccc1OCC#C)CO 10R-0812 COc1cc(ccc1OCC#C)/C=C/C(=O)O 10R-0813 CN(C)CCn1c(=N)c2cc(c(cc2[nH]c1=S)OC)OC 10R-0815 c1cnccc1c2ncc(s2)c3ccn[nH]3 10R-0818 C/C(=N\NC(=O)N)/c1cnc(s1)c2cccs2 10R-0819 c1cc(ccc1c2ccnc(n2)NS(=O)(=O)c3ccc(cc3)N)F 10R-0824 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccc[n+](c3)C.[I-] 10R-0826 c1cc(sc1)c2ncc(s2)c3ccno3 10R-0827 C[C@@H](c1ccccc1)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 10R-0828 COC(=O)c1c(ccs1)n2cc(nn2)c3ccccc3 10R-0829 c1cc(sc1)C2CC(=O)CC(=O)C2n3cncn3 10R-0830 c1c(cnc(c1Cl)CC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 10R-0831 COC(=O)Cc1c(ccn(c1=O)C2CCCC2)O 10R-0833 COc1ccc(cc1)C(=O)NCCN2CCN(CC2)C(=O)c3ccc(cc3)OC 10R-0834 c1cc(cc(c1)Cl)N2CCN(CC2)C(=O)Cc3c(cc(cn3)C(F)(F)F)Cl 10R-0835 c1c(cnc(c1Cl)CC(=O)NC2CCCCCCC2)C(F)(F)F 10R-0836 c1ccc2c(c1)CCNC2C3C(=O)CC(C(C3=O)n4cncn4)c5ccc(cc5)Cl 10R-0837 Cc1c(c(c(c(c1C)C)C(=O)C2CCN(CC2)C(=O)C)C)C 10R-0839 Cc1c(c(c(c(c1C)C)C(=O)C2CCNCC2)C)C 10R-0841 C/C(=N/c1ccc(cc1)N(C)C)/c2cnc(s2)c3ccncc3 10R-0843 COc1ccc(cc1OCC#C)C=O 10R-0844 c1ccc2c(c1)c(c[nH]2)CCNc3cccc(c3C#N)F 10R-0846 c1cc(sc1)CNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 10R-0847 c1c(cc(c(c1[N+](=O)[O-])NCCN2CCNCC2)[N+](=O)[O-])C(F)(F)F 10R-0848 Cc1c(c(n2c(n1)cc(n2)c3ccc(c(c3)Cl)Cl)C)Cc4cccc(c4)F 10R-0849 Cc1c(sc2n1ccn2)C(C)OC(=O)Nc3ccc(cc3)Cl 10R-1000 Cc1ccc(n1c2ccccc2CNC(=O)c3ccc(cc3)F)C 10R-1001 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CCC(C(C(F)(F)F)(F)F)O 10R-1060 c1ccc(cc1)CN(CCO)/C=C/C(=O)C(C(F)(F)F)(F)F 10R-1061 C[C@H](c1ccccc1)NC(=O)C(F)(F)Cl 10R-1064 c1cnc(nc1)N2CCN(CC2)/C=C/C(=O)C(F)(F)F 10R-1066 c1ccc(cc1)c2c(c3ccccc3[nH]2)C(=O)C(F)(F)F 10R-1067 c1cnc(nc1)SC(C(=O)O)F 10R-1075 c1ccc2c(c1)CCC(C2=O)NC(=O)c3ccc(cc3)F 10R-1121 Cc1ccc(cc1)C(=O)O/N=C/2\CCCc3c2cccc3 10R-1125 c1ccc\2c(c1)CCC/C2=N\OC(=O)c3cccs3 10R-1126 Cc1cccc(c1)C(=O)O/N=C/2\CCCc3c2cccc3 10R-1127 c1ccc\2c(c1)CCC/C2=N\OC(=O)c3ccc(c(c3)Cl)Cl 10R-1130 c1ccc\2c(c1)CCC/C2=N\OC(=O)c3cccc(c3)C(F)(F)F 10R-1131 c1ccc\2c(c1)CCC/C2=N\OC(=O)c3cccc(c3)Cl 10R-1132 c1ccc\2c(c1)CCC/C2=N\OC(=O)C3CC3 10R-1136 c1ccc\2c(c1)CCC/C2=N\OCc3ccc(cc3)Cl 10R-1138 c1ccc(cc1)CC(=O)O/N=C/2\CCCc3c2cccc3 10R-1140 c1cc(cc(c1)Cl)n2c(=O)cc(cn2)O 10R-1141 Cc1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3)F)/CCS2 10R-1144 Cc1ccc2c(c1)/C(=N/OC(=O)c3cccs3)/CCS2 10R-1145 Cc1ccc(cc1)C(=O)O/N=C/2\CCSc3c2cc(cc3)C 10R-1146 Cc1ccc2c(c1)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/CCS2 10R-1147 Cc1ccc2c(c1)/C(=N/OC(=O)C3CC3)/CCS2 10R-1154 Cc1cccc(c1)C(=O)O/N=C/2\CCSc3c2cc(cc3)C 10R-1155 COc1ccc(cc1C(=O)OC)S(=O)(=O)N2CCOCC2 10R-1161 Cc1ccc2c(c1)/C(=N/OC(=O)c3cccc(c3)Cl)/CCS2 10R-1162 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Cl 10R-1164 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCCC2 10R-1165 c1cc(c(c(c1)Cl)N2CCCCC2)NC(=O)c3ccc(cc3)Cl 10R-1181 c1cc(c(c(c1)Cl)N2CCCCC2)NC(=O)c3ccc(c(c3)Cl)Cl 10R-1182 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2cccc(c2N3CCCCC3)Cl 10R-1184 Cc1cc(c(n1c2ccc(c(c2)Cl)N3CCOCC3)C)C(=O)C(=O)NC 10R-1194 Cc1cc(c(n1c2ccc(c(c2)Cl)N3CCOCC3)C)C(=O)C(=O)Nc4ccc(cc4)Cl 10R-1199 Cc1cc(c(n1c2ccc(c(c2)Cl)N3CCOCC3)C)C(=O)C(=O)Nc4ccc(cc4)[N+](=O)[O-] 10R-1200 Cc1cc(c(n1c2ccc(c(c2)Cl)N3CCOCC3)C)C(=O)C(=O)Nc4ccccc4 10R-1201 Cc1cc(c(n1c2ccc(c(c2)Cl)N3CCOCC3)C)C(=O)C(=O)Nc4ccc(cc4)Br 10R-1202 Cc1cc(c(n1c2ccc(c(c2)Cl)N3CCOCC3)C)C(=O)C(=O)Nc4ccc(cc4)F 10R-1203 Cc1cc(c(n1c2ccc(c(c2)Cl)N3CCOCC3)C)C(=O)C(=O)Nc4ccc(cc4Cl)Cl 10R-1204 c1cc(n(c1)c2ccc(cc2Cl)[N+](=O)[O-])C(=O)C(=O)Nc3ccc(cc3)Cl 10R-1207 c1cc(n(c1)c2ccc(cc2Cl)[N+](=O)[O-])C(=O)C(=O)Nc3ccc(cc3)Br 10R-1209 CCOC(=O)COc1cccc2c1cccc2 10R-1240 CCn1c(nnc1S(=O)(=O)Cc2ccc(c(c2)Cl)Cl)COc3cccc(c3)C(F)(F)F 10R-1241 c1ccc2c(c1)cccc2OCC(=O)NN 10R-1242 c1ccc(cc1)n2c(nnc2S)COc3cccc4c3cccc4 10R-1243 c1ccc(cc1)n2c(nnc2S)COc3cccc(c3)C(F)(F)F 10R-1244 CCn1c(nnc1S(=O)(=O)C)COc2cccc(c2)C(F)(F)F 10R-1245 CCn1c(nnc1S(=O)Cc2ccc(c(c2)Cl)Cl)COc3cccc(c3)C(F)(F)F 10R-1248 CCn1c(nnc1S(=O)Cc2ccc(cc2)C)COc3cccc(c3)C(F)(F)F 10R-1251 c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)COc4cccc(c4)C(F)(F)F 10R-1252 Cc1ccc(cc1)CSc2nnc(n2c3ccccc3)COc4cccc(c4)C(F)(F)F 10R-1253 c1ccc(cc1)n2c(nnc2SCc3ccc(c(c3)Cl)Cl)COc4cccc(c4)C(F)(F)F 10R-1254 CSc1nnc(n1c2ccccc2)COc3cccc(c3)C(F)(F)F 10R-1255 c1ccc(cc1)n2c(nnc2SCC(=O)N)COc3cccc(c3)C(F)(F)F 10R-1256 c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)COc4cccc5c4cccc5 10R-1257 c1ccc(cc1)n2c(nnc2S(=O)Cc3ccc(cc3)Cl)COc4cccc(c4)C(F)(F)F 10R-1259 c1ccc(cc1)n2c(nnc2S(=O)(=O)Cc3ccc(cc3)Cl)COc4cccc(c4)C(F)(F)F 10R-1260 Cc1ccc(cc1)CS(=O)c2nnc(n2c3ccccc3)COc4cccc(c4)C(F)(F)F 10R-1261 Cc1ccc(cc1)CS(=O)(=O)c2nnc(n2c3ccccc3)COc4cccc(c4)C(F)(F)F 10R-1262 c1ccc(cc1)n2c(nnc2S(=O)Cc3ccc(c(c3)Cl)Cl)COc4cccc(c4)C(F)(F)F 10R-1263 c1ccc(cc1)n2c(nnc2SCc3ccc(c(c3)Cl)Cl)COc4cccc5c4cccc5 10R-1264 c1ccc(cc1)n2c(nnc2SCC(=O)N)COc3cccc4c3cccc4 10R-1265 CSc1nnc(n1c2ccccc2)COc3cccc4c3cccc4 10R-1266 c1ccc(cc1)n2c(nnc2SCc3ccc(cc3Cl)Cl)COc4cccc(c4)C(F)(F)F 10R-1267 c1ccc(cc1)n2c(nnc2S(=O)Cc3ccc(cc3)Cl)COc4cccc5c4cccc5 10R-1269 c1ccc(c(c1)N2CCN(CC2)CC(COc3ccc(cc3)C#N)O)F 10R-1421 Cn1c2c(cn1)c(c(cn2)C(=O)O)Oc3ccc(cc3)OC 10T-0002 c1ccc(c(c1)C(=O)NN)N2CCS(=O)(=O)CC2 10T-0005 CN1CCN(CC1)C(=O)c2ccccc2N3CCS(=O)(=O)CC3 10T-0006 c1ccc(cc1)CNC(=O)c2ccccc2N3CCS(=O)(=O)CC3 10T-0007 COC(=O)C(Cc1cccc(c1)Cl)(c2ccc(cc2)[N+](=O)[O-])C(=O)OC 10T-0008 CCCC(c1ccc(cc1)[N+](=O)[O-])(C(=O)OC)C(=O)OC 10T-0009 COC(=O)C(Cc1cnc(s1)Cl)(c2ccc(cc2)[N+](=O)[O-])C(=O)OC 10T-0010 CCN1C(=O)/C(=C/c2cc(ccc2OC)OC)/SC1=O 10T-0011 c1cnccc1/C=C\2/C(=O)NC(=O)S2 10T-0012 CCN1C(=O)/C(=C/c2ccc(c(c2)[N+](=O)[O-])Cl)/SC1=O 10T-0013 c1ccc(c(c1)NNC(=S)N)F 10T-0014 c1cc(ccc1NNC(=S)N)F 10T-0015 c1ccc(c(c1)NNC(=S)N)Cl 10T-0016 c1cc(c(cc1NNC(=S)N)Cl)Cl 10T-0017 CN1C(=O)/C(=C\c2c[nH]c3c2cccc3)/SC1=O 10T-0018 c1cc(cc(c1)N)CC2C(=O)NC(=O)S2 10T-0021 CCOC(=O)c1ccc(cc1)Nc2cnc3ccccc3n2 10T-0022 CCOC(=O)c1cnc2c(c1OC(CCN)C(F)(F)F)cnn2C 10T-0023 C1CCC(CC1)C(=O)NNC(=O)CN2CCS(=O)(=O)CC2 10T-0027 c1cc(sc1)S(=O)(=O)NNC(=O)CN2CCS(=O)(=O)CC2 10T-0028 CC(C)C/C=C/1\C(=O)N(C(=O)S1)C 10T-0029 C1CC1C(=O)NNC(=O)CN2CCS(=O)(=O)CC2 10T-0031 CCCC(c1ccc(cc1)[N+](=O)[O-])C(=O)O 10T-0033 CCOC(=O)c1cnc2c(c1OC(CCNS(=O)(=O)C)C(F)(F)F)cnn2C 10T-0034 Cc1ccc2ccccc2c1NS(=O)(=O)C 10T-0036 Cc1ccc2ccccc2c1NC(=S)NC 10T-0037 Cc1ccc2ccccc2c1NC(=O)C3CC3 10T-0038 Cc1ccc2ccccc2c1NS(=O)(=O)c3cccs3 10T-0039 Cc1ccc2ccccc2c1NC(=O)c3ccco3 10T-0040 CCCCCC(=O)Nc1c(ccc2c1cccc2)C 10T-0041 c1csc(n1)C(=O)CBr 10T-0046 Cc1ccc2ccccc2c1NC(=O)Nc3ccc(cc3)Cl 10T-0047 c1cc(cc(c1)F)NNC(=S)N 10T-0049 c1cc(cc(c1)Cl)CC(c2ccc(cc2)[N+](=O)[O-])C(=O)O 10T-0052 c1ccc(c(c1)C(=O)N/N=C/c2cccs2)N3CCS(=O)(=O)CC3 10T-0053 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NNC(=O)CN2CCS(=O)(=O)CC2 10T-0054 COC(=O)C(Cc1cnc(s1)Cl)(c2ccc(cn2)[N+](=O)[O-])C(=O)OC 10T-0055 CC(=O)N1CCCC(C1)/C(=N/O)/c2ccc(cc2F)F 10T-0056 CS(=O)(=O)Nc1ccc(cc1)c2cn3cccnc3n2 10T-0060 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)CC4C(=O)NC(=O)S4 10T-0062 CN1C(=O)/C(=C\N2CCN(CC2)c3ccccc3)/SC1=O 10T-0064 c1c(cnc(c1Cl)N)C#N 10T-0065 Cc1c(cccc1[N+](=O)[O-])n2cccc2 10T-0066 c1csc2c1C(CNC2=O)NC(=O)C(F)(F)F 10T-0068 CN1C(=O)/C(=C\c2ccc(cc2)[N+](=O)[O-])/SC1=O 10T-0069 c1cc2c(cn[nH]2)c(c1)NC(=O)c3ccco3 10T-0070 c1cc2c(cn[nH]2)c(c1)NC(=O)c3ccc(cc3)F 10T-0071 CC(C)(C)C(=O)Nc1cccc2c1cn[nH]2 10T-0072 c1cc(cc(c1)Cl)CCC(=O)c2cccs2 10T-0075 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccccc3Cl)SCc4ccccc4F 10T-0201 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)N 10T-0202 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccccc3Cl)SC/C=C/c4ccccc4 10T-0204 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccccc3Cl)SCc4cccc(c4)C(F)(F)F 10T-0206 CC(=C(C#N)C#N)c1ccc(cc1)Cl 10T-0209 COc1cccc(c1)CSc2nc3cc(c(cc3c(=N)n2Cc4ccccc4Cl)OC)OC 10T-0210 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccccc3Cl)SCC#N 10T-0211 Cc1cc(c(c(c1)C)CSc2nc3cc(c(cc3c(=N)n2Cc4ccccc4Cl)OC)OC)C 10T-0212 COC(=O)/C(=C/c1cn(nc1c2ccc(cc2)c3ccccc3)c4ccccc4)/C#N 10T-0214 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)/C=N/O 10T-0215 CC(=C(C#N)C#N)c1ccc2c(c1)OCO2 10T-0216 CCOC(=O)C1C(CC(=CC1=O)c2ccc(cc2)OC)c3ccccc3 10T-0218 Cc1nc2c3cc(c(cc3[nH]c(=S)n2n1)OC)OC 10T-0219 Cc1c2c(n3c(n1)c(cn3)C#N)N(CC2)CCN4CCOCC4 10T-0221 CCCCCC1CCC(CC1)c2nnc(o2)S 10T-0222 Cc1c2c(n3c(n1)c(cn3)C#N)N(CC2)Cc4cccc(c4)Cl 10T-0223 C/C(=N\Nc1ccccc1)/c2ccccn2 10T-0224 Cc1c(c(n(n1)C)Cl)C(=O)NC(c2ccccc2)C(=O)NCc3ccc(cc3)OC 10T-0225 Cc1cccc(c1NC(=O)C(c2ccccc2)NC(=O)c3c(nn(c3Cl)C)C)C 10T-0227 Cn1cc(c(n1)C(F)(F)F)C(=O)NCCCC(=O)NCc2ccc(cc2)OC 10T-0228 CC(C)c1ccc(cc1)NC(=O)CCCNC(=O)c2cn(nc2C(F)(F)F)C 10T-0229 Cc1ccc(cc1)CNC(=O)CCCNC(=O)c2cn(nc2C(F)(F)F)C 10T-0230 c1cc2c(cc1C(F)(F)F)c(=O)c(c[nH]2)C(=O)O 10T-0231 Cc1c2c(n3c(n1)c(cn3)C#N)N(CC2)Cc4ccco4 10T-0234 Cc1c2c(n3c(n1)c(cn3)C#N)N(CC2)CC4CCCO4 10T-0235 Cc1c2c(n3c(n1)c(cn3)C#N)N(CC2)Cc4ccccc4OC 10T-0236 CCCCCCCCN1CCc2c1n3c(c(cn3)C#N)nc2C 10T-0237 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)c3ccc(cc3)C 10T-0239 CC(C)Sc1nc2cc(c(cc2c(=N)n1Cc3ccccc3Cl)OC)OC 10T-0241 CCCSc1nc2cc(c(cc2c(=N)n1Cc3ccccc3Cl)OC)OC 10T-0242 CCSc1nc2cc(c(cc2c(=N)n1Cc3ccccc3Cl)OC)OC 10T-0244 c1cc(ccc1c2ccn(c(=N)c2C#N)N)Cl 10T-0248 CCOC(=O)/C=C/c1cc(cn1C)C(=O)c2ccc(cc2Cl)Cl 10T-0250 Cc1cc(cc(c1Br)CO)CO 10T-0251 CCOC(=O)C1C(CC(=CC1=O)c2ccccc2OC)c3ccsc3 10T-0254 Cc1c2c(n3c(n1)c(cn3)C#N)N(CC2)C(C(C)C)C(=O)OC 10T-0256 c1ccc(cc1)c2cnn3c2NC(=O)CC3 10T-0257 CCCCCC1CCC(CC1)c2nnc(o2)SCc3ccc(cc3)Cl 10T-0259 Cc1cc2nc(c3c(n2n1)N(CC3)Cc4ccccc4Cl)C 10T-0261 CCOC(=O)c1cnc2c(cnn2c1O)c3ccc(c(c3)OC)OC 10T-0262 Cc1c[nH]nc1c2ccc(c(c2)F)OC 10T-0263 Cc1c2c(n3c(n1)c(cn3)C#N)N(CC2)CC(OC)OC 10T-0264 Cn1cc(cc1C=O)C(=O)c2ccccc2F 10T-0265 CCc1nc2c3cc(c(cc3[nH]c(=S)n2n1)OC)OC 10T-0267 Cc1nc2c(c(ccn2n1)c3ccc(cc3)Cl)C#N 10T-0268 COC(=O)c1ccc(c(c1)[N+](=O)[O-])NCc2ccccc2N3CCC(CC3)CO 10T-0270 CCCc1c(c2cccc3c2n(c1=O)CCC3)O 10T-0272 CCOC(=O)/C=C/c1cc(cn1C)C(=O)c2ccccc2 10T-0273 c1cc(c(c(c1)F)c2nc3c(c(ccn3n2)c4ccc(cc4)Cl)C#N)F 10T-0274 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccc(cc4)C(C)(C)C)OC)OC 10T-0277 c1ccc(c(c1)CNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])N3CCC(CC3)CO 10T-0278 c1ccc(c(c1)CNc2ccc(cn2)[N+](=O)[O-])N3CCC(CC3)CO 10T-0279 CCCCCC1CCC(CC1)c2nnc(o2)SCc3c(cc(cc3C)C)C 10T-0281 CCCCCC1CCC(CC1)c2nnc(o2)SCc3ccc(cc3)C 10T-0282 COc1cc2c(cc1OC)[nH]c(=S)n3c2ncn3 10T-0283 CCCCCC1CCC(CC1)c2nnc(o2)SCCN3C(=O)c4ccccc4C3=O 10T-0286 CCCCCC1CCC(CC1)c2nnc(o2)SCc3ccc(cc3)[N+](=O)[O-] 10T-0287 Cc1c(c(n(n1)C)Cl)C(=O)NCC(=O)Nc2ccc(cc2)C(C)C 10T-0288 Cc1ccc(cc1)CNC(=O)CNC(=O)c2c(nn(c2Cl)C)C 10T-0289 Cc1c(c(n(n1)C)Cl)C(=O)NCC(=O)NCc2ccc(cc2)OC 10T-0290 c1cc(ccc1c2ccn3c(c2C#N)nc(n3)C4CCCCC4)Cl 10T-0293 c1cc(oc1)c2nc3c(c(ccn3n2)c4ccc(cc4)Cl)C#N 10T-0294 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)c3ccc(cc3)Cl 10T-0295 CCOC(=O)C1C(CC(=CC1=O)c2ccc(cc2)Cl)c3ccc(cc3)Cl 10T-0298 Cn1cc(cc1/C=C/C(=O)O)C(=O)c2ccccc2 10T-0299 Cc1cccc(c1NC(=O)c2cc3c4ccccc4n(c3s2)C)C 10T-0300 c1cc(cc(c1)Cl)c2nc3c(c(ccn3n2)c4ccc(cc4)Cl)C#N 10T-0301 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)c3ccc4ccccc4c3 10T-0303 c1ccc(c(c1)CNc2ccc(cc2[N+](=O)[O-])C#N)N3CCC(CC3)CO 10T-0306 Cn1cc(cc1/C=C(\C#N)/c2cccc(c2)C(F)(F)F)C(=O)c3ccccc3F 10T-0308 CCCCCC1CCC(CC1)c2nnc3n2N=C(CS3)c4ccc5ccccc5c4 10T-0311 CCCCCC1CCC(CC1)c2nnc3n2N=C(CS3)c4ccc(cc4)Cl 10T-0312 CC(=O)c1cccc(c1)N2Cc3ccccc3C2 10T-0313 CC(C)(C)c1nc2c(c(ccn2n1)c3ccc(cc3)Cl)C#N 10T-0314 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)c3c(ccs3)Cl 10T-0320 Cc1c(c(=O)n2c3ccccc3nc2[nH]1)CCOC(=O)C4CCCCC4 10T-0321 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3ccccc3F 10T-0322 Cc1nc2c3cc(c(cc3nc(n2n1)SCc4c(cccc4Cl)F)OC)OC 10T-0323 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)c3cc(c(c(c3)C)O)C 10T-0324 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)CC(=O)Nc3ccccc3 10T-0326 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3ccccc3 10T-0329 Cc1ccccc1C(=O)OCCc2c([nH]c3ncnn3c2=O)C 10T-0330 c1ccc2c(c1)CN(C2)Cc3ccccc3N4CCC(CC4)CO 10T-0331 c1ccc(cc1)S(=O)(=O)c2csc(c2N)C(=O)O 10T-0335 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3cc(c(c(c3)OC)OC)OC 10T-0338 CN(C)/C=C/C(=C(C#N)C#N)c1ccc2c(c1)OCO2 10T-0340 Cc1nc2c3cc(c(cc3nc(n2n1)SCc4ccc(cc4)C(C)(C)C)OC)OC 10T-0341 CCCCCC1CCC(CC1)c2nnc3n2N=C(CS3)c4cc(c(c(c4)C)O)C 10T-0342 CCCCCC1CCC(CC1)c2ccc(cc2)N3Cc4ccccc4C3 10T-0344 Cn1cc(c2c1cccc2)C(=O)CCl 10T-0345 Cc1ccc(cc1)C(=O)Nc2cscc2S(=O)(=O)c3ccccc3 10T-0349 c1cc2c(cc1c3ccn(c(=N)c3C#N)N)OCO2 10T-0350 CCCCCc1nc2c(c(ccn2n1)c3ccc(cc3)Cl)C#N 10T-0351 Cc1ccccc1c2nc3c(c(ccn3n2)c4ccc(cc4)Cl)C#N 10T-0352 Cc1nc2c3cc(c(cc3nc(n2n1)SCc4ccc(cc4Cl)Cl)OC)OC 10T-0353 Cc1nc2c3cc(c(cc3nc(n2n1)SCc4ccccc4)OC)OC 10T-0354 Cn1c2ccccc2c3c1sc(c3)C(=O)NCc4ccco4 10T-0358 CCCNC(=O)c1cc2c3ccccc3n(c2s1)C 10T-0359 Cc1c(c(n(n1)c2ccc(cc2)F)N)c3cccc(c3)C(F)(F)F 10T-0360 Cn1c2ccccc2c3c1sc(c3)C(=O)NCCOC 10T-0363 Cc1c(noc1c2nc3c(c(ccn3n2)c4ccc(cc4)Cl)C#N)c5c(cccc5Cl)F 10T-0364 c1ccc(c(c1)c2nc3c(c(ccn3n2)c4ccc(cc4)Cl)C#N)F 10T-0365 Cc1cc(c(c(c1)C)CSc2nc3cc(c(cc3c4n2nc(n4)C)OC)OC)C 10T-0368 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)c3cccc(c3)[N+](=O)[O-] 10T-0369 CCCCCC1CCC(CC1)c2nnc(o2)SCC(=O)C 10T-0370 c1cn(nc1C2CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl 10T-0371 CC(=O)c1cc2c(cc1N3Cc4ccccc4C3)OCO2 10T-0372 Cn1c2ccccc2c3c1sc(c3)C(=O)Nc4cccc(c4)Cl 10T-0373 CCc1nc2c(c(ccn2n1)c3ccc(cc3)Cl)C#N 10T-0374 CC(C)c1ccc(cc1)NC(=O)c2cc3c4ccccc4n(c3s2)C 10T-0375 Cn1c2ccccc2c3c1sc(c3)C(=O)NCCCN(C)C 10T-0377 Cc1c(c(on1)N)c2cccc(c2)C(F)(F)F 10T-0381 Cc1c(c([nH]n1)N)c2cccc(c2)C(F)(F)F 10T-0382 Cc1c(c(n(n1)c2cccc(n2)Cl)N)c3cccc(c3)C(F)(F)F 10T-0383 Cn1c2ccccc2c3c1sc(c3)C(=O)N4CCOCC4 10T-0385 CCCCCC1CCC(CC1)c2nnc3n2N=C(CS3)c4cccc(c4)[N+](=O)[O-] 10T-0390 CC(=O)C1(C(C1(C#N)S(=O)(=O)c2ccccc2)c3ccc(cc3)Cl)C(=O)C 10T-0603 c1cc(cc(c1)Oc2ncccn2)C=O 10T-0605 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)S(=O)(=O)c3ccccc3)c4ccc(cc4)Cl 10T-0620 Cc1ccc(cc1)S(=O)(=O)C2=C(OC3=C(C2c4ccc(cc4)Cl)C(=O)CC(C3)(C)C)N 10T-0622 CSc1ccc(cc1)c2[nH]c3cnccc3n2.Cl 10T-0627 Cc1c(sc(n1)c2ccc(cc2)Cl)c3cc(c(c(n3)OC)C#N)c4ccc(cc4)Cl 10T-0628 c1ccnc(c1)/C=C/C(=O)c2cnc(s2)c3ccc(cc3)Cl 10T-0629 CCC(=O)C(C(=O)CC)C(=O)OC 10T-0632 c1cc(ccc1C(=O)NNC(=S)N)F 10T-0800 c1ccc(cc1)c2csc(n2)NNC(=O)c3ccc(cc3)F 10T-0801 c1cc(ccc1c2csc(n2)NNC(=O)c3ccc(cc3)F)Cl 10T-0802 Cc1c(nnn1c2ccsc2C(=O)OC)C(=O)OC(C)(C)C 10T-0804 CN(C)/C=C(/C(=O)c1c(cc(cn1)C(F)(F)F)Cl)\C(=O)C2CC2 10T-0805 c1ccc(cc1)c2c(nnc(n2)S)c3ccccc3 10T-0809 Cc1cc(n(n1)c2nc(cs2)C(=O)N3CCN(CC3)c4ccccc4)C(F)(F)F 10T-0811 Cc1cc(n(n1)c2nc(cs2)C(=O)Nc3ccc(cc3)F)C(F)(F)F 10T-0812 Cc1cc(n(n1)c2nc(cs2)C(=O)Nc3cccnc3)C(F)(F)F 10T-0813 Cc1cc(n(n1)c2nc(cs2)C(=O)NCc3ccccc3OC)C(F)(F)F 10T-0814 Cc1cc(n(n1)c2nc(cs2)C(=O)N3CCOCC3)C(F)(F)F 10T-0815 Cc1ccc(n1NC(=O)c2ccco2)C 10T-0818 Cc1cc(n(n1)c2nc(cs2)C(=O)Nc3ccccc3Oc4ccccc4)C(F)(F)F 10T-0821 c1csc(c1)/C=C/C(=O)/C=C/c2sccc2 10T-0823 c1cc(c(cc1F)C2CC(=O)C=C(C2n3cncn3)O)F 10T-0824 C/C(=N/OC(=O)Nc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)N3CCCC3 10T-0826 C/C(=N/OC(=O)c1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)N3CCCC3 10T-0846 c1ccc(cc1)Cn2cc(c3c2cccc3)C(=O)Nc4ccccc4 10T-1480 COc1ccc(cc1)NC(=O)c2cn(c3c2cccc3)Cc4ccccc4 10T-1481 c1ccc(cc1)CNC(=O)c2cn(c3c2cccc3)Cc4ccccc4 10T-1482 CNC(=O)c1cn(c2c1cccc2)Cc3ccccc3 10T-1484 c1ccc(cc1)Cn2cc(c3c2cccc3)C(=O)N4CCCCC4 10T-1485 c1ccc(cc1)CNC(=O)c2cn(c3c2cccc3)Cc4ccc(cc4)Cl 10T-1487 COc1ccc(cc1)NC(=O)c2cn(c3c2cccc3)Cc4ccc(cc4)Cl 10T-1488 c1ccc(cc1)NC(=O)c2cn(c3c2cccc3)Cc4ccc(cc4)Cl 10T-1490 Cc1ccc(nc1)NC(=O)C2CC2 10W-0019 Cn1c(c(c(n1)C(F)(F)F)CNS(=O)(=O)c2ccccc2Cl)Oc3ccccc3 10W-0021 Cn1c(c(c(n1)C(F)(F)F)CNC(=O)c2cccs2)Oc3ccccc3 10W-0022 Cn1c(c(c(n1)C(F)(F)F)CNC(=O)c2ccc(cc2)OC)Oc3ccccc3 10W-0023 Cn1c(c(c(n1)C(F)(F)F)CNC(=O)c2cccc(c2)C(F)(F)F)Oc3ccccc3 10W-0024 CC(C)(C)C(=O)NCc1c(nn(c1Oc2ccccc2)C)C(F)(F)F 10W-0040 Cn1c(c(c(n1)C(F)(F)F)CNS(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl)Oc3ccccc3 10W-0045 CCOC(=O)C(=CNc1cccnc1)C(=O)OCC 10W-0074 COC(=O)c1ccc2c(c1)NC(=O)C3N2CCC3 10W-0201 c1cc(cc(c1)C(F)(F)F)CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N5CCOCC5 10W-0202 CN(C)/C=C/C(=O)c1ccc(cc1O)OCCCCl 10W-0203 c1cc(cc(c1)C(F)(F)F)COc2ccc(c(c2)O)C=O 10W-0206 COC(=O)c1cc(c[nH]c1=O)Br 10W-0208 c1cc2c(cc1S(=O)(=O)N3CCOCC3)N(C(=O)C4N2CCC4)CC#N 10W-0213 c1ccc(c(c1)CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N5CCOCC5)F 10W-0217 c1cc2c(cc1C(=O)O)NC(=O)C3N2CCC3 10W-0218 COC(=O)c1cc2ccccc2n1Cc3ccc(cc3)Cl 10W-0220 CS(=O)(=O)Nc1ccc2c(c1)NCC2.Cl 10W-0222 c1cc2c(cc1[N+](=O)[O-])OC(C(=O)N2)CCN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 10W-0225 CN(C)/C=C(\CCN1CCOCC1)/C(=O)c2ccc(cc2)F 10W-0228 c1ccc(cc1)/C=C/CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N5CCOCC5 10W-0229 Cc1c(c(=O)n(c(n1)N)N)Cc2ccccc2 10W-0230 Cc1c(c(=O)n([nH]1)c2ccccc2)CCOC(=O)c3ccc(cc3)C(F)(F)F 10W-0233 Cc1c(c(=O)n(n1C(=O)c2cccc(c2)[N+](=O)[O-])C)CCOC(=O)c3cccc(c3)[N+](=O)[O-] 10W-0235 Cc1ccc(cc1)CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N5CCOCC5 10W-0237 c1cc(ccc1C(=O)CCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)F 10W-0238 COc1ccc-2c(c1)CCc3c2n[nH]c3 10W-0239 c1cc(ccc1c2c(c[nH]n2)CCN3CCOCC3)F 10W-0240 COC(=O)c1c(c2ccccc2[nH]1)I 10W-0241 Cc1c(c(=O)n([nH]1)c2ccccc2)CCOC(=O)c3cccc(c3)C(F)(F)F 10W-0242 Cc1c(c(=O)n([nH]1)c2ccccc2)CCOC(=O)c3cccs3 10W-0243 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NCc3cccc(c3)C(F)(F)F 10W-0244 COc1cccc(c1)CNC(=O)CC2C(=O)Nc3ccccc3S2 10W-0245 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NCc3ccc(c(c3)Cl)Cl 10W-0246 COC(=O)c1c(c2ccccc2[nH]1)C=C(C#N)C#N 10W-0249 CCOC(=O)CCc1c(nc([nH]c1=O)n2c(=O)c(c([nH]2)C)CCO)C 10W-0250 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cccc(c3)OC)C#N 10W-0251 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccccc3)C#N 10W-0252 CCOC(=O)C(=CNc1cc(nn1C(C)(C)C)C)C(=O)OCC 10W-0253 CSc1nc2nc(c(cn2n1)CCN3CCOCC3)c4ccc(cc4)F 10W-0255 c1cc(ccc1c2c(cn3c(n2)c(cn3)C#N)CCN4CCOCC4)F 10W-0256 COc1cccc(c1)CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N5CCOCC5 10W-0257 Cc1ccc(cc1)C2C(=C(NC3=C2C(=O)CC(C3)(C)C)C)C#N 10W-0259 CC1CN(CC(O1)C)CCC2C(=O)Nc3c(cccn3)O2 10W-0263 c1cc(c(cc1OCCCCl)O)c2cc[nH]n2 10W-0264 Cc1ccc(cc1)Cn2c3ccccc3cc2C(=O)OC 10W-0265 CCCCC1C(=C(NC2=C1C(=O)CC(C2)(C)C)C)C#N 10W-0267 CCOc1cc(ccc1O)C2C(=C(NC3=C2C(=O)CC(C3)(C)C)C)C#N 10W-0268 c1ccc(c(c1)N2CCN(CC2)CCC3C(=O)Nc4ccc(cc4O3)[N+](=O)[O-])F 10W-0270 CCN1CCN(CC1)CCC2C(=O)Nc3ccc(cc3O2)[N+](=O)[O-] 10W-0271 CN1C(=O)C(=Cc2c3ccccc3[nH]c2C(=O)OC)C(=O)N(C1=O)C 10W-0272 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccc(cc2)I)CCO 10W-0274 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccccc2[N+](=O)[O-])CCO 10W-0275 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cccc4c3cccc4)C#N 10W-0276 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3)F)C#N 10W-0277 CCN1CCN(CC1)CCC2C(=O)Nc3c(cccn3)O2 10W-0278 c1ccc(cc1)CN2CCN(CC2)CCC3C(=O)Nc4c(cccn4)O3 10W-0279 c1cc2c(nc1)NC(=O)C(O2)CCN3CCOCC3 10W-0280 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc4c(c3)OCO4)C#N 10W-0281 c1cc2c(nc1)NC(=O)C(O2)CCN3CCN(CC3)c4ccc(c(c4)Cl)Cl 10W-0282 Cc1ccc(cc1)S(=O)(=O)n2c(c(c(=O)[nH]2)CCO)C 10W-0283 c1ccc(cc1)CN2CCN(CC2)CCC3C(=O)Nc4ccc(cc4O3)[N+](=O)[O-] 10W-0285 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cccnc3)C#N 10W-0287 COc1ccc(cc1)CNC(=O)CC2C(=O)Nc3ccccc3S2 10W-0290 Cc1ccc(cc1)CNC(=O)CC2C(=O)Nc3ccccc3S2 10W-0291 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NCc3ccc(cc3)Cl 10W-0292 COc1ccccc1CNC(=O)CC2C(=O)Nc3ccccc3S2 10W-0293 Cc1c(c(=O)[nH]n1S(=O)(=O)c2cccs2)CCO 10W-0294 COC(=O)c1c(c2ccccc2n1S(=O)(=O)C)I 10W-0296 CC(=O)c1ccc(cc1O)OCc2cccc(c2)C(F)(F)F 10W-0298 Cc1c(c(=O)[nH]n1C(=O)c2ccc(cc2)[N+](=O)[O-])CCO 10W-0300 CCOC(=O)CC/C(=N\NC(=N)N)/C 10W-0302 CN(CC(=O)O)C1=N/C(=C/C=C/c2ccccc2)/C(=O)N1 10W-0303 CN1CCN(CC1)CCCC(=O)c2ccc(cc2)F 10W-0306 CN1CCN(CC1)S(=O)(=O)c2ccc3c(c2)NC(=O)C4N3CCC4 10W-0307 COC(=O)c1c(c2ccccc2[nH]1)C=C3C(=O)c4ccccc4C3=O 10W-0308 c1ccc(cc1)S(=O)(=O)N(n2c(=O)cc(nc2N)C(F)(F)F)S(=O)(=O)c3ccccc3 10W-0311 COC(=O)c1cc2ccccc2n1S(=O)(=O)C 10W-0313 COC(=O)c1c(c2ccccc2n1S(=O)(=O)C)C=O 10W-0315 CN1CC(=O)N2C1=N/C(=C/C=C/c3ccccc3)/C2=O 10W-0318 Cc1ccc(c(c1)CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N5CCOCC5)C 10W-0321 c1cc(c(nc1)N2CCCC2C(=O)O)[N+](=O)[O-] 10W-0322 COC(=O)c1c(c2ccccc2n1S(=O)(=O)c3ccccc3)I 10W-0324 COC(=O)c1c(c2ccccc2n1S(=O)(=O)c3ccc(cc3)Br)I 10W-0325 CN(C)/C=C/C(=O)c1ccc(cc1O)OCc2cccc(c2)C(F)(F)F 10W-0326 c1cc2c(cc1/C=C/3\C(=O)NC(=N3)N4CCOCC4)OCO2 10W-0328 CCOC(=O)C(=O)c1c[nH]c2c1cccn2 10W-0332 COC(=O)c1c(c2ccccc2[nH]1)/C=C/3\c4ccccc4NC3=O 10W-0335 c1cc2c(nc1)N3CCCC3C(=O)N2 10W-0336 CN(OC)S(=O)(=O)c1ccc(c(c1)[N+](=O)[O-])Cl 10W-0337 CN1CCN(CC1)CC/C(=C\N(C)C)/C(=O)c2ccc(cc2)F 10W-0338 COC(=O)c1cc2ccccc2n1S(=O)(=O)c3ccccc3 10W-0339 Cc1nn(c(=O)n1c2cccc(c2)Cl)CCN3C(=O)c4ccccc4C3=O 10W-0340 c1ccc(cc1)/C=C/C=N/Nc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N3CCC(CC3)C(=O)O 10W-0342 c1cc(cc(c1)[N+](=O)[O-])/C=N/Nc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N3CCC(CC3)C(=O)O 10W-0343 COc1ccc(c(c1)/C=N/Nc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N3CCC(CC3)C(=O)O)OC 10W-0344 c1cc2c(cc1/C=N/Nc3ccc(cc3[N+](=O)[O-])S(=O)(=O)N4CCC(CC4)C(=O)O)OCO2 10W-0345 c1ccc(c(c1)/C=N/Nc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N3CCC(CC3)C(=O)O)C(F)(F)F 10W-0348 CCOC(=O)c1ccc(nc1C)c2ccc3c(c2)CCC3 10W-0349 CN(OC)S(=O)(=O)c1ccc2c(c1)NC(=O)C3N2CCC3 10W-0350 c1cc(cc(c1)C(F)(F)F)COc2ccc(c(c2)O)c3cc[nH]n3 10W-0351 COC(=O)c1c(c2ccccc2[nH]1)/C=C/3\C(=O)NC(=O)S3 10W-0356 Cc1ccc2c(c1)NC(=O)C(O2)CCCl 10W-0359 c1cc(cc(c1)C(F)(F)F)CSC2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)N2 10W-0360 CN1CCN(CC1)CCc2cn3c(nc2c4ccc(cc4)F)nc(n3)SC 10W-0362 CN1CCN(CC1)CCc2c[nH]nc2c3ccc(cc3)F 10W-0363 CN1CCN(CC1)CCc2cn3c(ncn3)nc2c4ccc(cc4)F 10W-0365 CN1CCN(CC1)CCc2cn3c(c(cn3)C#N)nc2c4ccc(cc4)F 10W-0366 C/C(=N/O)/c1cccc(c1)N2Cc3ccccc3C2 10W-0370 COC(=O)c1c(c2ccccc2[nH]1)/C=C(\C#N)/S(=O)(=O)C 10W-0373 COC(=O)c1cc2ccccc2n1S(=O)(=O)c3ccc(cc3)Br 10W-0374 CCOC(=O)C(=O)c1cn(c2c1cccn2)S(=O)(=O)c3ccc(cc3)OC 10W-0375 CCCCCC1CCC(CC1)c2ccc(cc2)n3c(n[nH]c3=O)C 10W-0378 CC(C)(C)OC(=O)N1CC(C1)OS(=O)(=O)C 10W-0604 c1cc(cc(c1)Nc2ncnc(n2)c3cccnc3)C(F)(F)F 10W-0639 c1ccc(c(c1)CO)Oc2ccccc2C#N 10W-0703 COC(=O)c1cc(cc(c1)OCC=C)OCC=C 10W-0705 c1cc(ncc1C(=O)NN)N 10W-0706 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccccc2C#N 10W-0707 c1c(cnc(c1C(=O)O)Cl)Br 10W-0709 COC(=O)c1cc(cnc1Cl)Br 10W-0710 c1cc(cc(c1)OCCCOc2cccc(c2)C(F)(F)F)C(F)(F)F 10W-0712 c1ccc(cc1)C(=O)CC(=O)CCCO 10W-0715 CC(C)(C(=O)O)n1cccn1 10W-0717 c1ccc2c(c1)c(no2)CC(=O)O 10W-0718 c1cc(sc1)C(CCO)N 10W-0800 COc1ccc(cc1OC)C(CCO)NC(=S)N 10W-0801 c1ccc(c(c1)/C=C\2/c3ccccc3NC2=O)N 10W-0802 c1cc(ccc1n2cnn(c2=O)CC(=O)O)OC(F)(F)F 10W-0803 Cc1ccc(cc1)n2cnn(c2=O)CC(=O)O 10W-0804 c1ccc2c(c1)c3c([nH]2)-c4c(c[nH]n4)CC3 10W-0809 COc1cccc(c1)N/C=C/2\CCc3c4ccccc4[nH]c3C2=O 10W-0811 c1ccc2c(c1)c3c([nH]2)/C(=N/OC(=O)c4ccco4)/CCC3 10W-0812 c1ccc2c(c1)c3c([nH]2)/C(=N/OC(=O)C4CCCCC4)/CCC3 10W-0813 CCCCCC(=O)O/N=C/1\CCCc2c1[nH]c3c2cccc3 10W-0814 CN1C(=O)C(=Cc2c(ccc(c2[N+](=O)[O-])OC)OC)C(=O)N(C1=O)C 10W-0817 c1ccc2c(c1)cc3c(n2)-c4c(c5ccccc5n4Cc6cccc(c6)C(F)(F)F)CC3 10W-0819 c1ccc(cc1)NC(=O)O/N=C/2\CCCc3c2[nH]c4c3cccc4 10W-0821 c1ccc2c(c1)c3c([nH]2)/C(=N/OC(=O)Nc4cccc(c4)C(F)(F)F)/CCC3 10W-0822 CC(C)(C)NC(=O)O/N=C/1\CCCc2c1[nH]c3c2cccc3 10W-0823 CCOC(=O)c1csc(n1)Nc2ccc(c(c2)C(F)(F)F)Cl 10W-0824 CNC(=O)c1ccc2c(c1)OCO2 10W-0825 COc1ccc(c2c1cc[nH]2)OC 10W-0828 c1ccc2c(c1)c3c([nH]2)/C(=N/OCc4ccc(cc4)Cl)/CCC3 10W-0829 c1ccc(c(c1)CO/N=C/2\CCCc3c2[nH]c4c3cccc4)F 10W-0830 COc1ccc(cc1)CO/N=C/2\CCCc3c2[nH]c4c3cccc4 10W-0831 c1ccc2c(c1)c3c([nH]2)/C(=N/OCc4cccc(c4)C(F)(F)F)/CCC3 10W-0832 c1ccc2c(c1)c3c([nH]2)/C(=N/OC(=O)c4cccs4)/CCC3 10W-0833 c1ccc2c(c1)c3c([nH]2)/C(=N\CCO)/CCC3 10W-0835 c1ccc2c(c1)c3c(n2CCC#N)C(=O)CCC3 10W-0836 COc1ccc(c(c1C=O)N)OC 10W-0837 c1ccc(c(c1)C(CCO)N)F 10W-0838 Cc1c(nnn1c2ccc(cc2)C(F)(F)F)C(=O)c3c(cc(cn3)C(F)(F)F)Cl 10W-0840 Cc1c(nnn1c2ccc(c(c2)Cl)Cl)C(=O)c3c(cc(cn3)C(F)(F)F)Cl 10W-0841 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/Nc4ccc(cc4)F)/CC3 10W-0843 CC(C)c1ccc(cc1)N/C=C/2\CCc3c4ccccc4[nH]c3C2=O 10W-0844 c1ccc(cc1)Oc2cccc(c2)N/C=C/3\CCc4c5ccccc5[nH]c4C3=O 10W-0845 CN(C)Cc1cc(cc(c1O)OC)C=O 10W-0846 c1ccc2c(c1)ccc(n2)c3c(ccs3)Cl 10W-0847 c1cc(nc2c1cc(cc2Br)Br)c3c(ccs3)Cl 10W-0848 c1cnn(c1)c2cncc(n2)n3cccn3 10W-0849 Cc1n[nH]c(=O)n1c2ccc(cc2)C(C)(C)C 10W-0850 CN(C)Cc1cc(cc(c1O)OC)C=C(C#N)C#N 10W-0851 COc1ccc(cc1)c2ccc3c(ccc(c3n2)OC)OC 10W-0854 COc1ccc(cc1)c2ccc3cc(cc(c3n2)Br)Br 10W-0855 Cn1cc(c(=O)n(c1=O)C)c2c(=O)n(c(=O)n(c2Cl)C)C 10W-0856 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/Nc4ccc(cc4)OC(F)(F)F)/CC3 10W-0857 COc1ccc(cc1)C/N=C\2/CCCc3c2[nH]c4c3cccc4 10W-0859 c1cc(cc(c1)C(F)(F)F)C(CCO)N 10W-0861 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)C(F)(F)F 10W-0863 Cc1cc(nc(n1)n2cc(nn2)c3ccccc3)C(F)(F)F 10W-0864 c1cc(ccc1C(F)(F)F)NC(=S)N 10W-0866 Cc1n[nH]c(=O)n1c2ccc(cc2)Br 10W-0867 c1ccc2c(c1)c3c([nH]2)C(CCC3)NCCO 10W-0868 CCOC(=O)c1c(n2cccnc2n1)Cl 10W-0870 c1cscc1C(CCO)N 10W-0871 COC(=O)c1cccc(c1CBr)[N+](=O)[O-] 10W-0872 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)C(C)(C)C 10W-0873 Cc1n[nH]c(=O)n1c2ccc(cc2)OC(F)(F)F 10W-0874 Cc1nn(c(=O)n1c2ccc(cc2)C(C)(C)C)c3c(cc(cn3)C(F)(F)F)Cl 10W-0875 c1cnc2nc(cn2c1)C(=O)O 10W-0876 Cc1nn(c(=O)n1c2ccc(cc2)C(C)(C)C)CC#N 10W-0877 COc1ccc2c(c1)c(c[nH]2)CCn3ccc(c(c3=O)CC(=O)OC)O 10W-0880 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SCCCCOc4ccccc4)C(F)(F)F 10W-0881 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SCc4ccc(cc4)F)C(F)(F)F 10W-0882 c1ccc2c(c1)cc3c(n2)-c4c(c5ccccc5n4Cc6ccc(cc6)Cl)CC3 10W-0883 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)Br 10W-0884 Cc1nn(c(=O)n1c2ccc(cc2)Br)c3c(cc(cn3)C(F)(F)F)Cl 10W-0885 COc1cccc(c1O)CC2C(=O)NC(=O)S2 10W-0886 Cc1cc(cc(c1O)OC)C=O 10W-0887 CCc1ccc(cc1)Cn2c3ccccc3c4c2-c5c(cc6ccccc6n5)CC4 10W-0890 Cc1ccc(c(c1)Cn2c3ccccc3c4c2-c5c(cc6ccccc6n5)CC4)C 10W-0891 c1ccc2c(c1)cc3c(n2)-c4c(c5ccccc5n4Cc6ccccc6F)CC3 10W-0892 COc1ccc(cc1)c2csc(n2)Nc3ccc(cc3)C(F)(F)F 10W-0893 Cc1nn(c(=O)n1c2ccc(cc2)C(C)(C)C)CC(=O)O 10W-0894 Cc1cc(cc(c1O)OC)C=C2C(=O)N(C(=O)N(C2=O)C)C 10W-0895 c1cc(ccc1c2cnco2)[N+](=O)[O-] 10W-0897 COc1ccc(cc1)C(CCO)N2Cc3ccccc3C2 10W-0898 COc1cc(ccc1OCc2ccc(nc2)Cl)C=O 10W-0899 COC(=O)c1cccc(c1CN2CCC(CC2)Cc3ccccc3)[N+](=O)[O-] 10W-0900 c1ccc2c(c1)cc3c(n2)-c4c(c5ccccc5n4Cc6ccc(cc6)[N+](=O)[O-])CC3 10W-0903 CC1(c2cc(ccc2N(C13C=Cc4cc(ccc4O3)OC)C)Cl)C 10W-0904 COc1cccc(c1O)CC2C(=O)N(C(=O)S2)CC=C 10W-0905 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)c4cc([nH]n4)c5ccco5 10X-0019 c1cc(c(nc1)N2CCC(CC2)c3cc([nH]n3)c4ccco4)[N+](=O)[O-] 10X-0026 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)c3cc([nH]n3)c4ccco4 10X-0028 COc1ccc(c(c1)C2C3=C(C4CCN3CC4)NC(=S)N2)OC 10X-0040 c1cc(sc1)C2C3=C(C4CCN3CC4)NC(=S)N2 10X-0047 COc1ccc(c(c1)C2C3=C(C4CCN3CC4)N=C5N2C(=O)CS5)OC 10X-0058 c1cc(sc1)C2C3=C(C4CCN3CC4)N=C5N2C(=O)CS5 10X-0063 CC1=C(C(C2=C(N1)C3CCN2CC3)c4cc(ccc4OC)OC)C#N 10X-0111 CC1=C(C(C2=C(N1)C3CCN2CC3)c4ccc(cc4)Cl)C#N 10X-0112 CC1=C(C(C2=C(N1)C3CCN2CC3)c4cccs4)C#N 10X-0113 Cc1c(c(c2c(n1)C3CCN2CC3)c4ccco4)C#N 10X-0126 CC(=O)c1cc(cs1)Br 10X-0139 Cc1cc(c(s1)C)C(=O)/C=C/Nc2ccc(cc2)Br 10X-0200 Cc1cc(c(s1)C)c2ccnc3n2ncc3C#N 10X-0201 Cc1c(c(c2cc(ccc2n1)Oc3ccccc3)Nc4cccc(c4)SC)CCCl 10X-0203 COC(=O)C1CC(CN1C2=NC(=O)/C(=C\c3ccc(cc3)SC)/S2)O 10X-0204 CSc1ccc(cc1)/C=C/2\C(=O)N=C(S2)NC(CO)CO 10X-0205 CC(=O)OCCC1C(=O)Nc2cc(ccc2O1)CC(=O)OC 10X-0207 Cc1cc(c(s1)C)c2ccnc3n2ncn3 10X-0208 Cc1c(n(c(c1S(=O)(=O)c2ccccc2)N)C3CCCCC3)C 10X-0210 CCS(=O)(=O)c1ccc2c(c1)NC(=O)C(O2)CCO 10X-0211 Cc1c(n(c(c1S(=O)(=O)c2ccccc2)n3cccc3)C4CCCCC4)C 10X-0219 c1cc(ccc1CN2CCCCC2)OCCCF 10X-0220 COC(=O)Cc1ccc2c(c1)NC(=O)C(O2)CCOC(=O)C3CCCCC3 10X-0222 Cc1ccc(n1c2c(c(c(n2C3CCCCC3)C)C)S(=O)(=O)c4ccccc4)C 10X-0223 c1cc2c(cc1C3c4c(c(=O)cc(o4)CO)OC(=C3C#N)N)OCO2 10X-0224 CSc1ccc(cc1)/C=C\2/C(=O)N=C(S2)NO 10X-0226 CC(C)(C)c1ccc(cc1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N 10X-0230 CCS(=O)(=O)c1ccc2c(c1)NC(=O)C(O2)CCCl 10X-0232 Cc1c(n(c(c1S(=O)(=O)c2ccccc2)n3cccc3)CCCn4ccnc4)C 10X-0235 c1ccc2c(c1)cccc2C3c4c(c(=O)cc(o4)CO)OC(=C3C#N)N 10X-0237 CCCCCCCCN1CCc2c1n3c(cc(n3)C)nc2C 10X-0241 c1c(oc2c(c1=O)OC(=C(C2C3CCCCC3)C#N)N)CO 10X-0249 c1ccc(cc1)COc2ccc(cc2)C3c4c(c(=O)cc(o4)CO)OC(=C3C#N)N 10X-0250 CCOc1ccccc1C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N 10X-0251 Cc1c(n(c(c1S(=O)(=O)c2ccccc2)N)CCOC)C 10X-0268 c1ccc(cc1)COc2ccc(cc2)/C=C/c3c4c(c5cccc(c5n3)Oc6ccccc6)SCC4 10X-0276 c1ccc(cc1)Oc2cccc3c2nc(c4c3SCC4)/C=C/c5cccc6c5cccc6 10X-0277 c1cnccc1C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N 10X-0278 c1cc(cc(c1)C(F)(F)F)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N 10X-0279 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)CNC(=O)c3cc(c([nH]3)Br)Br 10X-0283 Cc1c(n(c(c1S(=O)(=O)c2ccccc2)n3cccc3)CCOC)C 10X-0285 CNc1c(ccs1)C#N 10X-0292 C#CCOc1ccc2ccccc2c1CN3CCN(CC3)c4ccccc4 10X-0293 Cc1ccc(n1c2c(c(c(n2CCOC)C)C)S(=O)(=O)c3ccccc3)C 10X-0294 COC(CNC(=O)c1cc(c([nH]1)Br)Br)OC 10X-0295 C#CCOc1ccc2ccccc2c1CN3CCOCC3 10X-0300 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3cc(c([nH]3)Br)Br 10X-0304 C#CCOc1ccc2ccccc2c1CN3CCc4ccccc4C3 10X-0306 c1cc2c(cc1CNC(=O)c3cc(c([nH]3)Br)Br)OCO2 10X-0311 CC1CCCCN1CCCNC(=O)c2cc(c([nH]2)Br)Br 10X-0312 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0319 c1cc(cc(c1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)[N+](=O)[O-] 10X-0320 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0321 c1cc(ccc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)Cl 10X-0322 c1cc(sc1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0323 Cc1cccc(c1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0324 c1ccc(c(c1)F)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0325 Cc1ccc(cc1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0326 COc1ccc(cc1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0327 c1cc(cc(c1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)C(F)(F)F 10X-0331 CCS(=O)(=O)Oc1c(c(c(c(c1F)F)F)F)F 10X-0332 c1ccc2cc(ccc2c1)S(=O)(=O)Oc3c(c(c(c(c3F)F)F)F)F 10X-0340 CC(C)(C)c1ccc(cc1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0341 c1cc(ccc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)I 10X-0342 c1cc(c(cc1Cl)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)Cl 10X-0343 c1cc(ccc1c2nc(on2)CCl)Cl 10X-0347 c1cc(ccc1CSC2=N/C(=C\c3ccc(cc3)n4cncn4)/C(=O)N2)F 10X-0348 CCc1ccc(cc1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0349 c1ccc(cc1)CS(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 10X-0350 c1cc(cc(c1)C(F)(F)F)c2nc(on2)CCl 10X-0355 c1cc(c(c(c1)Cl)CSC2=N/C(=C/c3ccc(cc3)n4cncn4)/C(=O)N2)F 10X-0357 c1cc(ccc1/C=C/2\C(=O)NC(=N2)SCCCF)n3cncn3 10X-0358 c1cc(ccc1/C=C/2\C(=O)N3CCSC3=N2)n4cncn4 10X-0361 Cc1c2cc(c(c(c2oc(=O)c1Br)Br)O)O 10X-0362 CN1CCCN(CC1)Cc2nc(no2)c3ccc(cc3)Cl 10X-0363 c1c(c(nnc1Cl)Cl)Cl 10X-0364 CC(C)(C)OC(=O)N1CCCn2c(cc(n2)CO)C1 10X-0603 c1c(c([nH]c1C(=O)C(Cl)(Cl)Cl)Br)Br 10X-0700 c1c(c([nH]c1C(=O)O)Br)Br 10X-0701 COC(=O)c1cc(c([nH]1)Br)Br 10X-0702 c1c(c([nH]c1C(=O)NN)Br)Br 10X-0703 COc1ccc(cc1)c2ccc(s2)C=O 10X-0704 COC(=O)c1ccc(cc1)c2ccc(s2)C=O 10X-0705 c1c(c([nH]c1C(=O)NCCCO)Br)Br 10X-0706 c1cc(cc(c1)Cl)C(=O)CBr 10X-0707 c1cscc1C(=O)CBr 10X-0708 Cc1cc(cc(c1O)OC)/C=N/NC(=O)c2ccncc2 10X-0800 Cc1cc(cc(c1O)OC)/C=C\2/c3ccccc3NC2=O 10X-0801 c1cc2nc(c(n2cc1I)C(=O)O)C(F)(F)F 10X-0802 c1cnc(cn1)NN 10X-0803 COc1ccc2cc(c(=O)oc2c1)C(=O)O 10X-0804 CCOC(=O)c1c(nn(c1C)c2ccc(nn2)O)C 10X-0805 c1cc(ncc1c2cnco2)Cl 10X-0806 Cc1ccc2c(c1N)NCCC2 10X-0807 c1cc(cc(c1)C(F)(F)F)c2ccc(cn2)C(=O)c3cccc(c3)C(F)(F)F 10X-0813 c1c(nc[nH]1)CCNC(=O)Cn2cncn2 10X-0814 CCOC(=O)c1c(nn(c1C)c2cc(ccc2Cl)Cl)C 10X-0815 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)C)C 10X-0816 c1cc(cc(c1)N)c2cnco2 10X-0817 Cc1ccc(cc1)S(=O)(=O)c2cc(nc(n2)N)C 10X-0818 Cc1cc(nc(n1)N)Nc2ccc(cc2)Cl 10X-0819 CC(C)(C)c1ccc(cc1)Oc2cccc(c2)C3CC(=O)C(C(=O)C3n4cncn4)C5c6ccccc6CCN5 10X-0820 Cc1c2c(nc(n1)n3cc(nn3)C(=O)c4cccc(c4)C(F)(F)F)CCC2 10X-0821 c1ccc2c(c1)CCNC2C3C(=O)CC(C(C3=O)n4cncn4)c5cccc(c5)Cl 10X-0822 CCOC(=O)c1c(nn(c1C)c2ccc(cc2Cl)Cl)C 10X-0824 c1cc(cc(c1)OCc2cnc(s2)Cl)C#N 10X-0825 CCOC(=O)c1ccccc1c2cn3cc(cc(c3n2)Cl)C(F)(F)F 10X-0830 c1cc(c(cc1Cn2c3ccc(cc3c(c2C(=O)O)I)I)Cl)Cl 10X-0833 Cc1c(c(n(n1)c2cc(ccc2Cl)Cl)C)C(=O)O 10X-0834 Cc1ccc(cc1)n2c(c(c(n2)C)C(=O)O)C 10X-0835 CCOC(=O)c1c([nH]nc1C)C 10X-0839 CN(c1cnccn1)N 10X-0840 COC(=O)C1CCN(CC1)c2cnccn2 10X-0841 Cc1c(c(on1)/C=C/c2c[nH]c3c2cc(cc3)OC)[N+](=O)[O-] 10X-0842 CC1=C(/C(=C/c2c[nH]c3c2cc(cc3)OC)/C(=O)N1CCc4ccc(c(c4)OC)OC)C(=O)OC 10X-0844 Cc1cc(nc(n1)N)Nc2ccc(cc2)F 10X-0845 Cc1cc(nc(n1)N)Nc2cccc(c2)C(F)(F)F 10X-0846 Cc1c(c(nc(n1)N)Nc2ccc(cc2)Cl)Br 10X-0847 CN(C)/C=C/C(=O)c1cc(cc(c1)F)C(F)(F)F 10X-0850 c1cc(cc(c1)OCc2cnc(s2)Cl)/C(=N\O)/N 10X-0852 c1cc2c(cc1C=O)CCO2 10X-0855 Cc1c(c(n[nH]1)C)C(=O)O 10X-0856 Cc1ccc(c2c1c3ccccc3n2Cc4cccc(c4)C(F)(F)F)C 10X-0857 CN(C)/C=C/C(=O)c1ccc(cc1F)C(F)(F)F 10X-0858 Cc1c(c(n(n1)c2ccc(cc2Cl)Cl)C)C(=O)O 10X-0860 c1ccc(c(c1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)C(=O)O 10X-0861 c1cc(ccc1c2cnco2)/C(=N\O)/N 10X-0862 c1cc(ccc1OCc2cnc(s2)Cl)S(=O)(=O)NC3CC3 10X-0863 CC1CCN(CC1)S(=O)(=O)c2ccc(cc2)OCc3cnc(s3)Cl 10X-0864 c1cc(ccc1OCc2cnc(s2)Cl)S(=O)(=O)NN3CCOCC3 10X-0865 c1c(c(c(nc1O)O)C#N)C(F)(F)F 10X-0866 Cc1cc(ccc1N)C(=O)O 10X-0868 CCCCCCC(c1ccno1)C(=O)OC 10X-0869 c1ccc(c(c1)C#N)N2CCCCC2 10X-0870 c1cc(ccc1N(S(=O)(=O)c2ccc(cc2)OCc3cnc(s3)Cl)S(=O)(=O)c4ccc(cc4)OCc5cnc(s5)Cl)OC(F)(F)F 10X-0871 c1csc(c1Br)C=O 10X-0872 c1cc(ccc1c2ccc(cn2)C(=O)c3ccc(cc3F)C(F)(F)F)C(F)(F)F 10X-0874 CCOC(=O)/C(=C\N(C)C)/C(=O)c1ccc(nc1)Cl 10X-0875 COC(=O)c1ccc(c(c1)N)N 10X-0878 c1ccc2c(c1)/C(=C/c3c(ccs3)Br)/C(=O)N2 10X-0879 c1ccn2c(c1)ncc2Br 10X-0880 c1ccc2c(c1)CCNC2c3c(c4ccccc4oc3=O)O 10X-0884 CCC(CC)c1c(nc(s1)N)C(=O)OC 10X-0900 Cc1cc(c(c(c1)OS(=O)(=O)c2ccc(cc2)OC)CN3CCOCC3)C 10X-0902 CCn1c2ccccc2c(c(c1=O)C(=O)C)O 10X-0920 CCn1c2ccccc2c3c(c1=O)c(c(c(=O)o3)Cc4ccc(cc4)[N+](=O)[O-])O 10X-0925 c1cc(ccc1C=O)OCCCN2CCCCC2 10X-0928 CSC1=N/C(=C/c2ccc(cc2)n3cncn3)/C(=O)N1 10X-0929 CCOC(=O)CSc1ccccc1 10X-0932 c1cc(ccc1CN2CCCCC2)OCCCN3CCCCC3 10X-0933 c1cc(ccc1CN2CCN(CC2)c3ccc(cc3)O)OCCCN4CCCCC4 10X-0934 CC(=O)c1c(c2ccccc2n(c1=O)C)O 10X-0936 CC(=O)c1c(c2ccccc2n(c1=O)Cc3ccccc3)O 10X-0937 CC(=O)c1c(c2cccc3c2n(c1=O)CC3)O 10X-0938 CCOC(=O)CS(=O)(=O)c1ccccc1 10X-0939 CN1CCN(CC1)c2ccc(cc2)/C=C/3\C(=O)NC(=S)N3 10X-0940 COC(=O)C1CCN(CC1)CCCOc2ccc(cc2)C=O 10X-0941 c1cc(ccc1C=O)OCCCN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 10X-0942 CCOC(=O)C1(CCN(CC1)Cc2ccc(cc2)Cl)S(=O)(=O)c3ccccc3 10X-0943 c1c(sc(n1)N2CCOCC2)/C=C/3\C(=O)NC(=S)N3 10X-0944 Cc1cc(c(cc1OS(=O)(=O)c2ccc(cc2)OC)C)CN3CCOCC3.Cl 10X-0948 Cc1cc(c(cc1OS(=O)(=O)c2ccc(cc2)Cl)C)CN3CCOCC3.Cl 10X-0949 CCOC(=O)C1(CCN(CC1)Cc2ccc(cc2)C)S(=O)(=O)c3ccccc3 10X-0950 CCOC(=O)C1(CCN(CC1)Cc2ccccc2)S(=O)(=O)c3ccccc3 10X-0951 CC(C)n1c2ccccc2c(c(c1=O)C(=O)C)O 10X-0952 CCCCn1c2ccccc2c(c(c1=O)C(=O)C)O 10X-0953 CC(=O)c1c(c2ccccc2n(c1=O)C3CCCCC3)O 10X-0954 CC(C)c1cc(cc(c1O)C(C)C)CN2CCC(CC2)C(=O)O 10X-0956 CC(C)c1cc(cc(c1O)C(C)C)CN2CCN(CC2)c3ccc(cc3)OC 10X-0958 Cn1c(c(cn1)C#N)/N=C/N(C)C 10X-0960 Cn1c2ccccc2c3c(c1=O)c(c(c(=O)o3)[N+](=O)[O-])O 10X-0963 COC(=O)C1CCN(CC1)Cc2ccc(cc2)OCCCN3CCN(CC3)c4ccc(cc4)[N+](=O)[O-] 10X-0966 CCOC(=O)CSc1ccccc1C(=O)O 10X-0968 CC(=O)c1c(c2cccc3c2n(c1=O)CCC3)O 10X-0969 CN1CCN(CC1)c2ccc(cc2)/C=C\3/C(=O)NC(=N3)SCc4ccc(c(c4)Cl)Cl 10X-0970 Cc1cc(c(cc1OS(=O)(=O)c2ccccc2[N+](=O)[O-])C)CN3CCOCC3 10X-0972 Cc1cc(c(c(c1)OS(=O)(=O)c2ccc(cc2)I)CN3CCOCC3)C 10X-0973 Cc1cc(c(cc1OS(=O)(=O)c2ccc(cc2)I)C)CN3CCOCC3.Cl 10X-0974 Cc1cc(c(cc1OS(=O)(=O)c2ccc(cc2)F)C)CN3CCOCC3.Cl 10X-0975 Cn1c(c(cn1)C#N)N/C=N/O 10X-0976 c1cc(ccc1/C=C/2\C(=O)NC(=N2)N3CCOCC3)n4cncn4 10X-0977 Cc1cc(c(c(c1)O)CN2CCC(CC2)C(=O)O)C 10X-0981 c1ccc(cc1)n2c3ccccc3c4c(c2=O)c(cc(=O)o4)O 10X-0984 COC(=O)C1CCN(CC1)CCCOc2ccc(cc2)CN3CCN(CC3)c4ccc(cc4)[N+](=O)[O-] 10X-0986 c1ccc(cc1)Oc2ccc(cn2)C=O 10X-0989 Cc1cc(c(c(c1)OS(=O)(=O)c2ccccc2[N+](=O)[O-])CN3CCOCC3)C 10X-0990 Cn1c2c(cn1)c(ncn2)NO 10X-0991 COC(=O)c1ccccc1C=O 10X-0992 Cc1cc(c(cc1OC(=O)c2ccc(cc2)Cl)C)CN3CCOCC3.Cl 10X-0995 COC(=O)c1c(sc(n1)N)c2ccc(cc2)F 10X-0996 COC(=O)c1c(sc(n1)N)c2ccc(cc2)Cl 10X-0997 c1cc(ccc1CN2CCC(CC2)C(=O)O)OCCCN3CCN(CC3)c4ccc(cc4)[N+](=O)[O-] 10X-0999 Cc1ccc(cc1)CNC(=O)c2cnc(nc2C(F)(F)F)c3ccccc3 10X-5006 CC1(C(=O)Nc2ccccc2O1)C(=O)N3CCOCC3 10X-5007 c1ccc(c(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)C(F)(F)F 10X-5024 CCOC(=O)C(=O)c1c[nH]c2c1cc(cc2)Br 10X-5043 CCOC(=O)C(=O)c1c[nH]c2c1cc(cc2)OC 10X-5059 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N 10Y-0603 COC(=O)c1cc(c(c(c1)Br)N)[N+](=O)[O-] 10Y-0604 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2ccc(cc2)N 10Y-0700 c1cc2c(cc1Br)[nH]nc2N 10Y-0701 c1cc2c(cc1C(F)(F)F)c(n[nH]2)N 10Y-0702 c1cc2c(c(c1)Cl)c(n[nH]2)N 10Y-0704 COc1ccc(cc1)OC2=C(C(OC2=O)O)Cl 10Y-0706 c1cc2c(cc1Br)c(n[nH]2)N 10Y-0709 COC(=O)c1c(c2c(s1)cccc2Cl)N 10Y-0710 COc1ccc(cc1)c2ccc(c(c2)F)C#N 10Y-0711 c1cc(ccc1c2ccc(c(c2)F)C#N)Cl 10Y-0713 c1cc(ccc1C=O)c2ccc(cn2)C(F)(F)F 10Y-0717 c1cc(ccc1C(CN)O)Cl 10Y-0719 COc1ccc(cc1)c2ccc(c(c2)C#N)F 10Y-0721 c1ccc(cc1)c2ccc(c(c2)F)C#N 10Y-0723 c1cc(sc1)c2nc(cs2)C(=O)NN 10Y-0724 c1ccc(cc1)c2ccc3c(c2)[nH]nc3N 10Y-0725 c1cc(ccc1C2CNC(=O)CO2)Cl 10Y-0726 c1cc(ccc1C(=O)CO)F 10Y-0727 C#CCN1C(=O)c2ccccc2C1=O 10Y-0730 CCOc1c(cnc(n1)c2ccccc2)C(=O)O 10Y-0731 c1ccc(cc1)c2ncc(c(n2)O)C(=O)O 10Y-0732 CN(C)/C=C/C(=O)c1cc(c(s1)Br)Br 10Y-0801 c1ccc(c(c1)C(=O)N)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Cl 10Y-0804 c1c[nH]nc1c2ccncc2 10Y-0805 CC(C)(CCl)C(=O)Nc1ccccc1 10Y-0806 CC(C)(C)c1ccc(cc1)NC2CCN(CC2)C(=O)OC(C)(C)C 10Y-0808 CCC1CCCCN1c2ccc(cc2[N+](=O)[O-])c3c4ccccc4c(=O)[nH]n3 10Y-0814 Cc1ccc(cc1)/C(=C/N(C)C)/C=O 10Y-0816 Cc1ccc(cc1)c2cnc3cc(nn3c2)c4ccc(cc4)Cl 10Y-0819 CNC(=O)c1cc(c[nH]1)Br 10Y-0822 CNNC(=O)c1cc(c[nH]1)Br 10Y-0823 c1c(c[nH]c1C(=O)N2CCCCC2)Br 10Y-0824 CC(C)CNC(=O)c1cc(c[nH]1)Br 10Y-0825 Cc1ccc(n1c2ccccc2C(=O)OC)C 10Y-0826 c1cnccc1CNC(=O)c2cc(c[nH]2)Br 10Y-0829 c1c(c[nH]c1C(=O)NCCN2CCCC2)Br 10Y-0830 CCCCc1nc2cc(ccc2o1)C(=O)O 10Y-0833 c1c(c[nH]c1C(=O)N2CCSCC2)Br 10Y-0834 CC1CCN(CC1)C(=O)c2cc(c[nH]2)Br 10Y-0837 CCN(CC)C(=O)c1cc(c[nH]1)Br 10Y-0842 c1cc(ccc1C2c3ccsc3CCN2)[N+](=O)[O-] 10Y-0844 CC(C)CCOc1ccc(cc1)C(=O)OC 10Y-0923 COc1ccc(cc1)OC2CCNCC2.Cl 10Y-7005 c1c(cnc(c1Cl)CN)C(F)(F)F.Cl 10Z-0006 COc1ccc(cc1)C(=O)c2c(cc(cn2)C(F)(F)F)c3cccc(c3)C(F)(F)F 10Z-0014 c1cc(c(c(c1)Cl)C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl)Cl 10Z-0024 c1cc(c(c(c1)Cl)C(=O)NCCS(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl 10Z-0027 c1cc(c(c(c1)Cl)c2nnnn2CCSc3c(cc(cn3)C(F)(F)F)Cl)Cl 10Z-0028 COc1ccc(cc1)C(=O)c2c(cc(cn2)C(F)(F)F)c3ccccc3OC 10Z-0030 CN/C(=N\CCSc1c(cc(cn1)C(F)(F)F)Cl)/c2c(cccc2F)F 10Z-0039 Cc1ccccc1C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl 10Z-0046 Cc1ccccc1C(=O)NCCS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F 10Z-0050 Cc1ccccc1c2nnnn2CCSc3c(cc(cn3)C(F)(F)F)Cl 10Z-0055 c1cc(cc(c1)C(F)(F)F)c2nnnn2CCSc3c(cc(cn3)C(F)(F)F)Cl 10Z-0064 c1cc(c(c(c1)F)C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)F 10Z-0067 c1ccc(c(c1)C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl 10Z-0068 c1cc(c(cc1C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl)Cl 10Z-0071 COc1ccccc1C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl 10Z-0073 Cc1ccccc1C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl 10Z-0074 c1cc(cc(c1)[N+](=O)[O-])N2CCN(CC2)CCC3C(=O)Nc4c(cccn4)O3 10Z-0209 c1ccc(c(c1)C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl)Cl 10Z-0222 c1cc(ccc1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)O 10Z-0223 COc1ccccc1C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl 10Z-0237 c1ccc(c(c1)C(=O)NCCS(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl 10Z-0238 c1cc(cc(c1)C(F)(F)F)C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl 10Z-0240 c1ccc(c(c1)c2nnnn2CCSc3c(cc(cn3)C(F)(F)F)Cl)Cl 10Z-0242 c1cc(ccc1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NN 10Z-0245 c1cc(cc(c1)C(F)(F)F)C(=O)NCCS(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl 10Z-0247 c1cc(ccc1C#N)c2ccc(cc2)OCCCBr 10Z-0248 c1ccc(cc1)NC(=O)NNC(=O)c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 10Z-0251 COc1ccccc1C(=O)NCCS(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl 10Z-0261 CN1CCN(CC1)C(=O)c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 10Z-0263 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)O 10Z-0700 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)NN 10Z-0701 c1cc(ccc1C=O)c2ccc(cc2)C(F)(F)F 10Z-0702 c1cc(cc(c1)[N+](=O)[O-])c2ccc(cc2)C=O 10Z-0703 COC(=O)c1cc(c(=O)[nH]c1)I 10Z-0704 Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)CO 10Z-0705 COc1ccc(cc1)c2ccc(cc2)C=O 10Z-0706 c1ccc(c(c1)C=O)c2cccc(c2)[N+](=O)[O-] 10Z-0707 COC(=O)c1ccc(cc1)c2ccccc2C=O 10Z-0710 CCOC(=O)c1cc(cnc1N)Br 10Z-0715 c1c(cnc(c1C(=O)O)Cl)I 10Z-0716 COC(=O)c1cc(c(nc1)Cl)I 10Z-0717 CCOC(=O)c1csc(n1)c2ccc(cc2)OC 10Z-0718 c1cc(ccc1C(=O)CN)Br.Cl 10Z-0719 c1cc(cc(c1)C(F)(F)F)c2nc(cs2)C(=O)NN 10Z-0720 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 10Z-0803 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 10Z-0804 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(cc3)O 10Z-0807 Cn1ccnc1C(=O)N2CCOCC2 10Z-0809 CCC1CCCCN1Cc2cnc(s2)Cl 10Z-0813 CC1CCCC(N1Cc2cnc(s2)Cl)C 10Z-0814 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)Br 10Z-0815 Cn1cc(cc1C(=O)OC)Br 10Z-0817 c1ccc(cc1)N2CCN(CC2)C(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 10Z-0826 Cc1cc(n[nH]1)c2cccc(c2)Br 10Z-0827 Cn1cc(cc1C(=O)N2CCN(CC2)C)Br 10Z-0829 CCOC(=O)C1CCN(CC1)Cc2c(cc(cn2)C(F)(F)F)Cl 10Z-0831 c1cc(cc(c1)NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)C(F)(F)F 10Z-0833 c1cnc(nc1)N2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl 10Z-0834 c1ccc(c(c1)N2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl 10Z-0835 c1c(cnc(c1Cl)CN2CCC(CC2)C(=O)NN)C(F)(F)F 10Z-0837 CCOC(=O)C1CCN(CC1)c2ncc(s2)C=C3C(=O)N(C(=O)N(C3=O)C)C 10Z-0840 CCOC(=O)C1CCN(CC1)c2ncc(s2)/C=N/CCc3ccccc3 10Z-0842 COCCCNC(=O)c1cn2cc(cc(c2n1)Cl)C(F)(F)F 10Z-0843 c1cnccc1CNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 10Z-0844 c1cc2c(cc1CN3CCN(CC3)Cc4c(cc(cn4)C(F)(F)F)Cl)OCO2 10Z-0845 CCc1ccc(cc1)/C=N/NC(=O)c2cn3cc(ccc3n2)I 10Z-0849 CCOC(=O)C1CCN(CC1)c2ncc(s2)C=C3C(=O)OC(OC3=O)(C)C 10Z-0851 c1cc(ccc1c2cn3cc(ccc3n2)N)Br 10Z-0852 c1cc(ccc1c2cn3cc(cc(c3n2)Cl)C(F)(F)F)NC(=O)c4cn5cc(cc(c5n4)Cl)C(F)(F)F 10Z-0854 c1cc2c(cc1Br)nc([nH]2)Cl 10Z-0926 c1cc2c(cc1Br)nc([nH]2)NN 10Z-0929 c1cc2c(cc1[N+](=O)[O-])nc([nH]2)Cl 10Z-0930 COC(=O)c1cc2ccc(cc2o1)Br 10Z-0931 COCCOc1c(cc(cn1)C(F)(F)F)Cl 10Z-5010 CCNCc1cccnc1 10Z-5027 c1c(cnc(c1Cl)OCC[NH3+])C(F)(F)F.[Cl-] 10Z-5043A c1ccc(cc1)NC(=O)OCCOc2c(cc(cn2)C(F)(F)F)Cl 10Z-5044 c1c(cc(nc1C(F)(F)F)C(F)(F)F)Cl 10Z-7005 CN(C)/C=C\C(=O)c1ccc(cc1)n2ccnc2 11A-003 C/C(=N\O)/c1ccc(cc1)n2ccnc2 11A-011 CN(C)/C=C(\C#N)/C(=O)/N=C/N(C)C 11A-012 c1cc(ccc1c2ccn[nH]2)n3ccnc3 11A-013 c1cc(ccc1c2ccno2)n3ccnc3 11A-014 c1ccc(cc1)NC(=O)n2ccc(n2)c3ccc(cc3)n4ccnc4 11A-015 c1cc(ccc1c2ccn(n2)C(=O)Nc3ccc(cc3)Cl)n4ccnc4 11A-016 c1ccc(cc1)n2c(ccn2)c3ccc(cc3)n4ccnc4 11A-018 Cc1ccc(cc1)NC(=O)n2ccc(n2)c3ccc(cc3)n4ccnc4 11A-020 C1CCn2c(nnc2CC#N)C1 11A-021 C/C(=N\OC(=O)Nc1ccccc1)/c2ccc(cc2)n3ccnc3 11A-024 CC(=O)c1ccc(cc1)n2cc[n+](c2)C.[I-] 11A-025 C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/c2ccc(cc2)n3ccnc3 11A-026 CC(C)(C)NC(=O)n1ccc(n1)c2ccc(cc2)n3ccnc3 11A-027 c1ccc(c(c1)C#N)n2ccnc2 11A-029 CN(C)C(=S)Cc1ccccc1 11A-030 c1ccc(c(c1)C(=O)N)n2ccnc2 11A-032 C[n+]1ccn(c1)c2ccccc2C#N.[I-] 11A-033 c1cc(ccc1c2ccnc(n2)N)n3ccnc3 11A-034 c1ccc(c(c1)C(=O)N/C=N/O)n2ccnc2 11A-037 COC(=O)c1ccc(cc1)n2ccnc2 11A-039 c1ccc(cc1)C(=O)Cn2cccn2 11A-040 Cc1cc(n(n1)CC(=O)c2ccccc2)C 11A-042 c1ccc(cc1)S(=O)(=O)NN/C=C/2\CCNC2=O 11A-044 c1ccc2c(c1)C(OC2=O)CC(=O)c3ccc(cc3)n4ccnc4 11A-050 c1cc(ccc1C(=O)CC(=O)N)n2ccnc2 11A-053 CC(=O)CC(=O)C1C(=O)N(C(=O)N(C1=O)C)C 11A-054 Cc1cc([nH]n1)C2C(=O)N(C(=O)N(C2=O)C)C 11A-055 Cc1cc(n(n1)C)c2c(n(c(=O)n(c2=O)C)C)O 11A-057 CC(=O)CC(=O)C1C(=O)NC(=O)NC1=O 11A-058 CC(C)(C)N1C(CC(=O)CC1=O)c2ccccc2 11A-061 C1C[NH2+]NC1=O.[Cl-] 11A-062 CC(=O)c1ccc([nH]c1=O)C(C)(C)C 11A-063 c1cc(ccc1c2nnc3n2CCCC3)Cl 11A-064 C1CN(NC1=O)C(=O)CCl 11A-065 c1ccc(cc1)S(=O)(=O)N2CCC(=O)N2 11A-066 c1cc(ccc1S(=O)(=O)N2CCC(=O)N2)Cl 11A-067 COc1ccc(cc1)S(=O)(=O)N2CCC(=O)N2 11A-068 Cc1ccc(cc1)S(=O)(=O)N2CCC(=O)N2 11A-069 c1cc(ccc1SCC(=O)N2CCC(=O)N2)Cl 11A-070 c1cc(ccc1C(=O)N2CCC(=O)N2)Cl 11A-071 c1ccc(c(c1)C(=O)N2CCC(=O)N2)Cl 11A-072 Cn1c(c(c(=O)n(c1=O)C)C=C2C(=O)N(C(=O)N(C2=O)C)C)O 11A-076 CN1C(=O)C(C(=O)N(C1=O)C)/C=N/O 11A-077 Cc1cc(on1)c2c(n(c(=O)n(c2=O)C)C)O 11A-081 c1ccc(cc1)SCC(=O)N2CCC(=O)N2 11A-082 c1cc(ccc1CSCC(=O)N2CCC(=O)N2)Cl 11A-083 Cc1c(c(on1)/C=C/Nc2ccccc2SC)[N+](=O)[O-] 11B-001 Cc1c(c(no1)c2ccccc2)C(=O)OC 11B-004 c1cc(cc(c1)C(F)(F)F)CNC=C2C=NNC2=O 11B-008 CC1=NNC(=O)C1=CNCc2cccc(c2)C(F)(F)F 11B-009 c1cc(cc(c1)C(F)(F)F)CNC=C2C(=NNC2=O)C(F)(F)F 11B-010 c1ccc(cc1)C2=NNC(=O)C2=CNCc3cccc(c3)C(F)(F)F 11B-011 COCC1=NNC(=O)C1=CNCc2cccc(c2)C(F)(F)F 11B-012 c1cc(sc1)c2cn(nc2N)c3ccc(cc3Cl)Cl 11B-013 c1ccc(cc1)n2cc(c3ccccc3c2=O)C(=O)O 11B-016 CN(C)/C=C/c1c(c(no1)c2ccccc2)C(=O)OC 11B-018 c1cc(c(cc1Cl)Cl)n2c(c(cn2)c3ccsc3)N 11B-019 c1ccc(cc1)n2c(c(cn2)c3ccsc3)N 11B-020 c1ccc2c(c1)c(cn(c2=O)c3ccc(cc3)Cl)C(=O)O 11B-021 c1ccc(cc1)n2cc(c(n2)N)c3cccs3 11B-022 COC(=O)c1c(onc1c2ccccc2)/C=C/Nc3ccccc3 11B-023 c1ccc(cc1)c2c(c(on2)/C=C/Nc3ccccc3)C#N 11B-024 COC(Cc1nnc(n1c2cccc(c2)C(F)(F)F)S)OC 11B-026 COC(=O)c1cn(c(=O)c2c1cccc2)c3ccccc3 11B-029 COC(=O)c1cn(c(=O)c2c1cccc2)c3ccc(cc3)Cl 11B-030 CN(C)C(=O)c1cn(c(=O)c2c1cccc2)c3ccc(cc3)Cl 11B-031 CNC(=O)c1cn(c(=O)c2c1cccc2)c3ccccc3 11B-032 CNC(=O)c1cn(c(=O)c2c1cccc2)c3ccc(cc3)Cl 11B-033 CN(C)C(=O)c1cn(c(=O)c2c1cccc2)c3ccccc3 11B-034 c1ccc(cc1)n2cc(c3ccccc3c2=O)C(=O)Nc4ccc(cc4)Cl 11B-035 c1ccc2c(c1)c(cn(c2=O)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)Cl 11B-036 c1ccc(cc1)c2c(c(on2)C/C=N/O)C#N 11B-038 COC(Cc1nnc(n1c2cccc(c2)C(F)(F)F)SCc3ccccc3)OC 11B-039 c1ccc(cc1)N/C=C(/C#N)\c2ccsc2 11B-040 COc1ccc(cc1)N/C=C(/C#N)\c2ccsc2 11B-041 CN(c1ccc(cc1)Cl)C(=O)c2cn(c(=O)c3c2cccc3)c4ccccc4 11B-042 CN(c1ccc(cc1)Cl)C(=O)c2cn(c(=O)c3c2cccc3)c4ccc(cc4)Cl 11B-043 c1ccc(cc1)N/C=C(/C2=NCCCCC2)\[N+](=O)[O-] 11B-045 c1ccc(cc1)Oc2ccc(cc2)NC=C3C=NNC3=O 11B-052 CC1=NNC(=O)C1=CNc2ccc(cc2)Oc3ccccc3 11B-053 c1ccc(cc1)Oc2ccc(cc2)NC=C3C(=NNC3=O)C(F)(F)F 11B-054 c1ccc(cc1)C2=NNC(=O)C2=CNc3ccc(cc3)Oc4ccccc4 11B-055 COCC1=NNC(=O)C1=CNc2ccc(cc2)Oc3ccccc3 11B-056 c1ccc(cc1)/C=C(\c2ccno2)/Oc3ccc(cc3)Cl 11B-058 c1ccnc(c1)c2cnc(nc2N3CCOCC3)N 11B-059 c1ccc(cc1)CN/C=C/c2c(c(no2)c3ccccc3)C#N 11B-063 CN(C)/C=C\1/C(=NOC1=O)c2ccccc2 11B-067 COC(CC(=O)NNC(=S)Nc1ccc(cc1)Cl)OC 11B-070 COC(=O)CN/C=C\1/C(=NOC1=O)c2ccccc2 11B-073 COC(Cc1nnc(n1c2ccc(cc2)Cl)S)OC 11B-074 c1ccc2c(c1)c(cn(c2=O)Cc3cccnc3)C(=O)O 11B-079 c1cc(ccc1C(F)(F)F)NC=C2C(=NNC2=O)C(F)(F)F 11B-080 CC1=NNC(=O)C1=CNc2ccc(cc2)C(F)(F)F 11B-082 c1ccc(cc1)C2=NNC(=O)C2=CNc3ccc(cc3)C(F)(F)F 11B-083 COCC1=NNC(=O)C1=CNc2ccc(cc2)C(F)(F)F 11B-084 c1ccc(cc1)C2=NNC(=O)C2=CN3CCCCC3 11B-086 Cc1ccc(cc1)N/C=C(/C#N)\c2ccsc2 11B-088 Cc1ccc(cc1C)N/C=C(/C#N)\c2ccsc2 11B-089 c1ccc(cc1)Oc2ccc(cc2)N/C=C(/C#N)\c3ccsc3 11B-091 CCSC(c1ccnn1C(=O)Nc2ccccc2)SCC 11B-092 COC(Cc1nnc(n1c2ccc(cc2)Cl)SCc3ccccc3)OC 11B-093 c1ccc2c(c1)c(cn(c2=O)Cc3ccccn3)C(=O)O 11B-102 CCSC(c1ccnn1S(=O)(=O)c2ccc(cc2)Cl)SCC 11B-107 c1ccc(cc1)C\2=NOC(=O)/C2=C\Nc3ccc(cc3)Cl 11B-109 Cc1c(cnc(n1)N)C(=O)Nc2ccccc2 11B-114 COc1ccc(c(c1)OC)N/C=C(/C#N)\c2ccsc2 11B-120 CSc1cccc(c1)N/C=C(/C#N)\c2ccsc2 11B-121 c1cc(ccc1N/C=C(/C#N)\c2ccsc2)Cl 11B-122 c1cc(ccc1N/C=C(\C#N)/c2ccsc2)F 11B-124 CN(C)/C=C\1/c2ccccc2C(=O)O1 11B-126 COC(=O)c1cn(c(=O)c2c1cccc2)Cc3cccnc3 11B-128 Cc1cc(n(n1)C)C 11B-132 CN(C)/C=C\1/C(=NN(C1=O)c2ccccc2)C(F)(F)F 11B-133 c1cc(c(cc1Cl)Cl)N/C=C(/C#N)\c2ccsc2 11B-134 c1ccc(cc1)N/C=C\2/c3ccccc3C(=O)O2 11B-135 c1cc(ccc1C(=O)O)N/C=C(/C#N)\c2ccsc2 11B-136 Cc1c(cnc(n1)N)C(=O)NCc2ccccc2 11B-138 c1cc(c(cc1Cl)Cl)N2C(=O)CC(=N2)C(F)(F)F 11B-140 COC(=O)c1ccc(cc1)N/C=C(/C#N)\c2ccsc2 11B-141 COC(=O)CN/C=C\1/C(=NN(C1=O)c2ccccc2)C(F)(F)F 11B-142 c1ccc(cc1)N/C=C\2/C(=NN(C2=O)c3ccccc3)C(F)(F)F 11B-143 c1ccc(cc1)N2C(=O)/C(=C\Nc3ccccc3Cl)/C(=N2)C(F)(F)F 11B-144 c1ccc(cc1)N2C(=O)/C(=C\Nc3cccc(c3)Cl)/C(=N2)C(F)(F)F 11B-145 c1ccc(cc1)N2C(=O)/C(=C\Nc3ccc(cc3)Cl)/C(=N2)C(F)(F)F 11B-146 c1ccc(cc1)N2C(=O)/C(=C\Nc3ccccc3C(F)(F)F)/C(=N2)C(F)(F)F 11B-147 c1ccc(cc1)N2C(=O)/C(=C\Nc3cccc(c3)C(F)(F)F)/C(=N2)C(F)(F)F 11B-148 c1ccc(cc1)N2C(=O)/C(=C\Nc3ccc(cc3)C(F)(F)F)/C(=N2)C(F)(F)F 11B-149 c1ccc(cc1)N2C(=O)/C(=C\NN3CCOCC3)/C(=N2)C(F)(F)F 11B-150 c1ccc(cc1)N2C(=O)/C(=C\NCc3cccnc3)/C(=N2)C(F)(F)F 11B-151 Cc1c(c(n(n1)C)C)[N+](=O)[O-] 11B-153 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)Cl)/OC2=O 11B-154 COc1ccc(cc1)N/C=C(/C#N)\c2cccs2 11B-155 c1cc(sc1)/C(=C\Nc2ccc(cc2)C(=O)O)/C#N 11B-156 CN(C)/C=C/C(=O)/C=C/c1ccccc1 11C-001 CN(C)C=CC(=O)c1ccc(cc1)OC 11C-002 COc1ccc(cc1)C(=O)C/C=N/OC 11C-003 Cc1ccc(cc1)C(=O)/C=C/N(C)C 11C-009 Cc1ccc(cc1)C(=O)C/C=N/OC 11C-010 CN(C)/C=C/C(=O)c1ccco1 11C-011 c1cc2c(cc1CN3CCN(CC3)c4[nH]nc(n4)N)OCO2 11C-014 CO/N=C/C(=C(c1ccc(cc1)Cl)O)/C=N\OC 11C-032 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)S(=O)(=O)C)/C#N 11C-045 CC(c1ccnn1C(=O)Nc2ccccc2)Oc3ccc(cc3Cl)Cl 11C-046 CCNC(=O)n1c(ccn1)C(C)Oc2ccc(cc2Cl)Cl 11C-047 CN(C)c1nnc(o1)c2ccc(cc2)Cl 11C-062 CC(c1ccnn1S(=O)(=O)c2ccccc2)Oc3ccc(cc3Cl)Cl 11C-063 CC(c1ccnn1S(=O)(=O)C)Oc2ccc(cc2Cl)Cl 11C-064 CC(c1ccnn1C(=O)c2ccccc2)Oc3ccc(cc3Cl)Cl 11C-065 CC(c1ccnn1C(=O)C)Oc2ccc(cc2Cl)Cl 11C-067 CSc1nc2nccc(n2n1)c3ccc(cc3)Cl 11C-068 c1cc(c(cc1Cl)Cl)CO/N=C\CC(=O)Nc2ccc(cc2Cl)Cl 11D-001 c1cc(c(cc1CO/N=C\CC(=O)Nc2ccc(cc2Cl)Cl)Cl)Cl 11D-002 c1ccc(cc1)Oc2ccc(cc2)NC(=O)C/C=N\OCc3ccc(cc3Cl)Cl 11D-003 CO/N=C\CC(=O)Nc1ccc(cc1)Oc2ccccc2 11D-004 c1cc(c(cc1NC(=O)CC(=O)O)Cl)Cl 11D-005 c1cc(nn2c1n[nH]c2=O)Cl 11D-006 CN(C)/C=C/C(=O)Nc1ccc(c(c1)Cl)Cl 11D-007 CN(C)/C=C(/C=N/OC)\C(=O)Nc1ccc(cc1)Cl 11D-008 c1cc(c(cc1NC(=O)C/C=N\OCc2ccc(cc2Cl)Cl)Cl)Cl 11D-009 c1cc(c(c(c1)Cl)CO/N=C\CC(=O)Nc2ccc(c(c2)Cl)Cl)Cl 11D-010 c1cc(ccc1CO/N=C\CC(=O)Nc2ccc(c(c2)Cl)Cl)[N+](=O)[O-] 11D-011 c1cc(c(cc1CO/N=C\CC(=O)Nc2ccc(c(c2)Cl)Cl)Cl)Cl 11D-012 c1ccc(cc1)NC(=O)O/N=C\CC(=O)Nc2ccc(cc2Cl)Cl 11D-013 c1cc(ccc1/N=C/c2c(nc3n2ccs3)Cl)S(=O)(=O)N 11D-014S CC(C)/N=C/c1c(nc2n1ccs2)Cl 11D-015S CCC(C)/N=C/c1c(nc2n1ccs2)Cl 11D-017S C/N=C/c1c(nc2n1ccs2)Cl 11D-018S c1csc2n1c(c(n2)Cl)/C=N/C3CCCCC3 11D-019S COC(=O)c1c(ccs1)c2ccc(o2)C(=O)Nc3cccc(c3)Cl 11D-021 COC(=O)c1c(ccs1)c2ccc(o2)C(=O)N3CCOCC3 11D-022 COC(=O)c1c(ccs1)c2ccc(o2)C(=O)NCc3ccccc3 11D-023 CNC(=O)c1ccc(o1)c2ccsc2C(=O)OC 11D-024 CN(C)/C=C/C(=O)Nc1ccccc1 11D-025 c1cc(c(cc1NC(=O)C/C=N\O)Cl)Cl 11D-026 c1cc(c(c(c1)Cl)CO/N=C\CC(=O)Nc2ccc(cc2)Cl)Cl 11D-027 c1cc(ccc1CO/N=C\CC(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] 11D-028 c1ccc(cc1)NC(=O)C/C=N\OCc2ccc(c(c2)Cl)Cl 11D-029 c1ccc(cc1)NC(=O)C/C=N\OCc2ccc(cc2Cl)Cl 11D-030 CO/N=C\CC(=O)Nc1ccc(c(c1)Cl)Cl 11D-031 COC(=O)c1c(ccs1)c2ccc(o2)C(=O)Nc3cccnc3 11D-032 COC(=O)c1ccc(o1)c2ccsc2C(=O)OC 11D-033 COCCCNc1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F 11D-034 CN(C)/C=C(\C=N\OCc1ccc(cc1Cl)Cl)/C(=O)Nc2ccc(c(c2)Cl)Cl 11D-035 c1cc(ccc1N2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)Cl 11D-036 COc1ccc(cc1)CNc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 11D-037 c1cc(ccc1N2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)F 11D-038 c1cc(ccc1/C=C/C(=O)/C=C/NNc2ccc(nn2)Cc3ccc(cc3Cl)Cl)Cl 11D-039 c1cc(sc1)/C=C\C(=O)/C=C/NNc2ccc(nn2)Cc3ccc(cc3Cl)Cl 11D-040 c1cnc(nc1)N2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 11D-041 c1cc(cc(c1)N2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)C(F)(F)F 11D-042 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ccc5c(cc(nc5n4)C(F)(F)F)C(F)(F)F 11D-043 COC(=O)c1c(ccs1)c2ccc(o2)C(=O)N 11D-044 CCCCOC(=O)c1ccc(o1)c2ccsc2C(=O)OC 11D-045 COc1ccc(cc1)/C=C/C(=O)/C=C/NNc2ccc(nn2)Cc3ccc(cc3Cl)Cl 11D-046 c1ccc(cc1)/C=C/C(=O)/C=C/NNc2ccc(nn2)Cc3ccc(cc3Cl)Cl 11D-048 c1cc(cc(c1)C(F)(F)F)CNc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 11D-049 c1cc(ccc1c2cnn(c2N)c3ccc(nn3)Cc4ccc(cc4Cl)Cl)Cl 11D-050 c1cc(sc1)c2cnn(c2N)c3ccc(nn3)Cc4ccc(cc4Cl)Cl 11D-051 COc1ccc(cc1)c2cnn(c2N)c3ccc(nn3)Cc4ccc(cc4Cl)Cl 11D-052 c1cc(ccc1c2cnn(c2N)c3ccc(nn3)Cc4ccc(cc4Cl)Cl)F 11D-053 c1ccc(cc1)c2cnn(c2N)c3ccc(nn3)Cc4ccc(cc4Cl)Cl 11D-054 CN(C)/C=N/C(=S)Nc1ccc(cc1)Cl 11D-055 Cc1c2c([nH]c(=O)n1)CCC2 11D-056 COC(=O)c1cc2c(s1)nc3n2ccs3 11D-057S Cc1c2c(nc(n1)Cl)CCC2 11D-058 CN(C)/C=N/C(=S)Nc1ccc(cc1Cl)Cl 11D-059 CN(C)/C=N/C(=S)Nc1cccc(c1)C(F)(F)F 11D-060 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=N/O)Cl 11D-061S CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Sc2ccc(cc2)Cl 11D-062S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(cc3Cl)Cl)Cl 11D-063S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(c(c3)Cl)Cl)Cl 11D-064S C[N+](=C/N=C(\Nc1ccc(cc1)Cl)/SC)C.[I-] 11D-065 CN(C)/C=C/C(=O)c1ccc(cc1Cl)Oc2ccc(cc2)Cl 11D-066 c1cc(ccc1Nc2[nH]ncn2)Cl 11D-067 c1cc(ccc1F)Sc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 11D-068 CC(=O)c1ccc(cc1Cl)Oc2ccc(cc2)Cl 11D-069 c1cc(ccc1CSc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 11D-071 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)Cl 11D-072S c1cc(c(cc1Cl)Cl)Nc2[nH]ncn2 11D-073 c1ccc(cc1)Cn2c(=O)n3c(n2)ccc(n3)Cl 11D-075 c1cc(ccc1CO/N=C/c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)[N+](=O)[O-] 11D-077S c1cc(cc(c1)Nc2[nH]ncn2)C(F)(F)F 11D-079 CN(C)/C=N/C(=S)Nc1ccccc1F 11D-080 CN(C)/C=N/C(=S)Nc1cc(cc(c1)Cl)Cl 11D-081 c1ccc(cc1)CSc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 11D-082 c1cc(ccc1Oc2ccc(c(c2)Cl)c3cc[nH]n3)Cl 11D-083 C[N+](=C/N=C(\Nc1ccccc1F)/SC)C.[I-] 11D-085 Cc1c2c(nc(n1)SCc3ccc(cc3)Cl)CCC2 11D-087 Cc1c2c(nc(n1)SCc3ccccc3Cl)CCC2 11D-090 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OC 11D-091S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/O 11D-092S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(cc3Cl)Cl 11D-093S c1cc(ccc1SC2CC(=O)OC2=O)Cl 11D-094 COC\1=CC(=O)O/C1=C\Nc2ccccc2 11D-096 COC\1=CC(=O)O/C1=C\Nc2ccc(cc2)Cl 11D-097 CO/N=C/C(/C=N/O)C(=O)Nc1ccc(cc1)Cl 11D-098 Cc1c2c(nc(n1)S(=O)(=O)Cc3ccc(cc3)Cl)CCC2 11D-099 Cc1c2c(nc(n1)S(=O)(=O)Cc3ccccc3Cl)CCC2 11D-100 c1c(cc(cc1Cl)Cl)Nc2[nH]ncn2 11D-102 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3c(cccc3Cl)Cl 11D-103S COC\1=CC(=O)O/C1=C\Nc2ccc(cc2Cl)Cl 11D-104 c1cc(cc(c1)Sc2ccc(cc2[N+](=O)[O-])C=O)C(F)(F)F 11D-106 COC\1=CC(=O)O/C1=C\Nc2ccc(cc2)Oc3ccccc3 11D-107 COC\1=CC(=O)O/C1=C\Nc2ccc(cc2)C(=O)O 11D-108 c1cc(ccc1Oc2ccc(c(c2)Cl)c3ccnc(n3)N)Cl 11D-109 c1cc(ccc1Nc2ncnc(n2)N)Cl 11D-110 c1c(c(cnn1)C(=O)N)C(=O)N 11D-111 COC\1=CC(=O)O/C1=C\Nc2ccc(cc2)C(F)(F)F 11D-112 COC(=O)c1c(ccs1)/N=C/c2c(nc3n2ccs3)Cl 11D-113S CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Sc2cccc(c2)C(F)(F)F 11D-114S c1cc(cc(c1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(c(c3)Cl)Cl)C(F)(F)F 11D-115S c1cc(cc(c1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3c(cccc3Cl)Cl)C(F)(F)F 11D-116S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(c(c3)Cl)Cl 11D-119S CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2 11D-120S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(cc3Cl)Cl 11D-121S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(c(c3)Cl)Cl 11D-122S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/OCc3c(cccc3Cl)Cl 11D-123S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=N/O 11D-124S c1ccc(c(c1)CSc2ccc(cc2[N+](=O)[O-])/C=N/O)Cl 11D-125S CO/N=C/c1ccc(c(c1)[N+](=O)[O-])SCc2ccccc2Cl 11D-126S Cc1c2c(nc(n1)SCc3ccccc3)CCC2 11D-127 Cc1c2c(nc(n1)S(=O)(=O)Cc3ccccc3)CCC2 11D-128 COc1ccc(cc1)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 11D-130 c1cc(ccc1Sc2c(n3ccsc3n2)C#N)Cl 11D-133S c1cc(cc(c1)C(F)(F)F)CSc2ccc(cc2[N+](=O)[O-])C=O 11D-134S c1cc(ccc1Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)F 11D-135 c1cc(ccc1C(F)(F)F)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 11D-136 COC(=O)c1cn(nc1c2ccncc2)c3ccccc3 11D-510 c1ccc(c(c1)CN2c3ccccc3C4(C5CC6CC(C5)CC4C6)OC2=O)Cl 11D-511 Cc1cc(n2c(n1)nc(n2)SCc3ccccc3)O 11D-541 Cc1ncc(c(n1)c2ccncc2)C(=O)OC 11D-546 c1ccc(cc1)CSc2nc3nc(cc(n3n2)O)O 11D-555 Cc1cc(n2c(n1)nc(n2)SCc3ccccc3)OC 11D-557 Cc1ccn2c(c1)nc(c2C(=O)Nc3ccc(cc3)F)C 11D-572 Cc1cccn2c1nc(c2C(=O)Nc3ccc(cc3F)F)C 11D-573 Cc1c(n2ccccc2n1)C(=O)Nc3ccc(cc3)Cl 11D-575 Cc1cc(n2c(n1)nc(n2)S(=O)(=O)Cc3ccccc3)OC 11D-582 COc1cc(n2c(n1)nc(n2)S(=O)(=O)Cc3ccccc3)OC 11D-595 c1ncn(n1)CC(=N)N.Cl 11E-001 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccccc2C(F)(F)F 11E-002 c1c(cnc(c1Cl)NNC(=N)Cn2cncn2)C(F)(F)F 11E-003 c1cc(nnc1NNC(=N)Cn2cncn2)Cl 11E-004 Cc1nc(cn1Cc2c(cccc2Cl)Cl)C(=O)C 11E-005 c1cc(nc(c1)Cl)NNC(=N)Cn2cncn2 11E-007 c1cc(nc(c1)Cl)n2cnc(n2)Cn3cncn3 11E-008 c1ncn(n1)CC(=N)NNC(=O)CC#N 11E-010 c1cc(nc(c1)F)NNC(=N)Cn2cncn2 11E-011 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)Br 11E-012 c1cc(c(cc1Cl)Cl)CO/N=C\NC(=S)Nc2cc(cc(c2)Cl)Cl 11E-013 c1cc(c(cc1Cl)Cl)CONC(=N)Cn2cncn2.Cl 11E-014 c1ncn(n1)Cc2nc([nH]n2)CC#N 11E-015 CNC(=O)c1cc(c[nH]1)C(=O)c2ccccc2Br 11E-016 c1cnccc1C(=O)NNC(=N)Cn2cncn2 11E-017 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2F)C(F)(F)F 11E-018 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccccc2Br 11E-019 c1cnccc1c2nc([nH]n2)Cn3cncn3 11E-020 Cc1nc(cn1Cc2c(cccc2Cl)Cl)/C(=N\O)/C 11E-023 Cc1nc(cn1Cc2c(cccc2Cl)Cl)C(=O)/C=C/N(C)C 11E-024 c1ncn(n1)CC(=O)NN 11E-025 CN(C)/C=N/C(=S)Nc1ccc(cc1)F 11E-027 c1cc(c(cc1F)C(F)(F)F)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 11E-028 Cc1nc(cn1Cc2c(cccc2Cl)Cl)c3cc[nH]n3 11E-029 CNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2C(F)(F)F)F 11E-030 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2C(F)(F)F)F 11E-031 c1cc(ccc1NC(=S)N/C=N\OCc2ccc(cc2Cl)Cl)F 11E-032 CN(C)/C=N/C(=S)Nc1ccc(cc1F)Br 11E-033 c1cc(c(cc1Cl)Cl)CO/N=C\NC(=S)Nc2ccc(cc2F)Br 11E-035 c1cc(c(c(c1)Cl)CONC(=N)Cn2cncn2)Cl.Cl 11E-037 c1cc(c(cc1F)Cl)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 11E-038 c1csc(c1Cl)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 11E-039 CNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)F 11E-040 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2c(ccs2)Cl 11E-041 Cc1cc(n(n1)c2ncc(cn2)C#N)C 11E-042 COc1ccc(cc1)c2ccnn2c3ncc(cn3)C#N 11E-043 c1ccc(cc1)S(=O)(=O)n2ccc(n2)c3cccc(c3)Oc4c(cc(cn4)C(F)(F)F)Cl 11E-044 Cc1nc(cn1Cc2c(cccc2Cl)Cl)c3ccnc(n3)N 11E-045 c1cc(cc(c1)Cl)OC/C(=N/NC(=O)c2ccncc2)/N 11E-046 c1cc(cc(c1)Cl)OCc2nc([nH]n2)c3ccncc3 11E-047 c1cc(c(cc1Cl)Cl)c2ccnn2c3ncc(cn3)C#N 11E-048 c1cc(cc(c1)Cl)OC/C(=N/Nc2cccc(n2)Cl)/N 11E-051 c1cc(cc(c1)Cl)OCc2ncn(n2)c3cccc(n3)Cl 11E-052 c1cc(ccc1OC/C(=N/NC(=O)c2ccncc2)/N)F 11E-053 c1cc(ccc1OCc2nc([nH]n2)c3ccncc3)F 11E-054 c1cc(ccc1OC/C(=N/NC(=O)CC#N)/N)F 11E-055 COc1ccc(cc1)/N=C(\C[N+](=O)[O-])/NN/C=C\2/c3ccccc3C(=O)O2 11E-057 CCOC(=O)C(=O)NNc1c(cc(cn1)C(F)(F)F)Cl 11E-058 CS(=O)(=O)n1ccc(n1)c2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl 11E-059 c1c(cnc(c1Cl)NNC(=O)C(=O)N)C(F)(F)F 11E-060 c1ccc2c(c1)/C(=C/NN/C(=N/c3ccc(cc3)F)/C[N+](=O)[O-])/OC2=O 11E-061 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)N=[N+]=[N-] 11E-062 Cn1cc(cc1C=O)C(=O)c2ccc(cc2Cl)Cl 11E-065 c1ccc(cc1)NC(=O)Nc2cc(c[nH]2)C(=O)c3ccc(cc3Cl)Cl 11E-067 COC(=O)Nc1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 11E-068 CCOC(=O)C(=O)Nc1ccc(cc1Cl)Cl 11E-069 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)c3nnco3 11E-070 c1cc(c(cc1Cl)Cl)NC(=O)C(=O)NN 11E-071 c1cc(c(cc1Cl)Cl)NC(=O)C(=O)N 11E-072 CN(C)/C=N/C(=O)C(=O)Nc1ccc(cc1Cl)Cl 11E-073 c1ccc2c(c1)/C(=C/NNC(=O)C(=O)Nc3ccc(cc3Cl)Cl)/OC2=O 11E-075 c1cc(c(cc1Cl)Cl)CO/N=C/NC(=O)C(=O)Nc2ccc(cc2Cl)Cl 11E-076 c1ccc(cc1)n2cnc(n2)OCC#N 11E-077 CC(=O)/C(=C/c1ccccc1)/Oc2ccc(cc2)C#N 11E-078 c1cc(cc(c1)C(F)(F)F)Cn2cc(ccc2=O)C(=O)NN 11E-301S c1ccnc(c1)NC(=S)Nc2cccnc2 11E-302S CSc1nnc(o1)c2ccc(=O)n(c2)Cc3ccccc3 11E-303S C#CCSc1nnc(o1)c2ccc(=O)n(c2)Cc3ccccc3 11E-304S CNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2cccc(c2)C(F)(F)F 11E-305S C=CCNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2cccc(c2)C(F)(F)F 11E-306S c1cc(cc(c1)Cl)Cn2cccc(c2=O)c3nnc(o3)SCc4ccc(cc4Cl)Cl 11E-308S CSc1nnc(o1)c2cccn(c2=O)Cc3cccc(c3)Cl 11E-309S C=CCSc1nnc(o1)c2ccc(=O)n(c2)Cc3ccccc3 11E-310S c1ccc(cc1)Cn2cc(ccc2=O)c3nnc(o3)SCc4ccc(c(c4)Cl)Cl 11E-311S Cn1c(nnc1S)c2ccc(=O)n(c2)Cc3cccc(c3)C(F)(F)F 11E-312S C=CCn1c(nnc1S)c2ccc(=O)n(c2)Cc3cccc(c3)C(F)(F)F 11E-313S Cc1c(c(n(n1)c2ccccc2)N)c3ccccc3 11E-314S Cc1c(c(n(n1)c2cccc(c2)[N+](=O)[O-])N)c3ccccc3 11E-315S Cc1c(c(n(n1)c2ccccc2)N)c3ccc(cc3)Cl 11E-316S c1cc(cc(c1)C(F)(F)F)Cn2cc(ccc2=O)c3nnc(o3)S 11E-317S c1ccc(cc1)Cn2cc(ccc2=O)c3nnc(n3N)S 11E-318S c1ccc(cc1)Cn2cccc(c2=O)c3nnc(o3)SCc4ccc(cc4)C(F)(F)F 11E-319S c1ccc(cc1)Cn2cccc(c2=O)c3nnc(o3)SCc4cccc(c4)C(F)(F)F 11E-320S C=CCn1c(n[nH]c1=S)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 11E-322S CCOC(=O)CSC(=S)Nc1cccnc1 11E-323S CCOC(=O)CS/C(=N/c1cccnc1)/SC.I 11E-324S CCNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2cccc(c2)C(F)(F)F 11E-326S Cc1c(c(n(n1)c2cccc(c2)[N+](=O)[O-])N)c3ccc(cc3)Cl 11E-327S Cc1c(c(n(n1)c2cccc(c2)Cl)N)c3ccc(cc3)Cl 11E-328S CCn1c(nnc1S)c2ccc(=O)n(c2)Cc3cccc(c3)C(F)(F)F 11E-329S c1ccnc(c1)N2CCN(CC2)C(=O)c3ccc(=O)n(c3)Cc4ccc(c(c4)Cl)Cl 11E-330S CNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2Cl)Cl 11E-332S C=CCNC(=S)NNC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2Cl)Cl 11E-333S C=CCNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 11E-334S Cc1c(c(n(n1)c2ccccc2)N)c3cccc(c3)C(F)(F)F 11E-335S Cc1c(c(n(n1)c2cccc(c2)Cl)N)c3cccc(c3)C(F)(F)F 11E-336S CSc1nnc(n1CC=C)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-340S C=CCn1c(nnc1SCC=C)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-341S C=CCn1c(nnc1SCc2ccc(cc2Cl)Cl)c3cccn(c3=O)Cc4ccc(cc4Cl)Cl 11E-342S C=CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3cccn(c3=O)Cc4ccc(cc4Cl)Cl 11E-343S C=CCn1c(nnc1SCc2ccc(cc2)C(F)(F)F)c3cccn(c3=O)Cc4ccc(cc4Cl)Cl 11E-344S c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)c3nnc(o3)S 11E-345S Cc1c(c(n(n1)c2cccc(c2)[N+](=O)[O-])N)c3cccc(c3)C(F)(F)F 11E-346S Cc1c(c(n(n1)c2cccc(c2)[N+](=O)[O-])N)c3cccc(c3)Cl 11E-347S C=CCn1c(nnc1S)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 11E-348S Cn1c(nnc1S)c2ccc(=O)n(c2)Cc3ccc(cc3Cl)Cl 11E-349S C=CCn1c(nnc1S)c2ccc(=O)n(c2)Cc3ccc(cc3Cl)Cl 11E-350S Cn1c(nnc1SC)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 11E-351S Cn1c(nnc1SCc2ccccc2)c3cccn(c3=O)Cc4ccc(c(c4)Cl)Cl 11E-352S Cn1c(nnc1SCC#C)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 11E-353S Cc1c(c(n(n1)c2cccc(c2)C(F)(F)F)N)c3ccc(cc3)Cl 11E-354S Cc1ccccc1n2c(c(c(n2)C)c3ccc(cc3)Cl)N 11E-356S Cc1c(c(n(n1)c2ccc(cc2)OC)N)c3ccc(cc3)Cl 11E-357S Cc1c(c(n(n1)c2ccc(cc2)Cl)N)c3ccc(cc3)Cl 11E-358S C=CCSc1nnc(o1)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-359S c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)c3nnc(o3)SCc4ccc(cc4)Cl 11E-360S CCNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccc(cc2)Cl 11E-362S C=CCNC(=S)NNC(=O)c1cccn(c1=O)Cc2ccc(cc2)Cl 11E-363S CCn1c(nnc1S)c2cccn(c2=O)Cc3ccc(cc3)Cl 11E-364S C=CCn1c(nnc1S)c2cccn(c2=O)Cc3ccc(cc3)Cl 11E-365S Cn1c(nnc1SC)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-366S Cn1c(nnc1SCC=C)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-367S Cn1c(nnc1SCC#C)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-368S Cn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3cccn(c3=O)Cc4ccc(cc4Cl)Cl 11E-369S Cn1c(nnc1SCc2cccc(c2)C(F)(F)F)c3cccn(c3=O)Cc4ccc(cc4Cl)Cl 11E-370S CCn1c(nnc1SC)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-371S CCn1c(nnc1SC)c2cccn(c2=O)Cc3ccc(cc3)Cl 11E-373S CCn1c(nnc1SCC=C)c2cccn(c2=O)Cc3ccc(cc3)Cl 11E-374S CSc1nnc(n1CC=C)c2cccn(c2=O)Cc3ccc(cc3)Cl 11E-375S C=CCn1c(nnc1SCC#C)c2cccn(c2=O)Cc3ccc(cc3)Cl 11E-377S C=CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3cccn(c3=O)Cc4ccc(cc4)Cl 11E-378S C=CCn1c(nnc1SCc2c(cccc2Cl)F)c3cccn(c3=O)Cc4ccc(cc4)Cl 11E-379S c1cc(ccc1N2C(=O)CC(=N2)C(F)(F)F)Cl 11E-380S CCn1c(nnc1SCC=C)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 11E-381S CCn1c(nnc1SCC(=O)c2ccccc2)c3cccn(c3=O)Cc4ccc(cc4Cl)Cl 11E-382S CN(C)/C=C(/c1ccccc1)\C(=O)OC 11E-384S C=CCn1c(nnc1SCC#C)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 11E-389S C=CCn1c(nnc1SCc2ccccc2)c3cccn(c3=O)Cc4ccc(c(c4)Cl)Cl 11E-390S CSc1nnc(n1CC=C)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 11E-394S CO/N=C\1/c2ccccc2N(C1=O)Cc3ccc(c(c3)Cl)Cl 11E-395S c1ccc(cc1)c2c[nH]n(c2=O)c3ccccc3 11E-396S c1ccc(cc1)c2c[nH]n(c2=O)c3cccc(c3)Cl 11E-397S c1ccc(cc1)c2c[nH]n(c2=O)c3cccc(c3)C(F)(F)F 11E-398S c1ccc2c(c1)C(=O)C(=O)N2Cc3cccc(c3)C(F)(F)F 11E-400S c1ccc2c(c1)/C(=N/OCc3ccc(cc3Cl)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11E-403S c1ccc2c(c1)/C(=N/OCc3ccc(cc3)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11E-404S c1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3ccc(c(c3)Cl)Cl 11E-405S Cc1c(c(=O)n([nH]1)c2ccccc2)c3ccccc3 11E-408S Cc1c(c(=O)n([nH]1)c2cccc(c2)Cl)c3ccccc3 11E-409S Cc1c(c(=O)n([nH]1)c2cccc(c2)C(F)(F)F)c3ccccc3 11E-410S Cc1c(c(=O)n([nH]1)c2cccc(c2)[N+](=O)[O-])c3ccccc3 11E-411S c1ccc(cc1)C(=O)O/N=C\2/c3ccccc3N(C2=O)Cc4ccc(c(c4)Cl)Cl 11E-413S c1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11E-414S c1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3Cl)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11E-415S c1ccc(cc1)c2c[nH]n(c2=O)c3cccc(c3)[N+](=O)[O-] 11E-420S CN(C)/C=C(\c1cccc(c1)Cl)/C(=O)OC 11E-423S c1ccc2c(c1)/C(=N/OCc3ccc(cc3)Cl)/C(=O)N2Cc4cccc(c4)C(F)(F)F 11E-424S c1ccc2c(c1)/C(=N/OCc3ccc(cc3Cl)Cl)/C(=O)N2Cc4cccc(c4)C(F)(F)F 11E-425S c1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3cccc(c3)C(F)(F)F 11E-432S c1ccc(cc1)n2c(=O)c(c[nH]2)c3ccc(cc3)Cl 11E-433S c1cc(cc(c1)Cl)n2c(=O)c(c[nH]2)c3ccc(cc3)Cl 11E-434S c1cc(cc(c1)n2c(=O)c(c[nH]2)c3ccc(cc3)Cl)C(F)(F)F 11E-435S c1cc(cc(c1)[N+](=O)[O-])n2c(=O)c(c[nH]2)c3ccc(cc3)Cl 11E-436S CO/N=C\1/c2ccccc2N(C1=O)Cc3cccc(c3)C(F)(F)F 11E-437S c1ccc2c(c1)/C(=N/OCc3c(cccc3Cl)Cl)/C(=O)N2Cc4cccc(c4)C(F)(F)F 11E-438S c1ccc(cc1)n2c(=O)c(c[nH]2)c3cccc(c3)Cl 11E-439S c1cc(cc(c1)Cl)c2c[nH]n(c2=O)c3cccc(c3)Cl 11E-440S c1cc(cc(c1)Cl)c2c[nH]n(c2=O)c3cccc(c3)[N+](=O)[O-] 11E-441S CN(C)c1nc(c(c(=O)o1)C#N)Nc2ccccc2 11E-900 CN(C)c1nc(c(c(=O)o1)C#N)N2CCN(CC2)c3ccccc3 11E-901 COc1ccc(cc1)C(=O)C[n+]2ccccc2.[I-] 11E-902 CC(=O)N1CN(C=C1)C(=O)C 11E-903 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3ccc(cc3Cl)Cl 11E-904 CN(C)c1nc(c(c(=O)o1)C#N)OC 11E-905 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3ccc(cc3)[N+](=O)[O-] 11E-906 c1ccc(cc1)c2nnc3n2c4ccccc4[nH]c3=O 11E-907 c1ccc2c(c1)nc(c3n2cnn3)Sc4ncccn4 11E-909 CN1CCN(CC1)c2c(c(=O)oc(n2)N(C)C)C#N 11E-910 c1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccc(cc5Cl)Cl 11E-911 COc1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccc(cc5Cl)Cl 11E-912 c1ccc2c(c1)c3nnc(n3c(n2)Nc4ccc(c(c4)Cl)Cl)c5ccc(cc5Cl)Cl 11E-913 Cc1cc(n(n1)CCOC(=O)c2ccccc2)c3c(nn(c3O)c4ccccc4)C 11E-914 COc1ccc(cc1)Oc2nc3ccccc3c4n2c(nn4)c5ccccc5F 11E-915 CNc1nc2ccccc2c3n1c(nn3)c4ccc(c(c4)Cl)Cl 11E-916 CN1CCN(CC1)c2nc3ccccc3c4n2c(nn4)c5ccc(c(c5)Cl)Cl 11E-917 CCOC(=O)C(=C1OCCO1)C#N 11E-918 C(COc1c(c(=O)[nH]c(n1)N)C#N)O 11E-920 CCOC(=O)c1c(n(nc1OCCO)c2ccccc2)N 11E-921 c1ccc2c(c1)CCN2C(=O)CC(=O)N3CCc4c3cccc4 11E-922 CCOC(=O)NC(=O)CC#N 11E-923 CCO/C=C(\C#N)/C(=O)NC(=O)OCC 11E-924 Cn1cc(c(=O)[nH]c1=O)C#N 11E-925 c1ccc(cc1)Cn2cc(c(=O)[nH]c2=O)C#N 11E-926 CCOC(=O)NC(=O)/C(=C\Nc1ccc(cc1)Cl)/C#N 11E-927 c1ccc(cc1)CN2CC(C(=O)NC2=O)C(=N)N 11E-928 CN1CC(C(=O)NC1=O)C(=N)N 11E-929 c1ccc(cc1)Oc2nc3ccccc3c4n2c(nn4)c5ccccc5F 11E-930 COc1ccc(cc1)Oc2nc3ccccc3c4n2c(nn4)c5ccc(cc5)Br 11E-931 c1cc(ccc1n2cc(c(=O)[nH]c2=O)C#N)Cl 11E-932 c1ccc2c(c1)c3nnc(n3c(n2)Oc4ccc(cc4Cl)Cl)c5ccccc5F 11E-933 c1ccc(cc1)Oc2nc3ccccc3c4n2c(nn4)c5ccc(c(c5)Cl)Cl 11E-934 c1ccc(cc1)Oc2nc3ccccc3c4n2c(nn4)c5ccc(cc5)Br 11E-935 c1cc[nH+]c(c1)c2[nH]c(=O)c(c(n2)OCCO)C#N.[Cl-] 11E-937 c1cc(ccc1N2CC(C(=O)NC2=O)C(=N)N)Cl 11E-938 c1ccc2c(c1)c3nnc(n3c(n2)Oc4ccc(cc4Cl)Cl)c5ccc(cc5)Br 11E-939 c1ccc2c(c1)c3nnc(n3c(n2)Oc4ccc(cc4Cl)Cl)c5ccc(c(c5)Cl)Cl 11E-940 CCOC(=O)NC(=O)/C(=C\Nc1ccccc1)/C#N 11E-941 c1ccc(cc1)n2cc(c(=O)[nH]c2=O)C#N 11E-942 c1ccc(cc1)N2C(=O)NC3(N2)CCCc4c3cccc4 11E-943 CCOC(=O)NC(=O)C(/C=N/OCc1ccc(cc1)Cl)C#N 11E-944 CCOC(=O)NC(=O)/C(=C/N1CCN(CC1)Cc2ccccc2)/C#N 11E-945 CCOC(=O)NC(=O)/C(=C\Nc1cccnc1)/C#N 11E-946 c1cc(ccc1COn2cc(c(=O)[nH]c2=O)C#N)Cl 11E-947 CCOC(=O)NC(=O)/C(=C\Nc1ccc(cc1)C(=O)C)/C#N 11E-948 c1ccc(cc1)N2CC(C(=O)NC2=O)C(=N)N 11E-949 CC(=O)c1ccc(cc1)n2cc(c(=O)[nH]c2=O)C#N 11E-950 c1cc(cnc1)n2cc(c(=O)[nH]c2=O)C#N 11E-951 CCOC(=O)NC(=O)c1c[nH]n(c1=N)c2ccccc2 11E-952 CCOC(=O)NC(=O)/C(=C\Nc1ccc(cc1)OC)/C#N 11E-953 CCOC(=O)NC(=O)/C(=C\Nc1ccsc1C(=O)OC)/C#N 11E-954 CCOC(=O)NC(=O)C(/C=N/OC)C#N 11E-955 COc1ccc(cc1)n2cc(c(=O)[nH]c2=O)C#N 11E-956 COn1cc(c(=O)[nH]c1=O)C#N 11E-957 CC(=O)c1cn(c(=O)[nH]c1=O)OCc2ccc(cc2)Cl 11E-960 COC(=O)c1c(ccs1)n2cc(c(=O)[nH]c2=O)C#N 11E-961 CCOC(=O)c1c(onc1OCCO)N 11E-962 CCOC(=O)c1c(onc1OCCOC(=O)c2ccc(cc2)Cl)N 11E-963 CCOC(=O)c1c(n(nc1OCCO)c2ccc(cc2)Cl)N 11E-964 CC(=O)c1cn(c(=O)[nH]c1=O)OC 11E-965 CCOC(=O)c1c(onc1OCCOC(=O)c2ccc(cc2Cl)Cl)N 11E-968 Cn1c(ccc1C(=O)OC)/C(=C/c2ccc(cc2)Cl)/C#N 11F-001 CC1(OCC(O1)C2C(=C(C(=O)O2)O)O)C 11F-002 c1c(cnc(c1Cl)NCC(=O)NN)C(F)(F)F 11F-003 c1cc(cc(c1)N/C=C/c2nc(c(s2)C#N)C(F)(F)F)C(F)(F)F 11F-004 Cn1c(ccc1C(=O)O)/C(=C/c2ccc(cc2)Cl)/C#N 11F-006 c1cc(ccc1COc2ccsc2C(=O)O)F 11F-007 c1ccc(cc1)COC(=O)/C=C/c2c(cc(cn2)C(F)(F)F)Cl 11F-008 Cn1c(ccc1C(=O)NCCCOC)/C(=C/c2ccc(cc2)Cl)/C#N 11F-009 c1ccc(cc1)COc2ccsc2C(=O)O 11F-010 CCOC(=O)C(C)(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)OCC 11F-011 c1ccnc(c1)SCc2c(cc(cn2)C(F)(F)F)Cl 11F-018 CCc1c(cc(cn1)C(F)(F)F)Cl 11F-019 c1cc(ccc1OCC(=N)NNC(=O)CNc2c(cc(cn2)C(F)(F)F)Cl)Cl 11F-020 c1ccc(cc1)COc2ccsc2NC(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 11F-021 c1cc(ccc1COc2ccsc2NC(=O)NNc3c(cc(cn3)C(F)(F)F)Cl)F 11F-022 c1cc(c(cc1Cl)Cl)COc2ccsc2NC(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 11F-023 CNC(=S)NNC(=O)CNc1c(cc(cn1)C(F)(F)F)Cl 11F-024 c1cc(cc(c1)C(F)(F)F)COc2ccsc2NC(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 11F-025 Cn1c(nnc1S)CNc2c(cc(cn2)C(F)(F)F)Cl 11F-026 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)Nc2ccc(cc2)Cl 11F-030 c1cc(ccc1OCc2[nH]c(nn2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl 11F-031 Cc1nc(c(s1)C(=O)OCC(=O)c2ccccc2)C(F)(F)F 11F-032 CN(C)/C=N/NC(=O)CNc1c(cc(cn1)C(F)(F)F)Cl 11F-033 CN(C)/C=N/C(=O)CNc1c(cc(cn1)C(F)(F)F)Cl 11F-034 c1ccc(c(c1)c2nnco2)Oc3c(cc(cn3)C(F)(F)F)Cl 11F-037 COc1ccc(cc1)OCC(=N)NNC(=O)c2cccnc2Oc3ccccc3 11F-044 Cc1nc(c(s1)C(=O)OCC(=O)c2cccc(c2)C(F)(F)F)C(F)(F)F 11F-045 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)N2CCN(CC2)c3ccc(cc3)Cl 11F-046 COC(=O)/C=C/c1c(cc(cn1)C(F)(F)F)Cl 11F-049 CO/N=C/NC(=O)CNc1c(cc(cn1)C(F)(F)F)Cl 11F-050 c1c(cnc(c1Cl)n2cc(cn2)C#N)C(F)(F)F 11F-051 c1cc(ccc1C(F)(F)F)N/N=C(\C#N)/N=N/c2ccc(cc2)C(F)(F)F 11F-052 c1ccc2c(c1)/C(=C/c3c(cc(cn3)C(F)(F)F)Cl)/OC2=O 11F-055 c1ccc2c(c1)c(n[nH]c2=O)Cc3c(cc(cn3)C(F)(F)F)Cl 11F-056 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)OCC(=O)c2ccc(cc2)Cl 11F-057 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)Cl)O 11F-059 CC(C)(C(=O)O)n1cncn1 11F-063 c1c(cnc(c1Cl)NNC=C2C(=O)CCCC2=O)C(F)(F)F 11F-100 CCN(Cc1cccc(c1)C(F)(F)F)C(=O)c2cc(cc(c2)Cl)Cl 11F-301S C#CCN(Cc1cccc(c1)C(F)(F)F)C(=O)c2cc(cc(c2)Cl)Cl 11F-302S c1cc(ncc1[N+](=O)[O-])n2cncn2 11F-303S CC1(C=C(N=C(N1)SC)/C=C/c2ccc(cc2)Cl)C 11F-304S CCCCC(=O)OCc1c(nn(c1Cl)C)C(F)(F)F 11F-305S Cn1c(c(c(n1)C(F)(F)F)COC(=O)CCl)Cl 11F-307S c1ccc2c(c1)C(=O)C(=O)N2Cc3ccc(cc3)Cl 11F-308S CC1(C=C(N=C(N1)SC)/C=C/c2ccc(cc2)C(F)(F)F)C 11F-309S c1cc(cc(c1)C(F)(F)F)CN(C2CC2)C(=O)c3cc(cc(c3)Cl)Cl 11F-310S CC(=O)OCc1c(nn(c1Cl)C)C(F)(F)F 11F-312S Cc1ccc(cc1)COn2c3cc(ccc3nc2c4ccccc4)[N+](=O)[O-] 11F-314S Cc1cc(cc(c1)COn2c3cc(ccc3nc2c4ccccc4)[N+](=O)[O-])C 11F-315S Cc1ccc(cc1)c2nc3ccc(cc3n2OCC(=O)O)Cl 11F-316S Cc1ccc(cc1)c2nc3ccc(cc3n2OC(C)C(=O)O)Cl 11F-317S COC(=O)c1cc(c(nc1)n2cncn2)Cl 11F-319S c1cc(ncc1C#N)n2cncn2 11F-320S c1ccc(cc1)Cc2nc3ccccc3c(n2)S 11F-321S CN(C)C(=O)On1c2cc(ccc2nc1c3ccccc3)Cl 11F-322S c1ccc(cc1)c2nc3ccc(cc3n2OCc4c(cccc4Cl)F)Cl 11F-323S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(c(c4)Cl)Cl)Cl 11F-324S c1ccc(cc1)c2nc3ccc(cc3n2OCc4c(cccc4Cl)Cl)Cl 11F-325S CC1(C=C(N=C(N1)SC)/C=C/c2ccc(cc2)F)C 11F-326S CC1(C=C(N=C(N1)SC)/C=C/c2ccc(cc2Cl)F)C 11F-327S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F 11F-332S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(cc2)F 11F-333S C/N=C(\c1ccc(cc1Cl)S(=O)(=O)C)/Nc2ccc(cc2)Cl 11F-334S CCSC1=NC(=CC(N1)(C)C)/C=C/c2c(cccc2Cl)Cl 11F-335S CCSC1=NC(=CC(N1)(C)C)/C=C/c2ccc(cc2Cl)Cl 11F-336S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4)Br)[N+](=O)[O-] 11F-337S c1ccc(cc1)c2nc3ccc(cc3n2OCc4c(cccc4Cl)Cl)[N+](=O)[O-] 11F-338S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4Cl)Cl)[N+](=O)[O-] 11F-342S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(c(c4)Cl)Cl)[N+](=O)[O-] 11F-344S c1cc(ncc1/C(=N/O)/N)n2cncn2 11F-345S c1cc(cc(c1)Cl)c2nc3ccc(cc3n2O)[N+](=O)[O-] 11F-347S CCOC(=O)C(C)On1c2cc(ccc2nc1c3ccccc3)[N+](=O)[O-] 11F-348S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)C(F)(F)F 11F-350S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(cc2F)F 11F-352S CCC/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(cc2)Cl 11F-354S CCCC/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(cc2)Cl 11F-355S COc1cccc(c1)c2nc3ccc(cc3n2O)[N+](=O)[O-] 11F-359S CCSC1=NC(=CC(N1)(C)C)/C=C/c2ccc(cc2)OC(F)(F)F 11F-360S CC1=CC(NC(=N1)SCC=C)(C)C 11F-361S CN(c1ccc(cc1)Cl)C(=O)c2cccc(c2)C(F)(F)F 11F-362S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(cc2)C(F)(F)F 11F-364S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(cc2)Br 11F-365S c1cc(ccc1C(=O)Nc2ccc(cc2)Cl)C(F)(F)F 11F-366S c1cc(ccc1NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl 11F-367S Cc1cccc(c1)C(=O)Nc2ccc(cc2)Cl 11F-368S CCSC1=NC(=CC(N1)(C)C)/C=C/c2cccnc2 11F-369S CCOC(=O)c1ccc(nc1)n2cncn2 11F-370S Cc1ccc(cc1)CN2c3ccccc3/C(=N/O)/C2=O 11F-371S c1ccc(cc1)c2nc3ccc(cc3n2OCC(=O)O)[N+](=O)[O-] 11F-372S c1ccc(cc1)Cc2nc3ccccc3c(n2)SCc4c(cccc4Cl)Cl 11F-373S c1ccc(cc1)Cc2nc3ccccc3c(n2)SCc4ccccc4 11F-374S c1ccc2c(c1)C(=O)C(=O)N2Cc3cccc(c3)Cl 11F-375S Cc1ccc(cc1)c2nc3ccc(cc3n2OCC(=O)N)Cl 11F-376S COc1cccc(c1)c2nc3ccccc3n2O 11F-377S CCOC(=O)COn1c2cc(ccc2nc1c3cccc(c3)Cl)[N+](=O)[O-] 11F-378S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)S 11F-379S COc1cccc(c1)C(=O)Nc2ccc(cc2)Cl 11F-380S C/N=C(\c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/Nc2ccc(cc2)Cl 11F-381S C/N=C(\c1ccc(cc1)C(F)(F)F)/Nc2ccc(cc2)Cl 11F-384S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)SCc4ccc(c(c4)Cl)Cl 11F-385S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)SCc4ccc(cc4Cl)Cl 11F-386S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)SCc4cccc(c4)C(F)(F)F 11F-387S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)CCl)/C2=O 11F-388S C#CCSc1c2ccccc2nc(n1)Cc3ccc(cc3)Cl 11F-389S C=CCSc1c2ccccc2nc(n1)Cc3ccc(cc3)Cl 11F-390S c1cc(cc(c1)Cl)c2nc3ccc(cc3n2OCc4ccc(cc4Cl)Cl)[N+](=O)[O-] 11F-391S c1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3cccc(c3)Cl 11F-392S c1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3ccc(cc3)Cl 11F-393S CC1(C=C(N=C(N1)SCC=C)/C=C/c2c(cccc2Cl)Cl)C 11F-394S Cc1cccc(c1)/C(=N\C)/Nc2ccc(cc2)Cl 11F-395S C/N=C(\c1cccc(c1)OC)/Nc2ccc(cc2)Cl 11F-396S CSc1c2ccccc2nc(n1)Cc3ccc(cc3)Cl 11F-397S Cc1ccc(cc1)COn2c3cc(ccc3nc2c4cccc(c4)Cl)[N+](=O)[O-] 11F-398S c1ccc(c(c1)COn2c3cc(ccc3nc2c4cccc(c4)Cl)[N+](=O)[O-])Cl 11F-399S CN(C)C(=O)On1c2cc(ccc2nc1c3cccc(c3)Cl)[N+](=O)[O-] 11F-400S c1cc(cc(c1)C(F)(F)F)COn2c3cc(ccc3nc2c4cccc(c4)Cl)[N+](=O)[O-] 11F-401S CC1(C=C(N=C(N1)SCC=C)/C=C/c2ccc(cc2Cl)Cl)C 11F-402S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)C)/C2=O 11F-405S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)C(Cl)Cl)/C2=O 11F-406S CCOC(=O)CSc1c2ccccc2nc(n1)Cc3ccc(cc3)Cl 11F-408S CCOC(=O)C(C)Sc1c2ccccc2nc(n1)Cc3ccc(cc3)Cl 11F-409S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)SCc4ccc(cc4)Cl 11F-410S c1ccc2c(c1)c(nc(n2)Cc3cccc(c3)Cl)SCc4ccc(cc4Cl)Cl 11F-411S C#CCSc1c2ccccc2nc(n1)Cc3cccc(c3)Cl 11F-412S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)CCCCl)/C2=O 11F-413S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)CC(C)C)/C2=O 11F-414S CCCCC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3)C 11F-415S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)C(C)(C)CCl)/C2=O 11F-416S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)NCc4ccc(c(c4)Cl)Cl 11F-417S Cc1cc(n(n1)C)O 11F-418S Cc1c(c(n(n1)C)Cl)C=O 11F-419S Cc1c(c(n(n1)C)O)C(=O)Nc2ccccc2 11F-420S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)C(C)Cl)/C2=O 11F-423S Cc1ccc(cc1)CN2c3ccccc3/C(=N/OC(=O)CCCl)/C2=O 11F-424S C=CCNc1c2ccccc2nc(n1)Cc3ccc(cc3)Cl 11F-425S CCOC(=O)C(C)On1c2cc(ccc2nc1c3cccc(c3)Cl)[N+](=O)[O-] 11F-427S Cc1c(c(n(n1)C)Cl)C(=O)Nc2ccccc2 11F-428S C/N=C(\c1ccc(cc1[N+](=O)[O-])C(F)(F)F)/Nc2ccc(cc2)Cl 11F-429S Cc1c(c(n(n1)C)Oc2ccc(cc2)Cl)C=O 11F-431S Cc1c(c(n(n1)C)Oc2ccc(cc2)Cl)C(=O)O 11F-432S c1ccc2c(c1)/C(=N/OC(=O)CCl)/C(=O)N2Cc3ccc(cc3)Cl 11F-433S c1ccc2c(c1)/C(=N/OC(=O)CCCl)/C(=O)N2Cc3ccc(cc3)Cl 11F-434S CC(C(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3)Cl)Cl 11F-435S c1ccc2c(c1)/C(=N/OC(=O)CCCCl)/C(=O)N2Cc3ccc(cc3)Cl 11F-436S CC(C)CC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3)Cl 11F-437S c1ccc(cc1)CNc2c3ccccc3nc(n2)Cc4ccc(cc4)Cl 11F-438S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)NCc4ccc(cc4Cl)Cl 11F-439S Cc1c(c(n(n1)C)Sc2ccc(cc2)Cl)C(=O)Nc3ccccc3 11F-440S Cc1c(c(n(n1)C)Sc2cccc(c2)C(F)(F)F)C(=O)Nc3ccccc3 11F-441S Cc1c(c(n(n1)C)Oc2cccc(c2)C(F)(F)F)C=O 11F-442S Cc1c(c(n(n1)C)Oc2cccc(c2)Cl)C=O 11F-443S c1cc2c(cc1[N+](=O)[O-])C(=O)C(=O)N2Cc3ccc(cc3Cl)Cl 11F-446S CCCCC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3)Cl 11F-447S Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C#N 11F-448S c1cc(ccc1/C(=N\O)/N)NS(=O)(=O)c2ccc(cc2)Cl 11F-449S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)NCc4cccc(c4)C(F)(F)F 11F-450S c1ccc2c(c1)c(nc(n2)Cc3ccc(cc3)Cl)NCc4ccc(cc4)Cl 11F-451S c1cc(c(nc1)Cl)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 11F-901 c1cc(nnc1N2CCC(=O)CC2)Cl 11F-902 c1ccc(cc1)c2c[nH]c(c2C#N)N 11F-903 c1ccc(cc1)c2c[nH]c(c2C#N)/N=C/c3ccc(cc3)Cl 11F-904 c1cc(nnc1N2CCC(CC2)C(=O)N)Cl 11F-905 c1cc(nnc1N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 11F-906 C=CCOc1ccc2ccccc2c1C=O 11F-907 c1cc(c(nc1)Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)O 11F-908 C=CCOc1ccc2ccccc2c1/C=N/O 11F-909 c1ccc(cc1)c2cn(c(c2C#N)/N=C/c3ccc(cc3)Cl)Cc4ccc(cc4Cl)Cl 11F-910 c1ccc2c(c1)ccc3c2C4C(CO3)CON4 11F-911 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)Nc5ccc(cc5)Cl 11F-912 CCOC(=O)c1c(c[nH]c1NC(=O)Nc2ccc(cc2)Cl)c3ccc(cc3)Cl 11F-913 c1ccc(cc1)c2nc(cs2)c3ccccc3C(=O)O 11F-915 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)c5ccc(cc5)Cl 11F-916 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)N 11F-917 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)CCl 11F-918 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)CSc5ccc(cc5)Cl 11F-919 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)N4C5c6c7ccccc7ccc6OCC5CO4 11F-920 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)CON5C(=O)c6ccccc6C5=O 11F-921 c1ccc(cc1)c2cn(c(c2C#N)N)Cc3ccc(cc3Cl)Cl 11F-922 c1ccc2c(c1)C(=O)N(C2=O)OCC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 11F-924 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)CON)C(F)(F)F.Cl 11F-925 c1ccc(cc1)C(=O)NOCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 11F-926 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)CO/N=C/C3C(=O)CCCC3=O)C(F)(F)F 11F-927 CC(=O)Nc1ccc(cc1)S(=O)(=O)NOCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 11F-928 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)CONC(=O)N)C(F)(F)F 11F-929 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)Nc5cccc(c5)C(F)(F)F 11F-930 c1cc(ccc1C(/C=N\OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C#N)F 11F-931 CCOC(=O)c1ccccc1c2csc(n2)N(c3ccccc3)C(=O)Nc4cccc(c4)Cl 11F-932 c1ccc(cc1)Nc2nc(cs2)c3ccccc3C(=O)O 11F-934 COc1ccc(cc1)NC(=O)c2ccccc2c3csc(n3)c4ccccc4 11F-935 C=CC[n+]1ccccc1/C=N/O.[Br-] 11F-936 CCOC(=O)C1C(N(OC1(C(F)(F)F)O)C)c2ccc(cc2)OC 11F-937 CCOC(=O)C1C(N(OC1(C(F)(F)F)O)C)c2ccccc2 11F-939 c1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 11F-942 C=CCOc1ccc(cc1/C=N/O)Br 11F-943 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)CNC(=O)c5ccc(cc5)Cl 11F-944 c1c(cnc(c1Cl)N2CCN(CC2)C(=S)N)C(F)(F)F 11F-945 c1cc(ccc1c2csc(n2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 11F-946 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)N3CCCC3)C(F)(F)F 11F-947 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)N3CCOCC3)C(F)(F)F 11F-948 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 11F-949 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)N3CCCCC3)C(F)(F)F 11F-950 c1c(cnc(c1Cl)N2CCN(CC2)c3nc(cs3)CCl)C(F)(F)F 11F-952 CC(=O)CC(=O)Nc1ncccn1 11F-953 CC(=O)CC(=O)Nc1nccs1 11F-954 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)NCCO)C(F)(F)F 11F-955 CN(CCO)C(=O)C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 11F-957 CN1CCN(CC1)C(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 11F-958 Cc1ccc(cc1)S(=O)(=O)NC(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 11G-003 c1cc(c(nc1)Cl)C(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 11G-004 c1cc(cc(c1)S(=O)(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 11G-007 CSc1nc(nc(n1)N/C=N\O)Cn2cncn2 11G-008 CC(C)(C)C(=O)n1cc(cn1)c2c(cc(cn2)C(F)(F)F)Cl 11G-009 c1ccc(cc1)CSc2nc([nH]n2)N 11G-010 c1cc(c(cc1Cl)Cl)CSc2nc([nH]n2)N 11G-011 COc1cc(=O)n(nc1C(=N)OC)c2cccc(c2)C(F)(F)F 11G-014 CSc1cc(=O)n(nc1C(=N)SC)c2cccc(c2)C(F)(F)F 11G-015 COC(=O)CC(=O)/C(=N\Nc1ccccc1C(F)(F)F)/C(=O)OC 11G-016 c1cc(c(c(c1)F)C#N)C(C#N)c2ccc(cc2)F 11G-017 CC(C)(C)c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)O 11G-018 CCOC(=O)c1cnc2nc(nn2c1N)Sc3c(cc(cn3)C(F)(F)F)Cl 11G-019 COc1ccc(cc1)/C=C\c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 11G-020 c1cc(oc1)c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 11G-021 CN(C)/N=C/c1ccc(cc1)Cl 11G-022 c1ccc(cc1)S(=O)(=O)c2cc(ccc2O)O 11G-023 c1cc(cc(c1)Cl)n2c(=O)cc(c(n2)C(=O)N)O 11G-025 CC(C)(C)c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)O 11G-026 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 11G-030 CC(C)(C)c1ccc(cc1)n2c(=O)cc(c(n2)C#N)Cl 11G-031 COc1cccc(c1)N/N=C(\C(=O)CC(=O)OC)/C(=O)OC 11G-032 c1cc2c(c(c1)F)C(=C(C2(C#N)c3ccc(cc3)F)C#N)N 11G-033 c1cc(cc(c1)Cl)n2c(=O)cc(c(n2)C#N)Cl 11G-034 COC(=O)C1=C(c2c(cccc2F)C1(C#N)c3ccc(cc3)F)N 11G-035 c1ccc(cc1)CSc2nc3ncc(cn3n2)C#N 11G-036 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)/C(=N/OCc3ccc(cc3)Cl)/C 11G-037 c1cc(c(cc1Cl)Cl)CSc2nc3ncc(cn3n2)C#N 11G-039 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)c3ccn[nH]3 11G-042 COc1ccc(cc1)c2cn[nH]c2N 11G-044 Cn1cccc1C(C#N)c2cccc(c2C#N)F 11G-045 c1cc(cc(c1)C(F)(F)F)CSc2nc([nH]n2)N 11G-047 COc1ccc(cc1)c2cnn3c2ncc(c3)C#N 11G-049 c1cc(cc(c1)C(F)(F)F)CSc2nc3ncc(cn3n2)C#N 11G-050 C#CCSc1nc([nH]n1)N 11G-051 CC(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-301S CN1CCN(CC1)c2ccc(cc2)NC(=O)C(Cl)Cl 11G-302S CN1CCN(CC1)c2ccc(cc2)NC(=O)C(Cl)(Cl)Cl 11G-303S CN1CCN(CC1)c2ccc(cc2)NC(=O)c3cccc(c3)Cl 11G-304S CN1CCN(CC1)c2ccc(cc2)NC(=O)c3cccc(c3)C(F)(F)F 11G-305S CC(C(=O)OC)NS(=O)(=O)c1ccc(cc1)F 11G-306S CC(C(=O)OC)NS(=O)(=O)c1ccc(cc1)OC 11G-309S CN1CCN(CC1)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl 11G-310S CCCC(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-311S CC(C)C(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-312S c1cc(ccc1NC(=O)C(F)(F)F)N2CCOCC2 11G-314S c1cc(ccc1NC(=O)C(F)(F)F)N2CCCCC2 11G-316S CC(C)(C)C(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-317S CCCCC(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-318S CC(C)CC(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-319S c1csc(c1SCC#N)C(=O)O 11G-320S c1cc(ccc1CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)Cl)Cl 11G-322S c1ccc(c(c1)S(=O)(=O)NC(Cc2ccc(cc2)Cl)C(=O)O)Cl 11G-323S c1cc(ccc1CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)Br)Cl 11G-324S c1cc(cc(c1)S(=O)(=O)NC(Cc2ccc(cc2)Cl)C(=O)O)C(F)(F)F 11G-326S c1cc(ccc1NC(=O)c2c(ccs2)SCC#N)F 11G-328S CC(C(=O)Nc1ccc(cc1)N2CCN(CC2)C)Cl 11G-329S c1ccc(c(c1)N)N2CCOCC2 11G-330S CN1CCN(CC1)c2ccc(cc2)NC(=O)CCCl 11G-331S Cc1cccc(c1)C(=O)Nc2ccc(cc2)N3CCN(CC3)C 11G-332S c1ccc(cc1)S(=O)(=O)C(CCC(=O)c2ccc(cc2)F)C(=O)N 11G-333S Cc1ccc(cc1)S(=O)(=O)C(CCC(=O)c2ccc(cc2)Br)C(=O)N 11G-334S COc1ccc(cc1)OC(C(=O)Nc2ccc(cc2)Cl)(F)F 11G-336S COc1ccc(cc1)OC(C(=O)Nc2ccc(cc2F)F)(F)F 11G-337S COc1ccc(cc1)OC(C(=O)Nc2ccc(cc2)OC(F)(F)F)(F)F 11G-338S CN1CCN(CC1)c2ccc(cc2)NC(=O)C(c3ccccc3)Cl 11G-339S c1ccc(cc1)S(=O)(=O)NC(Cc2ccc(cc2)Cl)C(=O)O 11G-340S Cc1ccc(cc1)S(=O)(=O)NC(Cc2ccc(cc2)Cl)C(=O)O 11G-341S c1csc(c1SCC(=O)N)C(=O)O 11G-342S c1cc(c(cc1F)F)NC(=O)c2c(ccs2)SCC#N 11G-343S COc1ccc(cc1)NC(=O)c2c(ccs2)SCC#N 11G-345S CCC(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-346S Cc1ccc(cc1)C(=O)CCC(C(=O)N)S(=O)(=O)c2ccccc2 11G-347S c1ccc(cc1)S(=O)(=O)C(CCC(=O)c2ccc(cc2)Br)C(=O)N 11G-348S Cc1ccc(cc1)C(=O)CCC(C(=O)N)S(=O)(=O)c2ccc(cc2)Cl 11G-349S c1ccc(cc1)C(=O)CCC(C(=O)N)S(=O)(=O)c2ccc(cc2)Cl 11G-350S Cc1cccc(c1NC(=O)c2c(ccs2)SCC#N)C 11G-351S CC(C)(CCl)C(=O)Nc1ccc(cc1)N2CCN(CC2)C 11G-354S c1ccc(cc1)S(=O)(=O)C(CCC(=O)c2cccs2)C(=O)N 11G-355S CN1CCN(CC1)c2ccc(cc2)NC(=O)c3c(cccc3F)F 11G-356S CN1CCN(CC1)c2ccc(cc2)NC(=O)c3cccc(c3)OC 11G-358S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccccc2)C 11G-361S c1ccc(cc1)S(=O)(=O)C(CCC(=O)c2ccc(cc2)Cl)C(=O)N 11G-363S CC(=O)Nc1ccc(cc1)N2CCN(CC2)Cc3ccccc3 11G-364S c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)NC(=O)c4cccc(c4)C(F)(F)F 11G-365S c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)NC(=O)c4ccc(cc4)F 11G-369S c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)NC(=O)c4ccc(cc4Cl)Cl 11G-370S CC(C)(C)c1ccc(cc1)OC(C(=O)NC2CCCCC2)(F)F 11G-371S CC(C)(C)c1ccc(cc1)OC(C(=O)NCC2CC2)(F)F 11G-372S COC(=O)CSc1ccsc1C(=O)Nc2ccc(cc2)Cl 11G-374S COC(=O)CSc1ccsc1C(=O)Nc2ccc(cc2F)F 11G-375S c1ccc(cc1)C(CN2CCN(CC2)c3ccccc3)O 11G-406S c1ccc(cc1)C(CN2CCN(CC2)c3ccc(cc3)F)O 11G-407S c1ccc(cc1)C(CN2CCN(CC2)c3cccc(c3)Cl)O 11G-408S Cc1ccc(c(c1)N2CCN(CC2)CC(c3ccccc3)O)C 11G-409S c1ccc(cc1)C(CN2CCN(CC2)c3ccccc3F)O 11G-410S Cc1ccc(c(c1)C)N2CCN(CC2)CC(c3ccccc3)O 11G-411S COc1cccc(c1)N2CCN(CC2)CC(c3ccccc3)O 11G-412S c1ccc(cc1)N2CCN(CC2)CC(c3ccc(cc3)Cl)O 11G-413S c1cc(cc(c1)Cl)N2CCN(CC2)CC(c3ccc(cc3)Cl)O 11G-414S c1cc(ccc1C(CN2CCN(CC2)c3ccc(cc3)F)O)Cl 11G-415S c1ccc(c(c1)N2CCN(CC2)CC(c3ccc(cc3)Cl)O)F 11G-416S Cc1ccc(c(c1)N2CCN(CC2)CC(c3ccc(cc3)Cl)O)C 11G-417S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(c4ccc(cc4)Cl)O 11G-418S c1ccc(cc1)N2CCN(CC2)CC(c3ccc(cc3)F)O 11G-419S c1cc(cc(c1)Cl)N2CCN(CC2)CC(c3ccc(cc3)F)O 11G-420S c1cc(ccc1C(CN2CCN(CC2)c3ccc(cc3)F)O)F 11G-421S c1ccc(c(c1)N2CCN(CC2)CC(c3ccc(cc3)F)O)F 11G-422S c1ccc(cc1)N2CCN(CC2)CC(c3ccc(cc3)Br)O 11G-423S c1ccc(c(c1)N2CCN(CC2)CC(c3ccc(cc3)Br)O)F 11G-424S c1ccc(cc1)CN2CCN(CC2)CC(c3ccccc3)O 11G-425S c1cc(cc(c1)Cl)N2CCN(CC2)CC(c3ccc(cc3)Br)O 11G-426S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(c4ccc(cc4)Br)O 11G-427S Cc1ccc(c(c1)N2CCN(CC2)CC(c3ccc(cc3)Br)O)C 11G-428S c1ccc(c(c1)N2CCN(CC2)CC(c3ccc(cc3)C(F)(F)F)O)F 11G-429S c1cc(cc(c1)Cl)N2CCN(CC2)CC(c3ccc(cc3)C(F)(F)F)O 11G-430S COc1ccc(cc1)C(CN2CCN(CC2)c3ccccc3)O 11G-431S COc1ccc(cc1)C(CN2CCN(CC2)c3ccccc3F)O 11G-432S COc1ccc(cc1)C(CN2CCN(CC2)c3ccc(cc3)F)O 11G-433S COc1ccc(cc1)C(CN2CCN(CC2)c3cccc(c3)Cl)O 11G-434S c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)NC(=O)C(Cl)Cl 11G-436S c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)NC(=O)c4ccc(cc4)Cl 11G-437S CC(C)(C)C(=O)Nc1ccc(cc1)N2CCN(CC2)Cc3ccccc3 11G-438S CCCC(=O)Nc1ccc(cc1)N2CCN(CC2)Cc3ccccc3 11G-439S Cc1ccc(cc1Cl)NC(=O)C(Oc2ccc(cc2)OC)(F)F 11G-442S COc1ccc(cc1)OC(C(=O)Nc2ccccc2C(=O)OC)(F)F 11G-443S COc1ccc(cc1)OC(C(=O)Nc2c(cccc2Cl)Cl)(F)F 11G-444S Cc1c(cccc1Cl)NC(=O)C(Oc2ccc(cc2)OC)(F)F 11G-445S CCCCC(=O)Nc1ccc(cc1)N2CCN(CC2)Cc3ccccc3 11G-446S CC(C)CC(=O)Nc1ccc(cc1)N2CCN(CC2)Cc3ccccc3 11G-447S CC(=O)Nc1ccc(cc1)N2CCN(CC2)c3ccc(cc3)F 11G-448S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)N3CCN(CC3)c4ccc(cc4)F 11G-449S CCCCC(=O)Nc1ccc(cc1)N2CCN(CC2)c3ccc(cc3)F 11G-450S CC(C)C(=O)Nc1ccc(cc1)N2CCN(CC2)c3ccc(cc3)F 11G-451S c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)N3CCN(CC3)c4ccc(cc4)F)F 11G-452S c1ccc(cc1)Oc2ccc(c3c2nccc3)Cl 11G-453S CC(=O)Nc1ccccc1N2CCOCC2 11G-454S c1ccc(c(c1)NC(=O)CCl)N2CCOCC2 11G-455S c1ccc(c(c1)NC(=O)C(Cl)Cl)N2CCOCC2 11G-456S c1ccc(c(c1)NC(=O)C(Cl)(Cl)Cl)N2CCOCC2 11G-457S COC(=O)CS(=O)(=O)c1ccsc1C(=O)Nc2ccc(c(c2)F)F 11G-458S CC(C)(C)c1ccc(cc1)OC(C(=O)Nc2ccccc2C(=O)OC)(F)F 11G-459S CC(C)(C)c1ccc(cc1)OC(C(=O)Nc2ccc(cc2)Cl)(F)F 11G-460S CC(C)(C)c1ccc(cc1)OC(C(=O)NCC=C)(F)F 11G-461S CC(C)(C)c1ccc(cc1)OC(C(=O)N2CCOCC2)(F)F 11G-462S c1ccc(c(c1)NC(=O)c2ccc(cc2)F)N3CCOCC3 11G-465S c1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)N3CCOCC3 11G-466S c1cc(sc1)C(=O)CCC(C(=O)N)S(=O)(=O)c2ccc(c(c2)Cl)Cl 11G-467S c1ccc(cc1)NC(=O)c2c(snn2)Sc3ccc(cc3)Cl 11G-469S c1cc(cc(c1)NC(=O)c2c(snn2)Sc3ccc(cc3)Cl)C(F)(F)F 11G-470S c1cc(ccc1Sc2c(nns2)C(=O)Nc3ccc(c(c3)Cl)Cl)Cl 11G-471S CNC(=O)c1c(snn1)Sc2ccc(cc2)Cl 11G-472S CN(C)C(=O)c1c(snn1)Sc2ccc(cc2)Cl 11G-473S c1cc(ccc1Sc2c(nns2)C(=O)N3CCOCC3)Cl 11G-474S c1cc(ccc1Sc2c(nns2)C(=O)N3CCCCC3)Cl 11G-475S C=CCSc1ccsc1C(=O)O 11G-476S c1ccc(c(c1)C(=O)Nc2ccccc2N3CCOCC3)Cl 11G-477S c1ccc(c(c1)NC(=O)c2cccc(c2)Cl)N3CCOCC3 11G-478S CNC(=O)c1c(ccs1)SCc2ccc(cc2Cl)Cl 11G-479S c1ccc(cc1)C(CN2CCN(CC2)c3cccc(c3)C(F)(F)F)O 11G-480S c1cc(cc(c1)Cl)C(CN2CCN(CC2)c3cccc(c3)C(F)(F)F)O 11G-481S c1cc(cc(c1)N2CCN(CC2)CC(c3ccc(cc3)Cl)O)C(F)(F)F 11G-482S CCCCC(=O)Nc1ccccc1N2CCOCC2 11G-484S CC(C)(C)C(=O)Nc1ccccc1N2CCOCC2 11G-485S c1ccc(cc1)NC(=O)c2c(snn2)S(=O)(=O)c3ccc(cc3)Cl 11G-486S CC(C)C(=O)Nc1ccccc1N2CCOCC2 11G-487S c1ccc2c(c1)c(ccc2Cl)Oc3ccccc3[N+](=O)[O-] 11G-488S CCCNC(=O)c1c(snn1)Sc2ccc(cc2)Cl 11G-496S Cc1ccc(cc1)C(=O)ON(C)/C=C/C(=O)c2ccc(cc2)Br 11G-900 CN(/C=C/C(=O)c1ccc(cc1)Br)OC(=O)Nc2ccccc2Cl 11G-902 CN(/C=C/C(=O)c1ccc(cc1)Br)OC(=O)c2cccc(c2)C(F)(F)F 11G-904 c1ccc(cc1)NC(=O)N2CCOC23CCN(CC3)c4cccc(n4)F 11G-906 c1cc(nc(c1)F)N2CCC3(CC2)N(CCO3)C(=O)C4CC4 11G-908 c1ccc(cc1)C2C(CON2c3ccccc3)S(=O)(=O)c4ccccc4 11G-909 Cc1c(c(n(n1)c2ccccc2)Cl)C=O 11G-910 Cc1c(c(no1)c2ccccc2)C(=O)N3CCOC34CCN(CC4)c5cccc(n5)F 11G-913 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCOC34CCN(CC4)c5cccc(n5)F 11G-914 Cc1c2c(n(n1)c3ccccc3)OCC4C2N(OC4)C 11G-916 c1ccnc(c1)c2cc(nc(n2)c3ccccn3)O 11G-917 COC(=O)CC(=O)N1CCN(CC1)c2ccc(cc2)F 11G-918 c1cc(ccc1N2CCC3(CC2)N(CCO3)Cc4ccc(cc4Cl)Cl)[N+](=O)[O-] 11G-920 c1ccc(cc1)N2C(=O)C3CC(CN3C2=O)O 11G-921 c1cc(ccc1SC2CC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)Cl 11G-922 c1ccnc(c1)c2cc(nc(n2)c3ccccn3)Cl 11G-924 c1ccc(cc1)C2C3C(C(=O)N(C3=O)CCNc4c(cc(cn4)C(F)(F)F)Cl)ON2c5ccccc5 11G-925 Cn1c(c(c(n1)C(F)(F)F)C=O)OCC=C 11G-927 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)N3CCC4(CC3)OCCO4 11G-930 COc1ccc(cc1)N2CCN(CC2)C(=O)CC(=O)OC 11G-933 COC(=O)C1CC(CN1C(=O)N)O 11G-934 CC(=O)NCCn1cccc1 11G-936 Cc1c(c(n(n1)c2ccccc2)OCC=C)/C=N/O 11G-937 COc1ccc(cc1)CN2CCOC23CCN(CC3)c4ccc(cc4)[N+](=O)[O-] 11G-938 C/[N+](=C\CC(=O)c1ccc(cc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)/[O-] 11G-940 Cc1ccc(cc1)C(=O)ON(C)/C=C/C(=O)c2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 11G-941 c1cc(ccc1C(=O)NOCC(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 11G-943 c1c(cnc(c1Cl)NCC[NH3+])C(F)(F)F.[Cl-] 11G-944 c1ccc(cc1)CCN2CCC3=C(C2)CCc4c3cccc4.Cl 11G-945 c1c(cnc(c1Cl)NCCNC(=O)CO/N=C/C2=C(CCCC2=O)O)C(F)(F)F 11G-946 Cc1c(c(n(n1)c2ccccc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C=O 11G-947 c1cc(ccc1C(/C=N/OCC(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)C#N)Cl 11G-949 Cc1ccc(o1)C(=O)/C=C/N(C)C 11G-950 c1c(cnc(c1Cl)NCCNc2c[nH]c(=O)[nH]c2=O)C(F)(F)F 11G-951 CN(C)/C=C/C(=O)c1cccs1 11G-952 c1c(cnc(c1Cl)NCCNC(=O)CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 11G-953 COC(=O)CC(=O)N1CCN(CC1)c2ccc(c(c2)Cl)Cl 11G-954 CN(C)/C=C(\C(=O)N1CCN(CC1)c2ccc(c(c2)Cl)Cl)/C(=O)OC 11G-957 COC(=O)C1(C2C(C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)ON1)C(=O)OC 11G-958 CS(=O)(=O)NOCC(=O)NCCNc1c(cc(cn1)C(F)(F)F)Cl 11G-960 c1cc(c(cc1Cl)Cl)C(c2c(cc(cn2)C(F)(F)F)Cl)O 11H-001 Cc1c(c(=O)cco1)Oc2c(cc(cn2)C(F)(F)F)Cl 11H-002 Cc1c(c(=O)cc[nH]1)OCc2ccc(cc2)Cl 11H-003 c1cc(cc(c1)NC(=O)OC(c2ccc(cc2Cl)Cl)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 11H-004 c1ccc(cc1)S(=O)(=O)C(C2c3ccccc3CCN2C(=O)Nc4cccc(c4)C(F)(F)F)[N+](=O)[O-] 11H-005 Cc1c(c(=O)ccn1c2c(cc(cn2)C(F)(F)F)Cl)OCc3ccc(cc3)Cl 11H-006 CC(c1ccnc2n1ncc2C#N)Sc3c(cc(cn3)C(F)(F)F)Cl 11H-007 CC(c1ccnc2n1ncn2)Sc3c(cc(cn3)C(F)(F)F)Cl 11H-008 Cc1c(c(=O)cc[nH]1)Oc2c(cc(cn2)C(F)(F)F)Cl 11H-009 Cc1c(c(=O)cco1)OCC(=O)c2ccccc2 11H-010 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)n3cnc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 11H-013 c1cc(c(nc1)Sc2ncn(n2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] 11H-014 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)n3cnc(n3)Sc4ccc5c(cc(nc5n4)C(F)(F)F)C(F)(F)F 11H-016 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c3ccccc3c2=O)C#N 11H-018 Cc1c(c(=O)ccn1c2c(cc(cn2)C(F)(F)F)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 11H-019 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)Sc3nc[nH]n3 11H-022 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 11H-023 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)NCC=C 11H-024 COc1cccc(c1)c2c(c(nc(n2)c3ccccc3)O)C#N 11H-025 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)N3CCOCC3 11H-026 COC(=O)C1CC(=O)NN(C1)C(=O)Nc2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl 11H-028 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c3ccccc3c2=O)NC(=O)N4CCOCC4 11H-029 COc1cccc(c1)c2c(c(nc(n2)c3ccccc3)Cl)C#N 11H-030 CN1CCN(CC1)c2c(c(nc(n2)c3ccccc3)c4cccc(c4)OC)C#N 11H-031 Cc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)O)C#N 11H-032 CC(C(=O)C)n1cnc(n1)Sc2c(cccn2)[N+](=O)[O-] 11H-033 Cc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)Cl)C#N 11H-034 Cc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)N4CCN(CC4)C)C#N 11H-035 c1ccc(cc1)c2nc(c(c(n2)Cl)C#N)c3ccc(cc3)F 11H-036 CN1CCN(CC1)c2c(c(nc(n2)c3ccccc3)c4ccc(cc4)F)C#N 11H-037 c1ccc(cc1)c2nc(c(c(n2)O)C#N)c3ccc(cc3)F 11H-038 Cc1c(c(ccn1)Cl)Oc2c(cc(cn2)C(F)(F)F)Cl 11H-039 Cc1c(c(ccn1)N2CCOCC2)Oc3c(cc(cn3)C(F)(F)F)Cl 11H-040 Cc1c(c(ccn1)Sc2ccc(cc2)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 11H-041 c1ccc(cc1)C(=O)c2c(cc(cn2)C(F)(F)F)N3CCOCC3 11H-042 c1cc(ccc1/C(=N/Nc2c(cc(cn2)C(F)(F)F)Cl)/c3c(cc(cn3)C(F)(F)F)Cl)Cl 11H-043 c1cc(nc(c1)Cl)N/N=C(/c2ccc(cc2)Cl)\c3c(cc(cn3)C(F)(F)F)Cl 11H-046 c1cc(ccc1c2c3c(cc(cn3)C(F)(F)F)n(n2)c4c(cc(cn4)C(F)(F)F)Cl)Cl 11H-048 COc1ccccc1c2c(c(nc(n2)c3ccccc3)O)C#N 11H-049 COc1ccccc1c2c(c(nc(n2)c3ccccc3)Cl)C#N 11H-050 CC(c1[nH]c2ccccc2n1)O 11H-051 c1ccc(cc1)C(=O)CSc2ncc(c(n2)C(F)(F)F)C#N 11H-052 c1cc(nc(c1)Cl)n2c3cc(cnc3c(n2)c4ccc(cc4)Cl)C(F)(F)F 11H-053 CN1CCN(CC1)c2c(c(nc(n2)c3ccccc3)c4ccccc4OC)C#N 11H-054 Cc1c(c(=O)c(c[nH]1)Br)Oc2c(cc(cn2)C(F)(F)F)Cl 11H-057 c1ccc(cc1)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 11H-301S c1cc(ccc1NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-])F 11H-304S c1cc(ccc1C(CS(=O)(=O)c2ccc(cc2)Cl)(c3ccc(cc3)F)O)F 11H-306S c1cc(ccc1C(CS(=O)(=O)c2ccc(cc2)F)(c3ccc(cc3)F)O)F 11H-307S c1ccc(cc1)CS(=O)(=O)CC(c2ccc(cc2)F)(c3ccc(cc3)F)O 11H-308S c1cc(ccc1C(CSc2ccc(cc2)Cl)(c3ccc(cc3)F)O)F 11H-309S c1ccc(cc1)CSCC(c2ccc(cc2)F)(c3ccc(cc3)F)O 11H-310S c1cc(ccc1C(CSc2ccc(cc2)F)(c3ccc(cc3)F)O)F 11H-311S c1cc(ccc1CSCC(c2ccc(cc2)F)(c3ccc(cc3)F)O)Cl 11H-312S COc1ccc(cc1)SCC(c2ccc(cc2)F)(c3ccc(cc3)F)O 11H-313S c1cc(ccc1C(CS(=O)(=O)c2ccc(c(c2)Cl)Cl)(c3ccc(cc3)Cl)O)Cl 11H-314S COc1ccc(cc1)c2ccc(c(=O)[nH]2)C#N 11H-315S COc1cccc(c1)c2ccc(c(=O)[nH]2)C#N 11H-316S c1cc(ccc1C(CS(=O)(=O)c2ccc(cc2)Br)(c3ccc(cc3)Cl)O)Cl 11H-318S Cc1ccc(cc1)S(=O)(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 11H-319S CN(C)c1nc2cc(cc(c2c(=O)o1)Cl)Cl 11H-321S COC(=O)c1c(ccs1)Oc2ccc(cn2)[N+](=O)[O-] 11H-323S COC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])F 11H-324S c1cc(c(cc1F)[N+](=O)[O-])Oc2ccsc2C(=O)O 11H-325S COc1ccc(cc1)c2ccc(c(n2)OC(=O)c3c(cccc3Cl)Cl)C#N 11H-329S c1cc(ccc1C(CSc2ccc(cc2)F)(c3ccc(cc3)Cl)O)Cl 11H-330S c1cc(ccc1C(CSc2ccc(cc2)Br)(c3ccc(cc3)Cl)O)Cl 11H-331S COc1cccc(c1)c2ccc(c(n2)OC(=O)c3c(cccc3Cl)Cl)C#N 11H-332S c1cc(c(c(c1)Cl)C(=O)Oc2c(ccc(n2)c3ccc(cc3Cl)Cl)C#N)Cl 11H-333S c1cc(ccc1C(=O)Oc2c(ccc(n2)c3ccc(cc3Cl)Cl)C#N)F 11H-334S c1cc(c(c(c1)F)C(=O)Oc2c(ccc(n2)c3ccc(cc3Cl)Cl)C#N)F 11H-335S COc1cccc(c1)c2ccc(c(n2)OC(=O)c3ccc(cc3)Cl)C#N 11H-336S COc1cccc(c1)c2ccc(c(n2)OC(=O)c3cccc(c3)C(F)(F)F)C#N 11H-337S COc1cccc(c1)c2ccc(c(n2)OC(=O)c3ccc(cc3F)F)C#N 11H-339S Cc1cccc(c1)SCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 11H-340S c1cc(ccc1C(CS(=O)c2ccc(cc2)F)(c3ccc(cc3)Cl)O)Cl 11H-341S c1cc(ccc1C(CS(=O)c2ccc(cc2)Cl)(c3ccc(cc3)F)O)F 11H-343S c1cc(ccc1C(CSc2ccc(c(c2)Cl)Cl)(c3ccc(cc3)Cl)O)Cl 11H-344S c1cc(c(c(c1)Cl)SCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 11H-345S Cc1cccc(c1)S(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 11H-346S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2)Cl 11H-352S c1cc(ccc1C(CS(=O)c2ccc(cc2)Br)(c3ccc(cc3)Cl)O)Cl 11H-353S c1cc(ccc1C(CS(=O)c2ccc(c(c2)Cl)Cl)(c3ccc(cc3)Cl)O)Cl 11H-354S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2)F 11H-355S CC(=O)c1ccccc1NS(=O)(=O)c2cccc(c2)C(F)(F)F 11H-356S c1cc(c(c(c1)Cl)S(=O)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 11H-359S c1ccc(cc1)C(CS(=O)(=O)c2ccccc2)(c3ccccc3)O 11H-360S CC1CN(CC(O1)C)C(=O)CS(=O)(=O)c2ccc(cc2)F 11H-362S CC1CN(CC(O1)C)C(=O)CS(=O)(=O)c2ccc(cc2)OC 11H-363S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2)Br 11H-364S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2Cl)Cl 11H-365S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(c(c2)Cl)Cl 11H-366S CC(=O)c1ccccc1NS(=O)(=O)c2ccccc2Cl 11H-367S CC(=O)c1ccccc1NS(=O)(=O)c2cccc(c2Cl)Cl 11H-368S CC(=O)c1ccccc1NS(=O)(=O)c2cc(cc(c2)Cl)Cl 11H-369S Cc1ccc(cc1)SCC(c2ccccc2)(c3ccccc3)O 11H-370S COc1ccc(cc1)SCC(c2ccccc2)(c3ccccc3)O 11H-371S c1ccc(cc1)C(CSc2ccc(c(c2)Cl)Cl)(c3ccccc3)O 11H-372S COc1ccc(cc1)S(=O)CC(c2ccccc2)(c3ccccc3)O 11H-373S COC(=O)c1c(ccs1)Oc2ccc(c(c2)C(F)(F)F)[N+](=O)[O-] 11H-374S CN(c1ccccc1)C(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 11H-375S c1cc(cc(c1)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-])C(F)(F)F 11H-376S c1ccc(c(c1)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-])F 11H-377S c1cc(c(cc1[N+](=O)[O-])F)Oc2ccsc2C(=O)Nc3cc(cc(c3)Cl)Cl 11H-378S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2)OC 11H-380S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2)NC(=O)C 11H-381S CC(=O)c1ccccc1NS(=O)(=O)c2ccccc2[N+](=O)[O-] 11H-382S Cc1c(cccc1Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 11H-383S c1cc(ccc1C(F)(F)F)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 11H-384S C=CCNC(=O)c1c(ccs1)Oc2ccc(cc2F)[N+](=O)[O-] 11H-385S CCOC(CNC(=O)c1c(ccs1)Oc2ccc(cc2F)[N+](=O)[O-])OCC 11H-386S Cc1ccc(cc1)S(=O)CC(c2ccccc2)(c3ccccc3)O 11H-387S c1ccc(cc1)C(CS(=O)c2ccc(c(c2)Cl)Cl)(c3ccccc3)O 11H-388S CC(C)(C#C)NC(=O)c1c(ccs1)Oc2ccc(cc2F)[N+](=O)[O-] 11H-389S c1cc(c(cc1Oc2ccsc2C(=O)O)C(F)(F)F)[N+](=O)[O-] 11H-390S CC(=O)c1ccccc1NS(=O)(=O)C 11H-392S Cc1ccc(cc1)S(=O)(=O)CC(=O)N2CC(OC(C2)C)C 11H-394S CC1CN(CC(O1)C)C(=O)CS(=O)(=O)Cc2ccccc2 11H-395S CC1CN(CC(O1)C)C(=O)CS(=O)(=O)Cc2ccc(cc2)Cl 11H-396S CC(=O)c1ccccc1NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl 11H-397S c1ccc(cc1)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F 11H-399S c1ccc(c(c1)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F)F 11H-400S c1cc(cc(c1)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F)C(F)(F)F 11H-401S c1cc(ccc1NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F)Cl 11H-402S CN(c1ccccc1)C(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F 11H-403S c1cc(c(cc1F)F)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F 11H-404S c1cc(ccc1NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F)S(=O)(=O)N 11H-405S COc1ccc(c(c1)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F)OC 11H-406S CNC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])F 11H-407S CN(C)C(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])F 11H-408S C=CCNC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])F 11H-409S c1cc(c(cc1F)[N+](=O)[O-])Oc2ccsc2C(=O)N3CCOCC3 11H-410S c1ccc(cc1)Oc2c(ccc(n2)c3cccc(c3)C(F)(F)F)C#N 11H-507S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Oc3cccc(c3)C(F)(F)F)C#N 11H-508S c1cc(cc(c1)C(F)(F)F)c2ccc(c(n2)Oc3cccc(c3)Cl)C#N 11H-509S c1ccc2c(c1)c(=O)oc(n2)Nc3ccc(cc3)F 11H-525S c1ccc2c(c1)c(=O)oc(n2)Nc3ccccc3F 11H-534S c1ccc2c(c1)c(=O)oc(n2)Nc3cccc(c3)F 11H-535S c1ccc2c(c1)c(=O)oc(n2)Nc3ccccc3Cl 11H-536S c1ccc2c(c1)c(=O)oc(n2)Nc3cccc(c3)Cl 11H-537S c1ccc2c(c1)c(=O)oc(n2)Nc3cccc(c3)C(F)(F)F 11H-538 c1ccc2c(c1)c(=O)oc(n2)Nc3ccc(cc3F)F 11H-540S c1ccc2c(c1)c(=O)oc(n2)Nc3ccc(cc3)C(F)(F)F 11H-542S CN(C)/C=C(\C#N)/c1ccc(cc1)[N+](=O)[O-] 11H-545S c1cc(ccc1c2c3c(n[nH]2)CCCC3)Cl 11H-549S c1ccc2c(c1)C3=NC(CN3C(=O)N2)CN4CCN(CC4)c5cccc(c5)Cl 11H-550S c1ccc2c(c1)CC(C2N3CCOCC3)NC(=O)N4CCOCC4 11H-901 C/C(=C(/C#N)\C(=O)N)/N(C)C 11H-902 c1ccc2c(c1)C(=O)C=C(C2=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl 11H-903 c1cc(ccc1/C=N\NC(=O)C2=NOC3C2COC4(CCN(CC4)c5ccc(cc5)[N+](=O)[O-])OC3)Cl 11H-904 c1ccc2c(c1)c(c(n2c3c(cc(cn3)C(F)(F)F)Cl)CSc4cccc(c4)C(F)(F)F)Br 11H-905 CCOC(=O)C1=NOC2C1COC3(CCN(CC3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])OC2 11H-906 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)c4c[nH][nH]c4=O 11H-907 COC(=O)C(/C=N/OCc1ccc(cc1)[N+](=O)[O-])c2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl 11H-908 COc1ccc(cc1)N/C=C(/c2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl)\C(=O)OC 11H-909 C/C(=C(\C#N)/C(=O)N)/NCCNc1c(cc(cn1)C(F)(F)F)Cl 11H-910 C/C(=C(\C#N)/C(=O)N)/Nc1ccc(cc1)OC 11H-911 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)N 11H-913 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)CC#N 11H-915 CCOC(=O)C1=NOC2C1COC3(CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)OC2 11H-916 CCOC(=O)NC1Cc2ccccc2C1N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 11H-917 Cc1c(c(=O)ncn1CCNc2c(cc(cn2)C(F)(F)F)Cl)C#N 11H-918 CN(C)/C=C/c1c(c(=O)ncn1CCNc2c(cc(cn2)C(F)(F)F)Cl)C#N 11H-920 CCOC(=O)C1=NOC2C1COC3(CCN(CC3)c4ncccn4)OC2 11H-921 c1c(cnc(c1Cl)N2CCC3(CC2)OCC4C(CO3)ON=C4C(=O)NN)C(F)(F)F 11H-923 c1cnc(nc1)N2CCC3(CC2)OCC4C(CO3)ON=C4C(=O)NN 11H-924 c1c(cc(c(c1[N+](=O)[O-])N2CCC3(CC2)OCC4C(CO3)ON=C4C(=O)NN)[N+](=O)[O-])C(F)(F)F 11H-926 C/C(=C(\C#N)/C(=O)N)/Nc1ccc(cc1)Cl 11H-929 C/C(=C(\C#N)/C(=O)N)/NCc1ccncc1 11H-930 CCOC(=O)/C=C(\NC(=O)NC(C)(C)C)/N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 11H-931 C/C(=C(\C#N)/C(=O)N)/NN(C)c1c(cc(cn1)C(F)(F)F)Cl 11H-932 Cc1c(c(=O)ncn1N(C)c2c(cc(cn2)C(F)(F)F)Cl)C#N 11H-933 C/C(=C(/C#N)\C(=O)N)/Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 11H-934 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)N 11H-935 c1c(cnc(c1Cl)NCCNC(=O)N)C(F)(F)F 11H-936 c1c(cnc(c1Cl)NCCn2cc(c(=O)[nH]c2=O)C(=O)O)C(F)(F)F 11H-937 CC(=O)C1=NOC2C1COC(OC2)c3ccccc3F 11H-939 c1c(cnc(c1Cl)NCCN2C(=O)CC(=O)NC2=O)C(F)(F)F 11H-940 CN(C)/C=C\1/C(=O)NC(=O)N(C1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl 11H-941 c1cc(ccc1N/C=C/2\C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)OC(F)(F)F 11H-942 c1c(cnc(c1Cl)NCCNC=C(C#N)C#N)C(F)(F)F 11H-943 COC(=O)/C(=C(\C(=O)N)/Cl)/Cl 11H-944 CON/C=N/C(=O)C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 11H-945 CON/C=N\C(=O)Cc1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 11H-947 COC(=O)C1CCN(CC1)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 11H-948 COC(=O)C1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 11H-949 c1ccc(cc1)S(=O)(=O)CC2=C(CC(CC2=O)c3ccc(cc3)Cl)Sc4ccccn4 11H-950 c1cc(ccc1N2CCC(CC2)C(=O)O)[N+](=O)[O-] 11H-951 COC(=O)C1CCN(CC1)c2ncccn2 11H-952 c1c(cc(c(c1[N+](=O)[O-])N2CCC(CC2)C(=O)O)[N+](=O)[O-])C(F)(F)F 11H-953 c1cnc(nc1)N2CCC(CC2)C(=O)O 11H-955 C=CCNC(=O)C1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 11H-956 C=CCNC(=O)C1CCN(CC1)c2ncccn2 11H-958 CCOC(=O)C1=NOC(C1)CNC(=O)C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 11H-960 Cn1ccc(n1)c2ccc(cc2)Oc3cccc(c3C#N)Cl 11J-001 c1c(cnc(c1Cl)n2cnc(n2)N)C(F)(F)F 11J-002 C#CCNC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3cccs3 11J-003 Cc1c(cnc2n1ncc2C#N)C(=O)C 11J-004 CC(=O)c1cnc2c(cnn2c1/C=C/N(C)C)C#N 11J-005 c1ccc(c(c1)C(=O)c2ccc(s2)CC#N)F 11J-006 c1cc(oc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)O 11J-007 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)NN 11J-008 Cc1c(c(=O)cco1)OCc2c(cccc2Cl)Cl 11J-009 Cc1c(c(=O)cco1)OCc2c(cccc2Cl)F 11J-010 CNC(=S)NNC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3cccs3 11J-011 Cn1c(nnc1S)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 11J-012 c1cc(ccc1C(=O)c2ccc(s2)CC(=S)N)Cl 11J-013 c1ccc(cc1)C(=O)c2ccc(s2)CC#N 11J-014 Cn1c(nnc1SC)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 11J-015 c1cc(ccc1c2csc(n2)Cc3ccc(s3)C(=O)c4ccc(cc4)Cl)Cl 11J-016 c1cc(ccc1C(=O)c2ccc(s2)Cc3nc(cs3)c4ccc(c(c4)Cl)Cl)Cl 11J-017 c1cc(ccc1NC(=O)Nc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 11J-018 COC(=O)NC(=O)CCl 11J-019 c1ccc(cc1)C(=O)c2[nH]ccn2 11J-020 c1ccn(c1)c2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl 11J-022 c1cc(ccc1C(=O)Nc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 11J-023 CN(C)/C=N/c1ncn(n1)c2c(cc(cn2)C(F)(F)F)Cl 11J-028 Cc1c(c(=O)cc[nH]1)OCc2c(cccc2Cl)F 11J-029 Cc1c(c(=O)cco1)OCc2ccc(cc2Cl)Cl 11J-030 Cn1c(cc(n1)C(F)(F)F)Oc2c(cc(cn2)C(F)(F)F)Cl 11J-033 CC(C(=O)C)Oc1cc(nn1C)C(F)(F)F 11J-034 Cc1c(c(=O)cc[nH]1)OCc2c(cccc2Cl)Cl 11J-035 Cc1c2cnc3c(cnn3c2ccn1)C#N 11J-036 Cc1c(c(sc1C(=O)N/C=N/OC)C#N)c2ccccc2 11J-037 Cc1c(c(=O)ccn1Cc2ccc(cc2)F)OCc3c(cccc3Cl)F 11J-038 CN(C)/C=C\c1c2cnc3c(cnn3c2ccn1)C#N 11J-039 CC(C)(CNC(=O)c1ccccc1)SCc2ccc(cc2)Cl 11J-040 Cc1c(c(=O)ccn1c2c(cccn2)[N+](=O)[O-])OCc3c(cccc3Cl)F 11J-041 CO/N=C/CC(=O)Nc1ccc(cc1F)F 11J-043 COC(=O)c1c(onc1c2ccccc2)/C=C/c3cnc(c4c3onc4c5ccccc5)O 11J-044 Cc1ccc(cc1)Cn2ccc(=O)c(c2C)OCc3c(cccc3Cl)F 11J-045 Cc1c(c(=O)ccn1Cc2ccc(cc2)Cl)OCc3c(cccc3Cl)F 11J-046 Cc1c(c(=O)ccn1Cc2ccc(cc2)[N+](=O)[O-])OCc3c(cccc3Cl)F 11J-047 Cc1c(c(=O)ccn1Cc2ccc(cc2Cl)Cl)OCc3c(cccc3Cl)F 11J-048 Cc1c(c(=O)ccn1Cc2c(cccc2Cl)F)OCc3c(cccc3Cl)F 11J-049 Cc1c(c(=O)ccn1Cc2ccccc2)OCc3c(cccc3Cl)F 11J-050 c1c(cnc(c1Cl)n2cnc(n2)c3ncn(n3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 11J-053 CO/N=C/C(=C/c1ccc(cc1Cl)Cl)/C(=O)Nc2ccc(cc2F)F 11J-054 CC(C)(CNC(=O)CCl)SCc1ccc(cc1)Cl 11J-055 Cc1c(c(=O)ccn1c2c(cc(cn2)C(F)(F)F)Cl)OCc3c(cccc3Cl)F 11J-056 c1ccc(cc1)N/C=C\c2c3cnc4c(cnn4c3ccn2)C#N 11J-057 CO/N=C/Cc1c2cnc3c(cnn3c2ccn1)C#N 11J-058 Cc1c(c(=O)cco1)OCc2ccccc2 11J-059 c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)c3nc4ccc(cc4s3)Cl 11J-301S Cc1ccccc1Cn2c3cc(c(cc3nc2c4ccc(nc4)Cl)Cl)Cl 11J-302S c1ccc(c(c1)Cn2c3cc(c(cc3nc2c4ccc(nc4)Cl)Cl)Cl)Cl 11J-303S CNC(=O)c1ccc(cc1)Cl 11J-306S CC(C)c1ccc2c(c1)C(=O)C(=O)N2 11J-308S c1cc(c(nc1)Cl)c2nc3ccc(cc3s2)Cl 11J-309S c1cc(c(cc1Cl)Cl)Cn2c3cc(c(cc3nc2c4ccc(nc4)Cl)Cl)Cl 11J-310S c1cc(c(=O)[nH]c1)c2nc3cc(c(cc3s2)Cl)Cl 11J-311S Cn1c(nnn1)c2ccc(cc2)Cl 11J-313S c1cc(cc(c1)Cl)Cn2c(nnn2)c3ccc(cc3)Cl 11J-314S CCCn1c(nnn1)c2ccc(cc2)Cl 11J-318S CC(C)n1c(nnn1)c2ccc(cc2)Cl 11J-319S c1ccc(c(c1)c2nc(on2)c3ccc(nc3)Cl)Cl 11J-320S COc1c(cccn1)c2nc3ccc(cc3s2)Cl 11J-321S CN(C)c1c(cccn1)c2nc3ccc(cc3s2)Cl 11J-322S c1cc(cc(c1)C(F)(F)F)Cn2c(nnn2)c3ccc(cc3)Cl 11J-324S c1cc(c(nc1)Cl)c2nc3cc(c(cc3s2)Cl)Cl 11J-326S c1cc(c(cc1Cn2c3cc(c(cc3nc2c4ccc(nc4)Cl)Cl)Cl)Cl)Cl 11J-327S c1ccc(cc1)Cn2c3ccc(cc3nc2c4ccc[nH]c4=O)Cl 11J-329S c1ccc(cc1)Cn2c3ccc(cc3nc2c4cccnc4Cl)Cl 11J-330S C=CCn1c(nnn1)c2ccc(cc2)Cl 11J-333S c1ccc(cc1)Sc2c(cccn2)c3nc4ccc(cc4s3)Cl 11J-334S CN(C)c1c(cccn1)c2nc3cc(c(cc3s2)Cl)Cl 11J-335S CNC(=O)c1cccc(c1)C(F)(F)F 11J-336S CC(C)NC(=O)c1cccc(c1)C(F)(F)F 11J-337S c1cc(cc(c1)Cl)CNC(=O)c2cccc(c2)C(F)(F)F 11J-338S c1ccc(cc1)Cn2c3ccc(cc3nc2c4ccc(=O)[nH]c4)Cl 11J-339S CCCNC(=O)c1cccc(c1)C(F)(F)F 11J-340S C=CCNC(=O)c1cccc(c1)C(F)(F)F 11J-341S c1cc(cc(c1)Cl)Cn2c(nnn2)c3cccc(c3)Cl 11J-342S c1cc(cc(c1)C(F)(F)F)Cn2c(nnn2)c3cccc(c3)Cl 11J-343S c1ccc(cc1)Cn2c3ccc(cc3nc2c4ccc(nc4)Cl)Cl 11J-346S c1cc(cc(c1)Cl)Cn2c(nnn2)c3cccc(c3)C(F)(F)F 11J-347S CC(C)n1c(nnn1)c2cccc(c2)C(F)(F)F 11J-348S Cn1c2ccc(cc2nc1c3ccc[nH]c3=O)Cl 11J-351S CNC(=O)c1cc(cc(c1)Cl)Cl 11J-352S CC(C)NC(=O)c1cc(cc(c1)Cl)Cl 11J-353S Cn1c2ccc(cc2nc1c3cccnc3Cl)Cl 11J-354S c1cc(cc(c1)Cl)CNC(=O)c2cc(cc(c2)Cl)Cl 11J-355S CCCNC(=O)c1cc(cc(c1)Cl)Cl 11J-356S C=CCNC(=O)c1cc(cc(c1)Cl)Cl 11J-357S Cn1c(nnn1)c2cc(cc(c2)Cl)Cl 11J-358S Cn1c(nnn1)c2cccc(c2)Cl 11J-360S CC(C)n1c(nnn1)c2cccc(c2)Cl 11J-362S C=CCNC(=O)c1cccc(c1)Cl 11J-363S CCCn1c(nnn1)c2cccc(c2)Cl 11J-365S c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cc(cc(c2)Cl)Cl 11J-367S c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cccc(c2)C(F)(F)F 11J-368S CC(C)n1c(nnn1)c2cc(cc(c2)Cl)Cl 11J-369S c1cc(cc(c1)Cl)Cn2c(nnn2)c3cc(cc(c3)Cl)Cl 11J-370S c1cc(cc(c1)C(F)(F)F)Cn2c(nnn2)c3cccc(c3)C(F)(F)F 11J-371S C=CCn1c(nnn1)c2cc(cc(c2)Cl)Cl 11J-372S CCCn1c(nnn1)c2cc(cc(c2)Cl)Cl 11J-373S c1cc(cc(c1)C(F)(F)F)Cn2c(nnn2)c3cc(cc(c3)Cl)Cl 11J-374S c1ccc2c(c1)nc(n2Cc3ccc(cc3)Cl)c4ccc[nH]c4=O 11J-375S CC(C)C(=O)Nc1ccc(cc1)Cl 11J-376S C=CCn1c(nnn1)c2cccc(c2)Cl 11J-378S CCOC(=O)NC(=S)Nc1ccccn1 11J-380S CC(C)c1nnnn1c2ccc(cc2)Cl 11J-382S Cn1c2ccc(cc2nc1c3ccc(nc3)Cl)Cl 11J-383S Cc1ccc(cc1)C(=O)Nc2ccc([n+](c2)[O-])OC 11J-384S CC(C)C(=O)Nc1cc(cc(c1)Cl)Cl 11J-385S CCCC(=O)Nc1cc(cc(c1)Cl)Cl 11J-386S CSc1nc2ccccn2c(=O)n1 11J-389S c1ccc(cc1)CSc2nc3ccccn3c(=O)n2 11J-390S c1ccn2c(c1)nc(nc2=O)SCc3ccc(cc3)Cl 11J-391S COc1ccc(cc1)CSc2nc3ccccn3c(=O)n2 11J-392S Cn1c2ccc(cc2nc1c3ccc(=O)[nH]c3)Cl 11J-393S c1ccc2c(c1)nc(n2Cc3cccc(c3)Cl)c4ccc[nH]c4=O 11J-394S CCOC(=O)CSc1nc2ccccn2c(=O)n1 11J-396S c1ccn2c(c1)nc(nc2=O)SCc3cccc(c3)C(F)(F)F 11J-397S CC(C)(C)c1ccc(cc1)CSc2nc3ccccn3c(=O)n2 11J-398S C=CCSc1nc2ccccn2c(=O)n1 11J-400S COc1ccc(cc1)NCc2ccccc2 11J-507S Cc1ccc(cc1)c2nc(on2)c3ccc(nc3)Cl 11J-509S COc1cccc(c1)c2nc(on2)c3ccc(nc3)Cl 11J-510S Cc1cccc(c1)c2nc(on2)c3ccc(nc3)Cl 11J-513S c1cc(c(cc1c2nc(on2)c3ccc(nc3)Cl)Cl)Cl 11J-514S CC(=O)c1cc(cc(c1O)Br)Br 11J-517S Cc1c2cc(cc(c2oc1C(=O)c3ccccc3)Br)Br 11J-523S Cc1c2cc(cc(c2oc1C(=O)c3ccc(cc3)Cl)Br)Br 11J-525S Cc1c2cc(cc(c2oc1C(=O)c3ccc(c(c3)Cl)Cl)Br)Br 11J-529S c1ccc(cc1)c2ccc(c(=O)[nH]2)C(=O)O 11J-531S Cc1c2cc(ccc2oc1C(=O)c3ccccc3)Br 11J-533S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)Cl)Br 11J-534S Cc1c2ccccc2oc1C(=O)c3ccc(cc3)F 11J-536S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)F)Br 11J-537S Cc1c2cc(cc(c2oc1C(=O)c3ccc(cc3)F)Br)Br 11J-538S c1ccc(cc1)c2cccc(=O)n2Cc3ccc(cc3)Cl 11J-541S Cc1c2cc(ccc2oc1C(=O)c3ccc(c(c3)Cl)Cl)Br 11J-543S Cc1c2cc(ccc2oc1C(=O)c3ccc(c(c3)Cl)Cl)Cl 11J-544S Cc1c2cc(ccc2oc1C(=O)c3ccc(c(c3)Cl)Cl)[N+](=O)[O-] 11J-545S Cc1c2cc(ccc2oc1C(=O)c3ccccc3)Cl 11J-547S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)Cl)Cl 11J-548S Cc1c2ccc(cc2oc1C(=O)c3ccccc3)OC 11J-549S Cc1c2ccc(cc2oc1C(=O)c3ccc(cc3)Cl)OC 11J-550S COC(=O)c1c2n(c(c1C(=O)OC)c3ccccc3)CCC2 11J-555S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)F)CCC2 11J-556S Cc1ccc(cc1)c2c(c(c3n2CCC3)C(=O)OC)C(=O)OC 11J-557S Cc1c2ccc(cc2oc1C(=O)c3ccc(cc3)F)OC 11J-559S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(c(c3)Cl)Cl)CCC2 11J-560S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)Cl)CCC2 11J-561S COc1ccc(cc1)c2c(c(c3n2CCC3)C(=O)OC)C(=O)OC 11J-562S COC(=O)c1c2n(c(c1C(=O)OC)c3cccc(c3)C(F)(F)F)CCC2 11J-563S Cc1ccc(cc1)c2c(c(c3n2CCC3)C(=O)O)C(=O)O 11J-564S Cc1c2cc(ccc2oc1C(=O)c3ccccc3)[N+](=O)[O-] 11J-567S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 11J-568S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)F)[N+](=O)[O-] 11J-569S c1ccc(cc1)c2c(c(c3n2CCC3)C(=O)O)C(=O)O 11J-570S c1cc(cc(c1)Cl)c2c(c(c3n2CCC3)C(=O)O)C(=O)O 11J-572S c1cc(ccc1c2c(c(c3n2CCC3)C(=O)O)C(=O)O)Cl 11J-573S c1cc(ccc1c2c(c(c3n2CCC3)C(=O)O)C(=O)O)F 11J-574S COc1ccc(cc1)c2c(c(c3n2CCC3)C(=O)O)C(=O)O 11J-575S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)[N+](=O)[O-])[N+](=O)[O-] 11J-577S Cc1c2cc(ccc2oc1C(=O)c3ccccc3)OC 11J-578S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)Cl)OC 11J-579S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)F)OC 11J-581S c1ccc(c(c1)C(=O)NO)N 11J-582S c1ccc(cc1)c2cccc(=O)n2Cc3ccc(c(c3)Cl)Cl 11J-585S COC(=O)c1ccc(cc1)Cn2c(cccc2=O)c3ccccc3 11J-586S Cc1ccn2c(c1)nc(nc2=O)SCc3ccc(cc3)Cl 11J-590S Cc1ccn2c(c1)nc(nc2=O)SCc3ccc(cc3)OC 11J-591S CC(C)(C)c1ccc(cc1)Cn2c(cccc2=O)c3ccccc3 11J-593S COc1ccc(cc1)Cn2c(cccc2=O)c3ccccc3 11J-594S Cc1c(c(no1)C#N)C(=O)Nc2ccc(cc2)OC 11J-900 Cc1c(c(no1)C#N)C(=O)Nc2c(cc(cn2)C(F)(F)F)Cl 11J-901 Cc1cc(n(n1)C2CCS(=O)(=O)C2)c3c(nn(c3O)c4nc(cs4)c5c(ccs5)Cl)C 11J-902 CN(C)/C=C/C(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 11J-903 COc1ccc(cc1)NC(=O)c2cccnc2Cl 11J-904 COC(=O)C1CCN(CC1)c2c(cc([nH]2)c3c(ccs3)Cl)C#N 11J-905 COc1ccc(cc1)NC(=O)c2cccnc2OC 11J-906 c1ccc(cc1)c2nccc(n2)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-] 11J-907 c1cc(cnc1)c2nccc(n2)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-] 11J-908 Cc1c(c(no1)C#N)C(=O)Nc2ccccn2 11J-909 Cc1c(c(no1)C#N)C(=O)N(C)c2ccccc2 11J-910 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)CBr)Cl 11J-911 Cc1ccc(cc1)c2nccc(n2)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-] 11J-912 Cc1nccc(n1)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 11J-913 COC(=O)C1CCN(CC1)c2c(cc([nH]2)c3c(ccs3)Br)C#N 11J-914 c1ccc(cc1)C2C3C(CCCC3=O)ON2c4ccccc4 11J-915 CO/N=C/CC(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 11J-916 COC(=O)c1cc([nH]c1N2CCC(CC2)C(=O)OC)c3c(ccs3)Br 11J-918 COC(=O)c1cc([nH]c1N2CCC(CC2)C(=O)OC)c3c(ccs3)Cl 11J-919 c1csc(c1Cl)C(=O)C[N+]23CN4CN(C2)CN(C4)C3.[Br-] 11J-920 COc1ccc(cc1OC)/C=C/[N+](=O)[O-] 11J-921 c1ccc(cc1)N2Cc3ccsc3C=N2 11K-001 c1ccc2c(c1)-c3c(cc(nn3)c4ccc(cc4)O)C2=O 11K-002 c1ccc2c(c1)-c3c(cc(nn3)c4ccncc4)C2=O 11K-003 c1ccc2c(c1)-c3c(cc(nn3)c4cccnc4)C2=O 11K-004 c1cc(ccc1N2Cc3ccsc3C=N2)F 11K-005 c1ccc2c(c1)-c3c(cc(nn3)c4ccc(cc4)Br)C2=O 11K-006 c1ccc2c(c1)-c3c(cc(nn3)c4ccccc4F)C2=O 11K-007 c1ccc2c(c1)-c3c(cc(nn3)c4ccc(cc4Cl)Cl)C2=O 11K-008 COc1ccc(cc1)/N=c\2/c(nss2)Cl 11K-010 c1cc(ccc1/N=c\2/c(nss2)Cl)Cl 11K-011 Cc1ccc(cc1)c2cc3c(nn2)-c4ccccc4C3=O 11K-012 c1ccc2c(c1)-c3c(cc(nn3)c4cccc(c4)Cl)C2=O 11K-013 c1ccc2c(c1)-c3c(cc(nn3)c4ccc(c(c4)Cl)Cl)C2=O 11K-014 c1cc(ccc1c2ccnc3n2nc(n3)N)Cl 11K-015 COC(=O)c1ccc(cc1)/N=c\2/c(nss2)Cl 11K-016 COc1ccc(cc1)c2ccnc3n2nc(n3)N 11K-017 Cc1cc(ccc1/N=c\2/c(nss2)Cl)Cl 11K-019 c1ccc(cc1)c2ccnc3n2nc(n3)N 11K-020 c1ccc(cc1)Oc2ccc(cc2)c3ccnc4n3nc(n4)N 11K-021 c1cnccc1c2ccnc3n2nc(n3)N 11K-022 c1cc(cc(c1)Cl)c2ccnc3n2nc(n3)N 11K-023 c1ccnc(c1)c2ccnc3n2nc(n3)N 11K-024 c1cc(ccc1c2cnc3nc(nn3c2N)N)Cl 11K-025 c1cscc1c2cnc3nc(nn3c2N)N 11K-026 COc1ccc(cc1)c2cnc3nc(nn3c2N)N 11K-027 CC(=O)CCS(=O)(=O)c1ccccc1 11K-028 c1cc(ccc1/C=C\c2ccnc3n2nc(n3)N)Cl 11K-029 COc1ccc(cc1)/C=C\c2ccnc3n2nc(n3)N 11K-030 Cc1ccc(o1)c2ccnc3n2nc(n3)N 11K-031 CN(C)/C=N/c1nc2nccc(n2n1)c3ccc(cc3)Cl 11K-032 CN(C)/C=N/c1nc2nccc(n2n1)c3ccncc3 11K-033 CN(C)/C=N/c1nc2nccc(n2n1)c3ccc(cc3)OC 11K-034 CN(C)/C=N/c1nc2nccc(n2n1)c3ccccc3 11K-035 COC(=O)c1c(ccs1)/N=c\2/c(nss2)Cl 11K-036 c1cc(c(cc1F)F)/N=c\2/c(nss2)Cl 11K-037 CN(C)/C=N\c1nc2nccc(n2n1)c3ccc(cc3)Oc4ccccc4 11K-038 CN(C)/C=N/c1nc2nccc(n2n1)c3cccc(c3)Cl 11K-039 CN(C)/C=N/c1nc2nccc(n2n1)/C=C\c3ccc(cc3)OC 11K-040 CO/N=C/Nc1nc2nccc(n2n1)c3ccc(cc3)Cl 11K-041 Cc1ccc(o1)c2ccnc3n2nc(n3)/N=C/N(C)C 11K-042 CO/N=C/Nc1nc2nccc(n2n1)c3ccncc3 11K-043 COc1ccc(cc1)c2ccnc3n2nc(n3)N/C=N/OC 11K-044 CN(C)/C=N/c1nc2nccc(n2n1)/C=C\c3ccc(cc3)Cl 11K-045 c1cc(ccc1/N=c\2/c(nss2)Cl)Br 11K-046 CN(C)/C=N/c1c(cnc2n1nc(n2)/N=C/N(C)C)c3ccsc3 11K-047 CN(C)/C=N/c1c(cnc2n1nc(n2)/N=C/N(C)C)c3ccc(cc3)Cl 11K-048 COC(=O)c1cccc(c1)/N=c\2/c(nss2)Cl 11K-049 CN(C)/C=N/c1c(cnc2n1nc(n2)/N=C/N(C)C)c3cccs3 11K-050 CN(C)/C=N/c1nc2nccc(n2n1)c3ccco3 11K-051 CN(C)/C=N/c1c(cnc2n1nc(n2)/N=C/N(C)C)c3ccc(cc3)OC 11K-052 CN(C)/C=N/c1nc2nccc(n2n1)c3cccnc3 11K-053 CN(C)/C=N/c1nc2nccc(n2n1)c3cccs3 11K-054 c1cc(c(cc1[N+](=O)[O-])Cl)/N=c\2/c(nss2)Cl 11K-055 CN(C)/C=N/c1nc2nccc(n2n1)c3ccccn3 11K-056 CO/N=C/Nc1nc2nccc(n2n1)/C=C\c3ccc(cc3)Cl 11K-057 c1c(cc(cc1Cl)Cl)/N=c/2\c(nss2)Cl 11K-058 Cc1ccc(cc1)/N=c\2/c(nss2)Cl 11K-059 CO/N=C/Nc1nc2nccc(n2n1)c3cccnc3 11K-060 CO/N=C/Nc1nc2nccc(n2n1)c3ccc(cc3)Oc4ccccc4 11K-061 c1cc(ccc1C#N)/N=c\2/c(nss2)Cl 11K-062 COc1ccc(cc1)/C=C\c2ccnc3n2nc(n3)N/C=N/OC 11K-063 c1cc(c(cc1Cl)Cl)/N=c\2/c(nss2)Cl 11K-064 Cc1ccc(o1)c2ccnc3n2nc(n3)N/C=N/OC 11K-065 c1cc(ccc1/N=c/2\c(nss2)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 11K-066 CO/N=C/Nc1nc2nccc(n2n1)c3ccco3 11K-067 CO/N=C/Nc1nc2nccc(n2n1)c3cccs3 11K-068 CO/N=C/Nc1nc2nccc(n2n1)c3cccc(c3)Cl 11K-069 CO/N=C/Nc1nc2nccc(n2n1)c3ccccn3 11K-070 c1ccn(c1)c2nc3nccc(n3n2)c4cccc(c4)Cl 11K-071 c1ccc(cc1)Oc2ccc(cc2)c3ccnc4n3nc(n4)n5cccc5 11K-072 c1cc(cc(c1)/N=c\2/c(nss2)Cl)C#N 11K-073 COc1ccc(cc1)/C=C/c2ccnc3n2nc(n3)n4cccc4 11K-074 COc1ccc(cc1)c2ccnc3n2nc(n3)n4cccc4 11K-075 c1ccn(c1)c2nc3nccc(n3n2)c4ccc(cc4)Cl 11K-076 c1ccn(c1)c2nc3nccc(n3n2)c4ccncc4 11K-077 c1ccn(c1)c2nc3nccc(n3n2)/C=C/c4ccc(cc4)Cl 11K-078 c1ccc(cc1)c2ccnc3n2nc(n3)n4cccc4 11K-079 CC(c1ccnc2n1nc(n2)n3cccc3)Oc4ccsc4C(=O)OC 11K-081 Cc1ccc(o1)c2ccnc3n2nc(n3)n4cccc4 11K-082 c1ccn(c1)c2nc3nccc(n3n2)c4ccco4 11K-083 C/C(=N/OC)/CCS(=O)(=O)c1ccccc1 11K-084 c1ccnc(c1)c2ccnc3n2nc(n3)n4cccc4 11K-085 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3ccc(cc3)F 11K-086 CC(c1ccnc2n1nc(n2)n3cccc3)Oc4ccc(cc4)F 11K-087 CC(c1ccnc2n1nc(n2)N/C=N/OC)Oc3ccc(cc3)F 11K-088 C/C(=N/O)/CCS(=O)(=O)c1ccccc1 11K-089 Cc1c(cc(c(n1)Cl)C#N)C(=O)OC 11K-301S CCSc1c(cc(c(n1)C)C(=O)C)C#N 11K-303S CCCSc1c(cc(c(n1)C)C(=O)C)C#N 11K-304S Cc1c(cc(c(n1)SC(C)C)O)C(=O)C 11K-305S C/C=C/CSc1c(cc(c(n1)C)C(=O)C)C#N 11K-306S Cc1c(cc(c(n1)SCC#C)C#N)C(=O)C 11K-307S Cc1c(cc(c(n1)SCC(C)C)C#N)C(=O)C 11K-308S Cc1c(cc(c(n1)OC)C#N)C(=O)OC 11K-309S Cc1c(cc(c(n1)Oc2ccc(cc2)F)C#N)C(=O)OC 11K-310S Cc1c(cc(c(n1)Sc2ccc(cc2)OC)C#N)C(=O)OC 11K-311S Cc1c(cc(c(n1)Oc2ccc(cc2)OC)C#N)C(=O)OC 11K-313S Cc1c(cc(c(n1)OC(C)C)C#N)C(=O)OC 11K-314S CCCn1c(c(cc(c1=O)C#N)C(=O)C)C 11K-315S Cc1c(cc(c(n1)Oc2ccccc2)C#N)C(=O)OC 11K-319S Cc1c(cc(c(n1)Oc2cccc(c2)C(F)(F)F)C#N)C(=O)OC 11K-320S Cc1ccc(cc1)/C=C/c2ccc(=O)n(n2)CC=C 11K-321S CCOC(=O)Cn1c(=O)ccc(n1)/C=C/c2ccc(cc2)C 11K-322S Cn1c(=O)ccc(n1)/C=C/c2ccc(cc2)OC 11K-323S COc1ccc(cc1)/C=C/c2ccc(=O)n(n2)CC=C 11K-324S Cc1c(cc(c(n1)Oc2ccccc2OC)C#N)C(=O)OC 11K-325S Cc1c(cc(c(n1)Oc2ccc(cc2Cl)Cl)C#N)C(=O)OC 11K-326S Cc1c(cc(c(n1)Sc2ccccc2)C#N)C(=O)OC 11K-327S Cc1c(cc(c(n1)Sc2ccc(cc2)Cl)C#N)C(=O)OC 11K-328S Cc1c(cc(c(n1)Sc2ccccc2Cl)C#N)C(=O)OC 11K-329S Cc1c(cc(c(n1)SCc2ccccc2)C#N)C(=O)OC 11K-330S Cc1c(cc(c(=O)n1C)C#N)C(=O)OC 11K-334S Cc1cccc(c1C)Oc2c(cc(c(n2)C)C(=O)OC)C#N 11K-336S Cc1c(cc(c(n1)Oc2ccccc2)C#N)C(=O)C 11K-338S Cc1c(cc(c(n1)Sc2ccccc2)C#N)C(=O)C 11K-339S c1cc(ccc1NC(=O)C(F)(F)F)Cl 11K-343S Cc1c(cc(c(n1)Oc2cc(c(cc2Cl)Cl)Cl)C#N)C(=O)OC 11K-345S CCOc1ccc(cc1)/C=C/C(=O)CCC(=O)O 11K-347S CCOc1ccc(cc1)/C=C/C2=NNC(=O)CC2 11K-348S COc1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccccc3 11K-349S CCOC(=O)C(C(=O)c1ccccc1)C(=O)OCC 11K-351S COc1ccc(cc1)Oc2c(nccn2)C#N 11K-352S CCOC(=O)Cn1c(=O)ccc(n1)/C=C/c2ccc(cc2)OC 11K-353S CCOC(=O)C(C)n1c(=O)ccc(n1)/C=C/c2ccc(cc2)OC 11K-354S COc1ccc(cc1)CN(c2ccc(cc2)Cl)C(=O)C(F)(F)F 11K-355S CCOC(=O)C(C)N1C(=O)CCC(=N1)/C=C/c2ccc(cc2)OC 11K-358S Cc1c(cc(c(n1)N(C)C)C#N)C(=O)OC 11K-359S CC(C)c1ccc(cc1)/C=C/C(=O)CCC(=O)O 11K-363S CC(C)c1ccc(cc1)/C=C/C2=NNC(=O)CC2 11K-364S CCOc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccccc3 11K-365S CCOc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)CC(=O)OCC 11K-366S Cc1c(cc(c(n1)Oc2cccc(c2)C(F)(F)F)C#N)C(=O)C 11K-367S Cc1c(cc(c(n1)Oc2ccc(cc2Cl)Cl)C#N)C(=O)C 11K-368S Cc1c(cc(c(n1)Sc2ccc(cc2)Cl)C#N)C(=O)C 11K-369S Cc1c(cc(c(n1)Sc2ccccc2Cl)C#N)C(=O)C 11K-370S c1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3cccc(c3)C(F)(F)F 11K-371S Cc1ccccc1CN2C(=O)CCC(=N2)/C=C/c3ccccc3 11K-372S Cc1c(cc(c(n1)Oc2ccc(cc2)F)C#N)C(=O)C 11K-373S Cc1c(cc(c(n1)Oc2ccccc2OC)C#N)C(=O)C 11K-374S Cc1cc(cc(c1)Oc2c(cc(c(n2)C)C(=O)C)C#N)C 11K-375S CCOC(=O)c1cc(c(=O)[nH]c1c2ccccc2)C#N 11K-377S CCOC(=O)c1cc(c(=S)[nH]c1c2ccccc2)C#N 11K-378S c1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccccc3Cl 11K-379S CC(C)(C)c1ccc(cc1)CN2C(=O)CCC(=N2)/C=C/c3ccccc3 11K-380S c1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccc(c(c3)Cl)Cl 11K-381S c1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccc(cc3)F 11K-382S Cc1c(cc(c(n1)N2CCCC2)C#N)C(=O)OC 11K-383S Cc1c(cc(c(n1)NC)C#N)C(=O)C 11K-384S c1cc(ccc1Sc2c(nccn2)C#N)Cl 11K-386S c1ccc(c(c1)Sc2c(nccn2)C#N)Cl 11K-387S c1cc(cc(c1)Sc2c(nccn2)C#N)C(F)(F)F 11K-388S COc1ccc(cc1)Sc2c(nccn2)C#N 11K-389S Cc1ccc(cc1)Sc2c(nccn2)C#N 11K-390S Cc1c(cc(c(n1)NCc2ccccc2)C#N)C(=O)C 11K-391S c1cc(ccc1F)Sc2c(nccn2)C#N 11K-392S COC(=O)c1ccccc1Sc2c(nccn2)C#N 11K-394S c1cc(ccc1Oc2c(nccn2)C#N)Cl 11K-395S c1cc(cc(c1)Oc2c(nccn2)C#N)C(F)(F)F 11K-396S c1ccc(cc1)Oc2c(nccn2)C#N 11K-397S CCOC(=O)CN1C(=O)CCC(=N1)/C=C/c2ccc(cc2)C(C)C 11K-398S CC(C)c1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3cccc(c3)C(F)(F)F 11K-399S Cc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccccc3Cl 11K-400S Cc1ccc(cc1)/C=C/C2=NN(C(=O)CC2)Cc3ccc(c(c3)Cl)Cl 11K-401S CC(C)c1ccc(cc1)/C=C/c2ccc(nn2)O 11K-402S Cc1c(cc(c(n1)NCc2ccccc2)C#N)C(=O)OC 11K-403S Cc1c(cc(c(n1)NCC=C)C#N)C(=O)OC 11K-404S CCCNc1c(cc(c(n1)C)C(=O)OC)C#N 11K-405S Cc1c(cc(c(n1)NCC=C)C#N)C(=O)C 11K-406S c1cc(c(cc1F)F)Oc2c(nccn2)C#N 11K-407S c1ccc(c(c1)Oc2c(nccn2)C#N)Cl 11K-408S c1cc(c(cc1Cl)Cl)Oc2c(nccn2)C#N 11K-409S CCOC(=O)c1cc(c(nc1c2ccccc2)Cl)C#N 11K-410S c1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccc(cc3)F 11K-411S CCN(CC)c1c(cc(c(n1)C)C(=O)C)C#N 11K-412S Cc1c(cc(c(n1)N2CCOCC2)C#N)C(=O)C 11K-413S Cc1c(cc(c(n1)N2CCCCC2)C#N)C(=O)C 11K-414S CC(C)c1ccc(cc1)/C=C/c2ccc(=O)n(n2)C 11K-415S CCOC(=O)Cn1c(=O)ccc(n1)/C=C/c2ccc(cc2)C(C)C 11K-416S Cc1c(cc(c(n1)N2CCCC2)C#N)C(=O)C 11K-417S CCCNc1c(cc(c(n1)C)C(=O)C)C#N 11K-418S Cc1c(cc(c(n1)N2CCN(CC2)C)C#N)C(=O)C 11K-419S Cc1ccc(cc1)Sc2ccc(cc2NC(=O)c3cccc(c3)C(F)(F)F)C#N 11K-504S Cc1ccc(cc1)Sc2ccc(cc2NC(=O)c3ccc(cc3Cl)Cl)C#N 11K-505S Cc1ccc(cc1)Sc2ccc(cc2NC(=O)c3ccc(cc3)Cl)C#N 11K-506S c1ccc(cc1)Oc2cc(nc(n2)c3ccncc3)CS(=O)(=O)c4ccccc4 11K-507S CCOC(=O)CSc1cc(nc(n1)c2ccncc2)CS(=O)(=O)c3ccccc3 11K-508S c1ccc(cc1)Oc2cc(nc(n2)c3ccccn3)CS(=O)(=O)c4ccccc4 11K-509S c1ccc(cc1)Sc2cc(nc(n2)c3ccccn3)CS(=O)(=O)c4ccccc4 11K-511S COc1cc(nc(n1)c2ccccn2)CS(=O)(=O)c3ccccc3 11K-512S c1ccc(cc1)c2nc(cc(n2)Sc3ccccc3)CSc4ccc(cc4)Cl 11K-513S c1ccc(cc1)c2nc(cc(n2)Oc3ccc(cc3)Cl)CSc4ccc(cc4)Cl 11K-514S Cc1ccc(cc1)Sc2ccc(cc2NC(=O)c3ccccc3C)C#N 11K-515S Cc1ccc(cc1)Sc2ccc(cc2NC(=O)c3cc(c(c(c3)OC)OC)OC)C#N 11K-516S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)CSc4ccccc4 11K-518S CCOC(=O)CSc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 11K-519S CCOC(=O)C(C)Sc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 11K-520S COc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 11K-521S CSc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 11K-522S CSc1ccc(cc1NC(=O)c2ccc(cc2Cl)Cl)C#N 11K-523S CSc1ccc(cc1NC(=O)c2ccc(cc2)Cl)C#N 11K-524S Cc1ccc(cc1)Sc2ccc(cc2NC(=O)C3CC3)C#N 11K-525S Cc1ccc(cc1)Sc2ccc(cc2NC(=O)c3ccc(cc3)F)C#N 11K-526S CSc1ccc(cc1NC(=O)c2ccc(c(c2)Cl)Cl)C#N 11K-527S CSc1ccc(cc1NC(=O)c2cccc(c2Cl)Cl)C#N 11K-528S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C#N)Cl 11K-529S CSc1ccc(cc1NC(=O)c2cccnc2Cl)C#N 11K-530S CSc1ccc(cc1NC(=O)c2ccc(nc2)Cl)C#N 11K-531S Cc1ccccc1C(=O)Nc2cc(ccc2SC)C#N 11K-532S COc1ccc(cc1)C(=O)Nc2cc(ccc2SC)C#N 11K-533S c1cc(ccc1Sc2ccc(cc2N)C#N)Cl 11K-534S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3cccnc3)Cl 11K-536S COc1cccc(c1)C(=O)Nc2cc(ccc2Sc3ccc(cc3)Cl)C#N 11K-537S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc(ccc2Sc3ccc(cc3)Cl)C#N 11K-538S c1ccc(c(c1)C(=O)Nc2cc(ccc2Sc3ccc(cc3)Cl)C#N)Cl 11K-539S Cc1cccc(c1)C(=O)Nc2cc(ccc2Sc3ccc(cc3)Cl)C#N 11K-540S c1ccc(cc1)Sc2cc(nc(n2)c3cccnc3)CS(=O)(=O)c4ccccc4 11K-541S c1ccc(cc1)SCc2cc(nc(n2)c3cccnc3)O 11K-546S c1cc(ccc1Sc2ccc(cc2NC(=O)c3ccc(nc3)Cl)C#N)Cl 11K-548S c1cc(c(c(c1)Cl)Sc2ccc(cc2N)C#N)Cl 11K-550S CSc1cc(nc(n1)c2ccccn2)CSc3ccc(cc3)Cl 11K-554S c1ccc(cc1)c2nc(cc(n2)Cl)CS(=O)(=O)c3ccccc3 11K-555S c1cc(c(c(c1)Cl)Sc2ccc(cc2NC(=O)c3ccc(cc3)Cl)C#N)Cl 11K-558S c1ccc(cc1)c2nc(cc(n2)Sc3ccccc3)CS(=O)(=O)c4ccccc4 11K-559S c1ccc(cc1)c2nc(cc(n2)Oc3ccccc3)CS(=O)(=O)c4ccccc4 11K-560S CCOC(=O)CSc1cc(nc(n1)c2ccccc2)CS(=O)(=O)c3ccccc3 11K-561S COc1cc(nc(n1)c2ccccc2)CS(=O)(=O)c3ccccc3 11K-562S CSc1cc(nc(n1)c2ccccc2)CS(=O)(=O)c3ccccc3 11K-563S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3)Cl)CS(=O)(=O)c4ccccc4 11K-564S CSc1ccc(cc1NC(=O)c2ccccc2)C#N 11K-565S CSc1ccc(cc1NC(=O)c2cccc(c2)Cl)C#N 11K-566S CSc1ccc(cc1NC(=O)C2CC2)C#N 11K-568S CCOC(=O)C(C)Sc1cc(nc(n1)c2ccccc2)CS(=O)(=O)c3ccccc3 11K-572S c1ccc(cc1)Sc2cc(nc(n2)c3cccnc3)CS(=O)c4ccccc4 11K-573S CCOC(=O)CSc1cc(nc(n1)c2cccnc2)CS(=O)c3ccccc3 11K-574S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc(ccc2Sc3c(cccc3Cl)Cl)C#N 11K-576S c1ccc(c(c1)C(=O)Nc2cc(ccc2Sc3c(cccc3Cl)Cl)C#N)Cl 11K-577S Cc1ccccc1C(=O)Nc2cc(ccc2Sc3c(cccc3Cl)Cl)C#N 11K-580S c1cc(cc(c1)Cl)C(=O)Nc2cc(ccc2Sc3c(cccc3Cl)Cl)C#N 11K-581S CSC(=CC(=O)c1ccccc1)SC 11K-591S CSc1cc([nH]c(=O)c1C#N)c2ccccc2 11K-592S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3ccccn3)N4CCOCC4 11K-593S c1ccc(cc1)CNc2cc(nc(n2)c3ccccn3)CS(=O)(=O)c4ccccc4 11K-594S c1ccc(cc1)N2CCN(CC2)c3cc(nc(n3)c4ccccn4)CS(=O)(=O)c5ccccc5 11K-595S c1ccc(cc1)CNc2cc(nc(n2)c3cccnc3)CSc4ccc(cc4)Cl 11K-596S CN(C)c1cc(nc(n1)c2cccnc2)CSc3ccccc3 11K-598S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3ccncc3)N4CCCCC4 11K-599S c1ccc(cc1)Sc2ccc(cc2C#N)N 11K-601S c1ccc2c(c1)-c3c(cc(nn3)c4cccc(c4)C(F)(F)F)C2=O 11K-606S c1ccc(cc1)SCc2cc(nc(n2)c3ccncc3)N4CCOCC4 11K-607S c1ccc(cc1)SCc2cc(nc(n2)c3ccncc3)N4CCCC4 11K-608S CNc1cc(nc(n1)c2ccncc2)CSc3ccccc3 11K-609S COC(=O)c1ccccc1Sc2cc(nc(n2)c3ccccc3)CSc4ccccc4 11K-610S COC(=O)c1ccccc1Oc2cc(nc(n2)c3ccccc3)CSc4ccccc4 11K-611S CCOC(=O)CSc1cc(nc(n1)c2ccccc2)CSc3ccccc3 11K-613S CCOC(=O)C(C)Sc1cc(nc(n1)c2ccccc2)CSc3ccccc3 11K-614S c1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl 11K-615S c1cc(ccc1Sc2ccc(cc2C#N)N)Cl 11K-616S CN(C)c1cc(nc(n1)c2ccccc2)CSc3ccccc3 11K-623S c1ccc(cc1)c2nc(cc(n2)N3CCCC3)CSc4ccccc4 11K-624S CC(C)Nc1cc(nc(n1)c2ccccc2)CSc3ccccc3 11K-625S c1ccc(cc1)CNc2cc(nc(n2)c3ccccc3)CSc4ccccc4 11K-626S c1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3cccc(c3)C(F)(F)F 11K-627S c1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccc(cc3)Cl 11K-629S C=CCNc1cc(nc(n1)c2ccncc2)CS(=O)(=O)c3ccccc3 11K-630S C=CCNc1cc(nc(n1)c2ccccc2)CSc3ccccc3 11K-631S CCOC(=O)CSc1cc(nc(n1)c2ccccn2)CS(=O)c3ccc(cc3)Cl 11K-632S c1cc(ccc1Oc2cc(nc(n2)c3ccncc3)CS(=O)c4ccc(cc4)Cl)Cl 11K-633S COC(=O)c1ccccc1Sc2cc(nc(n2)c3ccncc3)CS(=O)c4ccc(cc4)Cl 11K-634S c1ccc(cc1)Sc2cc(nc(n2)c3ccccn3)CS(=O)c4ccc(cc4)Cl 11K-635S Cc1ccc(cc1)Sc2ccc(cc2C#N)[N+](=O)[O-] 11K-645S Cc1ccc(cc1)Sc2ccc(cc2C#N)N 11K-646S Cc1cccc(c1)c2cc3c(nn2)-c4ccccc4C3=O 11K-647S Cc1c(c(c(c(n1)C/C=N/OCc2ccc(cc2)[N+](=O)[O-])C#N)c3ccc(cc3)Cl)C#N 11K-900 CCOC(=O)c1c(con1)c2c(c(c(c(n2)C)C#N)c3ccc(cc3)Cl)C#N 11K-902 CNC1c2cc(ccc2OCC1CO)Br.Cl 11K-903 Cc1c(c(c(c(n1)/C=C/N(C)C)C#N)c2c(cccc2Cl)Cl)C#N 11K-904 CNC1c2cccc(c2OCC1CO)OC.Cl 11K-905 Cc1c(c(c(c(n1)/C=C/Nc2ccc(cc2)F)C#N)c3c(cccc3Cl)Cl)C#N 11K-906 Cc1c(c(c(c(n1)/C=C/Nc2cccc(c2)Cl)C#N)c3c(cccc3Cl)Cl)C#N 11K-907 Cc1c(c(c(c(n1)/C=C/Nc2ccc(cc2)OC(F)(F)F)C#N)c3c(cccc3Cl)Cl)C#N 11K-908 c1ccc2c(c1)ccc3c2C(C(CO3)CO)N.Cl 11K-910 c1c(c(c(=O)n(n1)C(=O)N)Cl)Cl 11K-911 c1c(c(c(=O)[nH]n1)Cl)Cl 11K-912 c1ccc2c(c1)nc(c(n2)Cl)NN=C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 11K-913 c1ccc2c(c1)nc(c(n2)Cl)NNC(=O)Nc3ccc(cc3)Cl 11K-914 C/C(=C(\C#N)/C(=O)N)/NCCc1ccc(c(c1)OC)OC 11K-915 CN(C)/C=C/c1c(c(=O)ncn1N(C)c2c(cc(cn2)C(F)(F)F)Cl)C#N 11K-916 COc1ccc(cc1)/N=C/Cc2c(c(=O)ncn2CCNc3c(cc(cn3)C(F)(F)F)Cl)C#N 11K-918 Cc1c(c(=O)ncn1CCc2ccc(c(c2)OC)OC)C#N 11K-919 Cc1c(c(=O)ncn1Cc2ccncc2)C#N 11K-920 CN(C)/C=C/c1c(c(=O)ncn1CCc2ccc(c(c2)OC)OC)C#N 11K-921 CO/N=C/Cc1c(c(=O)ncn1CCNc2c(cc(cn2)C(F)(F)F)Cl)C#N 11K-922 COc1ccc(cc1OC)CCn2cnc(=O)c(c2C/C=N/OCc3ccc(cc3)Cl)C#N 11K-923 COc1ccc(cc1OC)CCn2cnc(=O)c(c2C/C=N/OC/C=C/Cl)C#N 11K-924 CCOC(=O)CNC(=S)N(C)C1c2cccc(c2OCC1CO)OC 11K-925 c1cc[n+](cc1)CC(=O)c2c(ccs2)Br.[I-] 11K-927 c1cc[n+](cc1)CC(=O)c2cccs2.[I-] 11K-928 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3cccs3 11K-929 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3c(ccs3)Br 11K-930 CCn1c(=O)c(c(cn1)Cl)Cl 11K-931 C/C(=N\NC(=O)OC)/c1cccs1 11L-001 Cc1ccc(cc1)c2nnc3n2c(nc4c3cccc4)C(F)(F)F 11L-002 C/C(=N\NC(=O)OC)/c1ccncc1 11L-003 c1ccc(c(c1)c2csnn2)O 11L-004 C/C(=N\NC(=O)OC)/c1ccc(cc1)F 11L-005 C/C(=N\NC(=O)OC)/c1cccc(c1)C(F)(F)F 11L-006 c1cnccc1c2csnn2 11L-007 Cc1cc(n(n1)c2c3ccccc3nc(n2)C(F)(F)F)C 11L-008 c1ccc2c(c1)c(nc(n2)C(F)(F)F)N/N=C/c3ccc(cc3)Cl 11L-009 Cc1ccsc1/C=N/Nc2c3ccccc3nc(n2)C(F)(F)F 11L-012 C/C(=N\NC(=O)OC)/c1cccc(c1)O 11L-013 c1cc(sc1)c2csnn2 11L-014 c1ccc(c(c1)c2csnn2)OC(=O)c3cccs3 11L-015 c1ccc(c(c1)c2csnn2)OS(=O)(=O)c3ccc(cc3)Cl 11L-016 C/C(=N/NC(=O)OC)/c1ccc(cc1)Sc2ccccc2 11L-017 C/C(=N\NC(=O)OC)/c1ccc(cc1)n2ccnc2 11L-018 COc1ccc(cc1)C(=O)Oc2ccccc2c3csnn3 11L-019 c1cc(ccc1c2csnn2)F 11L-020 c1cc(cc(c1)C(F)(F)F)c2csnn2 11L-021 c1ccc(cc1)Sc2ccc(cc2)c3csnn3 11L-022 c1cc(ccc1c2csnn2)[NH+]3C=CN=C3.[Cl-] 11L-023 c1cc(ccc1c2csnn2)n3ccnc3 11L-024 CN(c1c2ccccc2nc(n1)C(F)(F)F)N 11L-025 Cc1cc(ccc1Oc2c3ccccc3nc(n2)C(F)(F)F)Cl 11L-026 c1ccc2c(c1)c(nc(n2)C(F)(F)F)Oc3ccc(cc3)[N+](=O)[O-] 11L-027 c1ccc2c(c1)c(nc(n2)C(F)(F)F)N/N=C/c3cccc(c3)[N+](=O)[O-] 11L-029 c1ccc2c(c1)c3nnc(n3c(n2)C(F)(F)F)c4ccc(cc4)Cl 11L-031 c1ccc(cc1)c2nnc3n2c(nc4c3cccc4)C(F)(F)F 11L-032 c1cc(cc(c1)O)c2csnn2 11L-033 COc1ccc(cc1)c2nnc3n2c(nc4c3cccc4)C(F)(F)F 11L-034 c1ccc2c(c1)c3nnc(n3c(n2)C(F)(F)F)c4cccc(c4)[N+](=O)[O-] 11L-035 c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)Cl)C#N)c3ccc(cc3)Cl 11L-304S c1ccc(cc1)N2c3ccccc3/C(=N/c4ccc(cc4)Cl)/C2=O 11L-309S COc1ccc(cc1)/C(=N/O)/Cl 11L-310S Cc1c(n(c2c1c(ncn2)Sc3ccc(cc3)C(C)C)Cc4ccccc4)C 11L-314S Cc1cccc(c1)Sc2c3c(c(n(c3ncn2)Cc4ccccc4)C)C 11L-315S Cc1c(n(c2c1c(ncn2)Sc3ccc(cc3)Br)Cc4ccccc4)C 11L-316S c1ccc(cc1)N2c3ccccc3/C(=N/c4ccc(cc4)C(F)(F)F)/C2=O 11L-318S c1c(c(cc(c1O)Cl)F)[N+](=O)[O-] 11L-319S c1ccc(cc1)N2c3ccccc3/C(=N/c4ccccc4C(F)(F)F)/C2=O 11L-320S c1ccc(cc1)N2c3ccccc3/C(=N/c4cccc(c4)Cl)/C2=O 11L-321S CCOC(=O)COc1cc(c(cc1Cl)F)[N+](=O)[O-] 11L-322S c1ccc(cc1)N2c3ccccc3/C(=N/c4cc(cc(c4)Cl)Cl)/C2=O 11L-324S Cc1ccc(cc1)/N=C\2/c3ccccc3N(C2=O)c4ccccc4 11L-325S COc1ccc(cc1)c2cc(on2)CO 11L-326S COc1ccc(cc1)c2cc(on2)C(=O)O 11L-327S c1cc(ccc1c2cc(nc(c2C#N)N3CCCC3)c4ccc(c(c4)Cl)Cl)Cl 11L-328S c1cc(ccc1c2cc(nc(c2C#N)N3CCOCC3)c4ccc(c(c4)Cl)Cl)Cl 11L-331S CC(=O)Nc1c2c(nn(c2ncn1)C(C)(C)C)c3ccc(cc3)Cl 11L-332S c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)Oc3ccc(cc3)Cl)C#N)c4ccc(cc4)Cl 11L-333S CC(=O)Nc1cccc(c1)Oc2c(c(cc(n2)c3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl)C#N 11L-334S Cc1cccc(c1C)Oc2c(c(cc(n2)c3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl)C#N 11L-335S c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)Oc3ccc(cc3)F)C#N)c4ccc(cc4)Cl 11L-336S Cc1cccc(c1)/N=C\2/c3ccccc3N(C2=O)c4ccccc4 11L-337S Cc1cc(cc(c1)/N=C\2/c3ccccc3N(C2=O)c4ccccc4)C 11L-338S c1ccc(c(c1)/C=N/O)Cl 11L-339S c1ccc(c(c1)c2cc(on2)CO)Cl 11L-341S c1ccc(cc1)N2c3ccccc3/C(=N/c4ccc(cc4)Br)/C2=O 11L-342S c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)Sc3ccc(cc3)F)C#N)c4ccc(cc4)Cl 11L-343S COc1ccc(cc1)Sc2c(c(cc(n2)c3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl)C#N 11L-344S Cc1ccc(cc1)Sc2c(c(cc(n2)c3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl)C#N 11L-345S c1cc(ccc1c2cc(nc(c2C#N)N3CCCCC3)c4ccc(c(c4)Cl)Cl)Cl 11L-349S c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)N3CCCCC3)C#N)c4ccc(cc4Cl)Cl 11L-350S CCOc1ccc(cc1)/N=C\2/c3ccccc3N(C2=O)c4ccccc4 11L-351S c1ccc(cc1)N2c3ccccc3/C(=N/c4ccc(cc4)Oc5ccccc5)/C2=O 11L-352S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3C(=O)C2=O)Cl 11L-353S c1c(c(cc(c1O)Cl)F)N 11L-354S CCOC(=O)COc1cc(c(cc1Cl)F)N 11L-355S COc1ccc(cc1)N/N=C\2/c3ccccc3N(C2=O)c4ccccc4 11L-357S c1ccc(cc1)N/N=C\2/c3ccccc3N(C2=O)c4ccccc4 11L-358S Cc1ccccc1N/N=C\2/c3ccccc3N(C2=O)c4ccccc4 11L-359S CC(C)(C)n1c(c(c(n1)c2ccc(cc2)Cl)C#N)NC(=O)c3cccc(c3)C(F)(F)F 11L-361S Cc1ccc(cc1)N/N=C\2/c3ccccc3N(C2=O)c4ccccc4 11L-363S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4ccc(c(c4)Cl)Cl)/C2=O 11L-364S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4cc(cc(c4)Cl)Cl)/C2=O 11L-365S c1cc(ccc1c2cc(on2)C(=O)O)Cl 11L-366S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4cc(ccc4Cl)Cl)/C2=O 11L-367S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4ccc(cc4)[N+](=O)[O-])/C2=O 11L-368S c1ccc(c(c1)c2cc(on2)C(=O)O)Cl 11L-369S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])/C2=O 11L-371S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N\Nc4c(cc(cc4Cl)C(F)(F)F)Cl)/C2=O)Cl 11L-372S c1ccc(cc1)N/N=C/2\c3cc(ccc3N(C2=O)Cc4cccc(c4)C(F)(F)F)Cl 11L-373S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N\Nc4ccc(cc4)[N+](=O)[O-])/C2=O)Cl 11L-374S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N\Nc4c(cc(cc4Cl)Cl)Cl)/C2=O)Cl 11L-375S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4c(cc(cc4Cl)Cl)Cl)/C2=O 11L-376S c1ccc(cc1)N2c3ccccc3/C(=N\Nc4c(cc(cc4Cl)C(F)(F)F)Cl)/C2=O 11L-377S Cc1ccc(cc1)c2cc(c(c(n2)N3CCN(CC3)C)C#N)c4ccc(cc4Cl)Cl 11L-382S CN1CCN(CC1)c2c(c(cc(n2)c3cccc(c3)C(F)(F)F)c4ccc(cc4Cl)Cl)C#N 11L-383S Cc1ccc(cc1)CN2c3ccccc3C(=O)C2=O 11L-384S c1ccc2c(c1)/C(=N\Nc3ccc(cc3)[N+](=O)[O-])/C(=O)N2Cc4cccc(c4)C(F)(F)F 11L-386S c1ccc2c(c1)/C(=N\Nc3cc(cc(c3)Cl)Cl)/C(=O)N2Cc4cccc(c4)C(F)(F)F 11L-387S c1ccc2c(c1)/C(=N\Nc3ccc(cc3)Br)/C(=O)N2Cc4cccc(c4)C(F)(F)F 11L-388S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4ccc(cc4)Cl)/C2=O 11L-390S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4ccc(cc4)F)/C2=O 11L-391S CN1c2ccccc2/C(=N/Nc3ccccc3)/C1=O 11L-395S CN1c2ccccc2/C(=N\Nc3ccc(cc3)OC)/C1=O 11L-396S COc1ccc(cc1)N/N=C/2\c3ccccc3N(C2=O)Cc4cccc(c4)C(F)(F)F 11L-397S Cc1ccc(cc1)CN2c3ccccc3/C(=N\Nc4ccc(cc4)Cl)/C2=O 11L-398S Cc1ccc(cc1)CN2c3ccccc3/C(=N\Nc4cccc(c4)F)/C2=O 11L-399S CN1c2ccccc2/C(=N\Nc3ccc(cc3)Cl)/C1=O 11L-400S CN1c2ccccc2/C(=N\Nc3ccc(cc3)Br)/C1=O 11L-401S COc1ccc(cc1)CSc2nc(cc(n2)Sc3ccc(cc3)OC)CSC 11L-502S Cn1c(c(c(n1)c2ccccc2)/C=N/OC)Sc3ccccc3C(=O)OC 11L-503S Cc1ccc(cc1)c2c(c(nc(n2)SC)Sc3ccc(cc3Cl)Cl)C#N 11L-504S Cc1ccc(cc1)c2c(c(nc(n2)SC)Sc3ccc(cc3)Cl)C#N 11L-505S Cc1ccc(cc1)c2c(c(nc(n2)SC)Sc3cccc(c3)C(F)(F)F)C#N 11L-506S CSCc1cc(nc(n1)SCc2ccc(cc2)Cl)O 11L-507S COc1ccc(cc1)CSc2nc(cc(n2)N3CCOCC3)CSC 11L-508S Cc1ccc(cc1)c2c(c(nc(n2)SC)Sc3cccc(c3)C)C#N 11L-513S c1ccc(cc1)CSc2nc(c(c(n2)O)C#N)c3ccccc3 11L-514S CC(c1cc(no1)c2ccc(cc2)Cl)O 11L-518S c1ccc(cc1)CSc2nc(c(c(n2)Cl)C#N)c3ccccc3 11L-519S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)O)C#N 11L-520S c1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3Cl)O)C#N 11L-521S c1ccc(cc1)c2c(c(nc(n2)SCc3cccc(c3)C(F)(F)F)O)C#N 11L-522S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)Cl)C#N 11L-523S c1ccc(cc1)CSc2nc(c(c(n2)Sc3cccc(c3)C(F)(F)F)C#N)c4ccccc4 11L-524S c1ccc(cc1)C2N=C(SC(=N2)c3ccc(cc3)Cl)c4ccc(cc4)Cl 11L-525S Cc1ccc(cc1)c2c(c(nc(n2)SC)Sc3cccc(c3Cl)Cl)C#N 11L-526S c1ccc(cc1)c2c(c(nc(n2)SCc3cccc(c3)C(F)(F)F)Cl)C#N 11L-530S Cc1ccc(cc1)CSc2nc(c(c(n2)O)C#N)c3ccccc3 11L-531S c1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3Cl)Cl)C#N 11L-532S Cc1ccc(cc1)CSc2nc(c(c(n2)Cl)C#N)c3ccccc3 11L-533S CS(=O)(=O)c1nccc(n1)c2ccccc2 11L-534S c1ccc(cc1)N2C(=O)CSC2=O 11L-536S c1cc(cc(c1)Cl)N2C(=O)CSC2=O 11L-537S Cc1c(c(on1)C)CS(=O)c2ccc(cc2)Br 11L-540S Cc1c(c(on1)C)CS(=O)(=O)c2ccc(cc2)Br 11L-541S Cc1c(c(on1)C)CSC 11L-542S Cc1ccc(cc1)N2C(=O)CSC2=O 11L-543S c1cc(cc(c1)N2C(=O)CSC2=O)C(F)(F)F 11L-544S Cc1ccccc1N2C(=O)CSC2=O 11L-545S c1cc(ccc1N2C(=O)CSC2=O)Cl 11L-546S c1ccc(cc1)CSc2nc(c(c(n2)N3CCOCC3)C#N)c4ccccc4 11L-550S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)NC)C#N 11L-551S c1c(cc(cc1Cl)Cl)N2C(=O)CSC2=O 11L-552S Cc1cccc(c1N2C(=O)CSC2=O)C 11L-553S Cc1c(c(on1)C)CSCc2ccc(cc2)Cl 11L-554S Cc1cc([nH]c(=S)c1C#N)C 11L-559S Cc1c(c(on1)C)CS(=O)(=O)C2CCCCC2 11L-563S c1ccc(cc1)N/N=C\2/c3ccccc3N(C2=O)Cc4ccc(c(c4)Cl)Cl 11L-564S c1ccc2c(c1)/C(=N\Nc3c(cc(cc3Cl)C(F)(F)F)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11L-565S c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11L-566S c1ccc2c(c1)/C(=N\Nc3cccc(c3)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11L-567S CC(=O)c1cc(no1)c2ccc(cc2)Cl 11L-568S c1ccc2c(c1)/C(=N\Nc3ccccc3Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 11L-569S C=CCN1c2ccccc2C(=O)C1=O 11L-570S Cc1c(c(on1)C)CS(=O)(=O)CC(=O)OC 11L-572S Cc1c(c(on1)C)CS(=O)(=O)Cc2ccc(cc2)Cl 11L-573S Cc1c(c(on1)C)CS(=O)Cc2ccc(cc2)Cl 11L-574S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SC)/C=C/c3ccc(cc3)C 11L-577S Cc1c(c(on1)C)CSc2ccc(cc2)[N+](=O)[O-] 11L-579S Cc1c(c(on1)C)CSc2ccc(cc2)NC(=O)C 11L-580S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCC=C)/C=C/c3ccc(cc3)C 11L-581S CCCSc1c(c(cc(n1)/C=C/c2ccc(cc2)C)/C=C\c3ccc(cc3)C)C#N 11L-583S CSc1c(c(cc(n1)/C=C/c2ccccc2)/C=C/c3ccccc3)C#N 11L-584S CCOC(=O)c1c(cc([nH]c1=O)C)O 11L-585S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3ccc(cc3)F)/C=C/c4ccc(cc4)C 11L-586S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3cccc(c3)C(F)(F)F)/C=C/c4ccc(cc4)C 11L-587S Cc1c(c(on1)C)CNc2ccc(cc2)Cl 11L-588S Cc1c(c(on1)C)CN2CCOCC2 11L-590S Cc1c(c(on1)C)CS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] 11L-591S c1cc(ccc1c2cc(on2)C(=O)CBr)Cl 11L-593S c1ccc2c(c1)/C(=N\Nc3c(cc(cc3Cl)C(F)(F)F)Cl)/C(=O)N2Cc4cccc(c4)C(F)(F)F 11L-594S c1ccc(cc1)N/N=C/2\c3ccccc3N(C2=O)Cc4cccc(c4)C(F)(F)F 11L-595S Cc1nc(cs1)c2cc(no2)c3ccc(cc3)Cl 11L-596S c1ccc2c(c1)c(c(s2)C#N)OCc3ccc(cc3)Cl 11L-597S C=CCOc1c2ccccc2sc1C#N 11L-598S c1ccc2c(c1)c(c(s2)C#N)OCc3c(cccc3Cl)Cl 11L-599S Cc1c(c(on1)C)CN(C)C 11L-600S CNc1cc(nc(n1)SCc2ccc(cc2)OC)CSC 11L-601S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3ccccc3C)/C=C/c4ccc(cc4)C 11L-602S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3cccc(c3)C)/C=C/c4ccc(cc4)C 11L-603S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3cccc(c3)Cl)/C=C/c4ccc(cc4)C 11L-604S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3ccc(cc3)Cl)/C=C/c4ccc(cc4)C 11L-605S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3ccc(cc3)C(C)(C)C)/C=C/c4ccc(cc4)C 11L-606S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3ccc(c(c3)Cl)Cl)/C=C/c4ccc(cc4)C 11L-607S Cc1c(c(on1)C)CNc2ccccc2 11L-609S Cc1c(c(on1)C)CN2CCCC2 11L-610S Cc1c(c(on1)C)CNc2ccc(cc2)OC 11L-612S Cc1c(c(on1)C)CN2CCN(CC2)C 11L-613S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCC#C)/C=C/c3ccc(cc3)C 11L-614S Cc1ccc(cc1)CSc2c(c(cc(n2)/C=C/c3ccc(cc3)C)/C=C\c4ccc(cc4)C)C#N 11L-615S Cc1ccc(cc1)/C=C\c2cc(nc(c2C#N)SCc3ccccc3)/C=C/c4ccc(cc4)C 11L-616S COc1c2ccccc2sc1C#N 11L-617S c1ccc2c(c1)c(c(s2)C#N)OCc3c(cccc3Cl)F 11L-618S Cc1c(c(on1)C)COC 11L-619S Cc1c(c(on1)C)COC(C)C 11L-620S Cc1c(c(on1)C)COc2ccccc2 11L-621S Cc1c(c(on1)C)COc2ccc(cc2)Cl 11L-622S c1ccc2c(c1)c(c(s2)C#N)OCc3ccc(cc3Cl)Cl 11L-623S c1ccc2c(c1)c(c(s2)C#N)OCc3ccc(cc3)[N+](=O)[O-] 11L-624S c1ccc2c(c1)c(c(s2)C#N)OCc3ccc(cc3)F 11L-625S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)NC(C)C)C#N 11L-627S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)NCC=C)C#N 11L-629S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)N4CCCCC4)C#N 11L-631S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)N4CCN(CC4)C)C#N 11L-632S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)NCc4ccccc4)C#N 11L-633S Cc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)NC4CCCCC4)C#N 11L-634S CCN(CC)c1c(c(nc(n1)SCc2ccccc2)c3ccc(cc3)C)C#N 11L-635S C=CCNc1c(c(nc(n1)SCc2cccc(c2)C(F)(F)F)c3ccccc3)C#N 11L-636S c1ccc(cc1)c2c(c(nc(n2)SCc3cccc(c3)C(F)(F)F)NC4CCCCC4)C#N 11L-637S CN1CCN(CC1)c2c(c(nc(n2)SCc3cccc(c3)C(F)(F)F)c4ccccc4)C#N 11L-638S CCN(CC)c1c(c(nc(n1)SCc2cccc(c2)C(F)(F)F)c3ccccc3)C#N 11L-639S CNc1c(c(nc(n1)SCc2ccccc2Cl)c3ccccc3)C#N 11L-640S C=CCNc1c(c(nc(n1)SCc2ccccc2Cl)c3ccccc3)C#N 11L-641S c1ccc(cc1)c2c(c(nc(n2)N3CCCC3)N4CCCC4)C#N 11L-643S CCN(CC)c1c(c(nc(n1)SCc2ccccc2Cl)c3ccccc3)C#N 11L-644S CCCNc1c(c(nc(n1)SCc2ccccc2Cl)c3ccccc3)C#N 11L-645S c1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3Cl)N4CCOCC4)C#N 11L-646S CC(C)Nc1c(c(nc(n1)SCc2ccccc2Cl)c3ccccc3)C#N 11L-647S C=CCNc1c(c(nc(n1)SCc2c(cccc2Cl)Cl)c3ccccc3)C#N 11L-648S CCCNc1c(c(nc(n1)SCc2c(cccc2Cl)Cl)c3ccccc3)C#N 11L-649S c1ccc(cc1)c2c(c(nc(n2)SCc3c(cccc3Cl)Cl)NC4CCCCC4)C#N 11L-650S c1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3Cl)NC4CCCCC4)C#N 11L-652S COc1ccc(cc1)C2C(=C(OC3=C2/C(=N/OCc4ccc(cc4)Cl)/CCC3)n5cccc5)C#N 11L-700 CC(C)(CCl)C(=O)Nc1cccc(c1)[N+](=O)[O-] 11L-701 CN1C(=O)c2ccccc2/C(=N\Nc3ccc(cc3)Cl)/C1=O 11L-702 CC1(CN(C1=O)c2cccc(c2)[N+](=O)[O-])C 11L-703 CC(C)(CCl)C(=O)Nc1ccc(cc1C(=O)c2ccccc2)Cl 11L-704 CC1(CN(C1=O)c2ccc(cc2C(=O)c3ccccc3)Cl)C 11L-705 CC1=C(C(NC(=S)N1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3Cl)Cl 11L-706 c1ccc2c(c1)c(c(s2)C=O)Cl 11L-707 c1ccc2c(c1)/C(=N\Nc3cccc(c3)[N+](=O)[O-])/C(=O)OC2=O 11L-708 c1ccc2c(c1)/C(=N/Nc3ccc(nc3)Cl)/C(=O)OC2=O 11L-710 C1C2C=CC1C3C2C(=O)N(C3=O)N4C(=O)CSC4=S 11L-711 Cc1ccc(cc1)CO/N=C/2\CCCC3=C2C(C(=C(O3)n4cccc4)C#N)c5ccc(cc5)OC 11L-712 c1cc(sc1c2ccno2)S(=O)(=O)N3CCCCC3 11L-713 CC1(CN(C1=O)c2ccc(cc2)c3ccno3)C 11L-714 CCOC(=O)c1c2c(sc1N)CCCC2 11L-717 CN(C)/C=C\1/C(=O)N(C(=S)S1)N2C(=O)C3C4CC(C3C2=O)C=C4 11L-718 CC1(CN(C1=O)c2nccs2)C 11L-719 CC1(CN(C1=O)c2ccc(cc2)c3ccnc4n3ncn4)C 11L-720 CC1(CN(C1=O)c2ccc(cc2)/C(=C/N(C)C)/C#N)C 11L-721 c1ccn(c1)C2=C(C(C3=C(O2)CCCC3=O)c4cccs4)C#N 11L-722 COc1ccc(cc1)N/C=C\2/C(=O)N(C(=S)S2)N3C(=O)CCC3=O 11L-724 c1ccc(cc1)COc2ccc(cc2)/C=C\3/C(=O)N(C(=S)S3)N4C(=O)c5ccccc5C4=O 11L-725 CC(=C)C(=O)Nc1ccc(cc1Cl)[N+](=O)[O-] 11L-726 Cc1ccc(cc1)NC(=O)C(=C)C 11L-727 CC(=C)C(=O)Nc1ccsc1C(=O)OC 11L-730 COc1ccc(cc1)NC(=O)C(=C)CS(=O)(=O)c2ccccc2 11L-731 CC1(CN(C1=O)c2ccc(cc2)c3ccnc4n3ncc4c5ccc(cc5)Cl)C 11L-732 CC(C)(CCl)C(=O)NN(C)c1c(cc(cn1)C(F)(F)F)Cl 11L-733 CC1(CN(C1=O)N(C)c2c(cc(cn2)C(F)(F)F)Cl)C 11L-734 CC1(CN(C1=O)c2ccc(cc2)C(=O)C/C=N/OCc3ccc(cc3)Cl)C 11L-735 CC1(CN(C1=O)c2ccc(cc2)OC(F)(F)F)C 11L-736 COc1ccc(cc1)CN2C(=O)c3ccccc3C(C2=O)/C=N/OCc4ccc(cc4)Cl 11L-738 CC1(CN(C1=O)c2ccc(cc2)C(/C=N/OCc3ccc(cc3Cl)F)C#N)C 11L-739 COc1ccc(cc1)C2C(=C(OC3=C2/C(=N/OCc4ccc(cc4)F)/CCC3)n5cccc5)C#N 11L-740 CC(C)c1ccc(cc1)NC(=O)C(C)(C)CCl 11L-741 CC(C)c1ccc(cc1)N2CC(C2=O)(C)C 11L-742 CC(C)(CCl)C(=O)Nc1cccc(c1)O 11L-744 CC1(CN(C1=O)c2cccc(c2)O)C 11L-745 CC1=C(C(NC(=N1)SCc2ccc(cc2)OC)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4Cl)Cl 11L-746 Cc1ccc(cc1)CO/N=C\C2c3ccccc3C(=O)N(C2=O)Cc4ccc(cc4)OC 11L-747 CC1(CN(C1=O)c2ccc(cc2)c3ccnc4n3nc(n4)SCc5cccc(c5)Cl)C 11L-748 COc1ccc(cc1)CN2C(=O)c3ccccc3C(C2=O)/C=N\OCc4ccc(cc4)F 11L-749 c1ccc2c(c1)c(c(s2)/C=N/OCc3ccc(cc3)Cl)Cl 11L-750 c1cc(ccc1/C=C\2/C(=O)N(C(=S)S2)N3C(=O)C4C5CC(C4C3=O)C=C5)[N+](=O)[O-] 11L-751 CC(C)(CCl)C(=O)Nc1cccc(n1)NC(=O)C(C)(C)CCl 11L-753 CC1(CN(C1=O)c2cccc(n2)N3CC(C3=O)(C)C)C 11L-754 c1ccc(cc1)CN2C(=O)c3ccccc3C(C2=O)/C=N/OCc4c(cccc4Cl)F 11L-755 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C4CC(C3C2=O)C(C4C#N)O 11L-901 Cc1ccc(cc1)c2ccnc(n2)C3CN(C(=O)NC3=O)Cc4ccc(cc4)OC 11L-902 c1cc2c(cc1Cl)[nH]c(=O)c(=O)n2CCNc3c(cc(cn3)C(F)(F)F)Cl 11L-903 c1cc(c(cc1Cl)NC(=O)N)NCCNc2c(cc(cn2)C(F)(F)F)Cl 11L-904 c1cc(c2ccoc2c1)CC(=O)O 11L-905 c1cc2c(cc1Cl)nc(c(=O)n2CCNc3c(cc(cn3)C(F)(F)F)Cl)Cl 11L-906 CCOC(=O)NC(=O)C(=NNc1ccc(cc1F)F)C(=O)C 11L-908 CCOC(=O)NC(=O)/C(=N\Nc1ccc(cc1)Cl)/C(=O)C 11L-909 c1cc2c(cc1Cl)nc(c(=O)n2CCNc3c(cc(cn3)C(F)(F)F)Cl)N4CCCC4 11L-910 COCCNc1c(=O)n(c2ccc(cc2n1)Cl)CCNc3c(cc(cn3)C(F)(F)F)Cl 11L-911 COC(=O)c1cc(c(=O)oc1C/C=N\OCc2ccc(cc2Cl)Cl)NC(=O)c3ccccc3 11L-912 COC(=O)c1cc(c(=O)oc1C/C=N\OCc2ccc(c(c2)Cl)Cl)NC(=O)c3ccccc3 11L-913 CC(=O)c1c(=O)[nH]c(=O)n(n1)c2ccc(cc2F)F 11L-915 c1cc(oc1)CNc2c(=O)n(c3ccc(cc3n2)Cl)CCNc4c(cc(cn4)C(F)(F)F)Cl 11L-916 c1cc2c(cc1Cl)nc(c(=O)n2CCNc3c(cc(cn3)C(F)(F)F)Cl)N4CCOCC4 11L-917 CC(=O)c1c(=O)[nH]c(=O)n(n1)c2ccc(cc2)Cl 11L-918 c1cc2c(cc1Cl)n3cnnc3c(=O)n2CCNc4c(cc(cn4)C(F)(F)F)Cl 11L-920 Cc1nnc2n1c3cc(ccc3n(c2=O)CCNc4c(cc(cn4)C(F)(F)F)Cl)Cl 11L-921 c1cc2c(cc1Cl)n3c(c(=O)n2CCNc4c(cc(cn4)C(F)(F)F)Cl)nnc3C(F)(F)F 11L-922 CC(=O)c1c(=O)n(c(=O)n(n1)c2ccc(cc2F)F)C 11L-923 CCOC(=O)NC(=O)/C(=N\Nc1cc(cc(c1)Cl)Cl)/C(=O)C 11L-924 Cn1c(=O)c(nn(c1=O)c2ccc(cc2F)F)C(=O)CBr 11L-925 Cn1c(=O)c(nn(c1=O)c2ccc(cc2)Cl)C(=O)/C=C/N(C)C 11L-926 c1ccc(cc1)NC(=O)N2C3(CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)CC(=O)N2 11L-927 CC(=O)c1c(=O)[nH]c(=O)n(n1)c2cc(cc(c2)Cl)Cl 11L-928 Cn1c(=O)c(nn(c1=O)c2ccc(cc2)Cl)c3ccnn3c4ccccc4 11L-929 Cn1c(=O)c(nn(c1=O)c2ccc(cc2)Cl)c3ccnn3C4CCS(=O)(=O)C4 11L-930 Cn1c(=O)c(nn(c1=O)c2ccc(cc2F)F)c3csc(n3)c4ccccc4 11L-931 CCOC(=O)C1=NOC2C1C3CC2C4C3C(=O)N(C4=O)CCc5ccc(c(c5)OC)OC 11L-932 COc1ccc(cc1OC)CCN2C(=O)C3C4CC(C3C2=O)C5C4C(=NO5)C(=O)NN 11L-933 Cc1ccc(cc1C)N/C=C/C(=O)c2c(=O)n(c(=O)n(n2)c3ccc(cc3)Cl)C 11L-934 Cn1c(=O)c(nn(c1=O)c2ccc(cc2)Cl)c3ccnc(n3)c4ccccc4 11L-935 CCOC(=O)NC(=O)/C(=N\Nc1ccc(cc1)OC)/C(=O)C 11L-936 c1ccc2c(c1)C(=O)C(=C(C#N)C#N)C2=O 11L-937 Cn1c(=O)c(nn(c1=O)c2ccc(cc2F)F)C(=O)/C=C/N(C)C 11L-938 COc1ccc(cc1OC)CCN2C(=O)C3C4CC(C3C2=O)C5C4C(=NO5)C(=O)O 11L-939 COc1ccc(cc1OC)CCN2C(=O)C3C4CC(C3C2=O)C5C4C(=NO5)C(=O)N/N=C\c6ccc(cc6)Cl 11L-940 CC(=O)c1c(=O)[nH]c(=O)n(n1)c2ccc(cc2)OC 11L-941 c1ccc(cc1)N2C(=O)C3C(NC(=C4C(=O)c5ccccc5C4=O)C3C2=O)c6ccccn6 11L-942 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C(NC(=C4C(=O)c5ccccc5C4=O)C3C2=O)c6ccccn6 11L-943 Cn1c(=O)c(nn(c1=O)c2ccc(cc2F)F)c3ccn[nH]3 11L-944 Cn1c(=O)c(nn(c1=O)c2ccc(cc2F)F)c3ccnc(n3)c4ccncc4 11L-945 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)c5ccccn5)C(=O)N(C4=O)c6ccc(cc6Cl)Cl)C2=O 11L-947 COC(=O)c1c(ccs1)N2C(=O)C3C(NC(=C4C(=O)c5ccccc5C4=O)C3C2=O)c6ccccn6 11L-948 COc1ccc(cc1OC)CCN2C(=O)C3C4CC(C3C2=O)C5C4C(=NO5)C(=O)N 11L-950 CC(=O)c1c(=O)n(c(=O)n(n1)c2cc(cc(c2)Cl)Cl)C 11L-951 Cn1c(=O)c(nn(c1=O)c2cc(cc(c2)Cl)Cl)c3csc(n3)c4cccnc4 11L-953 c1ccc(cc1)/C=C/C2C3C(C4N2CSC4)C(=O)N(C3=O)c5ccccc5 11L-954 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)c5ccccn5)C(=O)N(C4=O)CCNc6c(cc(cn6)C(F)(F)F)Cl)C2=O 11L-955 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)c5ccccn5)C(=O)N(C4=O)c6ccc(cc6)Cl)C2=O 11L-956 Cn1c(=O)c(nn(c1=O)c2cc(cc(c2)Cl)Cl)c3csc(n3)N 11L-957 c1ccc2c(c1)C(=O)C(=C(C#N)NCc3ccccn3)C2=O 11L-958 c1ccc2c(c1)C(=O)C(=C(C#N)NCC(=O)O)C2=O 11L-959 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)C(=O)O)C(=O)N(C4=O)c5ccc(cc5)Cl)C2=O 11L-960 CCOC(=O)NC(=O)/C(=N/Nc1cccc(c1)C(F)(F)F)/C(=O)C 11L-961 CC(=O)c1c(=O)[nH]c(=O)n(n1)c2cccc(c2)C(F)(F)F 11L-962 C/C(=N\OC)/C1CC1c2ccc(cc2)Cl 11M-001 c1ccc(cc1)OCCN2C(=O)C(=O)N(C2=O)Cc3cccc(c3)Cl 11M-002 c1ccc(cc1)CN2C(=O)C(=O)N(C2=O)Cc3ccccc3[N+](=O)[O-] 11M-003 C/C(=N\OCc1ccccc1)/C2CC2c3ccc(cc3)Cl 11M-004 COc1ccccc1CN2C(=O)C(=O)N(C2=O)CC(=O)c3ccc(cc3)F 11M-005 c1ccc(c(c1)CNC(=O)N)F 11M-006 c1ccc(c(c1)CN2C(=O)C(=O)NC2=O)F 11M-007 CN(C)c1ccnc(c1C#N)n2ccnc2 11M-008 CN(C)c1ccnc(c1C#N)n2cccc2 11M-009 CN(C)c1ccnc(c1C#N)n2cncn2 11M-011 Cc1ccc(cc1)C(=O)CN2C(=O)C(=O)N(C2=O)Cc3cccc(c3)C(F)(F)F 11M-012 c1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC(=O)c3ccccc3Cl 11M-013 c1cc(cc(c1)Cl)CN2C(=O)C(=O)N(C2=O)CC(=O)c3cccc(c3)C(F)(F)F 11M-014 c1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC(=O)c3ccc(cc3)c4ccccc4 11M-015 CN(C)c1ccnc(c1C#N)n2cccc2C=O 11M-016 CN(C)c1ccnc(c1C#N)n2cccc2/C=N/O 11M-017 CN(C)c1ccnc(c1C#N)n2cccc2/C=N/OC 11M-018 c1cc(cc(c1)Cl)CN2C(=O)C(=O)N(C2=O)CC(=O)c3ccc(cc3)Br 11M-019 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2c(cc(cc2C)C)C 11M-020 Cc1cc(c(c(c1)C)CN2C(=O)C(=O)N(C2=O)Cc3ccccc3F)C 11M-021 CN(C)c1ccnc(c1C#N)n2cccc2/C=N/OCc3ccc(cc3)[N+](=O)[O-] 11M-022 CN(C)c1ccnc(c1C#N)n2cccc2/C=N/OCc3cccc(c3)F 11M-023 CN(C)c1ccnc(c1C#N)n2cccc2/C=N/OCc3ccccc3OC 11M-024 CN(C)c1ccnc(c1C#N)n2cccc2/C=N/OCc3ccc(cc3Cl)F 11M-025 c1cc(cc(c1)Cl)CN2C(=O)C(=O)N(C2=O)CC#N 11M-026 Cc1cc(c(c(c1)C)CN2C(=O)C(=O)N(C2=O)CC(=O)O)C 11M-027 CN(C)c1ccnc(c1C#N)n2cccc2/C=N/OCc3ccccc3 11M-028 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2ccccc2F 11M-029 Cc1cc(c(c(c1)C)CN2C(=O)C(=O)N(C2=O)OC)C 11M-030 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2c(cccc2Cl)F 11M-031 COc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC(=O)N 11M-032 c1cc(c(c(c1)Cl)CN2C(=O)C(=O)N(C2=O)CC(=O)O)F 11M-033 c1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC#N 11M-034 c1ccc(c(c1)n2cccc2)F 11M-035 Cc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC#N 11M-036 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2ccc(cc2Cl)Cl 11M-037 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2ccccc2 11M-038 Cc1cc(c(c(c1)C)CN2C(=O)C(=O)N(C2=O)OCc3ccc(cc3Cl)F)C 11M-039 c1ccc(c(c1)CN2C(=O)C(=O)N(C2=O)CC(=O)O)F 11M-040 c1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC(=O)O 11M-041 c1cc(c(c(c1)Cl)CON2C(=O)C(=O)N(C2=O)Cc3ccc(c(c3)Cl)Cl)F 11M-042 c1ccc(c(c1)C(=O)CN2C(=O)C(=O)N(C2=O)Cc3cccc(c3)C(F)(F)F)Cl 11M-043 Cc1ccccc1CN2C(=O)C(=O)N(C2=O)OCc3ccccc3F 11M-044 c1cc(cc(c1)Cl)CN2C(=O)C(=O)N(C2=O)CC(=O)N 11M-045 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2ccc(cc2)[N+](=O)[O-] 11M-046 c1cc(c(cc1Cl)Cl)CN2C(=O)C(=O)N(C2=O)CC(=O)O 11M-047 Cc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC(=O)N 11M-048 CON1C(=O)C(=O)N(C1=O)Cc2ccc(cc2)[N+](=O)[O-] 11M-050 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2ccc(cc2)C(F)(F)F 11M-051 CC(C)c1ccc(cc1)/C=C/C(=O)/C=C/N(C)C 11M-052 c1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC(=O)N 11M-053 c1cc(ccc1CN2C(=O)C(=O)N(C2=O)CC(=O)O)[N+](=O)[O-] 11M-054 c1cc(ccc1CN2C(=O)C(=O)N(C2=O)CC(=O)O)C(F)(F)F 11M-055 CC(C)c1ccc(cc1)C2CC2C(=O)C 11M-056 c1cc(ccc1CN2C(=O)C(=O)N(C2=O)CC(=O)N)F 11M-057 CC(C)c1ccc(cc1)/C=C\c2ccnc3n2nc(n3)SC/C=C/c4ccccc4 11M-058 CC(C)c1ccc(cc1)/C=C\c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 11M-059 CC(C)c1ccc(cc1)/C=C\c2ccnc3n2nc(n3)SC 11M-060 c1ccc(c(c1)CN2CCn3c(cc(n3)C(=O)O)C2=O)Cl 11M-301S C=CCSc1ncc(n1Cc2ccccc2)/C=N/Nc3c(cc(cc3Cl)Cl)Cl 11M-309S C=CCSc1ncc(n1Cc2ccccc2)/C=N/Nc3ccc(cc3)Cl 11M-310S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)c2ccc(cc2)OC)c3ccccc3 11M-312S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)c2cccc(c2)C(F)(F)F)c3ccccc3 11M-313S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)c2ccc(cc2)Cl)c3ccccc3 11M-314S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)c2c(cccc2F)F)c3ccccc3 11M-315S C=CCSc1ncc(n1Cc2ccccc2)/C=N/O 11M-316S c1ccc(cc1)C(=N)NCC(=O)O 11M-317S c1ccc(cc1)c2[nH]c(c(n2)C=O)Cl 11M-318S COc1ccc(cc1)CN2CCn3c(cc(n3)C(=O)O)C2=O 11M-319S CCOC(=O)c1cn(nc1C(F)(F)F)C 11M-320S Cn1cc(c(n1)C(F)(F)F)C(=O)O 11M-321S Cn1cc(c(n1)C(F)(F)F)C(=O)N2CCN(CC2)C 11M-323S Cn1cc(c(n1)C(F)(F)F)C(=O)N2CCN(CC2)c3ccccc3F 11M-324S Cc1ccnc(c1)NC(=O)c2cn(nc2C(F)(F)F)C 11M-325S Cn1cc(c(n1)C(F)(F)F)C(=O)Nc2cccnc2 11M-326S Cn1cc(c(n1)C(F)(F)F)C(=O)Nc2ncccn2 11M-327S Cc1ccc(cc1)Sc2c(nc([nH]2)c3ccccc3)C=O 11M-328S CCSc1c(nc(n1C)c2ccccc2)/C=N/NC 11M-329S CCSc1ncc(n1C)/C=N/Nc2ccc(cc2)F 11M-331S CCSc1ncc(n1C)/C=N/Nc2ccc(cc2)Cl 11M-332S COc1ccc(cc1)CN2CCn3c(c(cn3)C(=O)Nc4ccc(cc4Cl)Cl)C2=O 11M-333S Cc1cc(cc(c1)NC(=O)c2cnn3c2C(=O)N(CC3)Cc4ccc(cc4)OC)C 11M-334S c1cc(cc(c1)C(F)(F)F)C(=N)NCC(=O)O 11M-335S COc1ccc(cc1)CN2CCn3c(c(cn3)C(=O)Nc4ccccc4)C2=O 11M-336S Cc1cccc(c1)NC(=O)c2cnn3c2C(=O)N(CC3)Cc4ccc(cc4)OC 11M-337S COc1ccc(cc1)CN2CCn3c(cc(n3)C(=O)Nc4ccc(cc4)OC)C2=O 11M-338S Cc1cc(ccc1NC(=O)c2cc3n(n2)CCN(C3=O)Cc4ccc(cc4)OC)Cl 11M-339S CCSc1ncc(n1C)/C=N/c2ccc(cc2)OC 11M-340S CCSc1ncc(n1C)/C=N/c2ccc(cc2)F 11M-341S CCSc1ncc(n1C)/C=N/c2ccc(cc2F)F 11M-342S CCSc1ncc(n1C)/C=N/c2ccc(c(c2)C)C 11M-343S Cc1ccc(cc1)Sc2c(nc([nH]2)c3ccccc3)/C=N/Nc4ccccc4 11M-344S Cc1ccc(cc1)Sc2c(nc([nH]2)c3ccccc3)/C=N/Nc4c(cc(cc4Cl)Cl)Cl 11M-345S Cc1ccc(cc1)Sc2c(nc([nH]2)c3ccccc3)/C=N/c4ccc(cc4)Cl 11M-346S Cc1ccc(cc1)Sc2c(nc([nH]2)c3ccccc3)/C=N/c4ccc(c(c4)C)C 11M-347S Cc1c2ccccc2nc(c1C(=O)C)Sc3ccccc3 11M-501S Cc1c2ccccc2nc(c1C(=O)C)Sc3cccc(c3)Cl 11M-502S CCOC(=O)c1cnc(nc1NC)c2ccccc2 11M-503S CCOC(=O)c1cnc(nc1N2CCOCC2)c3ccccc3 11M-504S Cc1c2ccccc2nc(c1C(=O)C)Sc3ccc(cc3Cl)Cl 11M-507S CCOC(=O)c1cnc(nc1NCc2ccccc2)c3ccccc3 11M-508S CCOC(=O)c1cnc(nc1Sc2ccc(cc2)Cl)c3ccccc3 11M-509S c1ccc(cc1)c2ncc(c(n2)Sc3ccc(cc3)Cl)C(=O)O 11M-510S CCOC(=O)c1cnc(nc1NCC=C)c2ccccc2 11M-511S CCOC(=O)c1cnc(nc1N2CCN(CC2)C)c3ccccc3 11M-512S CCOC(=O)c1cnc2ccccn2c1=O 11M-514S CCOC(=O)c1cnc(nc1Sc2ccccc2)c3ccccc3 11M-515S c1ccc(cc1)c2ncc(c(n2)Sc3ccccc3)C(=O)O 11M-516S CCOC(=O)c1cnc(nc1Sc2ccc(cc2)C)c3ccccc3 11M-517S Cc1ccc(cc1)Sc2c(cnc(n2)c3ccccc3)C(=O)O 11M-518S CCOC(=O)c1cnc(nc1Sc2cccc(c2)Cl)c3ccccc3 11M-519S c1ccc(cc1)c2ncc(c(n2)Sc3cccc(c3)Cl)C(=O)O 11M-520S CCOC(=O)c1cnc(nc1Sc2cccc(c2)C(F)(F)F)c3ccccc3 11M-521S c1ccc(cc1)c2ncc(c(n2)Sc3cccc(c3)C(F)(F)F)C(=O)O 11M-522S CCOC(=O)c1cnc(nc1Sc2cccc(c2)C)c3ccccc3 11M-523S Cc1cccc(c1)Sc2c(cnc(n2)c3ccccc3)C(=O)O 11M-524S CCOC(=O)c1cnc(nc1N2CCSCC2)c3ccccc3 11M-525S CCOC(=O)c1cnc(nc1N2CC(OC(C2)C)C)c3ccccc3 11M-526S CCOC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)C(F)(F)F 11M-528S CCOC(=O)c1cnc(nc1Sc2ccc(cc2)OC)c3ccccc3 11M-534S COc1ccc(cc1)Sc2c(cnc(n2)c3ccccc3)C(=O)O 11M-535S CCOC(=O)c1cnc(nc1Sc2cc(ccc2C)C)c3ccccc3 11M-536S Cc1ccc(c(c1)Sc2c(cnc(n2)c3ccccc3)C(=O)O)C 11M-537S CCOC(=O)c1cnc(nc1Sc2ccccc2Cl)c3ccccc3 11M-538S c1ccc(cc1)c2ncc(c(n2)Sc3ccccc3Cl)C(=O)O 11M-539S CCOC(=O)c1cnc(nc1Oc2cccc(c2)C(F)(F)F)c3ccccc3 11M-540S CCOC(=O)c1cnc(nc1NC2CCCCC2)c3ccccc3 11M-544S CCOC(=O)c1cnc(nc1N2CCCC2)c3ccccc3 11M-545S CCOC(=O)c1cnc(nc1Oc2ccc(c(c2)Cl)Cl)c3ccccc3 11M-546S CCOC(=O)c1cnc(nc1Sc2ccc(cc2Cl)Cl)c3ccccc3 11M-548S c1ccc(cc1)c2ncc(c(n2)Sc3ccc(cc3Cl)Cl)C(=O)O 11M-549S c1ccc(cc1)c2ncc(c(n2)Sc3ccc(cc3)Cl)C(=O)N4CCOCC4 11M-555S CC(=O)Nc1ccc(cc1)OCC(=O)NN 11M-557S CCOC(=O)c1c(cc(=O)n(n1)c2ccccc2)C(F)(F)F 11M-558S c1cc(cc(c1)n2c(=O)cc(c(n2)C(=O)Nc3ccc(cc3)C(F)(F)F)C(F)(F)F)C(F)(F)F 11M-560S c1cc(cc(c1)NC(=O)c2c(cc(=O)n(n2)c3cccc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F 11M-561S c1ccc(cc1)NC(=O)c2c(cc(=O)n(n2)c3cccc(c3)C(F)(F)F)C(F)(F)F 11M-562S c1ccc(cc1)c2ncc(c(n2)Sc3ccc(cc3)Cl)C(=O)Nc4cccc(c4)C(F)(F)F 11M-571S c1ccc(cc1)c2ncc(c(n2)Sc3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)Cl 11M-573S CCOC(=O)c1cnc(nc1Oc2ccccc2)c3ccccc3 11M-574S CCOC(=O)c1cnc(nc1Oc2ccc(cc2)Cl)c3ccccc3 11M-575S CCOC(=O)c1cnc(nc1Oc2cccc(c2C)C)c3ccccc3 11M-577S CCOC(=O)c1cnc(nc1Oc2ccc(cc2)C)c3ccccc3 11M-578S CCOC(=O)c1cnc(nc1Oc2ccc(cc2)F)c3ccccc3 11M-579S CCOC(=O)c1cnc(nc1Oc2cc(c(cc2Cl)Cl)Cl)c3ccccc3 11M-580S c1cc(ccc1C(F)(F)F)OCC(=O)NN 11M-581S CCOC(=O)c1cnc(nc1Oc2ccc(cc2)OC)c3ccccc3 11M-582S CCOC(=O)c1cnc(nc1Oc2cccc(c2)Cl)c3ccccc3 11M-583S c1ccc(cc1)c2ncc(c(n2)Oc3ccccc3)C(=O)O 11M-584S c1ccc(cc1)c2ncc(c(n2)Oc3ccc(cc3)F)C(=O)O 11M-585S c1cc(cc(c1)NC(=O)c2c(cc(=O)n(n2)c3ccc(cc3)Cl)C(F)(F)F)C(F)(F)F 11M-588S c1ccc(cc1)NC(=O)c2c(cc(=O)n(n2)c3ccc(cc3)Cl)C(F)(F)F 11M-589S c1cc(ccc1NC(=O)c2c(cc(=O)n(n2)c3ccc(cc3)Cl)C(F)(F)F)Cl 11M-590S Cc1ccc(cc1)/C=N/NC(=O)COc2ccc(cc2)C(F)(F)F 11M-593S COc1ccc(cc1OC2CCCC2)C(CC(=O)OC)C#N 11M-702 c1cc(c(c(c1)Cl)Cc2c(ccc(c2O)C=O)O)F 11M-703 C/C(=C\C(=O)C(F)(F)F)/Nc1ccccc1O 11M-704 CN(C)/C=C/C(=O)C(Cc1c(cccc1Cl)F)C(=O)c2ccccc2 11M-708 Cc1ccc(cc1)C(=O)Nc2cccc(n2)Nc3c(cc(cn3)C(F)(F)F)Cl 11M-711 Cc1cc(nc(c1C#N)SC(F)F)C 11M-712 c1cc(ccc1CN2CCc3cncn3C2=O)[N+](=O)[O-] 11M-713 C/C(=C/C(=O)C(F)(F)F)/Nc1ccc(cc1)OC 11M-714 CC(=O)CC(=O)NC(=O)C 11M-717 c1cc(c(c(c1)Cl)Cc2c(ccc(c2O)/C=N/CCc3ccc(cc3)S(=O)(=O)N)O)F 11M-719 c1cc(ccc1c2ccnc(n2)[S-])F.[K+] 11M-720 CC(=O)Nc1cccc(n1)NC(=O)C 11M-721 Cc1ccc(cc1)/C=C/C(=O)CCc2c(cccc2Cl)Cl 11M-722 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)S 11M-724 c1cc(ccc1c2ccnc(n2)S)F 11M-725 CN(C)/C=C\C(=C\C(=O)C(F)(F)F)\Nc1ccccc1O 11M-727 c1cc(ccc1N2CC2c3ccncc3)OC(F)(F)F 11M-728 c1cc(ccc1CN2CCc3cncn3C2=O)Br 11M-729 C/C(=C\C(=O)C(F)(F)F)/NOCc1ccc(cc1)F 11M-732 c1cc(ccc1c2ccnc(n2)SC(F)F)F 11M-735 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)SC(F)F 11M-736 C/C(=N\Nc1ccc(cc1)Cl)/CC(=O)C(F)(F)F 11M-739 CC1(CC(=CC(=O)C1)OC(=O)c2ccccc2F)C 11M-901 Cc1ccc(cc1)C(=O)Oc2cc(no2)c3ccccc3 11M-902 c1ccc(cc1)c2cc(on2)OC(=O)c3ccc(cc3)Cl 11M-903 c1ccc(cc1)c2cc(=O)on2C(=O)C3CC3 11M-904 c1ccc(cc1)c2cc(on2)OC(=O)c3ccc(cc3)F 11M-905 Cc1ccc(cc1)C(=O)OC2=CC(=O)CC(C2)(C)C 11M-906 CN(C)/C=C/C(=O)c1ccoc1 11M-908 CC1(CC(=CC(=O)C1)OC(=O)c2ccc(cc2)Cl)C 11M-909 COc1ccc(cc1)N/C=C/C(=O)c2ccoc2 11M-910 c1ccc(cc1)c2cc(on2)OC(=O)c3cccc(c3)C(F)(F)F 11M-911 Cc1c(c(no1)c2ccccc2Cl)C(=O)Oc3cc(no3)c4ccccc4 11M-914 COc1cccc(c1)C(=O)Oc2cc(no2)c3ccccc3 11M-916 c1ccc(cc1)c2cc(=O)on2S(=O)(=O)c3ccc(cc3)Br 11M-917 c1ccc(cc1)c2cc(=O)on2C(=O)c3ccc(cc3Cl)Cl 11M-919 c1ccc(cc1)c2cc(=O)on2C(=O)c3ccccc3Cl 11M-920 c1ccc(cc1)c2cc(=O)on2S(=O)(=O)c3ccc4ccccc4c3 11M-921 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Oc3cc(no3)c4ccccc4 11M-922 c1ccc(cc1)c2cc(=O)on2C(=O)c3c(cccc3Cl)Cl 11M-923 COc1ccc(cc1OC)S(=O)(=O)n2c(cc(=O)o2)c3ccccc3 11M-924 COc1ccc(cc1)S(=O)(=O)n2c(cc(=O)o2)c3ccccc3 11M-925 c1ccc(cc1)c2ccc(cc2)c3ccc4ccccc4c3 11N-001 c1cc(cc(c1)[N+](=O)[O-])/C=N/OC(=O)c2ccco2 11N-002 c1cc(ccc1C(=O)N/N=C/c2cnc(s2)N3CCCCC3)Cl 11N-003 c1cc(cc(c1)[N+](=O)[O-])/C=N/OC(=O)c2c(cccc2F)F 11N-004 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)O/N=C/c3cccc(c3)[N+](=O)[O-] 11N-005 c1cc(cc(c1)[N+](=O)[O-])/C=N\OC(=O)c2ccc(cc2)C(F)(F)F 11N-006 Cc1cccc(c1)C(=O)O/N=C/c2cccc(c2)[N+](=O)[O-] 11N-007 COc1ccc(cc1OC)/C=N\NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl 11N-008 CN(CCO)c1ccccn1 11N-009 c1cc(ccc1/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl)F 11N-011 c1c(sc(n1)N2CCCC2)C=O 11N-012 c1ccc(cc1)Oc2ccccc2C=O 11N-013 CCN(CC)c1ncc(s1)C=O 11N-014 COC(=O)/C=C\1/C(=O)OCCN1 11N-015 c1cc(cc(c1)[N+](=O)[O-])NC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O 11N-017 CCN(CC)c1ncc(s1)C=C2C(=O)OC(OC2=O)(C)C 11N-018 c1ccnc(c1)/C=N/OCc2cnc(s2)Cl 11N-019 Cc1ccc(cc1)CO/N=C/c2cccc(c2)[N+](=O)[O-] 11N-022 c1ccc(cc1)CNC(=O)c2c(c3cccc4c3n(c2=O)CC4)O 11N-023 c1ccc(cc1)CN2CCN(CC2)c3ncc(s3)C=O 11N-024 c1ccc(cc1)Oc2ccccc2/C=C/C(=O)O 11N-025 c1cc(c(c(c1)Cl)COc2ccc(cc2)C(=O)NN)F 11N-026 c1cc2c3c(c1)c(c(c(=O)n3CC2)C(=O)NC45CC6CC(C4)CC(C6)C5)O 11N-027 c1ccc(cc1)C(=O)NCCc2ccccn2 11N-028 c1ccc(cc1)C(=O)N/N=C/c2cnc(s2)N3CCOCC3 11N-029 CC(=O)O/N=C/c1cccc(c1)[N+](=O)[O-] 11N-030 c1cc(cc(c1)[N+](=O)[O-])/C=N/OC(=O)C2CC2 11N-031 CCN(CC)c1ncc(s1)/C=N/NC(=S)N 11N-033 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)Nc4cc(ccc4F)F)O 11N-034 COC(=O)C1=C2C(=O)OCCN2C(=O)CC1 11N-035 CCCNC(=O)c1c(c2cccc3c2n(c1=O)CCC3)O 11N-038 Cc1ccc(cc1)/C=N/NC(=O)c2ccc(cc2)OCc3c(cccc3Cl)F 11N-039 c1ccc(cc1)C/N=C/c2cnc(s2)Cl 11N-040 Cc1cccc(c1C)NC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O 11N-041 CC1CN(CC(O1)C)c2ncc(s2)C=C(C#N)C#N 11N-042 c1cc(sc1)C(=O)O/N=C(/c2ccc(cc2)OCc3cnc(s3)Cl)\N 11N-043 c1cc(cc(c1)Br)/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl 11N-044 c1cc(cc(c1)[N+](=O)[O-])/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl 11N-045 COc1ccc(cc1)Oc2ccccc2C=O 11N-047 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)c4ccc(cc4)NC(=O)c5c(c6cccc7c6n(c5=O)CCC7)O 11N-048 CCN(CC)c1ncc(s1)C=C2C(=O)N(C(=O)N(C2=O)C)C 11N-049 c1ccc(c(c1)C=O)Oc2ccc(cc2)Cl 11N-050 COC(=O)/C=C\1/C(=O)OCC(N1)Cc2ccccc2 11N-051 c1ccc(cc1)Oc2ccccc2/C=N/NC(=O)c3ccc(cc3)OCc4ccc(c(c4)Cl)Cl 11N-053 c1cc(cc(c1)[N+](=O)[O-])/C=N/OCc2ccc(cc2Cl)Cl 11N-054 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)Nc4c(c(c(c(c4F)F)F)F)F)O 11N-055 c1cc(cc(c1)[N+](=O)[O-])/C=N/OC(=O)Nc2cccc(c2)Cl 11N-056 COc1cc2c(cc1OC)ncnc2Nc3ccccc3 11N-058 COc1cc2c(cc1OC)ncnc2Nc3ccccc3Cl 11N-059 Cc1ccc(cc1C)Nc2c3cc(c(cc3ncn2)OC)OC 11N-060 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3F)F 11N-061 c1cc2c3c(c1)c(c(c(=O)n3CC2)C(=O)Nc4c(cccc4Br)Br)O 11N-062 COCCCNCc1cnc(s1)Cl 11N-063 COC(=O)C1=C2C(=O)OCC(N2C(=O)CC1)Cc3ccccc3 11N-064 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3)OC(F)(F)F 11N-065 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3)Br 11N-066 Cc1ccc(c(c1)C)Nc2c3cc(c(cc3ncn2)OC)OC 11N-068 Cc1cc(ccc1Nc2c3cc(c(cc3ncn2)OC)OC)OC 11N-069 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3)I 11N-070 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)Nc4ccc(cc4)I)O 11N-071 CCONc1c2cc(c(cc2ncn1)OC)OC 11N-072 c1cc(cc(c1)[N+](=O)[O-])/C=N/OC(=O)Nc2ccc(c(c2)Cl)Cl 11N-075 CC(C)c1ccc(cc1)Nc2c3cc(c(cc3ncn2)OC)OC 11N-076 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3Cl)Cl 11N-078 COc1cc2c(cc1OC)ncnc2Nc3ccc4c(c3)OCO4 11N-079 Cc1c(cccc1Cl)Nc2c3cc(c(cc3ncn2)OC)OC 11N-080 COc1cc2c(cc1OC)ncnc2Nc3c(cccc3F)F 11N-081 c1cc(cc(c1)[N+](=O)[O-])/C=N/Oc2c(cccn2)[N+](=O)[O-] 11N-082 c1c(sc(n1)Cl)/C=N/O 11N-083 COc1cc2c(cc1OC)ncnc2Nc3ccc(c(c3)Cl)Cl 11N-084 Cc1cccc(c1C)Nc2c3cc(c(cc3ncn2)OC)OC 11N-085 COc1ccc(c(c1)OC)Nc2c3cc(c(cc3ncn2)OC)OC 11N-086 Cc1cc(ccc1Nc2c3cc(c(cc3ncn2)OC)OC)Cl 11N-089 Cc1ccc(c(c1)Nc2c3cc(c(cc3ncn2)OC)OC)C 11N-090 c1ccc(cc1)N2CCN(CC2)c3ncc(s3)C=O 11N-091 CCN(CC)c1ncc(s1)/C=N/NC(=O)c2ccncc2 11N-092 Cc1ccc(cc1)Oc2ccccc2C=O 11N-093 c1ccc(cc1)NC(=O)O/N=C/c2cccc(c2)[N+](=O)[O-] 11N-094 Cc1ccc(cc1)NC(=O)O/N=C/c2cccc(c2)[N+](=O)[O-] 11N-095 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3)N4CCOCC4 11N-096 COc1cc(ccc1O)/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl 11N-097 c1cc(cc(c1)F)CO/N=C/c2cccc(c2)[N+](=O)[O-] 11N-098 CC(=O)Nc1ccc(cc1)c2[nH]c(c(n2)c3ccccc3)c4ccccc4 11N-099 COc1cc2c(cc1OC)ncnc2NCc3ccc(cc3)Cl 11N-100 c1cc(ccc1Cc2ccncc2)[N+](=O)[O-] 11N-102 COc1cc2c(cc1OC)ncnc2NCc3ccc(cc3Cl)Cl 11N-103 COc1cc2c(cc1OC)ncnc2NCc3ccccc3 11N-104 COc1cccc(c1)CNc2c3cc(c(cc3ncn2)OC)OC 11N-105 COc1cc2c(cc1OC)ncnc2NCc3ccc(cc3)F 11N-106 COc1cc2c(cc1OC)ncnc2NCc3ccccc3C(F)(F)F 11N-109 COc1cc2c(cc1OC)ncnc2NCc3ccccc3F 11N-110 Cc1ccccc1CNc2c3cc(c(cc3ncn2)OC)OC 11N-111 COc1cc2c(cc1OC)ncnc2Nc3cccc(c3)F 11N-112 c1ccc(c(c1)N2CCN(CC2)Cc3cnc(s3)Cl)F 11N-113 Cc1ccc(cc1)CNc2c3cc(c(cc3ncn2)OC)OC 11N-114 COc1cc2c(cc1OC)ncnc2NCc3ccco3 11N-115 COc1cc2c(cc1OC)ncnc2NCCc3ccccc3 11N-116 COc1ccc(cc1OC)CC/N=C/c2cnc(s2)Cl 11N-118 Cc1ccc(c(c1)C)OCc2cnc(s2)Cl 11N-119 Cc1ccc(cc1)/C=N/NC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O 11N-120 c1cc(ccc1C(=O)N/N=C/c2c(c(c(c(c2F)F)F)F)F)OCc3ccc(c(c3)Cl)Cl 11N-121 c1cc(oc1)/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl 11N-122 CN1c2ccsc2/C(=N/NC(=O)c3cccc(c3)C(F)(F)F)/CS1(=O)=O 11N-301S CN1c2ccsc2/C(=N/NC(=O)c3ccc(cc3)F)/CS1(=O)=O 11N-302S CN1c2ccsc2/C(=N/NC(=O)c3c(cccc3F)F)/CS1(=O)=O 11N-304S CN1c2ccsc2/C(=N/NC(=O)c3ccc(cc3)Cl)/CS1(=O)=O 11N-305S CCOC(=O)C1=C(OC2=C(C1c3ccc(cc3)Cl)C(=O)CCC2)N 11N-322S c1cc(c(cc1Cl)Cl)C2C(=C(OC3=C2C(=O)CCC3)N)C#N 11N-323S CCOC(=O)C1=C(OC2=C(C1c3ccc(cc3Cl)Cl)C(=O)CCC2)N 11N-324S CCCC(=O)N/N=C/1\CS(=O)(=O)N(c2c1scc2)C 11N-325S CN1c2ccsc2/C(=N/NC(=O)Cc3cccs3)/CS1(=O)=O 11N-326S Cc1cccc(c1)C(=O)N/N=C/2\CS(=O)(=O)N(c3c2scc3)C 11N-328S c1cc(c(c(c1)Cl)CN2c3cc(ccc3SCCC2=O)Cl)Cl 11N-329S c1cc(c(c(c1)Cl)CN2c3cc(ccc3SCCC2=O)Cl)F 11N-330S Cc1cccc(c1)CN2c3cc(ccc3SCCC2=O)Cl 11N-331S CCN1c2cc(ccc2SCCC1=O)Cl 11N-332S CCOC(=O)CN1c2cc(ccc2SCCC1=O)Cl 11N-333S C#CCN1c2cc(ccc2SCCC1=O)Cl 11N-334S COc1ccc(cc1)C(=O)CN2c3cc(ccc3SCCC2=O)Cl 11N-336S c1cc2c(cc1Cl)NC(=S)CCS2 11N-337S CCOC(=O)c1cc2c3ccccc3n(c2s1)C 11N-339S Cn1c2ccccc2c3c1sc(c3)C(=O)NN 11N-340S Cn1c2ccccc2c3c1sc(c3)C(=O)OC 11N-341S c1ccc(cc1)CSC2=Nc3cc(ccc3SCC2)Cl 11N-342S CCCN1c2cc(ccc2SCCC1=O)Cl 11N-343S CCOC(=O)C1=C(OC2=C(C1c3ccc(cc3)OC)C(=O)CCC2)N 11N-346S C=CCN1c2cc(ccc2SCCC1=O)Cl 11N-350S Cc1ccc(cc1)CSC2=Nc3cc(ccc3SCC2)Cl 11N-351S c1ccc(c(c1)CSC2=Nc3cc(ccc3SCC2)Cl)Cl 11N-352S CSc1nc2c(c(n1)OC(=O)c3ccc(cc3)Cl)CCCC2 11N-353S CC(C)(C)C(=O)Oc1c2c(nc(n1)SC)CCCC2 11N-354S CSc1nc2c(c(n1)OC(=O)c3ccccc3Cl)CCCC2 11N-355S CSc1nc2c(c(n1)OC(=O)c3cccs3)CCCC2 11N-356S CSc1nc2c(c(n1)OC(=O)c3cccc(c3)Cl)CCCC2 11N-357S Cc1cccc(c1)C(=O)Oc2c3c(nc(n2)SC)CCCC3 11N-358S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)Br)Br 11N-359S c1cc(ccc1C(=O)Cn2c(=O)c(c(cn2)Br)Br)Cl 11N-360S CO/N=C(\Cn1c(=O)c(c(cn1)Br)Br)/c2ccc(cc2)Cl 11N-361S CC(=O)Cn1c(=O)c(c(cn1)NC)Br 11N-362S CC(=O)Cn1c(=O)c(c(cn1)NC)Cl 11N-363S CC(=O)Cn1c(=O)c(c(cn1)NCC=C)Cl 11N-364S COc1ccc(cc1)Oc2c3c(nc(n2)SC)CCCC3 11N-365S CCOC(=O)C1=C(OC2=C(C1c3ccccc3Cl)C(=O)CCC2)N 11N-366S CCOC(=O)C1=C(OC2=C(C1c3ccc(cc3)[N+](=O)[O-])C(=O)CCC2)N 11N-367S CN1c2ccsc2C(=C(S1(=O)=O)C(=O)Nc3ccccc3)O 11N-370S c1cc(ccc1C(=O)Cn2c(=O)c(c(cn2)Cl)Cl)Cl 11N-372S CO/N=C(\Cn1c(=O)c(c(cn1)Cl)Cl)/c2ccc(cc2)Cl 11N-373S c1cc(ccc1C(=O)Cn2c(=O)c(c(cn2)N3CCOCC3)Br)Cl 11N-374S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)N2CCOCC2)Br 11N-375S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)N2CCOCC2)Cl 11N-376S CO/N=C(\Cn1c(=O)c(c(cn1)N2CCOCC2)Br)/c3ccc(cc3)Cl 11N-377S CCOC(=O)C1=C(OC2=C(C1c3ccccc3)C(=O)CCC2)N 11N-378S CCOC(=O)C1=C(OC2=C(C1c3c(cccc3Cl)F)C(=O)CCC2)N 11N-379S CN1c2ccsc2C(=C(S1(=O)=O)C(=O)Nc3cccc(c3)C(F)(F)F)O 11N-380S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)c4c(cccc4F)F 11N-382S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)c4ccccc4 11N-383S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)c4ccc(cc4)F 11N-384S CC(=O)NNC(=O)c1cc2c3ccccc3n(c2s1)C 11N-385S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)CCl 11N-386S c1ccc(cc1)SCC2CSc3n2c(=O)c4ccccc4n3 11N-387S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccc(cc4)Cl 11N-388S CC(C)(C)c1ccc(cc1)CSC2=Nc3cc(ccc3SCC2)Cl 11N-389S c1cc(ccc1CSC2=Nc3cc(ccc3SCC2)Cl)Cl 11N-390S c1cc(ccc1CSC2=Nc3cc(ccc3SCC2)Cl)F 11N-391S c1cc(cc(c1)Cl)CSC2=Nc3cc(ccc3SCC2)Cl 11N-392S c1cc(cc(c1)C(F)(F)F)CSC2=Nc3cc(ccc3SCC2)Cl 11N-393S Cc1cccc(c1)CSC2=Nc3cc(ccc3SCC2)Cl 11N-394S CC(C)(C)C(=O)NNC(=O)c1cc2c3ccccc3n(c2s1)C 11N-395S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)c4cccc(c4)C(F)(F)F 11N-396S Cc1ccccc1C(=O)NNC(=O)c2cc3c4ccccc4n(c3s2)C 11N-397S Cc1cccc(c1)C(=O)NNC(=O)c2cc3c4ccccc4n(c3s2)C 11N-398S Cc1ccc(cc1)C(=O)NNC(=O)c2cc3c4ccccc4n(c3s2)C 11N-399S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)c4cccs4 11N-400S CN1c2ccsc2C(=C(S1(=O)=O)C(=O)Nc3ccc(cc3)Cl)O 11N-401S Cc1ccc(cc1)NC(=O)C2=C(c3c(ccs3)N(S2(=O)=O)C)O 11N-402S Cc1cccc(c1NC(=O)C2=C(c3c(ccs3)N(S2(=O)=O)C)O)C 11N-403S CN1c2ccsc2C(=C(S1(=O)=O)C(=O)Nc3ccc(cc3)F)O 11N-404S CN1c2ccsc2C(=C(S1(=O)=O)C(=O)Nc3ccc(c(c3)Cl)Cl)O 11N-405S CN1c2ccsc2C(=C(S1(=O)=O)C(=S)Nc3ccccc3)O 11N-406S CC(=O)Cn1c(=O)c(c(cn1)N(C)C)Cl 11N-407S CCN(CC)c1cnn(c(=O)c1Cl)CC(=O)C 11N-408S CC(=O)Cn1c(=O)c(c(cn1)NC2CCCCC2)Cl 11N-409S CC(=O)Cn1c(=O)c(c(cn1)NC2CC2)Cl 11N-410S C=CCNc1cnn(c(=O)c1Cl)CC(=O)c2ccc(cc2)Cl 11N-411S c1cc(ccc1C(=O)Cn2c(=O)c(c(cn2)N3CCOCC3)Cl)Cl 11N-412S c1cc(ccc1C(=O)Cn2c(=O)c(c(cn2)N3CCCC3)Cl)Cl 11N-413S CO/N=C(\Cn1c(=O)c(c(cn1)N2CCOCC2)Cl)/c3ccc(cc3)Cl 11N-414S CO/N=C(\Cn1c(=O)c(c(cn1)N2CCCC2)Cl)/c3ccc(cc3)Cl 11N-415S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)N2CCCC2)Br 11N-416S c1cc(ccc1C(=O)Cn2c(=O)c(c(cn2)N3CCCC3)Br)Cl 11N-417S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccc(cc4Cl)Cl 11N-420S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccc(cc4)F 11N-421S Cc1c(c(n(n1)C)Cl)C(=O)OC 11N-503S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C(=O)O)Cl 11N-505S CC(C)(C)NC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccc(cc2)Cl 11N-510S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C(=O)N3CCCCC3)Cl 11N-511S CN(C)C(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccc(cc2)Cl 11N-512S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C(=O)N3CCOCC3)Cl 11N-513S Cc1cc(nc2c1c(c(s2)C(=O)OC)N)C 11N-515S c1ccc2c(c1)c(nc3n2ncc3C#N)N4CCCCC4 11N-519S c1ccc2c(c1)c(nc3n2ncc3C#N)N4CCOCC4 11N-520S COC(=O)CSc1ccc(cc1[N+](=O)[O-])C(=O)OC 11N-522S COC(=O)c1ccc2c(c1)NC(=O)CS2 11N-523S CN1c2cc(ccc2SCC1=O)C(=O)OC 11N-524S CN1c2cc(ccc2SCC1=O)C(=O)O 11N-526S COC(=O)c1ccc2c(c1)N(C(=O)CS2)Cc3ccc(cc3)Cl 11N-527S COC(=O)c1ccc2c(c1)N(C(=O)CS2)Cc3cccc(c3)C(F)(F)F 11N-528S c1ccc2c(c1)CCCC(=O)N2Cc3ccc(cc3)F 11N-562S Cc1c(c(n(n1)C)Cl)/C=N/OC(=O)c2ccccc2 11N-565S Cc1c(c(n(n1)C)Cl)/C=N/OC(=O)c2ccc(cc2)F 11N-566S Cc1c(c(n(n1)C)Cl)/C=N/OC(=O)c2cccc(c2)C(F)(F)F 11N-567S Cc1c(c(n(n1)C)Cl)/C=N/OC(=O)c2ccc(nc2)Cl 11N-569S Cc1c(c(n(n1)C)Cl)/C=N/OC(=O)c2c(cccc2F)F 11N-570S Cc1ccc(cc1)C(=O)O/N=C/c2c(nn(c2Cl)C)C 11N-571S Cc1c(c(n(n1)C)Cl)C(=O)N 11N-575S Cc1c(c(n(n1)C)Sc2ccc(cc2)Cl)C(=O)N 11N-576S c1ccc2c(c1)CCCC(=O)N2Cc3c(cccc3Cl)F 11N-578S Cc1c(c(n(n1)C)Cl)/C=N/OC(=O)c2ccc(cc2)[N+](=O)[O-] 11N-579S Cc1c(c(n(n1)C)Cl)C#N 11N-580S COc1ccc(cc1)CN2c3ccccc3CCCC2=O 11N-581S c1ccc2c(c1)CCCC(=O)N2Cc3cccc(c3)Cl 11N-582S CC(C)(C)c1ccc(cc1)CN2c3ccccc3CCCC2=O 11N-583S CCN1c2ccccc2CCCC1=O 11N-585S c1ccc2c(c1)CCCC(=O)N2Cc3ccc(c(c3)Cl)Cl 11N-586S Cc1cccc(c1)CN2c3ccccc3CCCC2=O 11N-587S c1ccc2c(c1)CCCC(=O)N2Cc3ccc(cc3)Cl 11N-588S c1ccc2c(c1)CCCC(=O)N2Cc3cccc(c3)F 11N-590S c1ccc2c(c1)CCCC(=O)N2Cc3ccccc3Cl 11N-593S c1ccc2c(c1)CCCC(=O)N2Cc3ccc(cc3Cl)Cl 11N-594S c1ccc2c(c1)CCCC(=O)N2Cc3c(cccc3Cl)Cl 11N-595S Cc1ccccc1CN2c3ccccc3CCCC2=O 11N-596S CSc1nc(cc(n1)Sc2ccc(cc2)F)C(F)(F)F 11N-644S CSc1nc(cc(n1)Oc2ccc(cc2)F)C(F)(F)F 11N-646S CSc1nc(cc(n1)Oc2ccc(cc2F)F)C(F)(F)F 11N-647S COC(=O)c1c(ccs1)Oc2cc(nc(n2)SC)C(F)(F)F 11N-648S CSc1nc(cc(n1)Oc2cccc(c2)C(F)(F)F)C(F)(F)F 11N-649S Cc1ccc(cc1)Oc2cc(nc(n2)SC)C(F)(F)F 11N-651S CSc1nc(cc(n1)Oc2ccc(cc2)[N+](=O)[O-])C(F)(F)F 11N-652S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)OC 11N-654S CSc1nc(cc(n1)Oc2ccncc2)C(F)(F)F 11N-655S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)O 11N-656S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)N3CCOCC3 11N-658S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)NC3CC3 11N-659S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)NC3CCCCC3 11N-660S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)NC(C)C 11N-661S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)NCC=C 11N-662S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)N(C)C 11N-663S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CO 11N-664S COC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2 11N-665S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)Nc3cccc(c3)C(F)(F)F 11N-666S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)Nc3ccc(cc3)OC 11N-667S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)Nc3ccc(cc3)F 11N-668S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)O 11N-670S Cc1cccc(c1C)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 11N-671S COc1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 11N-672S Cc1ccccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 11N-673S c1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 11N-674S CCc1cccc(c1NC(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)CC 11N-675S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)N3CCOCC3 11N-678S C=CCNC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2 11N-679S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)NC3CCCCC3 11N-680S CC(C)(C)NC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2 11N-681S CC(C)NC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2 11N-682S COc1ccc(c(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccccc3)OC 11N-683S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)Nc3ccc(cc3F)F 11N-684S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)Nc3cccc(c3)C(F)(F)F 11N-685S COc1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccccc3 11N-686S Cc1ccc(cc1)Sc2cc(nc(n2)SC)C(F)(F)F 11N-687S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)c3ccc(cc3)Cl 11N-689S c1cc(c(nc1)Sc2nnc(s2)SCCCF)[N+](=O)[O-] 11N-700 C1CCC(C1)Sc2nnc(s2)SC3CCCC(=O)C3 11N-701 c1c[n+](cn1O)[O-] 11N-702 c1ccc(cc1)CSc2nnc(s2)S 11N-703 c1ccc(cc1)CC(CO)n2ccc(c(c2=O)Cc3ccc(cc3)F)O 11N-705 c1cc(cc(c1)Cl)Cn2ccc(c(c2=O)Cc3ccc(cc3)F)O 11N-706 Cc1[nH+]c(cs1)C(=O)C.[Br-] 11N-708 c1ccc(cc1)OCCSc2nnc(s2)S 11N-710 Cc1ccc(cc1)c2n(cc[n+]2[O-])O 11N-711 c1cc(oc1)Cn2ccc(c(c2=O)Cc3ccc(cc3)F)O 11N-712 Cc1ccc(cc1)Cn2cc(c(c(c2=O)Cc3ccc(cc3)F)O)/C=N/OCc4ccc(cc4Cl)Cl 11N-713 c1cc(ccc1Cc2c(ccn(c2=O)C3CCCCC3)O)F 11N-716 c1ccc(cc1)OCCSc2nnc(s2)SCC(=O)c3ccc(cc3)Cl 11N-719 c1ccc(cc1)C(=O)Sc2nnc(s2)SCCOc3ccccc3 11N-720 COc1ccccc1Cn2ccc(c(c2=O)Cc3ccc(cc3)F)O 11N-721 c1ccc(cc1)COn2ccnc2 11N-722 c1ccc(cc1)CSc2nnc(s2)SC(C(=O)O)(F)F 11N-724 c1([nH]nc(n1)Br)Br 11N-725 C=CCOn1ccnc1 11N-729 CN(C)C(=O)Sc1nnc(s1)SCCOc2ccccc2 11N-730 c1cc(c(cc1COn2ccnc2)Cl)Cl 11N-732 c1cc(ccc1N2C(=O)CC(C2=O)Sc3c(cc(cn3)C(F)(F)F)Cl)Cl 11N-733 c1cc(ncc1[N+](=O)[O-])Sc2nccn2c3c(cc(cn3)C(F)(F)F)Cl 11N-734 Cc1ccc(cc1)C(=O)CSc2nccn2c3c(cc(cn3)C(F)(F)F)Cl 11N-735 COC(=O)COc1ccc(c(c1Cc2c(cccc2Cl)F)OCC(=O)OC)C=O 11N-739 CCOC(=O)CSc1nnc(s1)SCCN2C(=O)c3ccccc3C2=O 11N-744 c1c(cnc(c1Cl)Sc2nnc(s2)Sc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 11N-745 CC(C)CSc1nnc(s1)Sc2c(cccn2)[N+](=O)[O-] 11N-746 CCOC(=O)C(Cc1c(cccc1Cl)F)C(=O)C 11N-747 c1cc(ccc1C(=O)CSc2nccn2c3c(cc(cn3)C(F)(F)F)Cl)Br 11N-753 Cc1ccc(cc1)/C(=N\O)/CSc2nccn2c3c(cc(cn3)C(F)(F)F)Cl 11N-755 CC(C)Oc1ccc(c(c1Cc2c(cccc2Cl)F)OC(C)C)/C=C(\C#N)/S(=O)(=O)c3ccccc3 11N-756 c1cc(c(c(c1)Cl)Cc2c(ccc(c2O)C=O)OC3CCCC3)F 11N-757 c1cc(ccc1COn2ccnc2)C(F)(F)F 11N-760 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)Cc3ccc(cc3)F)O)F 11N-762 c1ccc(cc1)Cn2c(nc(n2)Br)Br 11N-763 c1cc(c(cc1Cl)Cl)COn2ccnc2 11N-765 COc1ccc(cc1OC)CCn2ccc(c(c2=O)Cc3c(cccc3Cl)F)O 11N-767 CCOC(=O)C(Cc1c(cccc1Cl)F)c2ccnc3n2nc(n3)N 11N-768 COc1ccc(cc1OC)CCn2ccc(c(c2=O)Cc3ccc(cc3)Cl)O 11N-801 CC(=O)C(=Cc1ccc(cc1)[N+](=O)[O-])C(=O)C 11N-802 c1ccc(c(c1)Nc2c3ccc(cc3ncn2)Cl)Cl 11N-807 c1cc(cc(c1)Cl)Nc2c3ccc(cc3ncn2)Cl 11N-808 c1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)Cl 11N-809 C=CCn1ccc(c(c1=O)Cc2ccc(cc2)Cl)O 11N-810 CC1=C(C(n2c(ncn2)N1)c3ccc(cc3)[N+](=O)[O-])C(=O)C 11N-811 c1ccc(cc1)Nc2c3ccc(cc3ncn2)Cl 11N-813 c1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)F 11N-814 c1cc(c(cc1F)F)Nc2c3ccc(cc3ncn2)Cl 11N-815 c1cc2c(cc1Cl)ncnc2Nc3ccc(cc3Cl)Cl 11N-820 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3)F 11N-821 CCOC(CCn1ccc(c(c1=O)Cc2ccc(cc2)Cl)O)OCC 11N-822 Cc1ccc(cc1C)Nc2c3ccc(cc3ncn2)Cl 11N-823 c1ccc(cc1)Oc2ccc(cc2)Nc3c4ccc(cc4ncn3)Cl 11N-824 CC(=O)C(=Cc1ccc(c(c1)OC)O)C(=O)C 11N-825 c1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)Br 11N-826 c1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)OC(F)(F)F 11N-827 c1cc(ccc1Cc2c(ccn(c2=O)Cc3ccncc3)O)Cl 11N-828 CC(=O)C(=Cc1ccc2c(c1)OCO2)C(=O)C 11N-831 CN(C)/C=N/c1cc(ccc1C(=O)O)Cl 11N-832 c1cc(c(cc1Nc2c3ccc(cc3ncn2)Cl)Cl)Cl 11N-833 COc1ccc(c(c1)OC)Nc2c3ccc(cc3ncn2)Cl 11N-834 CC(C)c1ccc(cc1)Nc2c3ccc(cc3ncn2)Cl 11N-835 Cc1ccc(c(c1)C)Nc2c3ccc(cc3ncn2)Cl 11N-836 c1cc(c(c(c1)F)Nc2c3ccc(cc3ncn2)Cl)F 11N-837 CC1=C(C(n2c(ncn2)N1)c3ccc4c(c3)OCO4)C(=O)C 11N-838 CC1=C(C(n2c(ncn2)N1)c3ccc(c(c3)OC)O)C(=O)C 11N-839 c1cc(sc1)Cn2ccc(c(c2=O)Cc3ccc(cc3)Cl)O 11N-841 c1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)N4CCOCC4 11N-842 c1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)I 11N-843 c1cc2c(cc1Cl)ncnc2Cl 11N-844 COc1cc(cc(c1)OC)Nc2c3ccc(cc3ncn2)Cl 11N-846 c1cc(cc(c1)F)Nc2c3ccc(cc3ncn2)Cl 11N-847 c1cc2c(cc1Nc3c4ccc(cc4ncn3)Cl)OCO2 11N-848 Cc1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)OC 11N-849 Cc1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)Cl 11N-850 Cc1ccc(c(c1)Nc2c3ccc(cc3ncn2)Cl)C 11N-851 CCOC(=O)C(=Cc1cccc(c1)C#N)C#N 11N-903 c1cc(cc(c1)c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N)C#N 11N-909 COC(=O)C1CCN(CC1)C(=O)c2cccc(c2)[N+](=O)[O-] 11N-917 COC(=O)C1CCN(CC1)C(=O)c2ccc(cc2)Cl 11N-918 COc1ccc(cc1)C(=O)N2CCC(CC2)C(=O)OC 11N-919 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)OC 11N-921 COC(=O)C1CCN(CC1)C(=O)CCC(=O)O 11N-923 c1cc(ccc1C(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-] 11N-927 Cc1ccc(cc1)CN2CCC(CC2)C(=O)OC 11N-930 c1cc(ccc1C(=O)N2CCC(CC2)C(=O)N)[N+](=O)[O-] 11N-931 COC(=O)C1CCN(CC1)C(=O)/C=C/C(=O)O 11N-932 c1cc(ccc1C(=O)N2CCC(CC2)C#N)[N+](=O)[O-] 11N-933 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)O 11N-934 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)N 11N-936 CC(C)(C)c1cc(c(c(c1)C=O)O)C=O 11N-950 CC(C)(C)c1ccc(c(c1)C=O)O 11N-951 c1c(cc(c(c1C=O)O)C=O)Cl 11N-952 CC(C)(C)c1ccc(c(c1)/C=N\O)O 11N-953 CC(c1cc(c(c(c1)/C=N\O)O)/C=N\O)(C)C 11N-954 CC(C)(C)c1cc(c(c(c1)C#N)O)C#N 11N-960 Cc1cc(c(c(c1)C=O)O)C=O 11N-961 Cc1cc(c(c(c1)/C=N/O)O)/C=N/O 11N-966 CC(C)(C)c1cc(c(c(c1)C#N)OCc2ccc(cc2)C(F)(F)F)C#N 11N-971 CC(C)(C)c1cc(c(c(c1)C(=O)O)O)C(=O)O 11N-975 c1cc(ccc1c2nccc(n2)c3ccc(cc3Cl)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 11P-001 COc1ccc(cc1)C(=O)CSc2nnc(o2)c3ccco3 11P-003 c1ccc(cc1)C(=O)CSc2nnc(o2)c3ccco3 11P-004 c1ccc(c(c1)C(=O)CSc2nnc(o2)c3ccco3)Cl 11P-005 c1ccc(cc1)OCCSc2nnc(o2)c3ccco3 11P-006 c1ccc(cc1)CCNc2ccc(cc2Br)[N+](=O)[O-] 11P-007 CC(C(=O)OC)Oc1ccc(cc1)c2nccc(n2)c3cccs3 11P-009 CC(c1ccn(n1)S(=O)(=O)c2ccc(cc2)OC)Oc3ccc(c(c3)F)c4ccccc4 11P-011 c1cc(c(cc1[N+](=O)[O-])Br)n2ccnc2 11P-014 Cc1ccc(c(c1)/C=C/c2nnc(o2)C)C 11P-015 Cc1ccc(cc1)C(=O)n2ccc(n2)C(C)Oc3ccc(c(c3)F)c4ccccc4 11P-016 Cc1cccc(c1)CSc2nnc(o2)c3ccco3 11P-017 CC(c1ccn(n1)C(=O)c2ccc(cc2)Cl)Oc3ccc(c(c3)F)c4ccccc4 11P-018 Cn1cccc1c2nnc(o2)S 11P-019 CC(=O)NC1c2ccccc2-c3c1cccn3 11P-022 CC(C)(C)OC(=O)CSCC(C(=O)O)NC(=O)OC(C)(C)C 11P-023 CC(C)(C)OC(=O)CSc1nnc(o1)c2ccco2 11P-024 c1cc(ccc1c2nccc(n2)c3ccc(cc3)Br)OCCCF 11P-025 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCCOCCOc4ccc(cc4)F 11P-027 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OCCCF 11P-029 CC(c1ccn(n1)C(=O)c2ccco2)Oc3ccc(c(c3)F)c4ccccc4 11P-030 COc1ccc(cc1)C2=Nn3c(nnc3SC2)c4ccco4 11P-032 c1ccc(cc1)C2=Nn3c(nnc3SC2)c4ccco4 11P-033 c1cc(ccc1c2nccc(n2)c3ccc(cc3)Cl)O 11P-034 CCOC(=O)/C(=N\Nc1ccccc1[N+](=O)[O-])/Cl 11P-035 c1cc(ccc1c2nccc(n2)c3ccc(cc3)F)OCCCF 11P-036 COc1ccc(cc1)c2nnc(o2)S 11P-037 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)c4ccc(cc4)OCCCF 11P-038 CCC(=O)NC1=C(Cc2c1cccc2)C3=CCc4c3cccc4 11P-039 CC(=O)NC1=C(c2ccccc2C1)C3=Cc4ccccc4C3 11P-040 c1ccc(cc1)C2(c3ccccc3-c4c2cccn4)O 11P-042 CCOC(=O)C1(CC(=C(CC1C(=O)OC(C)(C)C)C)C)C(=O)OCC 11P-043 Cn1cccc1c2nnc(o2)SCc3ccc(cc3)Br 11P-044 Cc1ccccc1CSc2nnc(o2)c3cccc(c3)OCc4ccc(cc4Cl)Cl 11P-046 CCCCCc1ccc(cc1)c2ccc(cc2)CC(=O)OC 11P-049 CCOC(=O)/C(=N\Nc1ccccc1[N+](=O)[O-])/N 11P-053 c1cc\2c(nc1)-c3ccc(cc3/C2=N\O)[N+](=O)[O-] 11P-054 c1cc(ccc1C=O)OCCCF 11P-060 CCOC(=O)C(CSCC(=O)NCCc1ccccc1)NC(=O)OC(C)(C)C 11P-061 COc1ccc(cc1)c2nnc(o2)SCC(=O)c3ccc(cc3)OC 11P-062 COc1ccc(cc1)c2nnc(o2)SCCCF 11P-063 COc1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)C(F)(F)F 11P-064 CCOC(=O)CN1CCS(=O)(=O)CC1 11P-0640 COc1ccc(cc1)c2nnc(o2)SCC(=O)c3ccc(cc3Cl)Cl 11P-066 COc1ccc(cc1)c2nnc(o2)SCc3ccc(cc3Cl)Cl 11P-067 CCOC(=O)COc1ccc(cc1)c2nccc(n2)c3ccc(cc3)Cl 11P-068 c1cc(ccc1c2nccc(n2)c3ccc(cc3)Cl)OCCCF 11P-069 c1ccc2c(c1)-c3ccccc3C2=NN 11P-072 Cc1ccc(cc1)/C(=N/NC(=O)N)/C 11P-074 c1cc(c(cc1N)Br)N2CCOCC2 11P-075 COC(=O)COc1ccc(cc1)c2nccc(n2)c3ccc(cc3)Br 11P-079 c1ccc(cc1)c2nnc(o2)SCc3cccc(c3)F 11P-081 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCc4[nH]nnn4 11P-082 CCOC(=O)C1(CC1c2ccc(cc2)Cl)C(=O)OCC 11P-083 CCOC(=O)C(CSC(=O)CCC(=O)NCCc1ccccc1)NC(=O)OC(C)(C)C 11P-085 CCOC(=O)C(CS)NC(=O)OCc1ccccc1 11P-086 c1cc(ccc1c2nccc(n2)c3ccc(cc3Cl)Cl)Oc4cc(cc(n4)C(F)(F)F)C(F)(F)F 11P-091 CCCCCCCc1ccc(cc1)/C=C\2/C(=O)NC(=O)S2 11P-094 c1cc2c(cc[nH]2)c(c1)OCCOCCOc3ccc(cc3)F 11P-097 CCOC(=O)C(CSC(=O)Cc1ccccc1)[NH3+].C(=O)(C(F)(F)F)[O-] 11P-098 CCCCCCCc1ccc(cc1)/C=N/c2ccc(cc2)C(=O)OCC 11P-102 CCCCCCCc1ccc(cc1)CNc2ccc(cc2)C(=O)OCC 11P-106 CCOC(=O)C(=Cc1ccc(cc1)OC)C(=O)OCC 11P-107 c1cc(ccc1C(=O)CSc2nnc(o2)c3ccncc3)Cl 11P-109 c1cc(c(c(c1)Cl)CSc2nnc(o2)c3ccncc3)F 11P-110 CCOC(=O)C(CSC(=O)c1ccc(cc1)[N+](=O)[O-])[NH3+].C(=O)(C(F)(F)F)[O-] 11P-111 CC(C(=O)OC)Oc1ccc(cc1)c2nccc(n2)c3ccc(cc3)F 11P-114 CC1=C(CC(=C(C1)C(=O)OC)C(=O)OC)C 11P-115 COC(=O)CCCOc1ccc(cc1)c2nccc(n2)c3ccc(cc3)F 11P-116 CC(C)(C)c1ccc(cc1)C(=O)NN 11P-118 COc1ccc(cc1)c2nnc3n2N=C(CS3)c4ccc(cc4Cl)Cl 11P-121 COc1cccc(c1Br)F 11P-122 c1cnccc1c2nnc(o2)SCC#N 11P-124 c1cc(ccc1Oc2ccc(cc2Br)[N+](=O)[O-])F 11P-125 Cc1ccc(cc1)S(=O)(=O)n2ccc-3c2CCc4c3nc(s4)CN5CCN(CC5)c6ccccc6OC 11P-128 c1ccc(c(c1)/C=C/2\C(=O)NC(=O)S2)Oc3ccc(cc3Cl)Cl 11P-129 c1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)Oc3ccc(cc3)Cl 11P-130 c1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)Oc3ccc(cc3Cl)Cl 11P-131 c1ccc(c(c1)/C=C\2/C(=O)NC(=O)S2)Oc3ccc(cc3F)Br 11P-132 c1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)Oc3ccc(cc3)F 11P-133 c1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)Oc3ccc(cc3F)Br 11P-135 c1cc(ccc1CSc2nnc(o2)c3ccncc3)[N+](=O)[O-] 11P-136 CCCCCCCc1ccc(cc1)C=C2C(=O)NC(=O)NC2=O 11P-139 c1cc(c(cc1[N+](=O)[O-])Br)N2CCC(CC2)C(=O)O 11P-142 c1cnccc1c2nnc(o2)SCCCF 11P-144 c1cc(ccc1C2=Nn3c(nnc3SC2)c4ccncc4)Cl 11P-145 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)O 11P-148 CC1=C(C[C@@H]([C@@H](C1)C(=O)OC)C(=O)OC)C 11P-149 c1ccc(c(c1)/C=C/2\C(=O)NC(=O)S2)Oc3ccc(c(c3)F)F 11P-153 c1ccc(c(c1)/C=C\2/C(=O)NC(=O)S2)Oc3ccc(c(c3)F)Cl 11P-154 CN1C(=O)C(=Cc2ccccc2Oc3ccc(cc3)Cl)C(=O)N(C1=O)C 11P-155 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OS(=O)(=O)c4ccc(cc4)OC 11P-158 CN1C(=O)C(=Cc2ccccc2Oc3ccc(cc3F)Br)C(=O)N(C1=O)C 11P-159 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCc4nnc(o4)C 11P-160 CN1C(=O)C(=Cc2ccccc2Oc3ccc(cc3Cl)Cl)C(=O)N(C1=O)C 11P-163 CCCCCCCc1ccc(cc1)CNc2ccc(cc2)C(=O)O 11P-165 Cc1ccc(cc1)C(=O)CSc2nnc(o2)c3ccc(cc3)C(F)(F)F 11P-166 Cc1ccccc1CSc2nnc(o2)c3ccncc3 11P-167 Cc1ccc(cc1)c2c(c[nH]n2)C=O 11P-168 c1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)Oc3cccc(c3)C(F)(F)F 11P-173 CN1C(=O)C(=Cc2ccccc2Oc3cccc(c3)C(F)(F)F)C(=O)N(C1=O)C 11P-174 Cc1ccc(cc1)C2=Nn3c(nnc3SC2)c4ccc(cc4)C(F)(F)F 11P-176 CC(C)(C)c1ccc(cc1)c2nnc(o2)S 11P-179 c1cc(cc(c1)F)CSc2nnc(o2)c3ccc(cc3)C(F)(F)F 11P-180 c1ccc(cc1)OCCSc2nnc(o2)c3ccc(cc3)C(F)(F)F 11P-181 c1cc(ccc1c2nnc(o2)SCc3ccc(c(c3)Cl)Cl)C(F)(F)F 11P-183 c1cc(ccc1c2nnc(o2)SCC(=O)c3ccc(cc3)Cl)C(F)(F)F 11P-184 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OS(=O)(=O)c4ccc(c(c4)OC)OC 11P-185 COc1ccc(cc1)c2nnc(o2)SCc3cccc(c3)C(F)(F)F 11P-186 c1cc(c(cc1[N+](=O)[O-])Br)NC2CCCC2 11P-187 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OS(=O)(=O)c4ccc(cc4)Br 11P-188 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3nnc(o3)SCc4ccc(c(c4)Cl)Cl 11P-191 Cc1ccc(cc1)C(=O)CSc2nnc(o2)c3ccc(cc3)OC 11P-192 COc1ccc(cc1)S(=O)(=O)Oc2ccc(c(c2)F)c3ccccc3 11P-194 c1ccc(cc1)c2ccc(cc2F)OC(=O)c3cccc(c3)C(F)(F)F 11P-195 COc1ccc(cc1)Oc2ccccc2C#N 11P-196 COC(=O)COc1ccc(cc1)c2nccc(n2)c3ccccn3 11P-197 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)c3nccc(n3)c4ccc(cc4)OC 11P-199 c1cc(c(c(c1)Cl)CSc2nnc(o2)c3ccc(cc3)C(F)(F)F)F 11P-200 c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)OCCCF 11P-201 CN1C(=O)C(=Cc2ccc(cc2)OCCCF)C(=O)N(C1=O)C 11P-202 c1cc(ccc1C=C2C(=O)NC(=O)NC2=O)OCCCF 11P-206 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4cccs4 11P-207 c1c2c(cc(c1Cl)Cl)nc(c(n2)C(F)(F)F)O 11P-209 CCc1ccc(cc1)CSc2nnc(o2)c3ccc(cc3)OC 11P-210 CC(C)(C)OC(=O)CSc1nnc(o1)c2ccc(cc2)OC 11P-211 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccco4 11P-212 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4cccs4 11P-213 CC1=C(C[C@H]([C@@H](C1)C(=O)OC)C(=O)OC)C 11P-214 c1cc(oc1)C(=O)Oc2ccc(cc2)c3nccc(n3)c4cccs4 11P-216 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccco4 11P-217 CCCCCCCCSc1nnc(o1)c2ccc(cc2)OC 11P-220 COc1ccc(cc1)c2nnc(o2)SC/C=C/c3ccccc3 11P-221 Cc1ccc(cc1)C(=O)CSc2nnc(o2)c3ccc(cc3)C(C)(C)C 11P-222 CC1(OCCO1)c2cccc(c2)[N+](=O)[O-] 11P-223 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccc(cc4)F 11P-227 Cc1c[nH]c(c1C#N)NC(=O)C 11P-228 CCOC(=O)/C(=N\Nc1ccccc1[N+](=O)[O-])/NC(=O)c2ccccc2 11P-229 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)c3nccc(n3)c4ccccn4 11P-230 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccc(cc4)F 11P-231 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4cccc(c4)C(F)(F)F 11P-232 c1ccc(cc1)CC(=O)Oc2ccc(cc2)c3nccc(n3)c4ccccn4 11P-233 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccc(cc4)Cl 11P-234 CCCCCCCCS(=O)(=O)c1nnc(o1)c2ccc(cc2)OC 11P-235 c1cc(c(cc1C(=O)O)F)[N+](=O)[O-] 11P-237 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)O 11P-238 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NN 11P-239 c1cc(ccc1Oc2ccc(cc2Br)N)F 11P-242 COC(=O)c1cc2n(n1)CCCNC2=O 11P-243 CC(C)(C)c1ccc(cc1)c2nnc(o2)SCCN3C(=O)c4ccccc4C3=O 11P-244 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccc(c(c2)F)c3ccccc3 11P-245 c1ccc(cc1)c2ccc(cc2F)OC(=O)c3cccc(c3Cl)Cl 11P-246 c1cc(c(c(c1)Cl)COc2ccc(cc2)C=O)F 11P-248 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OS(=O)(=O)c4ccc(cc4)Cl 11P-250 c1ccc(cc1)c2ccc(cc2F)OC(=O)c3ccco3 11P-251 c1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)c3nccc(n3)c4ccccn4 11P-254 CCOC(=O)C(C#N)c1ccc(cc1[N+](=O)[O-])C(F)(F)F 11P-255 c1cc(cc(c1)NC(=O)c2ccncc2)C(=O)O 11P-304S c1c(nns1)C(=O)NN 11P-305S COc1cnc(nc1OC)c2ccccc2 11P-309S c1ccc(cc1)n2c(c(cn2)C(=O)NN)n3cccc3 11P-313S c1cc2ccn(c2nc1)S(=O)(=O)c3ccc(cc3)Cl 11P-314S c1cc2ccn(c2nc1)S(=O)(=O)c3ccc(cc3)F 11P-315S COc1ccc(cc1)NC(=O)c2cnn(c2n3cccc3C(=O)C(=O)Nc4ccc(cc4)OC)c5ccccc5 11P-320S c1ccc(cc1)c2c3c(c(ncn3)O)sc2SCC#N 11P-321S c1ccc(cc1)S(=O)(=O)n2ccc3c2nccc3 11P-322S Cc1ccc(cc1)S(=O)(=O)OCC2(CCN(CC2)C(=O)c3ccc(c(c3)Cl)Cl)F 11P-324S c1cc(ccc1F)S(=O)(=O)OCC2(CCN(CC2)C(=O)c3ccc(c(c3)Cl)Cl)F 11P-330S c1cc(c(cc1C(=O)N2CCC(CC2)(COS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)F)Cl)Cl 11P-331S c1ccc(cc1)c2c3c(c(ncn3)Cl)sc2SCC#N 11P-334S COC(=O)c1ccc(o1)NC(=O)c2ccccc2 11P-337S COC(=O)c1ccc(o1)NC(=O)c2ccc(cc2)F 11P-338S COC(=O)c1ccc(o1)NS(=O)(=O)c2ccccc2 11P-339S COC(=O)c1ccc(o1)NS(=O)(=O)c2ccc(cc2)Cl 11P-340S CC(C)(C)C(=O)Nc1c(sc(c1c2ccccc2)SCC#N)C#N 11P-343S Cc1ccc(cc1)C(=O)Nc2ccc(o2)C(=O)OC 11P-345S COC(=O)c1ccc(o1)NC(=O)c2cccc(c2)Cl 11P-346S COC(=O)c1ccc(o1)NC(=O)C2CC2 11P-347S CCN(CC)C(=O)C(=O)c1cccn1c2c(cnn2c3ccccc3)C(=O)OCC 11P-350S CCOC(=O)c1cnn(c1n2cccc2C(=O)C(=O)NCC=C)c3ccccc3 11P-351S c1cc(sc1)c2nnc(n2N)S 11P-352S Cn1c(nnc1S)c2cnn(c2n3cccc3)c4ccccc4 11P-353S c1cc(sc1)c2nnc(n2/N=C/c3ccc(cc3)F)S 11P-356S CCOC(=O)c1cnn(c1n2cccc2C(=O)C(=O)N(C)C)c3ccccc3 11P-357S CCCNC(=O)C(=O)c1cccn1c2c(cnn2c3ccccc3)C(=O)OCC 11P-358S CCOC(=O)c1cnn(c1n2cccc2C(=O)C(=O)N3CCCC3)c4ccccc4 11P-359S CCOC(=O)c1cnn(c1n2cccc2C(=O)C(=O)Nc3ccc(cc3)F)c4ccccc4 11P-360S CCOC(=O)c1cnn(c1n2cccc2C(=O)C(=O)Nc3ccccc3)c4ccccc4 11P-361S CCOC(=O)c1cnn(c1n2cccc2C(=O)C(=O)Nc3ccc(cc3)OC)c4ccccc4 11P-362S CCOC(=O)c1cnn(c1n2cccc2C(=O)C(=O)Nc3ccccc3C(F)(F)F)c4ccccc4 11P-363S Cn1c(nnc1SCC=C)c2cnn(c2n3cccc3)c4ccccc4 11P-364S Cn1c(nnc1SCc2ccccc2)c3cnn(c3n4cccc4)c5ccccc5 11P-365S Cn1c(nnc1SC)c2cnn(c2n3cccc3)c4ccccc4 11P-366S c1ccc(cc1)S(=O)(=O)n2c(cc3c2nccc3)C(c4ccc(cc4)Cl)O 11P-368S CSc1nnc(n1N)c2cccs2 11P-374S Cn1c(nnc1SCc2ccc(cc2)Cl)c3ccn(c3n4cccc4)c5ccccc5 11P-375S Cn1c(nnc1SCc2ccc(cc2)F)c3cnn(c3n4cccc4)c5ccccc5 11P-376S Cn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])c3cnn(c3n4cccc4)c5ccccc5 11P-377S Cc1ccc(cc1)CSc2nnc(n2C)c3cnn(c3n4cccc4)c5ccccc5 11P-378S Cn1c(nnc1SCc2ccc(cc2)OC)c3cnn(c3n4cccc4)c5ccccc5 11P-379S CCCSc1nnc(n1C)c2cnn(c2n3cccc3)c4ccccc4 11P-380S CCSc1nnc(n1C)c2cnn(c2n3cccc3)c4ccccc4 11P-381S CCCCCCSc1nnc(n1C)c2cnn(c2n3cccc3)c4ccccc4 11P-382S c1ccc(cc1)S(=O)(=O)n2c(cc3c2nccc3)C(c4cccs4)O 11P-384S c1ccnc(c1)SCCC(=O)O 11P-385S c1ccc(cc1)c2c3c(c(ncn3)Oc4ccc(cc4)Cl)sc2SCC#N 11P-386S Cc1ccc(cc1)CSc2nnc(n2N)c3cccs3 11P-387S Cc1ccc(cc1)/C=N/n2c(nnc2S)c3cccs3 11P-388S COc1ccc(cc1)/C=N/n2c(nnc2S)c3cccs3 11P-389S Cc1ccc(cc1)Oc2ncc(cn2)c3ccc(cc3)Cl 11P-391S c1ccc(cc1)c2c(cc(=O)[nH]n2)Br 11P-396S COc1cnc(nc1Sc2ccc(cc2)Cl)c3ccccc3 11P-397S c1cc(cc(c1)[N+](=O)[O-])/C=N/n2c(nnc2S)c3cccs3 11P-398S c1ccc(c(c1)/C=N/n2c(nnc2S)c3cccs3)O 11P-399S c1ccn(c1)c2ccc(cc2)[N+](=O)[O-] 11P-400S COC(=O)c1c(c2ccccc2s1)n3cccc3 11P-411S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCNCC3 11P-412S c1ccc(cc1)n2c(c(cn2)c3nnc(o3)S)n4cccc4 11P-416S c1ccc(cc1)n2c(c(cn2)c3nnc(n3c4ccccc4)S)n5cccc5 11P-417S c1cc(ccc1C2NC(CS2)C(=O)O)Cl 11P-420S Cc1ccc(cc1)C2NC(CS2)C(=O)O 11P-421S Cc1ccc(cc1)C(=O)NNC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 11P-502S Cc1ccc(cc1)c2nnc(o2)c3cc4cc(ccc4s3)[N+](=O)[O-] 11P-504S c1ccc(cc1)c2c(snn2)C(=O)N3CCOCC3 11P-507S CN(C)C(=O)c1c(nns1)c2ccccc2 11P-508S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)N3CCOCC3 11P-514S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)N3CCCC3 11P-515S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)N3CCCCC3 11P-516S CC1CN(CC(O1)C)C(=O)C(=O)c2cccn2c3ccsc3C(=O)OC 11P-517S CCCNC(=O)C(=O)c1cccn1c2ccsc2C(=O)OC 11P-519S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)NCC=C 11P-520S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)Nc3ccc(cc3)F 11P-521S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)Nc3cccc(c3)C(F)(F)F 11P-522S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)Nc3ccc(cc3)C(F)(F)F 11P-523S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)Nc3ccccc3C(F)(F)F 11P-524S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)Nc3ccc(cc3)Cl 11P-525S COC(=O)c1c(ccs1)n2cccc2C(=O)C(=O)Nc3ccc(cc3)Br 11P-526S c1ccc(cc1)c2c(snn2)C(=O)Nc3ccc(cc3)Cl 11P-528S c1ccc(cc1)c2c(snn2)C(=O)Nc3ccc(cc3)Br 11P-529S c1ccc(cc1)c2c(snn2)C(=O)Nc3cc(cc(c3)Cl)Cl 11P-530S c1ccc(cc1)c2c(snn2)C(=O)Nc3cccc(c3Cl)Cl 11P-531S c1ccc(cc1)c2c(snn2)C(=O)Nc3cccc(c3)C(F)(F)F 11P-532S c1ccc(cc1)c2c(snn2)C(=O)Nc3ccc(cc3)C(F)(F)F 11P-533S c1ccn(c1)c2ccsc2 11P-535S COC(=O)c1ccc(cc1)NC(=O)c2c(nns2)c3ccccc3 11P-536S c1ccc(cc1)c2c(snn2)C(=O)Nc3cc(ccc3O)Cl 11P-538S Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3ccco3 11P-540S Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3ccc(cc3)OC 11P-541S COC(=O)c1c(cc(s1)SC)c2ccc(cc2)Cl 11P-543S CSc1cc(c(s1)C(=O)O)c2ccc(cc2)Cl 11P-544S Cc1c(sc(n1)c2ccccc2)/C(=N/O)/C 11P-545S CC(C)NC(=O)c1ccc(cc1)CNC(=O)OCC(F)(F)F 11P-547S c1cc(ccc1CNC(=O)OCC(F)(F)F)C(=O)Nc2ccc(cc2)Cl 11P-548S c1cc(ccc1CNC(=O)OCC(F)(F)F)C(=O)Nc2ccc(cc2Cl)Cl 11P-549S COc1ccc(cc1)NC(=O)c2ccc(cc2)CNC(=O)OCC(F)(F)F 11P-550S CNC(=O)c1ccc(cc1)CNC(=O)OCC(F)(F)F 11P-551S CNC(=O)c1c(cc(s1)SC)c2ccc(cc2)Cl 11P-553S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)c3cccs3)/C 11P-554S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)Nc3cccc(c3)Cl)/C 11P-555S CC(C)NC(=O)c1c(cc(s1)SC)c2ccc(cc2)Cl 11P-556S CSc1cc(c(s1)C(=O)N2CCCC2)c3ccc(cc3)Cl 11P-557S CSc1cc(c(s1)C(=O)Nc2ccc(cc2)Cl)c3ccc(cc3)Cl 11P-558S CSc1cc(c(s1)C(=O)Nc2ccc(cc2F)F)c3ccc(cc3)Cl 11P-559S COc1ccc(cc1)NC(=O)c2c(cc(s2)SC)c3ccc(cc3)Cl 11P-560S CSc1cc(c(s1)C(=O)Nc2ccc(cc2)Oc3ccccc3)c4ccc(cc4)Cl 11P-561S CSc1cc(c(s1)C(=O)N2CCN(CC2)Cc3ccccc3)c4ccc(cc4)Cl 11P-562S CSc1cc(c(s1)C(=O)NCC=C)c2ccc(cc2)Cl 11P-563S CSc1cc(c(s1)C(=O)Nc2ccc(cc2)Br)c3ccc(cc3)Cl 11P-564S CSc1cc(c(s1)C(=O)Nc2ccc(cc2)C(F)(F)F)c3ccc(cc3)Cl 11P-565S CSc1cc(c(s1)C(=O)Nc2ccc(c(c2)Cl)Cl)c3ccc(cc3)Cl 11P-566S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)C3CC3)/C 11P-568S Cc1cccc(c1)C(=O)O/N=C(\C)/c2c(nc(s2)c3ccccc3)C 11P-569S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/C 11P-570S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)c3ccc(cc3)F)/C 11P-571S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)c3ccc(c(c3)Cl)Cl)/C 11P-572S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)c3ccc(cc3)Cl)/C 11P-573S c1cc(ccc1c2nc(on2)c3ccc(=O)n(c3)Cc4ccc(c(c4)Cl)Cl)Cl 11P-581S c1cc(ccc1Cn2cc(ccc2=O)c3nc(no3)c4ccc(cc4)Cl)Cl 11P-582S c1cc(ccc1Cn2cc(ccc2=O)c3nc(no3)c4ccncc4)Cl 11P-584S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)NC3CCCCC3)/C 11P-585S Cc1ccc(cc1)NC(=O)O/N=C(\C)/c2c(nc(s2)c3ccccc3)C 11P-586S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)Nc3ccccc3)/C 11P-587S c1ccnc(c1)/C(=N/OC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3)Cl)/N 11P-590S c1cc(c(cc1c2nc(on2)c3cc(cn(c3=O)Cc4ccc(cc4Cl)Cl)Cl)[N+](=O)[O-])Cl 11P-591S c1cc(ccc1c2nc(on2)c3cc(cn(c3=O)Cc4ccc(cc4Cl)Cl)Cl)Cl 11P-592S CSc1cc(c(s1)C(=O)NN)c2ccc(cc2)Cl 11P-593S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)Nc3ccc(cc3Cl)Cl)/C 11P-594S Cc1c(sc(n1)c2ccccc2)/C(=N/OC(=O)NC(C)C)/C 11P-595S CCNC(=O)O/N=C(\C)/c1c(nc(s1)c2ccccc2)C 11P-596S c1cc(ccc1c2cnc(nc2)Sc3ccc(cc3)Cl)Cl 11P-599S C1CN(CCN1CC(C(F)(F)F)O)CC(C(F)(F)F)O 11P-600 c1c(cc(c(c1C=O)O)Br)[N+](=O)[O-] 11P-605 c1cc2c(cc1CN3CCS(=O)(=O)CC3)OCO2 11P-607 C1CC1CN2CCS(=O)(=O)CC2 11P-608 c1c(cnc(c1Cl)N2CCN(CC2)CC(C(F)(F)F)O)C(F)(F)F 11P-609 COc1ccc(cc1OC)CN2CCS(=O)(=O)CC2 11P-610 c1cc(c(c(c1)Cl)/C=C\2/C(C3CCN2CC3)O)F 11P-611 c1cc(cnc1)CN2CCS(=O)(=O)CC2 11P-614 C1CCCC(CC1)N2CCS(=O)(=O)CC2 11P-615 c1cc(ccc1CN2CCS(=O)(=O)CC2)F 11P-616 COc1cccc(c1)CN2CCS(=O)(=O)CC2 11P-617 c1ccc2c(c1)c(c[nH]2)CCN3CCS(=O)(=O)CC3 11P-618 c1ccc(cc1)C(C(=O)O)N2CCS(=O)(=O)CC2 11P-619 COc1ccc2c(c1)cc(o2)C#N 11P-620 CC(C)C(C(=O)O)N1CCS(=O)(=O)CC1 11P-621 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)I 11P-622 c1cc(nnc1NCCO)Cl 11P-623 COc1ccc2c(c1)cc(o2)C(=O)N 11P-624 c1ccc(cc1)C(=O)NC(=S)N2CCCc3c2cccc3 11P-626 c1cc(c(cc1CN2CCS(=O)(=O)CC2)Cl)Cl 11P-628 C(CCNCC(C(F)(F)F)O)CNCC(C(F)(F)F)O 11P-630 CN(CC(C(F)(F)F)O)C1CCCCC1 11P-632 c1ccc(cc1)/C(=N\OC(=O)c2cccs2)/c3cc4cc(cc(c4o3)Br)Br 11P-633 CCC(C)NCC(C(F)(F)F)O 11P-634 C([C@@H](C(F)(F)F)O)N 11P-636 Cc1ccc(cc1)CN2CCS(=O)(=O)CC2 11P-638 COc1ccc(cc1)C(=O)COc2c(cc(cc2Br)OC)C=O 11P-639 c1ccc2c(c1)c(c[nH]2)CC(C(=O)O)N3CCS(=O)(=O)CC3 11P-641 c1cc(c(cc1Cl)Cl)C(c2cc3cc(cc(c3o2)Br)Br)O 11P-642 c1ccc(cc1)C(c2cc3cc(cc(c3o2)Br)Br)O 11P-643 COc1cc(cc(c1O)CO)Br 11P-644 CC1CN(CC(O1)C)CC(C(F)(F)F)O 11P-647 C1CCN(C(C1)CO)CC(C(F)(F)F)O 11P-648 COCCCNCC(C(F)(F)F)O 11P-649 CC(C)CC(C(=O)O)N1Cc2ccccc2C1=O 11P-650 C1CCC(C1)NCC(C(F)(F)F)O 11P-653 c1cc(ccc1c2nnc(n2N)c3ccc(cc3)Cl)Cl 11P-656 c1c(cc(c(c1CO)O)Br)[N+](=O)[O-] 11P-658 c1cc(ccc1C(c2cc3cc(cc(c3o2)Br)Br)O)Br 11P-659 c1cc(cnc1)c2nnc(n2N)c3cccnc3 11P-660 CCC(C)(C)c1ccc(c(c1)C(C)(C)CC)OCCCCNCC(C(F)(F)F)O 11P-661 C1CCC(CC1)N(CCO)CC(C(F)(F)F)O 11P-662 CC(C)N(CC(C(F)(F)F)O)C(C)C 11P-663 COc1cccc2c1oc(c2)C(c3ccc(cc3Cl)Cl)O 11P-665 COc1cc(ccc1C(=O)OC)N 11P-667 CC(C)(CO)N1Cc2ccccc2C1=O 11P-668 c1ccc(cc1)/C=C/2\COc3ccccc3C2=O 11P-669 c1ccc2c(c1)CN(C2=O)C(Cc3ccc(cc3)O)C(=O)O 11P-670 c1cc(ccc1c2nnc(n2N)c3ccc(cc3)O)O 11P-672 COc1ccc(c(c1)/C=N/c2ccccc2C#N)O 11P-676 COc1cccc2c1oc(c2)C(c3ccccc3Cl)O 11P-677 c1cn(cn1)CCCN2CCS(=O)(=O)CC2 11P-678 CN(C)CCn1cc2cc(ccc2n1)[N+](=O)[O-] 11P-680 c1ccc(cc1)NC(=O)OC(CN2CCN(CC2)c3ccccc3)C(F)(F)F 11P-681 Cn1c2ccc(cc2cn1)[N+](=O)[O-] 11P-682 Cn1cc2cc(ccc2n1)[N+](=O)[O-] 11P-683 c1ccc(cc1)C2CC23COc4ccccc4C3=O 11P-684 c1ccc(cc1)c2nnc(n2n3cccc3)c4ccccc4 11P-685 COc1cc(c(cc1C(=O)OC)Br)N 11P-687 COc1cccc(c1)C(=O)OC(CN2CCN(CC2)c3ccccc3)C(F)(F)F 11P-689 Cc1ccccc1c2nnc(n2N)c3ccccc3C 11P-690 c1ccc(cc1)NC(=O)OC\2C3CCN(/C2=C\c4c(cccc4Cl)F)CC3 11P-691 Cn1c2ccc(cc2cn1)N 11P-692 COc1ccc(cc1)NC(=O)OC\2C3CCN(/C2=C\c4c(cccc4Cl)F)CC3 11P-693 COc1ccc(cc1)NC(=O)OC(CN2CCN(CC2)c3ccccc3)C(F)(F)F 11P-694 Cn1c2ccc(cc2cn1)NC(=S)NC(=O)c3ccccc3 11P-695 COc1ccc(c(c1)O)/C=N/c2ccc(c(c2)OC)C(=O)OC 11P-700 c1ccc(cc1)C(=O)NC(=S)NCCN2CCOCC2 11P-701 Cn1c2ccc(cc2cn1)NC(=S)N 11P-703 c1ccc(c(c1)/C=C/2\COc3ccccc3C2=O)F 11P-704 COc1cc(ccc1C(=O)O)N 11P-705 COC(=O)c1ccc(cc1O)N 11P-706 c1ccc(cc1)C(C(=O)O)N2Cc3ccccc3C2=O 11P-707 c1ccc2c(c1)C(=O)/C(=C/c3ccc(c(c3)Cl)Cl)/CO2 11P-708 c1ccc(c(c1)/C=C/2\COc3ccccc3C2O)F 11P-709 CC(=O)C(Cc1c(cccc1Cl)Cl)C(=O)c2cn(nn2)c3cc(cc(c3)Cl)Cl 11P-802 Cc1c(sc(n1)c2cccnc2)c3cc[nH]n3 11P-803 COc1ccc2c(c1)[nH]c(n2)OCc3ccc(cc3)F 11P-806 COC(C(=O)c1cn(nn1)c2cc(cc(c2)Cl)Cl)OC 11P-807 Cc1c(nnn1c2cc(cc(c2)Cl)Cl)C(=O)c3ccc(cc3)OC 11P-809 Cc1cccc(n1)n2cc(nc2)C(=O)N/N=C\c3cccs3 11P-811 c1c(cc(cc1Cl)Cl)n2cc(nn2)c3cnc4cc(c(cc4n3)Cl)Cl 11P-814 CN(C)C(=O)C(Cc1ccccc1)C(=O)c2cn(nn2)c3cc(cc(c3)Cl)Cl 11P-817 Cc1c(sc(n1)c2ccccn2)C(=O)/C=C/N(C)C 11P-818 CN(C)/C=C/C(=O)C(CC(=O)OC)C(=O)OC 11P-819 COC(=O)Cc1c(ccn(c1=O)Cc2ccc(c(c2)Cl)Cl)O 11P-820 Cc1c(sc(n1)c2ccccc2)c3ccnn3C 11P-821 c1cc(cc(c1)F)CC(Cc2cccc(c2)F)C(=O)c3cn(nn3)c4cc(cc(c4)Cl)Cl 11P-822 CN(C)/C=C/c1c(nnn1c2cc(cc(c2)Cl)Cl)C(=O)c3ccc(cc3)OC 11P-823 CC[NH+](CC)CC.CC1(OC(=O)[C-](C(=O)O1)C(c2ccc3c(c2)OCO3)C(C#N)C(=C(C#N)C#N)N)C 11P-824 Cc1c(sc(n1)c2ccccc2)c3ccnn3c4ccccc4 11P-825 CCOC(=O)COc1c2cc(cc1Cc3cc(cc(c3OCC(=O)OCC)Cc4cc(cc(c4OCC(=O)OCC)Cc5cc(cc(c5OCC(=O)OCC)C2)C(C)(C)C)C(C)(C)C)C(C)(C)C)C(C)(C)C 11P-831 COC(=O)CC(c1ccno1)C(=O)OC 11P-833 Cc1cccc(n1)n2cc(nc2)C(=O)N/N=C(/C)\c3ccc(cc3)[N+](=O)[O-] 11P-835 Cc1ccc(cc1)/C(=N\NC(=O)c2cn(cn2)c3cccc(n3)C)/C 11P-836 CN(C)/C=C/c1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)c3ccncc3 11P-841 COC(=O)Cc1c(ccn(c1=O)Cc2cccs2)O 11P-842 COC(=O)Cc1c(ccn(c1=O)CCc2c[nH]c3c2cccc3)O 11P-843 COC(=O)Cc1c(ccn(c1=O)Cc2ccc(cc2)F)O 11P-844 COc1ccc(c(c1Br)F)Br 11P-845 Cc1cc(ccc1NC(=O)c2cc(ccc2Cl)[N+](=O)[O-])C34CC5CC(C3)CC(C5)C4 11P-847 c1cnccc1c2c3c(ccn2)n(nn3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F 11P-848 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)CCc5ccccc5)C 11R-0001 Cc1c(c(nc(n1)C)NNC(=O)C(C)(C)C)I 11R-0002 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)F)C 11R-0004 c1cc(ccc1c2cnc3cc(nn3c2N)c4ccc(c(c4)Cl)Cl)F 11R-0005 Cc1cc2ncc(c(n2n1)C(F)(F)F)C(=O)O 11R-0006 c1ccnc(c1)c2ccnc3n2nc(c3Cl)c4ccc(c(c4)Cl)Cl 11R-0007 Cc1cc2nc(c(c(n2n1)N)c3ccccc3)C 11R-0008 Cc1c(c(nc(n1)C)Oc2ccc(cc2)C#N)I 11R-0011 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)N)c5ccccc5)C)C 11R-0013 Cc1c(c(n2c(n1)cc(n2)c3ccc(c(c3)Cl)Cl)N)c4ccccc4 11R-0015 Cc1c(c(nc(n1)C)N2CCOCC2)I 11R-0017 Cc1c(c(nc(n1)C)NC2CCCCC2)I 11R-0018 CCOC(=O)/C(=C\Nc1cc(n[nH]1)C)/C(=O)C(F)(F)F 11R-0021 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)C(C)Oc5ccc(cc5Cl)Cl)C 11R-0022 c1cc(sc1)c2cc(n3c(n2)c(c(n3)c4ccc(c(c4)Cl)Cl)Cl)C(F)(F)F 11R-0025 c1ccc(cc1)c2cc(n3c(n2)c(c(n3)c4ccc(c(c4)Cl)Cl)Cl)C(F)(F)F 11R-0026 c1cc(cc(c1)Cl)c2cc(n3c(n2)c(c(n3)c4ccc(c(c4)Cl)Cl)Cl)C(F)(F)F 11R-0027 c1cc(c(cc1c2c(c3nc(cc(n3n2)C(F)(F)F)c4ccc(o4)Cl)Cl)Cl)Cl 11R-0030 Cc1cc2ncc(c(n2n1)O)NC(=O)c3ccccc3 11R-0032 Cc1cc2nccc(n2n1)C(C)Oc3ccc(cc3Cl)Cl 11R-0033 Cc1cc2nccc(n2n1)c3cnc4n(c3=O)ccs4 11R-0035 Cc1cc2nccc(n2n1)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-] 11R-0036 Cc1cc2nccc(n2n1)c3cnc4n(c3=O)CCS4 11R-0037 Cc1cc2ncc(c(n2n1)C)C(=O)Nc3ccsc3C(=O)OC 11R-0044 Cc1cc2nc(cc(n2n1)O)CSc3ccc(cc3)Cl 11R-0045 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)CSc5ccc(cc5)Cl)C 11R-0046 Cc1cc2nc(cc(n2n1)O)CS(=O)(=O)c3ccccc3 11R-0047 c1ccc(cc1)/C=C/c2ccccc2O 11R-0052 Cc1cc2ncc(c(n2n1)N)c3ccsc3 11R-0054 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)C)C(=O)Nc5ccsc5C(=O)O)C 11R-0055 C1(C(NC(=O)N1)O)O 11R-0058 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc(cc5)N6CCN(CC6)C)C 11R-0061 COC1=C(C2(C=CC(=O)C=C2)OC1=O)C(=O)OC 11R-0062 Cc1cc(n(n1)c2nc(cs2)c3cccc(c3)[N+](=O)[O-])C 11R-0067 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)OC)C 11R-0068 Cc1cc2ncc(c(n2n1)C)C(=O)Nc3ccsc3C(=O)O 11R-0070 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)Cl)C 11R-0071 Cc1cc2nccc(n2n1)c3cnc4n(c3=O)c5ccccc5s4 11R-0072 CCOC(=O)c1cnc2cc(nn2c1C(F)(F)F)C 11R-0073 Cc1cc(n2c(n1)cc(n2)C)N 11R-0075 c1ccc2c(c1)c(cn2C(=O)c3ccccc3F)c4ccc(nn4)Cl 11R-0200 c1ccc2c(c1)c(cn2C(=O)C3CC3)c4ccc(nn4)Cl 11R-0201 c1ccc2c(c1)c(cn2C(=O)C3CCCCC3)c4ccc(nn4)Cl 11R-0202 COC(=O)c1ccccc1Sc2c(cc(cn2)C(F)(F)F)Cl 11R-0203 C#CCOc1ccccc1C(=O)O 11R-0204 COc1ccc(cc1)c2cn3c(n2)ccc4c3nc(cc4C(F)(F)F)C(F)(F)F 11R-0205 CCOC(=O)C1=C(N=C2N(C1c3ccccc3)C(=O)CCS2)C 11R-0206 CCOC(=O)C1=C([NH+]=C2N(C1c3ccccc3)CCS2)C.[Br-] 11R-0207 CCN1C(=C(C(NC1=O)c2cccc(c2)[N+](=O)[O-])C(=O)OCC)C 11R-0208 CCOC(=O)C1=C(N=C2N(C1c3ccc(cc3)F)C(=O)CCS2)C 11R-0209 c1cc2nc(cn2c3c1c(cc(n3)C(F)(F)F)C(F)(F)F)C(=O)O 11R-0211 c1cc(ccc1c2c3c(no2)CCCC3)Cl 11R-0212 CCOC(=O)C1=C(NC(=S)NC1c2ccc(cc2)F)C 11R-0213 CCOc1ccccc1C=C2C(=O)c3ccccc3C2=O 11R-0215 c1ccc(cc1)c2c3c(no2)CCCC3 11R-0216 c1ccc(c(c1)COC(=O)NC2=C(C(=O)c3ccccc3C2=O)Cl)Cl 11R-0219 COc1cc(c(cc1OC)NC(=S)NCc2cccc(c2)C(F)(F)F)C#N 11R-0220 CC(=O)c1cc([nH]c1)C(=O)N2CCN(CC2)Cc3ccccc3 11R-0221 CCOC(=O)C1=C([NH+]=C2N(C1c3ccc(cc3)F)CCS2)C.[Br-] 11R-0222 CCOC(=O)C1=C(NC(=S)N(C1c2ccccc2)C=O)C 11R-0223 CCOC(=O)C1=C(NC(=O)N(C1c2ccccc2)C=O)C 11R-0224 CC(=O)c1cc([nH]c1)C(=O)NN 11R-0225 CCOC(=O)C1=C(N=C2N(C1c3ccccc3)C(=O)C(S2)C)C 11R-0226 CCOC(=O)C1=C(N(C(=S)N(C1c2ccccc2)C(=O)C)C)C 11R-0227 c1ccc(cc1)C=C2C(=O)c3ccccc3C2=O 11R-0228 c1ccc2c(c1)C(=O)C(=Cc3cccs3)C2=O 11R-0229 CCOc1ccccc1c2c(c(nc-3c2C(=O)c4c3cccc4)C)C#N 11R-0230 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NN 11R-0231 CC1=C2C(c3ccccc3C2=O)NC(=O)N1 11R-0235 CCOC(=O)C1=C(NC(=S)NC1c2cccc3c2cccc3)C 11R-0236 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)Cc3cccc(c3)C(F)(F)F 11R-0238 c1cc2nc(cn2c3c1c(cc(n3)C(F)(F)F)C(F)(F)F)C(=O)NN 11R-0239 CC#N.c1ccc2c(c1)c(cn2C(=O)c3cccc(c3)C(F)(F)F)c4ccc(nn4)Cl 11R-0242 CC#N.c1ccc2c(c1)c(cn2C(=O)c3cccc(c3)Br)c4ccc(nn4)Cl 11R-0243 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NC(=O)OC3CCCCCCC3 11R-0244 c1ccc(cc1)c2cn3c(n2)ccc4c3nc(cc4C(F)(F)F)C(F)(F)F 11R-0245 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccc(c3)C(F)(F)F)SCc4ccc(cc4)F 11R-0246 Cc1ccc(c(c1)CSc2nc3cc(c(cc3c(=N)n2Cc4cccc(c4)C(F)(F)F)OC)OC)C 11R-0247 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccc(c3)C(F)(F)F)SCc4ccc(cc4)Cl 11R-0248 CC(C)(C)c1ccc(cc1)CSc2c(c3c(c(n2)c4ccc(cc4)Cl)CCCC3)C#N 11R-0253 c1cc(ccc1c2c3c(c(c(n2)SCCCF)C#N)CCCC3)Cl 11R-0254 CCOC(=O)c1cn2cc(cc(c2n1)Cl)C(F)(F)F 11R-0255 c1cc2nc(cn2c3c1c(cc(n3)C(F)(F)F)C(F)(F)F)c4nnco4 11R-0257 CCOC(=O)C1=C(N=C(SC1c2ccccc2)/N=C/N(C)C)C 11R-0259 c1cc(ccc1C(=O)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)F)[N+](=O)[O-] 11R-0260 c1cc(ccc1C(=O)N2CCN(CC2)C(=O)C3CCCCC3)[N+](=O)[O-] 11R-0262 c1cc(ccc1CSc2c(c3c(c(n2)c4ccc(cc4)Cl)CCCC3)C#N)C(F)(F)F 11R-0264 c1ccc2c(c1)C(C(N(C2=O)CCCCl)c3ccc4c(c3)OCO4)C(=O)O 11R-0265 COc1ccc(cc1OC)C2C(c3ccccc3C(=O)N2CCCCl)C(=O)O 11R-0266 CCOC(=O)C1=C(N=C2N(C1c3cccc4c3cccc4)C(=O)CCS2)C 11R-0270 c1cc(ccc1c2cn3c(n2)ccc4c3nc(cc4C(F)(F)F)C(F)(F)F)F 11R-0271 c1cc(ccc1c2cn3c(n2)ccc4c3nc(cc4C(F)(F)F)C(F)(F)F)Br 11R-0272 COC(=O)c1ccccc1SCc2ccc(cc2Cl)Cl 11R-0273 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NC(=O)OCc3ccc(cc3)[N+](=O)[O-] 11R-0279 COc1cccc(c1)CSc2nc3cc(c(cc3c(=N)n2Cc4cccc(c4)C(F)(F)F)OC)OC 11R-0280 COc1ccc(cc1)CSc2nc3cc(c(cc3c(=N)n2Cc4cccc(c4)C(F)(F)F)OC)OC 11R-0281 c1ccc(cc1)c2c3c(c(c(n2)SCc4ccc(cc4)F)C#N)CCC3 11R-0282 Cc1ccc(cc1)c2c3c(c(c(n2)SCc4ccc(cc4)F)C#N)CCCC3 11R-0283 Cc1ccc(cc1)c2c3c(c(c(n2)SCc4ccc(cc4)C(C)(C)C)C#N)CCCC3 11R-0284 Cc1ccc(cc1)c2c3c(c(c(n2)SCCC(=C(F)F)F)C#N)CCCC3 11R-0285 c1ccc(c(c1)C(=O)O)SCc2ccc(cc2Cl)Cl 11R-0286 COC(=O)c1ccccc1SCc2cccc(c2)F 11R-0287 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccc(c3)C(F)(F)F)SCCC(=O)OC 11R-0288 CCCSc1nc2cc(c(cc2c(=N)n1Cc3cccc(c3)C(F)(F)F)OC)OC 11R-0289 CCOC(=O)C1=C(NC(=O)N(C1c2ccccc2)C(=O)C)C 11R-0290 CCOC(=O)C1=C(NC(=S)N(C1c2ccccc2)C(=O)C)C 11R-0291 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)c3ccc(cc3)[N+](=O)[O-] 11R-0292 Cc1ccc(c(c1)CSc2ccccc2C(=O)OC)C 11R-0295 COc1ccc(cc1)c2cn3ccsc3n2 11R-0296 c1ccc(c(c1)C(=O)O)SCc2cccc(c2)F 11R-0298 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccc(c3)C(F)(F)F)SCc4ccncc4 11R-0302 Cc1c(c(c2c(n1)-c3ccccc3C2=O)c4cccs4)C#N 11R-0303 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2CCCCl)C(=O)O 11R-0306 Cc1ccc(c(c1)CSc2ccccc2C(=O)O)C 11R-0307 CC(=O)/C=C/c1c(nc2n1ccs2)SCc3ccccc3 11R-0313 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccc(c3)C(F)(F)F)SCc4c(cccc4Cl)F 11R-0318 CCOC(=O)C1CSC2(N1C(=O)c3c2cccc3)C 11R-0319 CC(=O)c1ccc2c(c1)c(on2)c3ccc(cc3)OC 11R-0320 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccc(c3)C(F)(F)F)SC 11R-0322 COc1ccccc1C2C(c3ccccc3C(=O)N2C4CCCC4)C(=O)O 11R-0325 COc1ccc(cc1)c2c(n3ccsc3n2)C=O 11R-0327 c1ccc2c(c1)C(C(N(C2=O)C3CCCCC3)c4ccc(cc4)Cl)C(=O)O 11R-0329 CC(C)CSc1nc2cc(c(cc2c(=N)n1Cc3cccc(c3)C(F)(F)F)OC)OC 11R-0331 CCSc1nc2cc(c(cc2c(=N)n1Cc3cccc(c3)C(F)(F)F)OC)OC 11R-0336 CCOC(=O)CC(=O)NC(CC(=O)OC)c1ccc(cc1)C(C)C 11R-0600 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2NC(=O)C3CC3)C(=O)OC 11R-0601 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2NC(=O)c3cccs3)C(=O)OC 11R-0603 CC(C)c1ccc(cc1)C(CC(=O)OC)NC(=O)c2cccs2 11R-0605 CC(C)c1ccc(cc1)C(CC(=O)OC)NS(=O)(=O)c2ccc(cc2)Br 11R-0606 c1ccn(c1)c2ccc(cc2)OC(F)(F)F 11R-0607 Cc1ccc(cc1)C(CC(=O)O)NC(=O)C(F)(F)F 11R-0609 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2N)C(F)(F)F 11R-0611 c1ccn(c1)c2nccs2 11R-0613 c1ccc(cc1)N2CCN(CC2)Cc3cnc(s3)n4ccc5c4cccc5 11R-0614 CN1CCN(CC1)c2ccc(cn2)N 11R-0615 CC(=O)c1ccc(cc1)n2cccc2 11R-0616 CC(C)c1ccc(cc1)/C=C/C(=O)O 11R-0617 COC(=O)c1ccc(cc1)/C=C/[N+](=O)[O-] 11R-0618 c1ccc2c(c1)ccn2Cc3cnc(s3)Oc4cccc(c4)Cl 11R-0619 Cc1ccc(cc1)Oc2ncc(s2)CN3CCOCC3 11R-0620 c1cc(cc(c1)Cl)Oc2ncc(s2)CN3CCOCC3 11R-0621 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)C=O 11R-0622 c1cc(ccc1n2ccc(c2)C=O)OC(F)(F)F 11R-0623 c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cccn2c3ccc(cc3)Br 11R-0624 c1cc(n(c1)c2nccs2)C=O 11R-0625 c1cc(ncc1N)N2CCOCC2 11R-0626 c1cc(ccc1C(CC(=O)O)NC(=O)C(F)(F)F)[N+](=O)[O-] 11R-0627 c1cc(cc(c1)Br)C(CC(=O)O)NC(=O)C(F)(F)F 11R-0628 Cc1ccc(cc1)Oc2ncc(s2)Cn3ccc4c3cccc4 11R-0629 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)/C=N/O 11R-0630 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)C#N 11R-0632 COC(=O)CC(c1ccc(cc1)Br)n2cccc2 11R-0633 c1cc(ccc1n2ccc(c2)C=C(C#N)C#N)OC(F)(F)F 11R-0636 CCOC(=O)CC(=O)NC(CC(=O)OC)c1ccc(cc1)Br 11R-0637 Cc1ccc(cc1)Oc2ncc(s2)CN3CC(OC(C3)C)C 11R-0638 Cc1ccc(cc1)Oc2ncc(s2)CN3CCN(CC3)C 11R-0639 Cc1ccc(cc1)Oc2ncc(s2)Cn3cccn3 11R-0640 Cc1cc(c(cc1OC(=O)c2ccc(cc2)OC)C(C)C)Br 11R-0641 c1cc(ccc1n2ccc(c2)/C=N/O)Br 11R-0642 c1cc(ccc1n2ccc(c2)C=C(C#N)C#N)Br 11R-0643 c1cc2c(cc1C(CC(=O)O)NC(=O)C(F)(F)F)OCO2 11R-0645 Cc1cc(c(c(c1OC(=O)c2ccco2)Br)C(C)C)Br 11R-0646 Cc1cc(c(c(c1OC(=O)c2cccc(c2)[N+](=O)[O-])Br)C(C)C)Br 11R-0647 c1ccc2c(c1)/C(=C/c3ccn(c3)c4ccc(cc4)Br)/C(=O)N2 11R-0648 c1ccnc(c1)CCNC(=O)c2cccn2c3ccc(cc3)Br 11R-0649 c1c2c(cc3c1OCO3)C(=O)CC2NC(=O)C(F)(F)F 11R-0650 Cc1cc(c(cc1OC(=O)c2ccc(cc2Cl)Cl)C(C)C)Br 11R-0651 Cc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)n3cccc3 11R-0652 Cc1c(sc(n1)N(c2cccc(c2)C(F)(F)F)C(=O)OC(C)(C)C)C(=O)C 11R-0802 Cc1c(c(n2c(n1)cc(n2)c3ccc(c(c3)Cl)Cl)C)Cc4c(cccc4Cl)Cl 11R-0803 c1ccc2c(c1)c(c[nH]2)CCNc3ccc(nn3)Cl 11R-0804 c1ccc(c(c1)C2CC(=O)CC(=O)C2n3cncn3)Oc4cccc(c4)Cl 11R-0805 c1ccnc(c1)N2CCN(CC2)C(=O)Cc3c(cc(cn3)C(F)(F)F)Cl 11R-0806 COc1ccc(cc1OCC#C)CO 11R-0807 COc1ccc(cc1OCC#C)/C=C/C(=O)O 11R-0808 CC(=O)C(Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cl 11R-0810 COc1ccc(cc1OCC#C)/C=N/O 11R-0812 Cc1c(sc(n1)N(c2cccc(c2)C(F)(F)F)C(=O)c3ccccc3)C(=O)C 11R-0816 COC(=O)c1c(ccs1)n2cc(nn2)C(=O)c3ccccn3 11R-0818 CC(=O)N1CCC(CC1)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl 11R-0819 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Cc4c(cc(cn4)C(F)(F)F)Cl 11R-0820 COc1cc(ccc1OCc2cn(nn2)c3ccccc3)C=O 11R-0821 CC(=O)c1cnc(s1)c2ccccn2 11R-0822 Cc1c(sc(n1)N(c2cccc(c2)C(F)(F)F)C(=O)c3ccccc3)C(=O)/C=C/N(C)C 11R-0823 CC(=O)c1cc([nH]c1)C(=O)OC 11R-0827 COC(=O)c1cc(c[nH]1)C(=O)Cc2ccc(cc2)Cl 11R-0828 CN(C)CCNC(=O)Cc1c(cc(cn1)C(F)(F)F)Cl 11R-0829 Cc1cc(nc(n1)C(C)C)NCC=C 11R-1000 Cc1cc(nc(n1)C(C)C)NC 11R-1001 c1ccc(cc1)c2c(c3ccccc3[nH]2)C(=O)C(F)(F)Cl 11R-1060 c1ccc(cc1)c2c(c3ccccc3[nH]2)C(C(F)(F)Cl)O 11R-1061 Cn1cc(c2c1cccc2)/C=C/C(=O)C(F)(F)F 11R-1064 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCOCC2 11R-1121 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCCCC2 11R-1122 CN1CCN(CC1)c2ccc(cc2[N+](=O)[O-])/C=N/OC 11R-1123 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(c3ccccc3)c4ccccc4 11R-1126 c1ccc(cc1)n2c(c(cn2)C(=O)NN)C(F)(F)F 11R-1130 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3ccc(cc3)F 11R-1132 CCn1c(nnc1S)c2cnn(c2C(F)(F)F)c3ccccc3 11R-1133 CCn1c(nnc1SC)c2cnn(c2C(F)(F)F)c3ccccc3 11R-1134 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=N/OC 11R-1136 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F 11R-1137 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3cccs3 11R-1138 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3cccc(c3)Cl 11R-1139 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3ccc(cc3Cl)Cl 11R-1140 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=N/OC 11R-1141 CCn1c(nnc1SCc2ccc(cc2)Cl)c3cnn(c3C(F)(F)F)c4ccccc4 11R-1142 CO/N=C\c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 11R-1143 CO/N=C/c1cc(ccc1Cl)[N+](=O)[O-] 11R-1144 CCn1c(nnc1SCc2cccc(c2)OC)c3cnn(c3C(F)(F)F)c4ccccc4 11R-1145 CCn1c(nnc1SCc2ccc(cc2Cl)Cl)c3cnn(c3C(F)(F)F)c4ccccc4 11R-1146 CCn1c(nnc1SCc2ccc(cc2)F)c3cnn(c3C(F)(F)F)c4ccccc4 11R-1147 CCn1c(nnc1SCc2cccc(c2)Cl)c3cnn(c3C(F)(F)F)c4ccccc4 11R-1148 CCn1c(nnc1SCc2ccc(cc2)C)c3cnn(c3C(F)(F)F)c4ccccc4 11R-1149 COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=N/OC 11R-1150 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)c3ccccc3 11R-1151 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)C 11R-1152 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])N2CCCN(CC2)C(=O)c3cccc(c3)Cl 11R-1153 c1ccc(cc1)n2c(c(cn2)C(=O)O)C(F)(F)F 11R-1154 CO/N=C\c1cc(ccc1N2CCCC2)[N+](=O)[O-] 11R-1155 c1ccc(cc1)n2c(c(cn2)C(=O)N3CCOCC3)C(F)(F)F 11R-1157 c1ccc(cc1)NS(=O)(=O)NC(=O)c2cccn2c3ccc(cc3Cl)[N+](=O)[O-] 11R-1181 c1ccn(c1)c2ccc(cc2)n3cccc3 11R-1182 c1ccn(c1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl 11R-1183 COc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)n3cccc3 11R-1184 c1ccn(c1)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl 11R-1185 c1ccn(c1)c2ccc(cc2)NC(=O)c3cccc(c3)[N+](=O)[O-] 11R-1186 c1ccn(c1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3Cl)Cl 11R-1187 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)n3cccc3 11R-1188 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)n3cccc3 11R-1190 c1ccn(c1)c2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl 11R-1191 c1ccn(c1)c2ccc(cc2)NC(=O)c3ccc(cc3)F 11R-1192 c1ccn(c1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)F 11R-1193 c1ccn(c1)c2ccc(cc2)NC(=O)C3CC3 11R-1194 c1ccn(c1)c2ccc(cc2Cl)NC(=O)c3cccc(c3)[N+](=O)[O-] 11R-1197 CN1CCN(CC1)c2ccc(cn2)NC(=O)c3ccc(cc3)Cl 11R-1198 Cc1ccc(cc1)C(=O)Nc2ccc(nc2)N3CCN(CC3)C 11R-1199 c1cc(ccc1C(=O)Nc2ccc(nc2)N3CCOCC3)Cl 11R-1200 Cc1ccc(cc1)C(=O)Nc2ccc(nc2)N3CCOCC3 11R-1201 CN1CCN(CC1)c2ccc(cn2)NS(=O)(=O)c3ccc(cc3)Cl 11R-1202 c1cc(n(c1)c2ccc(cc2Cl)[N+](=O)[O-])NS(=O)(=O)Nc3ccc(cc3)F 11R-1209 Cc1c(c2ccccc2[nH]1)C(=O)NS(=O)(=O)Nc3ccc(cc3)Cl 11R-1240 Cc1c(c2ccccc2[nH]1)C(=O)NS(=O)(=O)Nc3ccc(cc3)F 11R-1241 c1c2c([nH]c(=O)c1C#N)CCCC2 11R-1253 c1ccc2c(c1)/C(=N/NC(=S)N)/C(=O)N2 11R-1254 c1ccc(c(c1)c2nc3ccsc3c(n2)Cl)Cl 11R-1300 Cc1ccc(cc1)Oc2c3c(ccs3)nc(n2)c4ccccc4 11R-1301 COc1ccc(cc1)CNc2c3c(ccs3)nc(n2)c4ccccc4Cl 11R-1303 Cc1cc(nc(n1)c2ccccn2)Cl 11R-1482 c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)[N+](=O)[O-] 11T-0001 COC(=O)CC(c1cccc(c1)F)NC(=O)CN2CCN(CC2)c3ccc(cc3)F 11T-0002 c1cc2c(cn[nH]2)c(c1)NS(=O)(=O)c3ccc(cc3)I 11T-0004 Cc1ccc(cc1)C(=O)CCc2ccc(cc2)N 11T-0007 c1cc2c(cn[nH]2)c(c1)NS(=O)(=O)c3cccs3 11T-0010 c1cc(cc(c1)Cl)CCC(c2cccs2)O 11T-0011 COC(=O)C(C(CC(=O)c1cccs1)c2cccc(c2)Cl)C(=O)OC 11T-0012 COc1ccccc1C(CC(=O)c2cccs2)C(C(=O)OC)C(=O)OC 11T-0014 Cc1ccc(cc1)C(=O)CC(c2cc(c(c(c2)OC)OC)OC)C(C(=O)OC)C(=O)OC 11T-0016 COc1ccccc1CCC(=O)c2cccs2 11T-0018 COC(=O)C(c1ccc(cn1)[N+](=O)[O-])(C(=O)OC)Br 11T-0034 c1cc2c(cc1F)onc2C3CCNCC3.Cl 11T-0035 COc1ccccc1CCC(c2cccs2)O 11T-0040 COC(=O)C(c1ccc(cn1)N)C(=O)OC 11T-0041 c1ccc2c(c1)CN(C2)c3ccc(c(c3)c4nc5ccccc5o4)F 11T-0204 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)c3nc4ccccc4o3)F 11T-0205 C/C(=N/Nc1ccccc1)/c2ccc(c(c2)OC)OC 11T-0206 Cc1c(noc1c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N)c6ccccc6Cl 11T-0207 Cc1c(noc1c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N)c6c(cccc6Cl)F 11T-0208 CC(C)(C)c1nc2c(c(ccn2n1)c3ccc4c(c3)OCO4)C#N 11T-0209 Cc1c(noc1c2nc3c(c(ccn3n2)c4ccc(cc4)Cl)C#N)c5ccccc5Cl 11T-0210 Cc1ccc(cc1)CSc2nc3cc(c(cc3c4n2nc(n4)C)OC)OC 11T-0211 Cc1nc2c3cc(c(cc3nc(n2n1)SCc4cccc(c4)OC)OC)OC 11T-0212 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccc(cc4)C)OC)OC 11T-0213 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4cccc(c4)OC)OC)OC 11T-0214 c1ccc(c(c1)CNS(=O)(=O)c2cccs2)N3CCC(CC3)CO 11T-0215 C/C(=C\1/CCOC1=O)/Nc2ccc(cc2OC)OC 11T-0219 CCCCCC1CCC(CC1)C(=O)N/N=C\c2cn(nc2c3ccc(cc3)c4ccccc4)c5ccccc5 11T-0220 Cc1c(c(n(n1)c2ccc(cc2)[N+](=O)[O-])N)c3cccc(c3)C(F)(F)F 11T-0223 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)/C=N/NC(=O)c5ccccc5 11T-0226 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4cc(ccc4C)C)OC)OC 11T-0227 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)C=C5C(=O)c6ccccc6C5=O 11T-0228 c1ccc2c(c1)CN(C2)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl 11T-0229 C/C(=N/Nc1ccccc1)/c2ccc3ccccc3c2 11T-0231 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)/C=N/NC(=O)c5ccc(cc5)Cl 11T-0232 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)/C=N\NC(=O)c5ccncc5 11T-0233 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4c(cc(cc4C)C)C)OC)OC 11T-0234 CCOC(=O)C1CCN(CC1)c2ccc(cc2)C#N 11T-0236 Cc1ccc(cc1)S(=O)(=O)N/N=C\c2cn(nc2c3ccc(cc3)c4ccccc4)c5ccccc5 11T-0238 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4cccc(c4)C)OC)OC 11T-0239 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)C=O 11T-0241 Cc1c2c(n3c(n1)c(cn3)c4ccc(c(c4)OC)OC)N(CC2)C5CCCC5 11T-0243 c1cc(ccc1C#N)c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N 11T-0244 c1cc(cc(c1)NC(=O)C(F)(F)F)C(F)(F)F 11T-0245 c1ccc2c(c1)CN(C2)c3ccc4c(c3)NC(=O)CO4 11T-0246 c1cc(oc1)c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N 11T-0247 c1cc(cc(c1)C(F)(F)F)c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N 11T-0248 Cc1c2c(n3c(n1)c(cn3)c4ccc(c(c4)OC)OC)N(CC2)C(C)C 11T-0249 Cc1ccc(cc1)c2cn3c(cc(nc3n2)C)O 11T-0250 c1cc2c(cc1c3cc[nH]c(=O)c3C#N)OCO2 11T-0251 Cc1c(c(c2cc(cc(c2n1)OC)OC)Cl)CCCl 11T-0252 c1cc(ccc1c2csc(n2)CC#N)Cl 11T-0253 Cc1cc([nH]n1)C(F)(F)F 11T-0255 Cc1c2c(n3c(n1)c(cn3)c4ccc(c(c4)OC)OC)N(CC2)C5CCCCCC5 11T-0256 CCCCCCCN1CCc2c1n3c(c(cn3)c4ccc(c(c4)OC)OC)nc2C 11T-0257 Cc1c2c(n3c(n1)c(cn3)c4ccc(c(c4)OC)OC)N(CC2)CCOC 11T-0258 Cc1c2c(n3c(n1)c(cn3)c4ccc(c(c4)OC)OC)N(CC2)C5CCCCCCC5 11T-0259 CCc1nc2c3cc(c(cc3nc(n2n1)SC/C=C/c4ccccc4)OC)OC 11T-0260 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccccc4C)OC)OC 11T-0261 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccccc4)OC)OC 11T-0262 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)C=O 11T-0263 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3ccc(cc3)C#N 11T-0265 Cc1c2cn[nH]c2n(n1)C 11T-0266 C1CC1c2n[nH]nn2 11T-0268 c1ccc2c(c1)C(=O)N(C2=O)CCOc3ccc(cc3)OCCN4C(=O)c5ccccc5C4=O 11T-0270 CS(=O)(=O)C/C(=N/O)/N 11T-0271 CC(C)(C)c1ccc(cc1)c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N 11T-0274 COc1cccc(c1)c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N 11T-0275 CCCCCc1nc2c(c(ccn2n1)c3ccc4c(c3)OCO4)C#N 11T-0279 c1ccc(cc1)/C(=N\O)/N 11T-0283 c1cc(c(cc1C(F)(F)F)NC(=O)C/C(=N/O)/N)Cl 11T-0286 c1cc(ccc1C#N)Oc2ccc(cn2)C(F)(F)F 11T-0288 c1ccc2c(c1)CN(C2)c3cc(c(cc3F)Cl)O 11T-0289 C/C(=C/1\CCOC1=O)/Nc2ccccc2C(F)(F)F 11T-0291 c1cc(ccc1c2csc(n2)C/C(=N\O)/N)Cl 11T-0296 COc1cc(cc(c1)OC)/C(=N\O)/N 11T-0297 c1ccc(cc1)OC(=O)Nc2ccc(cc2)Cl 11T-0298 c1ccc(c(c1)c2nc3c(c(ccn3n2)c4ccc5c(c4)OCO5)C#N)F 11T-0300 c1cc2c(cc1c3ccn4c(c3C#N)nc(n4)C5CCCCC5)OCO2 11T-0301 c1cc(ccc1NC(=O)NN)Cl 11T-0302 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)NN 11T-0303 c1cc2c(cc1C(=O)CBr)OCO2 11T-0305 C/C(=C\1/CCOC1=O)/Nc2ccccc2OC 11T-0306 c1ccc(c(c1)COc2ccc(cc2)C#N)F 11T-0307 CCOC(=O)CN1CCc2c1n3c(c(cn3)c4ccc(c(c4)OC)OC)nc2C 11T-0308 CC(=O)NCCNS(=O)(=O)c1cccs1 11T-0310 CCOC(=O)c1cnc2c(c(nn2c1N)C)c3cccc(c3)C(F)(F)F 11T-0314 CN1CCN(CC1)c2ccc(cc2)NC(=O)NN 11T-0315 c1cc(cc(c1)Oc2ncccn2)CO 11T-0316 c1cc2c(cc1c3csc(n3)N)OCO2 11T-0317 Cn1c2ccccc2c3c1sc(c3)C(=O)NCc4ccc(cc4)OC 11T-0319 Cn1c2ccccc2c3c1sc(c3)C(=O)N4CCN(CC4)CCO 11T-0326 c1cc2c(cc1Cl)cc(o2)c3cc[nH]n3 11T-0327 c1cc(sc1)c2cc(n[nH]2)C(F)(F)F 11T-0328 c1cc(ccc1/C(=N/O)/N)Oc2ccc(cn2)C(F)(F)F 11T-0329 c1ccc(cc1)c2ccnc(c2C#N)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 11T-0330 CCCOc1ccc2c(c1)OC(CC2=O)(C)C 11T-0331 c1ccc2c(c1)NC(=O)C(O2)CCO 11T-0333 c1ccc2c(c1)C(=O)N(C2=O)CCCOc3ccc(cc3)OCCCN4C(=O)c5ccccc5C4=O 11T-0334 CCCCCC1CCC(CC1)c2nnc(o2)SCc3ccc(c(c3)Cl)Cl 11T-0335 c1cc(ccc1C2OCCO2)/C(=N/O)/N 11T-0339 c1cc(ccc1/C=C/c2cc[nH]n2)Cl 11T-0340 c1ccc(c(c1)COc2ccc(cc2)/C(=N/O)/N)F 11T-0341 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)Oc2ccccc2 11T-0342 c1cc2c(cc1O)c(c(o2)/C=C/c3ccoc3)C=O 11T-0343 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C(C(F)(F)F)(C(F)(F)F)O 11T-0346 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)/C=C(/C#N)\c4ccc(cc4)F 11T-0347 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)/C=C\C(=O)O 11T-0348 Cc1cccc(c1)/C(=C\c2cn(nc2c3ccc(c(c3)OC)OC)c4ccccc4)/C#N 11T-0351 Cc1c(c(c2cccc(c2n1)C(F)(F)F)Cl)CCCl 11T-0352 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)/C=C(/C#N)\c4ccc5c(c4)OCO5 11T-0353 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)/C=C(/C#N)\c4ccccc4 11T-0355 CC1CCN(CC1)c2c(c(ccn2)c3ccccc3)C#N 11T-0356 COc1cccc(c1)/C(=C\c2cn(nc2c3ccc(c(c3)OC)OC)c4ccccc4)/C#N 11T-0357 c1ccc2c(c1)c(cn2c3ccc(cc3)/C=C(/C#N)\c4ccc5c(c4)OCO5)C=O 11T-0358 Cc1n[nH]c(=O)n1c2cccc(c2)F 11T-0359 c1cc(c(cc1OC/C(=N/O)/N)Cl)Cl 11T-0360 Cc1c2c(n3c(n1)ncn3)N(CC2)Cc4ccc(cc4)OC 11T-0364 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)NN 11T-0366 Cc1nn(c(=O)n1c2cccc(c2)F)Cc3ccc(cc3)OC 11T-0368 Cc1n[nH]c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl 11T-0373 Cc1nn(c(=O)n1c2cccc(c2)F)Cc3ccc(cc3)Cl 11T-0374 Cc1n[nH]c(=O)n1c2ccc(cc2)Cl 11T-0376 COC(=O)N/N=C/c1ccccc1Cl 11T-0619 c1cc(c(cc1Br)/C=N/NCCO)O 11T-0620 c1ccc(cc1)c2ccc(cc2)C(=O)Nc3ccncc3 11T-0621 c1ccc(c(c1)/N=N/c2c(nc(nc2O)S)O)F 11T-0622 c1cc(ccc1F)Sc2c3c([nH]cn3)nc(n2)N 11T-0623 COC(=O)N/N=C/c1ccccc1 11T-0624 c1ccc(cc1)NC(=O)N/N=C/c2ccccc2O 11T-0625 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=N/NC(=O)OC 11T-0626 COC(=O)N/N=C/c1cc(ccc1O)Br 11T-0627 CCOC(=O)c1ccc(cc1)NC(=O)Nc2ccccc2 11T-0628 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F 11T-0629 CN(C)CCC[NH2+]c1ccc(cc1[N+](=O)[O-])C(F)(F)F.[Cl-] 11T-0630 CN(Cc1ccccc1)c2cc(nc(n2)N)Cl 11T-0631 CCOC(=O)N1CCN(CC1)c2cc(nc(n2)N)Cl 11T-0632 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F 11T-0633 c1c(nc(nc1Cl)N)N2CCCC2 11T-0634 CSc1nc(cc(n1)Sc2ccc(cc2)F)Sc3ccc(cc3)F 11T-0635 CCN(CCO)c1cc(nc(n1)SC)Cl 11T-0636 c1ccc2c(c1)C(=O)N(C2=O)Nc3cccc4c3nccc4 11T-0637 c1cnccc1c2nnc(s2)c3ccncc3 11T-0638 CCOC(=O)c1ccc(cc1)Nc2cc(c3ccccc3n2)C 11T-0639 COC(=O)N/N=C/c1cccc(c1Cl)Cl 11T-0640 c1cc2ccc3c(c2nc1)[NH2+]C4=C3CCC4.[Cl-] 11T-0641 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)N 11T-0642 c1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl 11T-0643 CN(C)CCC[NH2+]C1=C(C(=O)c2ccccc2C1=O)Cl.[Cl-] 11T-0644 Cc1nc(cs1)c2ccc(cc2)Cl 11T-0645 c1cnccc1c2ccnc(n2)N 11T-0646 c1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Sc4ccccc4 11T-0647 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Nc3ccc(c(c3)C(=O)O)O 11T-0648 c1ccc(cc1)NC(=S)N/N=C/c2ccccc2Cl 11T-0650 c1ccc(cc1)NC(=S)N/N=C/c2ccccc2O 11T-0651 c1ccc2c(c1)c(c[nH]2)CCCC(=O)OCC(=O)c3ccc(cc3)Cl 11T-0652 c1cc2ccc3cc([nH]c3c2nc1)c4ccncc4 11T-0653 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCCCC3 11T-0654 CN1CCN(CC1)C2=C(C(=O)c3ccccc3C2=O)Cl 11T-0655 C/C(=N\Nc1cccc2c1nccc2)/c3ccccn3 11T-0656 C/C(=N\Nc1cccc2c1nccc2)/c3ccc[nH]3 11T-0657 Cc1c2ccccc2c(=O)n(n1)c3cccc4c3nccc4 11T-0658 CN(C)CCC[NH2+]c1ccc(cc1C(F)(F)F)[N+](=O)[O-].[Cl-] 11T-0659 CCOC(=O)[C@@H](CC(C)C)NS(=O)(=O)c1ccc(cc1)CSc2nc(cc(n2)O)C 11T-0660 CCOC(=O)[C@H](CC(C)C)N(C)S(=O)(=O)c1ccc(cc1)C[NH3+].[Cl-] 11T-0661 CCOC(=O)[C@H](CC(C)C)N(C)S(=O)(=O)c1ccc(cc1)C[NH2+]c2ccncc2[N+](=O)[O-].[Cl-] 11T-0662 c1ccnc(c1)c2cc3ccc4cccnc4c3[nH]2 11T-0663 C/C(=N/Nc1ccccc1)/c2ccccc2C(=O)O 11T-0664 C/C(=N\Nc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/c2ccccc2C(=O)O 11T-0665 CC(C)(C)C1=CC(C=C(C1=O)C(C)(C)C)[N+](=O)[O-].C(=[NH2+])(N)N 11T-0666 CCOC(=O)C1CCN(CC1)C2=C(C(=O)c3ccccc3C2=O)Cl 11T-0667 c1ccc(cc1)c2c(sc(n2)N)C(=O)NN 11T-0668 c1ccc(cc1)/C=N/NC(=O)Nc2ccccc2 11T-0669 Cc1cc([n+]2n1C(=C(C2=O)c3ccccc3)[O-])C 11T-0670 CCCCCCCCCCCCNC1=C(C(=O)c2ccccc2C1=O)Cl 11T-0671 c1ccc(cc1)n2c(ccn2)c3ccc(cc3)F 11T-0672 COc1ccc(cc1)c2ccc(c(=O)[nH]2)C(=O)O 11T-0673 CCN1C(=O)C(SC1=O)C(c2ccc(c(c2)[N+](=O)[O-])Cl)O 11T-0800 CNC(=S)Nc1cccc2c1cn[nH]2 11T-0801 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccc(cc3)F)C(F)(F)F 11T-0802 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccc(cc3)Br)C(F)(F)F 11T-0803 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccc(c(c3)OC)OC)C(F)(F)F 11T-0804 c1cc2c(cc1C3CC(=O)C=C(C3n4cncn4)O)OCO2 11T-0807 c1ccc(cc1)Cc2c(ccn(c2=O)CCc3c[nH]c4c3cccc4)O 11T-0808 Cc1c2c(nc3n1nnn3)CCCC2 11T-0809 Cc1cc(ccc1Nc2nc(cs2)c3ccc(cc3)OC)[N+](=O)[O-] 11T-0810 COc1ccc(cc1)c2csc(n2)NNc3ccc(cc3Cl)Cl 11T-0811 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cccc3c2cn[nH]3 11T-0812 CS(=O)(=O)Nc1cccc2c1cn[nH]2 11T-0813 C=CCNC(=S)Nc1cccc2c1cn[nH]2 11T-0814 c1cc2c(cn[nH]2)c(c1)NC(=O)NC3CCCCC3 11T-0817 COc1ccc(cc1)c2ccc3ccccc3n2 11T-0819 Cc1ccc(cc1)c2ccc3ccccc3n2 11T-0820 c1ccc2c(c1)ccc(n2)c3ccccn3 11T-0821 c1c(cc(c2c1cn[nH]2)Br)[N+](=O)[O-] 11T-0822 c1c(cc(c2c1cn[nH]2)[N+](=O)[O-])Br 11T-0823 c1ccc2c(c1)ccc(n2)c3ccc(cc3)F 11T-0824 Cc1cc2ccccc2nc1C 11T-0826 CCN1C(=O)/C(=C\c2ccc(c(c2)[N+](=O)[O-])N3CCN(CC3)C)/SC1=O 11T-0827 c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)O 11T-0828 Cc1cc2c(cc1NC(=O)c3ccco3)cn[nH]2 11T-0829 c1ccc(cc1)c2ccc3ccccc3n2 11T-0830 c1ccc(cc1)c2ccc(cc2)c3ccc4ccccc4n3 11T-0831 c1ccc(cc1)/C=C/c2n[nH]nn2 11T-0832 Cc1ccc(cc1)c2n[nH]nn2 11T-0833 Cc1c2c(nc(n1)n3cc(nn3)c4ccccc4)CCCC2 11T-0835 c1ccc(cc1)Cc2c(ccn(c2=O)CCc3cnc[nH]3)O 11T-0836 COC(=O)c1c(ccs1)n2cc(nn2)c3c(cc(cn3)C(F)(F)F)Cl 11T-0837 Cc1c2c(nc(n1)n3c(c(nn3)C(=O)OC)C(=O)OC)CCCC2 11T-0838 Cc1cc(n2c(n1)nnn2)CC(C)C 11T-0839 Cc1c(c(n2c(n1)c(cn2)c3ccc(cc3)OC)C)Cc4cnc(s4)Cl 11T-0840 CN1C(=O)C(SC1=O)Cc2ccc(cc2)N 11T-0841 c1ccc2c(c1)ccc(n2)c3cccs3 11T-0842 c1ccc2c(c1)ccc(n2)c3ccncc3 11T-0843 Cc1c(c(n[nH]1)C)Cc2c(cccc2Cl)F 11T-0844 COC(=O)Cc1c(ccn(c1=O)CCc2cnc[nH]2)O 11T-0845 Cc1c(cccc1[N+](=O)[O-])n2cccc2C=O 11T-0847 CCOC(=O)/C=C(\C)/Nc1ccc2cn[nH]c2c1 11T-0848 Cc1cc(cc(c1n2cccc2)[N+](=O)[O-])Br 11T-0850 Cc1cc(cc(c1n2cccc2)Br)[N+](=O)[O-] 11T-0851 Cc1cc(cc(c1n2cccc2)Cl)[N+](=O)[O-] 11T-0852 c1ccc(cc1)CCNS(=O)(=O)c2ccc(cc2)CC3C(=O)NC(=O)S3 11T-0853 c1ccc2c(c1)ccc(n2)c3cccc(c3)c4ccc5ccccc5n4 11T-0854 CN1C(=O)/C(=C\c2ccc(cc2)N)/SC1=O 11T-0855 Cc1ccc(cc1)n2c(n[nH]c2=O)C 11T-0858 c1ccc2c(c1)ccc(n2)c3cccc(c3)O 11T-0859 Cc1c2c(nc(n1)n3cc(nn3)C(=O)C(C)Oc4ccc(cc4)Cl)CCCC2 11T-0861 c1cc(c(c(c1)F)/C=C/C(=O)/C=C/c2c(cccc2F)Cl)Cl 11T-0862 c1ccc2c(c1)cc(c(n2)N)C#N 11T-0863 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccc4ccccc4n3 11T-0864 COc1ccc(cc1OC)CNS(=O)(=O)c2ccc(cc2)CC3C(=O)NC(=O)S3 11T-0866 c1c(cc(c2c1cn[nH]2)Cl)[N+](=O)[O-] 11T-0867 c1ccc(cc1)C(c2ccccc2)c3ccn[nH]3 11T-0869 CN(C)/C=C/C(=O)C(c1ccccc1)c2ccccc2 11T-0870 Cc1c(cc2ccccc2n1)C(=O)O 11T-0872 Cc1n[nH]c(=O)n1c2ccc(cc2)F 11T-0875 CCOC(=O)C(=CNc1ccc2cn[nH]c2c1)C(=O)OCC 11T-0876 C/C(=N/OC(=O)c1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)N3CCOCC3 11T-0878 C/C(=N/OC(=O)N(C)C)/c1c(cc(cn1)C(F)(F)F)N2CCOCC2 11T-0879 C/C(=N/OC(=O)C)/c1c(cc(cn1)C(F)(F)F)N2CCOCC2 11T-0880 c1cc(cc(c1)[N+](=O)[O-])c2cn3cc(cc(c3n2)Cl)C(F)(F)F 11T-0881 CCCCCC(=O)Nc1ccc(cc1)CC2C(=O)N(C(=O)S2)C 11T-0883 Cc1c(cc2ccccc2n1)O 11T-0885 Cc1c2c(n3c(n1)nnn3)CCC2 11T-0887 Cc1ccc(cc1)n2c(nn(c2=O)Cc3ccc(cc3)Cl)C 11T-0888 c1ccc(cc1)c2csc(n2)NNC(=O)c3ccccc3 11T-0889 c1ccc(cc1)C(=O)NNc2nc(cs2)c3ccc(cc3)F 11T-0890 c1ccc(cc1)C(=O)NNc2nc(cs2)c3cccc(c3)[N+](=O)[O-] 11T-0891 Cc1nn(c(=O)n1c2ccc(cc2)F)Cc3ccccc3 11T-0892 Cc1nn(c(=O)n1c2ccc(cc2)F)CC#N 11T-0893 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)F 11T-0894 Cc1nn(c(=O)n1c2ccc(cc2)F)Cc3ccc(cc3)Cl 11T-0895 Cc1cc2ccccc2nc1c3ccccc3 11T-0896 Cc1nn(c(=O)n1c2ccc(cc2)F)Cc3cccc(c3)C(F)(F)F 11T-0897 Cc1nn(c(=O)n1c2ccc(cc2)F)Cc3ccc(cc3)[N+](=O)[O-] 11T-0898 c1ccc(cc1)c2ccc(cc2)c3cc[nH]n3 11T-0899 c1ccc(cc1)C(C(=O)Nc2ccc3c(c2)CCC3)Br 11T-1540 c1cc\2c(cc1C(F)(F)F)NC(=O)/C2=C\c3cc(ccc3O)Cl 11W-0037 CC(=O)Nc1ccc(cc1)/C=C\2/c3ccc(cc3NC2=O)C(F)(F)F 11W-0038 CCn1c(cc(n1)C)N 11W-0050 c1cc(c(cc1S(=O)(=O)N2CCCCC2)[N+](=O)[O-])Cl 11W-0055 c1cc2c(cc1C(F)(F)F)NC(=O)C3N2CCC3 11W-0200 COC(=O)c1c(c2ccccc2[nH]1)CC(C#N)C#N 11W-0206 Cc1ccccc1CN2C(=O)/C(=C\c3ccc4c(c3)OCO4)/N=C2SCc5cccc(c5)C(F)(F)F 11W-0209 CC(C)(C)c1ccc(cc1)C(=O)n2c3ccccc3c(c2C(=O)OC)I 11W-0210 c1cc(cc(c1)C(F)(F)F)CSC2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)N2CCCF 11W-0212 c1ccc(cc1)CCCN2C(=O)/C(=C\c3ccc4c(c3)OCO4)/N=C2SCc5cccc(c5)C(F)(F)F 11W-0214 c1ccc2c(c1)NC(=O)C(S2)CC(=O)Nc3ccc(cc3)Cl 11W-0217 c1cc(cc(c1)C(F)(F)F)CSC2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)N2CC#N 11W-0220 CSC1=NC(=O)CS1 11W-0222 c1cc2c(c[nH]c2nc1)C(=O)C(F)(F)F 11W-0223 COC1=C(Cc2c3ccccc3[nH]c2C(=O)N1)C#N 11W-0225 COc1cccc(c1)NC(=O)CC2C(=O)Nc3ccccc3S2 11W-0227 Cc1ccc(cc1)NC(=O)CC2C(=O)Nc3ccccc3S2 11W-0228 c1c(nc(s1)CC(=S)N)O 11W-0231 Cc1cc(ccc1NC(=O)C)Br 11W-0233 c1cc(c(cc1S(=O)(=O)N2CCCC2)[N+](=O)[O-])Cl 11W-0235 CN(OC)S(=O)(=O)c1ccc2c(c1)N(C(=O)C3N2CCC3)Cc4cccc(c4)C(F)(F)F 11W-0236 CC(=O)CCN1C(=O)c2ccccc2C1=O 11W-0240 CN(OC)S(=O)(=O)c1ccc2c(c1)N(C(=O)C3N2CCC3)Cc4ccccc4F 11W-0242 c1ccc(cc1)/C=C/C=C\2/C(=O)NC(=S)S2 11W-0245 CC(C)(C)n1cc(cn1)C(=O)c2ccccc2OS(=O)(=O)c3cccs3 11W-0246 c1ccc(c(c1)/C=C\2/C(=O)NC(=S)S2)C(F)(F)F 11W-0247 CCOC(=O)c1cnc2c(c1NCc3ccc(cc3)OC)c(n[nH]2)C 11W-0248 CSC1=NC(=O)/C(=C/C=C/c2ccccc2)/S1 11W-0250 CC(C)(C)n1cc(cn1)C(=O)c2ccccc2OCc3cccc(c3)C(F)(F)F 11W-0256 COc1cccc(c1)C(=O)n2c3ccccc3c(c2C(=O)OC)I 11W-0257 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C3=NC(=O)/C(=C/C=C/c4ccccc4)/S3 11W-0259 c1ccc(cc1)/C=C\C=C/2\C(=O)N=C(S2)N3CCOCC3 11W-0260 c1ccc(cc1)/C=C/C=C/2\C(=O)N=C(S2)N3CCN(CC3)Cc4ccc5c(c4)OCO5 11W-0261 CCOC(=O)c1cnn(c1C(F)(F)F)C(C)(C)C 11W-0263 c1ccc2c(c1)C(=O)N(C2=O)CCC3C(=O)Nc4c(cccn4)O3 11W-0268 c1ccc(cc1)/C=C/C=C/2\C(=O)N=C(S2)NCCCN3CCOCC3 11W-0271 COc1ccc(cc1)S(=O)(=O)n2cc(c3c2nccc3)C(=O)C(F)(F)F 11W-0274 Cc1ccc(cc1)CN2c3cccnc3N4CCCC4C2=O 11W-0275 Cc1cccc(c1)COc2ccccc2C(=O)c3cnn(c3)C(C)(C)C 11W-0276 CC(C)(C)n1cc(cn1)C(=O)c2ccccc2Oc3ccc(cn3)C(F)(F)F 11W-0278 CC(C)(C)n1c(c(cn1)C(=O)O)C(F)(F)F 11W-0279 COC(=O)Cc1c2ccccc2on1 11W-0280 Cc1ccc(cc1)CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N(C)OC 11W-0281 c1ccc(cc1)N2CCN(CC2)CCC3C(=O)Nc4c(cccn4)O3 11W-0282 CSc1ccccc1N2CCN(CC2)CCC3C(=O)Nc4c(cccn4)O3 11W-0283 CSC1=NC(=O)/C(=C/c2ccccc2C(F)(F)F)/S1 11W-0284 Cc1ccc(cc1)CNC(=O)Cc2c3ccccc3on2 11W-0285 c1ccc2c(c1)c(no2)CC(=O)NCc3cccc(c3)Cl 11W-0286 CC(C)(C)n1cc(cn1)C(=O)c2ccccc2OCCCF 11W-0288 CCOC(=O)c1c(nc(s1)Cc2nc(cs2)O)C 11W-0290 c1ccc(cc1)c2nc(cs2)CCN3C(=O)c4ccccc4C3=O 11W-0296 CC(C)(C)n1cc(cn1)C(=O)c2ccccc2OC(=O)c3ccco3 11W-0298 Cc1ccc(cc1)CN2c3cc(ccc3N4CCCC4C2=O)C(F)(F)F 11W-0301 Cc1ccc(c(c1)CN2c3cc(ccc3N4CCCC4C2=O)C(F)(F)F)C 11W-0302 c1cc2c(cc1S(=O)(=O)N3CCCC3)NC(=O)C4N2CCC4 11W-0303 c1ccc2c(c1)c(no2)CC(=O)NN 11W-0304 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)Cc3nc(cs3)O 11W-0307 c1c(nc(s1)Cc2nc(cs2)O)C(F)(F)F 11W-0308 c1cc(cc(c1)C(F)(F)F)CN2c3cc(ccc3N4CCCC4C2=O)C(F)(F)F 11W-0310 CC(C)(CCl)C(=O)n1c2ccccc2c(c1C(=O)OC)I 11W-0311 COc1ccc(cc1)c2csc(n2)Cc3nc(cs3)O 11W-0316 c1cc(ccc1c2csc(n2)Cc3nc(cs3)O)Cl 11W-0317 CCOC(=O)Cc1csc(n1)Cc2nc(cs2)O 11W-0318 c1ccc2cc(ccc2c1)c3csc(n3)Cc4nc(cs4)O 11W-0319 c1cc(c(cc1Cl)Cl)c2csc(n2)Cc3nc(cs3)O 11W-0320 CCNC(=S)NNC(=O)Cc1c2ccccc2on1 11W-0321 Cc1ccc(cc1)/C=N\NC(=O)Cc2c3ccccc3on2 11W-0322 COc1ccc(cc1)C(=O)NNC(=O)Cc2c3ccccc3on2 11W-0324 c1ccc(cc1)c2c(sc(n2)Cc3nc(cs3)O)CC(=O)O 11W-0326 Cc1ccc(cc1)c2csc(n2)Cc3nc(cs3)O 11W-0327 CCn1cc(c2c1nccc2)C(=O)C(F)(F)F 11W-0328 c1ccc(c(c1)C(=O)c2cnn(c2)c3cccc(c3)F)O 11W-0329 c1c(nc(s1)CC(=O)N)O 11W-0330 c1ccc(c(c1)c2csc(n2)Cc3nc(cs3)O)F 11W-0331 CCn1c(nnc1S)Cc2c3ccccc3on2 11W-0333 CCOC(=O)c1csc(n1)Cc2nc(cs2)O 11W-0334 Cc1c(sc(n1)Cc2nc(cs2)O)C 11W-0335 c1cc(cc(c1)C(F)(F)F)CN2c3cc(ccc3N4CCCC4C2=O)S(=O)(=O)N5CCCC5 11W-0347 c1cc2c(cc1C(F)(F)F)N3CCCC3C(=O)N2 11W-0348 c1ccc(cc1)c2c(sc(n2)Cc3nc(cs3)O)c4ccccc4 11W-0349 c1cc(cc(c1)C(F)(F)F)C(=O)NCCCOc2ccc(cc2)OCCCNC(=O)c3cccc(c3)C(F)(F)F 11W-0350 c1cc(sc1)C(=O)NCCCOc2ccc(cc2)OCCCNC(=O)c3cccs3 11W-0351 c1cc(oc1)C(=O)NCCCOc2ccc(cc2)OCCCNC(=O)c3ccco3 11W-0352 Cc1c(sc(n1)Cc2nc(cs2)O)C(=O)C 11W-0353 c1cc(ccc1c2csc(n2)Cc3nc(cs3)O)Br 11W-0354 c1ccc(cc1)c2csc(n2)Cc3nc(cs3)O 11W-0355 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)NN 11W-0356 c1ccc2c(c1)c(no2)CC(=O)NNC(=S)Nc3ccc(cc3)Cl 11W-0357 c1ccc(cc1)NC(=S)NNC(=O)Cc2c3ccccc3on2 11W-0358 c1cc2c(cc1C(F)(F)F)NCC3N2CCC3 11W-0361 CCOC(=O)N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 11W-0612 CCOC(=O)C1CCCN(C1)C(=O)OC(C)(C)C 11W-0613 Cc1c(c(n(n1)C)Sc2ccccc2C(=O)OC)C=O 11W-0701 Cc1cc(c(n1c2ccc(cc2)Br)C)C=O 11W-0702 c1c(cnc(c1C(=O)O)N)Br 11W-0705 COC(=O)c1cccc(c1CN2CCC(CC2)Cc3ccccc3)N 11W-0801 COc1ccc(cc1)Cn2c3ccccc3c4c2-c5c(cc6ccccc6n5)CC4 11W-0802 c1ccc2c(c1)cc3c(n2)-c4c(c5ccccc5n4Cc6ccc(cc6)Br)CC3 11W-0803 CCOC(=O)c1csc(n1)Nc2ccc(cc2)C(F)(F)F 11W-0804 C/C(=C(\Cc1ccc(cc1)Cl)/C(=O)C)/NCCc2c[nH]c3c2cc(cc3)OC 11W-0805 COc1cc(ccc1OCc2ccc(nc2)Cl)/C=C\3/C(=O)NC(=O)S3 11W-0806 COc1ccc(c2c1ccc(n2)c3cccc(c3)C(F)(F)F)OC 11W-0807 COc1ccc(c2c1ccc(n2)c3ccc4ccccc4c3)OC 11W-0808 c1cc(ccc1c2ccc3cc(cc(c3n2)Br)Br)F 11W-0810 COc1ccc(c2c1ccc(n2)c3ccc(cc3)F)OC 11W-0811 c1ccc(cc1)Oc2ccc(cc2)c3ccc4cc(cc(c4n3)Br)Br 11W-0812 COc1ccc(c2c1ccc(n2)c3ccc(cc3)Oc4ccccc4)OC 11W-0813 c1ccc2c(c1)cc3ccc4c5ccccc5n(c4c3n2)Cc6ccc(cc6)Br 11W-0814 Cc1c(c(nn2c1nnc2)C)Cc3cnc(s3)Cl 11W-0818 CCCCCCC(c1ccnc2n1nc(n2)N)C(=O)OC 11W-0819 Cc1cc2cc(cc(c2nc1c3ccc(cc3)OC)Br)Br 11W-0821 c1ccc(cc1)Oc2ccc(cc2)c3ccc4ccccc4n3 11W-0822 Cc1cc2ccccc2nc1c3ccc(cc3)OC 11W-0823 CCOC(=O)c1csc(n1)N(Cc2ccc(cc2)F)c3ccc(cc3)C(F)(F)F 11W-0825 CCOC(=O)c1csc(n1)N(c2ccc(cc2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)NC(=O)C 11W-0828 c1ccc(cc1)COC(=O)CCCc2c[nH]c3c2cccc3 11W-0829 COc1ccc(c2c1ccc(n2)c3cnccn3)OC 11W-0830 COc1ccc(c2c1ccc(n2)c3ccc(cc3)c4ccccc4)OC 11W-0831 CCOC(=O)c1csc(n1)N(c2ccc(cc2)C(F)(F)F)c3c(cc(cn3)C(F)(F)F)Cl 11W-0834 Cc1ccc(o1)CC2C(=O)NC(=O)S2 11W-0836 c1ccc2c(c1)c(c[nH]2)CCCC(=O)Nc3ccncc3 11W-0838 c1ccc2c(c1)c(c[nH]2)CCCC(=O)OCc3ccc(cc3)[N+](=O)[O-] 11W-0839 Cc1cc(cc(c1)COC(=O)CCCc2c[nH]c3c2cccc3)C 11W-0840 c1ccc2c(c1)c(c[nH]2)CCCC(=O)OCc3ccc(cc3)C(F)(F)F 11W-0841 Cc1c(sc2n1cc(n2)c3ccc(cc3)OC)C(=O)C 11W-0842 Cc1ccc(n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)C 11W-0843 COc1ccc2c(c1)c(c[nH]2)CCn3ccc(c(c3=O)C/C=C/c4ccccc4)O 11W-0845 c1ccc(c(c1)c2ccc3cc(cc(c3n2)Br)Br)O 11W-0846 c1ccn(c1)c2ccc(cn2)C#N 11W-0847 c1c(sc(n1)Cl)CN2CCC(CC2)C(=O)O.Cl 11W-0848 c1c(cc(c(c1I)O)I)c2c(cc(cn2)C(F)(F)F)Cl 11W-0851 c1c(cc(c(c1[N+](=O)[O-])O)I)c2c(cc(cn2)C(F)(F)F)Cl 11W-0852 Cc1ccc(cc1)c2ccc3c(ccc(c3n2)OC)OC 11W-0853 COc1ccc(c2c1ccc(n2)c3ccc(cc3)C4CCCCC4)OC 11W-0854 COc1ccc(c2c1ccc(n2)c3ccc4c(c3)OCO4)OC 11W-0855 CCOC(=O)CN(c1ccc(cc1)C(F)(F)F)c2nc(cs2)c3ccc(cc3)OC 11W-0857 COc1ccc(cc1)C(=C2C(=O)c3ccccc3C2=O)O 11W-0858 COC(=O)c1cccc(c1CN2CCN(CC2)c3ccc(cc3)F)[N+](=O)[O-] 11W-0859 CC1CCN(CC1)Cc2c(cccc2[N+](=O)[O-])C(=O)OC 11W-0860 Cc1cccc(c1N2CCN(CC2)Cc3c(cccc3[N+](=O)[O-])C(=O)OC)C 11W-0861 COC(=O)c1cccc(c1CN2CCN(CC2)c3ccccc3)[N+](=O)[O-] 11W-0862 COC(=O)c1cccc(c1CN2CCCCC2)[N+](=O)[O-] 11W-0863 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3cn4ccccc4n3 11W-0865 c1ccn2cc(nc2c1)c3cccc(c3)NC(=O)C4CC4 11W-0868 COc1ccc(c2c1cc3c(n2)-c4ccccc4CC3)OC 11W-0869 COc1cccc(c1)COc2ccccc2c3ccc4cc(cc(c4n3)Br)Br 11W-0870 c1ccn2cc(nc2c1)c3cccc(c3)NS(=O)(=O)c4cccc(c4)C(F)(F)F 11W-0871 c1ccc2c(c1)cc3c(n2)-c4ccccc4CC3 11W-0872 CN(C)c1c(cc(s1)C(=O)c2ccccc2)c3cccnc3 11W-7015 Cc1c(c(c2c(n1)C3CCN2CC3)c4cc(ccc4OC)OC)C#N 11X-0005 Cc1c(c(c2c(n1)C3CCN2CC3)c4ccc(cc4)Cl)C#N 11X-0006 Cc1c(c(c2c(n1)C3CCN2CC3)c4cccs4)C#N 11X-0018 Cn1cc(cc1C(=O)OC)/C=C\2/c3ccccc3NC2=O 11X-0058 Cc1cccc(c1[N+](=O)[O-])C(=O)OC 11X-0063 COC(=O)c1ccc(nc1)C(=O)O 11X-0066 Cc1cccc(c1N)C(=O)OC 11X-0097 COC(=O)/C=C/CSC1=N/C(=C/c2ccc(cc2)n3cncn3)/C(=O)N1 11X-0202 CCOC(=O)CSC1=N/C(=C/c2ccc(cc2)n3cncn3)/C(=O)N1 11X-0203 c1cc(ccc1/C=C/2\C(=O)N3CCCSC3=N2)n4cncn4 11X-0208 CCOC(=O)CSC1=N/C(=C/c2ccc(cc2)n3cncn3)/C(=O)N1C(=O)C 11X-0210 c1ccc(c(c1)/C=C\2/C(=O)NC(=S)S2)OCc3cnc(s3)Cl 11X-0213 CC(C(=O)OC)SC1=N/C(=C/c2ccc(cc2)n3cncn3)/C(=O)N1 11X-0214 c1cc(ccc1F)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 11X-0216 Cc1ccc(cc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)[N+](=O)[O-] 11X-0217 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)C 11X-0218 Cc1cccc(c1N2CCN(CC2)Cc3nc(no3)c4ccc(cc4)Cl)C 11X-0219 CN(Cc1nc(no1)c2ccc(cc2)Cl)C3CCCCC3 11X-0220 c1cc2cccnc2c(c1)S(=O)(=O)Oc3c(c(c(c(c3F)F)F)F)F 11X-0222 c1cc(ccc1c2nc(on2)CO)Cl 11X-0223 c1ccc(cc1)C2(CCOCC2)C=O 11X-0224 CN1CCCN(CC1)Cc2nc(no2)c3cccc(c3)C(F)(F)F 11X-0238 Cc1c(c(on1)C)C(=O)O 11X-0244 c1cc(cc(c1)C(F)(F)F)c2nc(on2)CO 11X-0245 c1cc(cc(c1)C(F)(F)F)c2nc(on2)CN3CCOCC3 11X-0247 COc1ccc2c(c1)sc(n2)c3ccc(cc3)[N+](=O)[O-] 11X-0248 c1cc(cc(c1)C(F)(F)F)c2nc(on2)COc3ccc(cc3)Cl 11X-0250 c1cc(cc(c1)C(F)(F)F)c2nc(on2)COc3cccc(c3)C(F)(F)F 11X-0251 Cc1c(c(on1)C)CO 11X-0256 c1ccc(cc1)c2ccc(cc2)S(=O)(=O)Oc3c(c(c(c(c3F)F)F)F)F 11X-0266 CCCOc1ccc(cc1)OCc2nc(no2)c3cccc(c3)C(F)(F)F 11X-0270 COc1ccc(cc1)OCc2nc(no2)c3cccc(c3)C(F)(F)F 11X-0271 c1cc(cc(c1)Cl)CS(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 11X-0282 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 11X-0283 CC(=O)N1CCC(CC1)N 11X-0603 C1CNC(=S)SC1 11X-0703 c1cc(ccc1c2cnco2)Br 11X-0800 Cc1cc(ccc1[N+](=O)[O-])C(=O)OC 11X-0801 COC(=O)c1ccc2c(c1)nccn2 11X-0803 c1c(c(c(nc1Cl)Cl)C#N)C(F)(F)F 11X-0804 c1cc(nc2c1cc(cc2Br)Br)c3ccsc3 11X-0806 c1ccc2c(c1)ccc(n2)c3ccsc3 11X-0807 Cc1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)OCc4cnc(s4)Cl)C 11X-0808 CC(C)(C)C(=O)Nc1ccccc1OC(F)(F)F 11X-0809 c1ccc2c(c1)/C(=C/c3cnc(s3)N4CCCCC4)/C(=O)N2 11X-0810 Cc1cc(ccc1N)C(=O)OC 11X-0812 c1cc(ccc1C(CC(=O)O)N)OC(F)(F)F 11X-0813 c1ccc2c(c1)/C(=C/c3ccc(cc3)OC(F)(F)F)/C(=O)N2 11X-0814 c1ccc2c(c1)/C(=C/c3cccc(c3)Oc4cccc(c4)C(F)(F)F)/C(=O)N2 11X-0815 c1ccc2c(c1)/C(=C\c3cc(ccc3F)F)/C(=O)N2 11X-0817 c1cc(cc(c1)Oc2cccc(c2)C(F)(F)F)C(CC(=O)O)N 11X-0819 c1c(cc(cc1F)F)C(CC(=O)O)N 11X-0820 COc1ccc(cc1)OCC(=O)N 11X-0822 CCOC(=O)c1cn(nn1)c2nc(cc(n2)C)C 11X-0824 c1cc2c(cc1C(=O)O)nccn2 11X-0826 CC(=O)c1c(cc(cn1)C(F)(F)F)c2cccc(c2)C(F)(F)F 11X-0827 c1ccc2c(c1)C(=O)C(=Cc3cnc(s3)N4CCCCC4)C2=O 11X-0828 c1cc(c(cc1F)F)C(CC(=O)O)N 11X-0829 Cc1c(c2ccccc2n1C)C(=O)O 11X-0830 c1cc2nc(cn2cc1I)C(=O)NN 11X-0831 COC(=O)Cc1ccc(cc1)OCc2ccc(nc2)Cl 11X-0833 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(cc3F)F 11X-0834 c1cc(ccc1CC(=O)O)OCc2ccc(nc2)Cl 11X-0835 CCOC(=O)c1c(n2cc(ccc2n1)I)Cl 11X-0839 c1cc2nc(c(n2cc1I)Cl)C(=O)O 11X-0840 c1ccc(c(c1)/C(=N/O)/N)N2CCCCC2 11X-0841 c1cc(ncc1C#N)Cl 11X-0845 CO/N=C(\c1ccc(nc1)C2CC2)/C3CC3 11X-0848 CCO/N=C(\c1ccc(nc1)C2CC2)/C3CC3 11X-0849 c1ccc(cc1)CO/N=C(\c2ccc(nc2)C3CC3)/C4CC4 11X-0850 c1cc(ccc1CO/N=C(\c2ccc(nc2)C3CC3)/C4CC4)Cl 11X-0851 c1ccc(cc1)CO/N=C(\c2cc3ccccc3nc2)/C4CC4 11X-0852 CC(C)Cc1c(nc(s1)N)C(=O)OC 11X-0920 c1ccc2c(c1)[nH]c(n2)C(=O)O 11X-0922 Cc1cc(c(c(c1)OS(=O)(=O)c2ccc(cc2)F)CN3CCOCC3)C.Cl 11X-0923 CCOC(=O)CC(=O)c1ccco1 11X-0925 CCOC(=O)c1nc2ccccc2s1 11X-0926 CC(=O)c1c(c2ccccc2n(c1=O)c3ccccc3)O 11X-0928 COc1cc(cc(c1OC)OC)C2c3ccc4ccccc4c3OC(=C2C#N)N 11X-0931 CC(C)(C)c1ccc(cc1)c2c(nc(s2)N)C(=O)OC 11X-0934 COC(=O)c1c(sc(n1)N)c2cccc(c2)F 11X-0938 COc1ccc(cc1)c2c(nc(s2)N)C(=O)OC 11X-0943 COC(=O)c1c(sc(n1)N)c2ccc(cc2)C#N 11X-0944 Cc1ccc(cc1)n2c(c(cn2)C#N)N 11X-0946 CN(C)/C=N/C1=C(C(c2ccc3ccccc3c2O1)c4cc(c(c(c4)OC)OC)OC)C#N 11X-0947 CC1(C(=O)Nc2cc(ccc2S1)[N+](=O)[O-])C 11X-0948 c1ccc2c(c1)ccc3c2OC(=C(C3c4ccc5c(c4)OCO5)C#N)N 11X-0950 COC(=O)c1c(sc(n1)N)c2ccccc2F 11X-0951 COC(=O)c1c(sc(n1)N)c2ccccc2Cl 11X-0952 c1cc(ccc1c2c(nc(s2)N)C(=O)O)F 11X-0953 c1ccc(cc1)n2c3c(cn2)c(ncn3)NO 11X-0954 c1ccc2c(c1)ccc3c2OC(=C(C3c4cccs4)C#N)N 11X-0955 COC(=O)c1c(sc(n1)N)c2ccc(c(c2)Cl)Cl 11X-0956 c1ccc2c(c1)ccc3c2OC(=C(C3c4ccc(cc4Cl)Cl)C#N)N 11X-0964 CN(C)/C=N/C1=C(C(c2ccc3ccccc3c2O1)c4ccc5c(c4)OCO5)C#N 11X-0965 Cc1ccc(cc1)n2c(c(cn2)C#N)/N=C/N(C)C 11X-0966 Cc1cc(cc(c1)NC(=O)CCl)C 11X-0967 CC(C)(C)c1ccc(cc1)c2c(nc(s2)N)C(=O)O 11X-0969 CC1(OCCO1)c2cccc(c2)NC(=O)OC(C)(C)C 11X-0971 c1ccc(cc1)COC(=O)N2CCNC(=O)C2 11X-0974 CC(=O)N(C)c1ccc(cc1)N 11X-7003 CSc1nc(c2c(n1)n(nn2)c3cccc(c3)F)Nc4cccc(c4)F 11X-9005 CC(C)(C)OC(=O)N1CCC2(CC1)NCCO2 11Y-0204 CCC(CC)N1C(C(CCC1=O)C(=O)O)c2ccc(cc2)Cl 11Y-0229 CC(=O)N(C)c1cccc(c1)[N+](=O)[O-] 11Y-0601 Cc1cc(cc(c1N)C(=O)OC)Br 11Y-0801 CC1c2ccsc2CCN1 11Y-0805 c1cc(ccc1c2nnc(o2)CCl)Cl 11Y-0809 c1cc(ccc1c2nnc(o2)CCl)C(F)(F)F 11Y-0812 COC(=O)c1cc(c[nH]1)C(=O)C2CC2 11Y-0814 CC(C)(C)c1ccc(cc1)c2nnc(o2)CCl 11Y-0815 c1cc(ccc1C(=O)NN)[N+](=O)[O-] 11Y-0817 Cn1cccc1C(=O)CC#N 11Y-0820 Cc1cc(c(c(=O)o1)C(=O)/C=C/c2ccccc2)O 11Y-0823 COc1ccc2c(c1)c(c[nH]2)C(=O)CC#N 11Y-0826 COC(=O)c1cc(ccc1F)C(F)(F)F 11Y-0828 COC(=O)c1ccc(cc1)I 11Y-0831 Cn1cccc1C(=O)/C(=C/c2ccccc2OC)/C#N 11Y-0832 COc1cc(cc(c1OC)OC)C2c3c(c4ccccc4oc3=O)Oc5c2c(=O)oc6c5cccc6 11Y-0833 c1cc(c(c(c1)Cl)c2ncc3n2cc(cc3Cl)C(F)(F)F)Cl 11Z-0018 c1cc(c(c(c1)F)C(=O)N2[C@H](NN=N2)c3c(cc(cn3)C(F)(F)F)Cl)F 11Z-0036 c1cc(c(c(c1)Cl)C(=O)N2[C@H](NN=N2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 11Z-0040 COc1ccccc1C(=O)N2[C@H](NN=N2)c3c(cc(cn3)C(F)(F)F)Cl 11Z-0053 c1cc(cc(c1)NC(=O)c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 11Z-0206 CCNC(=O)NNC(=O)c1ccc(cc1)c2c(cc(cn2)C(F)(F)F)Cl 11Z-0211 c1cc(ccc1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NNC(=O)NC3CCCC3 11Z-0212 CCn1c(n[nH]c1=O)c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 11Z-0222 c1cc(ccc1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)c4cn5cc(cc(c5n4)Cl)C(F)(F)F 11Z-0229 c1cc(ccc1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Cl 11Z-0248 COc1cccc(c1)NC(=O)c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 11Z-0250 c1ccnc(c1)NC(=O)c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 11Z-0251 c1cc(cnc1)NC(=O)c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 11Z-0252 CC(C)(C)OC(=O)n1cc(c2c1cccc2)CO 11Z-0700 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)OC)C=O 11Z-0701 COc1ccc(cc1)c2nc(cs2)CO 11Z-0702 COc1ccc2c(c1)c(c[nH]2)C=O 11Z-0705 c1cc(ccc1C=O)c2c(cc(cn2)C(F)(F)F)Cl 11Z-0706 c1cc(ccc1C=O)Oc2c(cc(cn2)C(F)(F)F)Cl 11Z-0707 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)OC)CO 11Z-0708 c1cc(ccc1C(CN)O)Br 11Z-0710 c1c(cnc(c1Cl)CN2CCN(CC2)C=O)C(F)(F)F 11Z-0712 c1cc(ccc1C=O)c2cc(ccn2)C(F)(F)F 11Z-0715 COC(=O)c1cc(on1)c2ccccc2 11Z-0717 c1cc(cc(c1)C(=O)O)c2ccc(cn2)C(F)(F)F 11Z-0719 c1cc(cc(c1)N)c2ccc(cn2)C(F)(F)F 11Z-0722 c1cc(ccc1NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)Cl 11Z-0802 c1ccc(c(c1)NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)F 11Z-0803 COc1cccc(c1)NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 11Z-0804 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 11Z-0808 c1cc(cc(c1)N2CCN(CC2)C(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F)C(F)(F)F 11Z-0809 c1ccnc(c1)CNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 11Z-0810 c1c(cnc(c1Cl)CNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)C(F)(F)F 11Z-0811 c1c(cn2cc(nc2c1Cl)C(=O)NN)C(F)(F)F 11Z-0813 Cc1nc2c(cccc2o1)[N+](=O)[O-] 11Z-0814 c1cc(ccc1S(=O)(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)Br 11Z-0817 CCCCc1nc2c(cccc2o1)[N+](=O)[O-] 11Z-0818 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCCCC2 11Z-0819 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCSCC2 11Z-0820 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCC(CC2)O 11Z-0822 c1cc(c(c(c1)F)C(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)F 11Z-0823 Cn1cc(cc1C(=O)NN)Br 11Z-0824 CCOC(=O)c1cc(cc(n1)C(=O)OCC)C(F)(F)F 11Z-0825 c1c(cn2cc(nc2c1Cl)C(=O)NNC(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F)C(F)(F)F 11Z-0826 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNC(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 11Z-0827 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNC(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 11Z-0828 CCCCc1nc2c(cccc2o1)N 11Z-0829 c1ccc(cc1)C(=O)NNC(=O)C2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl 11Z-0830 Cc1nc2c(cccc2o1)N 11Z-0831 Cn1cc(cc1C(=O)O)Br 11Z-0832 c1cc(cc(c1)N2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 11Z-0833 c1cc(c(c(c1)Cl)C(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)Cl 11Z-0835 c1cc(sc1)CC(=O)NNC(=O)C2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl 11Z-0836 c1cc(c(c(c1)F)C(=O)NNC(=O)C2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl)F 11Z-0837 CCOC(=O)c1c(cccn1)C(F)(F)F 11Z-0838 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNC(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 11Z-0839 COc1ccc(cc1)C(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 11Z-0840 c1cc(ccc1F)S(=O)(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 11Z-0841 CCOC(=O)c1cc(nc(c1)C(F)(F)F)C(F)(F)F 11Z-0842 c1ccc2c(c1)cccc2N3CCN(CC3)Cc4c(cc(cn4)C(F)(F)F)Cl 11Z-0843 c1cnccc1CN2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl 11Z-0845 c1cc(ccc1C(=O)NNC(=O)C2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 11Z-0847 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCN(CC2)C(=O)OC(C)(C)C 11Z-0848 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCC3(CC2)OCCO3 11Z-0849 CC1CCCN(C1)c2ccc(c(c2)C(=O)C)[N+](=O)[O-] 11Z-0854 CC1CCN(CC1)c2ccc(c(c2)C(=O)C)[N+](=O)[O-] 11Z-0855 c1c(cc(nc1C(F)(F)F)C(F)(F)F)C(=O)O 11Z-0856 c1c(cc(nc1C(=O)O)C(=O)O)C(F)(F)F.O 11Z-0858 c1cc(cc(c1)Br)C(=O)CC#N 11Z-0859 CCOC(=O)c1cc(cc(n1)C(F)(F)F)C(F)(F)F 11Z-0861 c1cc(ccc1C(=O)O)OCc2c(cc(cn2)C(F)(F)F)Cl 11Z-0862 CC(=O)c1cc(ccc1N)N2CCCCC2 11Z-0867 COC(=O)c1ccc(cc1)Oc2cc(ccn2)C(F)(F)F 11Z-0868 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCCC2 11Z-0869 CC(=O)NNC(=O)c1cn2cc(cc(c2n1)Cl)C(F)(F)F 11Z-0870 c1ccc(cc1)C(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 11Z-0871 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 11Z-0872 CC1CC2=C(CCCC2=O)NC1=O 11Z-0924 CC(C)c1cnc(nc1Nc2ccncc2F)c3c(cccn3)F 11Z-5043 C1CN(NC1=O)C(=O)CN2CCOCC2 12A-002 c1cc(c(cc1Oc2ccc(cn2)[N+](=O)[O-])F)N 12A-004 c1cc(ccc1C#N)n2ccnc2 12A-005 c1cc(ccc1C(=O)N)n2ccnc2 12A-006 CN(C)/C=N/C(=O)c1ccc(cc1)n2ccnc2 12A-008 C1CN(NC1=O)C(=O)C(Cl)Cl 12A-009 C1CN(NC1=O)C(=O)C(Cl)(Cl)Cl 12A-010 c1ccc(cc1)NC(=O)N2CCC(=O)N2 12A-011 c1cc(ccc1NC(=O)N2CCC(=O)N2)Cl 12A-012 c1cc(ccc1c2n[nH]nn2)n3ccnc3 12A-013 c1cc(ccc1C(=O)N/C=N/O)n2ccnc2 12A-014 Cc1ccc(cc1)NC(=O)N2CCC(=O)N2 12A-015 c1cc(cc(c1)Cl)NC(=O)N2CCC(=O)N2 12A-016 CN(C)/C=N/C(=O)/C(=C/c1ccc(cc1)Cl)/C#N 12A-018 c1cc(ccc1/C=C(\C#N)/C(=O)N/C=N/O)Cl 12A-019 CC(=O)C1C=CC(C2C1C(=O)OC2=O)c3ccccc3 12A-020 c1ccc(cc1)/C=C(\C#N)/C(=O)N 12A-022 c1cnccc1/C=C(\C#N)/C(=O)N 12A-023 c1ccc(cc1)NC(=S)N2CCC(=O)N2 12A-024 CN(C)/C=N/C(=O)/C(=C/c1ccncc1)/C#N 12A-025 CN(C)/C=N/C(=O)/C(=C/c1ccccc1)/C#N 12A-026 CN(C)/C=N/C(=O)/C(=C/c1ccc(cc1)OC)/C#N 12A-027 c1ccc(cc1)/C=C(\C#N)/C(=O)N/C=N/O 12A-028 COc1ccc(cc1)/C=C(\C#N)/C(=O)N/C=N/O 12A-029 c1cnccc1/C=C(\C#N)/C(=O)N/C=N/O 12A-030 COc1ccc(cc1)/C=C(\C#N)/C(=O)N/C=N/OC 12A-032 CC(C)(C)NC(=O)N1CCC(=O)N1 12A-033 c1cc(ccc1/N=N/N2CCC(=O)N2)Cl 12A-035 c1ccc(cc1)/N=N/N2CCC(=O)N2 12A-036 Cc1ccc(cc1)/N=N/N2CCC(=O)N2 12A-037 COc1ccc(cc1)/N=N/N2CCC(=O)N2 12A-038 c1cc(cc(c1)/N=N/N2CCC(=O)N2)C(F)(F)F 12A-039 CO/N=C/NC(=O)c1ccc(cc1)n2ccnc2 12A-040 c1cc[n+](cc1)CC(=O)N2CCC(=O)N2.[Cl-] 12A-044 Cn1c(c(c(=O)n(c1=O)C)/C=N/OC)O 12A-050 CC(C)(C)C(=O)/C(=C/N(C)C)/C#N 12A-051 c1cc(c(c(c1)Cl)COc2ccc(c(c2)F)N)Cl 12A-052 CNC(=S)N1CCC(=O)N1 12A-053 C/N=C(\[NH+]1CCC(=O)N1)/SCc2ccc(cc2)Cl.[Cl-] 12A-054 C/N=C(/[NH+]1CCC(=O)N1)\SCc2ccccc2Cl.[Cl-] 12A-056 C/N=C(\[NH+]1CCC(=O)N1)/SCc2cccc(c2)Cl.[Cl-] 12A-057 CC(C)(C)C(=O)NO 12A-058 C1CCn2c(nnc2CC(=O)N)C1 12A-060 CC(C)(C)C(=O)NOC(=O)c1ccc(cc1)Cl 12A-062 Cc1ccc(cc1)C(=O)ONC(=O)C(C)(C)C 12A-063 CC(C)(C)C(=O)NOC(=O)c1ccc(cc1)F 12A-065 CC(C)(C)c1c(sc(n1)N)C#N 12A-067 CC(C)(C)C(=O)ONC(=O)c1ccc(cc1)Cl 12A-069 CC(C)(C)C(=O)ONC(=O)c1ccc(cc1)F 12A-070 c1cc(sc1)/C=C(\C#N)/C(=O)N 12A-071 Cc1ccc(cc1)CS/C(=N\C)/[NH+]2CCC(=O)N2.[Cl-] 12A-072 CN(C)/C=N/C(=O)/C(=C/c1cccs1)/C#N 12A-074 c1cc(sc1)/C=C(\C#N)/C(=O)N/C=N/O 12A-075 CO/N=C/NC(=O)/C(=C/c1cccs1)/C#N 12A-076 CN(C)/C=C(\C#N)/C(=O)N/C=N/OC 12A-080 CN(C)/C=C(\C#N)/C(=O)N/C=N/O 12A-081 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)Cl)/C#N 12A-083 c1ccc(c(c1)/C=C(\C#N)/C(=O)N)O 12A-086 CN(C)/C=N/[N+](C)(C)C.[I-] 12A-087 CS/C(=C\[N+](=O)[O-])/Nc1ccccc1 12A-088 c1ccc(cc1)N/C(=C/[N+](=O)[O-])/NN 12A-090 CN(C)/C=N/[N+](C)(C)Cc1c(cccc1Cl)Cl.[Cl-] 12A-097 c1ccc(cc1)/C=C/C=C(\C#N)/C(=O)N 12A-098 CN(C)/C=N/C(=O)/C(=C/C=C/c1ccccc1)/C#N 12A-099 Cc1cc(n(n1)C(=O)N)C 12A-101 CC(=O)C(=C/C=C/c1ccccc1)C(=O)C 12A-102 Cc1cc(n(n1)C(=O)/C(=C/N(C)C)/C#N)C 12A-103 COC(=O)/C(=C\c1ccc(cc1)Cl)/C#N 12A-104 COC(=O)NN=C(/C=N/O)/C=N/O 12A-105 c1ccc(cc1)C(=O)CC(C#N)C#N 12A-107 C(C#N)C(=O)NNC(=O)CC#N 12A-109 c1c(ccc(c1)Cl)N=C(/C=N/O)/C=N/O 12A-111 CNN=C(/C=N/O)/C=N\O 12A-112 c1ccc(c(c1)NC(=O)N2CCC(=O)N2)Cl 12A-114 CCOC(=O)c1cc2c(=O)c3ccccc3oc2nc1/C=C/Nc4ccccc4 12B-001 CCOC(=O)c1cc2c(nc1/C=C/Nc3ccsc3C(=O)OC)Cc4ccccc4C2=O 12B-003 CCOC(=O)c1cc2c(=O)c3ccccc3oc2nc1/C=C/Nc4cccnc4 12B-004 COC(Cc1nnc(n1c2ccc(cc2)Cl)SCC=C)OC 12B-005 CCOC(=O)c1cc2c(=O)c3ccccc3oc2nc1/C=C/Nc4ccccn4 12B-008 Cc1ccc(cc1)N/C=C(\C#N)/c2cccs2 12B-010 Cc1ccc(cc1C)N/C=C(\C#N)/c2cccs2 12B-012 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3)Cl 12B-013 Cc1c(c(nc(n1)N)C)C(=O)NCc2ccccc2 12B-014 CN(C)C(=O)c1cn(c(=O)c2c1cccc2)Cc3cccnc3 12B-017 c1ccc(cc1)NC(=O)n2cc(c(n2)N3CCOCC3)c4ccccn4 12B-019 c1ccnc(c1)c2cn(nc2N3CCOCC3)C(=O)Nc4cccc(c4)C(F)(F)F 12B-020 c1ccc(cc1)C(=O)n2cc(c(n2)N3CCOCC3)c4ccccn4 12B-021 c1ccc(cc1)S(=O)(=O)n2cc(c(n2)N3CCOCC3)c4ccccn4 12B-022 c1ccc2c(c1)c(cn(c2=O)Cc3cccnc3)C(=O)Nc4ccc(cc4)Cl 12B-023 CN(C)C(=O)Nc1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F 12B-026 COC(=O)Nc1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F 12B-028 CC(=O)n1cc(c(n1)N2CCOCC2)c3ccccn3 12B-031 CS(=O)(=O)n1cc(c(n1)N2CCOCC2)c3ccccn3 12B-032 CC(=O)N1CC(=O)N(CC1=O)C(=O)C 12B-033 CN(C(=O)Nc1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F)OC 12B-034 CCSC(=O)Nc1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F 12B-035 CN(c1ccc(cc1)Cl)C(=O)c2cn(c(=O)c3c2cccc3)Cc4cccnc4 12B-038 CN(C)C(=O)c1cn(c(=O)c2c1cccc2)Cc3ccccn3 12B-042 COC(=O)c1cn(c(=O)c2c1cccc2)Cc3ccccn3 12B-043 c1ccc2c(c1)c(cn(c2=O)Cc3ccccn3)C(=O)Nc4ccc(cc4)Cl 12B-044 Cn1c(nnc1SCC=C)CC(OC)OC 12B-045 COC(Cc1nnc(n1c2ccccc2)SCC=C)OC 12B-046 COC(Cc1nnc(n1c2cccc(c2)C(F)(F)F)SCC=C)OC 12B-047 CN(c1ccc(cc1)Cl)C(=O)c2cn(c(=O)c3c2cccc3)Cc4ccccn4 12B-049 COC(=O)Nc1cn(c(=O)c2c1cccc2)Cc3cccnc3 12B-051 COC(Cc1nnc(n1c2ccccc2)SCC#C)OC 12B-052 COC(Cc1nnc(n1c2cccc(c2)C(F)(F)F)SCC#C)OC 12B-053 Cc1c(c(n(n1)C)/C=C/N(C)C)[N+](=O)[O-] 12B-054 CCOC(c1ccc(cc1)/C=C/c2c(c(no2)C)[N+](=O)[O-])OCC 12B-061 COC(Cc1nnc(n1c2ccc(cc2)Cl)SCC#C)OC 12B-064 Cc1c(c(on1)/C=C/c2ccc(cc2)C=O)[N+](=O)[O-] 12B-065 Cc1cc(nc(n1)Nc2ccccc2)C 12B-067 Cc1c(c(on1)/C=C/c2ccc(cc2)/C=N/c3ccccc3)[N+](=O)[O-] 12B-069 c1ccnc(c1)c2cn(nc2N3CCOCC3)S(=O)(=O)c4cccc(c4)C(F)(F)F 12B-070 CCSC(C(=O)NN)SCC 12B-071 c1ccc(cc1)NCc2c3ccccc3c(=O)[nH]n2 12B-072 CCOC(c1ccc(cc1)/C=C/C(=O)C)OCC 12B-075 Cc1c(c(n[nH]1)C)[N+](=O)[O-] 12B-076 c1ccc2c(c1)/C(=C/Nc3cccc(c3)C(F)(F)F)/OC2=O 12B-081 c1ccc(c(c1)C#N)N/C=C\2/c3ccccc3C(=O)O2 12B-082 COC(=O)Nc1cn(c(=O)c2c1cccc2)Cc3ccccn3 12B-083 c1ccc2c(c1)c(=O)c3cc4c(cc[nH]c4=O)nc3o2 12B-084 CN(C)n1ccc2c(c1=O)cc3c(=O)c4ccccc4oc3n2 12B-085 c1ccc2c(c1)c(=O)c3cc4c(ccn(c4=O)N5CCCCC5)nc3o2 12B-086 c1ccc2c(c1)c(=O)c3cc4c(ccn(c4=O)Cc5cccnc5)nc3o2 12B-087 c1ccc2c(c1)c(=O)c3cc4c(ccn(c4=O)Cc5ccncc5)nc3o2 12B-088 c1ccc2c(c1)c(n[nH]c2=O)CNc3cccc(c3)C(F)(F)F 12B-089 CC(=O)/C=C/c1ccc(cc1)C=O 12B-090 c1ccc(c(c1)C#N)NCc2c3ccccc3c(=O)[nH]n2 12B-091 COc1ccc(cc1)N/C=C\2/c3ccccc3C(=O)O2 12B-092 COc1ccc(cc1)NCc2c3ccccc3c(=O)[nH]n2 12B-093 c1ccc2c(c1)/C(=C/Nc3ccc(cc3Cl)Cl)/OC2=O 12B-094 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3Cl)Cl 12B-095 CN(/C=C\1/c2ccccc2C(=O)O1)c3ccccc3 12B-096 Cc1c(c(on1)/C=C/c2ccc(cc2)/C=C/C(=O)C)[N+](=O)[O-] 12B-098 CN(Cc1c2ccccc2c(=O)[nH]n1)c3ccccc3 12B-099 CN(C)Cc1c2ccccc2c(=O)[nH]n1 12B-101 C=CCn1ccc2c(c1=O)cccc2[N+](=O)[O-] 12B-103 c1ccnc(c1)C2CCCCC2=O 12B-104 CCOC(c1ccc(cc1)/C=C/C(=O)/C=C\N(C)C)OCC 12B-105 CCOC(c1ccc(cc1)/C=C\c2nccc(n2)N)OCC 12B-106 c1ccc(cc1)c2c(c(on2)/C=C/Nc3ccc(cc3)Cl)C#N 12B-108 Cc1ccc(cc1C)N/C=C/c2c(c(no2)c3ccccc3)C#N 12B-109 c1ccc(cc1)c2c(c(on2)/C=C/Nc3cccc(c3)C(F)(F)F)C#N 12B-110 COc1ccc(cc1)N/C=C/c2c(c(no2)c3ccccc3)C#N 12B-111 c1ccc(cc1)c2c(c(on2)/C=C/Nc3ccc(cc3)C(=O)O)C#N 12B-113 c1ccc(cc1)c2c(c(on2)/C=C/Nc3ccc(cc3F)O)C#N 12B-114 CSc1cccc(c1)N/C=C/c2c(c(no2)c3ccccc3)C#N 12B-115 COC(=O)c1c(onc1c2ccccc2)/C=C/Nc3ccc(cc3)C(=O)O 12B-116 c1ccc(cc1)c2c(c(on2)/C=C/Nc3ccc(cc3F)F)C#N 12B-119 c1ccc(cc1)c2c(c(on2)/C=C/Nc3cc(ccc3O)Cl)C#N 12B-120 c1ccc(cc1)/C=C(/c2ccnn2C(=O)c3ccc(cc3)Cl)\Oc4ccc(cc4)Cl 12B-122 c1ccnc(c1)C\2CCCC/C2=N\O 12B-125 C[N+](C)(C)Cc1c2ccccc2c(=O)[nH]n1.[I-] 12B-128 c1cc(ccc1NCCC(=O)O)Cl 12C-002 CN(C)/C=C/C(=O)c1ccc(cc1)Br 12C-005 CO/N=C/CC(=O)c1ccc(cc1)Br 12C-006 CN(C)/C=C/C(=O)c1ccc(cc1)c2ccccc2 12C-009 CO/N=C/CC(=O)c1ccc(cc1)c2ccccc2 12C-010 COC(=O)Cc1c(nnn1c2ccc(cc2)Cl)C(=O)OC 12C-015 COC(=O)Cc1c(nnn1c2ccc(cc2Cl)Cl)C(=O)OC 12C-019 CCC(=O)c1cc([nH]c1)C(=O)C(Cl)(Cl)Cl 12C-031 CSc1nc2nccc(n2n1)c3ccccn3 12C-040 CCC(=O)c1cc([nH]c1)C(=O)N2CCOCC2 12C-041 CCC(=O)c1cc([nH]c1)C(=O)N2CCN(CC2)c3ccccc3 12C-042 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 12C-044 c1ccc(cc1)N/C(=N/Nc2ccccc2)/S 12C-045 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccccc2 12C-046 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)Cl 12C-052 CNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)Cl 12C-054 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 12C-056 c1ccc(cc1)n2cnc(n2)O 12C-058 Cc1c(c(no1)c2ccccc2)C(=O)c3cc([nH]c3)C(=O)C(Cl)(Cl)Cl 12C-061 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 12C-063 COC(=O)Cc1c(nnn1c2ccc(cc2)[N+](=O)[O-])C(=O)OC 12C-066 COC(=O)Cc1c(nnn1c2ccc(cc2)C(F)(F)F)C(=O)OC 12C-069 COc1ccc(cc1)n2c(c(nn2)C(=O)OC)CC(=O)OC 12C-073 COC(=O)Cc1c(nnn1c2cccc(c2)C(F)(F)F)C(=O)OC 12C-075 COC(=O)Cc1c(nnn1c2ccc(cc2)OC(F)(F)F)C(=O)OC 12C-078 CSc1nc2nccc(n2n1)c3ccc(cc3)c4ccccc4 12C-084 CSc1nc2nccc(n2n1)c3ccc(cc3)Br 12C-085 COc1ccc(cc1)c2ccnc3n2nc(n3)SC 12C-086 CSc1nc2nccc(n2n1)c3ccc(cc3)Oc4ccccc4 12C-087 CSc1nc2nccc(n2n1)/C=C\c3ccccc3 12C-088 CSc1nc2ncc(c(n2n1)N)c3ccsc3 12C-089 c1ccc(c(c1)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3c(cccc3Cl)Cl)Cl 12D-003S c1cc(ccc1CSc2ccc(cc2[N+](=O)[O-])/C=N/O)Cl 12D-005S CO/N=C/c1ccc(c(c1)[N+](=O)[O-])SCc2ccc(cc2)Cl 12D-006S c1cc(ccc1CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(cc3Cl)Cl)Cl 12D-007S c1cc(c(c(c1)Cl)CO/N=C/c2ccc(c(c2)[N+](=O)[O-])SCc3ccc(cc3)Cl)Cl 12D-008S CO/N=C/c1ccc(c(c1)[N+](=O)[O-])SCc2cccc(c2)C(F)(F)F 12D-009S c1cc(cc(c1)C(F)(F)F)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(c(c3)Cl)Cl 12D-010S c1cc(cc(c1)C(F)(F)F)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3c(cccc3Cl)Cl 12D-011S c1cc(cc(c1)C(F)(F)F)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(cc3Cl)Cl 12D-012S c1cc(cc(c1)C(F)(F)F)CSc2ccc(cc2[N+](=O)[O-])/C=N/O 12D-013S c1cc(ccc1CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(c(c3)Cl)Cl)Cl 12D-017S COc1cccc(c1)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 12D-019 CN(C)/C=N/C(=S)Nc1ccc(cc1)OC 12D-020 c1cc(cc(c1)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)C(F)(F)F 12D-021 c1cc(nn2c1nnc2Cl)Cl 12D-022 c1cc(cc(c1)C(F)(F)F)CSc2ccc3nnc(n3n2)Cl 12D-023 CCOC(=O)CC1=CSC2=NCCN12.Cl 12D-024 c1cc(cc(c1)Sc2ccc3nnc(n3n2)Cl)C(F)(F)F 12D-025 c1cc(cc(c1)F)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 12D-026 c1ccc(cc1)CSc2ccc(cc2[N+](=O)[O-])/C=N/O 12D-031S c1ccc(cc1)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(cc3Cl)Cl 12D-033S c1ccc(cc1)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(c(c3)Cl)Cl 12D-034S c1ccc(cc1)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3c(cccc3Cl)Cl 12D-035S c1ccc(cc1)CSc2ccc(cc2[N+](=O)[O-])/C=N/OCc3ccc(cc3)[N+](=O)[O-] 12D-037S c1cc(ccc1CO/N=C/c2ccc(c(c2)[N+](=O)[O-])SCc3ccc(cc3)Cl)[N+](=O)[O-] 12D-038S c1cc(cc(c1)S(=O)c2ccc3nnc(n3n2)Cl)C(F)(F)F 12D-040 c1cc(cc(c1)Sc2ccc3n[nH]c(=O)n3n2)C(F)(F)F 12D-041 C1C[NH+]2C(=CSC2=N1)CC(=O)O.[Cl-] 12D-042S C[N+](=C/N=C(\Nc1ccc(cc1)OC)/SC)C.[I-] 12D-046 COc1ccc(cc1)Nc2[nH]ncn2 12D-047 Cc1cccc(c1NC(=S)/N=C/N(C)C)C 12D-048 Cc1cccc(c1N/C(=N\C=[N+](C)C)/SC)C.[I-] 12D-049 c1cc(ccc1O)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 12D-050 CC(C)Sc1ccc(cc1[N+](=O)[O-])C=O 12D-052S COC(=O)CSc1ccc(cc1[N+](=O)[O-])/C=N/OCc2c(cccc2Cl)Cl 12D-057S CC(C)(C)Sc1ccc(cc1[N+](=O)[O-])/C=N/O 12D-058S CC(C)(C)Sc1ccc(cc1[N+](=O)[O-])/C=N/OC 12D-059S CC(C)(C)Sc1ccc(cc1[N+](=O)[O-])/C=N/OCc2ccc(cc2Cl)Cl 12D-060S CC(C)(C)Sc1ccc(cc1[N+](=O)[O-])/C=N/OCc2c(cccc2Cl)Cl 12D-061S CC(C)Sc1ccc(cc1[N+](=O)[O-])/C=N/OCc2c(cccc2Cl)Cl 12D-063S c1cc(cc(c1)C(F)(F)F)CSc2ccc3n[nH]c(=O)n3n2 12D-064 CCOC(=O)CC1=CSC2=NCCN12 12D-065S c1cc(c(cc1OCC(F)(F)F)C(=O)NO)OCC(F)(F)F 12D-066S c1ccc(cc1)NC(=O)C/C=N\O 12D-067 c1ccc(cc1)NC(=O)C/C=N\OCc2ccc(cc2)[N+](=O)[O-] 12D-068 c1ccc(cc1)NC(=O)C/C=N\OCc2c(cccc2Cl)Cl 12D-069 c1cc(ccc1Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Oc4ccc5c(cc(nc5n4)C(F)(F)F)C(F)(F)F 12D-070 c1cc(ccc1CSc2c(n3ccsc3n2)C#N)Cl 12D-071S c1ccc(cc1)Sc2c(n3ccsc3n2)C#N 12D-072S c1ccc(cc1)CSc2c(n3ccsc3n2)C#N 12D-075S c1cc(cc(c1)C(F)(F)F)CSc2c(n3ccsc3n2)C=O 12D-076S c1cc(cc(c1)C(F)(F)F)CSc2c(n3ccsc3n2)/C=N/O 12D-077S Cc1ccc(cc1)Sc2c(n3ccsc3n2)C#N 12D-079S c1cc(cc(c1)C(F)(F)F)CSc2c(n3ccsc3n2)C#N 12D-080S Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2)S(=O)(=O)Oc3ccc(cc3)Cl 12D-081 c1ccc(cc1)NC(=O)C/C=N\OC(=O)Nc2ccccc2 12D-082 CN(C)/C=C(/C=N/OCc1ccc(cc1Cl)Cl)\C(=O)Nc2ccccc2 12D-083 Cc1c(c(ns1)SCc2ccc(cc2)Cl)C(=O)N 12D-084 Cc1c(n2ccccc2n1)c3c(cn(n3)C)Br 12D-806 Cc1ccn2c(c1)nc(c2CO)C 12D-808 CN(C)/C=C\1/C(=NOC1=O)c2ccncc2 12D-902 c1cc(c2c(c1)S(=O)(=O)NC2=O)O 12D-907 COC(=O)c1cn(nc1c2cccnc2)c3cccc(c3)C(F)(F)F 12D-914 c1cc(cc(c1)n2cc(c(n2)c3ccncc3)C(=O)O)C(F)(F)F 12D-916 c1cc(cc(c1)n2cc(c(n2)c3cccnc3)C(=O)O)C(F)(F)F 12D-917 Cc1ncc(c(n1)c2ccncc2)C(=O)NC 12D-919 CNC(=O)c1cn(nc1c2cccnc2)c3cccc(c3)C(F)(F)F 12D-923 CNC(=O)c1cn(nc1c2ccncc2)c3cccc(c3)C(F)(F)F 12D-924 c1cc(c(c(c1)Cl)CO/N=C/NC(=O)C(=O)Nc2ccc(cc2Cl)Cl)Cl 12E-002 CO/N=C/NC(=O)C(=O)Nc1ccc(cc1Cl)Cl 12E-003 CCOC(=O)COc1ncn(n1)c2ccccc2 12E-005 c1ccc(cc1)n2cnc(n2)OCC(=O)N 12E-006 CN(C)c1nc(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)N(C)C 12E-008 CC(C(=O)C)n1cncn1 12E-009 CN(C)c1nc(n(n1)c2cccc(n2)Cl)N(C)C 12E-010 c1cc(ccc1C(=O)Cn2cncn2)Cl 12E-011 CCNC(=O)n1cc(c(n1)c2ccccc2)n3cncn3 12E-012 CN(C)c1nc(n(n1)c2ccc(nn2)Cl)N(C)C 12E-015 CN(C)/C=C(/C(=O)c1ccc(cc1)Cl)\n2cncn2 12E-016 c1cc(ccc1c2c(c[nH]n2)n3cncn3)Cl 12E-018 CN(C)c1nc(n(n1)c2ccc(cc2Cl)Cl)N(C)C 12E-019 c1cc(ccc1c2c(cnc(n2)N)n3cncn3)Cl 12E-022 CC(=O)n1ccc(n1)c2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl 12E-028 CC(c1cc[nH]n1)n2cncn2 12E-029 CCNC(=O)n1cc(c(n1)c2ccc(cc2)Cl)n3cncn3 12E-030 CC(C(=O)/C=C/N(C)C)n1cncn1 12E-031 CC(c1ccnc(n1)N)n2cncn2 12E-032 c1ccc(cc1)S(=O)(=O)n2cc(c(n2)c3ccc(cc3)Cl)n4cncn4 12E-035 c1ccc(cc1)n2cnc(n2)OCC(=O)N/C=N\OCc3ccc(cc3Cl)Cl 12E-036 c1cc(ccc1/C=C(\C#N)/c2nc([nH]n2)Cn3cncn3)Cl 12E-040 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/c2nc([nH]n2)Cn3cncn3 12E-041 c1cc(ccc1/C=C(\C#N)/c2nc([nH]n2)Cn3cncn3)F 12E-042 COc1ccc(cc1)/C=C(\C#N)/c2nc([nH]n2)Cn3cncn3 12E-043 c1cc(cc(c1)Cl)/C=C(\C#N)/c2nc([nH]n2)Cn3cncn3 12E-044 c1cnccc1/C=C(\C#N)/c2nc([nH]n2)Cn3cncn3 12E-045 CN(C)c1ccc(cc1)/C=C(\C#N)/c2nc([nH]n2)Cn3cncn3 12E-046 c1ncn(n1)CC(=C(C#N)C#N)N 12E-047 Cc1c(c(=O)n([nH]1)c2ccccc2)c3ccc(cc3)Cl 12E-306S Cc1c(c(=O)n([nH]1)c2cccc(c2)Cl)c3ccc(cc3)Cl 12E-307S c1cc(cc(c1)Cl)c2c[nH]n(c2=O)c3cccc(c3)C(F)(F)F 12E-308S Cc1c(c(=O)n([nH]1)c2cccc(c2)C(F)(F)F)c3ccc(cc3)Cl 12E-309S Cc1c(c(=O)n([nH]1)c2cccc(c2)[N+](=O)[O-])c3ccc(cc3)Cl 12E-310S CC(C)C(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(c(c3)Cl)Cl 12E-311S CC(C)(C)C(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(c(c3)Cl)Cl 12E-312S Cc1c(c(=O)n([nH]1)c2ccccc2)c3cccc(c3)Cl 12E-313S Cc1c(c(=O)n([nH]1)c2cccc(c2)C(F)(F)F)c3cccc(c3)Cl 12E-314S Cc1c(c(=O)n([nH]1)c2cccc(c2)[N+](=O)[O-])c3cccc(c3)Cl 12E-315S c1ccc(cc1)c2c[nH]n(c2=O)c3ccc(cc3)Cl 12E-316S Cc1c(c(=O)n([nH]1)C(C)(C)C)c2ccc(cc2)Cl 12E-318S c1ccc2c(c1)/C(=N/OC(=O)C3CC3)/C(=O)N2Cc4cccc(c4)C(F)(F)F 12E-320S c1ccc2c(c1)/C(=N/OC(=O)CCl)/C(=O)N2Cc3cccc(c3)C(F)(F)F 12E-321S c1ccc2c(c1)/C(=N/OCc3c(cccc3Cl)Cl)/C(=O)N2Cc4ccc(c(c4)Cl)Cl 12E-322S c1ccc2c(c1)C(=O)C(=O)N2Cc3ccc(cc3Cl)Cl 12E-324S Cc1c[n+](ccc1OC)[O-] 12E-326S c1ccc(cc1)CN2c3ccccc3C(C2=O)OC(=O)Nc4ccccc4 12E-328S c1ccc(cc1)CN2c3ccccc3C(C2=O)OC(=O)Nc4ccc(cc4)Cl 12E-329S CCCCC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3cccc(c3)C(F)(F)F 12E-330S c1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3Cl)Cl)/C(=O)N2Cc4cccc(c4)C(F)(F)F 12E-331S c1ccc2c(c1)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/C(=O)N2Cc4cccc(c4)C(F)(F)F 12E-338S c1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3)Cl)/C(=O)N2Cc4cccc(c4)C(F)(F)F 12E-339S c1ccc2c(c1)C3(C(=O)N2)N(C(=O)CS3)c4ccc(cc4)Cl 12E-341S c1ccc(cc1)CN2c3ccccc3C(C2=O)OC(=O)Nc4cccc(c4)Cl 12E-342S c1ccc(cc1)CN2c3ccccc3C(C2=O)OC(=O)c4ccc(cc4)Cl 12E-343S c1ccc(c(c1)c2c[nH]n(c2=O)c3cccc(c3)[N+](=O)[O-])Cl 12E-346S c1ccc(c(c1)c2c[nH]n(c2=O)c3cccc(c3)Cl)Cl 12E-347S c1ccc(c(c1)c2c[nH]n(c2=O)c3ccc(cc3)Cl)Cl 12E-348S c1ccc(cc1)n2c(=O)c(c[nH]2)c3ccccc3Cl 12E-349S c1ccc2c(c1)/C(=N/OCc3ccc(cc3Cl)Cl)/C(=O)N2Cc4ccc(cc4Cl)Cl 12E-351S c1ccc2c(c1)/C(=N/OCc3ccc(c(c3)Cl)Cl)/C(=O)N2Cc4ccc(cc4Cl)Cl 12E-352S c1ccc2c(c1)/C(=N/OCc3ccc(cc3)Cl)/C(=O)N2Cc4ccc(cc4Cl)Cl 12E-353S c1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3ccc(cc3Cl)Cl 12E-354S CO/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3Cl)Cl 12E-355S CCCCC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3Cl)Cl 12E-356S c1ccc2c(c1)/C(=N/OC(=O)CCl)/C(=O)N2Cc3ccc(cc3Cl)Cl 12E-357S c1ccc2c(c1)C3(C(=O)N2)N(C(=O)CS3)c4ccc(cc4)F 12E-358S c1ccc2c(c1)C3(C(=O)N2Cc4ccc(c(c4)Cl)Cl)N(C(=O)CS3)c5ccc(cc5)Cl 12E-361S c1ccc(cc1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5ccc(cc5)F 12E-363S c1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3c(cccc3Cl)Cl 12E-364S c1ccc2c(c1)/C(=N/OCc3ccc(cc3)Cl)/C(=O)N2Cc4c(cccc4Cl)Cl 12E-365S c1ccc2c(c1)/C(=N/OCc3ccc(c(c3)Cl)Cl)/C(=O)N2Cc4c(cccc4Cl)Cl 12E-366S c1ccc2c(c1)/C(=N/OCc3c(cccc3Cl)Cl)/C(=O)N2Cc4c(cccc4Cl)Cl 12E-367S CC(C)(C)C(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3Cl)Cl 12E-369S CC(C)C(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3Cl)Cl 12E-370S c1ccc2c(c1)/C(=N/OC(=O)CCCCl)/C(=O)N2Cc3ccc(cc3Cl)Cl 12E-371S CCOC(=O)c1c(noc1/N=C/N(C)C)OCCOC(=O)c2ccc(cc2Cl)Cl 12E-900 CCOC(=O)c1c(noc1N/C=N/OCc2ccc(cc2)Cl)OCCOC(=O)c3ccc(cc3Cl)Cl 12E-901 CCOC(=O)c1c(noc1NC(=O)c2ccc(cc2)[N+](=O)[O-])OCCOC(=O)c3ccc(cc3)[N+](=O)[O-] 12E-903 COc1ccc(cc1)/C=C/C(=O)Cc2ccccc2 12E-910 Cc1ccc(cc1)/C=C/C(=O)Cc2ccccc2 12E-911 CCOC(=O)c1c(onc1OCCOC(=O)c2cccc(c2)C(F)(F)F)N 12E-913 c1ccc(cc1)C2CC(=O)C(=C(S2)Nc3ccccc3)c4ccccc4 12E-914 CCOC(=O)NC(=O)/C(=C\NNc1ccc(cc1Cl)Cl)/C#N 12E-915 CCOC(=O)c1c(noc1/N=C/N(C)C)OCCOC(=O)c2cccc(c2)C(F)(F)F 12E-916 Cc1ccc(cc1)CON2C(=O)c3ccccc3C2=O 12E-917 CCOC(=O)c1c(noc1NC(=O)c2cccc(c2)C(F)(F)F)OCCOC(=O)c3ccc(cc3Cl)Cl 12E-918 CS/C(=C(\c1ccccc1)/C(=O)/C=C/c2ccccc2)/Nc3ccccc3 12E-919 Cc1ccc(cc1)CON.Cl 12E-920 CCOC(=O)NC(=O)CC(=O)NC(=O)OCC 12E-921 c1ccc2c(c1)C(=O)N(C2=O)OCc3cccc(c3)C(F)(F)F 12E-923 COc1ccc(cc1)C2CC(=O)C(=C(S2)Nc3ccccc3)c4ccccc4 12E-924 c1ccc2c(c1)C(=O)N(C2=O)OCc3c(cccc3Cl)F 12E-925 c1cc(cc(c1)C(F)(F)F)CON.Cl 12E-926 CCOC(=O)c1c(noc1/N=C/NOCc2ccc(cc2)Cl)OCCOC(=O)c3cccc(c3)C(F)(F)F 12E-927 c1cc(c(c(c1)Cl)CON)F.Cl 12E-928 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)CCO 12E-929 c1cc[n+](cc1)CC(=O)c2cccc(c2)[N+](=O)[O-].[I-] 12E-930 Cc1c(c(n(n1)c2ccc(cc2Cl)Cl)O)C(=O)/C=C(/C)\O 12E-932 CN(C)c1nc(c(c(=O)o1)C#N)Nc2ccc(cc2)OC 12E-933 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3cccc(c3)[N+](=O)[O-] 12E-934 CN(C)c1nc(c(c(=O)o1)C#N)Nc2ccc(cc2)Cl 12E-935 CN(C)c1nc(c(c(=O)o1)C#N)N2CCOCC2 12E-936 CN(C)c1nc(c(c(=O)o1)C#N)N2CCCCC2 12E-937 CN(C)c1nc(c(c(=O)o1)C#N)Nc2ccc(cc2F)F 12E-938 Cc1nnc2n1c3ccccc3nc2Cl 12E-939 CCOC(=O)NC(=O)c1cn2c(nc1=O)OCC2 12E-940 Cc1nnc2n1c3ccccc3nc2SCC(=O)OC 12E-941 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)c2ccc(cc2)OC 12E-942 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)CCOC(=O)c2cccc(c2)Cl 12E-943 CN(C)c1nc(c(c(=O)o1)C#N)N2CCN(CC2)c3ccc(cc3)F 12E-944 Cc1cccc(c1N2CCN(CC2)c3c(c(=O)oc(n3)N(C)C)C#N)C 12E-945 Cc1ccc(cc1)C2CC(=O)C(=C(S2)Nc3ccccc3)c4ccccc4 12E-947 Cc1c(oc(n1)N)C(c2ccccc2)O 12E-950 CCOC(=O)c1c(onc1OCCOC(=O)C)N 12E-951 c1cc2c(cc1Cl)n3c(c(n2)Cl)nnc3C(F)(F)F 12E-952 CC1=C(C(=O)c2ccccc2C1=O)CC(=O)c3ccccc3F 12E-953 c1ccc(cc1)Sc2c3nnc(n3c4cc(ccc4n2)Cl)C(F)(F)F 12E-954 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)O 12F-001 CC(C)(C(=O)OCC(=O)c1ccc(cc1)Cl)n2cncn2 12F-002 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 12F-005 CCOC(=O)c1c(onc1c2c(cc(cn2)C(F)(F)F)Cl)C 12F-006 c1ccc(cc1)Sc2ccc(nn2)C(C#N)c3ccc(cc3)Cl 12F-007 c1ccnc(c1)/C(=N/OCc2c(cccc2Cl)F)/N 12F-008 c1cc(c(c(c1)Cl)CO/N=C(/c2cccnc2)\N)F 12F-009 c1cc(c(c(c1)Cl)CO/N=C(/c2ccncc2)\N)F 12F-010 c1cc(ccc1C(C#N)c2ccc(nn2)Sc3ccc(cc3)Cl)Cl 12F-011 CN(C)/C=C/C(=O)/C=C/c1c(cc(cn1)C(F)(F)F)Cl 12F-012 c1ccc(cc1)Sc2ccc(nn2)C(c3ccc(cc3)Cl)C(=O)N 12F-013 c1cc(ccc1C(c2ccc(nn2)Sc3ccc(cc3)Cl)C(=O)N)Cl 12F-014 c1cc(cc(c1)C(F)(F)F)CO/N=C(/c2ccncc2)\N 12F-015 c1c(cnc(c1Cl)c2c([n+](on2)[O-])c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 12F-017 CN(C)c1ccc(nn1)C(C#N)c2ccc(cc2)Cl 12F-018 CN(C)c1ccc(nn1)C(C#N)c2ccccc2 12F-019 c1cc(c(cc1Cl)Cl)C(C#N)c2ccc(nn2)N3CCCC3 12F-021 c1c(cnc(c1Cl)/C(=N/O)/N)C(F)(F)F 12F-022 c1c(cnc(c1Cl)/C(=N/O)/N2CCOCC2)C(F)(F)F 12F-023 c1cc(ccc1C(F)(F)F)N/N=C(\c2c(cc(cn2)C(F)(F)F)Cl)/N=N\c3ccc(cc3)C(F)(F)F 12F-026 c1cc(ccc1N2CCN(CC2)C(=O)c3cc4c(s3)cc(cn4)C(F)(F)F)Cl 12F-027 Cc1c(c(no1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)OC 12F-028 c1cnc(nc1/C=C/c2c(cc(cn2)C(F)(F)F)Cl)N 12F-034 c1cc(ccc1S/C(=N\O)/c2c(cc(cn2)C(F)(F)F)Cl)Cl 12F-037 c1cc(ccc1N/C(=N/O)/c2c(cc(cn2)C(F)(F)F)Cl)Cl 12F-038 c1c(cnc(c1Cl)c2nc(on2)C(F)(F)F)C(F)(F)F 12F-039 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)C(=O)CBr 12F-043 Cc1[nH+]c(cs1)c2cc(n(c2)C)C(=O)C(Cl)(Cl)Cl.[Br-] 12F-046 c1c(cnc(c1Cl)/C(=N/OC(=O)CCC(=O)O)/N)C(F)(F)F 12F-049 c1c(cnc2c1sc(c2)C(=O)N=N#N)C(F)(F)F 12F-051 c1cc(c(cc1Cl)Cl)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl 12F-052 COc1ccc(cc1)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl 12F-053 c1cc(cc(c1)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 12F-054 c1cc(c(c(c1)Cl)CO/N=C\Cc2c(cc(cn2)C(F)(F)F)Cl)Cl 12F-055 c1cc(ccc1C2=C(C(=O)OC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 12F-057 CC(C(=O)OC)n1cncn1 12F-058 CC(C(=O)N)n1cncn1 12F-059 c1ccc(cc1)Oc2ccccc2N/C=C/c3c(cc(cn3)C(F)(F)F)Cl 12F-060 CN(C)S(=O)(=O)c1ccc(cc1)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl 12F-070 c1ccc(c(c1)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl)Cl 12F-071 c1cc(cc(c1)Cl)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl 12F-072 c1cc(ccc1C#N)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl 12F-073 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)N/C=C/c3c(cc(cn3)C(F)(F)F)Cl 12F-074 c1cc(ccc1N/C=C/c2c(cc(cn2)C(F)(F)F)Cl)F 12F-075 c1ccc2c(c1)/C(=N/OC(=O)C(Cl)(Cl)Cl)/C(=O)N2Cc3ccc(cc3)Cl 12F-301S CC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3)Cl 12F-302S CCOC(=O)c1c(nc(s1)c2ccccc2)C 12F-303S Cc1c(c(n(n1)C)Oc2ccc(cc2)Cl)C(=O)Nc3ccccc3 12F-304S Cc1c(c(n(n1)C)Oc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)F 12F-305S Cc1c(c(n(n1)C)Oc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3F)F 12F-306S Cc1c(c(n(n1)C)Oc2cccc(c2)C(F)(F)F)C(=O)O 12F-307S c1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F 12F-308S c1ccc2c(c1)/C(=N/OC(=O)C(Cl)Cl)/C(=O)N2Cc3ccc(cc3)Cl 12F-309S CC(C)(CCl)C(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3)Cl 12F-310S Cc1c(c(n(n1)C)Oc2cccc(c2)Cl)C(=O)O 12F-311S Cc1c(c(n(n1)C)Oc2cccc(c2)C(F)(F)F)C(=O)Nc3ccccc3 12F-312S Cc1c(c(n(n1)C)Oc2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3)F 12F-313S Cc1c(c(n(n1)C)Oc2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F 12F-314S c1ccc2c(c1)/C(=N/OC(=O)CCl)/C(=O)N2Cc3c(cccc3Cl)Cl 12F-316S c1ccc(cc1)c2nc(cs2)C(=O)O 12F-317S c1cc2c(cc1[N+](=O)[O-])/C(=N/O)/C(=O)N2Cc3ccc(cc3Cl)Cl 12F-319S c1cc(ccc1CN2c3ccc(cc3C(=O)C2=O)[N+](=O)[O-])Cl 12F-320S c1cc(c(cc1CN2c3ccc(cc3C(=O)C2=O)Cl)Cl)Cl 12F-321S Cc1c(sc(n1)c2ccccc2)C(=O)O 12F-322S CCOC(=O)c1csc(n1)c2ccc(cc2)Cl 12F-323S Cc1c(c(n(n1)C)Oc2cccc(c2)Cl)C(=O)Nc3ccccc3 12F-327S Cc1c(c(n(n1)C)Oc2cccc(c2)Cl)C(=O)Nc3ccc(cc3)F 12F-328S Cc1c(c(n(n1)C)Oc2cccc(c2)Cl)C(=O)Nc3ccc(cc3F)F 12F-329S Cc1c(c(n(n1)C)Cl)C(=O)O 12F-330S Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc(cc3)Cl 12F-331S Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc(cc3F)F 12F-332S Cc1c(c(n(n1)C)Cl)C(=O)Nc2ccc(cc2)F 12F-336S Cc1c(c(n(n1)C)Cl)C(=O)Nc2ccc(cc2F)F 12F-337S Cc1c(c(n(n1)C)Sc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)F 12F-338S c1cc(ccc1c2nc(cs2)C(=O)O)Cl 12F-339S Cc1c(sc(n1)c2ccccc2)C(=O)Nc3cccc(c3)C(F)(F)F 12F-340S Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)O 12F-341S CC(C)CC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3c(cccc3Cl)Cl 12F-342S CCCCC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3c(cccc3Cl)Cl 12F-343S Cc1c(sc(n1)c2ccccc2Cl)C(=O)O 12F-344S c1ccc(cc1)NC(=O)c2csc(n2)c3ccc(cc3)Cl 12F-345S c1cc(ccc1c2nc(cs2)C(=O)Nc3ccc(cc3F)F)Cl 12F-346S Cc1c(c(n(n1)C)Sc2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3)F 12F-347S Cc1c(c(n(n1)C)Sc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3F)F 12F-348S Cc1c(c(n(n1)C)Sc2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F 12F-349S Cc1c(c(n(n1)C)Sc2cccc(c2)Cl)C(=O)Nc3ccccc3 12F-350S c1cc(c(cc1CN2c3ccc(cc3/C(=N/O)/C2=O)Cl)Cl)Cl 12F-351S CNC(=O)c1csc(n1)c2ccc(cc2)Cl 12F-352S Cc1ccc2c(c1)C(=O)C(=O)N2Cc3ccc(cc3)Cl 12F-353S c1cc2c(cc1[N+](=O)[O-])/C(=N/OC(=O)CCCCl)/C(=O)N2Cc3ccc(cc3Cl)Cl 12F-354S CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3Cl)Cl)[N+](=O)[O-] 12F-355S CC(C)SC1=NC(=CC(N1)(C)C)/C=C/c2c(cccc2Cl)Cl 12F-357S CC(C)CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3Cl)Cl)[N+](=O)[O-] 12F-358S CCCCC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3Cl)Cl)[N+](=O)[O-] 12F-359S c1cc(ccc1CN2c3ccc(cc3/C(=N/O)/C2=O)[N+](=O)[O-])Cl 12F-360S c1ccc2c(c1)/C(=N/OC(=O)C(Cl)Cl)/C(=O)N2Cc3cccc(c3)Cl 12F-361S Cc1c(c(n(n1)C)Sc2cccc(c2)Cl)C(=O)Nc3ccc(cc3)F 12F-362S Cc1c(c(n(n1)C)Sc2cccc(c2)Cl)C(=O)Nc3ccc(cc3F)F 12F-363S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Sc3cccc(c3)Cl 12F-364S CC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3cccc(c3)Cl 12F-365S c1ccc2c(c1)/C(=N/OC(=O)CCl)/C(=O)N2Cc3cccc(c3)Cl 12F-366S c1ccc(cc1)c2nc(cs2)C(=O)Nc3cccc(c3)C(F)(F)F 12F-367S c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccccc3 12F-368S c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc(cc3F)F 12F-369S c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc(cc3)OC(F)(F)F 12F-370S c1ccc2c(c1)/C(=N/OC(=O)CCCCl)/C(=O)N2Cc3cccc(c3)Cl 12F-371S CC(C)CC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3cccc(c3)Cl 12F-372S CCCCC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3cccc(c3)Cl 12F-373S c1cc(ccc1CN2c3ccc(cc3C(=O)C2=O)Cl)Cl 12F-374S c1ccc2c(c1)/C(=N/OC(=O)CCCl)/C(=O)N2Cc3cccc(c3)Cl 12F-375S c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc(cc3)C(F)(F)F 12F-376S CNC(=O)c1csc(n1)c2ccccc2 12F-377S CN(C)CCCNC(=O)c1csc(n1)c2ccccc2 12F-378S C=CCNC(=O)c1csc(n1)c2ccccc2 12F-380S c1ccc(cc1)c2nc(cs2)C(=O)Nc3cccc(c3)Cl 12F-381S c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccccc3Cl 12F-382S c1cc(cc(c1)NC(=O)c2csc(n2)c3ccc(cc3)Cl)C(F)(F)F 12F-383S c1cc(ccc1c2nc(cs2)C(=O)Nc3ccc(cc3)OC(F)(F)F)Cl 12F-384S CCCCC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3)Cl)[N+](=O)[O-] 12F-385S c1cc(ccc1CN2c3ccc(cc3/C(=N/OC(=O)CCl)/C2=O)[N+](=O)[O-])Cl 12F-386S c1cc(ccc1CN2c3ccc(cc3/C(=N/OC(=O)C(Cl)Cl)/C2=O)[N+](=O)[O-])Cl 12F-387S c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc(cc3)Cl 12F-389S c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc(c(c3)Cl)Cl 12F-390S Cc1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3ccc(cc3)Cl 12F-391S c1cc(ccc1CN2c3ccc(cc3/C(=N/O)/C2=O)Cl)Cl 12F-392S CC(C)CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3)Cl)[N+](=O)[O-] 12F-394S CCOC(=O)c1csc(n1)c2cccc(c2)C(F)(F)F 12F-395S c1cc(ccc1CN2c3ccc(cc3/C(=N/OC(=O)CCCl)/C2=O)[N+](=O)[O-])Cl 12F-396S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Sc3ccc(cc3)C(F)(F)F 12F-398S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Sc3ccc(c(c3)Cl)Cl 12F-399S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Sc3ccc(cc3Cl)Cl 12F-400S C/N=C(/c1cccc(c1)C(F)(F)F)\N(C)c2ccc(cc2)Cl 12F-401S CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(c(c3)Cl)Cl)Cl 12F-403S c1cc(c(cc1CN2c3ccc(cc3/C(=N/OC(=O)CCl)/C2=O)Cl)Cl)Cl 12F-404S CC(C)CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(c(c3)Cl)Cl)Cl 12F-405S CC(C)SC1=NC(=CC(N1)(C)C)/C=C/c2ccc(cc2Cl)Cl 12F-406S c1cc(cc(c1)C(F)(F)F)c2nc(cs2)C(=O)O 12F-407S c1cc(cc(c1)C(F)(F)F)c2nc(cs2)C(=O)Nc3cccc(c3)C(F)(F)F 12F-408S c1cc(cc(c1)C(F)(F)F)c2nc(cs2)C(=O)Nc3ccc(cc3F)F 12F-409S c1cc(cc(c1)C(F)(F)F)c2nc(cs2)C(=O)Nc3ccc(c(c3)Cl)Cl 12F-410S c1cc(cc(c1)C(F)(F)F)c2nc(cs2)C(=O)Nc3ccc(cc3)Cl 12F-411S COc1ccc(cc1)C2C(=C(C2=O)c3ccc(cc3)OC)O 12F-414S CCOC(=O)CN/C=C(\C(=O)C)/C(=O)Nc1nccs1 12F-900 CC(=O)CC(=O)NC(=O)CCl 12F-901 CC(=O)C(/C=N/OCc1ccc(cc1)[N+](=O)[O-])C(=O)Nc2nccs2 12F-902 c1cc(ccc1SCc2csc(n2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 12F-903 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)C4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 12F-904 Cc1cc(nc(c1)N/C=C(\C(=O)C)/C(=O)NC(=O)CCl)C 12F-905 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=S)NC(=O)N 12F-906 c1ccc(cc1)CN2CCN(CC2)C(=O)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 12F-907 c1cc(ccc1NC(=O)N)F 12F-908 c1cc(ccc1NC(=O)N)Cl 12F-909 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3nc(=O)[nH]s3 12F-910 Cc1ccc(cc1)C(=O)NC(=S)NC(=O)N 12F-911 c1cc(ccc1CONS(=O)(=O)c2ccc(cc2)Cl)Cl 12F-913 Cc1ccc(cc1)C(=O)Nc2nc(=O)[nH]s2 12F-914 c1ccc(cc1)C(=O)NC(=S)N2[C@H]3c4c5ccccc5ccc4OC[C@H]3CO2 12F-915 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=S)NC(=O)Nc3ccc(cc3)Cl 12F-916 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4C(=S)N 12F-918 c1cc(ccc1C(/C=N/OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C#N)Cl 12F-919 CC(=O)/C(=C\NCC(=O)O)/C(=O)Nc1nccs1 12F-920 Cc1ccc(cc1)c2ncc(c(n2)C)C(=O)Nc3nccs3 12F-921 CN1CCc2c(sc(c2C(=O)OC)N)C1.O 12F-922 Cc1c(cnc(n1)N)C(=O)Nc2nccs2 12F-923 Cc1cc(nc(n1)N/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl)C 12F-924 Cc1ccc(cc1)C2=N/C(=C/Nc3nc(cc(n3)C)C)/C(=O)O2 12F-925 Cc1cc(nc(n1)N/C=C/2\C(=O)OC(=N2)c3ccccc3)C 12F-926 Cc1cc(nc(n1)N/C=C/2\C(=O)OC(=N2)c3ccc(cc3)F)C 12F-927 Cc1cc(nc(n1)N/C=C/2\C(=O)OC(=N2)c3ccc(cc3)OC)C 12F-928 Cc1ccnc(n1)N/C=C(\C(=O)N/N=C\c2ccc(cc2)Cl)/NC(=O)c3ccccc3 12F-929 Cc1ccnc(n1)N/C=C(\C(=O)N/N=C\c2ccccc2)/NC(=O)c3ccccc3 12F-930 Cc1ccc(cc1)/C=N\NC(=O)/C(=C\Nc2nccc(n2)C)/NC(=O)c3ccccc3 12F-931 Cc1ccnc(n1)N/C=C(\C(=O)N/N=C\c2ccc(cc2)OC)/NC(=O)c3ccccc3 12F-932 Cc1ccnc(n1)N/C=C(\C(=O)N/N=C\c2ccc(cc2)F)/NC(=O)c3ccccc3 12F-933 CCCCOC(=O)CC(=O)C 12F-934 Cc1ccc(cc1)C(=O)NC(=S)NC(=O)NC 12F-935 CNC(=O)NC(=S)NC(=O)c1ccccc1 12F-936 CNC(=O)NC(=S)NC(=O)c1ccc(cc1)Cl 12F-937 CCCCOC(=O)c1cc2c(=O)c3cc(ccc3oc2nc1C)F 12F-939 Cn1c(=O)nc(s1)NC(=O)c2ccccc2 12F-940 Cn1c(=O)nc(s1)NC(=O)c2ccc(cc2)Cl 12F-941 Cc1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C 12F-942 CNC(=O)NC(=S)NC(=O)c1ccccc1Cl 12F-943 CNC(=O)NC(=S)NC(=O)c1ccc(cc1)OC 12F-944 Cc1ccc(cc1)NC(=O)ON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 12F-945 c1ccc(cc1)NC(=O)ON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 12F-946 c1cc(cc(c1)NC(=O)ON=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 12F-947 Cn1c(=O)nc(s1)NC(=O)c2ccccc2Cl 12F-948 Cn1c(=O)nc(s1)NC(=O)c2cccc(c2)Cl 12F-949 Cn1c(=O)nc(s1)NC(=O)c2ccc(cc2)OC 12F-950 c1c(cnc(c1Cl)N2CCC(CC2)O)C(F)(F)F 12F-951 COc1ccc(cc1)C(=O)OC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 12F-952 C1CN(CCC1=O)C(=O)N 12F-953 c1cc(ccc1C(=O)OCC(CO)n2cc(ccc2=O)[N+](=O)[O-])Cl 12F-955 CNC(=O)NC(=S)NC(=O)c1cccc(c1)Cl 12F-962 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Oc3ccccc3)O 12G-001 CCOC(=O)C(Cc1ccc(cc1)C(=O)OC)(C(=O)OCC)NC(=O)C 12G-002 Cc1nc(cn1c2c(cc(cn2)C(F)(F)F)Cl)/C(=N/OC(=O)c3ccc(cc3)Cl)/C 12G-003 c1ccc(cc1)Oc2ccc(cc2)n3c(=O)cc(c(n3)C(=O)N)O 12G-005 COc1cc(=O)n(nc1C#N)c2cccc(c2)C(F)(F)F 12G-006 C#CCSc1nc2ncc(cn2n1)C#N 12G-008 COc1cccc(c1)n2c(=O)cc(c(n2)C(=O)N)O 12G-009 Cn1cccc1C(CC#N)(C#N)c2cccc(c2C#N)F 12G-010 c1cc(c(c(c1)F)C#N)C(CCC#N)(C#N)c2ccc(cc2)F 12G-011 CCOC(=O)C(Cc1c(cc(cn1)C(F)(F)F)Cl)(C(=O)OCC)NC(=O)C 12G-012 c1ccc(cc1)Oc2ccc(cc2)n3c(=O)cc(c(n3)C#N)Cl 12G-013 COc1cccc(c1)n2c(=O)cc(c(n2)C#N)Cl 12G-014 Cn1cccc1C2(c3cccc(c3C(=C2C(=O)OC)N)F)C#N 12G-015 c1c(cnc(c1Cl)CC(C(=O)O)N)C(F)(F)F 12G-016 COc1cccc(c1)NS(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl 12G-017 c1cc(ccc1NS(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl 12G-018 c1cc(c(c(c1)F)C#N)C(C#N)c2cccs2 12G-019 c1cc2c(c(c1)F)C(=C(C2(C#N)c3cccs3)C#N)N 12G-020 COC(=O)C1=C(c2c(cccc2F)C1(C#N)c3cccs3)N 12G-021 C=CCNC(=S)n1cc(cn1)c2c(cc(cn2)C(F)(F)F)Cl 12G-022 c1c(cnc(c1Cl)c2cnn(c2)C(=O)C(F)(F)F)C(F)(F)F 12G-023 c1c(cn(n1)C2CCS(=O)(=O)C2)c3nc[nH]n3 12G-024 c1ccc(cc1)C2CC(=O)c3c2cccc3Sc4ccccc4 12G-026 c1cc(ccc1CON/C(=N\C(=O)Nc2ccc(cc2Cl)Cl)/Cn3cncn3)Cl 12G-027 CCCCCCCCCCC(=O)c1cc([nH]c1)C(=O)O 12G-030 Cn1cccc1C2(c3cccc(c3C(=C2C#N)N)F)C#N 12G-031 CSc1cc(=O)n(nc1C#N)c2cccc(c2)C(F)(F)F 12G-032 CCCCCCCCCCC(=O)c1cc([nH]c1)C(=O)[O-].[Na+] 12G-033 c1cc(c(c(c1)F)C#N)C(C#N)c2c(cccc2Cl)F 12G-034 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N3CCOCC3 12G-035 c1ccc(cc1)C2CC(=O)c3c2cccc3N4CCCC4 12G-036 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NN 12G-039 c1c(cnc(c1Cl)S)C(F)(F)F 12G-041 COc1cc(=O)n(nc1C(=N)NNC(=O)c2ccc(cc2)Cl)c3cccc(c3)C(F)(F)F 12G-042 c1cc(ccc1/C=N/NS(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl 12G-043 c1c(cnc(c1Cl)SCC#N)C(F)(F)F 12G-044 c1c(cnc(c1Cl)SCC(=C(C#N)C#N)N)C(F)(F)F 12G-045 c1cc(ccc1C(=O)NNC(=N)CSc2c(cc(cn2)C(F)(F)F)Cl)Cl 12G-046 c1cnccc1C(=O)NNC(=N)CSc2c(cc(cn2)C(F)(F)F)Cl 12G-047 c1c(cnc(c1Cl)SCC(=N)NNC(=O)CC#N)C(F)(F)F 12G-048 c1c(cnc(c1Cl)SCC(=[NH2+])N)C(F)(F)F.[Cl-] 12G-049 c1c(cnc(c1Cl)SCc2nc([nH]n2)CC#N)C(F)(F)F 12G-050 CC(C)OC(=O)c1c(snn1)Sc2ccc(cc2)Cl 12G-301S c1ccc(cc1)NC(=O)c2c(snn2)S(=O)c3ccc(cc3)Cl 12G-302S c1cc(ccc1S(=O)c2c(nns2)C(=O)Nc3ccc(c(c3)Cl)Cl)Cl 12G-303S CNC(=O)c1c(snn1)S(=O)c2ccc(cc2)Cl 12G-304S c1cc(ccc1S(=O)c2c(nns2)C(=O)N3CCOCC3)Cl 12G-305S c1cc(ccc1S(=O)c2c(nns2)C(=O)N3CCCCC3)Cl 12G-306S c1ccc(c(c1)NC(=O)c2cccnc2Cl)N3CCOCC3 12G-307S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccccc2N3CCOCC3 12G-308S c1ccc(c(c1)NC(=O)CCCCl)N2CCOCC2 12G-309S CC(C)(C)c1ccc(cc1)OC(C(=O)NC(C)(C)C)(F)F 12G-310S CC(C)(C)c1ccc(cc1)OC(C(=O)Nc2ccc(cc2)OC(F)(F)F)(F)F 12G-311S CC(C)(C)c1ccc(cc1)OC(C(=O)Nc2cc(cc(c2)Cl)Cl)(F)F 12G-312S CN(C)C(=O)c1c(snn1)S(=O)c2ccc(cc2)Cl 12G-314S c1cc(ccc1Sc2c(nns2)C(=O)OC3CCCCC3)Cl 12G-315S c1ccc2c(c1)c(ccc2Cl)Oc3ccc(cc3[N+](=O)[O-])F 12G-318S c1cc(cc(c1)NC(=O)c2c(snn2)S(=O)c3ccc(cc3)Cl)C(F)(F)F 12G-319S CCCNC(=O)c1c(snn1)S(=O)c2ccc(cc2)Cl 12G-320S CN1CCN(CC1)c2ccccc2NC(=O)c3ccc(cc3Cl)Cl 12G-321S CN1CCN(CC1)c2ccccc2NC(=O)c3ccccc3Cl 12G-323S CN(C)/C=C(\C#N)/S(=O)(=O)c1ccccc1 12G-324S CCOC(=O)c1c(snn1)Sc2ccc(cc2)C 12G-325S CCNC(=O)c1c(snn1)S(=O)c2ccc(cc2)Cl 12G-326S CN1CCN(CC1)c2ccccc2NC(=O)c3cccc(c3)Cl 12G-328S CN1CCN(CC1)c2ccccc2NC(=O)c3ccc(cc3)Cl 12G-330S CC(C)(C)C(=O)Nc1ccccc1N2CCN(CC2)C 12G-331S CN1CCN(CC1)c2ccccc2NC(=O)C(Cl)(Cl)Cl 12G-335S CN1CCN(CC1)c2ccccc2NC(=O)c3cccc(c3)C(F)(F)F 12G-336S CN1CCN(CC1)c2ccccc2NC(=O)c3c(cccc3F)F 12G-337S c1cc(ccc1S(=O)(=O)c2c(nns2)C(=O)N3CCCCC3)Cl 12G-341S c1cc(ccc1S(=O)(=O)c2c(nns2)C(=O)N3CCOCC3)Cl 12G-342S CN(C)C(=O)c1c(snn1)S(=O)(=O)c2ccc(cc2)Cl 12G-343S CC(C)(CCl)C(=O)Nc1ccccc1N2CCN(CC2)C 12G-344S CN1CCN(CC1)c2ccccc2NC(=O)C(c3ccccc3)Cl 12G-345S CCOC(=O)c1nc(n(n1)c2ccc(cc2)[N+](=O)[O-])C 12G-347S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)O 12G-348S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3ccc(cc3Cl)Cl 12G-351S CCOC(=O)c1c(snn1)Sc2cccc(c2)C(F)(F)F 12G-352S CCOC(=O)c1c(snn1)S(=O)(=O)c2ccc(cc2)C 12G-353S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)Cc3ccccc3)C 12G-355S CNC(=O)c1c(snn1)S(=O)(=O)c2ccc(cc2)Cl 12G-356S Cc1ccc(cc1)C(=O)Nc2ccccc2N3CCN(CC3)C 12G-361S CN1CCN(CC1)c2ccccc2NC(=O)c3cccnc3Cl 12G-362S CN1CCN(CC1)c2ccccc2NC(=O)c3ccc(cc3Cl)S(=O)(=O)C 12G-363S CN1CCN(CC1)c2ccccc2NC(=O)c3cc(cc(c3)Cl)Cl 12G-364S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)Cc3ccc(c(c3)Cl)Cl)C 12G-365S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)Cc3ccc(cc3)Cl)C 12G-366S CN1CCN(CC1)c2ccccc2NC(=O)c3ccc(c(c3)Cl)Cl 12G-367S CCOC(=O)c1nc(n(n1)c2ccc(cc2)Cl)C 12G-368S c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(c3c2nccc3)Cl 12G-369S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)O 12G-370S CCOC(=O)c1c(snn1)S(=O)(=O)c2ccccc2 12G-372S c1cc(ccc1NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Br)Cl 12G-376S c1cc(cc(c1)NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Br)C(F)(F)F 12G-377S c1ccc(cc1)NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Br 12G-378S c1cc(ccc1NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Br)F 12G-380S c1cc(ccc1S(=O)(=O)N2CCCC2C(=O)Nc3ccc(c(c3)F)F)Br 12G-381S c1cc(ccc1NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Cl)Cl 12G-382S c1ccc(cc1)NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Cl 12G-383S c1cc(cc(c1)NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F 12G-384S c1cc(ccc1NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)F)OC(F)(F)F 12G-386S c1cc(cc(c1)NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)F)C(F)(F)F 12G-387S c1cc(ccc1F)S(=O)(=O)N2CCCC2C(=O)Nc3ccc(c(c3)F)F 12G-388S c1cc(ccc1NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)F)Cl 12G-389S c1ccc(c(c1)S(=O)(=O)N2CCCC2C(=O)Nc3cccc(c3)C(F)(F)F)Cl 12G-391S CC(C)CC(C(=O)Nc1ccc(cc1)OC(F)(F)F)NS(=O)(=O)c2ccc(cc2)F 12G-392S CC(C)CC(C(=O)Nc1ccc(cc1)Cl)NS(=O)(=O)c2ccc(cc2)F 12G-393S CC(C)CC(C(=O)Nc1cccc(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)F 12G-394S Cc1ccc(cc1C)NC(=O)C(CC(C)C)NS(=O)(=O)c2ccc(cc2)F 12G-395S CC(C(=O)O)NS(=O)(=O)c1ccc(cc1)Cl 12G-396S CC(C(=O)Nc1cccc(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)Cl 12G-397S Cc1ccc(cc1C)NC(=O)C(C)NS(=O)(=O)c2ccc(cc2)F 12G-400S CC(C(=O)Nc1ccccc1Cl)NS(=O)(=O)c2ccc(cc2)F 12G-401S CC(C)C(C(=O)Nc1ccc(cc1)OC(F)(F)F)NS(=O)(=O)c2ccc(cc2)Cl 12G-402S Cc1ccc(cc1)NC(=O)C(C(C)C)NS(=O)(=O)c2ccc(cc2)Cl 12G-404S CC(C)C(C(=O)Nc1cccc(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)Cl 12G-405S CC(C)C(C(=O)Nc1cccc(c1)Cl)NS(=O)(=O)c2ccc(cc2)Cl 12G-407S c1cc(ccc1NC(=O)OCc2ccc(nc2)Cl)Cl 12G-412S c1cc(ccc1C(=O)OCc2ccc(nc2)Cl)Cl 12G-413S c1cc(cc(c1)Cl)NC(=O)C2CCCN2S(=O)(=O)c3ccc(cc3)Br 12G-414S c1cc(ccc1S(=O)(=O)N2CCCC2C(=O)N3CCOCC3)Br 12G-415S CC(C(=O)O)NS(=O)(=O)c1ccc(cc1)F 12G-417S c1cc(ccc1S(=O)(=O)NCC(=O)O)Cl 12G-418S c1cc(ccc1S(=O)(=O)NCC(=O)O)Br 12G-419S c1cc(ccc1NC(=O)CNS(=O)(=O)c2ccc(cc2)F)OC(F)(F)F 12G-422S CCOC(=O)c1c(snn1)S(=O)c2ccccc2 12G-424S c1cc(ccc1F)S(=O)(=O)NCC(=O)Nc2ccc(c(c2)F)F 12G-425S c1cc(ccc1S(=O)(=O)NOCC(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 12G-900 c1cc(ccc1NC(=O)NOCC(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 12G-901 CC1=CSC2=[N+](CCN12)CC(=O)c3ccccc3.[Br-] 12G-902 CCOC(=O)NC(=O)C(/C=N/CCNc1c(cc(cn1)C(F)(F)F)Cl)C#N 12G-904 c1c(cnc(c1Cl)N2CCC(=CC2)N3CCOCC3)C(F)(F)F 12G-905 CCOC(=O)/C=C\S/C=C(\C)/N1CCn2c1c(cc2C(=O)c3ccccc3)C(=O)OCC 12G-907 CCOC(=O)/C=C\S/C=C(\C)/N1CCn2c1c(cc2C(=O)C)C(=O)OCC 12G-909 c1c(cnc(c1Cl)N2CCC(=CC2)N3CCCCC3)C(F)(F)F 12G-911 CN1CCC(=CC1)N2CCN(CC2)c3ccccc3 12G-912 c1ccc2c(c1)CCC3=C2CCN(C3)CCNc4c(cc(cn4)C(F)(F)F)Cl.Cl 12G-913 CN1CCC(=CC1)N2CCOCC2 12G-915 CC(=O)CC(=O)Nc1cccc(c1)Cl 12G-916 CC(=O)CC(=O)Nc1ccccc1Cl 12G-917 C/C(=C\C(=O)Nc1ccccc1)/N2CCN(CC2)c3ccc(cc3)Cl 12G-918 C/C(=C\C(=O)Nc1ccc(cc1)Cl)/N2CCN(CC2)c3ccc(cc3)Cl 12G-919 C/C(=C\C(=O)Nc1cccc(c1)Cl)/N2CCN(CC2)c3ccc(cc3)Cl 12G-920 CN([C@H]1c2cc(ccc2OC[C@H]1CO)Br)C(=S)Nc3ccc(cc3)[N+](=O)[O-] 12G-921 C/C(=C\C(=O)Nc1ccccc1Cl)/N2CCN(CC2)c3ccc(cc3)Cl 12G-922 c1cc(c(cc1N2CCN(CC2)C(=O)CC(=O)N3CCN(CC3)c4ccc(c(c4)Cl)Cl)Cl)Cl 12G-923 c1cc(ccc1CC(C(=O)O)N)CO 12G-925 COC(=O)C(Cc1ccccc1)/N=C/c2ccc(cc2)Cl 12G-928 COC(=O)C1(C2C(C(N1)c3ccccc3)C(=O)N(C2=O)Cc4ccccc4)Cc5ccccc5 12G-932 COC(=O)C1(C2C(C(N1)c3ccc(cc3)Cl)C(=O)N(C2=O)Cc4ccccc4)Cc5ccccc5 12G-933 CCOC(=O)c1cc(c(=O)[nH]c1NN)C(=O)OCC 12G-934 COC(=O)C1(C2C(C(N1)c3cccc(c3)Cl)C(=O)N(C2=O)Cc4ccccc4)Cc5ccccc5 12G-935 COC(=O)C1(C2C(C(N1)c3ccccc3Cl)C(=O)N(C2=O)Cc4ccccc4)Cc5ccccc5 12G-936 c1cc(cnc1)/C(=N/Nc2ccc(cc2Cl)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 12H-001 c1cc(cnc1)c2c3c(cc(cn3)C(F)(F)F)n(n2)c4ccc(cc4Cl)Cl 12H-002 c1ccc(cc1)Oc2cc(cnc2C(=O)c3ccc(cc3Cl)Cl)C(F)(F)F 12H-003 c1cc(cnc1)/C(=N/Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])/c3c(cc(cn3)C(F)(F)F)Cl 12H-005 c1ccc(cc1)N/N=C(\c2cccnc2)/c3c(cc(cn3)C(F)(F)F)Cl 12H-006 c1ccc(cc1)n2c3cc(cnc3c(n2)c4cccnc4)C(F)(F)F 12H-008 c1cc(c(cc1Cl)Cl)C(=O)c2c(cc(cn2)C(F)(F)F)Oc3ccc(cc3Cl)Cl 12H-009 c1ccc(cc1)Oc2cc(cnc2C(c3ccc(cc3Cl)Cl)O)C(F)(F)F 12H-012 Cn1ccnc1CO 12H-013 CO/N=C/c1c(c(sc1Nc2ccccc2)C(=O)c3ccccc3)N 12H-014 c1cc(c(cc1Cl)Cl)C(c2c(cc(cn2)C(F)(F)F)Oc3ccc(cc3Cl)Cl)O 12H-016 Cc1c(c(ccn1)N2CCN(CC2)C)Oc3c(cc(cn3)C(F)(F)F)Cl 12H-017 Cc1cccc(c1)c2nc(c(c(n2)O)C#N)c3ccc(cc3)OC 12H-020 c1ccc(cc1)N/N=C(\c2ccc(cc2Cl)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 12H-021 c1ccc(cc1)n2c3cc(cnc3c(n2)c4ccc(cc4Cl)Cl)C(F)(F)F 12H-022 Cc1cccc(c1)c2nc(c(c(n2)Cl)C#N)c3ccc(cc3)OC 12H-024 Cc1cccc(c1)c2nc(c(c(n2)N3CCN(CC3)C)C#N)c4ccc(cc4)OC 12H-025 c1cn(cn1)c2c(cc(cn2)C(F)(F)F)Cl 12H-026 CN(C)c1cc(cnc1C(=O)c2ccccc2)C(F)(F)F 12H-031 c1cc(cc(c1)C(F)(F)F)C(=O)CSc2ncc(c(n2)C(F)(F)F)C#N 12H-033 CN(C)c1cc(cnc1C(=O)c2ccc(cc2)Cl)C(F)(F)F 12H-034 CN1CCN(CC1)c2cc(cnc2C(=O)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F 12H-035 c1cc(ccc1C(=O)c2c(cc(cn2)C(F)(F)F)N3CCOCC3)[N+](=O)[O-] 12H-036 c1ccc(cc1)N2CCN(CC2)c3cc(cnc3C(=O)c4ccc(cc4)Cl)C(F)(F)F 12H-038 CN(C)c1cc(cnc1C(=O)c2ccc(cc2)[N+](=O)[O-])C(F)(F)F 12H-040 CCC(C)(C)NC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])F 12H-301S CC(C)(C#C)NC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])F 12H-302S c1cc(ccc1c2c3c(n[nH]2)CCC3)Cl 12H-303S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4c(ccs4)Oc5ccc(cc5[N+](=O)[O-])F 12H-304S COC(=O)c1ccccc1NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F 12H-305S Cc1cccc(c1NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F)C 12H-306S c1ccc(cc1)Oc2ccc(cc2)NC(=O)c3c(ccs3)Oc4ccc(cc4[N+](=O)[O-])F 12H-307S Cc1c(cccc1Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F 12H-308S c1cc(c(cc1NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])F)F)F 12H-309S Cc1ccc(cc1)c2c3c(n[nH]2)CCC3 12H-311S c1ccc(cc1)NC(=O)c2c(ccs2)Oc3ccc(c(c3)C(F)(F)F)[N+](=O)[O-] 12H-312S c1cc(ccc1NC(=O)c2c(ccs2)Oc3ccc(c(c3)C(F)(F)F)[N+](=O)[O-])F 12H-313S c1cc(ccc1C(F)(F)F)NC(=O)c2c(ccs2)Oc3ccc(c(c3)C(F)(F)F)[N+](=O)[O-] 12H-314S CC(C)(C#C)NC(=O)c1c(ccs1)Oc2ccc(c(c2)C(F)(F)F)[N+](=O)[O-] 12H-315S c1ccc(cc1)C(CNCc2ccc(cc2)Cl)(c3ccccc3)O 12H-316S Cc1cc2c(c(c1C)[N+](=O)[O-])nc[nH]2 12H-317S Cc1ccc(cc1)CNCC(c2ccccc2)(c3ccccc3)O 12H-318S Cc1cc(nc(c1C#N)OC(=O)c2ccccc2C(=O)OC)C 12H-319S COc1ccc(cc1)CNCC(c2ccccc2)(c3ccccc3)O 12H-320S COc1cccc(c1)C[NH2+]CC(c2ccccc2)(c3ccccc3)O.[Cl-] 12H-321S Cc1cc2c(c(c1C)[N+](=O)[O-])ncn2Cc3ccccc3 12H-322S COc1cccc(c1)c2c3c(n[nH]2)CCC3 12H-323S c1ccc(cc1)C(C[NH2+]Cc2cccc[nH+]2)(c3ccccc3)O.[Cl-].[Cl-] 12H-324S c1ccc(cc1)C(C[NH2+]Cc2ccccc2Cl)(c3ccccc3)O.[Cl-] 12H-325S c1ccc(cc1)C(C[NH2+]Cc2cccc(c2)Cl)(c3ccccc3)O.[Cl-] 12H-326S c1ccc(cc1)C(CNCc2ccc(cc2)F)(c3ccccc3)O 12H-328S c1ccc(cc1)C(CNCc2ccc(cc2Cl)Cl)(c3ccccc3)O 12H-329S c1ccc(cc1)C(CNCc2cccc(c2)Cl)(c3ccc(cc3)Cl)O.Cl 12H-333S c1ccc(cc1)C(C[NH2+]Cc2ccc(cc2)Cl)(c3ccc(cc3)Cl)O.[Cl-] 12H-334S c1ccc(cc1)C(C[NH2+]Cc2ccc(c(c2)Cl)Cl)(c3ccc(cc3)Cl)O.[Cl-] 12H-335S c1cc(c(cc1Cl)Cl)c2c3c(n[nH]2)CCC3 12H-337S Cc1cc(nc(c1C#N)OC(=O)c2ccc(cc2)C(=O)OC)C 12H-338S Cc1ccc(cc1)CNCC(c2ccccc2)(c3ccc(cc3)Cl)O 12H-339S Cc1cc(nc(c1C#N)OC(=O)c2ccc(cc2)S(=O)(=O)N(C)C)C 12H-340S CC(=O)c1ccccc1NS(=O)(=O)c2ccccc2F 12H-341S CC(=O)c1ccccc1NS(=O)(=O)c2ccccc2C(F)(F)F 12H-342S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2)C(F)(F)F 12H-343S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2F)F 12H-344S CC(=O)c1ccccc1NS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] 12H-346S Cc1cc(nc(c1C#N)OC(=O)c2cccc(c2)S(=O)(=O)N(C)C)C 12H-347S c1ccc2c(c1)[nH]c(n2)/C=C/c3c(cccc3Cl)Cl 12H-348S c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4c(cccc4Cl)Cl 12H-349S COc1ccc(cc1)CNCC(c2ccccc2)(c3ccc(cc3)Cl)O 12H-350S c1ccc(cc1)C(CNCc2cccc(c2)C(F)(F)F)(c3ccc(cc3)Cl)O.Cl 12H-351S c1cc(c(cc1c2c3c(n[nH]2)CCC3)Cl)Cl 12H-352S COc1cccc(c1)C[NH2+]CC(c2ccccc2)(c3ccc(cc3)Cl)O.[Cl-] 12H-353S COc1ccccc1C[NH2+]CC(c2ccccc2)(c3ccccc3)O.[Cl-] 12H-354S c1ccc2c(c1)C3=NC(CN3C(=O)N2)CN4CCN(CC4)c5ccc(cc5)F 12H-503S c1ccc2c(c1)C3=NC(CN3C(=O)N2)CN4CCN(CC4)c5ccccc5F 12H-504S c1ccc2c(c1)C3=NC(CN3C(=O)N2)CN4CCN(CC4)c5cccc(c5)C(F)(F)F 12H-505S c1cc2c(cc1Cl)c(=O)oc(n2)Nc3ccc(cc3Cl)Cl 12H-512S c1cc(cc(c1)Nc2nc3ccc(cc3c(=O)o2)Cl)C(F)(F)F 12H-514S c1cc(ccc1C(F)(F)F)Nc2nc3ccc(cc3c(=O)o2)Cl 12H-515S c1ccc2c(c1)[nH]c(n2)/C=C/c3ccc(cc3)Cl 12H-516S c1ccc(cc1)/C=C/c2[nH]c3ccccc3n2 12H-517S c1ccc2c(c1)nc(n2Cc3cccc(c3)C(F)(F)F)/C=C/c4ccc(cc4)Cl 12H-518S c1ccc2c(c1)nc(n2Cc3ccc(c(c3)Cl)Cl)/C=C/c4ccc(cc4)Cl 12H-519S CCOC(=O)Cn1c2ccccc2nc1/C=C/c3ccc(cc3)Cl 12H-520S c1ccc(cc1)CN2CCN(CC2)CC3CN4C(=N3)c5ccccc5NC4=O 12H-522S c1ccc2c(c1)nc(n2Cc3cc(ccc3Cl)Cl)/C=C/c4ccc(cc4)Cl 12H-523S CC(C)(C)c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccc(cc4)Cl 12H-524S c1ccc(cc1)/C=C/c2nc3ccccc3n2Cc4ccc(cc4Cl)Cl 12H-527S c1ccc(cc1)/C=C/c2nc3ccccc3n2Cc4c(cccc4Cl)Cl 12H-528S COc1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccccc4 12H-529S CCOC(=O)Cn1c2ccccc2nc1/C=C/c3ccccc3 12H-530S c1ccc(cc1)/C=C/c2nc3ccccc3n2Cc4ccccc4Cl 12H-531S CC(C)(C)c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccccc4 12H-532S CC(C)Oc1c(ccc(n1)c2ccccc2Cl)C#N 12H-533S CCOCCOc1c(ccc(n1)c2ccccc2Cl)C#N 12H-534S COc1c(ccc(n1)c2ccccc2Cl)C#N 12H-535S COc1ccc(cc1)c2ccc(c(n2)Cl)C#N 12H-536S COc1ccc(cc1)c2ccc(c(n2)OC)C#N 12H-537S CC(C)Oc1c(ccc(n1)c2ccc(cc2)OC)C#N 12H-539S CCOCCOc1c(ccc(n1)c2ccc(cc2)OC)C#N 12H-540S c1ccc(c(c1)c2ccc(c(n2)Oc3ccccc3Cl)C#N)Cl 12H-541S c1ccc(c(c1)c2ccc(c(n2)Oc3ccc(cc3)F)C#N)Cl 12H-542S c1ccc(c(c1)c2ccc(c(n2)Oc3ccc(cc3F)F)C#N)Cl 12H-543S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC4CN5C(=N4)c6ccccc6NC5=O 12H-544S CCOc1c(ccc(n1)c2ccccc2Cl)C#N 12H-831S CNC(=S)NNC(=O)Cc1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 12H-900 C=CCNC(=O)C1CCN(CC1)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 12H-901 c1ccc(cc1)C2CC(ON2c3ccccc3)CNC(=O)C4CCN(CC4)c5ccc(cc5)[N+](=O)[O-] 12H-902 c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Cl 12H-903 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Cl)Cl 12H-904 Cn1c(nnc1S)Cc2c[nH]c3c2cccc3 12H-905 CC(=O)C1=NOC(C1)CNC(=O)C2CCN(CC2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 12H-906 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Cl 12H-907 C=CCN(c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl 12H-908 c1cc(cc(c1)N/C=C/2\C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 12H-909 CO/N=C\C1C(=O)NC(=O)N(C1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl 12H-910 C=CCN(c1ccccc1)S(=O)(=O)c2ccc(cc2)Cl 12H-911 c1c(cnc(c1Cl)NCCn2c(=O)cc([nH]c2=O)Cl)C(F)(F)F 12H-912 CCOC(=O)C1=NOC(C1)CNC(=O)C2CCN(CC2)c3ncccn3 12H-913 c1ccc(cc1)C2CC(=O)CC(=O)C2 12H-914 c1ccc(cc1)C2CC(ON2c3ccccc3)CN(c4ccccc4)S(=O)(=O)c5ccc(cc5)Cl 12H-915 c1ccc(cc1)C2CC(ON2c3ccccc3)CN(c4ccc(cc4)Cl)S(=O)(=O)c5ccc(cc5)Cl 12H-916 c1cc(ccc1/C=C/2\C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)Cl 12H-917 C=CCN(c1ccc(cc1)Cl)S(=O)(=O)c2ccccc2 12H-918 CC(=O)/C=C/c1ccc(cc1)OC 12H-919 CCOC(=O)C1=NOC(C1)CN(c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 12H-920 c1ccc(cc1)CNc2cc(=O)n(c(=O)[nH]2)CCNc3c(cc(cn3)C(F)(F)F)Cl 12H-921 c1ccnc(c1)Sc2cc(=O)n(c(=O)[nH]2)CCNc3c(cc(cn3)C(F)(F)F)Cl 12H-922 CCOC(=O)C1=NOC(C1)CN(c2ccccc2)S(=O)(=O)c3ccc(cc3)Cl 12H-923 c1ccc(cc1)C2CC(=O)C(C(=O)C2)CS(=O)(=O)c3ccccc3 12H-924 COc1ccc(cc1)C2CC(=O)CC(=O)C2 12H-925 CCOC(=O)C1=NOC(C1)CN(c2ccc(cc2)Cl)S(=O)(=O)c3ccccc3 12H-926 COc1ccc(cc1)C2CC(=O)C(C(=O)C2)CS(=O)(=O)c3ccccc3 12H-927 c1ccc(cc1)C2CC(=C(C(=O)C2)CS(=O)(=O)c3ccccc3)Cl 12H-929 c1ccc(cc1)C2CC(=C(C(=O)C2)CS(=O)(=O)c3ccccc3)Sc4ccccc4 12H-930 CCOC(=O)NC1Cc2ccccc2C1Sc3c(cc(cn3)C(F)(F)F)Cl 12H-932 CC1(OCCO1)c2ccc3c(c2)c(on3)c4ccc(cc4)F 12H-933 CCCON1C(=O)c2ccccc2C1=O 12H-934 CC(C)ON1C(=O)c2ccccc2C1=O 12H-935 CCOC(=O)NC1Cc2ccccc2C1Sc3ncccn3 12H-936 CC(=O)c1ccc2c(c1)c(on2)c3ccc(cc3)F 12H-937 CCOC(=O)NC1Cc2ccccc2C1Sc3ccccn3 12H-938 CCCON.Cl 12H-939 Cc1c(c[nH]n1)C(=O)NC(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl 12H-940 C/C(=N/Nc1ccccc1F)/c2ccc3c(c2)c(on3)c4ccc(cc4)F 12H-941 Cc1c(cn(n1)C)C(=O)N(Cc2ccc(cc2)F)C(=O)NN(C)c3c(cc(cn3)C(F)(F)F)Cl 12H-942 CC(C)ON.Cl 12H-943 CC(/C=N/OC)(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 12H-945 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C/C(C(=O)Nc2ccccc2Cl)C(=O)Nc3ccccc3Cl 12H-946 c1cc(ccc1CC2C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)Cl 12H-947 c1cc(ccc1[N+](=O)[O-])Sc2cc(=O)n(c(=O)[nH]2)CCNc3c(cc(cn3)C(F)(F)F)Cl 12H-948 CC(C)O/N=C/C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 12H-949 Cn1c(cc(n1)Oc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 12J-001 c1ccc2c(c1)nc(n2Cc3cccc(c3)C(F)(F)F)c4ccc[nH]c4=O 12J-301S c1ccc2c(c1)nc(n2Cc3c(cccc3Cl)Cl)c4ccc[nH]c4=O 12J-302S c1ccc2c(c1)nc(n2Cc3ccc(cc3Cl)Cl)c4ccc[nH]c4=O 12J-303S Cn1c2ccccc2nc1c3ccc[nH]c3=O 12J-304S COc1ccc(cc1)Cn2c3ccccc3nc2c4ccc[nH]c4=O 12J-305S c1ccc(c(c1)Cn2c3ccccc3nc2c4ccc(=O)[nH]c4)Cl 12J-307S COc1ccc(c[n+]1[O-])NC(=O)c2ccc(cc2)C#N 12J-308S c1ccc2c(c1)nc(n2Cc3ccc(cc3)Cl)c4ccc(=O)[nH]c4 12J-313S c1ccc2c(c1)nc(n2Cc3ccc(cc3Cl)Cl)c4ccc(=O)[nH]c4 12J-315S Cc1ccc(cc1)Cn2c3ccccc3nc2c4ccc(=O)[nH]c4 12J-316S Cc1ccccc1S(=O)(=O)c2c(cc(nc2Cl)C)C 12J-317S Cc1ccccc1Cn2c3ccccc3nc2c4ccc(=O)[nH]c4 12J-319S c1ccc2c(c1)[nH]c(n2)c3ccc(=O)[nH]c3 12J-320S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OC)C)C 12J-321S CCCOc1c(c(cc(n1)C)C)S(=O)(=O)c2ccccc2C 12J-322S Cc1cc2c(cc1C)nc([nH]2)c3ccc(=O)[nH]c3 12J-323S Cc1cc2c(cc1C)nc([nH]2)c3ccc[nH]c3=O 12J-324S CCCSc1c(c(cc(n1)C)C)S(=O)(=O)c2ccccc2C 12J-327S CCCCSc1c(c(cc(n1)C)C)S(=O)(=O)c2ccccc2C 12J-328S CCCCCOc1c(c(cc(n1)C)C)S(=O)(=O)c2ccccc2C 12J-329S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OCC(C)(C)C)C)C 12J-330S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OCCC(C)C)C)C 12J-331S CCC(C)Oc1c(c(cc(n1)C)C)S(=O)(=O)c2ccccc2C 12J-332S Cn1c2ccccc2nc1c3ccc(=O)[nH]c3 12J-333S CCOC(=O)C(C)Sc1nc2ccccn2c(=O)n1 12J-335S Cc1cc2c(cc1C)n(c(n2)c3ccc(=O)[nH]c3)Cc4ccc(cc4)Cl 12J-336S Cc1ccccc1S(=O)(=O)c2c(cc(nc2SC)C)C 12J-337S Cc1cc2c(cc1C)n(c(n2)c3ccc(=O)[nH]c3)Cc4ccc(c(c4)Cl)Cl 12J-338S CCSc1c(c(cc(n1)C)C)S(=O)(=O)c2ccccc2C 12J-339S c1ccc(cc1)c2c(cc(nc2Cl)O)O 12J-340S c1ccc(c(c1)c2c(cc(nc2Cl)O)O)Cl 12J-341S c1cc(ccc1c2c(cc(nc2Cl)O)O)Cl 12J-342S Cc1ccc(cc1)Cn2c3cc(c(cc3nc2c4ccc(=O)[nH]c4)C)C 12J-343S c1ccc2c(c1)nc(n2Cc3cccc(c3)C(F)(F)F)c4ccc(=O)[nH]c4 12J-344S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4ccc(cc4)Cl 12J-345S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4cccc(c4)Cl 12J-346S Cc1cc2c(cc1C)n(c(n2)c3ccc(=O)[nH]c3)C 12J-347S Cc1ccc(cc1)c2c(cc(nc2Cl)O)O 12J-348S Cc1cccc(c1)c2c(cc(nc2Cl)O)O 12J-349S c1cc(c(cc1c2c(cc(nc2Cl)O)O)Cl)Cl 12J-350S c1cc(c(cc1Cl)Cl)c2c(cc(nc2Cl)O)O 12J-351S Cc1ccn2c(c1)nc(nc2=O)SCc3cccc(c3)C(F)(F)F 12J-501S Cc1ccn2c(c1)nc(nc2=O)SCc3ccccc3 12J-508S Cc1ccn2c(c1)nc(nc2=O)SC 12J-509S CCOC(=O)CSc1nc2cc(ccn2c(=O)n1)C 12J-510S Cc1ccn2c(c1)nc(nc2=O)SCC=C 12J-511S CCOC(=O)C(C)Sc1nc2cc(ccn2c(=O)n1)C 12J-512S Cc1cccn2c1nc(nc2=O)SCc3ccccc3 12J-514S Cc1cccn2c1nc(nc2=O)SCc3ccc(cc3)Cl 12J-515S Cc1cccn2c1nc(nc2=O)SCc3ccc(cc3)C(C)(C)C 12J-516S Cc1cccn2c1nc(nc2=O)SCc3ccc(cc3)OC 12J-517S Cc1cccn2c1nc(nc2=O)SCc3cccc(c3)C(F)(F)F 12J-518S CCOC(=O)CSc1nc2c(cccn2c(=O)n1)C 12J-519S c1c(cc(c(c1C(=O)NO)N)Cl)Cl 12J-520S c1ccc2c(c1)c(=O)n(c(n2)c3cccc(c3)C(F)(F)F)O 12J-521S CCOC(=O)C(C)Sc1nc2c(cccn2c(=O)n1)C 12J-523S Cc1cccn2c1nc(nc2=O)SCC=C 12J-524S CCCSc1nc2c(cccn2c(=O)n1)C 12J-525S CCOC(=O)NC(=S)Nc1ccc(cn1)Cl 12J-530S c1cc(cc(c1)C(F)(F)F)c2nc3c(cc(cc3Cl)Cl)c(=O)n2O 12J-531S Cc1c2cc(cc(c2oc1C(=O)c3ccccc3)Cl)Cl 12J-534S Cc1c2cc(cc(c2oc1C(=O)c3ccc(cc3)Cl)Cl)Cl 12J-535S Cc1c2cc(cc(c2oc1C(=O)c3ccc(c(c3)Cl)Cl)Cl)Cl 12J-536S Cc1c2cc(cc(c2oc1C(=O)c3ccc(cc3)F)Cl)Cl 12J-537S Cc1c2cc(ccc2oc1C(=O)c3ccc(cc3)F)Cl 12J-540S c1cc2nc(nc(=O)n2cc1Cl)S 12J-544S Cc1c2cc(cc(c2oc1C(=O)c3ccc(cc3)[N+](=O)[O-])Cl)Cl 12J-546S c1ccc2c(c1)c(=O)n(c(n2)c3ccc(cc3)[N+](=O)[O-])O 12J-551S c1ccc(cc1)c2[nH]c(=O)c3cc(ccc3n2)Cl 12J-553S Cc1cccn2c1nc(nc2=O)SC 12J-557S CCOC(=O)NC(=S)Nc1ccc(cn1)C 12J-558S c1ccc2c(c1)c(=O)n(c(n2)c3ccccc3C(=O)O)O 12J-560S c1ccc2c(c1)c(=O)n(c(n2)c3ccc(c(c3)Cl)Cl)O 12J-561S CCOC(=O)/C=C/1\C(=O)N(C(=O)N1)C 12J-562S Cc1ccc2nc(nc(=O)n2c1)SCc3ccc(cc3)Cl 12J-563S Cc1ccc2nc(nc(=O)n2c1)SCc3cccc(c3)C(F)(F)F 12J-564S Cc1ccc2nc(nc(=O)n2c1)SCc3ccccc3 12J-565S Cc1ccc2nc(nc(=O)n2c1)SCc3ccc(cc3)OC 12J-567S Cc1ccc2nc(nc(=O)n2c1)SCc3ccc(cc3)C(C)(C)C 12J-568S CCOC(=O)CSc1nc2ccc(cn2c(=O)n1)C 12J-569S Cc1ccc2nc(nc(=O)n2c1)SCC=C 12J-570S CCOC(=O)C(C)Sc1nc2ccc(cn2c(=O)n1)C 12J-571S Cc1ccc2nc(nc(=O)n2c1)SC 12J-572S CCCSc1nc2ccc(cn2c(=O)n1)C 12J-573S c1csc(c1Cl)C(=O)C[NH3+].[Cl-] 12J-900 Cc1cc(n(n1)C(=O)Nc2cccc(c2)C(F)(F)F)C(F)(F)Cl 12J-901 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-])Cl 12J-902 Cc1cc(nc(n1)c2ccccc2)C(F)(F)Cl 12J-903 COc1ccc(cc1)C(=O)Nc2ncc3c(n2)-c4ccccc4CC3 12J-904 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)c4ccc(cc4)F 12J-905 Cc1cc(nc(n1)c2ccccc2)C(F)(F)Sc3cccc(c3)C(F)(F)F 12J-906 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)c4cccc(c4)C(F)(F)F 12J-907 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)C4CC4 12J-908 CCOC(=O)c1c(c[nH]c1N)c2c(ccs2)Cl 12J-909 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)c4cccc(c4)Cl 12J-910 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)c4cccc(c4)[N+](=O)[O-] 12J-911 CCOC(=O)c1c(cn2c1nc(cc2C)C)c3c(ccs3)Cl 12J-912 c1ccc(cc1)C2C\3C(CCC/C3=N\OCc4ccc(cc4)[N+](=O)[O-])ON2c5ccccc5 12J-913 c1ccc(cc1)C2C3C(CCCC34NC(=O)N(N4)c5ccccc5)ON2c6ccccc6 12J-914 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)c4cccs4 12J-915 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)Nc4ccc(cc4)Cl 12J-917 c1ccc-2c(c1)CCc3c2nc(nc3)NS(=O)(=O)c4ccc(cc4)Cl 12J-918 COC(=O)CSCC(=O)Nc1ncc2c(n1)-c3ccccc3CC2 12J-919 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)Nc4cccc(c4)Cl 12J-920 C/C(=N\OCc1ccc(cc1)[N+](=O)[O-])/CCS(=O)(=O)c2ccccc2 12K-001 C/C(=N/OCc1ccc(cc1)Cl)/CCS(=O)(=O)c2ccccc2 12K-002 C/C(=N/OC/C=C/Cl)/CCS(=O)(=O)c1ccccc1 12K-003 CC(C(=O)C)Oc1ccccc1Cl 12K-005 CC(C(=O)C)Oc1cccc(c1)OC 12K-006 Cc1cccc(c1)OC(C)C(=O)C 12K-007 CC(C(=O)/C=C/N(C)C)Oc1cccc(c1)OC 12K-008 COc1ccc(cc1)C(=O)Oc2ccc(cc2S(=O)(=O)c3ccccc3)Oc4c(cc(cn4)C(F)(F)F)Cl 12K-009 c1cc(c(cc1/N=c\2/c(nss2)Cl)C(F)(F)F)Cl 12K-010 CCOC(=O)c1ccc(cc1)/N=c\2/c(nss2)Cl 12K-011 c1cc(c(cc1/N=c/2\c(nss2)Cl)Cl)Cl 12K-012 c1ccc(c(c1)/N=c\2/c(nss2)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 12K-013 c1ccc(cc1)S(=O)(=O)c2cc(ccc2OCc3ccc(cc3)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 12K-014 Cc1cc(cc(c1)OC(C)C(=O)C)C 12K-015 COC(=O)c1ccc2c(c1)C(=O)c3ccccc3CO2 12K-016 CC(C(=O)C)Oc1ccc(cc1)C(C)(C)C 12K-017 CC(c1ccnc2n1nc(n2)N)Oc3cccc(c3)OC 12K-018 CC(C)(C=O)Sc1ccccc1 12K-019 Cc1ccc(cc1)OC(C)C(=O)C 12K-020 Cc1cccc(c1)OC(C)C(=O)/C=C/N(C)C 12K-021 CC(C)(C(OC)OC)Nc1ccc(cc1)Cl 12K-022 Cc1cccc(c1)OC(C)c2ccnc3n2ncn3 12K-023 c1ccc(cc1)S(=O)(=O)c2cc(ccc2OCc3cccc(c3)C(F)(F)F)Oc4c(cc(cn4)C(F)(F)F)Cl 12K-024 c1ccc(cc1)S(=O)(=O)c2cc(ccc2OCc3c(cccc3Cl)F)Oc4c(cc(cn4)C(F)(F)F)Cl 12K-025 CC(C(=O)C)Oc1ccc(cc1)C#N 12K-026 Cc1cccc(c1)OC(C)c2ccnc3n2nc(n3)N 12K-027 Cc1cc(ccc1OC(C)C(=O)C)Cl 12K-028 COc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2S(=O)(=O)c3ccccc3)Oc4c(cc(cn4)C(F)(F)F)Cl 12K-029 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1)C#N 12K-030 COC(=O)c1ccc2c(c1)C(c3ccccc3CO2)O 12K-031 CC(C(=O)C)Oc1cccc(c1)F 12K-032 Cc1cc(cc(c1)OC(C)C(=O)/C=C/N(C)C)C 12K-033 Cc1cccc(c1OC(C)C(=O)C)C 12K-034 CC(C)(C=O)Sc1ccc(cc1)Cl 12K-035 Cc1ccc(cc1)SC(C)(C)C=O 12K-036 Cc1cc(cc(c1)OC(C)c2ccnc3n2nc(n3)N)C 12K-037 CC(C(=O)C)Oc1ccc(cc1F)F 12K-038 CC(c1ccnc2n1nc(n2)N)Oc3cccc(c3)C(F)(F)F 12K-039 CC(C(=O)/C=C\N(C)C)Oc1cccc(c1)F 12K-040 Cc1cc(cc(c1)OC(C)c2ccnc3n2ncn3)C 12K-041 CC(C)(/C=N/OC)Sc1ccc(cc1)Cl 12K-042 CC(C(=O)C)Oc1ccc(cc1)[N+](=O)[O-] 12K-043 CC(C)(/C=N/OC)Sc1ccccc1 12K-044 Cc1ccc(cc1)SC(C)(C)/C=N/O 12K-045 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1F)F 12K-046 CC(C)(/C=N/O)Sc1ccc(cc1)Cl 12K-047 CC(C(=O)C)Oc1ccccc1F 12K-048 Cc1cc(ccc1OC(C)C(=O)/C=C/N(C)C)Cl 12K-049 CC(C)(/C=N/O)Sc1ccccc1 12K-050 Cc1ccc(cc1)SC(C)(C)/C=N/OCc2ccc(cc2)[N+](=O)[O-] 12K-051 Cc1ccc(cc1)SC(C)(C)/C=N/OC 12K-052 CC(C)(/C=N/OCc1ccc(cc1)[N+](=O)[O-])Sc2ccc(cc2)Cl 12K-053 CC(C)(/C=N/OCc1ccc(cc1)[N+](=O)[O-])Sc2ccccc2 12K-054 CC(C)c1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3cccc(c3)C(F)(F)F 12K-301S Cc1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccccc3Cl 12K-302S CCN(CC)c1c(cc(c(n1)C)C(=O)OC)C#N 12K-303S CCCCNc1c(cc(c(n1)C)C(=O)OC)C#N 12K-304S Cc1c(cc(c(n1)N2CCCCC2)C#N)C(=O)OC 12K-305S Cc1c(cc(c(n1)N2CCOCC2)C#N)C(=O)OC 12K-306S CCCCNc1c(cc(c(n1)C)C(=O)C)C#N 12K-307S Cc1c(cc(c(n1)NCCCN(C)C)C#N)C(=O)C 12K-308S Cc1c(cc(c(n1)N2CCN(CC2)c3ccccc3)C#N)C(=O)C 12K-309S Cc1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccc(cc3)F 12K-310S Cc1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccc(cc3)C(C)(C)C 12K-311S CCOC(=O)c1cc(c(nc1c2ccccc2)SC)C#N 12K-312S Cc1c(cc(c(n1)N2CCN(CC2)c3ccccc3)C#N)C(=O)OC 12K-315S Cc1c(cc(c(n1)N2CCN(CC2)C)C#N)C(=O)OC 12K-316S Cc1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccc(cc3Cl)Cl 12K-320S c1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccccc3Cl 12K-321S Cc1c(cc(c(n1)N(C)Cc2ccccc2)C#N)C(=O)OC 12K-322S Cc1c(cc(c(n1)N2CC(OC(C2)C)C)C#N)C(=O)C 12K-323S Cc1c(cc(c(n1)N(C)Cc2ccccc2)C#N)C(=O)C 12K-324S Cc1c(cc(c(n1)N2CC(OC(C2)C)C)C#N)C(=O)OC 12K-325S Cc1c(cc(c(n1)NCc2ccc(cc2Cl)Cl)C#N)C(=O)OC 12K-326S CCOC(=O)c1cc(c(nc1c2ccccc2)Sc3ccccc3)C#N 12K-327S CCOC(=O)c1cc(c(nc1c2ccccc2)Sc3ccc(cc3)Cl)C#N 12K-328S CCOC(=O)c1cc(c(nc1c2ccccc2)Sc3ccc(cc3)OC)C#N 12K-329S CCOC(=O)c1cc(c(nc1c2ccccc2)Sc3cccc(c3)C(F)(F)F)C#N 12K-330S CCOC(=O)c1cc(c(nc1c2ccccc2)SCc3ccc(cc3)Cl)C#N 12K-331S Cc1c(cc(c(n1)NCc2ccc(cc2)Cl)C#N)C(=O)C 12K-332S CC(C)(C)c1ccc(cc1)Cn2c(=O)ccc(n2)/C=C/c3ccccc3 12K-333S c1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccc(c(c3)Cl)Cl 12K-334S c1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3cccc(c3)C(F)(F)F 12K-335S CCOC(=O)c1cc(c(nc1c2ccccc2)SCc3cccc(c3)C(F)(F)F)C#N 12K-336S c1ccc(cc1)/C=C/c2ccc(=O)n(n2)Cc3ccc(cc3Cl)Cl 12K-343S Cc1ccccc1C(=O)NC2CCSC2=O 12K-344S Cc1cccc(c1)C(=O)NC2CCSC2=O 12K-345S c1cc(c(cc1Cl)Cl)C(=O)NC2CCSC2=O 12K-346S c1ccc(c(c1)C(=O)NC2CCSC2=O)Cl 12K-347S c1cc(cc(c1)Cl)C(=O)NC2CCSC2=O 12K-348S c1cc(c(cc1C(=O)NC2CCSC2=O)Cl)Cl 12K-349S c1cc(ccc1C(=O)NC2CCSC2=O)Cl 12K-350S CCOC(=O)c1cc(c(nc1c2ccccc2)SCc3ccc(cc3Cl)Cl)C#N 12K-353S CCOC(=O)c1cc(c(nc1c2ccccc2)Sc3ccccc3Cl)C#N 12K-354S CCOC(=O)c1cc(c(nc1c2ccccc2)Sc3ccc(cc3Cl)Cl)C#N 12K-355S c1cc(ccc1C(=O)NC2CCSC2=O)[N+](=O)[O-] 12K-359S c1cc(ccc1C#N)C(=O)NC2CCSC2=O 12K-360S c1cc(cc(c1)C(F)(F)F)C(=O)NC2CCSC2=O 12K-361S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3ccccc3)C#N 12K-362S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3cc(cc(c3)C)C)C#N 12K-363S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3cccc(c3)C(F)(F)F)C#N 12K-364S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3ccc(cc3)F)C#N 12K-365S Cc1ccc(cc1)Oc2ccc(cn2)C(=O)NC3CCSC3=O 12K-366S Cc1cccc(c1C)Oc2ccc(cn2)C(=O)NC3CCSC3=O 12K-367S c1cc(ncc1C(=O)NC2CCSC2=O)Oc3cc(c(cc3Cl)Cl)Cl 12K-368S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3ccc(cc3Cl)Cl)C#N 12K-369S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3ccccc3OC)C#N 12K-370S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3cccc(c3Cl)Cl)C#N 12K-371S CCOC(=O)c1cc(c(nc1c2ccccc2)Oc3ccc(cc3C)Cl)C#N 12K-372S Cc1c(nc(nn1)SC)/C=C/Nc2ccc(cc2)Cl 12K-373S Cc1c(nc(nn1)SC)/C=C/Nc2ccc(cc2)OC 12K-374S Cc1c(nc(nn1)SC)/C=C/Nc2ccc(cc2)C(F)(F)F 12K-375S Cc1c(nc(nn1)SC)/C=C/Nc2cc(cc(c2)Cl)Cl 12K-376S Cc1c(nc(nn1)SC)/C=C/Nc2ccc(cc2F)F 12K-377S CCOC(=O)c1cc(c(nc1c2ccccc2)Sc3ccccc3C(=O)OC)C#N 12K-378S c1cc(c(cc1Cl)Cl)Oc2ccc(cn2)C(=O)NC3CCSC3=O 12K-379S c1cc(ccc1Oc2ccc(cn2)C(=O)NC3CCSC3=O)F 12K-381S Cc1c(nc(nn1)SC)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F 12K-386S Cc1c(nc(nn1)SC)/C=C/Nc2ccc(c(c2)Cl)Cl 12K-387S Cc1c(nc(nn1)SC)/C=C/Nc2cccc(c2)C(F)(F)F 12K-388S Cc1c(nc(nn1)SC)/C=C/Nc2ccc(cc2)F 12K-389S Cc1ccc(cc1)N/C=C/c2c(nnc(n2)SC)C 12K-390S Cc1c(nc(nn1)SC)/C=C/NOC 12K-391S Cc1c(nc(nn1)SC)/C=C/NOCc2ccc(cc2)Cl 12K-392S c1ccnc(c1)c2nc(cc(n2)N3CCCC3)CS(=O)c4ccc(cc4)Cl 12K-503S c1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3cc(cc(c3)Cl)Cl 12K-504S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(c(c2)C#N)Sc3ccc(cc3)Cl 12K-505S c1cc(ccc1Sc2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl)Cl 12K-508S c1cc(c(c(c1)F)C(=O)c2ccc(c(c2)Cl)Cl)C(=O)O 12K-509S CCN(CC)c1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 12K-512S c1ccc(cc1)c2nc(cc(n2)N3CCCCC3)CSc4ccc(cc4)Cl 12K-513S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccc(cc3)F 12K-516S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccccc3C 12K-517S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl 12K-518S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3cccc(c3)C(F)(F)F 12K-519S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccccc3Cl 12K-520S c1cc(ccc1C(=O)Nc2ccc(c(c2)C#N)Sc3ccc(cc3)Cl)F 12K-521S CN(C)c1cc(nc(n1)c2ccccn2)CS(=O)c3ccc(cc3)Cl.O 12K-522S CCCNc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 12K-525S c1cc(ccc1C(=O)Nc2nc(=S)ss2)Cl 12K-526S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2nc(=S)ss2 12K-527S c1cc(ncc1C(=O)Nc2nc(=S)ss2)Cl 12K-528S CC(C)CC(=O)Nc1nc(=S)ss1 12K-529S C1CC1C(=O)Nc2nc(=S)ss2 12K-530S c1ccc(cc1)c2nc(cc(n2)Sc3ccccc3)CS(=O)c4ccc(cc4)Cl 12K-531S c1ccc(cc1)c2nc(cc(n2)Oc3ccccc3)CS(=O)c4ccc(cc4)Cl 12K-532S CCOC(=O)CSc1cc(nc(n1)c2ccccc2)CS(=O)c3ccc(cc3)Cl 12K-533S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3)Cl)CS(=O)c4ccc(cc4)Cl 12K-534S c1ccc(cc1)c2nc(cc(n2)Oc3ccc(cc3)Cl)CS(=O)c4ccc(cc4)Cl 12K-535S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)C3CC3 12K-538S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3cc(cc(c3)Cl)Cl 12K-539S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(c(c2)C#N)S(=O)(=O)c3ccc(cc3)Cl 12K-540S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)CS(=O)c4ccc(cc4)Cl 12K-541S c1ccc(cc1)c2nc(cc(n2)N3CCCCC3)CS(=O)c4ccc(cc4)Cl 12K-542S c1ccc(cc1)c2nc(cc(n2)N3CCCC3)CS(=O)c4ccc(cc4)Cl 12K-543S c1ccc2c(c1)-c3c(cc(nn3)c4ccc(c(c4)F)F)C2=O 12K-550S c1ccc2c(c1)-c3c(cc(nn3)c4cccc(c4)Br)C2=O 12K-551S Cc1ccccc1c2cc3c(nn2)-c4ccccc4C3=O 12K-554S CSc1ccc(cc1C#N)N 12K-558S c1ccc(cc1)c2nc(cc(n2)Cl)CS(=O)c3ccccc3 12K-559S CC(C)(C)C(=O)Nc1nc(=S)ss1 12K-560S c1cc(sc1)C(=O)Nc2nc(=S)ss2 12K-561S CCOC(=O)C(=O)Nc1nc(=S)ss1 12K-562S CCOC(=O)Nc1nc(=S)ss1 12K-563S Cc1ccccc1C(=O)Nc2ccc(c(c2)C#N)Sc3ccccc3C 12K-566S Cc1ccccc1Sc2ccc(cc2C#N)NC(=O)c3ccc(cc3)F 12K-567S Cc1ccccc1Sc2ccc(cc2C#N)NC(=O)c3ccccc3Cl 12K-568S c1cc(ccc1C(=O)Nc2nc(=S)ss2)F 12K-569S c1ccc(c(c1)C(=O)Nc2nc(=S)ss2)Cl 12K-570S Cc1ccccc1C(=O)Nc2nc(=S)ss2 12K-571S c1cc(cc(c1)Cl)C(=O)Nc2nc(=S)ss2 12K-572S COc1cccc(c1)C(=O)Nc2nc(=S)ss2 12K-573S Cc1ccccc1Sc2ccc(cc2C#N)NC(=O)c3cccc(c3)Cl 12K-574S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3cccc(c3)C 12K-575S Cc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccc(cc3Cl)Cl 12K-576S CSc1ccc(cc1C#N)NC(=O)c2ccc(c(c2)Cl)Cl 12K-577S CSc1ccc(cc1C#N)NC(=O)c2ccc(cc2Cl)Cl 12K-578S CSc1ccc(cc1C#N)NC(=O)c2ccc(cc2)Cl 12K-579S CSc1ccc(cc1C#N)NC(=O)c2ccccc2Cl 12K-580S CSc1ccc(cc1C#N)NC(=O)c2cccc(c2)C(F)(F)F 12K-581S CSc1ccc(cc1C#N)NC(=O)c2ccc(cc2)F 12K-582S Cc1ccccc1C(=O)Nc2ccc(c(c2)C#N)SC 12K-583S CSc1ccc(cc1C#N)NC(=O)c2cccc(c2)Cl 12K-584S CSc1ccc(cc1C#N)NC(=O)c2ccccc2 12K-585S CSc1ccc(cc1C#N)NC(=O)c2ccc(nc2)Cl 12K-586S COc1ccc(cc1)Sc2ccc(cc2C#N)[N+](=O)[O-] 12K-587S COc1ccc(cc1)Sc2ccc(cc2C#N)N 12K-588S Cc1cccc(c1)C(=O)Nc2ccc(c(c2)C#N)SC 12K-592S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3ccncc3)N4CCOCC4 12K-594S c1ccc(cc1)CNc2cc(nc(n2)c3ccncc3)CS(=O)(=O)c4ccccc4 12K-595S CSc1ccc(cc1C#N)NC(=O)c2c(cccc2F)F 12K-596S CS(=O)c1ccc(cc1C#N)NC(=O)c2cccc(c2)C(F)(F)F 12K-598S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccc(cc3)Cl 12K-599S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccc(cc3Cl)Cl 12K-600S Cc1ccccc1S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccccc3Cl 12K-601S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3cc(cc(c3)Cl)Cl 12K-602S Cc1ccccc1S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl 12K-603S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)CS(=O)c4ccccc4 12K-606S c1ccc(cc1)c2nc(cc(n2)Sc3ccccc3)CS(=O)c4ccccc4 12K-607S CSc1cc(nc(n1)c2ccccc2)CS(=O)c3ccccc3 12K-608S COc1cc(nc(n1)c2ccccc2)CS(=O)c3ccccc3 12K-609S CCOC(=O)CSc1cc(nc(n1)c2ccccc2)CS(=O)c3ccccc3 12K-610S Cc1ccccc1Sc2ccc(cc2C#N)NC(=O)c3cccc(c3)C(F)(F)F 12K-611S COc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccccc3Cl 12K-612S COc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3cccc(c3)Cl 12K-613S CSc1ccc(cc1C#N)NC(=O)c2cc(c(cc2Cl)F)F 12K-614S CSc1ccc(cc1C#N)NC(=O)c2cc(ccc2Cl)Cl 12K-615S COc1cccc(c1C(=O)Nc2ccc(c(c2)C#N)SC)OC 12K-616S c1cc(cc(c1)Sc2ccc(cc2C#N)[N+](=O)[O-])C(F)(F)F 12K-617S CSc1ccc(cc1C#N)NC(=O)c2cccnc2 12K-618S CSc1ccc(cc1C#N)NC(=O)c2ccccc2C(=O)c3ccc(cc3)F 12K-619S COc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3c(cccc3F)F 12K-620S COc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)C3CC3 12K-621S COc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccc(cc3)F 12K-622S c1cc(cc(c1)Sc2ccc(cc2C#N)N)C(F)(F)F 12K-623S Cc1cc(cc(c1)C(=O)Nc2ccc(c(c2)C#N)SC)C 12K-624S CSc1ccc(cc1C#N)NC(=O)c2cccc(c2)C#N 12K-625S CS(=O)(=O)c1ccc(cc1C#N)NC(=O)c2ccc(cc2)Cl 12K-626S CS(=O)(=O)c1ccc(cc1C#N)NC(=O)c2ccc(cc2Cl)Cl 12K-627S Cc1cccc(c1)C(=O)Nc2ccc(c(c2)C#N)S(=O)C 12K-628S CS(=O)c1ccc(cc1C#N)NC(=O)c2ccccc2 12K-629S CS(=O)c1ccc(cc1C#N)NC(=O)c2ccccc2Cl 12K-630S CS(=O)c1ccc(cc1C#N)NC(=O)c2cccc(c2)Cl 12K-631S CS(=O)(=O)c1ccc(cc1C#N)NC(=O)c2cc(ccc2Cl)Cl 12K-632S CS(=O)(=O)c1ccc(cc1C#N)NC(=O)c2cc(c(cc2Cl)F)F 12K-633S CS(=O)c1ccc(cc1C#N)NC(=O)c2ccc(c(c2)Cl)Cl 12K-637S CS(=O)(=O)c1ccc(cc1C#N)NC(=O)c2cccnc2 12K-638S CS(=O)c1ccc(cc1C#N)NC(=O)c2ccc(cc2Cl)Cl 12K-639S c1cc(cc(c1)Sc2ccc(cc2C#N)NC(=O)c3ccc(cc3)F)C(F)(F)F 12K-641S CCn1c(=O)c(c(cn1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 12K-900 CCn1c(=O)c(c(cn1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 12K-901 CCn1c(=O)c(c(cn1)N(C)N)Cl 12K-902 CCn1c(=O)c(c(cn1)N(C)NC(=O)Nc2ccc(cc2)Cl)Cl 12K-903 COc1ccc(cc1)n2c(=O)c(c(cn2)Cl)Cl 12K-905 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)Cl)Cl 12K-907 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)NN)Cl 12K-908 CN(c1cnn(c(=O)c1Cl)c2ccc(cc2)OC)N 12K-909 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)N3CCCC3)Cl 12K-910 COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCOCC3)Cl 12K-911 Cc1cc(n(n1)c2cnn(c(=O)c2Cl)c3cccc(c3)Cl)C 12K-912 CN(c1cnn(c(=O)c1Cl)c2ccc(cc2)OC)n3cccc3 12K-913 CCn1c(=O)c(c(cn1)N2CCOCC2)Cl 12K-914 CN(c1cnn(c(=O)c1Cl)c2ccc(cc2)OC)NC(=O)Nc3cccc(c3)C(F)(F)F 12K-915 COc1ccc(cc1)n2c(=O)c(c(cn2)ON3C(=O)CCC3=O)Cl 12K-917 c1ccc2c(c1)C(=O)N(C2=O)Oc3cnn(c(=O)c3Cl)c4cccc(c4)Cl 12K-918 CN1CCN(CC1)c2cnn(c(=O)c2Cl)c3cccc(c3)Cl 12K-919 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)O)Cl 12K-920 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)NCCO)Cl 12K-921 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)Sc3ccc(cc3)Br)Cl 12K-922 c1cc(sc1c2csnn2)S(=O)(=O)Cl 12L-001 CCOC(=O)c1coc(n1)/C=C/c2ccccc2 12L-002 c1ccc2c(c1)c3nncn3c(n2)C(F)(F)F 12L-003 CC(C)NS(=O)(=O)c1ccc(s1)c2csnn2 12L-004 CN1CCN(CC1)S(=O)(=O)c2ccc(s2)c3csnn3 12L-005 CN(C)S(=O)(=O)c1ccc(s1)c2csnn2 12L-006 C/C(=N\NC(=O)OC)/c1cc(c(cc1OC)OC)OC 12L-007 c1cc(cnc1)CNS(=O)(=O)c2ccc(s2)c3csnn3 12L-008 CCC(C)NS(=O)(=O)c1ccc(s1)c2csnn2 12L-009 CN(c1c2ccccc2nc(n1)C(F)(F)F)NC(=O)c3ccc(cc3)OC 12L-010 CN(c1c2ccccc2nc(n1)C(F)(F)F)NS(=O)(=O)c3ccc(cc3)OC 12L-011 c1ccc(c(c1)C(=O)NNc2cccc(n2)Cl)C(=O)O 12L-012 c1ccc2c(c1)C(=O)N(C2=O)Nc3cccc(n3)Cl 12L-013 c1ccc(c(c1)C(=O)NNc2ccc(cc2)Cl)C(=O)O 12L-014 c1ccc(c(c1)C(=O)NNc2ccc(cc2)F)C(=O)O 12L-015 Cc1ccc(cc1)NNC(=O)c2ccccc2C(=O)O 12L-016 c1ccc2c(c1)C(=O)N(C2=O)Nc3ccc(cc3)F 12L-017 Cc1ccc(cc1)NN2C(=O)c3ccccc3C2=O 12L-018 c1cc(oc1)CNS(=O)(=O)c2ccc(s2)c3csnn3 12L-019 CN(c1c2ccccc2nc(n1)C(F)(F)F)NS(=O)(=O)c3ccc(cc3)Cl 12L-020 c1ccc(c(c1)C(=O)NNc2ccc(cc2Cl)Cl)C(=O)O 12L-021 c1ccc2c(c1)C(=O)N(C2=O)Nc3ccc(cc3)Cl 12L-022 COc1cc(c(cc1OC)OC)c2csnn2 12L-023 CN(c1c2ccccc2nc(n1)C(F)(F)F)NS(=O)(=O)c3ccc(cc3)Br 12L-024 c1ccc2c(c1)C(=O)N(C2=O)Nc3ccc(cc3Cl)Cl 12L-025 c1ccc2c(c1)c[n+](nc2[O-])c3ccc(cc3)F 12L-026 c1ccc2c(c1)c[n+](nc2[O-])c3ccc(cc3Cl)Cl 12L-027 Cc1ccc(cc1)c2c3c(ncnc3n(n2)C(C)(C)C)NC(=O)c4ccc(cc4)F 12L-255S COc1ccc(cc1)c2cc(on2)C(=O)Nc3ccccc3 12L-301S CN(C)C(=O)c1cc(no1)c2ccc(cc2)OC 12L-302S CN1c2ccccc2/C(=N\Nc3ccc(cc3)F)/C1=O 12L-303S CC(C)N1c2ccccc2/C(=N\Nc3ccc(cc3)F)/C1=O 12L-304S c1ccc(cc1)c2cc(on2)CO 12L-305S Cc1ccc(cc1)CN2c3ccccc3/C(=N\Nc4ccc(cc4)[N+](=O)[O-])/C2=O 12L-306S Cc1ccc(cc1)CN2c3ccccc3/C(=N\Nc4c(cc(cc4Cl)Cl)Cl)/C2=O 12L-307S Cc1ccc(cc1)CN2c3ccccc3/C(=N\Nc4c(cc(cc4Cl)C(F)(F)F)Cl)/C2=O 12L-308S CC(C)N1c2ccccc2/C(=N\Nc3cc(ccc3Cl)Cl)/C1=O 12L-309S CC(C)N1c2ccccc2/C(=N\Nc3ccc(c(c3)Cl)Cl)/C1=O 12L-310S COc1ccc(cc1)c2cc(on2)C(=O)Nc3ccccc3F 12L-312S COc1ccc(cc1)c2cc(on2)C(=O)NCC=C 12L-313S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4ccccc4Cl)/C2=O 12L-314S c1ccc(cc1)N2c3ccccc3/C(=N/Nc4ccc(cc4Cl)Cl)/C2=O 12L-315S COc1ccc(cc1)N/N=C/2\c3ccccc3N(C2=O)CC=C 12L-316S C=CCN1c2ccccc2/C(=N\Nc3c(cc(cc3Cl)C(F)(F)F)Cl)/C1=O 12L-317S c1ccc(cc1)c2cc(on2)C(=O)O 12L-318S C=CCN1c2ccccc2/C(=N\Nc3cc(cc(c3)Cl)Cl)/C1=O 12L-320S C=CCN1c2ccccc2/C(=N\Nc3ccc(c(c3)Cl)Cl)/C1=O 12L-321S CC(C)N1c2ccccc2/C(=N\Nc3ccc(cc3Cl)Cl)/C1=O 12L-322S CC(C)N1c2ccccc2/C(=N\Nc3ccccc3Cl)/C1=O 12L-323S CC(C)N1c2ccccc2/C(=N\Nc3c(cc(cc3Cl)C(F)(F)F)Cl)/C1=O 12L-324S CN1c2ccccc2/C(=N\Nc3c(cc(cc3Cl)C(F)(F)F)Cl)/C1=O 12L-325S CN1c2ccccc2/C(=N\Nc3cc(ccc3Cl)Cl)/C1=O 12L-326S CN1c2ccccc2/C(=N\Nc3ccc(c(c3)Cl)Cl)/C1=O 12L-327S COc1ccc(cc1)c2cc(on2)C(=O)NCc3ccccc3 12L-328S COc1ccc(cc1)c2cc(on2)C(=O)Nc3cc(cc(c3)Cl)Cl 12L-329S Cc1ccc(cc1)c2c(c(n(n2)C(C)(C)C)N)C#N 12L-333S CC(C)(C)n1c(c(c(n1)c2ccc(cc2)Cl)C#N)NC(=O)c3ccccc3Cl 12L-334S CC(C)(C)n1c(c(c(n1)c2ccc(cc2)Cl)C#N)NC(=O)c3ccc(cc3)OC 12L-335S c1ccc(cc1)NC(=O)c2cc(no2)c3ccccc3Cl 12L-336S COc1ccc(cc1)NC(=O)c2cc(no2)c3ccccc3Cl 12L-337S c1ccc(c(c1)c2cc(on2)C(=O)Nc3cccc(c3)Cl)Cl 12L-338S CCNC(=O)c1cc(no1)c2ccccc2Cl 12L-339S Cc1ccc(cc1)c2c3c(nc(nc3n(n2)C(C)(C)C)c4ccc(cc4)C)N 12L-343S Cc1ccccc1C(=O)NC(C)C(=O)O 12L-346S c1ccc(cc1)c2cc(on2)C(=O)Nc3ccc(cc3)F 12L-347S c1ccc(cc1)c2cc(on2)C(=O)Nc3ccccc3 12L-348S c1ccc(cc1)c2cc(on2)C(=O)Nc3cccc(c3)C(F)(F)F 12L-349S Cc1c(cccc1Cl)NC(=O)c2cc(no2)c3ccccc3 12L-350S CN(C)C(=O)c1cc(no1)c2ccccc2 12L-351S Cc1ccc(cc1)c2c3c(ncnc3n(n2)C(C)(C)C)NC(=O)c4ccccc4Cl 12L-356S Cc1ccc(cc1)c2c3c(ncnc3n(n2)C(C)(C)C)NC(=O)c4ccc(cc4)C 12L-357S CC(C)(C)n1c(c(c(n1)c2ccc(cc2)F)C#N)N 12L-362S Cc1ccc(cc1)c2c3c(ncnc3n(n2)C(C)(C)C)NS(=O)(=O)c4ccc(cc4)C 12L-363S C#CCN1c2ccccc2C(=O)C1=O 12L-501S C#CCN1c2ccccc2/C(=N\Nc3c(cc(cc3Cl)C(F)(F)F)Cl)/C1=O 12L-502S C#CCN1c2ccccc2/C(=N\Nc3ccc(cc3)Cl)/C1=O 12L-503S Cc1ccc(cc1)CSc2nc(c(c(n2)NC)C#N)c3ccccc3 12L-504S Cc1ccc(cc1)CSc2nc(c(c(n2)NCc3ccccc3)C#N)c4ccccc4 12L-505S Cc1ccc(cc1)CSc2nc(c(c(n2)NCC=C)C#N)c3ccccc3 12L-506S Cc1ccc(cc1)CSc2nc(c(c(n2)NC3CCCCC3)C#N)c4ccccc4 12L-507S Cc1ccc(cc1)CSc2nc(c(c(n2)NC(C)C)C#N)c3ccccc3 12L-508S CC(C)(C)c1ccc(cc1)COc2c3ccccc3sc2C#N 12L-509S Cc1c(c(on1)C)CN2CCSCC2 12L-510S c1ccc2c(c1)c(c(s2)C#N)OCc3cccc(c3)Cl 12L-511S CNc1c(c(nc(n1)SCc2c(cccc2Cl)Cl)c3ccccc3)C#N 12L-513S C#CCN1c2ccccc2/C(=N\Nc3ccccc3)/C1=O 12L-514S c1ccc(cc1)COc2c3ccccc3sc2C#N 12L-515S c1ccc2c(c1)c(c(s2)C#N)OCc3ccc(c(c3)Cl)Cl 12L-516S CCOC(=O)c1cc2c(nn(c2s1)C)C(F)(F)F 12L-518S Cn1c2c(cc(s2)C(=O)O)c(n1)C(F)(F)F 12L-521S Cc1cc(c(c(n1)SC)C#N)/C=C\c2ccccc2 12L-522S Cc1cc(c(c(n1)SCC=C)C#N)/C=C\c2ccccc2 12L-523S CO/N=C(/CSCc1cccc(c1)Cl)\c2ccc(cc2)Cl 12L-524S CO/N=C(/COc1ccc(cc1)Cl)\c2ccc(cc2)Cl 12L-525S Cc1ccccc1COc2c3ccccc3sc2C#N 12L-526S CO/N=C(/CS(=O)c1ccc(cc1)Cl)\c2ccc(cc2)Cl 12L-528S CO/N=C(/CS(=O)(=O)c1ccc(cc1)Cl)\c2ccc(cc2)Cl 12L-529S Cn1c(c(c(n1)c2ccccc2)CNc3ccc(c(c3)Cl)Cl)Cl 12L-532S COc1ccc(cc1)SC/C(=N/OC)/c2ccc(cc2)Cl 12L-533S COc1ccc(cc1)CSC/C(=N\OC)/c2ccc(cc2)Cl 12L-534S CO/N=C(/CS(=O)Cc1ccc(cc1)Cl)\c2ccc(cc2)Cl 12L-536S CO/N=C(/CS(=O)(=O)Cc1ccc(cc1)Cl)\c2ccc(cc2)Cl 12L-537S COC(=O)/C(=C\c1cccs1)/CC(=O)c2ccccc2 12L-538S c1cc(ccc1S(=O)(=O)CC(c2ccc(c(c2)Cl)Cl)O)Cl 12L-541S c1cc(ccc1S(=O)(=O)CC(c2ccc(c(c2)Cl)Cl)O)Br 12L-542S COc1ccc(cc1)S(=O)(=O)CC(c2ccc(c(c2)Cl)Cl)O 12L-543S COc1ccc(cc1)S(=O)C/C(=N/OC)/c2ccc(cc2)Cl 12L-545S COc1ccc(cc1)S(=O)(=O)C/C(=N/OC)/c2ccc(cc2)Cl 12L-546S COc1ccc(cc1)CS(=O)C/C(=N\OC)/c2ccc(cc2)Cl 12L-547S COc1ccc(cc1)CS(=O)(=O)C/C(=N\OC)/c2ccc(cc2)Cl 12L-548S c1cc(ccc1F)S(=O)(=O)CC(c2ccc(c(c2)Cl)Cl)O 12L-549S c1ccc(cc1)C2=NC(N=C(S2)c3ccccc3)c4ccc(cc4)Cl 12L-550S Cn1c(c(c(n1)c2ccccc2)/C=N/c3ccc(cc3)Cl)Cl 12L-551S Cn1c(c(c(n1)c2ccccc2)/C=N/c3ccc(c(c3F)Cl)F)Cl 12L-552S Cc1ccc(cc1)C2N=C(SC(=N2)c3ccccc3)c4ccccc4 12L-553S Cc1ccc(cc1)SCCC(=O)c2ccc(cc2)Cl 12L-554S c1cc(ccc1C(=O)CCSc2ccc(cc2)Br)Cl 12L-555S c1cc(ccc1C(=O)CCSc2ccc(cc2)Cl)Cl 12L-556S COc1ccc(cc1)SCCC(=O)c2ccc(cc2)Cl 12L-557S c1cc(ccc1C(=O)CCSCc2ccc(cc2Cl)Cl)Cl 12L-558S Cc1ccc(cc1)SCCC(=O)c2ccc(cc2)OC 12L-560S c1cc(sc1)C(=O)CCSc2ccc(cc2)Cl 12L-561S c1cc(sc1)C(=O)CCSc2ccc(cc2)Br 12L-562S Cn1c(c(c(n1)c2ccccc2)/C=N/c3c(cccc3Cl)Cl)Cl 12L-563S Cn1c(c(c(n1)c2ccccc2)/C=N/c3cccc(c3)C(F)(F)F)Cl 12L-564S CC(C)(CCl)C(=O)NNc1c(cc(cn1)C(F)(F)F)Cl 12L-701 c1ccc2c(c1)C(=O)N(C2=O)N3C(=O)/C(=C/c4cccc(c4)Cl)/SC3=S 12L-702 CC1=CC(=O)/C(=C/N(C)C)/C(=O)O1 12L-704 CC1(CN(C1=O)c2ccc(cc2)C(=O)C/C=N/OCc3c(cccc3Cl)F)C 12L-705 CC1(CN(C1=O)Nc2c(cc(cn2)C(F)(F)F)Cl)C 12L-706 CC1=CC(=O)/C(=C/Nc2ccc(cc2)OC)/C(=O)O1 12L-707 COc1ccc(cc1O)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)CCC3=O 12L-711 c1cc(ccc1/C=C/2\C(=O)N(C(=S)S2)N3C(=O)C4C5CC(C4C3=O)C=C5)F 12L-712 c1ccc(cc1)c2nnc(o2)N 12L-713 CCOC(=O)c1cc2ccccc2nc1CCl 12L-714 CC(C)(CCl)C(=O)NNc1ccccc1 12L-715 COc1cccc(c1)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)CCCC3=O 12L-716 Cc1cccc(c1)N/C=C\2/C(=O)C=C(OC2=O)C 12L-721 COc1ccc(cc1)/C=N/NC(=O)N 12L-722 CC1(CN(C1=O)c2ccc(cc2)c3ccnn3c4ccc(cc4F)F)C 12L-723 Cc1cc(=O)c(cn1c2ccc(cc2)OC)C(=O)O 12L-724 c1cc(c(cc1/C=C/2\C(=O)N(C(=S)S2)N3C(=O)C4C5CC(C4C3=O)C=C5)[N+](=O)[O-])Cl 12L-725 CC(C)(CCl)C(=O)NNc1c(cc(cc1Cl)Cl)Cl 12L-726 CC1(CN(C1=O)Nc2c(cc(cc2Cl)Cl)Cl)C 12L-727 c1ccc(c(c1)CO/N=C/c2c(c3ccccc3s2)Cl)F 12L-728 c1ccc2c(c1)c(c(s2)/C=N/OCCOc3cccc(c3)C(F)(F)F)Cl 12L-729 Cc1cccc(c1)n2cc(c(=O)cc2C)C(=O)O 12L-730 Cc1ccc(cc1)CO/N=C/c2c(c3ccccc3s2)Cl 12L-731 Cc1ccc(c(c1)C)N/C=C\2/C(=O)C=C(OC2=O)C 12L-732 CC1=CC(=O)/C(=C/Nc2ccc(cc2)C(C)C)/C(=O)O1 12L-733 COc1ccccc1/C=C\2/C(=O)N(C(=S)S2)N3C(=O)CCCC3=O 12L-734 c1ccc2c(c1)c(c(s2)/C=N/O)Cl 12L-735 Cc1ccc(cc1)CO/N=C/c2c(cc(oc2=O)C)O 12L-736 c1ccc(c(c1)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)c4cccc5c4c(ccc5)C3=O)C(F)(F)F 12L-738 COc1ccc(cc1)c2nnc(o2)N 12L-739 c1ccc(cc1)N2C(=O)C3C4CSCN4C(C3C2=O)c5cccc(c5)Cl 12L-901 Cn1c(=O)c(nn(c1=O)c2cccc(c2)C(F)(F)F)C(=O)/C=C/N(C)C 12L-902 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)C(=O)O)C(=O)N(C4=O)c5cccc(c5)C(F)(F)F)C2=O 12L-903 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)C(=O)O)C(=O)N(C4=O)c5ccc(cc5Cl)Cl)C2=O 12L-904 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)C(=O)O)C(=O)N(C4=O)CCNc5c(cc(cn5)C(F)(F)F)Cl)C2=O 12L-905 CCCCCCCCCc1ccc(cc1)OCC(=O)OCC 12L-906 CCCCCCCCCc1ccc(cc1)OCC(=O)O 12L-907 c1ccc(cc1)/C=C/C2C3C(C4N2CSC4)C(=O)N(C3=O)c5ccc(cc5)Cl 12L-908 c1ccc(cc1)N2C(=O)C3C(C2=O)C(=C4C(=O)c5ccccc5C4=O)NC3C(=O)O 12L-910 Cc1ccc(cc1)n2c(ccn2)c3c(=O)n(c(=O)n(n3)c4cccc(c4)C(F)(F)F)C 12L-911 Cn1c(=O)c(nn(c1=O)c2cccc(c2)C(F)(F)F)c3ccnn3c4cccc(c4)Cl 12L-912 c1ccc(cc1)COC(=O)NC(Cc2cnc[nH]2)C(=O)NN 12L-913 Cn1c(=O)c(nn(c1=O)c2cccc(c2)C(F)(F)F)c3ccno3 12L-914 Cn1c(=O)c(nn(c1=O)c2cccc(c2)C(F)(F)F)c3ccnn3c4c(cc(cn4)C(F)(F)F)Cl 12L-915 c1c2n(cn1)C(=O)NC(C2)C(=O)NN 12L-916 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)c3ccc(cc3Cl)Cl 12L-917 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)c3ccc(cc3)Cl 12L-918 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F 12L-919 Cc1c(c(no1)C(=O)N)C(=O)N 12L-920 c1cc(cc(c1)NC(=O)NNC(=O)C2Cc3cncn3C(=O)N2)C(F)(F)F 12L-921 CCOC(=O)C1C2C(C(=C3C(=O)c4ccccc4C3=O)N1)C(=O)N(C2=O)c5cccc(c5)C(F)(F)F 12L-923 CCOC(=O)C1C2C(C(=C3C(=O)c4ccccc4C3=O)N1)C(=O)N(C2=O)c5ccc(cc5Cl)Cl 12L-924 CCOC(=O)C1C2C(C(=C3C(=O)c4ccccc4C3=O)N1)C(=O)N(C2=O)c5ccc(cc5)Cl 12L-925 CCOC(=O)C1C2C(C(=C3C(=O)c4ccccc4C3=O)N1)C(=O)N(C2=O)N(C)c5c(cc(cn5)C(F)(F)F)Cl 12L-926 CCOC(=O)Cc1c(cccn1)C(=O)Nc2ccc(cc2)Oc3ccccc3 12L-927 c1ccc(cc1)/C=C/C2C3C(C4N2CSC4)C(=O)N(C3=O)CCNc5c(cc(cn5)C(F)(F)F)Cl 12L-928 c1cc2ccn(c2nc1)c3c(cc(cn3)C(F)(F)F)Cl 12L-929 CCOC(=O)C1C2C(C(=C3C(=O)c4ccccc4C3=O)N1)C(=O)N(C2=O)c5ccsc5C(=O)OC 12L-930 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)N(C)c3c(cc(cn3)C(F)(F)F)Cl 12L-931 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 12L-932 Cc1cc2c([nH]1)cccc2OCC(CNC(C)(C)C)O 12L-933 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)c3ccsc3C(=O)OC 12L-934 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)c3ccccc3 12L-936 CCOC(=O)C1C2C1C(=O)N(C2=O)c3ccccc3 12L-937 Cc1cccc(c1)CN2C(=O)C(=O)N(C2=O)OCc3cccc(c3)Cl 12M-001 c1cc(cc(c1)C(F)(F)F)CN2C(=O)C(=O)N(C2=O)CC(=O)N 12M-002 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2ccc(c(c2)Cl)Cl 12M-003 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2cccc(c2)F 12M-004 c1cc(cc(c1)F)CN2C(=O)C(=O)N(C2=O)CC(=O)O 12M-005 c1cc(ccc1CN2C(=O)C(=O)N(C2=O)CC(=O)N)Cl 12M-006 CCOC(=O)CNC(=S)Nc1ccccc1 12M-007 c1ccc(cc1)N2C(=O)CNC2=S 12M-008 c1ccc(cc1)N2C(=O)/C(=C/c3ccc(cc3)Cl)/NC2=S 12M-009 CC(C)c1ccc(cc1)/C=C\2/C(=O)N(C(=S)N2)c3ccccc3 12M-010 CCOC(=O)CNC(=S)Nc1ccc(cc1)OC 12M-011 CN(C)/C=C\1/C(=O)N(C(=S)N1)c2ccccc2 12M-012 COc1ccc(cc1)N2C(=O)CNC2=S 12M-013 c1cc(cnc1)CN2C(=O)CNC2=S 12M-014 CCOc1ccc(cc1/C=C\2/C(=O)N(C(=S)N2)c3ccc(cc3)OC)Br 12M-015 CC(C)c1ccc(cc1)/C=C\2/C(=O)N(C(=S)N2)c3ccc(cc3)OC 12M-016 c1cc(c(cc1CN2C(=O)C(=O)N(C2=O)OCc3ccc(cc3Cl)Cl)Cl)Cl 12M-017 c1cc(c(cc1CN2C(=O)C(=O)N(C2=O)CC(=O)O)Cl)Cl 12M-018 COc1ccc(cc1)N2C(=O)/C(=C/c3ccc(cc3)Cl)/NC2=S 12M-019 CN(C)/C=C\1/C(=O)N(C(=S)N1)c2ccc(cc2)OC 12M-020 c1cc(cnc1)CN2C(=O)/C(=C/c3ccc(cc3)Cl)/NC2=S 12M-021 CCOc1ccc(cc1/C=C\2/C(=O)N(C(=S)N2)Cc3cccnc3)Br 12M-022 CC(C)c1ccc(cc1)/C=C\2/C(=O)N(C(=S)N2)Cc3cccnc3 12M-023 c1ccc(c(c1)CON2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)F)F 12M-025 c1cc(cc(c1)F)CN2C(=O)C(=O)N(C2=O)OCc3cccc(c3)Cl 12M-026 COc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC#N 12M-027 Cc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)OCc3ccc(cc3)F 12M-028 Cc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)OC 12M-029 c1ccc(c(c1)CN2C(=O)C(=O)N(C2=O)CC(=O)N)Cl 12M-030 c1cc(cc(c1)C(F)(F)F)CN2C(=O)C(=O)N(C2=O)CC#N 12M-031 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2c(cccc2Cl)Cl 12M-033 CCOC(=O)CN1C(=O)C(=O)N(C1=O)Cc2ccccc2Cl 12M-034 COc1ccc(cc1)c2c(cc(cn2)C(F)(F)F)Cl 12M-035 c1cc(c(c(c1)Cl)CN2C(=O)C(=O)N(C2=O)CC(=O)O)Cl 12M-036 c1ccc(c(c1)CN2C(=O)C(=O)N(C2=O)CC(=O)O)Cl 12M-037 c1cc(ccc1c2c(cc(cn2)C(F)(F)F)Cl)O 12M-039 CCc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)CC(=O)O 12M-040 c1ccc(c(c1)n2cccc2C=O)F 12M-041 Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)C(C)(C)C)c2ccccc2 12M-301S Cc1cc(nc(c1S(=O)(=O)C)N(C)NC(=O)C2CC2)c3ccccc3 12M-302S Cn1cc(c(n1)C(F)(F)F)NC(=O)OCc2ccc(cc2)OC 12M-304S Cn1cc(c(n1)C(F)(F)F)NC(=O)OCc2ccc(cc2)Cl 12M-305S Cn1cc(c(n1)C(F)(F)F)NC(=O)OCCc2ccc(c(c2)OC)OC 12M-306S CC(C)(C)COC(=O)Nc1cn(nc1C(F)(F)F)C 12M-307S Cn1cc(c(n1)C(F)(F)F)NC(=O)OCc2ccc(cc2Cl)Cl 12M-308S COc1ccc(cc1)CN2CCn3c(cc(n3)C(=O)NC4CC4)C2=O 12M-310S CC(C)NC(=O)c1cc2n(n1)CCN(C2=O)Cc3ccc(cc3)OC 12M-311S Cc1ccc(cc1)Sc2c(nc([nH]2)c3ccccc3)/C=N/c4cccc(c4)C(F)(F)F 12M-312S CCSc1ncc(n1C)/C=N/c2ccc(cc2)Cl 12M-314S CCSc1ncc(n1C)/C=N/c2ccc(cc2Cl)Cl 12M-315S CCSc1ncc(n1C)/C=N/c2ccc(cc2C)Cl 12M-316S CCSc1ncc(n1C)/C=N/c2nccs2 12M-317S CCSc1ncc(n1C)/C=C(\C#N)/c2ccc(cc2)OC 12M-318S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)C(=O)C(F)(F)F 12M-319S CCSc1ncc(n1C)/C=C(\C#N)/c2ccccc2 12M-320S CCSc1ncc(n1C)/C=C(\C#N)/c2cccc(c2)Cl 12M-321S CCSc1ncc(n1C)/C=C(\C#N)/c2ccc(c(c2)Cl)Cl 12M-322S CCSc1ncc(n1C)/C=C(/C#N)\S(=O)(=O)C 12M-323S C=CCSc1ncc(n1Cc2ccccc2)/C=N/OCc3ccc(cc3Cl)Cl 12M-324S CCSc1ncc(n1C)C=C(C#N)C#N 12M-325S CCOC(=O)/C(=C/c1cnc(n1C)SCC)/C#N 12M-326S Cn1cc(c(n1)C(F)(F)F)C(=O)Oc2ccc(cc2)OC 12M-329S Cc1cccc(c1C)OC(=O)c2cn(nc2C(F)(F)F)C 12M-330S Cn1cc(c(n1)C(F)(F)F)C(=O)Oc2cccc(c2)C(F)(F)F 12M-331S Cn1cc(c(n1)C(F)(F)F)C(=O)Oc2ccc(cc2)C#N 12M-332S Cn1cc(c(n1)C(F)(F)F)C(=O)Oc2ccc(cc2F)F 12M-333S Cn1cc(c(n1)C(F)(F)F)C(=O)Oc2cc(nn2C)C(F)(F)F 12M-335S Cn1cc(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC 12M-336S Cn1cc(c(n1)C(F)(F)F)NC(=O)c2ccc(cc2F)F 12M-337S Cn1cc(c(n1)C(F)(F)F)c2nnnn2c3ccc(cc3)OC 12M-338S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N\OC)/C(F)(F)F 12M-340S Cn1c2c(cn1)nc([nH]2)c3ccccc3 12M-341S Cc1c(sc2n1ncn2)C(C)OC(=O)Nc3cccc(c3)Cl 12M-501S Cc1c(sc2n1ncn2)C(C)OC(=O)Nc3ccccc3 12M-502S c1ccc(cc1)CNC(=O)c2cnc(nc2Sc3ccc(cc3)Cl)c4ccccc4 12M-506S c1cc(ccc1C(F)(F)F)NC(=O)c2c(cc(=O)n(n2)c3ccc(cc3)Cl)C(F)(F)F 12M-507S c1cc(ccc1C(F)(F)F)n2c(=O)cc(c(n2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F 12M-508S C=CCNC(=O)c1cnc(nc1Sc2ccc(cc2)Cl)c3ccccc3 12M-509S COc1ccc(cc1)Oc2c(cnc(n2)c3ccccc3)C(=O)O 12M-510S c1ccc(cc1)c2ncc(c(n2)Oc3ccc(cc3)Cl)C(=O)O 12M-511S c1ccc(cc1)c2ncc(c(n2)Oc3cc(c(cc3Cl)Cl)Cl)C(=O)O 12M-512S Cc1ccc(cc1)Oc2c(cnc(n2)c3ccccc3)C(=O)O 12M-516S Cc1cccc(c1C)Oc2c(cnc(n2)c3ccccc3)C(=O)O 12M-517S c1c(cc(c2c1[nH]c(n2)C(F)(F)F)Cl)Cl 12M-519S c1ccc(cc1)NC(=O)c2c(cc(=O)n(n2)c3ccccc3)C(F)(F)F 12M-525S Cc1ccc(cc1)C(=O)OC(C)c2c(n3c(s2)ncn3)C 12M-526S Cc1c(sc2n1ncn2)C(C)OC 12M-527S c1ccc(cc1)c2ncc(c(n2)Sc3cccc(c3)C(F)(F)F)C(=O)N4CCOCC4 12M-528S CN(C)C(=O)c1cnc(nc1Sc2cccc(c2)C(F)(F)F)c3ccccc3 12M-530S c1ccc(cc1)c2ncc(c(n2)Sc3cccc(c3)C(F)(F)F)C(=O)NC4CC4 12M-531S c1ccc(cc1)c2ncc(c(n2)Sc3cccc(c3)C(F)(F)F)C(=O)Nc4cccc(c4)C(F)(F)F 12M-532S c1ccc(cc1)c2ncc(c(n2)Sc3cccc(c3)C(F)(F)F)C(=O)Nc4ccc(cc4)C(F)(F)F 12M-533S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)C=O 12M-534S COC(C(=O)Nc1cc(cc(c1)Cl)Cl)C(=O)O 12M-535S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F 12M-536S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F 12M-537S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)Nc3ccc(cc3)C(F)(F)F)C(F)(F)F 12M-538S COC(=O)c1c(c(n(n1)c2ccccc2)Sc3ccc(cc3)Cl)C=O 12M-541S Cc1ccc(cc1)NC(=O)OC(C)c2c(n3c(s2)ncn3)C 12M-543S Cc1c(sc2n1ncn2)C(C)OC(=O)Nc3cccc(c3)C(F)(F)F 12M-544S Cc1c(sc2n1ncn2)C(C)OC(=O)Nc3ccc(cc3)F 12M-545S CCOC(=O)c1c(cc(=O)n(n1)c2cccc(c2)Cl)C(F)(F)F 12M-552S COC(=O)c1c(c(n(n1)c2ccccc2)Sc3ccc(cc3)Cl)/C=N/OCc4ccc(cc4Cl)Cl 12M-554S Cc1cccc(c1)NC(=O)OC(C)c2c(n3c(s2)ncn3)C 12M-557S Cc1c(sc2n1ncn2)C(C)OC(=O)Nc3ccc(c(c3)Cl)Cl 12M-558S Cc1ccc(cc1)S(=O)(=O)NC(=O)OC(C)c2c(n3c(s2)ncn3)C 12M-561S Cc1c(sc2n1ncn2)C(C)OC(=O)c3ccc(cc3)F 12M-562S CCOC(=O)/C(=N\Nc1ccc(cc1F)F)/C(=O)C(F)(F)F 12M-563S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OCc3ccc(cc3Cl)Cl 12M-564S c1cc(cc(c1)Cl)n2c(=O)cc(c(n2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F 12M-566S c1cc(c(cc1F)F)N/N=C(\C(=O)C(F)(F)F)/C(=O)O 12M-569S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OCc3c(cccc3Cl)Cl 12M-571S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OCc3cccc(c3)F 12M-572S Cc1ccc(cc1)CO/N=C/c2c(nn(c2Cl)c3ccccc3)C(=O)OC 12M-573S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OC 12M-574S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/O 12M-575S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OCc3ccc(cc3)F 12M-577S c1cc(ccc1C(F)(F)F)NC(=O)c2c(cc(=O)n(n2)c3ccc(cc3F)F)C(F)(F)F 12M-581S C1CCC(=NN=C(N)N)C1 12M-700 c1cc(nc(c1)Nc2c(cc(cn2)C(F)(F)F)Cl)Nc3c(cc(cn3)C(F)(F)F)Cl 12M-701 c1cc(c(c(c1)Cl)CCC(=O)/C=C/c2ccc3c(c2)OCO3)Cl 12M-703 COc1ccc(cc1)C2c3c(nn(c3OC(=C2C#N)N)c4ccccc4)c5ccccc5 12M-704 Cc1c2c(n(n1)c3ccccc3)OC(=C(C2c4ccc(cc4)OC)C#N)N 12M-706 Cc1ccc(cc1)c2ccnc(n2)[S-].[K+] 12M-707 Cc1ccc(cc1)c2ccnc(n2)S 12M-708 c1ccc(c(c1)c2ccnc(n2)S)O 12M-710 c1ccc(cc1)n2c(=O)c3c(ccs3)nc2SC(F)F 12M-711 c1ccc(c(c1)C(F)(F)F)N2CC2c3ccncc3 12M-713 Cc1cc(cc(c1)N/C(=C/C(=O)C(F)(F)F)/C)C 12M-714 Cc1ccc(cc1)c2ccnc(n2)SC(F)F 12M-718 c1ccc(c(c1)c2ccnc(n2)SC(F)F)O 12M-719 Cc1ccc(cc1)Cn2ccc(c(c2=O)Cc3ccccc3)O 12M-720 COC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)OC 12M-726 c1ccc(c(c1)[N+](=O)[O-])OC(F)F 12M-728 COc1ccc(cc1OC2CCCC2)C(CC(=O)OC)C[NH3+].[Cl-] 12M-729 CC(=O)Cc1c(cc(cn1)C(F)(F)F)Cl 12M-732 c1ccc(cc1)c2cc(on2)OS(=O)(=O)c3ccc(cc3Cl)Cl 12M-900 c1ccc(cc1)c2cc(=O)on2S(=O)(=O)c3ccccc3 12M-901 c1ccc(cc1)c2cc(=O)on2C(=O)Nc3cccc(c3)Cl 12M-902 CCNC(=O)n1c(cc(=O)o1)c2ccccc2 12M-907 c1ccc2c(c1)nc(o2)c3cnc(nc3)c4ccccn4 12M-908 c1ccc2c(c1)nc(o2)c3cnc(nc3)c4cccnc4 12M-909 c1ccc2c(c1)nc(o2)c3cnc(nc3)c4ccncc4 12M-910 c1ccc(cc1)c2cc(=O)on2C(=O)NC3CCCCC3 12M-912 COc1cc(c(cc1Cl)F)I 12M-918 CCC(=O)n1c(cc(=O)o1)c2ccccc2 12M-919 c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)(=O)c4ccccc4Cl 12M-920 C1c2c(c(c(c(n2)N)C#N)N)C(=O)NC1=O 12M-921 CCOC(=O)/C(=N\Nc1ccc(cc1)F)/c2c(c(c(c(n2)N)C#N)N)C#N 12M-923 CC(=O)c1cn(c2c1cccc2)C(=O)C 12M-924 CC(=O)n1cc(c2c1cccc2)C(=C)c3cn(c4c3cccc4)C(=O)C 12M-925 CC(=O)Nc1ccccc1OCc2cnc(s2)Cl 12N-001 CC(c1ccccc1)Nc2c3cc(c(cc3ncn2)OC)OC 12N-002 c1cc(ccc1C(=O)N/N=C/c2ccc(c(c2)Cl)Cl)OCc3ccc(c(c3)Cl)Cl 12N-003 CC(C)(C)c1ccc(cc1)/C=N\NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl 12N-004 c1cc(ccc1C(=O)N/N=C/c2cnc(s2)Cl)OCc3ccc(c(c3)Cl)Cl 12N-005 COc1cc2c(cc1OC)ncnc2Nc3cc(cc(c3)F)F 12N-006 c1cc(cc(c1)OCc2cnc(s2)Cl)C=O 12N-008 COc1ccc(cc1)Oc2ccccc2/C=N/NC(=O)c3ccc(cc3)OCc4ccc(c(c4)Cl)Cl 12N-009 c1ccc(c(c1)/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl)Oc4ccc(cc4)Cl 12N-010 CN1CCN(CC1)c2ncc(s2)C=O 12N-013 COc1cc(cc(c1)OC)Nc2c3cc(c(cc3ncn2)OC)OC 12N-014 c1cc(cc(c1)Cl)/C=N/NC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O 12N-017 COc1cc2c(cc1OC)ncnc2NCc3ccccn3 12N-020 Cc1ccc(cc1)Oc2ccccc2/C=N/O 12N-021 c1ccc(cc1)Oc2ccccc2/C=N/O 12N-022 COc1ccc(cc1)Oc2ccccc2/C=N/O 12N-027 c1ccc(c(c1)/C=N/O)Oc2ccc(cc2)Cl 12N-028 COc1ccc(cc1)CNc2c3cc(c(cc3ncn2)OC)OC 12N-029 COc1cc2c(cc1OC)ncnc2NCc3cccc(c3)Cl 12N-030 COc1cc2c(cc1OC)ncnc2NCc3ccc(c(c3)Cl)Cl 12N-031 COc1ccc(cc1OC)CNc2c3cc(c(cc3ncn2)OC)OC 12N-032 COc1cc2c(cc1OC)ncnc2NCc3cccc(c3F)F 12N-033 COc1cc2c(cc1OC)ncnc2NCc3cccc(c3)C(F)(F)F 12N-034 Cc1cc(cc(c1)Oc2ccccc2C=O)C 12N-035 COc1ccc(cc1)Oc2ccccc2/C=C/C(=O)O 12N-036 CC(C)(C)c1ccc(cc1)Oc2ccccc2C=O 12N-037 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccc(cc2)Cl 12N-039 Cc1ccc(cc1)Oc2ccccc2/C=C/C(=O)O 12N-040 COC(CNC(=O)c1c(c2cccc3c2n(c1=O)CC3)O)OC 12N-041 COc1cc2c(cc1OC)ncnc2NCC3CCCO3 12N-042 CC(C)(C)c1ccccc1NC(=O)c2c(c3cccc4c3n(c2=O)CC4)O 12N-043 c1cc2c3c(c1)c(c(c(=O)n3CC2)C(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)O 12N-044 COc1cc2c(cc1OC)ncnc2NCC=C 12N-045 c1ccc(cc1)/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl 12N-047 COc1ccc(cc1OC)CCNc2c3cc(c(cc3ncn2)OC)OC 12N-048 CCN(CC)c1ncc(s1)/C=N\O 12N-051 Cc1ccc(cc1)COc2ccc(cc2)C(=O)NN 12N-052 COc1cc(ccc1OCc2ccc(cc2)F)/C=N/NC(=O)c3ccc(cc3)OCc4ccc(c(c4)Cl)Cl 12N-053 c1cc(ccc1C(=O)N/N=C/c2ccc(o2)c3ccc(cc3Cl)Cl)OCc4ccc(c(c4)Cl)Cl 12N-054 COc1cc2c(cc1OC)ncnc2NCc3cccs3 12N-055 COC(=O)c1ccc(nc1)N 12N-057 c1ccc(c(c1)C=O)Oc2ccc(cc2Cl)Cl 12N-058 Cc1ccc(cc1)COc2ccc(cc2)C(=O)N/N=C/c3ccccc3Oc4cc(cc(c4)C)C 12N-060 COc1cc2c(cc1OC)ncnc2Nc3ccsc3C(=O)OC 12N-061 COc1cc2c(cc1OC)ncnc2NCCSc3ccc(cc3)Cl 12N-063 c1ccc(cc1)S(=O)(=O)Cc2cnc(s2)Cl 12N-064 COc1cc2c(cc1OC)ncnc2NCc3ccc4c(c3)OCO4 12N-066 c1ccc(c(c1)C=O)Oc2cccc(c2)Cl 12N-067 Cc1ccc(o1)CNc2c3cc(c(cc3ncn2)OC)OC 12N-069 c1ccc(c(c1)C=O)Oc2ccc(cc2)F 12N-071 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccc(cc2Cl)Cl 12N-072 Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)cn[nH]3 12N-074 CCOC(=O)C1CCN(CC1)c2ncc(s2)C=O 12N-075 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)C#N 12N-076 CC(=O)c1ccccc1OCc2cnc(s2)Cl 12N-077 Cc1ccc(cc1)COc2ccc(cc2)C(=O)N/N=C/c3ccc(c(c3)[N+](=O)[O-])Cl 12N-078 Cc1ccc(cc1)COc2ccc(cc2)C(=O)N/N=C/C=C\c3ccccc3 12N-079 COc1ccc(cc1)Oc2ccc(cc2)C#N 12N-080 Cc1ccc(cc1)COc2ccc(cc2)C(=O)N/N=C/c3ccc(cc3)NC(=O)C 12N-081 c1cc(ccc1CO)OCc2cnc(s2)Cl 12N-082 c1cc(ccc1C#N)Oc2ccc(cc2)F 12N-083 COc1cc2c(cc1OC)ncnc2NCc3ccccc3Cl 12N-085 CCCCCCCCCCCC(=O)NCCCN(C)C 12N-100 CCCc1ccc(c(c1)F)c2ccc(cc2)C(=O)Cc3ccc(cc3)Cl 12N-101 CCCCCCCCc1ccc(cc1)CCc2ccc(cc2)c3ccc(cc3)Br 12N-102 c1ccc(cc1)COc2ccc3cc(ccc3c2)Br 12N-104 CCC1CCC(CC1)C(=O)O 12N-105 CCOC(=O)C(c1ccccc1)Oc2ccc(cc2)c3ccc(cc3)OC(c4ccccc4)C(=O)OCC 12N-106 CCCCCCOc1ccc(cc1)/C=C/C(=O)Oc2ccc(cc2)CC(C)CC 12N-107 CCCCCCCCOc1ccc2ccccc2c1Cl 12N-108 CCCCOc1ccc2cc(ccc2c1)Br 12N-111 C=CCCCCCCCCCOc1ccc(cc1)C(=O)O 12N-112 CCCCCCCCOc1ccc(cc1)/C=C/C(=O)O 12N-113 CCCCCCOc1ccc(cc1)O 12N-116 CCCCCC1CCC(CC1)C(=O)O 12N-117 C=CCC(=O)OCCCCCCOc1ccc(cc1)C(=O)O 12N-118 CC(=C)C(=O)OCCCOc1ccc(cc1)C(=O)O 12N-119 CC(=C)C(=O)OCCCCOc1ccc(cc1)C(=O)O 12N-120 COC(c1ccccc1)C(=O)O 12N-121 CCOc1ccc2cc(ccc2c1)Br 12N-122 CCCCCCCCCCOc1ccc(cc1)/C=C\C(=O)O 12N-125 CC(C)CCCCC(C)CCOc1ccc(cc1)C(=O)O 12N-126 CCCCCC1COC(OC1)c2ccc(cc2)Br 12N-128 c1cc(ccc1C#N)c2ccc(cc2)C(=O)O 12N-132 c1cc(ccc1C(=O)O)OCCCCOC(=O)CCCl 12N-134 CCCCCCCCCCCC1CCC(CC1)CC(=O)O 12N-135 CCCCCCOc1ccc(cc1)OCC(=O)O 12N-137 CCCCCCCCOc1ccc(cc1)/C=C/C(=O)OC 12N-138 CCCCCC1CCC(CC1)c2ccc(cc2)Br 12N-139 CCCCCCCCCCc1ccc(cc1)C(=O)Oc2ccc(cc2)c3ccc(cc3)C#N 12N-140 C=CCCCCCCCOc1ccc(cc1)C(=O)O 12N-141 c1cc(ccc1C(=O)O)OCCO 12N-142 CC(=C)C(=O)OCCCCCCOc1ccc(cc1)C(=O)O 12N-145 CCCCCCCCOc1ccc2cc(ccc2c1Cl)C(=O)O 12N-149 COC(=O)c1ccc(cc1)c2ccc(cc2)O 12N-153 CCC(C)COc1ccc2cc(ccc2c1)Br 12N-158 CCc1ccc(cc1)C(=O)Oc2ccc(cc2)CC 12N-161 c1ccc(cc1)COc2ccc(cc2)c3c(c(c(c(c3F)F)Br)F)F 12N-162 C=CCOc1cc(cc(c1)OCC=C)C(=O)O 12N-164 C=CCC(=O)OCCCCCCCCCCCOc1ccc(cc1)C(=O)O 12N-165 CC(C(=O)O)Oc1ccc(cc1)OCc2ccccc2 12N-166 CCC(=O)OCCCCCCOc1ccc(cc1)C(=O)O 12N-167 CCCCCCCCOc1ccc(cc1F)c2ccc(cc2)O 12N-169 CC(=O)Oc1ccc(cc1F)c2ccc(cc2)OCc3ccccc3 12N-171 COC(=O)c1ccc(cc1)OCCCBr 12N-172 c1cc(ccc1c2ccc(cc2F)C(=O)O)OCCCCCO 12N-173 CC(CO)Oc1ccc(cc1)c2ccc(c(c2)F)c3ccc(cc3)OC(C)CO 12N-175 CCCCCCCCCCCCOc1ccc(cn1)C(=O)O 12N-176 CCCCCCCCCOc1ccc(cc1)c2ccc(cc2)CCC(=O)O 12N-177 CCCCCc1ccc(c(c1)F)C#Cc2ccc(cc2)Br 12N-178 CCCCCCCCCCOc1ccc(cn1)C(=O)O 12N-180 c1cc(ccc1CCc2ccc(cc2)Cl)O 12N-184 CCCCCCCCCCCCC/C=C/CC(CC(=O)O)C(=O)O 12N-186 CCCC1CCC(CC1)CCc2ccc(c(c2)F)OS(=O)(=O)C(F)(F)F 12N-187 c1ccc(cc1)COC(=O)CCCBr 12N-190 CCCCCc1ccc(cc1)Br 12N-191 CCCCCCCCCCCCCCCC[n+]1ccccc1.[Br-] 12N-193 CCCCCCCCCCCCCCCC[n+]1ccccc1.[I-] 12N-196 CCC(C)COc1ccc(cc1)O 12N-198 c1c(c[nH+]c([nH+]1)O)Br.[Cl-].[Br-] 12N-200 CCCCCCCCCCCCCCCCCC[n+]1ccccc1.[Cl-] 12N-201 CCCCCCCCCCCCCCCCCCCC[n+]1ccccc1.[Br-] 12N-203 c1ccc(cc1)COc2ccc(cc2F)O 12N-206 c1cc(c(c(c1)F)F)c2ccc(cc2)Cl 12N-207 COC(=O)c1ccc(cc1)OCCCCCCOc2ccc(cc2)C(=O)OC 12N-208 CSc1ccc(cc1)c2cccc(c2F)F 12N-209 c1ccc(cc1)COc2ccc3cc(ccc3c2)c4ccc(cc4F)Br 12N-212 c1cc(ccc1c2ccc(cc2)OCCCCCCCCCCO)C(=O)O 12N-213 C(C(C(C(C(C(C(C(C(C(C(F)F)(F)F)(F)F)(F)F)(F)F)(F)F)(F)F)(F)F)(F)F)(F)F)O 12N-214 CC(=O)Oc1ccc(cc1)c2ccc(cc2)C#N 12N-216 CCCC(=O)c1ccc(cc1)c2ccccc2 12N-223 c1ccc(cc1)c2ccc(cc2F)O 12N-225 CCCCCCCCCc1ccc(cc1)C(=O)O 12N-227 CCCCCOc1ccc(cc1)CC(=O)O 12N-228 CCCCCCC1CCC(CC1)C(=O)O 12N-229 CCCCCCCCOc1ccc(cc1F)Br 12N-231 CCCCCCCCCCOc1ccc(cc1)O 12N-236 CCCCCC1CCC(CC1)CC(=O)O 12N-237 CCCCCCCCOc1ccc(cc1)C(=[NH2+])N.[Cl-] 12N-238 CCC(=O)c1ccc(c(c1)F)OC 12N-239 c1cc(ccc1C2CCC(CC2)C(=O)O)Cl 12N-240 CCC(C)Cc1ccc(cc1)c2ccc(cc2)C(=O)O 12N-244 CCCCCC1(CCC(=O)CC1)C(=O)C 12N-245 CCCCCC1CCC(CC1)CBr 12N-247 CCCCCCCCCOc1ccc(cc1)c2ccc(cc2)C(=O)O 12N-248 C#Cc1ccc(cc1)OCc2ccccc2 12N-249 c1cc(ccc1C(=O)O)OCCCCCCOC2CCCCO2 12N-253 CCCC1CCC(CC1)C(=O)O 12N-254 CCCCCCCCCCCCCCCCCC[n+]1ccccc1.[Br-] 12N-255 CCc1ccc(c(c1)F)c2ccccc2 12N-256 CC(C)CCOc1ccc(cc1)C(=O)O 12N-257 CCCCCC1CCC(CC1)c2ccc(cc2)N 12N-259 CCNC(=O)C1=C(c2c(ccs2)N(S1(=O)=O)C)O 12N-301S CN1c2ccsc2C(=C(S1(=O)=O)C(=S)Nc3ccc(cc3)Cl)O 12N-302S Cc1ccc(cc1)NC(=S)C2=C(c3c(ccs3)N(S2(=O)=O)C)O 12N-303S Cc1ccccc1SCC2CSc3n2c(=O)c4ccccc4n3 12N-305S Cc1cccc(c1)SCC2CSc3n2c(=O)c4ccccc4n3 12N-306S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccc(cc4)Br 12N-307S CN1c2ccsc2C(=C(S1(=O)=O)C(=S)Nc3ccc(c(c3)Cl)F)O 12N-308S CN1c2ccsc2C(=C(S1(=O)=O)C(=S)Nc3ccccc3OC)O 12N-309S Cc1ccccc1NC(=S)C2=C(c3c(ccs3)N(S2(=O)=O)C)O 12N-310S CN1c2ccccc2C(=C(S1(=O)=O)C(=O)Nc3ccccc3)O 12N-311S c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccccc3 12N-312S CC(C)(C)OC(=O)CN1CCNCC1 12N-315S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccccc4Cl 12N-321S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4cccc(c4)Cl 12N-322S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4c(cccc4Cl)Cl 12N-323S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccccc4N 12N-324S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4cccc(c4Cl)Cl 12N-325S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4cc(ccc4Cl)Cl 12N-326S COc1cccc(c1)SCC2CSc3n2c(=O)c4ccccc4n3 12N-329S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSCc4ccc(cc4Cl)Cl 12N-330S c1ccc2c(c1)NC(=S)CS2 12N-331S c1ccc(cc1)CSCC2CSc3n2c(=O)c4ccccc4n3 12N-332S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSCc4ccc(cc4)Cl 12N-333S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSCc4cccc(c4)C(F)(F)F 12N-334S CN1c2ccccc2C(=C(S1(=O)=O)C(=O)Nc3cccc(c3)Cl)O 12N-336S CN1c2ccccc2C(=C(S1(=O)=O)C(=O)Nc3ccc(cc3)F)O 12N-337S CN1c2ccccc2C(=C(S1(=O)=O)C(=O)Nc3cccc(c3)C(F)(F)F)O 12N-338S Cc1cccc(c1)NC(=O)C2=C(c3ccccc3N(S2(=O)=O)C)O 12N-339S Cc1ccc(cc1)NC(=O)C2=C(c3ccccc3N(S2(=O)=O)C)O 12N-340S Cc1cccc(c1NC(=O)C2=C(c3ccccc3N(S2(=O)=O)C)O)C 12N-341S CN1c2ccccc2C(=C(S1(=O)=O)C(=O)Nc3ccc(cc3)Cl)O 12N-342S CCNC(=O)C1=C(c2ccccc2N(S1(=O)=O)C)O 12N-343S CN1c2ccccc2C(=C(S1(=O)=O)C(=O)Nc3ccc(c(c3)Cl)Cl)O 12N-345S CN1c2ccccc2C(=C(S1(=O)=O)C(=S)Nc3ccc(cc3)Cl)O 12N-346S CN1c2ccccc2C(=C(S1(=O)=O)C(=S)Nc3ccccc3)O 12N-347S CN1c2ccccc2C(=C(S1(=O)=O)C(=S)Nc3ccccc3OC)O 12N-348S Cc1ccc(cc1)NC(=S)C2=C(c3ccccc3N(S2(=O)=O)C)O 12N-349S CN1c2ccccc2C(=C(S1(=O)=O)C(=S)Nc3ccc(c(c3)Cl)F)O 12N-350S c1cc(cc(c1)F)CSC2=Nc3cc(ccc3SCC2)Cl 12N-352S c1cc(c(c(c1)Cl)CSC2=Nc3cc(ccc3SCC2)Cl)F 12N-353S c1cc(c(c(c1)Cl)CSC2=Nc3cc(ccc3SCC2)Cl)Cl 12N-354S COc1ccc(cc1)CSC2=Nc3cc(ccc3SCC2)Cl 12N-355S CC(=O)Cn1c(=O)c(c(cn1)Nc2ccc(cc2F)F)Br 12N-356S CC(=O)Cn1c(=O)c(c(cn1)NCC=C)Br 12N-357S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)NC2CC2)Br 12N-358S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)N(C)C)Br 12N-359S c1cc(ccc1C(=O)C(n2c(=O)c(c(cn2)Cl)Cl)(Br)Br)Cl 12N-360S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)N(C)C)Cl 12N-361S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)NCC=C)Cl 12N-362S CC(C)(C)C(=O)Cn1c(=O)c(c(cn1)NC2CC2)Cl 12N-363S c1ccc(cc1)C(=NNC(=O)COc2ccccc2)c3ccccc3 12N-364S Cc1ccccc1CSC2=Nc3cc(ccc3SCC2)Cl 12N-365S c1cc(c(cc1Cl)Cl)CSC2=Nc3cc(ccc3SCC2)Cl 12N-366S c1cc(ccc1C2C(=C(OC3=C2C(=O)CCC3)N)C#N)[N+](=O)[O-] 12N-372S c1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N 12N-373S Cc1cccc(c1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N 12N-374S Cn1c2ccccc2c3c1sc(c3)C(=O)NNS(=O)(=O)c4ccc(cc4)OC 12N-375S CC(=O)Nc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc3c4ccccc4n(c3s2)C 12N-376S Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc3c4ccccc4n(c3s2)C 12N-377S Cn1c2ccccc2c3c1sc(c3)C(=O)NNS(=O)(=O)c4ccc(cc4)F 12N-378S Cn1c2ccccc2c3c1sc(c3)C(=O)NNS(=O)(=O)c4ccc(cc4)Cl 12N-379S CO/N=C(\Cn1c(=O)c(c(cn1)NC2CCCCC2)Br)/c3ccc(cc3)Cl 12N-380S CCN(CC)c1cnn(c(=O)c1Br)C/C(=N\OC)/c2ccc(cc2)Cl 12N-381S CSC1=Nc2cc(ccc2SCC1)Cl 12N-386S CO/N=C(\Cn1c(=O)c(c(cn1)N2CCCC2)Br)/c3ccc(cc3)Cl 12N-418S c1ccc2c(c1)CCC(=C2Cl)C=O 12N-501S COC(=O)c1cc2c(s1)-c3ccccc3CC2 12N-502S c1ccc(cc1)N/N=C/C2=C(c3ccccc3CC2)Cl 12N-503S Cc1ccc(cc1)N/N=C/C2=C(c3ccccc3CC2)Cl 12N-505S c1ccc2c(c1)CCC(=C2Cl)/C=N/Nc3ccc(cc3)F 12N-506S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)O 12N-508S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)N4CCOCC4 12N-510S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)N4CCCCC4 12N-511S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)NC4CC4 12N-512S CNC(=O)c1cc2c(s1)-c3ccccc3CC2 12N-513S CN(C)C(=O)c1cc2c(s1)-c3ccccc3CC2 12N-514S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)Nc4ccc(cc4)Cl 12N-515S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)Nc4cc(cc(c4)Cl)Cl 12N-519S c1ccc2c(c1)[nH]c(n2)SCC(=O)c3ccc(cc3)Cl 12N-521S CCN1c2cc(ccc2SCC1=O)C(=O)OC 12N-523S Cc1cc\2c(n1c3ccc(cc3)OC)CCC/C2=N\Nc4ccccc4 12N-570S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)C3CC3 12N-641S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)c3cccc(c3)C(F)(F)F 12N-642S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)c3cccs3 12N-643S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3ccc(cc3)Cl 12N-645S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])CO)Cl 12N-646S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3cccc(c3)C(F)(F)F 12N-647S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3ccc(c(c3)Cl)Cl 12N-648S c1cc(cc(c1)Cl)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 12N-650S Cc1cccc(c1)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 12N-652S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)c3ccc(cc3)Cl 12N-655S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)c3cccc(c3)C(F)(F)F 12N-656S Cc1cccc(c1)NC(=O)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 12N-658S CCNC(=O)OCc1ccc(c(c1)[N+](=O)[O-])Sc2ccc(cc2)Cl 12N-659S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])COC(=O)NC3CCCCC3)Cl 12N-660S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)c3c(cccc3F)F 12N-661S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3cccc(c3)Cl 12N-662S c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3ccc(cc3)F 12N-663S Cc1cccc(c1)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Sc3nc4ccccc4s3 12N-664S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])COC(=O)c4cccc(c4)C(F)(F)F 12N-665S c1ccc(c(c1)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Sc3nc4ccccc4s3)Cl 12N-666S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CN3CCOCC3 12N-668S Cc1ccc(cc1)COn2ccnc2 12N-703 C#CCn1ccc(c(c1=O)Cc2c(cccc2Cl)F)O 12N-705 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)CCCN3CCOCC3)O)F 12N-706 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)CC3CCCO3)O)F 12N-707 CCOC(=O)C(Cc1c(cccc1Cl)F)c2ccnc3n2ncc3c4ccc(cc4)Cl 12N-708 c1cc(ccc1COn2ccnc2)F 12N-709 c1ccc(cc1)n2ccnc2 12N-710 c1c(cnc(c1Cl)n2c(nc(n2)Br)Br)C(F)(F)F 12N-712 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)Cc3ccncc3)O)F 12N-713 c1cc(ccc1Cn2c(nc(n2)Br)Br)F 12N-714 c1ccc(cc1)C(=O)Cn2c(nc(n2)Br)Br 12N-715 c1cc(ccc1S(=O)(=O)Cn2c(nc(n2)Br)Br)Cl 12N-716 c1ccc(cc1)COC(=O)n2c(nc(n2)Br)Br 12N-717 C1=CC(=O)C(C(C1=O)Br)Br 12N-719 CC(=O)C(Cc1cnc(s1)Cl)Cc2cnc(s2)Cl 12N-720 c1ccnc(c1)CCn2ccc(c(c2=O)Cc3c(cccc3Cl)F)O 12N-721 CCOC(=O)C(Cc1c(cccc1Cl)F)c2ccnc3n2nc(n3)SCc4cccc(c4)Cl 12N-723 c1ccc(cc1)COn2ccnc2C=O 12N-724 COc1cccc(c1)COn2ccnc2 12N-725 c1ccc(cc1)/C=C\COn2ccnc2 12N-726 c1cc(c(nc1)n2c(nc(n2)Br)Br)[N+](=O)[O-] 12N-727 c1cc(sc1)C(=O)n2c(nc(n2)Br)Br 12N-728 c1cc(ccc1COn2ccnc2)[N+](=O)[O-] 12N-730 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)Nc3cccc(n3)F)O)F 12N-732 CCOC(=O)C(Cc1c(cccc1Cl)F)c2ccnn2c3cccc(n3)F 12N-733 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)C3CC3)O)F 12N-735 CC(C(=O)C)n1c(nc(n1)Br)Br 12N-736 c1ccc(cc1)n2cc[nH+]c2S.[Cl-] 12N-737 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)CCc3ccc(cc3)S(=O)(=O)N)O)F 12N-740 c1cnc2ncnn2c1C(Cc3cnc(s3)Cl)Cc4cnc(s4)Cl 12N-741 c1cc(cc(c1)C(F)(F)F)Cn2ccc(c(c2=O)Cc3c(cccc3Cl)F)O 12N-742 c1ccc(cc1)CSC2=NCCN2C(=O)Oc3ccccc3 12N-746 Cc1ccc(cc1)S(=O)(=O)OCC(F)(F)F 12N-747 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)Nc3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)O)F 12N-748 CCCCCCCCCCCCn1ccc(c(c1=O)Cc2c(cccc2Cl)F)O 12N-750 Cc1cccc(c1C)Nc2c3ccc(cc3ncn2)Cl 12N-802 Cc1c(cccc1Cl)Nc2c3ccc(cc3ncn2)Cl 12N-803 c1cc2c(cc1Cl)ncnc2Nc3cc(cc(c3)F)F 12N-804 c1ccc(c(c1)CNc2c3ccc(cc3ncn2)Cl)F 12N-806 c1cc(cc(c1)Cl)CNc2c3ccc(cc3ncn2)Cl 12N-807 c1ccc(cc1)CNc2c3ccc(cc3ncn2)Cl 12N-808 c1cc(ccc1CNc2c3ccc(cc3ncn2)Cl)Cl 12N-809 Cc1ccc(cc1)CNc2c3ccc(cc3ncn2)Cl 12N-810 COc1ccc(cc1)CNc2c3ccc(cc3ncn2)Cl 12N-813 COc1ccc(cc1OC)CNc2c3ccc(cc3ncn2)Cl 12N-814 c1cc(c(c(c1)F)F)CNc2c3ccc(cc3ncn2)Cl 12N-815 c1cc(c(cc1CNc2c3ccc(cc3ncn2)Cl)Cl)Cl 12N-816 CC(c1ccccc1)Nc2c3ccc(cc3ncn2)Cl 12N-818 c1ccc(c(c1)CNc2c3ccc(cc3ncn2)Cl)C(F)(F)F 12N-819 c1cc(cc(c1)C(F)(F)F)CNc2c3ccc(cc3ncn2)Cl 12N-820 c1cc(c(cc1Cl)Cl)CNc2c3ccc(cc3ncn2)Cl 12N-821 c1cc(ccc1CNc2c3ccc(cc3ncn2)Cl)F 12N-822 COc1ccccc1CNc2c3ccc(cc3ncn2)Cl 12N-823 Cc1ccccc1CNc2c3ccc(cc3ncn2)Cl 12N-824 c1cc2c(cc1Cl)ncnc2NCC3CCCO3 12N-825 c1ccnc(c1)CNc2c3ccc(cc3ncn2)Cl 12N-826 C=CCNc1c2ccc(cc2ncn1)Cl 12N-827 c1cc(sc1)CNc2c3ccc(cc3ncn2)Cl 12N-828 c1ccc(cc1)CCNc2c3ccc(cc3ncn2)Cl 12N-829 CC1=NNC2(C1C(n3c(ncn3)N2)c4ccc(cc4)[N+](=O)[O-])C 12N-830 c1cc(oc1)CNc2c3ccc(cc3ncn2)Cl 12N-831 COCCCNc1c2ccc(cc2ncn1)Cl 12N-833 COc1ccc(cc1OC)CCNc2c3ccc(cc3ncn2)Cl 12N-834 c1cc2c(cc1CNc3c4ccc(cc4ncn3)Cl)OCO2 12N-835 CN(C)S(=O)(=O)CCN.Cl 12N-837 c1ccc(c(c1)CNc2c3ccc(cc3ncn2)Cl)Cl 12N-838 Cc1ccc(o1)CNc2c3ccc(cc3ncn2)Cl 12N-839 c1cc(ccc1SCCNc2c3ccc(cc3ncn2)Cl)Cl 12N-840 c1cc(ccc1CCNc2c3ccc(cc3ncn2)Cl)S(=O)(=O)N 12N-841 CCOC(=O)CN1CCC(CC1)C(=O)OC 12N-902 COC(=O)C1CCN(CC1)CC#N 12N-904 COC(=O)C1CCN(CC1)CC(=O)N 12N-905 COC(=O)CCN1CCC(CC1)C(=O)OC 12N-906 Cc1cc(c(c(c1)C#N)O)C#N 12N-951 CC(C)(C)c1cc(c(c(c1)C#N)OCc2ccc(cc2)[N+](=O)[O-])C#N 12N-952 CC(C)(C)c1cc(c(c(c1)C#N)OC(=O)c2ccc(cc2)C(F)(F)F)C#N 12N-960 COC(=O)/C=c\1/c(=O)[nH]c(=C)s1 12N-964 COC(=O)N1CCC(CC1)C(=O)O 12N-988 Cc1ccc(cc1)CSc2nnc(o2)c3ccc(cc3)C(C)(C)C 12P-002 CC(C)(C)c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)[N+](=O)[O-] 12P-003 CC(C)(C)c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)Cl 12P-004 CC(C)(C)c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)Br 12P-005 CN1C(=O)C(=Cc2ccc(cc2)OCc3c(cccc3Cl)F)C(=O)N(C1=O)C 12P-006 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/3\C(=O)NC(=O)S3)F 12P-008 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCCCF 12P-009 CC(C(=O)OC)Oc1ccc(cc1)c2nccc(n2)c3ccccn3 12P-010 c1cc(c(c(c1)Cl)COc2ccc(cc2)C=C3C(=O)NC(=O)NC3=O)F 12P-011 CC(C)(C)c1ccc(cc1)c2nnc(o2)SCC#N 12P-012 CCOC(=O)C/C(=N/NC(=O)CC#N)/c1ccccc1 12P-013 c1cc(cc(c1)Cl)COc2ccc(cc2)C=O 12P-014 CCOC(=O)C/C(=N/NC(=O)CC#N)/C(F)(F)F 12P-015 CC(C)(C)Oc1cccc(c1)C(=O)O 12P-016 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)c4ccc(cc4)Oc5cc(cc(n5)C(F)(F)F)C(F)(F)F 12P-018 c1cc(ccc1c2nccc(n2)c3ccc(cc3)F)OCC(=O)NN 12P-020 CCO/C(=N\NC(=O)c1ccc(cc1)C(F)(F)F)/C 12P-021 CCO/C(=N\NC(=O)c1ccccc1)/C 12P-022 CC(C(=O)NN)Oc1ccc(cc1)c2nccc(n2)c3ccccn3 12P-023 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=C/3\C(=O)NC(=O)S3 12P-024 CN1C(=O)C(=Cc2ccc(cc2)OCc3cccc(c3)Cl)C(=O)N(C1=O)C 12P-025 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCc4ccc(cc4)C(F)(F)F 12P-026 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCc4cc(cc(c4)C(F)(F)F)C(F)(F)F 12P-027 c1cc(ccc1CC#N)OCCCF 12P-028 c1cc(cc(c1)Cl)COc2ccc(cc2)C=C3C(=O)NC(=O)NC3=O 12P-029 c1ccc(cc1)SCC(CC(=O)c2ccc(cc2)c3ccc(cc3)Cl)C(=O)O 12P-030 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2CCC(C3=O)N4CCN(CC4)c5ccccc5OC 12P-032 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2CCC(C3=O)N4CCN(CC4)c5ccccc5F 12P-033 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCc4ccc(cc4)Br 12P-034 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)c3nccc(n3)c4cccs4 12P-035 CCOC(=O)C/C(=N/NC(=O)CC#N)/C 12P-036 C(C#N)C(=O)N/N=C(\CC(=O)C(F)(F)F)/C(F)(F)F 12P-040 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NN 12P-041 c1cc(oc1)/C(=N/NC(=O)CC#N)/CC(=O)C(F)(F)F 12P-043 c1cc(ccc1C=O)OCc2ccc(cc2Cl)Cl 12P-044 c1cc(ccc1COc2ccc(cc2)C=O)Br 12P-045 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCc4ccc(c(c4)Cl)Cl 12P-047 Cc1ccc(cc1)COc2ccc(cc2)c3nccc(n3)c4cccs4 12P-048 CCOC(=O)c1ccc(cc1)/N=C/c2ccccc2Oc3ccc(cc3)Cl 12P-049 CC(c1ccn(n1)C(=O)C2CC2)Oc3ccc(c(c3)F)c4ccccc4 12P-050 Cc1ccc(c(c1)/C=C/C(=O)N/N=C/c2ccc(cc2)OCc3c(cccc3Cl)F)C 12P-051 CC(c1ccn(n1)C(=O)c2ccc(cc2)F)Oc3ccc(c(c3)F)c4ccccc4 12P-056 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4cccs4 12P-057 Cc1cccc(c1)C(=O)Oc2ccc(cc2)c3nccc(n3)c4cccs4 12P-058 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OC(=O)C4CCCCC4 12P-059 Cc1nnc(o1)c2ccc(cc2)C(C)(C)C 12P-060 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)OCCCF 12P-061 c1cc(sc1)CNc2ccc(cc2Br)[N+](=O)[O-] 12P-062 COc1ccc(cc1)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 12P-064 c1ccc(cc1)CNC(=O)/C(=C/c2ccc(cc2)O)/C#N 12P-066 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl 12P-069 CC(c1ccn(n1)C(=O)c2cccs2)Oc3ccc(c(c3)F)c4ccccc4 12P-071 CC(c1ccn(n1)S(=O)(=O)c2cccc3c2cccc3)Oc4ccc(c(c4)F)c5ccccc5 12P-072 CCOC(=O)C(C)/C(=N/NC(=O)CC#N)/C 12P-073 c1cc(ccc1/C=N/NC(=O)c2ccc(cc2Cl)Cl)OCCCF 12P-074 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=N/NC(=O)c3ccc(cc3Cl)Cl)F 12P-075 c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)OCc3ccc(cc3Cl)Cl 12P-076 CC(c1ccn(n1)C(=O)c2ccc(cc2)I)Oc3ccc(c(c3)F)c4ccccc4 12P-077 COc1ccc(cc1)NC(=O)Oc2ccc(c(c2)F)c3ccccc3 12P-078 COc1ccccc1N2CCN(CC2)C3CCc4c(cc[nH]4)C3=O 12P-079 C/C(=N\NC(=O)CC#N)/CC(=O)c1ccccc1 12P-080 c1cc2c(cc[nH]2)c(c1)OCCOCCO 12P-081 c1cc(ccc1COc2ccc(cc2)/C=C/3\C(=O)NC(=O)S3)Br 12P-082 CN1C(=O)C(=Cc2ccc(cc2)OCc3ccc(cc3Cl)Cl)C(=O)N(C1=O)C 12P-083 CN1C(=O)C(=Cc2ccc(cc2)OCc3ccc(cc3)Br)C(=O)N(C1=O)C 12P-084 CC(c1ccn(n1)C(=O)C2CCCCC2)Oc3ccc(c(c3)F)c4ccccc4 12P-086 CCCCC(=O)n1ccc(n1)C(C)Oc2ccc(c(c2)F)c3ccccc3 12P-087 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(c(c2)F)c3ccccc3 12P-089 CC(c1ccn(n1)C(=O)c2c(cccc2F)F)Oc3ccc(c(c3)F)c4ccccc4 12P-090 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C4CCc5c(cc[nH]5)C4=O 12P-091 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OC(=O)NC4CCCCC4 12P-092 c1cc(ccc1/C=C/C(=O)O)OCCCF 12P-093 c1cc(cc(c1)Cl)COc2ccc(cc2)C=NNC(=O)c3ccc(cc3Cl)Cl 12P-095 Cc1ccccc1COc2ccc(cc2)C=O 12P-096 c1cc(ccc1CO)OCc2ccc(cc2Cl)Cl 12P-102 c1cc(ccc1CO)OCc2ccc(cc2)Br 12P-103 COc1ccc(cc1)c2ccnc(n2)c3ccc(cc3)OCc4cccc(c4)F 12P-105 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCCOCCNCc4ccc(cc4)F 12P-106 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCCOCCNCc4cccs4 12P-107 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCCOCCNCCN4CCOCC4 12P-108 Cc1ccc(cc1)NC(=O)n2ccc(n2)C(C)Oc3ccc(c(c3)F)c4ccccc4 12P-109 C/C(=N/NC(=O)CC#N)/CC(=O)C(F)(F)F 12P-110 CCOC(=O)C1(CC(=C(CC1C(=O)O)C)C)C(=O)OCC 12P-111 CCOC(=O)c1cn2ccccc2c1C(=O)OCC 12P-119 CC(c1ccnc(n1)N)Oc2ccc(c(c2)F)c3ccccc3 12P-120 CCOC(=O)c1c2ccccn2cc1c3ccccc3 12P-121 CCCc1c(nn(c1C)C(=O)CC#N)C 12P-122 CCc1c(nn(c1C)C(=O)/C(=C\N(C)C)/C#N)C 12P-124 CCOC(=O)c1c2ccccn2cc1c3ccc(cc3)Cl 12P-125 CCOC(=O)c1c2ccccn2cc1c3ccc(cc3)OC 12P-126 CCOC(=O)C(CSCCCN1C(=O)c2ccccc2C1=O)NS(=O)(=O)c3ccc(cc3Cl)Cl 12P-127 CCOC(=O)C(CSCC(CBr)O)NC(=O)OC(C)(C)C 12P-128 c1ccc(cc1)/C(=N/NC(=O)CC#N)/CC(=O)C(F)(F)F 12P-129 Cc1cccc(c1Oc2c(nc3ccccc3n2)C)C 12P-130 CC(C)(C)OC(=O)NC(CSCCCC(=O)O)C(=O)O 12P-131 CCOC(=O)C/C(=N/NC(=O)CC#N)/C(C)C 12P-132 CCc1c(nn(c1C)C(=O)CC#N)C 12P-133 CN1C(=O)C(=Cc2ccc(cc2)OCc3ccccc3)C(=O)N(C1=O)C 12P-134 c1ccc(cc1)COc2ccc(cc2)C=C3C(=O)NC(=O)NC3=O 12P-135 c1ccc(cc1)COc2ccc(cc2)/C=C/3\C(=O)NC(=O)S3 12P-137 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccc(cc4)I 12P-138 c1ccc(cc1)C(=O)Oc2ccc(cc2)c3nccc(n3)c4cccs4 12P-140 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccc(cc4)Cl 12P-141 COc1cc(ccc1Br)F 12P-143 CCC1c2c(c3ccccc3[nH]2)CCN1 12P-144 c1ccc(cc1)n2c(=N)c3ccccc3[nH]c2=S 12P-147 c1cc(ccc1CO)OCCCF 12P-148 c1ccc(cc1)COc2ccc(cc2)/C=N/Nc3ccc(cc3Cl)Cl 12P-149 CC(C)(C)c1ccc(cc1)N/N=C/c2ccc(cc2)OCc3ccccc3 12P-150 c1ccc(cc1)COc2ccc(cc2)/C=N/OCc3ccc(cc3Cl)Cl 12P-152 CCOC(=O)c1cc2cccn2cn1 12P-153 CC1(OC(=O)C(=Cc2ccc(cc2)OCc3ccccc3)C(=O)O1)C 12P-155 c1c2n(nc1C(=O)O)CCCNC2=O 12P-158 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=N/NC(=O)c3ccc(cc3)C(F)(F)F 12P-160 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=N/OCc3ccc(cc3Cl)Cl 12P-161 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)OCc3cccc(c3)Cl 12P-162 c1ccc(cc1)S(=O)(=O)n2c(cc3c2nccc3)C(c4ccc(cc4)F)O 12P-301S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCCCC3 12P-302S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCOCC3 12P-303S c1cc(c(c(c1)Cl)/C=N/n2c(nnc2S)c3cccs3)Cl 12P-304S c1cc(oc1)/C=N/n2c(nnc2S)c3cccs3 12P-306S c1cc(sc1)/C=N/n2c(nnc2S)c3cccs3 12P-307S c1ccc(cc1)CSc2nnc(o2)c3cnn(c3n4cccc4)c5ccccc5 12P-308S c1ccc(cc1)n2c(c(cn2)c3nnc(o3)SCc4ccc(cc4)F)n5cccc5 12P-309S C=CCSc1nnc(o1)c2cnn(c2n3cccc3)c4ccccc4 12P-310S c1ccc(cc1)CN2CCN(CC2)c3cc(=O)[nH]nc3c4ccccc4 12P-312S c1cc(c(nc1)Oc2ccc(c(c2)C(F)(F)F)Br)C(=O)Nc3ccc(cc3F)F 12P-314S COc1cccc(c1)/C=N/n2c(nnc2S)c3cccs3 12P-318S CC1C(=Nn2c(nnc2S1)c3cccs3)c4ccccc4 12P-325S CSc1nnc(n1c2ccccc2)c3cnn(c3n4cccc4)c5ccccc5 12P-331S CCCSc1nnc(n1c2ccccc2)c3cnn(c3n4cccc4)c5ccccc5 12P-332S COc1ccc(cc1)CSc2nnc(n2c3ccccc3)c4cnn(c4n5cccc5)c6ccccc6 12P-334S c1ccc(cc1)n2c(c(cn2)c3nnc(n3c4ccccc4)SCc5ccc(cc5)[N+](=O)[O-])n6cccc6 12P-335S CSc1nnc(o1)c2cnn(c2n3cccc3)c4ccccc4 12P-336S COc1ccc(cc1)CSc2nnc(o2)c3cnn(c3n4cccc4)c5ccccc5 12P-337S Cc1cccc(c1)CSc2nnc(n2c3ccccc3)c4cnn(c4n5cccc5)c6ccccc6 12P-340S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)c4ccccc4 12P-341S CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 12P-344S CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(cc2)C 12P-345S COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)NCC=C 12P-346S COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)N4CCOCC4 12P-347S COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)N4CCCC4 12P-348S c1ccc(cc1)C(=O)CCSc2ccccn2 12P-361S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)c4ccc(cc4)F 12P-362S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCC4(CC3)OCCO4 12P-363S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)C(=O)c4ccc(cc4)Cl 12P-364S c1cc(cc(c1)Oc2c(cccn2)C(=O)O)C(F)(F)F 12P-365S c1ccc(cc1)n2c(c(cn2)C(=O)NNS(=O)(=O)c3ccc(cc3)[N+](=O)[O-])n4cccc4 12P-367S c1ccc(cc1)n2c(c(cn2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl)n4cccc4 12P-368S c1ccc(cc1)n2c(c(cn2)C(=O)NNS(=O)(=O)c3ccccc3)n4cccc4 12P-369S Cc1ccc(cc1)C(=O)NNC(=O)c2cnn(c2n3cccc3)c4ccccc4 12P-370S Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cnn(c2n3cccc3)c4ccccc4 12P-371S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCCC3 12P-381S c1cc(c(c(c1)Cl)CSc2nnc(n2N)c3cccs3)Cl 12P-382S c1cc(sc1)c2nnc(n2N)SCc3ccc(cc3Cl)Cl 12P-383S c1cc(cc(c1)[N+](=O)[O-])CSc2nnc(n2N)c3cccs3 12P-384S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)C(=O)c4ccc(cc4)F 12P-389S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4Cl)Cl 12P-390S CC(C)(C)c1ccc(cc1)CSc2nnc(n2N)c3cccs3 12P-391S c1ccc(cc1)CSc2nnc(n2N)c3cccs3 12P-393S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)C(=O)c4cccs4 12P-394S Cc1ccc(cc1)C(=O)N2CCN(CC2)c3cc(=O)[nH]nc3c4ccccc4 12P-395S c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)C(=O)c4cccc(c4)C(F)(F)F 12P-402S c1ccc(cc1)c2c(snn2)C(=O)N3CCN(CC3)c4ccccc4F 12P-501S CNC(=O)c1c(nns1)c2ccccc2 12P-502S c1ccc(cc1)c2c(snn2)C(=O)N3CCCCC3 12P-503S COc1cnc(nc1N2CCOCC2)c3ccccc3 12P-504S COc1cnc(nc1N2CCCC2)c3ccccc3 12P-505S COc1cnc(nc1N2CCCCC2)c3ccccc3 12P-506S CNc1c(cnc(n1)c2ccccc2)OC 12P-507S COC(=O)c1c(ccs1)n2cccc2C(=O)C(Cl)(Cl)Cl 12P-511S COC(=O)c1c(ccs1)n2cccc2C(=O)N3CCOCC3 12P-512S COC(=O)c1c(ccs1)n2cccc2C(=O)NCc3ccccc3 12P-513S CC1CN(CC(O1)C)c2c(cnc(n2)c3ccccc3)OC 12P-514S COC(=O)c1c(ccs1)n2cccc2C(=O)NCC=C 12P-515S COc1cnc(nc1NCC=C)c2ccccc2 12P-518S COc1cnc(nc1N2CCN(CC2)C(c3ccccc3)c4ccccc4)c5ccccc5 12P-519S COc1cnc(nc1N2CCN(CC2)c3ccccc3F)c4ccccc4 12P-520S CNC(=O)c1cccn1c2ccsc2C(=O)OC 12P-521S CC(C)(C)OC(=O)N1CCC(CC1)Nc2ccc(cc2)OC 12P-542S c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)OC5=O 12P-545S CNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 12P-547S CC(C)NC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 12P-549S c1cc(c(cc1OCC(F)(F)F)C(=O)NC2CC2)OCC(F)(F)F 12P-550S C=CCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 12P-551S Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 12P-552S c1cc(c(cc1OCC(F)(F)F)C(=O)N/N=C\c2ccc(cc2Cl)Cl)OCC(F)(F)F 12P-553S CCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 12P-555S c1cc(c(cc1OCC(F)(F)F)C(=O)NC2CCCCC2)OCC(F)(F)F 12P-556S c1cc(ccc1F)S(=O)(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 12P-557S c1cc(ccc1S(=O)(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 12P-558S c1cc(ccc1S(=O)(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Br 12P-559S c1cc(c(cc1OCC(F)(F)F)C(=O)NNS(=O)(=O)c2ccc(cc2Cl)Cl)OCC(F)(F)F 12P-560S CS(=O)(=O)NNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 12P-562S CCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 12P-563S c1cc(ccc1/C=N\NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)F 12P-564S COc1ccc(cc1)/C=N\NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 12P-565S COc1cccc(c1)/C=N\NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 12P-566S c1ccc(cc1)Oc2ccc(cc2)/C=N\NC(=O)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F 12P-567S c1cc(sc1)/C=N\NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 12P-568S c1cc(ccc1/C=N\NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 12P-569S Cc1ccc(cc1)/C=N\NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 12P-570S CC(C)(C)OC(=O)N1CCC(CC1)Nc2cccc(c2)C(F)(F)F 12P-571S CC(C)(C)OC(=O)N1CCC(CC1)Nc2ccc(cc2Cl)Cl 12P-572S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)O/N=C(/c3ccccn3)\N 12P-578S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)O/N=C(/c3ccncc3)\N 12P-579S COc1cnc(nc1Sc2ccc(cc2)Br)c3ccccc3 12P-581S c1ccc(cc1)c2nnc(o2)c3ccccc3 12P-583S Cc1ccc(cc1)c2nnc(o2)c3ccc(cc3)C 12P-584S Cc1ccccc1c2nnc(o2)c3ccccc3C 12P-585S c1cc(cc(c1)F)c2nnc(o2)c3cccc(c3)F 12P-587S COc1cnc(nc1Sc2ccccc2Cl)c3ccccc3 12P-588S COc1cnc(nc1Oc2ccc(cc2)Cl)c3ccccc3 12P-590S Cc1ccc(cc1)Sc2c(cnc(n2)c3ccccc3)OC 12P-591S COC(=O)C(Cc1ccc(cc1)O)N2Cc3ccccc3C2=O 12P-600 c1ccc(c(c1)/C=C/2\CSc3ccc(cc3C2=O)Cl)F 12P-602 c1ccc(c(c1)C2CC23COc4ccccc4C3=O)F 12P-603 c1ccc2c(c1)C(/C(=C/c3ccc(c(c3)Cl)Cl)/CO2)O 12P-608 c1ccc(cc1)SCCCC(=O)O 12P-609 c1ccc(c(c1)CN2CCS(=O)(=O)CC2)Cl 12P-610 c1cc(ccc1CN2CCS(=O)(=O)CC2)Cl 12P-611 c1cc(cc(c1)Cl)CN2CCS(=O)(=O)CC2 12P-612 C1CCC(C1)CN2CCS(=O)(=O)CC2 12P-613 c1ccnc(c1)CN2CCS(=O)(=O)CC2 12P-614 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)[N+](=O)[O-])C 12P-615 CC(c1cc2cccc(c2o1)OC)O 12P-617 c1cc(ccc1CN2CCS(=O)(=O)CC2)OC(F)(F)F 12P-621 CC(CO)N1CCS(=O)(=O)CC1 12P-622 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)[N+](=O)[O-])/CO2 12P-624 c1cc2c(cc1[N+](=O)[O-])nccn2 12P-625 c1ccc(c(c1)c2nnc(n2N)c3ccccc3N)N 12P-626 c1ccc(c(c1)CN2CCS(=O)(=O)CC2)C(F)(F)F 12P-628 c1ccc2c(c1)C(/C(=C/c3ccc(cc3)[N+](=O)[O-])/CO2)O 12P-630 CN(C)/C=C/1\COc2ccccc2C1=O 12P-631 c1cc(ccc1CNCC(C(F)(F)F)O)OC(F)(F)F 12P-633 Cn1cnc2c1cc(cc2)[N+](=O)[O-] 12P-635 C1COCCN1CCNCC(C(F)(F)F)O 12P-637 c1ccc2c(c1)C(=O)CCCS2 12P-638 COc1cc(cc2c1oc(c2)C(=O)c3ccc(cc3)Br)Br 12P-639 CN(C)CCn1c2ccc(cc2cn1)NC(=S)N 12P-640 c1ccc(cc1)/C=C/2\COc3ccccc3C2O 12P-641 c1cnc(cn1)c2nnc(n2N)c3cnccn3 12P-644 c1ccc2c(c1)C(=O)/C(=C/c3cccs3)/CCS2 12P-648 c1cc(ncc1C#N)N 12P-651 CN(C)/C=C/1\CCSc2ccccc2C1=O 12P-652 c1ccc2c(c1)C(=O)/C(=C/c3cccs3)/CO2 12P-653 c1ccc(cc1)CC(CO)N2Cc3ccccc3C2=O 12P-654 c1ccc2c(c1)C(CCCS2)O 12P-655 c1ccc(cc1)/C=C/2\COc3ccccc3C2OCS(=O)(=O)c4ccc(cc4)Cl 12P-656 c1ccc(cc1)CN(Cc2cccs2)CC(C(F)(F)F)O 12P-658 CC(=O)c1[nH]c2ccccc2n1 12P-660 c1cc(sc1)c2nnc(n2N)c3cccs3 12P-661 c1cc(c(nc1)NN)C(F)(F)F 12P-663 CN1CCN(CC1)C(=O)CC#N 12P-665 Cc1cccc(n1)n2cc(nc2)C(=O)NCc3ccc(cc3)F 12P-800 Cc1ccc(cc1)NC(=O)c2cn(cn2)c3cccc(n3)C 12P-801 COC(=O)C1CC(=O)N(C1)CCc2c[nH]c3c2cccc3 12P-802 CN1CCN(CC1)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 12P-803 c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)CC(=O)N)Oc3c(cc(cn3)C(F)(F)F)Cl 12P-805 COC(=O)Cc1c(ccn(c1=O)Cc2cccc(c2)C(F)(F)F)O 12P-806 Cc1ccc(o1)Cn2ccc(c(c2=O)CC(=O)OC)O 12P-807 COC(=O)Cc1c(ccn(c1=O)CC(F)(F)F)O 12P-808 COC(=O)Cc1c(ccn(c1=O)CCc2ccc(cc2)S(=O)(=O)N)O 12P-810 Cc1ccc(cc1Cl)S(=O)(=O)N2c3ccccc3-c4ccccc4S2(=O)=O 12P-811 Cc1c(sc(n1)c2ccccn2)c3ccnn3c4ccc(cc4)Cl 12P-812 Cc1c(sc(n1)c2ccccn2)c3ccnn3c4ccc(cc4)F 12P-813 Cc1cccc(n1)n2cc(nc2)C(=O)N3CCN(CC3)c4ccccc4 12P-815 CCCCCCCNC(=O)c1cn(cn1)c2cccc(n2)C 12P-816 Cc1cccc(n1)n2cc(nc2)C(=O)NC3CCCCCC3 12P-817 COC(=O)Cc1c(ccn(c1=O)Cc2ccc3c(c2)OCO3)O 12P-818 Cc1cccc(n1)n2cc(nc2)C(=O)NNC(=O)NC3CCCCC3 12P-819 Cc1cccc(n1)n2cc(nc2)C(=O)NNC(=S)Nc3ccc(cc3)Cl 12P-820 Cc1c(sc(n1)c2ccccn2)c3ccnn3c4ccccc4 12P-821 COC(=O)Cc1c(ccn(c1=O)C2CC2)O 12P-822 Cc1c(sc(n1)c2ccccc2)C(=O)C3C(C3(C#N)C#N)c4ccccc4[N+](=O)[O-] 12P-831 CN1C(C(NC1=S)O)O 12R-0001 CC1(OC2COC(C2O1)C3CO3)C 12R-0004 c1ccc(cc1)CC2CC3(CCNCC3)OC2.Cl 12R-0005 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)N)C)C 12R-0011 Cc1cc2ncc(c(n2n1)N)c3ccc(cc3)Cl 12R-0012 Cc1cc2ncc(c(n2n1)C)C(=O)Nc3ccsc3C(=O)Nc4ccc(cc4)F 12R-0013 CCO/C=C(/C(=O)CCl)\C(=O)OCC 12R-0015 COc1ccc(cc1OCc2ccccc2)CO 12R-0016 Cc1cc([nH]n1)N/C=C(\C#N)/C(=O)OC 12R-0017 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)c5ccc(cc5)Cl)C 12R-0019 Cc1cc2ncc(c(n2n1)N)C(=O)OC 12R-0020 COc1ccc2cc(c(nc2c1)Cl)C=O 12R-0028 CCOC=C(C#N)C#N 12R-0029 c1ccc(cc1)CN(Cc2ccccc2)/C=C/C3=C(C(=O)c4ccccc4C3=O)Cl 12R-0201 Cc1ccc(cc1)c2c3cc(ccc3no2)C4(OCCO4)C 12R-0202 COc1cccc(c1)c2cn3ccsc3n2 12R-0203 CN(C)/C=C/C(=O)c1ccc2c(c1)c(on2)c3ccc(cc3)OC 12R-0204 CC1(CN2C(=O)c3ccccc3C2(S1)C)C 12R-0205 c1ccc2c(c1)C(=O)C(=Cc3ccc4c(c3)OCO4)C2=O 12R-0206 C(=O)c1c(nc(nc1Cl)N)Cl 12R-0210 Cc1ccc(cc1)c2cn3c(n2)ccc4c3nc(cc4C(F)(F)F)C(F)(F)F 12R-0211 c1cc(ccc1c2c(n3ccsc3n2)C=O)F 12R-0213 Cc1ccc(cc1)c2c3cc(ccc3no2)C(=O)C 12R-0214 c1cc(c(c(c1)F)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])F 12R-0216 CC(=O)/C=C/c1c(nc2n1ccs2)c3ccc(cc3)F 12R-0217 c1c[nH]c2c(c1=O)c(ncn2)N 12R-0218 CC1(OCCO1)c2ccc3c(c2)c(on3)c4cccc(c4)OC 12R-0219 COc1cccc(c1)c2c(n3ccsc3n2)C=O 12R-0221 CCCCCCCCCCCCSc1nc2cc(c(cc2c(=N)n1Cc3cccc(c3)C(F)(F)F)OC)OC 12R-0222 c1cc([nH]c1)C(c2ccc(cc2)C(=O)O)c3ccc[nH]3 12R-0223 Cc1cccc(c1)c2c3cc(ccc3no2)C4(OCCO4)C 12R-0226 CN1CCN(CC1)c2ccc(c(c2)N)[N+](=O)[O-] 12R-0229 Cc1ccc(cc1)c2c3cc(ccc3no2)C(=O)/C=C/N(C)C 12R-0230 CC(=O)c1ccc2c(c1)c(on2)c3cccc(c3)OC 12R-0235 CC(C)CSc1nc2cc(c(cc2c(=N)n1CCCn3ccnc3)OC)OC 12R-0236 c1cc(ccc1c2cn3ccsc3n2)[N+](=O)[O-] 12R-0238 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])C\2CCCC/C2=N\OC(=O)C3CCCC3 12R-0239 CN(C)/C=C/C(=O)c1ccc2c(c1)c(on2)c3cccc(c3)OC 12R-0240 Cc1cccc(c1)c2c3cc(ccc3no2)C(=O)C 12R-0241 CC1(CN2C(S1)c3ccccc3C2=O)C 12R-0242 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])C\2CCCC/C2=N\OC(=O)C3CCCCC3 12R-0243 Cc1cc(n2cc(nc2n1)c3ccccc3)O 12R-0246 Cc1ccc(cc1)c2c3cc(ccc3no2)c4ccnc(n4)N 12R-0248 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2C4CCCC4)C(=O)O 12R-0249 CCOC(=O)C1CSC2N1C(=O)c3c2cccc3 12R-0250 COc1cccc(c1)c2c(n3ccsc3n2)/C=C/c4ccn[nH]4 12R-0255 c1ccc2c(c1)C(C(N(C2=O)C3CCCC3)c4ccc(cc4)[N+](=O)[O-])C(=O)O 12R-0257 CC1=C(C(C2=C(N1)c3ccccc3C2=O)c4ccc5c(c4)OCO5)C#N 12R-0261 c1ccc(c(c1)c2cn3ccsc3n2)F 12R-0262 c1cc(oc1)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 12R-0263 COC(=O)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C=O 12R-0265 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 12R-0266 COc1cccc(c1)c2c3cc(ccc3no2)C(=O)/C=C/Nc4cc(cc(c4)OC)OC 12R-0268 Cc1ccc(cc1N/C=C/C(=O)c2ccc3c(c2)c(on3)c4cccc(c4)OC)F 12R-0269 Cc1cccc(c1)c2c3cc(ccc3no2)C(=O)/C=C/N(C)C 12R-0270 c1ccc2c(c1)C3=C(C2=O)C(NC(=S)N3)c4ccc5c(c4)OCO5 12R-0271 Cc1cccc(c1)c2c3cc(ccc3no2)C(=O)/C=C/Nc4cc(ccc4OC)OC 12R-0273 Cc1ccc(cc1)c2[nH]c(=O)c3cc(ccc3n2)N4CCOCC4 12R-0274 Cc1ccc(cc1)c2c(n3ccsc3n2)C=O 12R-0276 Cc1ccc(cc1)/C=C/C(=O)c2ccc3c(c2)c(on3)c4cccc(c4)OC 12R-0280 CN(C)C=C1C(=O)c2ccccc2C1=O 12R-0281 Cc1ccc(cc1)c2c3cc(ccc3no2)C(=O)/C=C/Nc4cc(c(c(c4)OC)OC)OC 12R-0282 c1ccc2c(c1)C3=C(C2=O)C(N=C(N3)SCc4cccc(c4)F)c5ccc6c(c5)OCO6 12R-0285 CCCSc1nc2cc(c(cc2c(=N)n1CCCN3CCOCC3)OC)OC 12R-0288 c1cc(ccc1c2[nH]c(=O)c3cc(ccc3n2)N4CCOCC4)F 12R-0289 c1ccc(c(c1)C=C2C(=O)c3ccccc3C2=O)F 12R-0291 Cc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O 12R-0292 COc1ccc(cc1OC)c2[nH]c(=O)c3cc(ccc3n2)N4CCCC4 12R-0293 c1ccc2c(c1)C(C(N(C2=O)C3CCCC3)c4ccc(cc4Cl)Cl)C(=O)O 12R-0294 c1ccc(cc1)C2C(c3ccccc3C(=O)N2C4CCCCC4)C(=O)O 12R-0295 CC(=O)OC(c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)C(=O)OC)OC(=O)C 12R-0296 CC1(OCCO1)c2ccc3c(c2)c(on3)c4cccc(c4)F 12R-0298 Cc1ccc(cc1)c2[nH]c(=O)c3cc(ccc3n2)N4CCCC4 12R-0299 c1cc2c(cc1N3CCCC3)c(=O)[nH]c(n2)C4CCCCC4 12R-0300 CC1(OCCO1)c2ccc3c(c2)c(c4ccccc4n3=O)C#N 12R-0301 C/C(=C\C(=O)c1ccc2c(c1)c(on2)c3ccc(cc3)F)/N(C)C 12R-0302 CC(=O)c1ccc2c(c1)c(on2)c3cccc(c3)F 12R-0304 c1cc(ccc1c2[nH]c(=O)c3cc(ccc3n2)N4CCCC4)Cl 12R-0305 Cc1ccc(cc1)C2C(=C(NC3=C2C(=O)c4c3cccc4)C)C#N 12R-0307 Cc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=S)N2 12R-0309 c1cc(ccc1C/N=C/c2ccn(c2)c3ccc(cc3)Br)F 12R-0600 Cn1ccc(c1)C=O 12R-0601 c1cc(ccc1n2ccc(c2)/C=N/c3ccc(c(c3)Cl)Cl)Br 12R-0602 COC(=O)CC(c1cccc2c1cccc2)N 12R-0603 c1ccn(c1)c2ccc3c(c2)OCO3 12R-0604 c1cc(c(nc1)N2CCOCC2)N 12R-0605 c1cc(ccc1n2ccc(c2)C(CC(=O)O)N)Br 12R-0606 COc1ccc(cc1OC)C(CC(=O)O)NC(=O)C(F)(F)F 12R-0607 COc1cc2c(cc1OC)C(=O)CC2NC(=O)C(F)(F)F 12R-0608 Cc1cccc(c1)C(CC(=O)O)NC(=O)C(F)(F)F 12R-0609 c1cc(ccc1n2ccc(c2)C=C(C(=O)O)C(=O)O)Br 12R-0610 CC(=O)O/N=C/c1ccn(c1)c2ccc(cc2)Br 12R-0611 CC(C)c1ccc(cc1)C(CC(=O)OC)NC(=O)Nc2ccc(cc2Cl)Cl 12R-0612 CN(C)/C=C(\C#N)/C(=O)Nc1cccc(c1)OC 12R-0613 c1cc(n(c1)c2nccs2)/C=N\O 12R-0614 Cc1ccc(o1)/C=C/C(=O)c2ccc(cc2)n3cccc3 12R-0615 CN(C)/C=C/C(=O)c1ccc(cc1)n2cccc2 12R-0616 CC(=O)c1ccc(cc1)n2cccc2C=O 12R-0617 CCOc1ccccc1/C=C/C(=O)c2ccc(cc2)n3cccc3 12R-0618 COc1ccc(cc1OC)/C=C/C(=O)c2ccc(cc2)n3cccc3 12R-0619 COC(=O)c1cccn1c2ccc(cc2)Br 12R-0620 c1ccn(c1)c2ccc(cc2)c3cc[nH]n3 12R-0621 c1ccn(c1)c2ccc(cc2)c3ccnc(n3)N 12R-0622 COc1cc2c(cc1OC)C(=O)CC2[NH3+].[Cl-] 12R-0623 Cc1cc(c(cc1Cl)NC(=O)C)N 12R-0624 Cc1cc(c(cc1Oc2cccc(c2)Cl)NC(=O)C)[N+](=O)[O-] 12R-0625 c1cc(n(c1)c2ccc3c(c2)OCO3)C(=O)C(Cl)(Cl)Cl 12R-0626 c1cc(n(c1)c2ccc3c(c2)OCO3)C=O 12R-0627 c1cc(n(c1)c2ncc(cn2)Br)C=O 12R-0628 c1cc(cc(c1)C(F)(F)F)C/N=C/c2cccn2c3nccs3 12R-0630 c1ccc2c(c1)cccc2C(CC(=O)O)NC(=O)C(F)(F)F 12R-0631 CC(=O)c1ccc(cc1)n2cccc2C=C(C#N)C#N 12R-0634 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)C(=O)C(Cl)(Cl)Cl 12R-0635 Cc1cc(c(cc1OC(=O)c2ccccc2F)C(C)C)Br 12R-0636 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)O 12R-0800 c1cc(ccc1CC(=O)c2cc([nH]c2)C(=O)O)Cl 12R-0802 c1cc(ccc1C(=O)NCCN2CCN(CC2)C(=O)c3ccc(cc3)Br)Br 12R-0809 COc1ccc(cc1OC)CCNC(=O)Cn2cncn2 12R-0810 c1cc(oc1)CNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 12R-0811 CC1=C(/C(=C/Nc2cc(c(c(c2)OC)OC)OC)/C(=O)N1CCc3ccccc3)C(=O)OC 12R-0812 CN(C)/C=C/C(=O)c1cnc(s1)c2ccccn2 12R-0813 c1ccc(cc1)c2c(c(oc2c3ccccc3)N)C#N 12R-0814 c1cc(cc(c1)C(F)(F)F)C(=O)NCC[NH+]2CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F.[Cl-] 12R-0816 COC(=O)c1coc(=O)c2c1cccc2 12R-0817 CC(C)(C)c1ccc(cc1)C(=O)NCC[NH+]2CCN(CC2)C(=O)c3ccc(cc3)C(C)(C)C.[Cl-] 12R-0819 COc1cc(cc(c1OC)OC)C(=O)NCCN2CCN(CC2)C(=O)c3cc(c(c(c3)OC)OC)OC 12R-0820 c1ccnc(c1)c2ncc(s2)c3ccnc(n3)N 12R-0822 c1c(cnc(c1Cl)CC(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 12R-0823 c1ccnc(c1)c2ncc(s2)c3ccn[nH]3 12R-0826 c1cc(oc1)c2c(c(oc2c3ccco3)N)C#N 12R-0827 Cc1c(oc(c1C#N)/N=C/c2ccc3c(c2)OCO3)C 12R-0830 Cc1c(c(n2c(n1)nc(n2)SC)O)C/C=C/c3ccccc3 12R-0840 c1ccc(cc1)n2c(c(cn2)C(=O)N3CCN(CC3)c4ccccc4)C(F)(F)F 12R-1120 CC(C)NC(=O)c1cnn(c1C(F)(F)F)c2ccccc2 12R-1121 C=CCNC(=O)c1cnn(c1C(F)(F)F)c2ccccc2 12R-1122 c1cc(ccc1NC(=O)C(F)(F)F)I 12R-1129 c1ccc(cc1)n2c(c(cn2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F 12R-1133 COc1ccc(cc1)NC(=O)c2cnn(c2C(F)(F)F)c3ccccc3 12R-1134 CO/N=C\c1cc(ccc1N2CCCCC2)[N+](=O)[O-] 12R-1136 COc1cccc(c1)Sc2ccc(cc2[N+](=O)[O-])/C=N\OC 12R-1138 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2N 12R-1139 COC(=O)c1ccccc1Sc2ccc(cc2[N+](=O)[O-])/C=N\OC 12R-1140 CO/N=C\c1ccc(c(c1)[N+](=O)[O-])Sc2c(cccc2Cl)Cl 12R-1141 CO/N=C/c1cc(ccc1Sc2ccc(cc2)Cl)[N+](=O)[O-] 12R-1144 CO/N=C/c1cc(ccc1Sc2c(cccc2Cl)Cl)[N+](=O)[O-] 12R-1145 CO/N=C/c1cc(ccc1Sc2cccc(c2Cl)Cl)[N+](=O)[O-] 12R-1146 Cc1ccc(cc1)Sc2ccc(cc2/C=N/OC)[N+](=O)[O-] 12R-1147 COC(=O)c1ccccc1Sc2ccc(cc2/C=N/OC)[N+](=O)[O-] 12R-1148 COc1cccc(c1)Sc2ccc(cc2/C=N/OC)[N+](=O)[O-] 12R-1152 CC(C)(C#Cc1ccc(cc1)NC(=O)C(F)(F)F)O 12R-1153 Cc1ccccc1C(=O)Nc2ccc(nc2)N3CCN(CC3)C 12R-1181 CN1CCN(CC1)c2ccc(cn2)NC(=O)c3ccc(cc3)C(F)(F)F 12R-1182 c1cc(ccc1C(=O)Nc2ccc(nc2)N3CCOCC3)F 12R-1184 Cc1ccccc1C(=O)Nc2ccc(nc2)N3CCOCC3 12R-1185 c1cc(sc1)C(=O)Nc2ccc(nc2)N3CCOCC3 12R-1186 c1cc(ccc1C(=O)Nc2ccc(nc2)N3CCOCC3)C(F)(F)F 12R-1187 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)N3CCN(CC3)C 12R-1189 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)N3CCOCC3 12R-1192 c1c2c(nc(c1C#N)Cl)CCCC2 12R-1240 COc1ccc(cc1)CSc2nc3c(c4ccccc4[nH]3)nn2 12R-1241 Cc1ccc(cc1)Sc2c(cc3c(n2)CCCC3)C#N 12R-1243 COC(=O)C(c1ccccc1[N+](=O)[O-])C(=O)OC 12T-0006 COC(=O)C(c1ccc(cc1)[N+](=O)[O-])(C(=O)OC)Br 12T-0012 COC(=O)C(CC=C)(c1ccc(cc1)[N+](=O)[O-])C(=O)OC 12T-0017 Cc1ccc(cc1)CC(c2ccc(cc2)[N+](=O)[O-])(C(=O)OC)C(=O)OC 12T-0020 COC(=O)C(CC=C)(c1ccc(cn1)[N+](=O)[O-])C(=O)OC 12T-0021 COC(=O)C(c1ccc(cn1)NC(=O)/C=C/C(=O)O)C(=O)OC 12T-0023 CCOC(=O)CSc1c(c(c(s1)C(=O)OCC)C)C(=O)OCC 12T-0027 c1cc(ccc1C(Cc2cnc(s2)O)C(=O)O)[N+](=O)[O-] 12T-0029 COC(=O)C(CC=C)(c1ccccc1[N+](=O)[O-])C(=O)OC 12T-0030 CC(c1ccccc1[N+](=O)[O-])(C(=O)OC)C(=O)OC 12T-0031 COC(=O)C(Cc1cnc(s1)Cl)(c2ccccc2[N+](=O)[O-])C(=O)OC 12T-0032 Cc1c(c(c2cccc(c2n1)OC)Cl)CCCl 12T-0200 Cc1nn(c(=O)n1c2cccc(c2)F)Cc3ccc(cc3)[N+](=O)[O-] 12T-0201 Cc1n[nH]c(=O)n1c2cccc(c2)OC 12T-0202 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)Cc3ccc(cc3)Cl 12T-0203 CN(C)/C=C/C(=O)/C=C/c1cccc(c1)OC 12T-0204 c1cc2c(cc1Cl)NC(=O)C(O2)CCO 12T-0207 c1cc2c(cc1[N+](=O)[O-])OC(C(=O)N2)CCO 12T-0208 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)Cc3ccc(cc3)[N+](=O)[O-] 12T-0210 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)C 12T-0211 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)Cc3ccc(cc3)OC 12T-0218 Cc1nn(c(=O)n1c2cccc(c2)F)C 12T-0219 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)CC#N 12T-0220 c1ccc(cc1)OC(=O)Nc2ccccc2F 12T-0221 Cc1c(c[nH]n1)c2ccccc2 12T-0222 c1cc(ccc1C(=O)OCCC2C(=O)Nc3ccc(cc3O2)[N+](=O)[O-])I 12T-0223 c1ccc(c(c1)NC(=O)NN)F 12T-0224 Cc1n[nH]c(=O)n1c2cccc(c2)Cl 12T-0225 Cc1nn(c(=O)n1c2cccc(c2)F)CC#N 12T-0226 Cc1nn(c(=O)n1c2cccc(c2)F)c3c(cc(cn3)C(F)(F)F)Cl 12T-0227 Cc1nn(c(=O)n1c2cccc(c2)OC)Cc3ccc(cc3)Cl 12T-0228 Cc1nn(c(=O)n1c2cccc(c2)OC)c3c(cc(cn3)C(F)(F)F)Cl 12T-0229 Cc1nn(c(=O)n1c2cccc(c2)F)CCOc3ccccc3 12T-0230 Cn1c(c(c(n1)c2ccccc2)C(=O)NCC(=O)OC)Cl 12T-0231 COc1cccc(c1)/C(=C/c2cn(nc2c3ccc(cc3)c4ccccc4)c5ccccc5)/C#N 12T-0233 Cc1c2c(n3c(n1)ncn3)N(CC2)CCN4CCCCC4 12T-0235 Cc1nn(c(=O)n1c2cccc(c2)OC)C 12T-0236 Cc1nn(c(=O)n1c2cccc(c2)OC)Cc3ccc(cc3)[N+](=O)[O-] 12T-0237 c1ccc(cc1)c2ccnc(c2C#N)N3CCN(CC3)c4ccc(cc4)F 12T-0241 COc1ccc(cc1)C(c2ccccc2)C(=O)O 12T-0244 COc1cccc(c1)/C=C/c2c(c3cc(ccc3o2)O)C=O 12T-0245 Cc1c2c(n3c(n1)c(cn3)C#N)N(N(CC2)Cc4ccccc4)C 12T-0247 Cn1c(c(c(n1)c2ccccc2)C(=O)NCC(=O)O)Cl 12T-0248 Cc1nn(c(=O)n1c2cccc(c2)F)Cc3cccc(c3)C(F)(F)F 12T-0249 Cc1nn(c(=O)n1c2cccc(c2)F)Cc3ccccc3 12T-0250 CCOC(=O)Cn1c(=O)n(c(n1)C)c2cccc(c2)F 12T-0251 CCOC(=O)Cn1c(=O)n(c(n1)C)c2cccc(c2)OC 12T-0252 Cc1n[nH]c(=O)n1c2ccc(cc2)OCc3ccccc3 12T-0254 Cc1nn(c(=O)n1c2cccc(c2)OC)Cc3ccccc3 12T-0255 CCCCCCCCn1c(=N)c2cc(c(cc2[nH]c1=S)OC)OC 12T-0256 Cc1nn(c(=O)n1c2cccc(c2)Cl)Cc3ccc(cc3)OC 12T-0257 Cc1nn(c(=O)n1c2cccc(c2)Cl)c3c(cc(cn3)C(F)(F)F)Cl 12T-0258 Cc1nn(c(=O)n1c2cccc(c2)Cl)Cc3ccc(cc3)Cl 12T-0259 Cn1c(c(c(n1)c2ccccc2)C(=O)NC(c3ccccc3)C(=O)OC)Cl 12T-0261 CC(C)CSc1nc2cc(c(cc2c(=N)n1C3CCCCCC3)OC)OC 12T-0262 Cc1nn(c(=O)n1c2cccc(c2)Cl)CCOc3ccccc3 12T-0263 Cc1nn(c(=O)n1c2cccc(c2)Cl)Cc3cccc(c3)C(F)(F)F 12T-0265 Cc1c(c(n(n1)C)Cl)NC(=O)OCC(C)(C)C 12T-0266 Cc1nn(c(=O)n1c2cccc(c2)Cl)Cc3ccccc3 12T-0267 Cc1nn(c(=O)n1c2cccc(c2)Cl)C 12T-0269 Cc1nn(c(=O)n1c2cccc(c2)OC)CC#N 12T-0270 Cc1nn(c(=O)n1c2cccc(c2)OC)Cc3cccc(c3)C(F)(F)F 12T-0271 Cc1nn(c(=O)n1c2cccc(c2)OC)CCOc3ccccc3 12T-0272 Cc1nn(c(=O)n1c2cccc(c2)OC)Cc3ccc(cc3)OC 12T-0273 Cc1n[nH]c(=O)n1c2ccccc2F 12T-0274 CCOC(=O)Cn1c(=O)n(c(n1)C)c2cccc(c2)Cl 12T-0276 Cc1nn(c(=O)n1c2cccc(c2)Cl)Cc3ccc(cc3)[N+](=O)[O-] 12T-0277 Cc1nn(c(=O)n1c2cccc(c2)Cl)CC3CC3 12T-0278 Cc1nn(c(=O)n1c2cccc(c2)Cl)CC#N 12T-0279 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3ccccc3F)OC)OC 12T-0280 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)Cc4cccc(c4)C(F)(F)F 12T-0281 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)Cc4ccc(cc4)Cl 12T-0282 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)Cc4ccc(cc4)OC 12T-0283 Cc1nn(c(=O)n1c2ccc(cc2)Cl)CCOc3ccccc3 12T-0284 Cc1nn(c(=O)n1c2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl 12T-0285 Cc1nn(c(=O)n1c2ccc(cc2)Cl)CC#N 12T-0286 Cc1nn(c(=O)n1c2ccc(cc2)Cl)Cc3ccc(cc3)Cl 12T-0287 Cc1nn(c(=O)n1c2ccc(cc2)Cl)Cc3cccc(c3)C(F)(F)F 12T-0288 Cc1nn(c(=O)n1c2ccc(cc2)Cl)Cc3ccc(cc3)[N+](=O)[O-] 12T-0289 Cc1nn(c(=O)n1c2ccc(cc2)Cl)Cc3ccccc3 12T-0290 Cc1nn(c(=O)n1c2ccc(cc2)Cl)Cc3ccc(cc3)OC 12T-0291 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)Cl 12T-0292 Cc1nn(c(=O)n1c2ccc(cc2)Cl)CC3CC3 12T-0293 Cc1nn(c(=O)n1c2ccc(cc2)Cl)C 12T-0294 Cn1c(c(c(n1)c2ccccc2)C(=O)NC(c3ccccc3)C(=O)O)Cl 12T-0295 COc1cccc(c1)/C=C/c2c(c3cc(c4ccccc4c3o2)O)C=O 12T-0296 CCOC(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 12T-0297 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)CCOc4ccccc4 12T-0298 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)Cc4ccc(cc4)[N+](=O)[O-] 12T-0299 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)C 12T-0300 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)c4c(cc(cn4)C(F)(F)F)Cl 12T-0301 Cc1nn(c(=O)n1c2ccccc2F)Cc3ccc(cc3)Cl 12T-0305 Cc1nn(c(=O)n1c2ccccc2F)c3c(cc(cn3)C(F)(F)F)Cl 12T-0306 c1ccc(cc1)Oc2ccc(cc2)NC(=O)Oc3ccccc3 12T-0307 Cc1nn(c(=O)n1c2ccccc2F)CCOc3ccccc3 12T-0308 c1ccc(cc1)Oc2ccc(cc2)NC(=O)NN 12T-0310 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)OCc3ccccc3 12T-0311 Cc1nn(c(=O)n1c2ccccc2F)CC#N 12T-0312 c1cc(cc(c1)OC/C(=N/O)/N)C(F)(F)F 12T-0313 Cc1c2c(c3cc(cc(c3n1)OC)OC)N(CC2)c4ccc(cc4)Oc5ccccc5 12T-0315 Cc1cccc(c1n2c(nn(c2=O)CCOc3ccccc3)C)C 12T-0316 Cc1nn(c(=O)n1c2cccc(c2)OC)CC3CC3 12T-0319 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)CC4CC4 12T-0320 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)CC#N 12T-0321 Cc1nn(c(=O)n1c2ccccc2F)Cc3ccc(cc3)OC 12T-0322 Cc1nn(c(=O)n1c2ccccc2F)Cc3ccccc3 12T-0323 CCOC(=O)/C(=C/NC(c1ccccc1)C(=O)O)/C(=O)C 12T-0325 Cc1nn(c(=O)n1c2ccccc2F)Cc3cccc(c3)C(F)(F)F 12T-0326 CCOC(=O)CCCNC(=O)c1c(nn(c1Cl)C)c2ccccc2 12T-0327 Cc1c(c(n(n1)C)Cl)NC(=O)OCc2ccccc2OC 12T-0328 c1cc(ccc1C2=NN=C(SC2)[NH3+])Cl.[Br-] 12T-0330 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccccc2F 12T-0331 Cc1cc(cc(=O)[nH]1)C(F)(F)F 12T-0332 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)c4c(cc(cn4)C(F)(F)F)Cl 12T-0333 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)CCOc4ccccc4 12T-0334 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)Cc4ccc(cc4)Cl 12T-0335 c1c2c(n3c(n1)c(c(n3)CC#N)C#N)CCCC2=O 12T-0336 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)Cc4ccc(cc4)[N+](=O)[O-] 12T-0337 c1cc(oc1)c2ccnc3n2nc(c3C#N)CC#N 12T-0340 Cc1nc(cn1Cc2c(cccc2Cl)Cl)c3ccc4ccccc4n3 12T-0801 c1ccc2c(c1)ccc(n2)c3ccc4c(c3)OCO4 12T-0802 Cc1ccc(cc1)n2c(nn(c2=O)C)C 12T-0803 Cc1nn(c(=O)n1c2ccc(cc2)F)c3c(cc(cn3)C(F)(F)F)Cl 12T-0804 Cc1nn(c(=O)n1c2ccc(cc2)F)CC3CC3 12T-0805 Cc1nn(c(=O)n1c2ccc(cc2)F)CCOc3ccccc3 12T-0806 Cc1nn(c(=O)n1c2ccc(cc2)F)Cc3ccc(cc3)OC 12T-0807 Cc1nn(c(=O)n1c2ccc(cc2)F)C 12T-0808 c1ccc2cc(ccc2c1)c3ccc4ccccc4n3 12T-0810 Cc1ccc(cc1)n2c(nn(c2=O)CC#N)C 12T-0811 COc1cc(c(cc1C(=O)OC)Br)NC(=O)CCl 12T-0813 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)N 12T-0815 Cc1c2c(nc(n1)n3cc(nn3)C(=O)OC)CCC2 12T-0816 COc1cc(c(cc1C(=O)OC)Br)N(S(=O)(=O)C)S(=O)(=O)C 12T-0817 c1cc(cc(c1)N)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 12T-0818 Cc1n[nH]c(=O)n1c2ccc(cc2)OC 12T-0819 Cc1n[nH]c(=O)n1c2ccccc2 12T-0820 COC(=O)c1cc2ccccc2n1Cc3cccc(c3)C(F)(F)F 12T-0821 Cc1n[nH]c(=O)n1c2ccc(cc2)C(C)C 12T-0822 COc1ccc(cc1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 12T-0824 c1ccc(cc1)NC(=O)Nc2ccc3c(c2)ocn3 12T-0825 C=CCNC(=O)Nc1ccc2c(c1)ocn2 12T-0826 c1cc(ccc1NC(=S)Nc2ccc3c(c2)ocn3)Cl 12T-0828 CCNC(=S)Nc1ccc2c(c1)ocn2 12T-0829 c1ccc(cc1)c2cnc3n(c2=O)CCS3 12T-0832 c1ccc(cc1)CN2CCc3c(cc4ccccc4n3)C2 12T-0833 c1cc(c(c(c1)F)NC(=O)NN)F 12T-0834 Cc1ccc(cc1)n2c(nn(c2=O)Cc3ccc(cc3)[N+](=O)[O-])C 12T-0835 Cc1ccc(o1)c2ccc3ccccc3n2 12T-0836 CCOC(=O)/C(=C/Nc1ccc2c(c1)ocn2)/C#N 12T-0837 Cc1nc(cn1Cc2ccc(cc2)F)C(=O)C 12T-0838 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)n4cccc4 12T-0839 c1ccc(c(c1)c2cc[nH]n2)Cl 12T-0845 c1ccn(c1)c2ccc3c(c2)ocn3 12T-0848 CN1C(=O)C(SC1=O)Cc2ccc(cc2)NS(=O)(=O)C 12T-0849 c1cc(ccc1C(=O)Nn2ccc3c(c2=O)c(cc(n3)C(F)(F)F)C(F)(F)F)Cl 12T-0852 Cc1c2c(nc(n1)n3c(c(nn3)CO)CO)CCC2 12T-0853 Cc1c2c(nc(n1)n3cc(nn3)C(=O)c4ccc5ccccc5c4)CCC2 12T-0854 C#CCN1CCN(CC1)c2cccc(c2)Cl 12T-0855 Cc1c(c(=O)ccn1CCc2c[nH]c3c2cccc3)Cc4c(cccc4Cl)Cl 12T-0856 c1cc2c(cc1NC(=O)/C=C/C(=O)O)ocn2 12T-0860 Cc1nc(cn1Cc2ccc(cc2)F)c3ccc4ccccc4n3 12T-0861 c1ccc2c(c1)ccc(n2)c3ccc(s3)Br 12T-0862 COC(=O)c1ccc(cc1O)NC(=O)/C=C/C(=O)O 12T-0864 Cc1c(nc(s1)c2ccc(cc2)Cl)c3ccccc3 12T-0865 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)Cc3ccccc3 12T-0867 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)C 12T-0868 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)CC#N 12T-0869 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)C(C)C 12T-0870 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)Cc3ccc(cc3)Cl 12T-0871 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)c3c(cc(cn3)C(F)(F)F)Cl 12T-0872 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)CC3CC3 12T-0873 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)Cc3cccc(c3)C(F)(F)F 12T-0874 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)Cc3ccc(cc3)[N+](=O)[O-] 12T-0875 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)CCOc3ccccc3 12T-0876 Cc1nn(c(=O)n1c2ccc(cc2)C(C)C)Cc3ccc(cc3)OC 12T-0877 c1cc(c(cc1N)O)C(=O)NN 12T-0878 Cc1ccc(cc1)/C=N/Nc2ccccc2c3ccccc3 12T-0879 c1ccc(cc1)c2ccccc2n3c(cc(n3)C(F)(F)F)C(F)(F)F 12T-0881 Cc1c(nn(c1C)c2ccccc2c3ccccc3)C 12T-0882 c1ccc(c(c1)NC(=O)NN)Cl 12T-0883 Cc1nc2ccc(cc2o1)[N+](=O)[O-] 12T-0885 CCOC(=O)c1c[nH]c2ccc3cn[nH]c3c2c1=O 12T-0886 c1ccc2c(c1)cc3c(n2)CCCC3 12T-0888 COc1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4cccnc4n3 12T-0889 COc1ccc(cc1)c2c(n3cc(cc(c3n2)Cl)C(F)(F)F)Cl 12T-0890 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)C 12T-0891 Cc1ccc(cc1)n2c(nn(c2=O)CC3CC3)C 12T-0893 c1ccc2c(c1)c3c([nH]2)C4Cc5c(c(cc(n5)C(F)(F)F)C(F)(F)F)C(=O)N4CC3 12T-0894 CCCCc1c(n(nn1)c2nc(c3c(n2)CCC3)C)CCCC 12T-0896 Cc1c(c(n2c(n1)c(cn2)c3cccs3)C)Cc4cccc(c4)C(F)(F)F 12T-0897 c1ccn(c1)c2ncc(cn2)Cl 12T-0898 Cc1nn(c(=O)n1c2ccccc2)Cc3ccccc3 12T-0899 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccccc2 12T-0900 Cc1nn(c(=O)n1c2ccccc2)CC#N 12T-0901 c1ccc2c(c1)ccc(n2)c3ccc(cc3)Br 12T-0902 CC1=NNC(=O)c2ccccc2O1 12T-0903 COc1ccc(c(c1)OC)NC(=O)NN 12T-0905 Cc1c2c(nc(n1)n3cc(nn3)C(=O)c4cccc(c4)N5CC(C5=O)(C)C)CCC2 12T-0916 COC(=O)C(c1ccc(cc1[N+](=O)[O-])S(=O)(=O)N2CCCCC2)C(=O)OC 12W-0002 c1ccc(cc1)CN2c3cccc(c3C(=O)C2=O)I 12W-0005 CCN(Cc1ccccc1)c2c3cnn(c3ncc2C(=O)O)C 12W-0008 c1ccc(cc1)N(c2ccccc2)C(=O)CCl 12W-0018 CCn1c2c(c(n1)C)c(c(cn2)C(=O)OCC)Cl 12W-0020 CCN(c1ccccc1)S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl 12W-0028 CN(c1ccccc1)S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl 12W-0029 c1ccc(cc1)N2c3ccccc3CC2=O 12W-0033 CCn1c2c(c(n1)C)c(c(cn2)C(=O)OCC)NC3CC3 12W-0034 CCn1c2c(c(n1)C)c(c(cn2)C(=O)OCC)NCc3ccc(cc3)OC 12W-0035 CCn1c2c(c(n1)C)c(c(cn2)C(=O)O)NCc3ccc(cc3)OC 12W-0036 CCn1c2c(c(n1)C)c(c(cn2)C(=O)OCC)NCCN3CCOCC3 12W-0037 CCn1c2c(c(n1)C)c(c(cn2)C(=O)OCC)NCc3cccc(c3)C(F)(F)F 12W-0043 CN(c1ccccc1)S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])C(C(=O)OC)C(=O)OC 12W-0044 CCN(c1ccccc1)C(=O)CCl 12W-0045 CCN(c1ccccc1)S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])C(C(=O)OC)C(=O)OC 12W-0048 CCn1c2c(c(n1)C)c(c(cn2)C(=O)OCC)NCc3ccc(cc3)C(F)(F)F 12W-0050 c1ccc(cc1)n2c(nnc2S)Cc3c4ccccc4on3 12W-0200 CC(C)(C)n1cc(cn1)C(=O)c2ccccc2OC(=O)c3cccc(c3)Br 12W-0201 c1cc(cc(c1)C(F)(F)F)Cn2cc(c3c2nccc3)C(=O)C(F)(F)F 12W-0203 c1ccc(cc1)c2ccc(cc2)c3csc(n3)Cc4nc(cs4)O 12W-0204 c1ccc2c(c1)c(no2)Cc3nnc(n3c4ccc(cc4)Cl)S 12W-0206 c1ccc(c(c1)Cn2cc(c3c2nccc3)C(=O)C(F)(F)F)F 12W-0207 CCOC(=O)C1(C(=O)Nc2ccccc2O1)C 12W-0208 CS(=O)(=O)c1ccc(cc1)c2csc(n2)Cc3nc(cs3)O 12W-0209 CCOC(=O)c1ccccc1c2csc(n2)Cc3nc(cs3)O 12W-0210 c1csc(c1Br)c2csc(n2)Cc3nc(cs3)O 12W-0211 CC1(C(=O)Nc2ccccc2O1)C(=O)O 12W-0216 Cc1nc(cs1)CCN2C(=O)c3ccccc3C2=O 12W-0221 COC(CCN1C(=O)c2ccccc2C1=O)(CBr)OC 12W-0222 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)c4cccnc4 12W-0226 CCOC(=O)C1(C(=O)Nc2c(cccn2)O1)C 12W-0227 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OC(=O)c4cccs4 12W-0229 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)Cn4cncn4 12W-0230 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)COc4cccc(c4)C(F)(F)F 12W-0232 c1cc(cc(c1)C(F)(F)F)C(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 12W-0236 CS(=O)(=O)N1CC2CCCN2c3c1cc(cc3)C(F)(F)F 12W-0237 COc1ccc(cc1)S(=O)(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 12W-0238 CC(C)(C)n1c(c(cn1)C(=O)NCc2cccc(c2)OC)C(F)(F)F 12W-0239 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OCc4cccc(c4)C 12W-0240 c1ccc(cc1)c2c(sc(n2)NC(=N)N)CC(=O)O 12W-0243 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)NNc4nc(cs4)CCN5C(=O)c6ccccc6C5=O 12W-0244 COc1cccc(c1)CN2CC3CCCN3c4c2cc(cc4)C(F)(F)F 12W-0245 c1ccc(cc1)CS(=O)(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 12W-0246 CC1(C(=O)Nc2c(cccn2)O1)C(=O)O 12W-0251 c1cc(ccc1F)S(=O)(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 12W-0254 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OC(=O)c4ccco4 12W-0256 CC1(C(=O)Nc2ccccc2O1)C(=O)NCc3cccc(c3)OC 12W-0257 CC1(C(=O)Nc2ccccc2O1)C(=O)NN 12W-0258 Cc1cccc(c1)COc2ccccc2C(=O)c3cnn(c3)c4ccc(cc4)Cl 12W-0262 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OS(=O)(=O)c4ccccc4 12W-0263 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)COc4ccccc4Cl 12W-0264 c1ccc2c(c1)C(=O)N(C2=O)CCc3cnc(s3)CC#N 12W-0265 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)c4ccccn4 12W-0266 c1cc2c(cc1C(F)(F)F)N3CCCC3CN2 12W-0267 c1cc2c(cc1C(F)(F)F)NC(=O)C3N2CSC3 12W-0268 c1ccc(cc1)S(=O)(=O)Oc2ccccc2C(=O)c3cnn(c3)c4ccc(cc4)Cl 12W-0269 c1c(c[nH]c1C=O)C(=O)CCl 12W-0270 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)Nc4nc(cs4)CCN5C(=O)c6ccccc6C5=O 12W-0271 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)c4ccc(cc4)F 12W-0272 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)c4cccc(c4)Cl 12W-0273 Cc1ccc(cc1)c2nc(cs2)CCN3C(=O)c4ccccc4C3=O 12W-0274 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)c4cccc(c4)F 12W-0275 COc1ccc(cc1)S(=O)(=O)N2CC3CCCN3c4c2ccc(c4)C(F)(F)F 12W-0282 COc1cccc(c1)CN2c3cc(ccc3N4CCCC4C2=O)C(F)(F)F 12W-0283 c1cc(cc(c1)F)CN2c3cc(ccc3N4CCCC4C2=O)C(F)(F)F 12W-0284 c1ccc(c(c1)C(=O)c2cnn(c2)c3ccc(cc3)Cl)OCCCF 12W-0288 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)c4nc(cs4)CCN5C(=O)c6ccccc6C5=O 12W-0290 CS(=O)(=O)N1CC2CCCN2c3c1ccc(c3)C(F)(F)F 12W-0293 c1ccc2c(c1)c(=O)c(co2)/C=C(\C#N)/C(=S)N 12W-0294 CCC1(CCCN(C1)C(=O)OC(C)(C)C)C(=O)O 12W-0604 COC(=O)c1cc(cnc1N)Br 12W-0701 c1cc(c(nc1)Cl)/C=N/O 12W-0708 Cc1ccc(cc1)S(=O)(=O)Cc2c(cccc2[N+](=O)[O-])C(=O)OC 12W-0801 COC(=O)c1cccc(c1CS(=O)(=O)c2ccccc2)[N+](=O)[O-] 12W-0802 c1ccc2c(c1)C=Cc3ccccc3N2Cc4ccc(cc4)F 12W-0804 COc1ccc(c2c1cc3c(n2)CCCCC3)OC 12W-0805 COc1ccc(c2c1cc3c(n2)-c4c(c5ccccc5[nH]4)CC3)OC 12W-0806 COc1ccc(cc1Cl)C=O 12W-0807 Cc1cc(nc2n1nc(n2)N)C(F)(F)F 12W-0809 COc1ccc2c(c1)c(c[nH]2)CCNC(=O)Nc3ccc(cc3)Cl 12W-0810 CCCCCCc1c(nc2nc(nn2c1O)N)C 12W-0811 COc1ccc2c(c1)c(c[nH]2)CCNC(=O)Nc3cccc(c3)C(F)(F)F 12W-0813 COc1ccc(c2c1cc3c(n2)CCCC3)OC 12W-0815 COc1ccc(c2c1cc3c(n2)CCCCCC3)OC 12W-0816 COc1ccc(c2c1cc3c(n2)CCC3)OC 12W-0817 c1ccc(c(c1)C#N)OCc2cnc(s2)Cl 12W-0819 Cn1c(cc(=O)n(c1=O)C)N(C)N 12W-0821 Cn1c(cc(=O)n(c1=O)C)N2CCN(CC2)c3ccc(cc3)OC 12W-0822 c1ccc2c(c1)ccc(c2/C=C\3/C(=O)NC(=O)S3)OCc4cnc(s4)Cl 12W-0823 Cn1c(=O)cc(n(c1=O)C)OC 12W-0824 c1ccc2c(c1)OCC(O2)C(=O)O 12W-0825 c1ccc(c(c1)/C(=N\O)/N)OCc2cnc(s2)Cl 12W-0826 c1cc2c(cc1C[NH+]3CC[NH+](CC3)CC#CCOc4ccc5c(c4)OCO5)OCO2.[Cl-].[Cl-] 12W-0827 c1ccc2c(c1)CN(C2=O)C(CO)C(=O)O 12W-0829 CC(C)(C)NC(=O)NCCc1c[nH]c2c1cc(cc2)OC 12W-0831 COc1ccc(c2c1cc3c(n2)-c4c(c5ccccc5n4Cc6ccc(cc6)Br)CC3)OC 12W-0833 Cc1ccc(c2c1c3ccccc3[nH]2)C 12W-0834 COc1ccc(cc1)Cn2c3ccccc3c4c2-c5c(cc6c(ccc(c6n5)OC)OC)CC4 12W-0835 COc1ccc(c2c1cc3c(n2)-c4c(c5ccccc5n4Cc6ccccc6F)CC3)OC 12W-0836 COc1ccc(c2c1cc3c(n2)-c4c(c5ccccc5n4Cc6ccc(cc6)[N+](=O)[O-])CC3)OC 12W-0837 CN1CCN(CC1)Cc2ccc(nc2)Cl 12W-0841 c1cc(ncc1CN2CCOCC2)Cl 12W-0842 c1ccc(cc1)N2CCN(CC2)Cc3ccc(nc3)Cl 12W-0843 c1cnn(c1)Cc2ccc(nc2)Cl 12W-0844 c1cc(ncc1Cn2ccnc2)Cl 12W-0845 c1cc(ncc1CN2CCCCC2)Cl 12W-0846 CCOC(=O)C1CCN(CC1)Cc2ccc(nc2)Cl 12W-0847 CC1CN(CC(O1)C)Cc2ccc(nc2)Cl 12W-0848 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)C(=O)O 12W-0849 c1ccc2c(c1)CN(C2=O)C(Cc3c[nH]c4c3cccc4)C(=O)O 12W-0850 CCOC(=O)c1cc2cc(cc(c2[nH]c1=O)Br)Br 12W-0851 COC(=O)CN1Cc2ccccc2C1=O 12W-0852 Cc1ccc(c2c1c3cc(ccc3[nH]2)[N+](=O)[O-])C 12W-0853 Cc1ccccc1Cn2c3ccccc3c4c2-c5c(cc6c(ccc(c6n5)OC)OC)CC4 12W-0854 COc1ccc(c2c1cc3c(n2)-c4c(c5ccccc5n4Cc6cccc(c6)C(F)(F)F)CC3)OC 12W-0855 Cc1cc(c(c(c1N)[N+](=O)[O-])C)[N+](=O)[O-] 12W-0857 COc1ccc(c2c1ccc(n2)c3ccncc3)OC 12W-0858 COc1ccc(c2c1ccc(n2)c3cccnc3)OC 12W-0859 c1ccc(c(c1)/C(=N/OC(=O)CCCl)/N)OCc2cnc(s2)Cl 12W-0860 c1ccc(cc1)C(=O)O/N=C(/c2ccccc2OCc3cnc(s3)Cl)\N 12W-0862 c1cc2c(cc1C(CCO)N)OCO2 12W-0863 CC(Cc1ccc(cc1)Cl)NC2CC2 12W-0865 CCOC(=O)C(=CNc1cccc(n1)N)C(=O)OCC 12W-0866 c1ccc2c(c1)cccc2CC(=O)NCC[NH3+].[Cl-] 12W-0867 Cc1cc2c(cc1C)NC(=O)CC(N2)C 12W-0869 c1ccc(cc1)CC(c2ccccc2)Nc3ccccn3 12W-0870 COc1cc(c(cc1S(=O)(=O)N)OC)N 12W-0871 CCOC(=O)C(c1ccccc1)Nc2ccc(cc2)SC 12W-0878 Cc1cccc(c1NC(=O)CN)Cl.Cl 12W-0880 CNc1ccc-2c(c1)Cc3c2cccc3.Cl 12W-0881 Cc1cc(nc(n1)Nc2[nH]c3ccccc3n2)C 12W-0882 Cc1nc2ccc(c(c2s1)[N+](=O)[O-])N 12W-0883 c1ccc(cc1)CN2CCC(CC2)Nc3ccccc3 12W-0887 COc1cc(c(c(c1OC)C(=O)O)OC)Br 12W-0890 c1cc(cc(c1)C(=O)Nc2ccc3c(c2)OCO3)CC(=O)O 12W-0891 COc1ccc(cc1)/C=N\c2ccc(cc2)/C=C\C(=O)O 12W-0892 c1cc(ccc1C(=O)NCC(=O)NCC(=O)O)[N+](=O)[O-] 12W-0893 c1c2c(cc(c1N)O)CCCC2 12W-0894 c1ccc(cc1)C(Cc2cc(c(c(c2)I)O)I)C(=O)O 12W-0895 c1cc2c(ccc(c2nc1)O)F 12W-0896 CC(=O)Nc1ccc(cc1)Oc2c(c(ncn2)Cl)[N+](=O)[O-] 12W-0900 COc1ccc-2c(c1)NC(c3n2ccc3)c4cc(cc(c4O)Cl)Cl 12W-0901 COc1ccc(cc1)Nc2[nH]c(nn2)NC(=O)Nc3ccc(cc3)Cl 12W-0902 CCOC(=O)c1cnc(nc1Nc2ccccc2Cl)C(F)(F)F 12W-0903 CC(C)CC(C)c1cc(nc2n1c3ccccc3n2)N 12W-0905 CCOC(=O)c1cnc(nc1N)Sc2c(cccn2)[N+](=O)[O-] 12W-0906 c1cc2c(cc1Cl)nc(s2)SCC(=O)O 12W-0907 CNc1ccc(cc1C(F)(F)F)CSc2ccc(cn2)C(F)(F)F 12W-0909 COc1nc(nc(n1)OC)Nc2cccc(c2)C(F)(F)F 12W-0910 C1CCC(CC1)NCCC#N 12W-0911 c1ccc2c(c1)nnn2CNc3cc(cc(c3)Cl)Cl 12W-0912 c1cc(ccc1CNCC(CSc2ccc(cc2)F)O)F.Cl 12W-0913 c1ccc2c(c1)c(nc3n2nnc3C(=O)N)N 12W-0915 CCCCNc1c(nc2ccccc2n1)Cl 12W-0916 c1cc(sc1)c2ccc(s2)c3ccnc(n3)N 12W-0918 c1ccc2c(c1)c(nc3n2nnc3c4ccc(cc4)[N+](=O)[O-])N 12W-0919 c1ccc(c(c1)NCN2C(=O)CCC2=O)n3cccc3 12W-0920 c1cc(c(c(c1)Cl)/C=C/c2ccnc(n2)N)F 12W-0921 c1cc(sc1)c2c(c(c(o2)N)c3ccc(cc3Cl)Cl)C#N 12W-0922 C=CCNCC(Cn1ccc2c1cccc2)O 12W-0924 Cc1c(c(n(n1)c2cc(ccc2Cl)C(F)(F)F)N)C(=S)N 12W-0925 c1ccc(c(c1)N)Sc2nccc(n2)C(F)(F)F 12W-0926 Cc1ccc(c(c1)[N+](=O)[O-])OCC2NCCS2 12W-0927 Cc1ccc(cc1NCN2C(=O)CNC2=S)Cl 12W-0929 c1cc(ccc1S(=O)(=O)CCNC2CCCCC2)Cl 12W-0933 c1c(c(sc1[N+](=O)[O-])N)[N+](=O)[O-] 12W-0934 c1cc(ccc1c2nnc(s2)N)[N+](=O)[O-] 12W-0935 CC1c2cnc(nc2-c3cc(ccc3S1)Cl)N 12W-0936 Cc1cccnc1NC2c3ccccc3C(=O)O2 12W-0937 c1ccc(c(c1)Nc2ncnc(n2)n3cccc3)Cl 12W-0938 c1cc(ccc1CNCC(Cn2ccc(n2)C(F)(F)F)O)C(F)(F)F 12W-0939 c1cc(ccc1c2cc(nc(n2)N)NS(=O)(=O)c3ccc(cc3)F)F 12W-0940 c1ccc(c(c1)N)SCc2cc(cc3c2OCOC3)[N+](=O)[O-] 12W-0941 Cc1ccc(c(c1)C)Nc2nc3ccccc3s2 12W-0942 COC(=O)/C=C/c1c(nc(s1)SC)N 12W-0944 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)N 12W-0946 Cc1ccc(cc1)CSC2=NCCN2.Cl 12W-0948 Cn1cc(c(n1)N)c2nc3ccccc3s2 12W-0950 CCOC(=O)C(=CNCCNc1c(cccn1)C(F)(F)F)C(=O)OCC 12W-0951 CCCCCNc1c(c(c(s1)Cl)[N+](=O)[O-])[N+](=O)[O-] 12W-0952 CSc1c(c(nc(n1)CSc2ccccc2)N)C#N 12W-0953 CNc1c(c(ncn1)Sc2nccn2C)[N+](=O)[O-] 12W-0959 c1cc2c(cc1Cl)Nc3c(cc(cc3O2)[N+](=O)[O-])[N+](=O)[O-] 12W-0960 Cc1cccc(c1Nc2nnc(s2)C(F)(F)F)C 12W-0963 c1cc(ccc1c2nc(on2)CSc3ncnc(n3)N)OC(F)(F)F 12W-0964 c1cc(ccc1CSc2nnc(s2)N)Cl 12W-0966 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2[nH]nc(n2)N 12W-0967 c1cc(ccc1c2csc(n2)c3cn[nH]c3N)Cl 12W-0969 c1ccc2c(c1)C(=O)NC(N2)c3ccc(c(c3)Cl)Cl 12W-0970 c1c(c(c(c(c1S(=O)(=O)N)Cl)Cl)N)S(=O)(=O)N 12W-0971 Cc1c(c(n(n1)C)Sc2ccccc2N)[N+](=O)[O-] 12W-0972 c1cc(c(cc1S(=O)(=O)N)[N+](=O)[O-])N 12W-0973 Cc1ccc(cc1Cl)Nc2nc(nc(n2)OC)OC 12W-0974 c1ccc2c(c1)c(c[nH]2)SC(=N)N.I 12W-5004 COc1cc(cc(c1O)C=O)O 12W-5015 COc1ccc(cc1OC)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 12X-0201 c1cc(ccc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)Br 12X-0202 COC(=O)c1ccccc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 12X-0203 COc1ccc2c(c1)nc(s2)c3ccc(cc3)N 12X-0205 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)C)C 12X-0206 c1ccc2c(c1)cccc2S(=O)(=O)Oc3c(c(c(c(c3F)F)F)F)F 12X-0207 CC(C)c1cc(c(c(c1)C(C)C)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)C(C)C 12X-0208 c1cc(c(cc1Br)Cl)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 12X-0210 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 12X-0211 CC(C)S(=O)(=O)Oc1c(c(c(c(c1F)F)F)F)F 12X-0217 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)S(=O)(=O)Oc3c(c(c(c(c3F)F)F)F)F 12X-0221 c1cc(cc(c1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)C(=O)O 12X-0230 COc1ccc(cc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)Cl 12X-0235 c1ccc(c(c1)C(=O)c2cnn(c2)c3cc(ccc3Cl)Cl)OS(=O)(=O)Cc4cccc(c4)Cl 12X-0237 c1ccc(cc1)CS(=O)(=O)Oc2ccccc2C(=O)c3cnn(c3)c4cc(ccc4Cl)Cl 12X-0243 c1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OS(=O)(=O)c4cccc5c4nccc5 12X-0248 CC1CCN(CC1)Cc2nc(no2)c3cccc(c3)C(F)(F)F 12X-0250 c1c(cnc(c1Cl)Cl)C(=O)O 12X-0700 CCOC(=O)c1ccc(s1)c2ccc(cc2)OC 12X-0701 CCOC(=O)c1ccc(s1)c2ccc(cc2)C=O 12X-0704 Cc1n[nH]c(=O)n1c2ccc(c(c2)OC)OC 12X-0801 Cc1c(nc2cc(ccc2n1)C(=O)OC)C 12X-0803 COc1ccc(cc1)OCCN 12X-0806 CC1(C(=O)N(C(=O)N1)Cc2ccc(cc2)Cl)C 12X-0807 c1cc(cc(c1)OCc2cnc(s2)Cl)/C(=N/OC(=O)c3cccs3)/N 12X-0808 CC1(C(=O)N(C(=O)N1)Cc2ccc(cc2)F)C 12X-0809 c1cc(sc1C(=O)CBr)Cl 12X-0810 c1cc(ccc1OCc2cnc(s2)Cl)S(=O)(=O)N3CCC(=O)CC3 12X-0811 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1F)F 12X-0812 Cc1c(nc2cc(ccc2n1)C(=O)O)C 12X-0813 Cc1c(nc2cc(ccc2n1)C(=O)NN)C 12X-0814 Cc1c2cc(ccc2[nH]c1C(=O)OC)OC 12X-0815 CC(=O)N1CCC(CC1)C(=O)c2ccc(cc2)Cl 12X-0816 Cc1cc(ccc1O)SC#N 12X-0817 Cc1cc(cc(c1N)Br)C(=O)OC 12X-0818 CS(=O)(=O)/C(=C/c1cn(c2c1cccc2)Cc3cnc(s3)Cl)/C#N 12X-0819 c1ccc2c(c1)c(cn2Cc3cnc(s3)Cl)/C=N/NC(=O)c4ccncc4 12X-0820 Cc1cc(cc(c1N)Br)C(=O)O 12X-0821 Cc1[nH]c(c(n1)C#N)C#N 12X-0823 Cc1c(nc2cc(ccc2n1)C(=O)N/N=C\c3cn(c4c3cccc4)Cc5cnc(s5)Cl)C 12X-0824 CCCCc1nc2ccc(cc2o1)C(=O)OC 12X-0825 CC(C)CC(=O)NNC(=O)c1cn2cc(ccc2n1)I 12X-0826 c1cc(ccc1C(=O)NNC(=O)c2cn3cc(ccc3n2)I)C(F)(F)F 12X-0827 CCCCc1[nH]c(c(n1)C#N)C#N 12X-0829 c1cc(c(cc1F)C(CC(=O)O)N)F 12X-0832 Cc1cn(c(=O)[nH]c1=O)CC(=O)OC 12X-0833 Cc1c(nc2cc(ccc2n1)C(=O)NNC(=O)C3CCN(CC3)C(=O)C)C 12X-0834 Cc1cc(nc(c1C#N)Cl)Cl 12X-0836 c1cc(ccc1C(=O)C2CCNCC2)Cl.Cl 12X-0837 CC(=O)Cc1nc(sn1)Nc2ccccc2 12X-0839 COC(=O)c1ccc(c(c1)F)F 12X-0841 c1ccc(cc1)c2[nH]c(c(n2)C#N)C#N 12X-0842 CCc1[nH]c(c(n1)C#N)C#N 12X-0843 Cc1cc(n[nH]1)C(=O)OC 12X-0844 Cc1cc(nc(n1)n2cc(nn2)c3cccc(c3)N)C(F)(F)F 12X-0852 COc1ccc(cc1OC)C2c3ccc4ccccc4c3OC(=C2C#N)N 12X-0920 c1ccc2c(c1)ccc3c2OC(=C(C3c4ccc(cc4)Br)C#N)N 12X-0921 Cc1ccc(cc1)C2c3ccc4ccccc4c3OC(=C2C#N)N 12X-0922 C1CC(OC1)CNC(=O)CCl 12X-0923 c1cc(cc(c1)C(=O)CBr)C#N 12X-0924 c1cc(oc1)CNC(=O)CCl 12X-0925 CN(C)/C=N/C1=C(C(c2ccc3ccccc3c2O1)c4cccs4)C#N 12X-0926 CN(C)/C=N/C1=C(C(c2ccc3ccccc3c2O1)c4ccc(c(c4)OC)OC)C#N 12X-0927 c1ccc(c(c1)c2c(nc(s2)N)C(=O)O)F 12X-0928 c1ccc(c(c1)c2c(nc(s2)N)C(=O)O)Cl 12X-0929 CCC(CC)c1c(nc(s1)N)C(=O)O 12X-0931 c1cc(oc1)CNS(=O)(=O)c2ccc(cc2)Cl 12X-0933 COc1cc(cc(c1OC)OC)OCC#C 12X-0936 C=CCN(Cc1ccco1)S(=O)(=O)c2ccc(cc2)Cl 12X-0937 c1ccc2c(c1)ccc3c2OC(=C(C3c4cccnc4)C#N)N 12X-0938 c1cc(ccc1c2c(nc(s2)N)C(=O)O)Cl 12X-0939 c1cnc(nc1)NC(=O)CCl 12X-0945 c1cc(ccc1S(=O)(=O)N2CC3CC4C=CC3(C2)O4)Cl 12X-0946 c1c(cnc(c1[N+](=O)[O-])O)Br 12X-0947 CN(C)/C=N/C1=C(C(c2ccc3ccccc3c2O1)c4ccc(cc4)Br)C#N 12X-0950 Cc1ccc(cc1)C2c3ccc4ccccc4c3OC(=C2C#N)/N=C/N(C)C 12X-0952 CC1(CNc2cc(ccc2S1)[N+](=O)[O-])C 12X-0955 COc1ccc(cc1)Oc2c3c(ccs3)nc(n2)c4ccccc4 12Y-0218 Cc1ccc(cc1)COc2ccc(cc2)CCCO 12Y-0700 c1cc(sc1C=O)N2CCCCC2 12Y-0702 c1cc(sc1C=O)N2CCOCC2 12Y-0703 CC(C)(C=O)N1CCCCC1 12Y-0705 Cc1ccc(cc1)COc2ccc(cc2)C(=O)O 12Y-0706 Cc1ccc(n1c2c(ccs2)c3cc([nH]n3)N)C 12Y-0800 Cn1cccc1C(=O)/C(=C/c2ccc(cc2)F)/C#N 12Y-0802 Cn1cccc1C(=O)/C(=C/c2ccccc2C(F)(F)F)/C#N 12Y-0803 Cn1cccc1C(=O)/C(=C/c2cccnc2)/C#N 12Y-0806 Cn1cccc1C(=O)/C(=C/c2ccsc2)/C#N 12Y-0807 Cn1cccc1C(=O)/C(=C/c2ccc(cc2)OC)/C#N 12Y-0808 c1cc(c(cc1Cl)Cl)c2nnc(o2)CCl 12Y-0810 c1cc(ccc1C(=O)NN)I 12Y-0812 CCCCc1nnc(o1)c2ccc(cc2)[N+](=O)[O-] 12Y-0813 CCOC(=O)c1ccc(cc1)N2CCOCC2 12Y-0815 c1cc2nc(cn2cc1Cl)C(=O)NN 12Y-0816 c1ccc2c(c1)nc(o2)CCl 12Y-0817 COc1ccc(c(c1)O)C(=O)NN 12Y-0818 c1cc(c(cc1C(=O)NN)Cl)Cl 12Y-0824 CCCCc1nnc(o1)c2ccc(cc2)N 12Y-0825 c1cc(c(cc1c2nnc(o2)CCl)Cl)Cl 12Y-0828 Cc1c(cccc1[N+](=O)[O-])C(=O)NN 12Y-0829 c1cc(ccc1c2nnc(o2)CCl)I 12Y-0830 CC(C)CC(=O)c1cc(n(c1)C)C(=O)OC 12Y-0831 Cc1c(nc2cc(ccc2n1)c3nnc(o3)CCl)C 12Y-0832 c1cc(ccc1c2nnc(o2)CCl)[N+](=O)[O-] 12Y-0833 Cc1c(c(=O)n([nH]1)C(=S)N)CCO 12Z-0221 CCOC(=O)c1ccc(cn1)C(F)(F)F 12Z-0603 CCOC(=O)c1c(cc(cn1)C(F)(F)F)Cl 12Z-0604 c1cc(ccc1C=O)N2CCOCC2 12Z-0700 c1cc(ccc1C=O)c2ccc(cn2)C#N 12Z-0702 c1cc(ccc1C=O)N2CCCCC2 12Z-0703 c1cc(ccc1C=O)N2CCSCC2 12Z-0704 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)C=O 12Z-0705 c1cc(c(cc1Br)C=O)N2CCCCC2 12Z-0707 c1cc(c(cc1Br)N2CCCCC2)C=O 12Z-0708 COC(=O)c1cnc2c(c(nn2c1N)CC#N)C#N 12Z-0709 CC(=O)c1cc(ccc1N)N2CCC(CC2)O 12Z-0800 Cc1ccc(cc1)CO/N=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 12Z-0806 c1cc(ccc1C(=O)NN)OCc2c(cc(cn2)C(F)(F)F)Cl 12Z-0808 C/C(=C\C(=O)C(F)(F)F)/NC1CCN(CC1)C 12Z-0811 c1cc(cc(c1)N2CCS(=O)(=O)CC2)C(=O)NN 12Z-0814 COc1cccc(c1)CO/N=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl 12Z-0819 COc1cccc(c1)CO/N=C/c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 12Z-0820 COc1cccc(c1)CO/N=C/c2ccc(cc2)c3cc(ccn3)C(F)(F)F 12Z-0821 c1cc(ccc1c2cnco2)N 12Z-0823 CC1CCCN(C1)c2ccc(c(c2)C(=O)C)N 12Z-0825 CC1CCN(CC1)c2ccc(c(c2)C(=O)C)N 12Z-0826 CC(=O)c1cc(ccc1N)N2CCCC2 12Z-0829 CO/N=C/c1ccc(cc1)c2c(cc(cn2)C(F)(F)F)Cl 12Z-0830 CO/N=C/c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 12Z-0831 CO/N=C/c1ccc(cc1)c2cc(ccn2)C(F)(F)F 12Z-0833 c1ccc2c(c1)nc(s2)NN 12Z-0921 c1cc2c(cc1[N+](=O)[O-])nc([nH]2)NN 12Z-0922 c1ccc(c(c1)C(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl)Cl 12Z-5004 c1cc(cc(c1)C(F)(F)F)C(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl 12Z-5005 Cc1ccccc1C(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl 12Z-5006 c1ccc(cc1)C(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl 12Z-5007 c1cc(c(c(c1)F)C(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl)F 12Z-5011 CC(=O)NCCOc1c(cc(cn1)C(F)(F)F)Cl 12Z-5013 c1ccc(c(c1)C(=O)NNc2cc(cc(n2)Cl)C(F)(F)F)Cl 12Z-5014 c1cc(cc(c1)C(F)(F)F)C(=O)NNc2cc(cc(n2)Cl)C(F)(F)F 12Z-5015 Cc1ccccc1C(=O)NNc2cc(cc(n2)Cl)C(F)(F)F 12Z-5016 CCc1cccc(n1)C#N 12Z-5017 c1ccc(c(c1)S(=O)(=O)NNc2cc(cc(n2)Cl)C(F)(F)F)Cl 12Z-5019 c1cc(c(c(c1)F)C(=O)NNc2cc(cc(n2)Cl)C(F)(F)F)F 12Z-5021 Cc1ccccc1S(=O)(=O)NNc2cc(cc(n2)Cl)C(F)(F)F 12Z-5032 Cc1ccccc1S(=O)(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl 12Z-5033 c1cc(c(c(c1)F)S(=O)(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl)F 12Z-5056 CC(C)(C)C(=O)Cc1nc(cs1)O 1B-001 c1cc(cc(c1)Cl)/N=N/N2CCC(=O)N2 1B-002 c1cc(ccc1C(=O)NC(=O)N2CCC(=O)N2)Cl 1B-004 CC(C)(C)C(=O)/C(=C/N(C)C)/c1nc(cs1)O 1B-007 c1cc(ccc1CN2CCC(=O)N2)Cl 1B-008 Cc1ccc(cc1)CN2CCC(=O)N2 1B-009 CC(C)(C)C(=O)/C(=C/c1ccccc1)/c2nc(cs2)O 1B-010 Cn1c(c(c(n1)N)CC(=O)c2ccccc2)N 1B-012 c1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccc(cc2F)O 1B-014 c1ccc(cc1)n2c(nnc2C(F)(F)F)C[N+](=O)[O-] 1B-015 Cc1cccc(c1)/N=N/N2CCC(=O)N2 1B-016 CN(C)/C=C(/c1nncn1c2ccccc2)\[N+](=O)[O-] 1B-017 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(cc1F)O 1B-020 CN/C(=C/[N+](=O)[O-])/SC 1B-021 CN/C(=C/[N+](=O)[O-])/NN 1B-022 Cn1c(nnc1C(F)(F)F)C[N+](=O)[O-] 1B-023 CCOC(=O)c1cc(c(nc1C)O)C(=O)C 1B-025 Cn1c(nnc1C(F)(F)F)/C(=C/N(C)C)/[N+](=O)[O-] 1B-026 CN(C)/C=C/C(=O)c1ccc(cc1)Cl 1B-027 CC(=O)c1ccccc1n2ccnc2 1B-028 c1ccc2c(c1)C(OC2=O)CC(=O)c3ccc(cc3)Cl 1B-035 CN(C)/C=C(\c1ccccc1)/C(=S)N(C)C 1B-041 CN(C)c1c(c[nH]n1)c2ccccc2 1B-048 c1ccc(cc1)n2c(nnn2)N 1B-050 CC(=O)C(=CN(C)C)C(=O)C 1B-052 Cc1c(cnn1c2ccccc2)C(=O)C 1B-053 CN(C)C(=S)Cc1ccc(cc1)Cl 1B-055 Cc1ccc(c(n1)O)c2ccn[nH]2 1B-056 CN(C)c1c(cnc(n1)N)c2ccccc2 1B-058 CS/C(=C\[N+](=O)[O-])/Nc1ccc(cc1)Cl 1B-059 c1ccc2c(c1)/C(=C/Nc3ccccc3N)/OC2=O 1C-001 Cn1ccc2c(c1=O)cccc2[N+](=O)[O-] 1C-003 CCOC(=O)/C=C(\C)/NN/C(=N/C)/C[N+](=O)[O-] 1C-004 c1ccnc(c1)Cn2ccc3c(c2=O)cccc3[N+](=O)[O-] 1C-005 CCS(=O)(=O)c1cc(cc(c1O)I)I 1C-006 CN(C)C(=S)Cc1ccc(cc1)Oc2ccccc2 1C-007 c1cc2c(ccn(c2=O)Cc3ccncc3)c(c1)[N+](=O)[O-] 1C-009 c1ccc2c(c1)C(OC2=O)C[N+](=O)[O-] 1C-013 c1ccn(c(=O)c1)c2cn(nc2c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)C(F)(F)F 1C-015 CN1c2ccccc2S(=O)(=O)N=C1Cl 1C-019 c1ccc2c(c1)c(=O)nc(s2)CC#N 1C-021 CC(=O)Nc1ccc(cc1)S(=O)(=O)N(C)C 1C-025 CC(=O)n1cc(c(n1)c2ccc(cc2)Cl)n3ccccc3=O 1C-026 CN(C)/C=C(\C#N)/c1nc(=O)c2ccccc2s1 1C-029 Cc1c(c(n(n1)C)/C=C/Nc2ccc(cc2)F)[N+](=O)[O-] 1C-030 CN(C)S(=O)(=O)c1ccc(cc1)N 1C-033 COC(Cc1nnc(n1c2ccc(cc2)Cl)SC)OC 1C-034 CN(C)/C=C(/c1ccc(cc1)Oc2ccccc2)\C(=S)N(C)C 1C-035 COC(Cc1nnc(n1c2cccc(c2)C(F)(F)F)SC)OC 1C-036 Cc1c(c(no1)c2ccccc2Cl)C(=O)N 1C-038 Cn1c(nnc1SC)CC(OC)OC 1C-039 COC(Cc1nnc(n1c2ccccc2)SC)OC 1C-041 Cc1c(c(n(n1)C)/C=C/Nc2ccc(cc2OC)OC)[N+](=O)[O-] 1C-043 CC\1=NN(C(=O)/C1=C\N(C)C)c2ccccc2 1C-045 Cc1c(c(no1)c2ccccc2Cl)C#N 1C-047 CC\1=NN(C(=O)/C1=C\Nc2ccc(cc2Cl)Cl)c3ccccc3 1C-048 CC\1=NN(C(=O)/C1=C\Nc2cc(cc(c2)Cl)Cl)c3ccccc3 1C-049 CC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)C(=O)OC)c3ccccc3 1C-050 CC\1=NN(C(=O)/C1=C\NCC(=O)OC)c2ccccc2 1C-051 CN1C(=O)CC(=N1)C(F)(F)F 1C-052 Cc1c(c(n(n1)C)/C=C/Nc2cc(ccc2O)Cl)[N+](=O)[O-] 1C-053 CN1C(=O)/C(=C\N(C)C)/C(=N1)C(F)(F)F 1C-054 Cc1cc(ccc1N/C=C/c2c(nn(c2[N+](=O)[O-])C)C)O 1C-055 CN(C)/C=C/c1c(c(no1)c2ccccc2Cl)C#N 1C-056 CC\1=NN(C(=O)/C1=C\Nc2ccccc2C(F)(F)F)c3ccccc3 1C-057 CC\1=NN(C(=O)/C1=C\Nc2cccc(c2)C(F)(F)F)c3ccccc3 1C-058 Cc1cccc(c1N/C=C\2/C(=NN(C2=O)c3ccccc3)C)C 1C-059 c1ccc2c(c1)/C(=C/NNC(=O)c3ccc(cc3)Cl)/OC2=O 1C-060 CN(C)c1c(c[nH]n1)c2ccc(cc2)Oc3ccccc3 1C-062 CN1C(=O)/C(=C\Nc2cc(cc(c2)Cl)Cl)/C(=N1)C(F)(F)F 1C-063 Cc1ccc(cc1C)N/C=C/c2c(c(no2)c3ccccc3Cl)C#N 1C-064 c1ccc(c(c1)c2c(c(on2)/C=C/Nc3ccc(cc3)Cl)C#N)Cl 1C-065 c1ccc(cc1)N/C=C/c2c(c(no2)c3ccccc3Cl)C#N 1C-066 c1ccc(c(c1)c2c(c(on2)/C=C/Nc3ccc(cc3)C(F)(F)F)C#N)Cl 1C-069 COc1ccc(cc1)N/C=C/c2c(c(no2)c3ccccc3Cl)C#N 1C-070 c1ccc(c(c1)c2c(c(on2)/C=C/Nc3ccc(cc3)C(=O)O)C#N)Cl 1C-072 COc1ccc(c(c1)OC)N/C=C/c2c(c(no2)c3ccccc3Cl)C#N 1C-074 CC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)OC)c3ccccc3 1C-076 Cc1c(c(no1)c2ccccc2Cl)C(=O)OC 1C-077 CC\1=NN(C(=O)/C1=C\Nc2ccccc2C#N)c3ccccc3 1C-079 Cc1ccc(cc1)N/C=C\2/C(=NN(C2=O)c3ccccc3)C 1C-080 c1ccc2c(c1)/C(=C/NNC(=O)c3ccccc3O)/OC2=O 1C-082 COC(=O)NN/C=C\1/c2ccccc2C(=O)O1 1C-083 c1ccc2c(c1)/C(=C/NNC(=S)N)/OC2=O 1C-084 c1ccc2c(c1)/C(=C/NNC(=O)c3ccncc3)/OC2=O 1C-086 C/N=C(\C[N+](=O)[O-])/NN/C=C\1/c2ccccc2C(=O)O1 1C-087 CN(C)/C=C/c1c(c(no1)c2ccccc2Cl)C(=O)OC 1C-088 Cc1cc(nc(n1)NC2=NS(=O)(=O)c3ccccc3[NH+]2C)C.[Cl-] 1C-089 CC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)[N+](=O)[O-])c3ccccc3 1C-092 CC\1=NN(C(=O)/C1=C\Nc2ccccc2OC)c3ccccc3 1C-093 CC\1=NN(C(=O)/C1=C\Nc2ccccc2O)c3ccccc3 1C-094 CC\1=NN(C(=O)/C1=C\Nc2cc(ccc2O)Cl)c3ccccc3 1C-095 CC\1=NN(C(=O)/C1=C\Nc2ccc(cc2OC)OC)c3ccccc3 1C-096 CN1C(=O)/C(=C\Nc2ccccc2O)/C(=N1)C(F)(F)F 1C-097 CN1C(=O)/C(=C\Nc2cc(ccc2O)Cl)/C(=N1)C(F)(F)F 1C-098 CN1C(=O)/C(=C\Nc2ccccc2C#N)/C(=N1)C(F)(F)F 1C-099 CN1C(=O)/C(=C\Nc2ccc(cc2OC)OC)/C(=N1)C(F)(F)F 1C-100 CN1C(=O)/C(=C\Nc2ccc(cc2)Cl)/C(=N1)C(F)(F)F 1C-101 CN1C(=O)/C(=C\Nc2ccc(cc2)[N+](=O)[O-])/C(=N1)C(F)(F)F 1C-102 CSc1cccc(c1)N/C=C/c2c(c(no2)c3ccccc3Cl)C#N 1C-105 CC\1=NN(C(=O)/C1=C\NCc2ccc(cc2)Cl)c3ccccc3 1C-106 c1ccc(cc1)C(=O)NN/C=C\2/c3ccccc3C(=O)O2 1C-107 CN1C(=O)/C(=C\Nc2ccc(cc2)C(=O)OC)/C(=N1)C(F)(F)F 1C-108 CN1C(=O)/C(=C\Nc2ccc(cc2Cl)Cl)/C(=N1)C(F)(F)F 1C-109 CC\1=NN(C(=O)/C1=C\NCc2cccnc2)c3ccccc3 1C-110 CC\1=NN(C(=O)/C1=C\NCc2ccncc2)c3ccccc3 1C-111 CN(C)c1nnnn1c2ccccc2 1C-112 c1ccc(c(c1)c2c(c(on2)/C=C/Nc3ccc(cc3)F)C#N)Cl 1C-114 c1ccc(c(c1)c2c(c(on2)/C=C/Nc3cc(cc(c3)Cl)Cl)C#N)Cl 1C-115 CN1C(=O)/C(=C\NCc2cccnc2)/C(=N1)C(F)(F)F 1C-116 CN1C(=O)/C(=C\NCc2ccc(cc2)Cl)/C(=N1)C(F)(F)F 1C-117 CN(C)c1nnnn1S(=O)(=O)c2cccc(c2)C(F)(F)F 1C-119 CN(C)S(=O)(=O)c1ccc(cc1)NC=C2C(=NNC2=O)C(F)(F)F 1C-120 CN1C(=O)/C(=C\Nc2ccc(cc2)S(=O)(=O)N(C)C)/C(=N1)C(F)(F)F 1C-121 CN(C)S(=O)(=O)c1ccc(cc1)NC=C2C=NNC2=O 1C-122 CN(C)c1nnnn1c2ncccn2 1C-123 c1c(cc(c(c1[N+](=O)[O-])N)[N+](=O)[O-])C(F)(F)F 1C-124 CN(C)S(=O)(=O)c1ccc(cc1)NC=C2C(=NNC2=O)c3ccccc3 1C-125 CN(C)S(=O)(=O)c1ccc(cc1)NC=C2C(=NNC2=O)COC 1C-126 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N 1C-130 c1ccc(c(c1)c2c(c(on2)/C=C/Nc3cccc(c3)Cl)C#N)Cl 1C-136 c1ccc(c(c1)c2c(c(on2)/C=C/Nc3ccccc3Cl)C#N)Cl 1C-137 Cc1c(c(no1)c2c(cccc2Cl)Cl)C#N 1C-138 CN(C)/C=C/c1c(c(no1)c2c(cccc2Cl)Cl)C#N 1C-139 CN1C(=O)/C(=C\NCC(=O)OC)/C(=N1)C(F)(F)F 1C-140 CN(C)c1c(cc(s1)C(=O)OC)c2ccccc2 1D-001 CN(C)C=C1C(=O)CCCC1=O 1D-002 CN(C)/C=C(\C#N)/c1ccccc1 1D-003 CN(C)/C=C/C(=O)c1ccc(cc1Cl)Cl 1D-004 c1cc(ccc1c2ccnc3n2nc(n3)N4CCOCC4)Br 1D-006 c1ccc(cc1)c2ccc(cc2)c3ccnc4n3nc(n4)N5CCOCC5 1D-007 c1ccc2c(c1)ncc(n2)Cl 1D-008 c1cc(nc(c1)Cl)NNC(=O)N 1D-009 COc1ccc(cc1)c2ccnc3n2nc(n3)N4CCOCC4 1D-010 c1ccc(cc1)c2cnc3nc(nn3c2N)N4CCOCC4 1D-011 CC(=O)C1C(=O)OC(OC1=O)(C)C 1D-012 c1cc(c(cc1Cl)Cl)c2ccnc3n2nc(n3)N4CCOCC4 1D-013 c1cscc1c2cnc3nc(nn3c2N)N4CCOCC4 1D-014 c1ccnc(c1)c2ccnc3n2nc(n3)N4CCOCC4 1D-015 CC(=O)/C=C/c1ccc(cc1)F 1D-016 CN(C)/C=C/C(=O)/C=C/c1ccc(cc1)Cl 1D-018 c1cc(ccc1c2cnc3nc(nn3c2N)N4CCOCC4)Cl 1D-021 c1cc(nc(c1)Cl)n2cnc(n2)O 1D-022 CN(C)/C=C/C(=O)/C=C/c1ccc(cc1)F 1D-023 c1cc(ccc1c2ccnc3n2nc(n3)N4CCOCC4)n5ccnc5 1D-024 c1ccc(cc1)Oc2ccc(cc2)c3ccnc4n3nc(n4)N5CCOCC5 1D-025 c1cc(oc1)c2ccnc3n2nc(n3)N4CCOCC4 1D-026 CN(C)/C=C/C(=O)/C=C/c1cccs1 1D-027 CN(C)/C=C/C(=O)/C=C/c1ccc(cc1)OC 1D-028 c1cc(ccc1c2ccnc3n2nc(n3)N4CCOCC4)F 1D-029 c1c2c(n3c(n1)nc(n3)N4CCOCC4)CCCC2=O 1D-030 CC(=O)COc1ncn(n1)c2ccccc2 1D-031 CC(C(=O)C)Oc1ncn(n1)c2ccccc2 1D-032 CO/N=C/C(=C(c1ccc(cc1)F)O)/C=N\OC 1D-034 c1c(cnc(c1Cl)NNC(=O)N)C(F)(F)F 1D-036 c1ccc(cc1)C(=O)C2C(O2)c3ccc(cc3)Cl 1D-038 c1ccc(cc1)C2C(O2)C(=O)c3ccc(cc3)Cl 1D-040 c1c(cnc(c1Cl)n2cnc(n2)O)C(F)(F)F 1D-041 c1cc(ccc1c2ccnc3n2ncn3)Cl 1D-042 c1cc(ccc1c2ccnc3n2ncn3)F 1D-043 c1cc(ccc1c2ccnc3n2ncn3)Br 1D-044 c1cc(oc1)c2ccnc3n2ncn3 1D-045 c1ccc(cc1)c2cnc3ncnn3c2N 1D-046 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C=O)Cl 1D-047 c1ccnc(c1)c2ccnc3n2ncn3 1D-048 c1cc(ccc1c2cnc3ncnn3c2N)Cl 1D-049 c1cscc1c2cnc3ncnn3c2N 1D-050 c1ccc(cc1)/C=C/c2ccnc3n2ncn3 1D-051 c1cc(ccc1/C=C/c2ccnc3n2ncn3)F 1D-052 c1cc(ccc1/C=C/c2ccnc3n2ncn3)Cl 1D-053 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])/C=N/O)Cl 1D-054 CC(c1ccnc(n1)N)Oc2ncn(n2)c3ccccc3 1D-056 c1c2c(n3c(n1)ncn3)CCCC2=O 1D-057 c1cc(sc1)/C=C/c2ccnc3n2ncn3 1D-058 COc1ccc(cc1)/C=C/c2ccnc3n2ncn3 1D-059 CC1(CC(=O)C(=CN(C)C)C(=O)C1)C 1D-061 c1c2c([nH]n1)-c3cnc4ncnn4c3CC2 1D-062 CN1CCC(=O)/C(=C/N(C)C)/C1 1D-063 CC1(Cc2c(cnc3n2ncn3)C(=O)C1)C 1D-064 c1cc(ccc1c2ccnc3n2ncn3)n4ccnc4 1D-065 c1ccc(cc1)Oc2ccc(cc2)c3ccnc4n3ncn4 1D-066 COC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)Cl 1D-067 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C=O)F 1D-068 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])/C=N\O)F 1D-069 CO/N=C\c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)Cl 1D-070 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])C=O)C(F)(F)F 1D-072 c1cc(ccc1c2ccnc3n2nnn3)Cl 1D-075 c1cc(c(cc1c2ccnc3n2ncn3)Cl)Cl 1D-077 CC(c1ccnc2n1ncn2)Oc3ccccc3 1D-081 c1ccc(cc1)C(=O)O/N=C/c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl 1D-082 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])/C=N/O)C(F)(F)F 1D-084 c1ccc(cc1)C(=O)O/N=C/c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)F 1D-085 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Oc2cccc(c2)C(F)(F)F 1D-086 CO/N=C/C(=C(c1ccc(cc1)c2ccccc2)O)/C=N\OC 1D-088 CC(c1ccnc2n1ncn2)Oc3ccc(cc3Cl)Cl 1D-089 CO/N=C/C(=C(c1ccc(cc1)Br)O)/C=N\OC 1D-091 CC(c1ccnc2n1ncn2)Oc3ccc(cc3)Cl 1D-092 CN(C)/C=C(\C#N)/c1ccc(cc1)F 1D-094 Cc1c(cnc2n1ncn2)C(=O)C 1D-095 CN(C)/C=C(/C#N)\c1ccc(cc1)OC 1D-096 CO/N=C/CC(=O)c1ccc(c(c1)Cl)Cl 1D-099 COc1ccc(cc1)c2cnc3ncnn3c2N 1D-100 c1cc(ccc1c2cnc3ncnn3c2N)F 1D-101 CO/N=C/C(=C(c1ccc(c(c1)Cl)Cl)O)/C=N\OC 1D-103 c1cnc2ncnn2c1N 1D-106 c1cc(c(cc1Cl)Cl)c2ccnc3n2ncn3 1D-111 c1cc(cc(c1)Cl)Oc2ccc(cc2[N+](=O)[O-])C=O 1D-113 Cc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C=O 1D-114 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Oc2cccc(c2)Cl 1D-115 c1cc(cc(c1)Cl)Oc2ccc(cc2[N+](=O)[O-])/C=N/O 1D-116 CN(C)/C=C/C(=O)c1ccccc1 1D-120 Cc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])/C=N/OC 1D-121 c1cnn(c1)CCCl 1D-124 c1ccc(cc1)C(=O)NCCCl 1D-126 COC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)F 1D-128 c1ccc(cc1)c2ccnc3n2ncc3C#N 1D-129 c1cc(c(cc1c2ccnc3n2ncc3C#N)Cl)Cl 1D-130 c1cc(ccc1c2ccnc3n2ncc3C#N)F 1D-131 c1ccnc(c1)c2ccnc3n2ncc3C#N 1D-132 c1ccc(cc1)c2ccnc3n2ncn3 1D-133 c1ccc(cc1)Oc2ccc(cc2)c3ccnc4n3ncc4C#N 1D-134 COc1ccc(cc1)c2ccnc3n2ncc3C#N 1D-135 Cc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])/C=N/OC(=O)c3ccccc3 1D-136 c1cc(ccc1c2ccnc3n2ncc3C#N)Br 1D-137 c1cc(ccc1c2ccnc3n2ncc3C#N)n4ccnc4 1D-138 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)NO)F 1D-139 c1ccc2c(c1)ncc(n2)Sc3ccc(cc3)Cl 1D-140 COC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2cccc(c2)C(F)(F)F 1D-141 CNc1c(cnn1c2ccc(cc2)Cl)[N+](=O)[O-] 1D-146 CNc1c(cnn1c2ccccn2)[N+](=O)[O-] 1D-147 c1ccc(cc1)/C=C\c2ccnc3n2ncc3C#N 1D-149 CC(=O)c1ccc(cc1)CCCl 1D-150 c1cc(ccc1/C=C\c2ccnc3n2ncc3C#N)Cl 1D-151 CC1(Cc2c(cnc3n2ncc3C#N)C(=O)C1)C 1D-152 c1ccc(cc1)c2cnc3c(cnn3c2N)C#N 1D-153 Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2)S(=O)(=O)Oc3cccc(c3)C(F)(F)F 1E-001 c1ccc(c(c1)C(=O)O)NC(=O)CC(=O)O 1E-002 CN(c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)N 1E-003 COc1ccc(cc1)Sc2c(n3ccsc3n2)C=O 1E-004S COc1ccc(cc1)Sc2c(n3ccsc3n2)/C=N/O 1E-005S c1ccc(cc1)c2c(c(nc(n2)c3cccnc3)O)C#N 1E-007S CN(c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)NC(=O)Nc3ccc(cc3)Cl 1E-009 c1ccc(cc1)c2c(c(nc(n2)c3ccncc3)O)C#N 1E-011S COc1ccc(cc1)Sc2c(n3ccsc3n2)C#N 1E-012S c1ccnc(c1)c2nc(c(c(n2)Sc3ccc(cc3)Cl)C#N)c4ccc(cc4)Cl 1E-013S CN(C)c1c(c(nc(n1)c2ccccc2)c3ccc(cc3)Cl)C#N 1E-014S c1cc(ccc1NC(=O)CC(=O)O)Br 1E-016 c1ccc(cc1)c2c(c(nc(n2)c3cccnc3)Cl)C#N 1E-020S CN(c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)NC(=S)Nc3ccccc3 1E-021 CN(C)/C=C/C(=O)Nc1ccc(cc1)Br 1E-022 c1ccnc(c1)C2=NN=C(NN2)c3ccccn3 1E-023 CC(C)Sc1c(n2ccsc2n1)C#N 1E-024S CN(C)c1c(c(nc(n1)c2cccnc2)c3ccc(cc3)Cl)C#N 1E-026S CNc1c(c(nc(n1)c2cccnc2)c3ccc(cc3)Cl)C#N 1E-027S CN(c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)NC(=O)c3ccc(cc3Cl)Cl 1E-029 CN(c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)NC(=O)c3ccc(cc3)F 1E-031 c1ccc(cc1)/C=C/C(/C=N\OCc2ccc(cc2Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl 1E-033 c1cc(cnc1)c2nc(c(c(n2)Cl)C#N)c3ccc(cc3)Cl 1E-035S COC(=O)c1c(ccs1)c2ccc(o2)C(=O)Nc3ccc(cc3)OC(F)(F)F 1E-036 COC(=O)c1c(ccs1)c2ccc(o2)COC(=O)Nc3cccc(c3)C(F)(F)F 1E-037 COc1ccc(cc1)NC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(cc4)Cl 1E-038 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)OC(F)(F)F 1E-039 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4F)F 1E-040 Cc1cc2nccc(n2n1)N 1E-041 c1ccc(cc1)c2c(c(nc(n2)c3ccccn3)O)C#N 1E-042S c1ccc(cc1)c2c(c(nc(n2)c3ccncc3)Cl)C#N 1E-043S c1cc(ccc1c2c(c(nc(n2)c3ccncc3)Cl)C#N)Cl 1E-044S c1ccc2c(c1)/C(=C/c3ccc(cc3Cl)Cl)/OC2=O 1E-046 c1cc(cnc1)c2nc(c(c(n2)N3CCOCC3)C#N)c4ccc(cc4)Cl 1E-047S c1ccc(cc1)c2c(c(nc(n2)c3cccnc3)N4CCOCC4)C#N 1E-048S CN(C)c1c(c(nc(n1)c2cccnc2)c3ccccc3)C#N 1E-049S CN(C)c1c(c(nc(n1)c2ccncc2)c3ccccc3)C#N 1E-050S c1cc(ccc1NC(=O)C/C=N\OCc2ccc(cc2Cl)Cl)Br 1E-051 COc1ccc(cc1)NC(=O)C/C=N\O 1E-052 c1cc(ccc1NC(=O)C/C=N\OCc2ccc(c(c2)Cl)Cl)Br 1E-053 c1ccnc(c1)c2nnc(n2N)c3ccccn3 1E-054 c1cc(c(c(c1)Cl)CO/N=C\CC(=O)Nc2ccc(cc2)Br)Cl 1E-055 c1cc(ccc1CO/N=C\CC(=O)Nc2ccc(cc2)Br)[N+](=O)[O-] 1E-056 c1ccc2c(c1)c(n[nH]c2=O)Cc3ccc(cc3Cl)Cl 1E-057 COC(=O)c1c(ccs1)c2ccc(o2)COC(=O)NC3CCCCC3 1E-058 COC(=O)c1c(ccs1)c2ccc(o2)COC(=O)c3ccc(cc3)Cl 1E-059 CC(C)Nc1c(c(nc(n1)c2cccnc2)c3ccccc3)C#N 1E-060S c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)N3CCNCC3 1E-061 CO/N=C\CC(=O)Nc1ccc(cc1)Br 1E-062 CN(C)/C=C(/C=N/OCc1c(cccc1Cl)Cl)\C(=O)Nc2ccc(c(c2)Cl)Cl 1E-063 c1ccc(cc1)c2cnn(c2N)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 1E-064 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)Nc4cccc(c4)C(F)(F)F 1E-065 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4Cl)Cl 1E-066 c1ccc(cc1)CNC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(cc4)Cl 1E-067 COc1ccc(cc1)c2cnn(c2N)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 1E-068 CN(C)/C=C(\C=N\OCc1ccc(cc1)[N+](=O)[O-])/C(=O)Nc2ccc(cc2)Cl 1E-069 c1cc(ccc1c2cnn(c2N)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)Cl 1E-070 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 1E-071 CC(C)Nc1c(c(nc(n1)c2cccnc2)c3ccc(cc3)Cl)C#N 1E-072S COC(=O)c1c(ccs1)c2ccc(o2)COC(=O)Nc3ccccc3 1E-073 CC(C)Nc1c(c(nc(n1)c2ccncc2)c3ccccc3)C#N 1E-074S CN(C)c1c(c(nc(n1)c2ccncc2)c3ccc(cc3)Cl)C#N 1E-075S c1cc(ccc1c2cnn(c2N)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)F 1E-076 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)N4CCCC4 1E-077 CNC(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)Cl 1E-078 CNC(=O)c1c2ccccc2c(=O)n(n1)c3ccccc3 1E-079 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F)Cl 1E-080 c1ccc(cc1)c2c(c(nc(n2)c3ccccc3)O)C#N 1E-084S c1ccc(cc1)c2c(c(nc(n2)c3ccccc3)Cl)C#N 1E-085S c1cc(c(cc1F)F)NC(=O)CC(=O)O 1E-086 c1ccc(cc1)Cc2c3ccccc3c(nn2)Cl 1E-087 CN(C)/C=C(/C=N/OCc1ccc(cc1Cl)Cl)\C(=O)Nc2ccc(cc2)Br 1E-088 CN(C)/C=C/C(=O)Nc1ccc(cc1F)F 1E-089 c1ccc(cc1)Cc2c3ccccc3c(nn2)N4CCOCC4 1E-091 c1ccc(cc1)Cc2c3ccccc3c(nn2)N4CCCCC4 1E-092 c1cc(c(cc1F)F)NC(=O)C/C=N\OCc2ccc(cc2Cl)Cl 1E-093 CC(C)Nc1c(c(nc(n1)c2ccncc2)c3ccc(cc3)Cl)C#N 1E-094S COC(=O)c1c(ccs1)c2ccc(o2)COC(=O)c3ccccc3 1E-095 COc1ccc(cc1)C(=O)OCc2ccc(o2)c3ccsc3C(=O)OC 1E-096 CCN(CC)c1c(c(nc(n1)c2ccccc2)c3ccc(cc3)Cl)C#N 1E-097S CC(C)Nc1c(c(nc(n1)c2ccccc2)c3ccc(cc3)Cl)C#N 1E-098S c1ccc(cc1)Cc2c3ccccc3c(nn2)N4CCN(CC4)c5ccccc5 1E-099 c1cc(ccc1CO/N=C\CC(=O)Nc2ccc(cc2F)F)[N+](=O)[O-] 1E-100 c1cc(c(cc1CO/N=C\CC(=O)Nc2ccc(cc2F)F)Cl)Cl 1E-101 c1cc(c(c(c1)Cl)CO/N=C\CC(=O)Nc2ccc(cc2F)F)Cl 1E-102 CC(=O)/C(=C/N(C)C)/C(=O)Nc1ccc(cc1Cl)Cl 1E-103 c1ccc(cc1)NC(=O)n2ccc(n2)c3ccc(cc3Cl)Oc4ccc(cc4)Cl 1E-104 CC(=O)C(/C=N/OCc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 1E-105 c1ccc(cc1)CSc2c(c(nc(n2)c3ccncc3)c4ccc(cc4)Cl)C#N 1E-106S c1ccc(cc1)Sc2c(c(nc(n2)c3ccncc3)c4ccc(cc4)Cl)C#N 1E-107S C=CCNc1c(c(nc(n1)c2ccccc2)c3ccc(cc3)Cl)C#N 1E-108S CN1CCN(CC1)c2c(c(nc(n2)c3ccccc3)c4ccc(cc4)Cl)C#N 1E-109S CCN(CC)c1c(c(nc(n1)c2ccccn2)c3ccccc3)C#N 1E-110S CCN(CC)c1c(c(nc(n1)c2ccccn2)c3ccc(cc3)Cl)C#N 1E-111S CN(C)c1c(c(nc(n1)c2ccccn2)c3ccccc3)C#N 1E-112S C=CCNc1c(c(nc(n1)c2ccccn2)c3ccc(cc3)Cl)C#N 1E-113S c1cc(c(cc1F)F)NC(=O)C/C=N\O 1E-116 CC(=O)C(/C=N/OC)C(=O)Nc1ccc(cc1Cl)Cl 1E-118 CC(C)(C)C(=O)OCc1ccc(o1)c2ccsc2C(=O)OC 1E-119 COC(=O)c1c(ccs1)c2ccc(o2)COC(=O)CCl 1E-120 CN1CCN(CC1)c2c(c(nc(n2)c3ccccn3)c4ccccc4)C#N 1E-121S CN1CCN(CC1)c2c(c(nc(n2)c3ccccn3)c4ccc(cc4)Cl)C#N 1E-122S c1ccc(cc1)NC(=O)Nn2c(nnc2c3ccccn3)c4ccccn4 1E-124 c1cc(ccc1NC(=O)n2ccc(n2)c3ccc(cc3Cl)Oc4ccc(cc4)Cl)Cl 1E-125 c1ccc(cc1)n2c(ccn2)c3ccc(cc3Cl)Oc4ccc(cc4)Cl 1E-128 CC(C)Nc1c(c(nc(n1)c2ccccn2)c3ccccc3)C#N 1E-129S CCN(CC)c1c(c(nc(n1)c2ccncc2)c3ccc(cc3)Cl)C#N 1E-130S C=CCNc1c(c(nc(n1)c2ccncc2)c3ccc(cc3)Cl)C#N 1E-131S CN1CCN(CC1)c2c(c(nc(n2)c3ccncc3)c4ccc(cc4)Cl)C#N 1E-132S c1cc(ccc1C(=O)n2ccc(n2)c3ccc(cc3Cl)Oc4ccc(cc4)Cl)Cl 1E-134 CN1CCN(CC1)c2c(c(nc(n2)c3ccccc3)c4ccccc4)C#N 1E-136S CCN(CC)c1c(c(nc(n1)c2ccccc2)c3ccccc3)C#N 1E-137S C=CCNc1c(c(nc(n1)c2ccccc2)c3ccccc3)C#N 1E-138S c1ccc(cc1)c2c(c(nc(n2)c3ccccc3)N4CCOCC4)C#N 1E-139S CNc1c(c(nc(n1)c2ccccc2)c3ccccc3)C#N 1E-140S c1cc(c(cc1Cl)Cl)n2c(c(nn2)C(=O)O)CC(=O)O 1E-141 CC(C)Oc1c(c(nc(n1)c2ccccc2)c3ccccc3)C#N 1E-142S CC(C)Oc1c(c(nc(n1)c2ccccc2)c3ccc(cc3)Cl)C#N 1E-143S c1cc(c(cc1OCC(F)(F)F)C(=O)NOCc2ccc(cc2Cl)Cl)OCC(F)(F)F 1E-144S c1cc(c(cc1CONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl)Cl 1E-145S c1cc(ccc1Oc2ccc(c(c2)Cl)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl)Cl 1E-147 CC(=O)C(/C=N/OC)C(=O)Nc1ccc(cc1)Cl 1E-149 c1ccnc(c1)c2nnc(n2NC(=O)Nc3ccc(cc3)OC(F)(F)F)c4ccccn4 1E-150 CC(=O)C(/C=N/OCc1c(cccc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 1E-152 c1cc(c(c(c1)Cl)CONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 1E-155S c1cc(ccc1CONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)[N+](=O)[O-] 1E-156S CONC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 1E-157S CCNC(=O)Nn1c(nnc1c2ccccn2)c3ccccn3 1E-159 c1ccc(cc1)c2c(c(nc(n2)c3ccccc3)Sc4ccccc4)C#N 1E-160S c1ccc(cc1)c2c(c(nc(n2)c3ccccc3)Sc4ccc(cc4)Cl)C#N 1E-161S c1cc(ccc1C(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 1E-163S c1cc(c(cc1C(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl)Cl 1E-164S c1ccc(cc1)c2nc(c(c(n2)Sc3ccccc3)C#N)c4ccc(cc4)Cl 1E-168S c1ccc(cc1)c2nc(c(c(n2)Sc3ccc(cc3)Cl)C#N)c4ccc(cc4)Cl 1E-169S c1ccnc(c1)c2nnc(n2N(S(=O)(=O)c3cccc(c3)C(F)(F)F)S(=O)(=O)c4cccc(c4)C(F)(F)F)c5ccccn5 1E-170 c1ccc(cc1)Cc2c3ccccc3c(nn2)Sc4ccccc4 1E-173 CNc1c(c(nc(n1)c2ccccc2)c3ccc(cc3)Cl)C#N 1E-177S COc1ccc(cc1)c2c(c(nc(n2)c3ccccn3)O)C#N 1E-178S COc1ccc(cc1)c2c(c(nc(n2)c3ccccn3)Cl)C#N 1E-179S c1ccc(cc1)Sc2c(c(nc(n2)c3cccnc3)c4ccc(cc4)Cl)C#N 1E-180S c1ccc(cc1)CNc2c(c(nc(n2)c3ccccc3)c4ccc(cc4)Cl)C#N 1E-181S c1ccc(cc1)Cc2c3ccccc3c(nn2)Oc4ccc(cc4)Cl 1E-182 CN(C)/C=N/n1c(nnc1c2ccccn2)c3ccccn3 1E-183 c1cc(ccc1C(=O)Cn2ccnc2)Cl 1E-184 Cc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)O 1E-189 c1cc(ccc1C(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)F 1E-190S c1cc(cc(c1)C(F)(F)F)C(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 1E-191S COc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)O)C#N 1E-192S COc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)Cl)C#N 1E-194S CNc1c(c(nc(n1)c2ccccn2)c3ccc(cc3)OC)C#N 1E-196S COC(=O)c1cnc(nc1c2cccnc2)SC 1E-902 COC(=O)c1cnc(nc1c2ccncc2)c3ccccn3 1E-903 c1ccnc(c1)c2ncc(c(n2)c3ccncc3)C(=O)O 1E-905 Cc1ccc(cc1)c2ncc(c(n2)c3ccncc3)C(=O)OC 1E-908 c1ccnc(c1)c2ncc(c(n2)c3ccncc3)C(=O)NN 1E-910 Cc1ccc(cc1)c2ncc(c(n2)c3ccncc3)C(=O)[NH2+][NH3+].[Cl-].[Cl-] 1E-912 Cc1ccc(cc1)c2ncc(c(n2)c3ccncc3)C(=O)NC 1E-914 COC(=O)/C(=C/N)/C(=O)c1ccncc1 1E-916 Cc1ccc(cc1)c2ncc(c(n2)c3cccnc3)C(=O)OC 1E-917 Cc1ccc(cc1)c2ncc(c(n2)c3ccncc3)C(=O)N 1E-919 Cc1ccc(cc1)c2ncc(c(n2)c3cccnc3)C(=O)NC 1E-920 Cc1ccc(cc1)c2ncc(c(n2)c3cccnc3)C(=O)N 1E-921 c1ncn(n1)C/C(=N/O)/[NH3+].[Cl-] 1F-001 c1cc(c(cc1Cl)Cl)NC(=O)C(=O)NNC(=N)Cn2cncn2 1F-002 CC(c1ccn(n1)C(=O)Nc2ccccc2)n3cncn3 1F-003 c1cc(c(cc1Cl)Cl)NC(=O)c2[nH]nc(n2)Cn3cncn3 1F-005 CNC(=O)c1cc(c[nH]1)C(=O)c2ccccc2C(F)(F)F 1F-006 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)F 1F-007 CC(c1ccn(n1)C(=O)C)n2cncn2 1F-010 c1ccc(c(c1)C(C#N)c2ccc(nn2)Cl)F 1F-011 c1cc(nc(c1)Cl)n2c(ccn2)O 1F-012 CC(c1ccn(n1)S(=O)(=O)c2ccccc2)n3cncn3 1F-013 CN(C)/C=C\1/C=NN(C1=O)c2cccc(n2)Cl 1F-014 c1cc(nc(c1)Cl)N2C(=O)/C(=C\Nc3ccc(cc3)Cl)/C=N2 1F-016 c1c(cnc(c1Cl)N2C(=O)CC=N2)C(F)(F)F 1F-017 CC(c1ccn(n1)S(=O)(=O)C)n2cncn2 1F-018 c1ccc(c(c1)Cc2ccc(nn2)O)F 1F-019 c1ccc\2c(c1)-c3c(cccn3)/C2=N/OCc4ccc(cc4)Cl 1F-020 c1ccc\2c(c1)-c3c(cccn3)/C2=N/OCc4ccc(cc4Cl)Cl 1F-021 c1ccc(c(c1)Cc2ccc(nn2)Cl)F 1F-023 c1cc(nc(c1)Cl)N2C(=O)/C(=C\Nc3ccc(cc3Cl)Cl)/C=N2 1F-026 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)C(=O)c2ccc(cc2Cl)Cl 1F-028 Cn1cc(cc1C(=O)OC)C(=O)c2ccc(cc2Cl)Cl 1F-029 c1ccc(c(c1)Cc2ccc(nn2)NN)F 1F-030 c1ccc(cc1)Oc2ccc(cc2)N/C=C\3/C=NN(C3=O)c4cccc(n4)Cl 1F-031 c1cc(cc(c1)N/C=C\2/C=NN(C2=O)c3cccc(n3)Cl)C(F)(F)F 1F-032 c1cc(nc(c1)Cl)N2C(=O)/C(=C\NOCc3ccc(cc3Cl)Cl)/C=N2 1F-033 c1cc(c(c(c1)Cl)CON/C=C\2/C=NN(C2=O)c3cccc(n3)Cl)Cl 1F-034 Cc1ccc(cc1)n2c(=O)cc(c(n2)C#N)Cl 1F-035 CC(C)OC(=O)Nc1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 1F-039 CCOC(=O)CC(=N)NNC(=O)c1ccncc1 1F-040 CCOC(=O)CC(=N)NNc1c(cc(cn1)C(F)(F)F)Cl 1F-042 CCOC(=O)Cc1[nH]nc(n1)c2ccncc2 1F-043 CC(C1c2ccccc2C(=O)O1)[N+](=O)[O-] 1F-045 Cn1cc(cc1C(=O)O)C(=O)c2ccc(cc2Cl)Cl 1F-048 c1cc(c(cc1Cl)Cl)n2c(=O)cc(c(n2)C(=O)N)O 1F-049 Cn1c(cc(c1)C(=O)c2c(cc(cc2)Cl)Cl)/C=C/C(=O)/C=C/c3n(cc(c3)C(=O)c4c(cc(cc4)Cl)Cl)C 1F-050 COC(=O)c1c(cc(=O)n(n1)c2ccccc2)Cl 1F-051 COC(=O)c1c(cc(=O)n(n1)c2ccccc2)Sc3ccc(cc3)Cl 1F-053 Cn1cc(cc1/C=N/OCc2ccc(cc2)Cl)C(=O)c3ccc(cc3Cl)Cl 1F-054 c1cc(c(cc1Cl)Cl)CO/N=C\CC(=O)NN 1F-055 c1cc(c(cc1Cl)Cl)n2c(=O)cc(c(n2)C#N)Cl 1F-056 c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)O 1F-057 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)O 1F-058 CN(C)/C=C/1\Cc2c(cc(cc2Cl)Cl)C1=O 1F-061 c1cc(c(c(c1)Cl)C(C#N)c2ccc(nn2)Cl)F 1F-062 CN(C)c1nc(n(n1)c2ccc(cc2)Cl)N(C)C 1F-064 c1cc(c(c(c1)Cl)Cc2ccc(nn2)O)F 1F-065 c1cc(c(c(c1)Cl)C(C#N)c2ccc(nn2)Cl)Cl 1F-066 Cc1cccc(c1C)n2c(nc(n2)N(C)C)N(C)C 1F-067 c1cc(c(c(c1)Cl)Cc2ccc(nn2)O)Cl 1F-068 c1cc(c(c(c1)Cl)Cc2ccc(nn2)Cl)F 1F-069 COc1ccc(cc1)Cn2cccc(c2=O)C(=O)O 1F-303S c1ccc2c(c1)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/C(=O)N2Cc4ccc(cc4Cl)Cl 1F-304S c1ccc(cc1)C(=O)O/N=C\2/c3ccccc3N(C2=O)Cc4ccc(cc4Cl)Cl 1F-305S c1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3Cl)Cl)/C(=O)N2Cc4ccc(cc4Cl)Cl 1F-306S c1ccc2c(c1)/C(=N/OC(=O)c3c(cccc3Cl)Cl)/C(=O)N2Cc4ccc(cc4Cl)Cl 1F-307S c1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3)Cl)/C(=O)N2Cc4ccc(cc4Cl)Cl 1F-308S c1ccc2c(c1)/C(=N/OC(=O)c3ccccc3Cl)/C(=O)N2Cc4ccc(cc4Cl)Cl 1F-309S CCC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3ccc(cc3Cl)Cl 1F-310S Cc1ccc(cc1)C(=O)O/N=C\2/c3ccccc3N(C2=O)Cc4ccc(cc4Cl)Cl 1F-311S c1ccc2c(c1)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/C(=O)N2Cc4c(cccc4Cl)Cl 1F-312S c1ccc2c(c1)/C(=N/OC(=O)c3ccc(cc3)Cl)/C(=O)N2Cc4c(cccc4Cl)Cl 1F-313S COc1ccc(cc1OC)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-315S COc1ccc(c(c1)OC)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-316S c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)C(=O)Nc3ccc4c(c3)OCO4 1F-317S c1ccc(c(c1)Cn2cccc(c2=O)C(=O)O)Cl 1F-318S COc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)Cl 1F-321S COc1ccc(cc1OC)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)Cl 1F-324S COc1ccccc1NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-325S COc1cccc(c1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-327S c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)C(=O)Nc3ccc(cc3)S(=O)(=O)N 1F-328S CCOc1ccccc1NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-329S CCOc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-330S COc1ccc(cc1)S(=O)(=O)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-331S c1ccc(cc1)NC2=NNc3ccccc3S2 1F-332S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)NS(=O)(=O)c3ccc(cc3)OC 1F-333S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3)OC 1F-334S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccc4c(c3)OCO4 1F-335S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3OC)OC 1F-336S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccc(c(c3)OC)OC 1F-337S CCOc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)Cl 1F-338S COc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccccc3Cl 1F-339S C=CCn1cccc(c1=O)C(=O)O 1F-340S c1cc(c(nc1)Cl)C(=O)NNc2cc(ccc2Cl)Cl 1F-341S COc1ccc(cc1)NC(=O)c2cccn(c2=O)CC=C 1F-343S c1cc2c(=O)[nH]n(c2nc1)c3ccc(cc3)Cl 1F-344S COC(=O)c1cccn(c1=O)Cc2ccccc2Cl 1F-345S COc1ccc(cc1OC)NC(=O)c2cccn(c2=O)Cc3ccccc3Cl 1F-346S c1cc(cc(c1)Cl)n2c3c(cccn3)c(=O)[nH]2 1F-347S COc1ccc(c(c1)OC)NC(=O)c2cccn(c2=O)CC=C 1F-349S COc1cc(cc(c1)OC)NC(=O)c2cccn(c2=O)CC=C 1F-350S COc1cc(cc(c1OC)OC)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-351S COc1cc(cc(c1)OC)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 1F-352S COc1ccc(c(c1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl)OC 1F-353S CCOc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccccc3Cl 1F-354S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3cc(c(c(c3)OC)OC)OC 1F-355S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3cc(cc(c3)OC)OC 1F-356S COc1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3cc(ccc3OC)OC 1F-357S COc1cc(cc(c1OC)OC)NC(=O)c2cccn(c2=O)CC=C 1F-359S COc1ccc(c(c1)NC(=O)c2cccn(c2=O)CC=C)OC 1F-360S C=CCn1cccc(c1=O)C(=O)Nc2ccc3c(c2)OCO3 1F-361S COc1ccc(cc1OC)NC(=O)c2cccn(c2=O)CC=C 1F-362S COc1cc(nc(n1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl)OC 1F-364S COc1ccc(c(c1)NC(=O)c2cccn(c2=O)Cc3ccccc3Cl)OC 1F-366S COc1cc(cc(c1)OC)NC(=O)c2cccn(c2=O)Cc3ccccc3Cl 1F-369S c1ccc(cc1)n2c3c(cccn3)c(=O)n2Cc4ccc(cc4)Cl 1F-373S c1ccc(cc1)n2c3c(cccn3)c(=O)n2Cc4c(cccc4Cl)Cl 1F-374S c1ccc(c(c1)Cn2cccc(c2=O)C(=O)Nc3ccc4c(c3)OCO4)Cl 1F-376S COc1ccccc1NC(=O)c2cccn(c2=O)Cc3ccccc3Cl 1F-377S c1cc(c(c(c1)Cl)Cn2c(=O)c3cccnc3n2c4cc(ccc4Cl)Cl)Cl 1F-378S c1cc2c(=O)[nH]n(c2nc1)c3ccc(cc3)F 1F-380S Cc1ccc(cc1)n2c3c(cccn3)c(=O)[nH]2 1F-382S c1ccc2c(c1)CSC(=N2)NCc3ccc(cc3)Cl 1F-385S COc1ccc(cc1)CNC2=Nc3ccccc3CS2 1F-386S c1ccc(cc1)Cc2[nH]c(=O)c3ccccc3n2 1F-389S c1ccc2c(c1)c(=O)[nH]c(n2)Cc3ccc(cc3)Cl 1F-390S c1ccc2c(c1)CSC(=N2)NCc3cccc(c3)C(F)(F)F 1F-393S c1ccc2c(c1)CSC(=N2)NCc3ccccc3Cl 1F-394S c1ccc2c(c1)CSC(=N2)NCc3cccnc3 1F-395S CCOC(=O)NC(=O)/C(=C\NN1CCCCC1)/C#N 1F-900 CCOC(=O)NC(=O)C(/C=N/OCc1ccc(cc1)Cl)C(=O)NC(=O)OCC 1F-901 c1c(c(=O)[nH]c(=O)n1N2CCCCC2)C#N 1F-903 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)OCc2ccc(cc2)Cl 1F-904 c1c(c(=O)[nH]c(=O)n1CCO)C#N 1F-905 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)N 1F-907 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)N2CCOCC2 1F-908 CC(=O)c1cn(c(=O)[nH]c1=O)N2CCN(CC2)C 1F-909 c1c(c(=O)[nH]c(=O)n1CC#N)C#N 1F-910 c1cc(cc(c1)C(F)(F)F)C(=O)OCCn2cc(c(=O)[nH]c2=O)C#N 1F-911 Cc1ccc(cc1)C(=O)OCCn2cc(c(=O)[nH]c2=O)C#N 1F-912 c1cc(sc1)C(=O)OCCn2cc(c(=O)[nH]c2=O)C#N 1F-913 c1ccc-2c(c1)CCc3c2nc(nc3)N 1F-915 CCOC(=O)NC(=O)/C(=C\NC#N)/C#N 1F-916 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)OC 1F-924 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)NC(=O)c2cccs2 1F-925 CC(=O)c1cn(c(=O)[nH]c1=O)C 1F-928 Cn1cc(c(=O)[nH]c1=O)C(=O)/C=C/c2ccccc2 1F-930 CCOC(=O)CNc1ccccc1C#N 1F-932 Cc1cc(n(n1)C(=S)N)c2c(nn(c2O)c3ccccc3)C 1F-933 CCOC(=O)c1c(c2ccccc2[nH]1)N 1F-936 c1ccc2c(c1)c3c([nH]2)c(=O)[nH]cn3 1F-937 CCOc1c(cc(c(=O)[nH]1)C(=O)OCC)C(=O)OCC 1F-938 c1ccc2c(c1)c3c([nH]2)c(nc[nH+]3)Cl.[Cl-] 1F-941 c1ccc(cc1)C(=O)NCC(=O)N2CCN(CC2)c3ccccc3 1F-942 c1ccc(cc1)C(=O)NCC(=O)NOCc2ccc(cc2)Cl 1F-943 c1ccc(cc1)N2CCN(CC2)C(=O)CNC(=O)c3ccc(cc3)Cl 1F-944 c1ccc(cc1)C(=O)NCC(=O)Nc2ccc(cc2)N 1F-946 CC(=O)c1ccc(cc1)NC(=O)CNC(=O)c2ccccc2 1F-950 c1ccc(cc1)N2CCN(CC2)c3c4c(c5ccccc5[nH]4)ncn3 1F-952 c1ccc2c(c1)c3c([nH]2)c(ncn3)Sc4ccc(cc4)Cl 1F-953 c1ccc2c(c1)c3c([nH]2)c(ncn3)N4CCOCC4 1F-954 c1ccc2c(c1)c3c([nH]2)c(ncn3)NN 1F-955 c1ccc(cc1)C(=O)NCC(=O)NNC(=S)N 1F-956 CCO/C(=C(/C=C(\C#N)/C(=O)OCC)\C(=O)OCC)/N 1F-957 c1ccc(cc1)C(=O)Nc2ncc3c(n2)-c4ccccc4CC3 1F-959 c1ccc2c(c1)CC(=O)N(C2=O)OCc3ccc(cc3)Cl 1F-960 CC(=NNc1c2c(c3ccccc3[nH]2)ncn1)C 1F-962 c1ccc(cc1)C(=O)NCc2nc([nH]n2)S 1F-963 COc1ccc(cc1)N/C=C\2/c3ccccc3C(=O)N(C2=O)OCc4ccc(cc4)Cl 1F-964 c1ccc(cc1)C(=O)NCC(=O)NCCO 1F-965 c1ccc(cc1)C(=O)NCC(=O)NCCOC(=O)c2cccs2 1F-966 CCOC(=O)c1cc(c(nc1NNc2ccccc2)O)C(=O)OCC 1F-967 c1ccc2c(c1)CC(=O)N(C2=O)OCc3ccc(cc3Cl)Cl 1F-968 Cc1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(=O)N 1F-971 c1cc(c(c(c1)Cl)CO/N=C/C(=C\Nc2ccc(cc2Cl)Cl)/c3c(cc(cn3)C(F)(F)F)Cl)Cl 1G-001 CC(=O)/C(=C\N(C)C)/c1ccc(c(c1)OC)OC 1G-002 c1cc(c(c(c1)Cl)CO/N=C/C(=C\Nc2ccc(cc2)C(F)(F)F)/c3c(cc(cn3)C(F)(F)F)Cl)Cl 1G-003 Cc1c(c[nH]n1)c2ccc(c(c2)OC)OC 1G-004 c1cc(ccc1N2CCN(CC2)/C(=N/O)/c3c(cc(cn3)C(F)(F)F)Cl)F 1G-005 c1cc(cnc1)CN/C(=N/O)/c2c(cc(cn2)C(F)(F)F)Cl 1G-006 c1cc(ccc1NC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F)Cl 1G-007 c1c(cnc(c1Cl)/C(=N\O)/N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 1G-008 c1ccc(cc1)CN2CCN(CC2)/C(=N/O)/c3c(cc(cn3)C(F)(F)F)Cl 1G-009 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3cc(cc(c3)Cl)Cl)/[N+](=O)[O-] 1G-011 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3cccc(c3)Cl)/[N+](=O)[O-] 1G-012 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3cc(ccc3O)Cl)/[N+](=O)[O-] 1G-013 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3cccc(c3)C(F)(F)F)/[N+](=O)[O-] 1G-014 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3ccc(cc3)OC(F)(F)F)/[N+](=O)[O-] 1G-015 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3ccc(cc3)C(=O)O)/[N+](=O)[O-] 1G-016 c1ccc(cc1)Oc2ccc(cc2)N/C=C(\C3c4ccccc4C(=O)O3)/[N+](=O)[O-] 1G-017 C#CCN/C(=N/O)/c1c(cc(cn1)C(F)(F)F)Cl 1G-018 c1cc(ccc1CN/C(=N/O)/c2c(cc(cn2)C(F)(F)F)Cl)Cl 1G-021 Cc1cccc(c1NC(=O)CBr)C 1G-022 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3ccc(cc3F)F)/[N+](=O)[O-] 1G-024 c1ccc(cc1)CN/C=C(\C2c3ccccc3C(=O)O2)/[N+](=O)[O-] 1G-025 Cc1ccc(c(c1)C)N/C=C(\C2c3ccccc3C(=O)O2)/[N+](=O)[O-] 1G-026 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)N/C(=N/O)/c3c(cc(cn3)C(F)(F)F)Cl 1G-027 CNC(=O)/C=C/c1c(cc(cn1)C(F)(F)F)Cl 1G-028 c1cc(c(cc1Cl)Cl)CO/N=C/C(=C\Nc2ccc(cc2Cl)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 1G-029 c1cc(ccc1/C=C\2/C(=C(C(=O)O2)c3c(cc(cn3)C(F)(F)F)Cl)c4ccc(cc4)Cl)Cl 1G-030 c1cc(ccc1NC(=O)Nc2cc3c(s2)cc(cn3)C(F)(F)F)Cl 1G-032 c1cc(ccc1/C(=C/c2c(cc(cn2)C(F)(F)F)Cl)/C#N)Cl 1G-033 c1cc(ccc1C\2=C(C(=O)O/C2=C\c3ccc(cc3Cl)Cl)c4c(cc(cn4)C(F)(F)F)Cl)Cl 1G-036 Cc1c(cnc(n1)N)c2ccc(c(c2)OC)OC 1G-037 Cc1c(cn(n1)S(=O)(=O)c2ccccc2)c3ccc(c(c3)OC)OC 1G-038 c1c(cnc(c1Cl)C/C=N/O)C(F)(F)F 1G-039 Cc1c(cn(n1)S(=O)(=O)c2ccc(cc2Cl)Cl)c3ccc(c(c3)OC)OC 1G-040 Cc1c(cn(n1)S(=O)(=O)C)c2ccc(c(c2)OC)OC 1G-041 Cc1nc(c(s1)C(=O)N/C=N\O)C(F)(F)F 1G-042 c1ccc(cc1)C2=C(C(=O)OC2)c3c(cc(cn3)C(F)(F)F)Cl 1G-044 CC(C)(C(=O)CC#N)n1cncn1 1G-047 CC(=O)O/N=C(/c1c(cc(cn1)C(F)(F)F)Cl)\NCc2cccnc2 1G-048 Cc1nc(c(s1)C(=O)NC(=O)Nc2ccccc2)C(F)(F)F 1G-050 Cc1nc(c(s1)C(=O)NC(=O)Nc2cccc(c2)C(F)(F)F)C(F)(F)F 1G-051 Cc1nc(c(s1)C(=O)NC(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F 1G-052 Cc1nc(c(s1)C(=O)NC(=O)Nc2ccc(cc2)OC(F)(F)F)C(F)(F)F 1G-053 CO/N=C/C(=C\Nc1ccc(cc1Cl)Cl)/c2c(cc(cn2)C(F)(F)F)Cl 1G-054 c1cc(ccc1S(=O)(=O)O/N=C(/c2c(cc(cn2)C(F)(F)F)Cl)\N)Cl 1G-055 c1ccc(cc1)C(=O)COC(=O)CC(=O)Nc2ccc(cc2)Cl 1G-056 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)c2csc([nH+]2)CC#N.[Br-] 1G-057 Cc1nc(c(s1)c2ncnn2c3ccc(cc3)Cl)C(F)(F)F 1G-058 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)O/N=C(\c2c(cc(cn2)C(F)(F)F)Cl)/N 1G-060 CNc1c(cnn1c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 1G-061 Cc1nc(c(s1)C(=O)NC)C(F)(F)F 1G-062 CC(C)(C(=O)/C(=C/N(C)C)/C#N)n1cncn1 1G-064 CC(C)(C(=O)/C(=C/c1ccc(cc1)Cl)/C#N)n2cncn2 1G-065 CO/N=C/C(=C\Nc1ccccc1)/c2c(cc(cn2)C(F)(F)F)Cl 1G-072 COC(=O)c1ccc(cc1)N/C=C(\C=N\OC)/c2c(cc(cn2)C(F)(F)F)Cl 1G-073 CO/N=C/C(=C\Nc1ccc(cc1)F)/c2c(cc(cn2)C(F)(F)F)Cl 1G-074 CO/N=C/C(=C\Nc1ccc(cc1)C(F)(F)F)/c2c(cc(cn2)C(F)(F)F)Cl 1G-075 COc1ccc(cc1)N/C=C(\C=N\OC)/c2c(cc(cn2)C(F)(F)F)Cl 1G-076 CCCCC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(c(c3)Cl)Cl)Cl 1G-301S c1cc(c(cc1CN2c3ccc(cc3/C(=N/OC(=O)CCCl)/C2=O)Cl)Cl)Cl 1G-304S c1cc(c(cc1CN2c3ccc(cc3/C(=N/OC(=O)C(Cl)Cl)/C2=O)Cl)Cl)Cl 1G-305S Cc1ccc2c(c1)C(=O)C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-306S c1cc(c(cc1CN2c3ccc(cc3/C(=N/OC(=O)CCCCl)/C2=O)Cl)Cl)Cl 1G-307S Cc1ccc2c(c1)/C(=N/OC(=O)CCCCl)/C(=O)N2Cc3ccc(cc3)Cl 1G-308S Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 1G-309S Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)NC 1G-310S CCOC(=O)c1c(nc(s1)c2cccc(c2)C(F)(F)F)C 1G-311S COC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(cc3Cl)Cl 1G-312S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N/O)/C2=O)Cl 1G-313S Cc1ccc2c(c1)/C(=N/OC(=O)C)/C(=O)N2Cc3ccc(cc3)Cl 1G-314S c1cc(cc(c1)C(F)(F)F)c2nc(cs2)C(=O)N 1G-319S Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)C(=O)O 1G-320S Cc1c(sc(n1)c2ccccc2)C(=O)NC 1G-321S Cc1c(sc(n1)c2ccccc2)C(=O)NCC=C 1G-322S Cc1ccc2c(c1)/C(=N/OC(=O)CCCl)/C(=O)N2Cc3ccc(cc3)Cl 1G-323S CCCCC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3)Cl)C 1G-324S Cc1ccc2c(c1)/C(=N/OC(=O)CC(C)C)/C(=O)N2Cc3ccc(cc3)Cl 1G-325S c1cc(ccc1c2nc(cs2)c3ccc(cc3Cl)Cl)C(=O)O 1G-326S Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc(c(c3)Cl)Cl 1G-327S CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3)Cl)Cl 1G-328S c1cc(ccc1CN2c3ccc(cc3/C(=N/OC(=O)CCl)/C2=O)Cl)Cl 1G-329S c1cc(ccc1CN2c3ccc(cc3/C(=N/OC(=O)C(Cl)Cl)/C2=O)Cl)Cl 1G-330S c1cnccc1c2nc(cs2)C(=O)O 1G-331S CCOC(=O)c1csc(n1)c2ccncc2 1G-332S c1cc(c(c(c1)Cl)CN2c3ccc(cc3C(=O)C2=O)Cl)Cl 1G-333S Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc(cc3)OC(F)(F)F 1G-334S COC(=O)c1ccc(cc1)c2nc(cs2)c3ccccc3 1G-335S Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)C(=O)Nc3cccc(c3)C(F)(F)F 1G-336S Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F 1G-337S c1cc(ccc1CN2c3ccc(cc3/C(=N/OC(=O)CCCl)/C2=O)Cl)Cl 1G-338S c1ccc(c(c1)N)Sc2c(cccn2)[N+](=O)[O-] 1G-339S CCCCC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3)Cl)Cl 1G-341S c1cc(ccc1c2nc(cs2)c3ccc(cc3Cl)Cl)C(=O)Nc4ccc(cc4F)F 1G-343S c1cc(ccc1NC(=O)c2csc(n2)c3ccncc3)Cl 1G-344S c1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)O 1G-345S CC(C)CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3ccc(cc3)Cl)Cl 1G-346S c1cc(ccc1CN2c3ccc(cc3/C(=N/OC(=O)CCCCl)/C2=O)Cl)Cl 1G-347S c1ccc(cc1)C2C(=O)N=C(S2)c3ccccc3 1G-348S CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3cccc(c3)C(F)(F)F)Cl 1G-349S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N/OC(=O)CCl)/C2=O)Cl 1G-350S c1cc(cc(c1)NC(=O)c2csc(n2)c3ccncc3)C(F)(F)F 1G-351S Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)C(=O)Nc3cc(cc(c3)Cl)Cl 1G-352S Cc1c(sc(n1)c2ccccc2)C(=O)Nc3cc(cc(c3)Cl)Cl 1G-353S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N/OC(=O)C(Cl)Cl)/C2=O)Cl 1G-354S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N/OC(=O)CCCl)/C2=O)Cl 1G-355S CNC(=O)c1ccc(cc1)c2nc(cs2)c3ccccc3 1G-356S c1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccccc4 1G-357S Cc1ccc2c(c1)/C(=N/O)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-358S c1cc(c(c(c1)Cl)CN2c3ccc(cc3/C(=N/O)/C2=O)Cl)Cl 1G-359S CNC(=O)c1csc(n1)c2ccncc2 1G-361S c1cnccc1c2nc(cs2)C(=O)N 1G-364S c1cc(ccc1C(F)(F)F)NC(=O)c2csc(n2)c3ccncc3 1G-365S c1cc(c(cc1F)F)NC(=O)c2csc(n2)c3ccncc3 1G-366S c1cc(cc(c1)C(F)(F)F)CN2c3ccc(cc3/C(=N/OC(=O)CCCCl)/C2=O)Cl 1G-367S CCCCC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3cccc(c3)C(F)(F)F)Cl 1G-368S CC(C)CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3cccc(c3)C(F)(F)F)Cl 1G-369S CCOC(=O)c1c(nc(s1)c2ccccc2)C(F)(F)F 1G-370S c1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)Nc4cccc(c4)C(F)(F)F 1G-371S c1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4F)F 1G-372S c1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4)Cl 1G-373S c1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(c(c4)Cl)Cl 1G-374S c1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4)OC(F)(F)F 1G-375S C=CCNC(=O)c1ccc(cc1)c2nc(cs2)c3ccccc3 1G-376S c1ccc2c(c1)/C(=N/OC(=O)CCCCl)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-377S c1ccc2c(c1)/C(=N/OC(=O)CCCl)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-378S CC(C)CC(=O)O/N=C\1/c2ccccc2N(C1=O)Cc3cccc(c3)C(F)(F)F 1G-379S Cc1c(sc(n1)c2cccnc2)C(=O)O 1G-380S C/N=C(\c1ccc(cc1)Cl)/Nc2cccnc2 1G-382S c1ccc2c(c1)N(c3c(cccn3)S2)Cc4ccc(c(c4)Cl)Cl 1G-384S CN(C)CCCNC(=O)c1csc(n1)c2ccncc2 1G-386S c1ccc(cc1)c2nc(c(s2)C(=O)O)C(F)(F)F 1G-387S COC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)F 1G-388S Cc1ccc2c(c1)/C(=N/OC(=O)C)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-389S Cc1ccc2c(c1)/C(=N/OC(=O)CCl)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-390S Cc1ccc2c(c1)/C(=N/OC(=O)C(Cl)Cl)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-391S c1cc(ccc1c2nc(cs2)c3ccc(cc3)F)C(=O)O 1G-392S CN(C)C(=O)c1ccc(cc1)c2nc(cs2)c3ccc(cc3Cl)Cl 1G-393S C=CCNC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(cc3Cl)Cl 1G-394S c1cnccc1c2nc(cs2)C(=O)Nc3cc(cc(c3)Cl)Cl 1G-395S Cc1c(sc(n1)c2cccnc2)C(=O)NC 1G-396S Cc1ccc2c(c1)/C(=N/OC(=O)CCCl)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-397S c1cc(ccc1NC(=O)c2csc(n2)c3ccncc3)Br 1G-398S CCCCC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3cccc(c3)C(F)(F)F)C 1G-399S c1cc(cc(c1)NC(=O)c2ccc(cc2)c3nc(cs3)c4ccc(cc4Cl)Cl)C(F)(F)F 1G-403S c1cc(ccc1c2nc(cs2)c3ccc(cc3Cl)Cl)C(=O)Nc4ccc(cc4)OC(F)(F)F 1G-404S c1cc(ccc1c2nc(cs2)c3ccc(cc3Cl)Cl)C(=O)Nc4ccc(cc4)F 1G-405S Cc1ccc2c(c1)/C(=N/OC(=O)CC(C)C)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-406S Cc1ccc2c(c1)/C(=N/OC(=O)CCCCl)/C(=O)N2Cc3cccc(c3)C(F)(F)F 1G-407S Cc1c(sc(n1)c2ccncc2)C(=O)O 1G-408S Cc1c(sc(n1)c2cccnc2)C(=O)N 1G-409S c1cc(ccc1C(=O)Nc2nccs2)Cl 1G-412S CC(C)CC(=O)O/N=C\1/c2cc(ccc2N(C1=O)Cc3c(cccc3Cl)Cl)Cl 1G-413S c1cc(c(c(c1)Cl)CN2c3ccc(cc3/C(=N/OC(=O)CCCCl)/C2=O)Cl)Cl 1G-414S Cc1c(sc(n1)c2cccnc2)C(=O)Nc3ccc(cc3)Cl 1G-415S Cc1c(sc(n1)c2cccnc2)C(=O)Nc3cccc(c3)C(F)(F)F 1G-416S Cc1c(sc(n1)c2cccnc2)C(=O)Nc3ccc(cc3)C(F)(F)F 1G-417S COC(=O)c1ccc(c(c1)[N+](=O)[O-])n2cccn2 1G-420S C/N=C(/c1cccc(c1)C(F)(F)F)\Nc2cccnc2 1G-421S c1cc(cnc1)NC(=N)c2ccc(cc2)Cl 1G-422S CC(C)/N=C(\c1ccc(cc1)Cl)/Nc2cccnc2 1G-423S c1ccc2c(c1)N(c3c(cccn3)S2)Cc4ccc(cc4)Br 1G-424S CC(=O)Nc1cccc(c1)c2nc(cs2)c3ccccc3 1G-425S COc1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)OC 1G-427S COC(=O)c1ccc(cc1)c2nc(cs2)c3cccc(c3)C(F)(F)F 1G-428S Cc1c(sc(n1)c2cccnc2)C(=O)Nc3ccc(cc3F)F 1G-430S COc1ccc(cc1)c2csc(n2)c3ccc(cc3)C(=O)O 1G-432S c1cc(cc(c1)C(F)(F)F)c2csc(n2)c3ccc(cc3)C(=O)O 1G-433S COC(=O)c1ccc(c(c1)[N+](=O)[O-])n2cncn2 1G-434S c1cc(ccc1c2nc(cs2)c3ccc(cc3)F)C(=O)Nc4ccc(cc4)F 1G-435S c1cc(ccc1c2nc(cs2)c3ccc(cc3)F)C(=O)Nc4ccc(cc4F)F 1G-436S COC(=O)c1c2ccc(cc2on1)[N+](=O)[O-] 1G-437S Cc1c(sc(n1)c2ccncc2)C(=O)Nc3ccc(cc3)Cl 1G-439S Cc1c(sc(n1)c2ccncc2)C(=O)Nc3ccc(cc3)Br 1G-440S c1ccc(cc1)c2csc(n2)c3cccc(c3)N 1G-444S C#CCN1c2ccccc2Sc3c1nccc3 1G-445S c1cc(cc(c1)C(F)(F)F)C(=N)Nc2cccnc2 1G-446S CNC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)OC 1G-447S c1cc(cc(c1)C(F)(F)F)c2csc(n2)c3ccc(cc3)C(=O)Nc4cccc(c4)C(F)(F)F 1G-448S c1cc(c(cc1C(=O)O)[N+](=O)[O-])n2ccnc2 1G-449S c1cnn(c1)c2ccc(cc2[N+](=O)[O-])C(=O)O 1G-450S c1ccc(cc1)C(=O)OC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 1G-900 CC(=O)CC(=O)Nc1c(cc(cn1)C(F)(F)F)Cl 1G-901 CC(=O)/C(=C\N(C)C)/C(=O)Nc1c(cc(cn1)C(F)(F)F)Cl 1G-903 Cc1c(cnc(n1)c2ccncc2)C(=O)Nc3c(cc(cn3)C(F)(F)F)Cl 1G-904 c1cc(cc(c1)C(F)(F)F)C(=O)OC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 1G-905 c1cc(ccc1C(=O)OC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 1G-906 COC(=O)c1c2c(sc1N)CN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 1G-907 CC(=O)OC1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 1G-908 COC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)Cl)CN(CC2)c4c(cc(cn4)C(F)(F)F)Cl 1G-909 Cc1c(cn(n1)c2ccc(cc2)F)C(=O)Nc3c(cc(cn3)C(F)(F)F)Cl 1G-910 c1ccc(c(c1)CON2C(=O)c3ccccc3C2=O)Br 1G-911 c1ccc(c(c1)CON2C(=O)c3ccccc3C2=O)[N+](=O)[O-] 1G-913 c1ccc2c(c1)C(=O)N(C2=O)OCc3ccc(cc3Cl)F 1G-914 c1ccc(c(c1)CON)Br.Cl 1G-915 c1ccc2c(c1)C(=O)N(C2=O)OCc3cc(ccc3Cl)Cl 1G-916 c1ccc2c(c1)C(=O)N(C2=O)OCc3cccc(c3Cl)Cl 1G-919 c1ccc(c(c1)CON2C(=O)c3ccccc3C2=O)C(F)(F)F 1G-921 COC(=O)c1c2c(sc1NC(=O)c3ccccc3Cl)CN(CC2)c4c(cc(cn4)C(F)(F)F)Cl 1G-922 CN(C)/C=N/c1c(c2c(s1)CN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)OC 1G-923 COC(=O)c1c2c(sc1/N=C/NOCc3ccc(cc3)Cl)CN(CC2)c4c(cc(cn4)C(F)(F)F)Cl 1G-924 c1cc(c(cc1F)Cl)CON.Cl 1G-925 c1cc(c(c(c1)Cl)Cl)CON.Cl 1G-926 c1cc(c(cc1Cl)CON)Cl.Cl 1G-927 c1ccc(c(c1)CON)[N+](=O)[O-].Cl 1G-928 c1c(cnc(c1Cl)N2CCc3c(sc(c3C#N)N)C2)C(F)(F)F 1G-929 COc1ccc(cc1)n2c(cc3c2CCCC3=O)c4ccccc4 1G-930 CN(C)/C=N/c1c(c2c(s1)CN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C#N 1G-931 CC(=O)c1ccc(cc1)C(=O)OC 1G-932 c1ccc(c(c1)CON)C(F)(F)F.Cl 1G-933 COc1ccccc1CON2C(=O)c3ccccc3C2=O 1G-936 c1ccc2c(c1)C(=O)N(C2=O)OCc3cccc(c3F)Cl 1G-937 Cc1ccc(cc1)CO/N=C\2/CCCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5 1G-938 COc1ccccc1CON.Cl 1G-939 c1ccc(cc1)C(=O)NC(=S)Nc2c(cc(cn2)C(F)(F)F)Cl 1G-940 COC(=O)c1c2c(sc1NS(=O)(=O)C)CN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 1G-941 c1c(cnc(c1Cl)NC(=S)N)C(F)(F)F 1G-942 c1cc(c(c(c1)Cl)F)CO[NH3+].[Cl-] 1G-943 CCOC(=O)/C(=N\O)/C(=O)C 1G-944 Cn1c(=O)c2c3c(sc2nc1S)CN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 1G-945 c1ccc2c(c1)C(=O)N(C2=O)OCc3c(cc(cn3)C(F)(F)F)Cl 1G-946 COC(=O)C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 1G-947 c1c(cnc(c1Cl)N2CCC(=CC(=O)NN)CC2)C(F)(F)F 1G-948 c1cc(ccc1NC(=O)NNC(=O)C=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 1G-951 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)NN)C(F)(F)F 1G-952 c1ccc(cc1)NC(=S)NNC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 1G-953 c1cc(ccc1C(=O)CC2=C(CCCC2=O)O)Cl 1G-954 Cc1cc\2c(o1)CC(C/C2=N/OCc3ccc(cc3)Cl)(C)C 1G-955 c1ccc(cc1)C(=O)CSC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl 1H-001 CC(C(=O)C)Oc1ccc(cc1)OC 1H-002 c1cc(c(cc1Cl)Cl)/C=C(/C#N)\c2[nH]nc(n2)CSc3c(cc(cn3)C(F)(F)F)Cl 1H-003 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1)OC 1H-005 c1cc(c(c(c1)Cl)CSc2c(cc(cn2)C#N)C#N)Cl 1H-006 c1c(cnc(c1C#N)SCc2c(cc(cn2)C(F)(F)F)Cl)C#N 1H-007 c1cc(ccc1CSc2c(cc(cn2)C#N)C#N)C(F)(F)F 1H-008 CC(=O)/C=C\c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)C)C 1H-009 c1c(cnc2c1c(c(s2)c3c(cc(cn3)C(F)(F)F)Cl)N)C#N 1H-010 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C/Nc4ccc(cc4)Cl)F 1H-013 CN1C(=O)C(=C(COc2ccccc2)N)C(=O)N(C1=O)C 1H-014 COC(=O)c1ccc(cc1)CSc2c(cc(cn2)C#N)C#N 1H-015 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C=O 1H-016 CN1C(=O)C(=C(COc2ccc(cc2)Cl)N)C(=O)N(C1=O)C 1H-019 COc1ccc(cc1)/C=C(/C#N)\c2[nH]nc(n2)CSc3c(cc(cn3)C(F)(F)F)Cl 1H-020 Cc1cc2ncc(cn2n1)C(=N)NNC(=O)CC#N 1H-021 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)/C=N/O 1H-022 c1ccc(cc1)OCC(=N)NNS(=O)(=O)c2ccccc2 1H-023 c1ccc(cc1)S(=O)(=O)NNC(=N)COc2ccc(cc2)Cl 1H-024 c1ccc2c(c1)C(CC(=O)O2)C(C#N)C(=O)N 1H-025 Cn1ccc2c1c(c3ccccc3c2NC(=O)Nc4ccccc4)C#N 1H-026 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C#N 1H-027 CN1C(=O)C(=C(COc2ccccc2Cl)N)C(=O)N(C1=O)C 1H-028 Cc1c2c(c(sc2ns1)c3c(cc(cn3)C(F)(F)F)Cl)N 1H-031 CN1C(=O)C(=C(COc2cccc(c2)Cl)N)C(=O)N(C1=O)C 1H-034 c1cc2c(cc1F)nc([nH]2)Cn3cncn3 1H-035 c1cc2c(cc1C(F)(F)F)nc([nH]2)Cn3cncn3 1H-036 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)/C=N/OCc3ccc(cc3)Cl 1H-037 CN(C)/C=N/C(=O)c1cnn(c1)c2c(cc(cn2)C(F)(F)F)Cl 1H-038 c1cc(ccc1OCC(=N)NNS(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl 1H-039 c1ccc(cc1)N2C(=O)CC(C2=O)Sc3c(cc(cn3)C(F)(F)F)Cl 1H-040 c1c(cnc(c1Cl)CSc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 1H-041 c1cc2c(cc1Cl)nc([nH]2)Cn3cncn3 1H-042 COc1cc(=O)n(nc1C(=N)[NH3+])c2cccc(c2)C(F)(F)F.[Cl-] 1H-043 CN(=CNC(=O)c1cnn(c1)c2c(cc(cn2)C(F)(F)F)Cl)=O 1H-044 c1cc(c(c(c1)Cl)CO/N=C/NC(=O)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 1H-045 c1c(cnc(c1Cl)CSC(=N)[NH3+])C(F)(F)F.[Br-] 1H-047 c1c(cnc(c1Cl)n2cc(cn2)c3nc[nH]n3)C(F)(F)F 1H-048 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)CO 1H-049 CCOC(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 1H-050 c1ccc(cc1)S(=O)(=O)NNC(=N)COc2cccc(c2)Cl 1H-051 COC(=O)c1c(ccs1)N2C(=O)CC(C2=O)Sc3c(cc(cn3)C(F)(F)F)Cl 1H-052 c1cc(c(cc1Cl)F)N2C(=O)CC(C2=O)Sc3c(cc(cn3)C(F)(F)F)Cl 1H-053 c1ccnc(c1)CNS(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl 1H-054 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)C#N 1H-055 c1ccc(cc1)/C=C/CSc2c(cc(cn2)C(F)(F)F)Cl 1H-056 CC(c1ccc(c(n1)O)C#N)Oc2ccc(cc2)OC 1H-057 c1cc(c(=O)[nH]c1)C(=O)Nc2ccncc2 1H-058 c1c(cnc(c1Cl)n2cncn2)C(F)(F)F 1H-059 c1cc(ccc1S(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl 1H-062 c1cc(ccc1F)S(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl 1H-063 c1ccc(cc1)S(=O)(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl 1H-066 CC(C(=O)C)Sc1c(cc(cn1)C(F)(F)F)Cl 1H-068 CC(C(=O)/C=C/N(C)C)Oc1cccnc1 1H-069 CCCNC(=O)c1c(snn1)S(=O)(=O)c2ccc(cc2)Cl 1H-301S CC(C)OC(=O)c1c(snn1)S(=O)(=O)c2ccc(cc2)Cl 1H-302S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3Cl)Cl 1H-303S c1cc(ccc1S(=O)(=O)c2c(nns2)C(=O)OC3CCCCC3)Cl 1H-305S CC(C)OC(=O)c1c(snn1)S(=O)c2ccc(cc2)Cl 1H-306S c1cc(ccc1S(=O)c2c(nns2)C(=O)OC3CCCCC3)Cl 1H-307S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccc(cc2)Cl)C 1H-308S c1cc2c(ccc(c2nc1)Oc3ccc(cc3[N+](=O)[O-])F)Cl 1H-309S CCOC(=O)/C(=N\Nc1cccc(c1)C(F)(F)F)/NC(=O)C 1H-311S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3ccccc3 1H-312S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3ccc(cc3)F 1H-313S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccc(cc2)Cl)CC#C)C 1H-314S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3ccc(cc3)Cl 1H-315S CCCNC(=O)c1nc(n(n1)c2ccc(cc2)[N+](=O)[O-])C 1H-316S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)N(C)C 1H-317S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)NC 1H-318S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3cccc(c3)C(F)(F)F 1H-319S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3ccc(cc3F)F 1H-320S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3ccccc3N4CCOCC4 1H-321S Cc1ccc(cc1)NC(=O)c2nc(n(n2)c3ccc(cc3)[N+](=O)[O-])C 1H-322S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccc(cc2)Cl)c3ccccc3 1H-323S Cc1nc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)Nc3ccc(cc3)OC 1H-324S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3ccccc3 1H-325S Cc1nc(nn1c2cccc(c2)C(F)(F)F)C(=O)O 1H-326S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)F 1H-328S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)Cl 1H-329S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 1H-330S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccccc2)c3ccccc3 1H-331S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3F)F 1H-332S CCOC(=O)/C(=N\Nc1ccc(cc1F)F)/NC(=O)C 1H-333S Cc1ccc(cc1)NC(=O)c2nc(n(n2)c3ccc(cc3)Cl)C 1H-334S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)Cc3ccc(cc3Cl)Cl)C 1H-336S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)OC 1H-337S Cc1nc(nn1c2ccc(cc2)Cl)C(=O)Nc3cc(cc(c3)Cl)Cl 1H-338S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)CC#C)C 1H-341S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)Cc3cccc(c3)C(F)(F)F)c4ccccc4 1H-342S Cc1nc(nn1c2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3Cl)Cl 1H-343S Cc1nc(nn1c2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3)Cl 1H-344S Cc1cccc(c1)S(=O)(=O)c2c(cc([nH]c2=O)c3ccccc3)C 1H-345S Cc1nc(nn1c2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3)F 1H-347S Cc1nc(nn1c2cccc(c2)C(F)(F)F)C(=O)Nc3cccc(c3)C(F)(F)F 1H-349S Cc1nc(nn1c2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(c(c3)F)F 1H-350S Cc1ccc(cc1)Cn2c(cc(c(c2=O)S(=O)(=O)c3cccc(c3)C)C)c4ccccc4 1H-351S CCn1c(cc(c(c1=O)S(=O)(=O)c2ccccc2C)C)C 1H-353S Cc1ccccc1S(=O)(=O)c2c(cc(n(c2=O)CC#C)C)C 1H-354S Cc1cccc(c1)S(=O)(=O)c2c(cc([nH]c2=O)C)C 1H-355S Cc1ccc(cc1)S(=O)(=O)c2c(c(c([nH]c2=O)C)C)C 1H-356S Cc1nc(nn1c2ccc(cc2F)F)C(=O)Nc3ccc(cc3)F 1H-358S Cc1nc(nn1c2ccc(cc2F)F)C(=O)Nc3ccc(cc3F)F 1H-359S Cc1ccccc1S(=O)(=O)c2c(cc(n(c2=O)CC(=C)C)C)C 1H-360S CCOC(=O)Cn1c(cc(c(c1=O)S(=O)(=O)c2ccccc2C)C)C 1H-361S Cc1nc(nn1c2ccc(cc2F)F)C(=O)Nc3ccc(cc3)Cl 1H-362S Cc1nc(nn1c2ccc(cc2F)F)C(=O)Nc3cccc(c3)C(F)(F)F 1H-363S COC(=O)C(c1ccccc1)NC(=O)CNS(=O)(=O)c2ccc(cc2)F 1H-364S COC(=O)C(c1ccccc1)NC(=O)CNS(=O)(=O)c2ccc(cc2)Cl 1H-366S CC(C(=O)OC)NC(=O)CNS(=O)(=O)c1ccc(cc1)F 1H-367S COC(=O)C(Cc1ccccc1)NC(=O)CNS(=O)(=O)c2ccc(cc2)F 1H-370S CC(C(=O)OC)NC(=O)CNS(=O)(=O)c1ccc(cc1)Br 1H-372S COC(=O)C(CCSC)NC(=O)CNS(=O)(=O)c1ccc(cc1)F 1H-373S c1cc(ccc1CSc2ccc(cc2)Cl)N 1H-402S c1cc(ccc1CSc2ccc(cc2)Cl)NC(=O)c3ccc(cc3)Cl 1H-403S c1cc(ccc1CSc2ccc(cc2)Cl)NC(=O)c3ccc(c(c3)Cl)Cl 1H-404S c1ccc(cc1)SCc2ccc(cc2)N 1H-406S c1cc(ccc1CSc2ccc(cc2)Br)NC(=O)c3ccc(cc3)Cl 1H-407S c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)Br)F 1H-408S c1ccc(cc1)C(=O)Nc2ccc(cc2)CSc3ccccc3 1H-409S c1ccc(cc1)SCc2ccc(cc2)NC(=O)c3cccc(c3)C(F)(F)F 1H-410S c1ccc(cc1)SCc2ccc(cc2)NC(=O)c3ccc(cc3)Cl 1H-411S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)Br 1H-412S c1cc(ccc1CSc2ccc(cc2)Br)NC(=O)c3cc(cc(c3)Cl)Cl 1H-413S c1cc(ccc1CSc2ccc(cc2)F)N 1H-415S c1ccc(cc1)SCc2ccc(cc2)NC(=O)c3cc(cc(c3)Cl)Cl 1H-417S c1ccc(cc1)SCc2ccc(cc2)NC(=O)c3ccc(cc3F)F 1H-418S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)CSc3ccccc3 1H-420S c1ccc(cc1)SCc2ccc(cc2)NC(=O)c3ccc(cc3)C(F)(F)F 1H-421S c1ccc(cc1)SCc2ccc(cc2)NS(=O)(=O)c3ccc(cc3)F 1H-422S c1ccc(cc1)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)Cl 1H-423S c1cc(ccc1CSc2ccc(cc2)Cl)NC(=O)c3cc(cc(c3)Cl)Cl 1H-424S c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)Cl)F 1H-425S c1cc(ccc1CSc2ccc(cc2)Cl)NC(=O)c3ccc(cc3)C(F)(F)F 1H-426S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)Cl 1H-805S CCOC(=O)c1cc(c(=O)[nH]c1NNC(=O)Nc2ccc(cc2)Cl)C(=O)OCC 1H-900 CCOC(=O)c1cc(c(=O)[nH]c1NNC(=O)C)C(=O)OCC 1H-901 CCOC(=O)c1cc(c(=O)[nH]c1N/N=C/N(C)C)C(=O)OCC 1H-902 c1c(cnc(c1Cl)N2CCN(CC2)CCNc3c[nH]c(=O)[nH]c3=O)C(F)(F)F 1H-905 COC(=O)C(c1ccccc1)/N=C/c2ccccc2 1H-906 CCOC(=O)NCCNc1c(cc(cn1)C(F)(F)F)Cl 1H-907 COC(=O)C(c1ccccc1)/N=C/c2ccc(cc2)Cl 1H-909 COC(=O)C1(C2C(C(N1)c3ccccc3)C(=O)N(C2=O)c4ccc(cc4)Cl)c5ccccc5 1H-911 COC(=O)C1(C2C(C(N1)c3ccc(cc3)Cl)C(=O)N(C2=O)c4ccc(cc4)Cl)c5ccccc5 1H-912 COc1cc(ccc1OCc2ccc(cc2)F)C=O 1H-913 c1c(cnc(c1Cl)N2CCN(CC2)c3c[nH]c(=O)[nH]c3=O)C(F)(F)F 1H-914 C/[N+](=C/c1ccc(c(c1)OC)OCc2ccc(cc2)F)/[O-] 1H-915 COC(=O)C(c1ccccc1)/N=C/c2ccccc2Cl 1H-916 COC(=O)C1(C2C(C(N1)c3cccc(c3)Cl)C(=O)N(C2=O)c4ccc(cc4)Cl)c5ccccc5 1H-917 c1ccc2c(c1)ccc(c2C=O)OCc3ccc(cc3Cl)Cl 1H-918 COC(=O)C1(C2C(C(N1)c3ccccc3Cl)C(=O)N(C2=O)c4ccc(cc4)Cl)c5ccccc5 1H-919 C/[N+](=C/c1c2ccccc2ccc1OCc3ccc(cc3Cl)Cl)/[O-] 1H-920 CCOC(=O)c1cc(c(nc1NN=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)O)C(=O)OCC 1H-921 c1cc(ccc1CCNc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N 1H-922 CCOC(=O)NC(=O)/C(=C\Nc1c(cc(cc1SCC(=O)OC)Cl)F)/C#N 1H-923 CN1C(C2C(O1)C(=O)N(C2=O)Cc3ccccc3)c4ccc(c(c4)OC)OCc5ccc(cc5)F 1H-924 CC(=O)CC(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 1H-925 CCOC(=O)NC(=O)/C(=C\Nc1ccc(cc1Cl)Cl)/C#N 1H-926 CC(=O)/C(=C\N(C)C)/C(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 1H-927 C=CCOc1ccccc1/C=C\2/C(=NN(C2=O)c3ccccc3)c4ccccc4 1H-928 C=CCOc1ccc2ccccc2c1/C=C\3/C(=NN(C3=O)c4ccccc4)c5ccccc5 1H-929 CN1C(=O)C(=Cc2c3ccccc3ccc2OCC=C)C(=O)N(C1=O)C 1H-930 c1ccc(cc1)c2c3c(n(n2)c4ccccc4)OC[C@@H]5[C@H]3c6c7ccccc7ccc6OC5 1H-931 COc1ccc(cc1)OCCN2C(=O)c3ccccc3C2=O 1H-933 CN1C(C(CO1)S(=O)(=O)c2ccccc2)c3ccc(c(c3)OC)OCc4ccc(cc4)F 1H-934 C/C(=C\C(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)/N3CCN(CC3)c4ccc(cc4)Cl 1H-935 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/c2cn(c(=O)n(c2=O)C)C 1H-936 Cn1c(=O)c2c(n(c1=O)C)OC[C@@H]3[C@H]2c4c5ccccc5ccc4OC3 1H-937 CN1C(=O)C(=Cc2ccccc2OCC=C)C(=O)N(C1=O)C 1H-938 Cn1c(=O)c2c(n(c1=O)C)OCC3C2c4ccccc4OC3 1H-939 CN1CCN(CC1)C2=CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 1H-940 CCOC(=O)NC(=O)/C(=C\Nc1ccc(cc1)Cl)/C(=O)C 1H-942 CC(=O)c1cn(c(=O)[nH]c1=O)c2ccc(cc2)Cl 1H-943 CCOC(=O)Cn1c(=O)ccn(c1=O)c2c(cc(cn2)C(F)(F)F)Cl 1H-945 COc1ccc(cc1)/C=C\2/C(=NN(C2=O)c3ccccc3)c4ccccc4 1H-947 c1c(cnc(c1Cl)NC2=NNC(=O)CN2)C(F)(F)F 1H-949 CCOC(=O)C1=NOC(C1)COc2ccc3ccccc3c2C=O 1H-950 CCOC(=O)C1=NOC(C1)COc2ccc3ccccc3c2/C=N\OCc4ccc(cc4)Cl 1H-953 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/c2cn(c(=O)[nH]c2=O)c3ccc(cc3)Cl 1H-954 c1cc(cc(c1)NC(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 1H-955 CC(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)Br)c3ccc(cc3)Cl 1H-956 CN1CCC(=CC1)N2CCCCC2 1H-957 CN(C)/C=N/C(=O)C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 1H-958 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC=C 1H-959 CN1CCN(CC1)C2=CCN(CC2)C 1H-960 CCOC(=O)C1=NOC(C1)CNC(=O)c2c(onc2c3ccccc3Cl)C 1H-961 COc1ccc(cc1)n2cc(c(=O)n(c2=O)Cc3ccc(cc3)F)C#N 1H-962 c1cc(cc(c1)C(F)(F)F)CON/C=N/C(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 1H-963 c1cc(ccc1C(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl 1H-964 c1ccc(cc1)C(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 1H-965 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 1H-966 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC3CC(=NO3)C(=O)NCC=C 1H-967 c1ccc2c(c1)C(=O)N(C2=O)CCOc3cccc(c3)C(F)(F)F 1H-968 C/[N+](=C\c1cccc(c1)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)/[O-] 1H-969 c1cc(ccc1n2cc(c(=O)n(c2=O)Cc3c(cc(cn3)C(F)(F)F)Cl)C#N)Cl 1H-971 c1cc(ccc1CN(CCNc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)C(F)(F)F)Cl 1H-972 C/C(=N/Nc1c(cc(cn1)C(F)(F)F)Cl)/c2ccc(cc2)n3cc(c(=O)[nH]c3=O)C#N 1H-974 c1c(cnc(c1Cl)NCCN(CCO)c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 1H-976 c1cc(ccc1/C(=N\Nc2ccc(nn2)Cl)/c3c(cc(cn3)C(F)(F)F)Cl)Cl 1J-001 CN(C)c1nnnn1c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 1J-002 CN(C)c1nnnn1c2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl 1J-003 CN(C)c1nnnn1c2ccccc2Oc3c(cc(cn3)C(F)(F)F)Cl 1J-004 COc1ccc(cc1)C(c2c(cc(cn2)C(F)(F)F)Cl)O 1J-006 c1cc(nc(c1)Nc2c(cc(cn2)C(F)(F)F)Cl)N 1J-007 c1cc(cnc1)/C(=N/OS(=O)(=O)c2ccc(cc2Cl)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 1J-008 Cc1ccc(cc1)S(=O)(=O)O/N=C(/c2cccnc2)\c3c(cc(cn3)C(F)(F)F)Cl 1J-009 Cn1ccnc1C(=O)NNc2ccccc2 1J-011 Cn1ccnc1C(=O)N 1J-012 Cn1ccnc1C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl 1J-014 CC(=O)c1ccc(cc1)Sc2ccccc2 1J-015 Cn1ccnc1C(=O)NNC2CCS(=O)(=O)C2 1J-016 CC(=O)c1ccc(cc1)S(=O)c2ccccc2 1J-017 CC(=O)c1ccc(cc1)S(=O)(=O)c2ccccc2 1J-018 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)n(n2)C(=O)Nc4ccc(cc4Cl)Cl 1J-019 CCOC(=O)Cn1c(nnn1)N(C)C 1J-020 c1ccc(cc1)NC(=O)Nc2cccc(n2)Nc3c(cc(cn3)C(F)(F)F)Cl 1J-021 CC(C)(CNc1c(cc(cn1)C(F)(F)F)Cl)S 1J-022 CN(C)c1nnnn1CC(=O)N 1J-023 CN(C)c1nnnn1CC(=O)NN 1J-024 c1cc(cc(c1)C(F)(F)F)C(C#N)N2CCOCC2 1J-026 CN(C)/C=C/C(=O)c1ccc(cc1)S(=O)c2ccccc2 1J-028 CN(C)/C=C/C(=O)c1ccc(cc1)S(=O)(=O)c2ccccc2 1J-029 CN(C)/C=C/C(=O)c1ccc(cc1)Sc2ccccc2 1J-030 CN(C)c1nnnn1CC(=O)N/C=N/OC 1J-031 c1cc(cc(c1)NC(=O)Nc2cccc(n2)Nc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 1J-035 c1cc(nc(c1)NC(=O)Nc2ccc(cc2)Cl)Nc3c(cc(cn3)C(F)(F)F)Cl 1J-036 c1ccc(cc1)/C=C/C(C#N)N2CCOCC2 1J-037 CC(C)(CNc1c(cc(cn1)C(F)(F)F)Cl)Sc2c(cc(cn2)C(F)(F)F)Cl 1J-039 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)O 1J-042 CC(=O)c1ccc(s1)Cc2c(cc(cn2)C(F)(F)F)Cl 1J-043 C/C(=N/O)/c1ccc(s1)Cc2c(cc(cn2)C(F)(F)F)Cl 1J-047 C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl 1J-049 c1ccc(cc1)/C=C/C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3 1J-050 c1cc(ccc1c2c3c(cc(cn3)C(F)(F)F)n(n2)c4ccc(nn4)Cl)Cl 1J-051 C/C(=N\N=C(\c1sc(cc1)Cc2ncc(cc2Cl)C(F)(F)F)/C)/c3sc(cc3)Cc4ncc(cc4Cl)C(F)(F)F 1J-052 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 1J-054 COc1ccc(cc1)NC(=O)c2ccccc2CC[N+](=O)[O-] 1J-055 c1cc(ccc1C(C#N)c2c(cc(cn2)C(F)(F)F)Cl)O 1J-056 c1ccc(cc1)C(CNCc2cccc(c2)C(F)(F)F)(c3ccccc3)O.Cl 1J-301S c1ccc(cc1)c2nc(cc(n2)O)O 1J-304S c1ccc(cc1)C(CNCc2ccc(c(c2)Cl)Cl)(c3ccccc3)O 1J-305S COc1ccc(cc1OC)CNCC(c2ccccc2)(c3ccccc3)O 1J-306S COc1cnc(nc1O)c2ccccc2 1J-310S COc1cnc(nc1O)c2ccccn2 1J-311S c1ccc(cc1)/C(=N\OCC2OCCO2)/C#N 1J-313S CC(C)NCC(c1ccccc1)(c2ccccc2)O 1J-314S c1ccc(cc1)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-315S Cc1ccc(cc1)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-316S CCCCCC(C)OC(=O)COc1ccc(c2c1nccc2)Cl 1J-317S c1cc(ccc1CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 1J-318S c1cc(ccc1CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)F 1J-319S c1cc(cc(c1)C(F)(F)F)C[NH2+]CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O.[Cl-] 1J-320S c1ccc(c(c1)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)F 1J-321S c1ccc(c(c1)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)Cl 1J-322S COc1cnc(nc1Cl)c2ccccn2 1J-324S COc1cccc(c1)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-325S COc1ccc(cc1)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-326S c1cc(cc(c1)Cl)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-327S c1ccc(cc1)c2nc(cc(n2)Cl)Cl 1J-330S CS(=O)(=O)c1ccc(c(c1)Cl)c2c3c(n[nH]2)CCC3 1J-331S c1cc(ccc1C(CNCc2ccc(cc2Cl)Cl)(c3ccc(cc3)Cl)O)Cl 1J-332S c1cc(ccc1C(CNCc2ccc(c(c2)Cl)Cl)(c3ccc(cc3)Cl)O)Cl 1J-333S COc1ccccc1CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-334S COc1ccc(cc1OC)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-335S c1ccc2c(c1)[nH]c(n2)CNS(=O)(=O)c3ccc(cc3)F 1J-338S CNCC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 1J-339S CCCCNCC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 1J-340S c1cc(ccc1C(CN)(c2ccc(cc2)Cl)O)Cl.Cl 1J-341S c1ccnc(c1)CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O.Cl.Cl 1J-342S CCC(C)NCC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 1J-343S c1cc(ccc1C(CN2CCOCC2)(c3ccc(cc3)Cl)O)Cl 1J-344S CC(C)(C)NCC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 1J-345S CC(C)NCC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 1J-346S CCN(CC)CCNCC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 1J-347S CC1CN(CC(O1)C)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-352S C=CCNCC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 1J-353S COc1cnc(nc1Sc2ccc(cc2)Cl)c3ccccn3 1J-355S CN1CCN(CC1)CC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O 1J-356S c1cc(cc(c1)Cl)N2CCN(CC2)CC(c3ccc(cc3)Cl)(c4ccc(cc4)Cl)O 1J-357S CC(c1[nH]c2ccccc2n1)NS(=O)(=O)c3ccc(cc3)Cl 1J-359S COc1cnc(nc1Sc2cccc(c2)C(F)(F)F)c3ccccn3 1J-360S COc1ccc(cc1)Sc2c(cnc(n2)c3ccccn3)OC 1J-361S COc1cnc(nc1Sc2ccc(cc2)F)c3ccccn3 1J-362S COc1cnc(nc1Sc2ccccc2)c3ccccn3 1J-363S Cc1cc2c(cc1C)nc([nH]2)/C=C/c3ccccc3 1J-502S CCOC(=O)c1cnc(nc1c2ccccc2)c3ccccc3 1J-510S CCOC(=O)c1nc(n(n1)c2ccc(c(c2)Cl)Cl)C(Cl)(Cl)Cl 1J-512S Cc1cc2c(cc1C)n(c(n2)/C=C/c3ccccc3)Cc4cccc(c4)F 1J-513S Cc1cc2c(cc1C)n(c(n2)/C=C/c3ccccc3)Cc4ccc(cc4)C(C)(C)C 1J-514S Cc1cc2c(cc1C)n(c(n2)/C=C/c3ccccc3)Cc4ccc(c(c4)Cl)Cl 1J-515S Cc1cc2c(cc1C)n(c(n2)/C=C/c3ccccc3)Cc4cccc(c4)OC 1J-516S Cc1cc2c(cc1C)n(c(n2)/C=C/c3ccccc3)Cc4ccc(cc4)C#N 1J-517S Cc1cc2c(cc1C)n(c(n2)/C=C/c3ccccc3)Cc4ccc(cc4)Cl 1J-518S CCOC(=O)Cn1c2cc(c(cc2nc1/C=C/c3ccccc3)C)C 1J-519S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)O 1J-521S c1ccc2c(c1)[nH]c(n2)/C=C/c3ccc(cc3Cl)Cl 1J-526S Cc1cc2c(cc1C)n(c(n2)/C=C/c3ccccc3)Cc4ccc(cc4)C(=O)OC 1J-530S c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccc(cc4Cl)Cl 1J-532S Cc1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccc(cc4Cl)Cl 1J-533S c1ccc2c(c1)nc(n2Cc3ccc(cc3)C(F)(F)F)/C=C/c4ccc(cc4Cl)Cl 1J-534S COC(=O)c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccc(cc4Cl)Cl 1J-535S Cc1ccc(cc1)/C=C/c2nc3ccccc3n2Cc4cccc(c4)C(F)(F)F 1J-536S Cc1ccc(cc1)/C=C/c2nc3ccccc3n2Cc4c(cccc4Cl)F 1J-537S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4ccc(cc4)F 1J-538S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4ccc(cc4)Cl 1J-539S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4cccc(c4)Cl 1J-540S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4ccccc4 1J-541S CCOC(=O)Cn1c2ccccc2nc1/C=C/c3ccc(cc3)C 1J-542S c1ccc2c(c1)nc(n2Cc3cccc(c3)C#N)/C=C/c4ccc(cc4Cl)Cl 1J-543S c1ccc2c(c1)nc(n2Cc3cccc(c3)Cl)/C=C/c4ccc(cc4Cl)Cl 1J-544S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4cccc(c4)C(F)(F)F 1J-550S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4ccc(cc4)Br 1J-552S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4cc(cc(c4)Cl)Cl 1J-553S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4ccc(cc4)C(F)(F)F 1J-555S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4ccc(cc4)OC(F)(F)F 1J-556S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)Nc4ccc(c(c4)F)F 1J-557S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)NCc4ccc(cc4)Cl 1J-558S c1ccc(cc1)c2cc(nc(n2)c3cccnc3)C(=O)Nc4cccc(c4)Cl 1J-565S CCCO/N=C/C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 1J-900 c1cnc(nc1)Sc2cc(=O)n(c(=O)[nH]2)CCNc3c(cc(cn3)C(F)(F)F)Cl 1J-901 c1cc(c(cc1Cl)Cl)NC(=O)C(/C=N/OCC(=O)N2CCOCC2)C(=O)Nc3ccc(cc3Cl)Cl 1J-902 CN(C)/C=C/C(=O)c1ccc2c(c1)c(on2)c3ccc(cc3)F 1J-903 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2ccc(cc2)Cl 1J-904 COC(=O)CSc1cc(=O)n(c(=O)[nH]1)CCNc2c(cc(cn2)C(F)(F)F)Cl 1J-906 CC(C)(C)ONC=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 1J-907 c1cc(cc(c1)F)n2ccc(n2)c3ccc4c(c3)c(on4)c5ccc(cc5)F 1J-908 c1ccc(c(c1)n2ccc(n2)c3ccc4c(c3)c(on4)c5ccc(cc5)F)F 1J-909 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC=C)S(=O)(=O)c2ccc(cc2)Cl 1J-910 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)/C(=C\c4ccc(cc4)Cl)/C#N 1J-911 c1ccc(c(c1)/C=C(/C#N)\c2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 1J-912 CN(C)/C=N/C(=O)NN(C)c1c(cc(cn1)C(F)(F)F)Cl 1J-913 COCCNC=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 1J-914 c1c[nH]c(=O)c(c1NCCNc2c(cc(cn2)C(F)(F)F)Cl)C#N 1J-915 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)/N=C/NOCc2ccc(cc2)[N+](=O)[O-] 1J-916 COC(=O)C(/C=N/Nc1c(cc(cn1)C(F)(F)F)Cl)c2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl 1J-918 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C(C2=O)ONC3(C(=O)OC)C(=O)OC 1J-920 CC1(NC(=O)N(N1)c2ccccc2F)c3ccc4c(c3)c(on4)c5ccc(cc5)F 1J-922 CC1(NC(=O)N(N1)c2cccc(c2)F)c3ccc4c(c3)c(on4)c5ccc(cc5)F 1J-923 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)/N=C/NOCc2ccc(cc2Cl)Cl 1J-924 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)/N=C/NOCc2ccc(cc2)OC 1J-925 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)/N=C/NOC 1J-926 CCOC(=O)C1=NOC2C1C(=O)N(C2=O)N(C)c3c(cc(cn3)C(F)(F)F)Cl 1J-927 c1ccc(cc1)CN2C(=O)CC(C2=O)Sc3ccc(cc3)Cl 1J-928 CN1C(C2C(O1)C(=O)N(C2=O)N(C)c3c(cc(cn3)C(F)(F)F)Cl)c4ccc(cc4)OC 1J-930 CC(=O)c1c(ccs1)Cl 1J-931 c1csc(c1Cl)C(=O)O 1J-932 c1ccc(cc1)CN2C(=O)CC(C2=O)(Sc3ccc(cc3)Cl)Cl 1J-933 c1cc(ccc1C(=O)O)N2CCN=C2S 1J-934 c1ccc(cc1)CN2C(=O)C=C(C2=O)Sc3ccc(cc3)Cl 1J-936 c1ccc(cc1)CN2C(=O)C(C(C2=O)Sc3ccc(cc3)Cl)Sc4ccc(cc4)Cl 1J-938 COc1ccc(cc1)NC2C(C(=O)N(C2=O)Cc3ccccc3)Sc4ccc(cc4)Cl 1J-939 CN(C)/C=C/C(=O)c1c(ccs1)Cl 1J-940 c1cc(ccc1C(=O)O)N2CCN=C2Sc3c(cc(cn3)C(F)(F)F)Cl 1J-941 c1ccc(cc1)CN2C(=O)C(C(C2=O)Sc3ccc(cc3)Cl)N4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 1J-942 c1cc(c(cc1Cl)Cl)NC(=O)C(F)(F)F 1J-944 c1ccnc(c1)CC2C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 1J-948 c1cc(ccc1N/C=C/C(=O)c2c(ccs2)Cl)OC(F)(F)F 1J-949 c1ccc2c(c1)c3c([nH]2)CCC4(C3)OCCO4 1J-952 Cc1ccc(cc1)SC2CC(=O)N(C2=O)c3ccc(cc3)Cl 1J-953 CN(c1ccc(cc1Cl)Cl)C(=O)CC(=O)N(C)c2ccc(cc2Cl)Cl 1J-954 Cc1ccc(cc1)SC2=CC(=O)N(C2=O)c3ccc(cc3)Cl 1J-955 c1cc(ccc1c2c3cc(ccc3no2)C(=O)/C=C/NNc4c(cc(cn4)C(F)(F)F)Cl)F 1J-956 CO/N=C/CC(=O)Oc1ccc(cc1Cl)Cl 1K-001 c1ccc(c(c1)NC(=O)CC(=O)O)Oc2c(cc(cn2)C(F)(F)F)Cl 1K-002 CCO/C=N/C(=C(/C#N)\N)/C#N 1K-003 c1cc(c(cc1NC(=O)CC(=O)O)Cl)Oc2ccc(cn2)C(F)(F)F 1K-004 CCOC(=O)c1c(c(on1)C)C(=O)CBr 1K-005 c1ccc(cc1)NS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 1K-010 Cc1c(c(no1)C(=O)NN)c2csc(n2)c3csc(n3)C 1K-011 Cc1c(c(no1)C(=O)N/N=C/c2ccc(cc2)Cl)c3csc(n3)c4csc(n4)C 1K-012 Cc1ccc(cc1)NS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 1K-013 Cc1cc(cc(c1)NS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl)C 1K-014 COc1ccc(cc1)NS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 1K-015 c1ccc2c(c1)nc(c(n2)Oc3ccc(cc3)Cl)C(F)(F)F 1K-016 CCCNS(=O)(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 1K-017 COCCNS(=O)(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 1K-018 CC(C)(CNS(=O)(=O)C)SCc1ccc(cc1)Cl 1K-019 c1ccc2c(c1)nc(c(n2)Oc3ccc(cc3)[N+](=O)[O-])C(F)(F)F 1K-020 COC(=O)c1ccc(cc1)Oc2c(nc3ccccc3n2)C(F)(F)F 1K-021 c1ccc2c(c1)nc(c(n2)Sc3ccc(cc3)Cl)C(F)(F)F 1K-022 c1cc(c(cc1Cl)Cl)CO/N=C/CC(=O)Oc2ccc(cc2Cl)Cl 1K-023 COC(=O)CSc1c(nc2ccccc2n1)C(F)(F)F 1K-024 CCOC(=O)CNC(=S)NNc1c(cc(cn1)C(F)(F)F)Cl 1K-027 c1ccc(cc1)NC(=O)CSc2c(nc3ccccc3n2)C(F)(F)F 1K-028 CCOC(=O)CNC(=S)NN 1K-029 CCOC(=O)CNC(=S)Nc1ccc(cc1)Cl 1K-030 c1ccc2c(c1)nc(c(n2)NCc3cccnc3)C(F)(F)F 1K-031 c1ccc(c(c1)C(=O)c2[nH]ccn2)Cl 1K-032 COC(=O)c1c(onc1c2ccccc2Cl)/C=C/c3cnc(c4c3onc4c5ccccc5Cl)O 1K-033 COC(=O)c1c(onc1c2ccccc2Cl)/C=C/c3cnc(c4c3onc4c5ccccc5Cl)Cl 1K-034 c1cc(ccc1N2C(=O)CNC2=S)Cl 1K-035 Cc1ccc(cc1)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 1K-037 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)F)/[N+](=O)[O-] 1K-038 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2cccc(c2)C(F)(F)F)/[N+](=O)[O-] 1K-039 Cc1c(cccc1Cl)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 1K-040 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)Br)/[N+](=O)[O-] 1K-041 COc1ccc(cc1)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 1K-042 Cc1cccc(c1C)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 1K-043 c1ccc2c(c1)nc(c(n2)NN)C(F)(F)F 1K-044 CN(c1c(nc2ccccc2n1)C(F)(F)F)N 1K-045 CN(C)/C=C\1/C(=O)N(C(=S)N1)c2ccc(cc2)Cl 1K-046 c1cc(ccc1/C=C\2/C(=O)N(C(=S)N2)c3ccc(cc3)Cl)Cl 1K-047 CO/N=C/C(C#N)c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F 1K-048 COc1ccc(cc1)/C=C\2/C(=O)N(C(=S)N2)c3ccc(cc3)Cl 1K-049 CCOC(=O)CNC(=S)Nc1ccc(cc1)C(F)(F)F 1K-050 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2F)F)/[N+](=O)[O-] 1K-051 c1ccc(cc1)Oc2ccc(cc2)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c3ccccc3 1K-052 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(c(c2)Cl)Cl)/[N+](=O)[O-] 1K-053 c1c(cnc(c1Cl)N/N=C/Nc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 1K-054 c1ccc(c(c1)C(=O)Nc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 1K-055 Cc1cccc(c1)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 1K-056 COC(=O)c1cccc(c1)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 1K-057 Cc1ccccc1S(=O)(=O)c2c(cc(nc2SCC(C)C)C)C 1K-301S Cc1ccc(c(c1S(=O)(=O)c2c(cc([nH]c2=O)C)C)C)Cl 1K-302S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4ccccc4Cl 1K-304S Cc1cccc(c1)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)C)C 1K-305S Cc1ccc(cc1)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)C)C 1K-306S Cc1ccc(c(c1)C)S(=O)(=O)c2c(cc([nH]c2=O)C)C 1K-307S c1cc(cc(c1)C(F)(F)F)c2c(cc(nc2Cl)O)O 1K-311S Cc1cc(nc(c1S(=O)(=O)c2cc(c(cc2C)Cl)C)Cl)C 1K-312S Cc1ccc(c(c1)C)S(=O)(=O)c2c(cc(nc2Cl)C)C 1K-313S Cc1ccccc1Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)C)C 1K-314S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4c(cccc4Cl)Cl 1K-315S Cc1ccc(cc1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)C)C 1K-316S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4cccc(c4)F 1K-317S Cc1cc(nc(c1S(=O)(=O)c2cc(c(cc2C)Cl)C)OCC(C)C)C 1K-318S Cc1ccc(c(c1)C)S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C 1K-319S Cc1ccc(c(c1)S(=O)(=O)c2c(cc([nH]c2=O)C)C)C 1K-320S CCn1c2cc(c(cc2nc1c3cccnc3Cl)C)C 1K-321S CCn1c2cc(c(cc2nc1c3ccc[nH]c3=O)C)C 1K-322S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4cccc(c4)F 1K-323S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4ccccc4F 1K-324S Cc1ccc(c(c1)S(=O)(=O)c2c(cc(nc2Cl)C)C)C 1K-326S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4cccc(c4)C(F)(F)F 1K-327S Cc1ccc(c(c1)S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C)C 1K-328S Cn1c(c(c(n1)C(F)(F)F)C#N)N(C)NC(=O)c2cccc(c2)C(F)(F)F 1K-329S Cn1c(c(c(n1)C(F)(F)F)C#N)N(C)NC(=O)c2ccc(cc2Cl)Cl 1K-330S CC(=O)NN(C)c1c(c(nn1C)C(F)(F)F)C#N 1K-331S Cc1c(snn1)C(=O)N(C)C 1K-333S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4c(cccc4Cl)F 1K-334S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OCC#C)C)C 1K-335S CCCn1c2cc(c(cc2nc1c3ccc[nH]c3=O)C)C 1K-336S Cc1c(snn1)C(=O)NC2CCCCC2 1K-337S Cc1c(snn1)C(=O)Nc2cccc(c2)C(F)(F)F 1K-338S Cc1c(snn1)C(=O)Oc2cccc(c2)C(F)(F)F 1K-339S c1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)C(F)(F)F 1K-340S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4ccc(cc4)C(C)(C)C 1K-341S CCCCc1cc(c(c(=O)[nH]1)S(=O)(=O)c2ccccc2C)C 1K-342S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4ccc(c(c4)Cl)Cl 1K-343S Cc1cc2c(cc1C)n(c(n2)c3ccc(=O)[nH]c3)Cc4ccccc4 1K-346S Cc1cc2c(cc1C)n(c(n2)c3ccc(=O)[nH]c3)Cc4ccc(cc4)C(F)(F)F 1K-347S CCc1ccccc1S(=O)(=O)c2c(cc(nc2Cl)C)C 1K-350S c1ccc2c(c1)c(=O)n(c(n2)c3cccc(c3)Cl)O 1K-501S Cc1ccc(cc1)c2nc3ccccc3c(=O)n2O 1K-502S COc1ccc(cc1)c2nc3ccccc3c(=O)n2O 1K-503S c1ccc2c(c1)c(=O)n(c(n2)c3ccccc3Cl)O 1K-506S c1ccc2c(c1)c(=O)n(c(n2)c3ccc(cc3Cl)Cl)O 1K-507S c1ccc2c(c1)c(=O)n(c(n2)c3ccc(cc3)C#N)O 1K-508S c1ccc(cc1)c2nc3cc(ccc3c(=O)n2O)Cl 1K-509S c1cc(ccc1c2nc3cc(ccc3c(=O)n2O)Cl)[N+](=O)[O-] 1K-510S c1ccc(c(c1)c2nc3cc(ccc3c(=O)n2O)Cl)Cl 1K-511S c1cc(ccc1c2nc3cc(ccc3c(=O)n2O)Cl)Cl 1K-513S c1ccc(c(c1)c2nc3cc(ccc3c(=O)n2O)Cl)C(=O)O 1K-514S c1cc(c(cc1c2nc3cc(ccc3c(=O)n2O)Cl)Cl)Cl 1K-516S Cc1ccccc1c2nc3ccccc3c(=O)n2O 1K-519S c1cc(ccc1C#N)c2nc3cc(ccc3c(=O)n2O)Cl 1K-521S Cn1c(cc(nc1=O)C(=O)O)O 1K-522S COc1ccc(cn1)NC(=O)c2ccc(cc2)Cl 1K-525S c1ccc(cc1)c2nc3ccc(cc3c(=O)n2O)Br 1K-528S c1cc(cc(c1)C(F)(F)F)c2nc3ccc(cc3c(=O)n2O)Br 1K-529S c1cc(c(cc1c2nc3ccc(cc3c(=O)n2O)Br)Cl)Cl 1K-530S COc1ccc(c[n+]1[O-])NC(=O)c2ccc(cc2)Cl 1K-531S c1cc(c(cc1Cl)Cl)c2nc3ccc(cc3c(=O)n2O)Br 1K-536S Cn1c(cc(nc1=O)C(=O)Nc2ccccc2)O 1K-550S Cn1c(cc(n1)c2ccccc2)O 1K-553S Cc1cc(n(n1)c2ccc(cc2F)F)c3c(nn(c3O)c4nc(cs4)c5c(ccs5)Cl)C 1K-900 Cc1cc(n(n1)c2ccc(cc2Cl)Cl)c3c(nn(c3O)c4nc(cs4)c5c(ccs5)Cl)C 1K-901 CC(=O)NC(=N)N 1K-902 c1ccc2c(c1)C(=O)N(C2=O)OCc3ccc(c(c3)Cl)Cl 1K-903 CCOC(=O)C1=NOC(C1)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 1K-904 Cc1ccc(cc1)C(=O)Nc2cc3c(n(c2=O)Cc4cccc(c4)OC)CCCC3=O 1K-905 CN1C(CC(O1)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)c4ccc(cc4)OC 1K-906 c1cc(ccc1C(=O)Nc2cc3c(n(c2=O)CCNc4c(cc(cn4)C(F)(F)F)Cl)CCCC3=O)Cl 1K-907 Cc1ccc(cc1)C(=O)Nc2cc(c(n(c2=O)Cc3ccccc3)C)C(=O)C 1K-908 c1ccc(cc1)C(=O)Nc2cc3c(n(c2=O)N4CCCCC4)CCCC3=O 1K-909 Cc1cc(n2cc(c(c2n1)C(=O)O)c3c(ccs3)Cl)C 1K-910 c1cc(cc(c1)Cl)Cn2c3c(cc(c2=O)NC(=O)c4cccc(c4)Cl)C(=O)CCC3 1K-911 Cc1c(cc(c(=O)n1CCc2ccc(c(c2)OC)OC)NC(=O)c3ccc(cc3)Cl)C(=O)C 1K-912 Cc1c(cc(c(=O)n1Cc2ccco2)NC(=O)c3ccc(cc3)Cl)C(=O)C 1K-913 c1cc(cc(c1)Cl)C(=O)Nc2cc3c(n(c2=O)Cc4ccco4)CCCC3=O 1K-914 CC(C)(/C=N/OCc1ccc(cc1)Cl)Sc2ccccc2 1L-001 Cc1ccc(cc1)SC(C)(C)/C=N/OCc2ccc(cc2)Cl 1L-002 CC(C)(/C=N/OCc1ccc(cc1)Cl)Sc2ccc(cc2)Cl 1L-003 CC(c1ccnc2n1nc(n2)N)Oc3ccc(cc3F)F 1L-004 Cc1ccc(cc1)OC(C)C(=O)/C=C/N(C)C 1L-005 CC(C(=O)/C=C/N(C)C)Oc1ccccc1F 1L-006 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1)C(C)(C)C 1L-007 CC(c1ccnc2n1ncn2)Oc3cccc(c3)C(F)(F)F 1L-008 CC(c1ccnc2n1nc(n2)N)Oc3cccc(c3)F 1L-009 Cc1cc(ccc1OC(C)c2ccnc3n2nc(n3)N)Cl 1L-010 CC(c1ccnc2n1nc(n2)N)Oc3ccc(cc3)C(C)(C)C 1L-012 CC(c1ccnc2n1ncn2)Oc3cccc(c3)F 1L-013 CC(c1ccnc2n1nc(n2)N)Oc3ccccc3 1L-014 c1cc(c(nc1)C(Cc2ccc(cc2Cl)Cl)(C#N)C#N)[N+](=O)[O-] 1L-015 CC(C)(C1OC(OC(O1)C(C)(C)Br)C(C)(C)Br)Br 1L-018 CC(c1ccnc2n1ncn2)Oc3ccccc3F 1L-020 CC(c1ccnc2n1nc(n2)N)Oc3ccccc3F 1L-021 Cc1cccc(c1OC(C)C(=O)/C=C/N(C)C)C 1L-022 Cc1ccc(cc1)OC(C)c2ccnc3n2nc(n3)N 1L-023 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1)[N+](=O)[O-] 1L-024 CC(c1ccnc2n1nc(n2)N)Oc3ccc(cc3)[N+](=O)[O-] 1L-025 CC(c1ccnc2n1ncn2)Oc3ccc(cc3)[N+](=O)[O-] 1L-026 CC(c1ccnc2n1ncn2)Oc3ccc(cc3F)F 1L-027 CC(C(=O)C)Oc1c(cccc1Cl)Cl 1L-028 c1ccnc(c1)SC(C#N)c2ccc(cc2Cl)Cl 1L-029 Cc1cccc(c1OC(C)c2ccnc3n2nc(n3)N)C 1L-030 c1ccnc(c1)SC(C#N)c2ccc(cc2)Cl 1L-031 c1cc(c(cc1Cl)Cl)C(C#N)Sc2c(cc(cn2)C(F)(F)F)Cl 1L-032 Cc1cc(ccc1OC(C)c2ccnc3n2ncn3)Cl 1L-033 CC(c1ccnc2n1ncn2)Oc3ccc(cc3)C(C)(C)C 1L-034 c1cc(ccc1C(C#N)Sc2c(cc(cn2)C(F)(F)F)Cl)Cl 1L-035 CC(c1ccnc2n1ncn2)Oc3ccc(cc3)C#N 1L-036 Cc1ccc(cc1)OC(C)c2ccnc3n2ncn3 1L-037 CC(C(=O)/C=C/N(C)C)Oc1ccccc1Cl 1L-038 c1cc(c(cc1Cl)Cl)C(C#N)Sc2nc[nH]n2 1L-039 c1cc(ccc1C(C#N)Sc2nc[nH]n2)Cl 1L-040 c1cc(ccc1C(C#N)Br)[N+](=O)[O-] 1L-041 CC(C(=O)/C=C/N(C)C)Oc1c(cccc1Cl)Cl 1L-042 CC(c1ccnc2n1nc(n2)N)Oc3ccccc3Cl 1L-043 c1cc(ccc1C(C#N)Sc2nc[nH]n2)[N+](=O)[O-] 1L-044 CC1=C(CC(=O)N1)C(=O)OC 1L-045 CC(c1ccnc2n1nc(n2)N)Oc3c(cccc3Cl)Cl 1L-046 CC1=C(/C(=C/N(C)C)/C(=O)N1)C(=O)OC 1L-047 CC(c1ccnc2n1ncn2)Oc3ccccc3Cl 1L-048 Cc1cc(nc(c1C#N)SC(C#N)c2ccc(cc2Cl)Cl)C 1L-049 Cc1cc(nc(c1C#N)SC(C#N)c2ccc(cc2)Cl)C 1L-050 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3ccc(cc3)C(C)(C)C 1L-051 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3ccc(cc3)[N+](=O)[O-] 1L-052 c1ccc(cc1)SC(C#N)c2ccc(cc2)Cl 1L-053 Cc1cc(ccc1OC(C)c2ccnc3n2nc(n3)/N=C/N(C)C)Cl 1L-054 Cc1cccc(c1)OC(C)c2ccnc3n2nc(n3)/N=C/N(C)C 1L-055 c1cc(cc(c1)/C=N/CC/N=C/c2cc(ccc2)Cl)Cl 1L-056 COc1ccc(cc1)/C=N/CC/N=C/c2ccc(cc2)OC 1L-057 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3cccc(c3)OC 1L-058 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3cccc(c3)F 1L-059 c1cc(cc(c1)Cl)CNCCNCc2cccc(c2)Cl 1L-060 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3ccc(cc3F)F 1L-062 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3ccccc3 1L-063 CC1=C(C(C(=O)N1)/C=N/OCc2ccc(cc2)Cl)C(=O)OC 1L-065 CC1=C(/C(=C/Nc2ccc(cc2)Oc3ccccc3)/C(=O)N1)C(=O)OC 1L-066 CC(c1ccnc2n1nc(n2)N/C=N/OC)Oc3cccc(c3)OC 1L-067 CC(c1ccnc2n1nc(n2)N/C=N/OC)Oc3ccccc3 1L-068 Cc1cc(cc(c1)OC(C)c2ccnc3n2nc(n3)/N=C/N(C)C)C 1L-069 Cc1cccc(c1)OC(C)c2ccnc3n2nc(n3)N/C=N/OC 1L-070 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3ccccc3F 1L-071 Cc1ccc(cc1)/C=N/CC/N=C/c2ccc(cc2)C 1L-072 CC(c1ccnc2n1nc(n2)N/C=N/OC)Oc3cccc(c3)F 1L-073 Cc1cc(cc(c1)OC(C)c2ccnc3n2nc(n3)N/C=N/OC)C 1L-074 c1cc(cc(c1)Cl)C[NH2+]CC[NH2+]Cc2cccc(c2)Cl.[Cl-].[Cl-] 1L-075 CC(c1ccnc2n1nc(n2)N/C=N/OC)Oc3ccc(cc3)[N+](=O)[O-] 1L-076 Cc1cc(ccc1OC(C)c2ccnc3n2nc(n3)N/C=N/OC)Cl 1L-077 c1csc(c1)/C=N/CC/N=C/c2sccc2 1L-078 CC1=C(/C(=C/Nc2ccc(cc2F)F)/C(=O)N1)C(=O)OC 1L-079 CC1=C(/C(=C/Nc2ccc(cc2)C#N)/C(=O)N1)C(=O)OC 1L-080 CC(c1ccnc2n1nc(n2)N/C=N/OC)Oc3ccc(cc3)C(C)(C)C 1L-081 CC(C(=O)C)Oc1cccc(c1)Cl 1L-082 CC(c1ccnc2n1ncn2)Oc3c(cccc3Cl)Cl 1L-083 Cc1ccc(cc1)CNCCNCc2ccc(cc2)C 1L-084 c1cc(sc1)CNCCNCc2cccs2 1L-085 CC1=C(/C(=C/Nc2ccc(cc2)C(C)C)/C(=O)N1)C(=O)OC 1L-088 c1cc(cc(c1)Cl)CN(CCN(Cc2cccc(c2)Cl)C(=O)Nc3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)Cl 1L-089 CC(C(=O)C)Oc1ccc(cc1)OC(C)C(=O)C 1L-090 CC(C(=O)/C=C/N(C)C)Oc1cccc(c1)Cl 1L-091 CC(c1ccnc2n1nc(n2)N)Oc3cccc(c3)Cl 1L-092 CC(Oc1ccc(cc1)OC(C(=O)/C=C/N(C)C)C)C(=O)/C=C/N(C)C 1L-093 COc1ccc(cc1)NC(=O)/C=C/c2ccco2 1L-303S c1ccc2c(c1)c(=N)n(nn2)c3ccc(cc3)C(F)(F)F 1L-304S c1ccc2c(c1)c(=N)n(nn2)c3cccc(c3)C(F)(F)F 1L-305S CCCNc1c(cc(c(n1)c2ccccc2)C(=O)OCC)C#N 1L-308S c1ccc2c(c1)c(nnn2)Nc3cccc(c3)C(F)(F)F 1L-309S c1ccc2c(c1)c(nnn2)Nc3ccc(cc3)C(F)(F)F 1L-310S Cc1c(nc(nn1)SCC=C)/C=C/Nc2ccc(cc2)OC 1L-312S Cc1ccc(cc1)N/C=C/c2c(nnc(n2)SCC=C)C 1L-314S Cc1c(nc(nn1)SCC=C)/C=C/Nc2cccc(c2)C(F)(F)F 1L-315S Cc1c(nc(nn1)SCC=C)/C=C/Nc2ccc(cc2)F 1L-316S Cc1c(nc(nn1)SCC=C)/C=C/Nc2ccc(cc2)Cl 1L-317S CCOC(=O)c1cc(c(nc1c2ccccc2)NCC=C)C#N 1L-318S CCCCNc1c(cc(c(n1)c2ccccc2)C(=O)OCC)C#N 1L-319S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCCC3)C#N 1L-320S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCCCC3)C#N 1L-321S CCOC(=O)c1cc(c(nc1c2ccccc2)NCc3ccccc3)C#N 1L-322S CCOC(=O)c1cc(c(nc1c2ccccc2)N(C)Cc3ccccc3)C#N 1L-323S CCOC(=O)c1cc(c(nc1c2ccccc2)N(C)C)C#N 1L-324S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCN(CC3)Cc4ccccc4)C#N 1L-325S CCOC(=O)c1cc(c(nc1c2ccccc2)NCc3ccc(cc3)Cl)C#N 1L-326S CCOC(=O)c1cc(c(nc1c2ccccc2)NCc3ccc(cc3Cl)Cl)C#N 1L-327S CCOC(=O)c1cc(c(nc1c2ccccc2)NCc3ccccc3OC)C#N 1L-332S CCOC(=O)c1cc(c(nc1c2ccccc2)NCc3cccc(c3)Cl)C#N 1L-333S Cc1c(nc(nn1)SCC=C)/C=C/NOCc2ccc(cc2Cl)Cl 1L-334S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCN(CC3)c4ccccc4F)C#N 1L-335S COc1ccccc1Oc2ccc(cn2)C(=O)NC3CCSC3=O 1L-336S c1cc(cc(c1)Oc2ccc(cn2)C(=O)NC3CCSC3=O)C(F)(F)F 1L-337S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCN(CC3)C)C#N 1L-338S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCN(CC3)c4ccccc4)C#N 1L-339S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCN(CC3)c4ccccn4)C#N 1L-340S CCOC(=O)c1cc(c(nc1c2ccccc2)NCc3ccc(cc3)C)C#N 1L-341S c1ccc2c(c1)c(=N)n(nn2)c3ccc(c(c3)Cl)Cl 1L-345S c1ccc2c(c1)c(nnn2)Nc3ccc(c(c3)Cl)Cl 1L-346S CCOC(=O)c1cc(c(nc1c2ccccc2)N3CCOCC3)C#N 1L-347S Cc1ccc(cc1)Oc2c(cccn2)C(=O)NC3CCSC3=O 1L-349S c1ccc(cc1)S(=O)(=O)Nc2[nH]c3ccccc3n2 1L-350S Cc1ccc(cc1)Cn\2c3ccccc3[nH]/c2=N\S(=O)(=O)c4ccccc4 1L-351S CC1(OC(=O)C(=COC)C(=O)O1)C 1L-352S Cc1ccc(cc1)SC=C2C(=O)OC(OC2=O)(C)C 1L-353S CCCSc1nc(c(nn1)C)/C=C/Nc2ccc(cc2)OC 1L-354S CCCSc1nc(c(nn1)C)/C=C/Nc2ccc(cc2)C 1L-355S CCCSc1nc(c(nn1)C)/C=C/Nc2ccc(cc2)Cl 1L-356S CCCSc1nc(c(nn1)C)/C=C/Nc2ccc(cc2)F 1L-357S CCCSc1nc(c(nn1)C)/C=C/Nc2cccc(c2)C(F)(F)F 1L-358S CC1(OC(=O)C(=CSc2ccc(cc2)OC)C(=O)O1)C 1L-362S CC1(OC(=O)C(=CSc2ccccc2Cl)C(=O)O1)C 1L-363S Cc1c(nc(nn1)SCc2ccccc2)/C=C/N(C)C 1L-364S CC1(OC(=O)C(=CSc2ccc(cc2)Cl)C(=O)O1)C 1L-365S CC1(OC(=O)C(=CSc2cccc(c2)Cl)C(=O)O1)C 1L-366S c1ccc(cc1)N2CCN(CC2)/C(=C/C#N)/N 1L-367S CC1(OC(=O)C(=CSc2ccccc2)C(=O)O1)C 1L-368S CC1(OC(=O)C(=CSc2ccc(cc2Cl)Cl)C(=O)O1)C 1L-369S c1ccc(cc1)CN2CCN(CC2)/C(=C/C#N)/N 1L-371S CC1(OC(=O)C(=CSc2ccc(cc2)Br)C(=O)O1)C 1L-373S CC1(OC(=O)C(=CSc2ccc(cc2)F)C(=O)O1)C 1L-374S CC1(OC(=O)C(=CSc2cccc(c2)C(F)(F)F)C(=O)O1)C 1L-375S CC1CN(CC(O1)C)/C(=C/C#N)/N 1L-376S C1CCN(C1)/C(=C/C#N)/N 1L-377S C[NH+]1CCN(CC1)c2c(ccc(n2)C(F)(F)F)C#N.[Cl-] 1L-378S CC1(OC(=O)C(=CSc2ccc(cc2)C(C)(C)C)C(=O)O1)C 1L-379S Cc1c(nnc(n1)SCc2ccc(cc2)Cl)C 1L-381S CCOC(=O)N1CCN(CC1)/C(=C/C#N)/N 1L-382S Cc1ccccc1SC=C2C(=O)OC(OC2=O)(C)C 1L-383S CC1(OC(=O)C(=CSCc2ccc(cc2)Cl)C(=O)O1)C 1L-384S CC1(OC(=O)C(=CSCc2ccc(cc2Cl)Cl)C(=O)O1)C 1L-385S CC1(OC(=O)C(=CSCc2cccc(c2)C(F)(F)F)C(=O)O1)C 1L-386S CC1(OC(=O)C(=CSCc2ccc(cc2)C(C)(C)C)C(=O)O1)C 1L-387S CC1(OC(=O)C(=CSCc2ccccc2)C(=O)O1)C 1L-388S Cc1c(nc(nn1)SCc2ccccc2)/C=C/Nc3ccc(cc3)OC 1L-389S Cc1ccc(cc1)N/C=C/c2c(nnc(n2)SCc3ccccc3)C 1L-390S Cc1c(nc(nn1)SCc2ccccc2)/C=C/Nc3cccc(c3)C(F)(F)F 1L-391S Cc1c(nc(nn1)SCc2ccccc2)/C=C/Nc3ccc(cc3)Cl 1L-392S Cc1c(nc(nn1)SCc2ccccc2)/C=C/Nc3ccc(cc3)F 1L-393S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/N(C)C 1L-397S c1ccc2c(c1)c(nnn2)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 1L-401S CC1(OC(=O)C(=CSC2CCCCC2)C(=O)O1)C 1L-402S Cc1c(nc(nn1)SCc2ccccc2)/C=C/NOCc3ccc(cc3Cl)Cl 1L-403S Cc1c(nc(nn1)SCc2ccccc2)/C=C/NOCc3ccc(cc3)Cl 1L-405S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/Nc3ccc(cc3)OC 1L-406S Cc1ccc(cc1)N/C=C/c2c(nnc(n2)SCc3ccc(cc3)Cl)C 1L-407S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/Nc3cccc(c3)C(F)(F)F 1L-408S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/Nc3ccc(cc3)Cl 1L-409S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/Nc3ccc(cc3)F 1L-410S CC1(OC(=O)C(=CN)C(=O)O1)C 1L-411S CC(C)SC=C1C(=O)OC(OC1=O)(C)C 1L-412S CC1(OC(=O)C(=CSC(C)(C)C)C(=O)O1)C 1L-413S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/NOCc3ccc(cc3Cl)Cl 1L-416S Cc1c(nc(nn1)SC)/C=C/NOCc2ccc(cc2Cl)Cl 1L-417S Cc1c(nc(nn1)SCc2ccccc2)/C=C/NOCc3ccc(cc3)F 1L-418S Cc1c(nc(nn1)SCc2ccccc2)/C=C/NOCc3c(cccc3Cl)Cl 1L-419S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/NOC 1L-421S Cc1c(nc(nn1)SCc2ccccc2)/C=C/NOC 1L-422S c1cc(cc(c1)Sc2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl)C(F)(F)F 1L-500S COc1ccc(cc1)S(=O)c2ccc(cc2C#N)NC(=O)C3CC3 1L-502S COc1ccc(cc1)S(=O)c2ccc(cc2C#N)NC(=O)c3ccc(cc3)F 1L-503S COc1ccc(cc1)S(=O)c2ccc(cc2C#N)NC(=O)c3c(cccc3F)F 1L-504S COc1ccc(cc1)S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccccc3Cl 1L-505S Cc1ccc(cc1)S(=O)c2ccc(cc2C#N)NC(=O)c3ccccc3Cl 1L-507S Cc1ccc(cc1)S(=O)c2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl 1L-508S c1cc(cc(c1)Cl)C(=O)Nc2ccc(c(c2)C#N)Sc3cccc(c3)C(F)(F)F 1L-509S COc1cccc(c1)C(=O)Nc2ccc(c(c2)C#N)Sc3cccc(c3)C(F)(F)F 1L-510S CS(=O)(=O)c1ccc(cc1C#N)NC(=O)c2ccccc2 1L-511S CS(=O)(=O)c1ccc(cc1C#N)NC(=O)c2cccc(c2)Cl 1L-512S CS(=O)c1ccc(cc1C#N)NC(=O)c2cccc(c2)C#N 1L-513S c1cc(c(c(c1)Cl)Sc2ccc(cc2C#N)C(F)(F)F)Cl 1L-514S COc1ccc(cc1)Sc2ccc(cc2C#N)NC(=O)c3ccc(cc3Cl)Cl 1L-516S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(c(c2)C#N)Sc3cccc(c3)C(F)(F)F 1L-517S c1cc(cc(c1)S(=O)c2ccc(cc2C#N)NC(=O)c3ccc(cc3)F)C(F)(F)F 1L-518S c1cc(cc(c1)S(=O)c2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl)C(F)(F)F 1L-519S COC(=O)c1ccccc1Sc2ccc(cc2C#N)C(F)(F)F 1L-520S c1cc(cc(c1)Cl)Sc2ccc(cc2C#N)C(F)(F)F 1L-521S c1ccc(c(c1)Sc2ccc(cc2C#N)C(F)(F)F)Cl 1L-523S COc1ccc(cc1)Sc2ccc(cc2C#N)C(F)(F)F 1L-524S C=CCNc1cc(nc(n1)c2ccccc2)CS(=O)c3ccccc3 1L-525S c1ccc(cc1)CNc2cc(nc(n2)c3ccccc3)CS(=O)c4ccccc4 1L-526S CCN(CC)c1cc(nc(n1)c2ccccc2)CS(=O)c3ccccc3 1L-527S CNc1cc(nc(n1)c2ccccc2)CS(=O)c3ccccc3 1L-528S c1ccc(cc1)c2nc(cc(n2)Oc3ccccc3)CS(=O)c4ccccc4 1L-529S c1cc(ccc1F)Sc2ccc(cc2C#N)C(F)(F)F 1L-530S c1cc(c(c(c1)Cl)Cl)Sc2ccc(cc2C#N)C(F)(F)F 1L-531S c1cc(c(cc1C(F)(F)F)C#N)Sc2ccc(cc2Cl)Cl 1L-532S c1ccc(cc1)SCCNC(=O)Cc2c(cccc2Cl)Cl 1L-533S COc1ccc(cc1)S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3cccc(c3)Cl 1L-534S c1cc(ccc1S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccc(c(c3)Cl)Cl)Cl 1L-537S Cc1nc(cc(n1)N2CCOCC2)CSc3ccc(cc3)Cl 1L-539S COc1ccc(cc1)S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccc(cc3)F 1L-540S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2C#N)NC(=O)c3ccccc3C 1L-541S c1cc(ccc1Sc2ccc(cc2C#N)C(F)(F)F)Cl 1L-543S c1ccnc(c1)c2nc(cc(n2)N3CCOCC3)CSc4ccc(cc4)Cl 1L-544S c1ccnc(c1)c2nc(cc(n2)N3CCCC3)CSc4ccc(cc4)Cl 1L-545S c1ccnc(c1)c2nc(cc(n2)N3CCCCC3)CSc4ccc(cc4)Cl 1L-546S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(c(c2)C#N)S(=O)(=O)c3cccc(c3)C(F)(F)F 1L-550S c1cc(cc(c1)Cl)C(=O)Nc2ccc(c(c2)C#N)S(=O)(=O)c3cccc(c3)C(F)(F)F 1L-551S COc1ccc(cc1)S(=O)c2ccc(cc2C#N)NC(=O)c3ccc(cc3Cl)Cl 1L-552S Cc1ccccc1Sc2ccc(cc2C#N)C(F)(F)F 1L-553S COc1cccc(c1)C(=O)Nc2ccc(c(c2)C#N)S(=O)c3cccc(c3)C(F)(F)F 1L-555S Cc1ccc(cc1)S(=O)c2ccc(cc2C#N)NC(=O)C3CC3 1L-556S c1(nc(=S)ss1)NC(=O)C(F)(F)F 1L-557S c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2nc(=S)ss2 1L-558S CCC(=O)Nc1nc(=S)ss1 1L-559S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)CS(=O)(=O)c4ccccc4 1L-560S c1ccc(cc1)CNc2cc(nc(n2)c3ccccc3)CS(=O)(=O)c4ccccc4 1L-561S c1ccc(cc1)c2nc(cc(n2)N3CCCC3)CS(=O)(=O)c4ccccc4 1L-562S C=CCNc1cc(nc(n1)c2ccccc2)CS(=O)(=O)c3ccccc3 1L-563S CNc1cc(nc(n1)c2ccccc2)CS(=O)(=O)c3ccccc3 1L-564S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)CSc4ccc(cc4)Cl 1L-565S c1cc(oc1)/C=C/C(=O)Nc2ccc(cc2)F 1L-566S c1cc(oc1)/C=C/C(=O)Nc2cc(cc(c2)Cl)Cl 1L-567S c1cc(oc1)/C=C/C(=O)Nc2ccc(cc2)Cl 1L-568S COc1ccc(cc1)Oc2ccc(cc2C#N)C(F)(F)F 1L-570S c1cc(c(cc1C(F)(F)F)C#N)Oc2ccc(cc2F)F 1L-571S c1ccc(cc1)c2nc(cc(n2)N3CCCC3)CSc4ccc(cc4)Cl 1L-572S CC(C)Nc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 1L-573S c1cc(oc1)/C=C/C(=O)Nc2ccc(cc2F)F 1L-574S c1cc(oc1)/C=C/C(=O)Nc2ccc(cc2Cl)Cl 1L-575S c1ccc(c(c1)NC(=O)/C=C/c2ccco2)Cl 1L-576S c1cc(oc1)/C=C/C(=O)Nc2cc(ccc2Cl)Cl 1L-577S c1cc(oc1)/C=C/C(=O)Nc2ccc(c(c2)Cl)Cl 1L-578S c1cc(oc1)/C=C/C(=O)Nc2ccc(c(c2)F)F 1L-579S c1cc(ccc1Sc2ccc(cc2C#N)C(F)(F)F)Br 1L-580S Cc1ccc(cc1)Sc2ccc(cc2C#N)C(F)(F)F 1L-581S Cc1cccc(c1C)Oc2ccc(cc2C#N)C(F)(F)F 1L-582S Cc1cc(cc(c1)Oc2ccc(cc2C#N)C(F)(F)F)C 1L-583S c1ccc(cc1)Sc2ccc(cc2C#N)C(F)(F)F 1L-584S CNc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 1L-585S C=CCNc1cc(nc(n1)c2ccccc2)CSc3ccc(cc3)Cl 1L-586S Cc1ccc(cc1)SCc2cc(n(n2)C)O 1L-588S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(cc3)C(C)C 1L-592S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3cccnc3)N4CCOCC4 1L-595S c1ccc(cc1)S(=O)(=O)Cc2cc(nc(n2)c3cccnc3)N4CCCC4 1L-596S C=CCNc1cc(nc(n1)c2ccccc2)CS(=O)c3ccc(cc3)Cl 1L-597S c1ccc(cc1)CNc2cc(nc(n2)c3ccccc3)CS(=O)c4ccc(cc4)Cl 1L-598S c1cc(oc1)/C=C/C(=O)Nc2ccc(cc2)Br 1L-599S c1cc(oc1)/C=C/C(=O)Nc2ccc(cc2)C(F)(F)F 1L-600S c1cc(cc(c1)NC(=O)/C=C/c2ccco2)C(F)(F)F 1L-601S CC(C)Nc1cc(nc(n1)c2cccnc2)CS(=O)(=O)c3ccccc3 1L-602S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(cc3)Br 1L-603S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3cccc(c3)Br 1L-604S c1cc(c(c(c1)F)C(=O)Nc2nc(=S)ss2)F 1L-605S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3c(cccc3Cl)F 1L-606S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(cc3)Cl 1L-607S c1ccc(c(c1)NC(=O)/C=C/c2ccco2)F 1L-608S COc1ccc(c(c1)NC(=O)/C=C/c2ccco2)OC 1L-609S c1ccc(cc1)NC(=O)/C=C/c2ccco2 1L-610S Cc1cccc(c1)NC(=O)/C=C/c2ccco2 1L-611S COc1cccc(c1)NC(=O)/C=C/c2ccco2 1L-612S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(cc3)C 1L-613S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(cc3)OC 1L-614S Cc1ccc(cc1)Oc2ccc(cc2C#N)C(F)(F)F 1L-615S c1ccc(cc1)c2cc\3c(nn2)-c4ccccc4/C3=N/O 1L-616S COc1ccc(cc1OC)c2cc\3c(nn2)-c4ccccc4/C3=N/O 1L-617S Cc1cccc(c1)c2cc\3c(nn2)-c4ccccc4/C3=N/O 1L-618S c1ccc\2c(c1)-c3c(cc(nn3)c4ccc(cc4)Br)/C2=N\O 1L-619S Cc1cc(cc(c1)NC(=O)/C=C/c2ccco2)C 1L-621S c1cc(oc1)/C=C/C(=O)Nc2ccc(c(c2F)Cl)F 1L-622S Cc1ccc(cc1NC(=O)/C=C/c2ccco2)Cl 1L-623S Cc1ccc(cc1)NC(=O)/C=C/c2ccco2 1L-624S c1c(cc(cc1Cl)Cl)C(=O)Nc2nc(=S)ss2 1L-625S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(cc3)F 1L-629S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(cc3)C(F)(F)F 1L-630S c1ccc(cc1)CC(=O)NCCSc2ccc(cc2)Cl 1L-636S c1cc(ccc1CC(=O)NCCSc2ccc(cc2)Cl)Cl 1L-637S Cc1ccc(cc1)CC(=O)NCCSc2ccc(cc2)Cl 1L-638S Cc1ccc(cc1)CC(=O)NCCS(=O)c2ccc(cc2)Cl 1L-641S c1cc(ccc1CC(=O)NCCS(=O)c2ccc(cc2)Cl)Cl 1L-642S c1ccc(cc1)CC(=O)NCCS(=O)c2ccc(cc2)Cl 1L-643S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)C=O 1L-644S Cc1ccc(cc1)SCc2c(c(n(n2)C)Sc3ccc(cc3)Br)C=O 1L-648S CCOC(=O)C1C(N=C(N=C1O)c2ccccc2)c3ccc(c(c3)OC)O 1L-650S Cc1nc(cc(n1)O)CSc2ccc(cc2)Cl 1L-712S c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)NCCOC(=O)c3cccs3)Cl 1L-900 c1cc(cc(c1)C(F)(F)F)C(=O)OCCNc2cnn(c(=O)c2Cl)c3cccc(c3)Cl 1L-901 CN(CCO)c1cnn(c(=O)c1Cl)c2ccc(cc2)OC 1L-902 CN(CCOC(=O)C1CC1)c2cnn(c(=O)c2Cl)c3ccc(cc3)OC 1L-904 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)N3CCNCC3)Cl 1L-905 CCOC(=O)CNC(=S)N1CCN(CC1)c2cnn(c(=O)c2Cl)c3cccc(c3)Cl 1L-906 CN(CCOC(=O)Nc1cccc(c1)C(F)(F)F)c2cnn(c(=O)c2Cl)c3ccc(cc3)OC 1L-907 CN(CCOC(=O)Nc1ccc(cc1)Cl)c2cnn(c(=O)c2Cl)c3ccc(cc3)OC 1L-908 CCOC(=O)/C(=C\N1CCN(CC1)c2cnn(c(=O)c2Cl)c3cccc(c3)Cl)/C#N 1L-909 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)F)Cl 1L-910 c1ccc(c(c1)C(=O)N2CCN(CC2)c3cnn(c(=O)c3Cl)c4cccc(c4)Cl)F 1L-911 c1cc(cc(c1)Cl)n2c(=O)c(c(cn2)N3CCN(CC3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl 1L-912 COc1cc(c(cc1OC)NC(=S)N2CCN(CC2)c3cnn(c(=O)c3Cl)c4cccc(c4)Cl)C#N 1L-913 COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCCCC3)Cl 1L-914 COc1ccc(cc1)n2c(=O)c(c(cn2)NCCc3ccccn3)Cl 1L-915 COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCN(CC3)C(c4ccccc4)c5ccccc5)Cl 1L-916 COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCN(CC3)c4cccc(c4)Cl)Cl 1L-917 COc1ccc(cc1)n2c(=O)c(c(cn2)NCC=C)Cl 1L-918 Cc1cc(=O)n(c(n1)/N=C/N(C)C)C 1L-919 c1c(cnc(c1Cl)N/N=C/C(=C(\C(=O)O)/Cl)/Cl)C(F)(F)F 1L-920 c1c(cnc(c1Cl)n2c(=O)c(c(cn2)Cl)Cl)C(F)(F)F 1L-921 CNc1nnc(s1)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 1L-922 Cc1ccc(cc1)N/N=C\2/CCCNC2=O 1L-923 Cc1ccc2c(c1)c3c([nH]2)C(=O)NCC3 1L-924 Cc1ccccc1N/N=C/2\CCCNC2=O 1L-925 c1ccc2c(c1)c(nc(n2)C(F)(F)F)NNC(=O)c3ccc(cc3)Cl 1M-001 c1ccc(c(c1)C(=O)NNc2ccc(cc2F)F)C(=O)O 1M-002 CN(c1c2ccccc2nc(n1)C(F)(F)F)NC(=O)c3ccccc3F 1M-003 CC(C)(C)NS(=O)(=O)c1ccc(s1)c2csnn2 1M-005 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)c4csnn4 1M-006 c1cc(sc1c2csnn2)S(=O)(=O)NC3CCCCC3 1M-007 c1ccc2c(c1)c[n+](nc2[O-])c3ccc(cc3)Cl 1M-008 COCCCNS(=O)(=O)c1ccc(s1)c2cnns2 1M-009 CCOC(=O)CNC(=O)c1ccccc1 1M-011 CCOC(=O)CNC(=O)c1cccs1 1M-012 CCOC(=O)CNC(=O)c1c(cccc1Cl)Cl 1M-013 CCOC(=O)CNC(=O)c1ccccc1F 1M-014 CCOC(=O)CNC(=O)c1ccco1 1M-015 CCOC(=O)CNC(=O)c1ccccc1Cl 1M-016 CCOC(=O)CNC(=O)c1ccc(cc1)F 1M-017 CCOC(=O)CNC(=O)c1ccc(cc1)OC 1M-018 CCOC(=O)CNC(=O)c1ccc(cc1)[N+](=O)[O-] 1M-019 CCOC(=O)CNC(=O)c1ccc(cc1)C 1M-020 CCOC(=O)CNC(=O)c1cccc(c1)C 1M-021 c1ccn(c1)c2c(c(c(c(c2n3cccc3)n4cccc4)n5cccc5)n6cccc6)n7cccc7 1M-022 CCOc1cnc(o1)c2ccc(cc2)OC 1M-023 CCOc1cnc(o1)c2ccc(cc2)[N+](=O)[O-] 1M-024 CCOc1cnc(o1)c2c(cccc2Cl)Cl 1M-025 CCOc1cnc(o1)c2ccc(cc2)F 1M-026 CCOc1cnc(o1)c2ccc(cc2)C 1M-027 COc1ccc(cc1)C(C#N)c2c(nc3ccccc3n2)C(F)(F)F 1M-028 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(c3ccc(cc3)Cl)C(=O)N/C=N/OCc4ccc(cc4)Cl 1M-029 CCOc1cnc(o1)c2ccccc2Cl 1M-030 CCOc1cnc(o1)c2cccs2 1M-031 CCOc1cnc(o1)c2ccccc2 1M-032 CCOc1cnc(o1)c2cccc(c2)C 1M-033 CCOC(=O)CNC(=O)c1c(onc1c2c(cccc2Cl)Cl)C 1M-034 CCOC(=O)CNC(=O)c1c(onc1c2c(cccc2Cl)F)C 1M-035 COc1cccc(c1)CO/N=C\NC(=O)C(c2ccc(cc2)Cl)c3c(nc4ccccc4n3)C(F)(F)F 1M-036 COc1ccc(cc1)CO/N=C/NC(=O)C(c2ccc(cc2)Cl)c3c(nc4ccccc4n3)C(F)(F)F 1M-037 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(c3ccc(cc3)Cl)C(=O)N/C=N\OCc4ccc(cc4Cl)Cl 1M-038 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(c3ccc(cc3)Cl)C(=O)N/C=N/OCc4cccc(c4)C(F)(F)F 1M-039 c1ccc(c(c1)CO/N=C/NC(=O)C(c2ccc(cc2)Cl)c3c(nc4ccccc4n3)C(F)(F)F)Br 1M-040 CCOc1cnc(o1)c2c(onc2c3c(cccc3Cl)Cl)C 1M-041 CCOc1cnc(o1)c2c(onc2c3c(cccc3Cl)F)C 1M-042 Cc1ccc(cc1)c2c3c(ncnc3n(n2)C(C)(C)C)NS(=O)(=O)c4ccc(cc4)Cl 1M-304S Cc1ccc(cc1)c2c3c(ncnc3n(n2)C(C)(C)C)NS(=O)(=O)c4ccc(cc4)[N+](=O)[O-] 1M-305S CC(C)(C)n1c2c(c(n1)c3ccc(cc3)F)c(ncn2)N 1M-307S c1ccc(cc1)N/N=C\2/c3ccccc3N(C2=O)CN4CCOCC4 1M-308S Cc1ccc(cc1)N/N=C\2/c3ccccc3N(C2=O)CN4CCOCC4 1M-309S c1ccc2c(c1)/C(=N/Nc3ccc(cc3)Cl)/C(=O)N2CN4CCOCC4 1M-310S CC(=O)N(c1c2c(nn(c2ncn1)C(C)(C)C)c3ccc(cc3)Cl)C(=O)C 1M-313S Cc1ccc2c(c1)N=C(CO2)c3ccc(cc3)F 1M-315S Cc1ccc2c(c1)N=C(CO2)c3ccc(cc3)Cl 1M-316S c1ccc2c(c1)/C(=N/Nc3ccc(c(c3)Cl)Cl)/C(=O)N2CN4CCOCC4 1M-318S c1ccc2c(c1)/C(=N/Nc3ccccc3Cl)/C(=O)N2CN4CCOCC4 1M-319S CN1CCN(CC1)CN2c3ccccc3/C(=N/Nc4ccccc4)/C2=O 1M-320S c1ccc2c(c1)/C(=N/Nc3ccc(cc3)F)/C(=O)N2CN4CCOCC4 1M-321S c1ccc2c(c1)/C(=N/Nc3ccc(cc3)F)/C(=O)N2CN4CCN(CC4)c5cccc(c5)Cl 1M-322S Cc1ccc2c(c1)N=C(CO2)c3ccc(cc3)OC 1M-324S Cc1ccc2c(c1)N=C(CO2)c3ccc(cc3)[N+](=O)[O-] 1M-326S CC(c1ccccc1)NC(=S)Nc2ccc(cc2)Cl 1M-328S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)Nc2ccccc2OC 1M-332S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)Nc2ccc(cc2)C(F)(F)F 1M-333S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)NCC=C 1M-334S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)N2CCOCC2 1M-335S c1cc(ccc1C2=Nc3cc(ccc3OC2)Cl)Cl 1M-337S c1cc(ccc1C2=Nc3cc(ccc3OC2)Cl)[N+](=O)[O-] 1M-338S CC(c1ccccc1)N/C(=N\c2ccc(cc2)Cl)/SC 1M-339S Cc1ccc(cc1)CNC(=S)Nc2ccccc2 1M-340S Cc1ccc(cc1)CN/C(=N\c2ccccc2)/SC 1M-344S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)Nc2cccc(c2)Cl 1M-345S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)NCc2ccc(cc2)Cl 1M-346S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)NC2CC2 1M-347S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)Nc2nccs2 1M-348S c1cc(ccc1C(CCSc2ccc(cc2)Br)O)Cl 1M-501S COc1ccc(cc1)SCC/C(=N/O)/c2ccc(cc2)Cl 1M-502S Cc1ccc(cc1)S(=O)(=O)CC(c2ccc(c(c2)Cl)Cl)O 1M-503S CC(=O)c1c(nn(c1Cl)C)c2ccccc2 1M-504S Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc(cc2)Cl 1M-506S Cc1ccc(cc1)SCCC(c2ccc(cc2)Cl)O 1M-507S Cc1ccc(cc1)S(=O)(=O)CCC(c2ccc(cc2)Cl)O 1M-509S Cc1ccc(cc1)S(=O)(=O)CC/C(=N\OCc2cccc(c2)F)/c3ccc(cc3)Cl 1M-510S Cc1ccccc1C2N=C(SC(=N2)c3ccccc3)c4ccccc4 1M-511S c1ccc(cc1)C2=NC(N=C(S2)c3ccccc3)c4cccc(c4)C(F)(F)F 1M-512S c1cc(ccc1c2csc(n2)NC(=O)CSCC(=O)O)Cl 1M-513S c1cc(ccc1c2csc(n2)N3C(=O)CSCC3=O)Cl 1M-514S COC(=O)c1c(ccs1)NC(=O)CSCC(=O)O 1M-519S COC(=O)c1c(ccs1)N2C(=O)CSCC2=O 1M-520S Cc1ccc(cc1)SCC/C(=N/O)/c2ccc(cc2)Cl 1M-521S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)NC 1M-526S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)Nc2ccccc2 1M-527S Cc1ccc(cc1)NC(=O)n2c(nnc2SC)N 1M-530S Cn1c(c(c(n1)c2ccccc2)C=O)Oc3ccc(cc3)Cl 1M-531S COC(=O)c1ccccc1SC/C(=N/OC)/c2ccc(cc2Cl)Cl 1M-532S CO/N=C(/CSCc1ccccc1Cl)\c2ccc(cc2Cl)Cl 1M-533S CSc1nnc(n1C(=O)Nc2ccc(cc2)Cl)N 1M-534S Cc1ccccc1NC(=O)n2c(nnc2SC)N 1M-535S Cc1ccc(cc1)SCC/C(=N\OC)/c2ccc(cc2)Cl 1M-536S Cc1ccc(cc1)S(=O)(=O)CC/C(=N/OC)/c2ccc(cc2)Cl 1M-537S Cc1ccc(cc1)SC/C(=N/OC)/c2ccc(cc2)Cl 1M-539S Cc1ccc(cc1)Sc2c(c3ccccc3nc2c4ccc(cc4)Cl)C(=O)O 1M-540S c1ccc2c(c1)C(=O)N3C2(NCC3)c4ccc(cc4)Cl 1M-541S Cc1ccc(cc1)Sc2cc3ccccc3nc2c4ccc(cc4)Cl 1M-543S CO/N=C(/COc1cc(c(cc1Cl)Cl)Cl)\c2ccc(cc2Cl)Cl 1M-547S c1ccc2c(c1)C(=O)N3C2(NCC3)c4ccc(cc4)F 1M-548S c1ccc(cc1)c2c(c(c3ccccc3n2)C(=O)O)Sc4ccc(cc4)Cl 1M-549S c1ccc(cc1)c2c(cc3ccccc3n2)Sc4ccc(cc4)Cl 1M-550S c1ccc2c(c1)cc(c(n2)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl 1M-551S c1cc(c(cc1CSc2[nH]c(nn2)N)Cl)Cl 1M-554S c1cc2c(cc1F)nc(s2)CSc3[nH]c(nn3)N 1M-555S CC(=O)c1cc(no1)c2ccccc2 1M-562S COc1ccc(cc1)Sc2c(c3ccccc3nc2c4ccc(cc4)Cl)C(=O)O 1M-564S Cc1ccc(cc1)Sc2c(c3ccccc3nc2c4ccc(cc4Cl)Cl)C(=O)O 1M-565S c1ccc(cc1)C(=O)N2CCN3C2(c4ccccc4C3=O)c5ccc(cc5)Cl 1M-566S CNC(=O)c1c2ccccc2nc(c1Sc3ccc(cc3)Cl)c4ccccc4 1M-569S c1ccc2c(c1)c(c(c(n2)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl)C(=O)O 1M-590S CC1(CN(C1=O)c2ccc(cc2)C(=O)/C=C/c3cccc(c3)Br)C 1M-700 CC(C)(CCl)C(=O)Nc1cccc(c1)Br 1M-701 CC1(CN(C1=O)c2cccc(c2)Br)C 1M-702 CCOC(=O)C(Cc1ccccc1)NC(=O)C(C)(C)CCl 1M-706 Cc1ccc(c(c1)C)n2cc(c(=O)cc2C)C(=O)O 1M-707 Cc1cc(c(c(=O)o1)/C=N/OCc2ccc(cc2Cl)Cl)O 1M-708 Cc1cc(=O)c(cn1c2ccc(cc2)C(C)C)C(=O)O 1M-709 Cc1ccc(cc1)N/N=C/c2c(cc(oc2=O)C)O 1M-710 Cc1nc2ccccc2c(=O)o1 1M-711 COC(=O)CN1C(=O)Cc2ccccc2C1=O 1M-713 c1ccc2c(c1)c(c(s2)C=O)Sc3ccc(cc3)Br 1M-714 c1ccc2c(c1)cc3c(n2)CN(C3=O)c4ccc(cc4)Cl 1M-715 CCOC(=O)C(C(=O)C)C(=O)c1ccccc1NC(=O)C 1M-716 C1CC(=COC1)C(=O)C(F)(F)F 1M-717 c1ccc2c(c1)c(c(s2)C#N)Cl 1M-718 CN1C(=O)c2ccccc2/C(=N/Nc3ccc(c4c3cccc4)Cl)/C1=O 1M-719 CC(=O)c1c(c2ccccc2[nH]c1=O)O 1M-720 Cc1cc(cc(c1)n2cc(c(=O)cc2C)C(=O)O)C 1M-721 CC1(CC(=CC(=O)C1)Nc2ccccc2N)C 1M-722 c1ccc2c(c1)CC(=O)N(C2=O)CC(=O)O 1M-724 c1ccc(c(c1)N(S(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl)Sc4c(cc(cn4)C(F)(F)F)Cl 1M-725 c1ccc2c(c1)c(c(s2)C#N)N3CCCC3 1M-727 Cc1ccc(cc1)Nn2cc(c(=O)cc2C)C(=O)O 1M-728 c1ccc2c(c1)/C(=N/Nc3ccc(cc3)Cl)/C(=O)N(C2=O)CC(=O)O 1M-729 CC1=CC(=O)/C(=C/Nc2ccc(cc2)N(C)C)/C(=O)O1 1M-731 c1c(c(n[nH]1)C(F)(F)F)CCCO 1M-732 Cc1cc(c(c(=O)o1)/C=N/Nc2ccc(cc2)F)O 1M-733 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)OC)C(=O)C1)C.CO 1M-735 Cc1c(c(on1)/C=C/c2c(c3ccccc3s2)Cl)[N+](=O)[O-] 1M-736 CN(C)/C=C/C(=O)c1c(c2ccccc2[nH]c1=O)O 1M-737 Cc1cc(c(c(=O)o1)/C=N/Nc2ccc(cc2)Cl)O 1M-738 Cc1cc(c(c(=O)o1)/C=N/Nc2cccc(c2)Cl)O 1M-739 CC1(OC(=O)C(=Cc2c(c3ccccc3s2)Cl)C(=O)O1)C 1M-740 COC1CCC(=CO1)C(=O)C(F)(F)F 1M-742 c1ccc2c(c1)c(c(s2)C=O)Sc3cc(c(cc3Cl)Cl)Cl 1M-743 CCO.CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)Cl)C(=O)C1)C 1M-744 COc1ccc(cc1)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)C4CCCCC4C3=O 1M-745 c1ccc2c(c1)c(c(s2)/C=C(\C#N)/C(=O)Nc3cccc(c3)C(F)(F)F)Cl 1M-746 COc1ccc(cc1)N2Cc3c(cc4ccccc4n3)C2=O 1M-747 Cc1cc(=O)c(cn1Nc2ccc(cc2)F)C(=O)O 1M-749 Cc1cc2c([nH]1)cccc2OCC(CN3CCCC3)O 1M-900 Cc1ccc(cc1)C(=O)Nc2cc(c(oc2=O)/C=C/Nc3ccc(cc3)C(=O)OC)C(=O)C 1M-901 Cc1ccc(cc1)C(=O)Nc2cc3c(nccc3oc2=O)C 1M-902 CCOC(=O)C1C(C1C(=O)NN)C(=O)Nc2ccccc2 1M-905 Cc1cc2c([nH]1)cccc2OCC(CNC3CCCCC3)O 1M-906 Cc1cc2c([nH]1)cccc2OCC(CN3CCOCC3)O 1M-907 CCOC(=O)Cc1c(cccn1)C(=O)Nc2ccc(cc2)F 1M-908 CCOC(=O)Cc1c(cccn1)C(=O)Nc2cccc(c2)C(F)(F)F 1M-909 CCOC(=O)Cc1c(cccn1)C(=O)Nc2ccc(cc2)OC(F)(F)F 1M-910 CCOC(=O)Cc1c(cccn1)C(=O)Nc2ccc(cc2)OC 1M-911 CCOC(=O)Cc1c(cccn1)C(=O)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 1M-912 Cc1cc2c([nH]1)cccc2OCC(CNCC=C)O 1M-913 Cc1cc2c([nH]1)cccc2OCC(CNCc3ccco3)O 1M-914 CCOC(=O)NC(=O)/C(=N\Nc1ccccc1)/C(=O)C 1M-916 Cc1cc2c([nH]1)cccc2OCC(CNCCCOC)O 1M-918 Cc1cc2c([nH]1)cccc2OCC(CN3CCCCC3)O 1M-919 CCOC(=O)c1cnc2cc(ccn2c1=O)C 1M-920 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)O 1M-922 c1cc(sc1)/C=N/O 1M-923 CC1=C(CCC(=O)N1)C#N 1M-925 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)Nc3ccc(cc3)OC 1M-926 CC1=C(/C(=C/N(C)C)/CC(=O)N1)C#N 1M-929 CC1=C(/C(=C/Nc2ccc(cc2)F)/CC(=O)N1)C#N 1M-930 CC1=C(/C(=C/Nc2ccc(cc2)OC(F)(F)F)/CC(=O)N1)C#N 1M-931 CC1=C(C(CC(=O)N1)/C=N/OCc2ccc(cc2Cl)F)C#N 1M-932 CC1(OC(=O)C(=C(Nc2ccc(c(c2)Cl)Cl)O)C(=O)O1)C 1M-933 COc1ccc(cc1)NC(=O)CC(=O)Nc2ccc(c(c2)Cl)Cl 1M-934 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)CC(=O)Nc2ccc(c(c2)Cl)Cl 1M-936 c1cc(c(cc1NC(=O)CC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl 1M-937 CCOC(=O)C1=C(NC(=O)CC1)C(F)(F)F 1M-938 CCOC(=O)C12CCCC=C1N(C(=O)CC2)Cc3ccccc3 1M-939 CN(c1ccccc1)C(=O)CC(=O)Nc2ccc(c(c2)Cl)Cl 1M-942 Cc1cnc(nc1)NC(=O)CC(=O)Nc2ccc(c(c2)Cl)Cl 1M-943 c1cc(c(cc1NC(=O)CC(=O)Nc2ccc(cn2)Cl)Cl)Cl 1M-947 c1cc(c(cc1NC(=O)CC(=O)Nc2cnccn2)Cl)Cl 1M-948 c1ccc(c(c1)n2cccc2/C=N/O)F 1N-001 c1ccc(c(c1)n2cccc2C#N)F 1N-002 c1cc(c(cc1c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-])O 1N-003 c1ccc2c(c1)[nH]c(=O)c3n2ccc3 1N-004 c1cc(c(cc1c2c(cc(cn2)C(F)(F)F)Cl)N)O 1N-005 CC(C)c1ccc(cc1)C2CC2/C(=N/O)/C 1N-006 CC(C)c1ccc(cc1)C2CC2/C(=N/OCc3ccc(cc3Cl)Cl)/C 1N-007 Cc1ccc(cc1)C(=O)O/N=C(\C)/C2CC2c3ccc(cc3)C(C)C 1N-011 CC(C)c1ccc(cc1)C2CC2/C(=N/OC(=O)C3CC3)/C 1N-013 Cc1ccc(cc1)C(=O)O/N=C(\C)/C2CC2c3ccc(cc3)OC 1N-014 Cc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)C(C)C(=O)C 1N-015 C/C(=N\OC(=O)c1ccc(cc1)[N+](=O)[O-])/C2CC2c3ccc(cc3)OC 1N-016 CC(C)c1ccc(cc1)C2CC2/C(=N/OCc3ccccc3F)/C 1N-017 CC(C(=O)C)N1C(=O)C(=O)N(C1=O)Cc2cccc(c2)Cl 1N-018 CC(C)c1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccc(cc3)[N+](=O)[O-])/C 1N-019 CC(C)c1ccc(cc1)C2CC2/C(=N/OC(=O)c3cccs3)/C 1N-020 CC(C(=O)C)N1C(=O)C(=O)N(C1=O)Cc2ccccc2C(F)(F)F 1N-021 CC(C)c1ccc(cc1)C2CC2/C(=N/OCCOc3ccccc3)/C 1N-022 CC(C)c1ccc(cc1)C2CC2/C(=N/OCc3c(cccc3Cl)Cl)/C 1N-023 CC(=O)C1CC1c2ccc(cc2)F 1N-029 CSc1ccc(cc1)NC(=S)NC(=O)c2ccccc2 1N-030 CCSc1ncc(n1C)c2cc(c3ccccc3n2)C(=O)O 1N-301S c1ccc(cc1)c2[nH]c(c(n2)/C=N/c3ccc(cc3)Cl)Cl 1N-302S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/O)/C(F)(F)F 1N-304S c1ccc2c(c1)c(cc(n2)c3ccc(cc3)Cl)C(=O)O 1N-306S CC(C)/N=C/c1c([nH]c(n1)c2ccccc2)Cl 1N-307S Cc1ccc(cc1)C/N=C/c2c([nH]c(n2)c3ccccc3)Cl 1N-308S Cc1ccc(cc1)C(=O)O/N=C(/c2cc(n(c2C)c3ccc(cc3)F)c4ccc(cc4)S(=O)(=O)C)\C(F)(F)F 1N-309S c1ccc(cc1)c2[nH]c(c(n2)/C=N/C3CCCCC3)Cl 1N-311S COc1ccc(cc1)C/N=C/c2c([nH]c(n2)c3ccccc3)Cl 1N-312S c1ccc(cc1)c2[nH]c(c(n2)/C=N/Cc3ccc(cc3)Cl)Cl 1N-313S Cn1cc(c(n1)C(F)(F)F)C(=O)NC2CC2 1N-314S Cc1cc(cc(c1)NC(=O)c2cn(nc2C(F)(F)F)C)C 1N-315S Cn1cc(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl 1N-316S Cn1cc(c(n1)C(F)(F)F)C(=O)Nc2cccc(c2)C(F)(F)F 1N-317S Cn1cc(c(n1)C(F)(F)F)c2nnnn2C3CC3 1N-318S Cc1cc(cc(c1)n2c(nnn2)c3cn(nc3C(F)(F)F)C)C 1N-319S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N\OC(=O)c4ccccc4)/C(F)(F)F 1N-320S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/OC(=O)c4ccc(cc4)F)/C(F)(F)F 1N-321S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/OC(=O)c4ccc(cc4)Cl)/C(F)(F)F 1N-322S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/OC(=O)c4cccc(c4)C(F)(F)F)/C(F)(F)F 1N-323S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N\OC(=O)C(C)C)/C(F)(F)F 1N-324S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/OC(=O)C4CC4)/C(F)(F)F 1N-325S CCOC(=O)Nc1cc(nc2c1cccc2)c3ccc(cc3)Cl 1N-327S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/OC(=O)c4ccc(cc4Cl)Cl)/C(F)(F)F 1N-328S Cc1c(cc(n1c2ccc(cc2)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/OC(=O)c4cccc(c4)OC)/C(F)(F)F 1N-329S Cn1cc(c(n1)C(F)(F)F)c2nnnn2c3ccc(cc3)Cl 1N-331S Cn1cc(c(n1)C(F)(F)F)c2nnnn2c3cccc(c3)C(F)(F)F 1N-332S c1ccc(cc1)c2[nH]c(c(n2)/C=N/c3cccc(c3)C(F)(F)F)Cl 1N-335S CC(=O)Nc1c(cc(c(c1Cl)O)Cl)Cl 1N-337S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OC(=O)c3ccc(c(c3)Cl)Cl 1N-502S c1ccnc(c1)c2nc(cc(n2)Cl)CS(=O)(=O)c3ccc(cc3)Cl 1N-503S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OC(=O)c3cccc(c3)Cl 1N-504S CC(C)(C)NC(=S)N1CCOCC1 1N-506S COC(=O)c1c(c(n(n1)c2ccccc2)Cl)/C=N/OC(=O)c3cccc(c3)C(F)(F)F 1N-507S Cn1cnnc1SCC(=O)c2ccc(cc2)Cl 1N-510S Cn1c(c(c(n1)c2ccccc2)/C=N/OC)O 1N-511S Cc1cc(c(cc1Cl)F)C(=O)C 1N-512S Cc1ccc(cc1)/C=N/c2ccc(cc2F)F 1N-529S c1cc(ccc1c2csc(n2)N3CCOCC3)Cl 1N-530S Cn1c(c(c(n1)c2ccccc2)/C=N/O)O 1N-531S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3Cl)Cl)O 1N-532S Cc1ccc(cc1)CSc2nc[nH]n2 1N-538S COc1ccc(cc1)c2csc(n2)N3CCOCC3 1N-539S c1cc(c(cc1Cl)Cl)c2csc(n2)N3CCOCC3 1N-540S c1ccc(cc1)c2csc(n2)N3CCOCC3 1N-541S c1cc(ccc1c2csc(n2)N3CCOCC3)[N+](=O)[O-] 1N-542S COC(=O)c1ccccc1NC(=O)C(F)(F)F 1N-543S CCOC(=O)/C=C/1\c2ccccc2N(C1=O)CC=C 1N-547S COc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)COCc3ccc(cc3)F 1N-551S c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)F)COCc3ccc(cc3)F 1N-552S c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)C(F)(F)F)COCc3ccc(cc3)F 1N-553S CC(C)(C)c1csc(n1)N2CCOCC2 1N-556S CCOC(=O)c1c(nc(s1)N2CCOCC2)C(F)(F)F 1N-557S c1cc(ccc1c2csc(n2)N3CCSCC3)F 1N-559S Cn1cnnc1SC/C(=N\O)/c2ccc(cc2)Cl 1N-564S COc1ccc(cc1)c2csc(n2)N3CCSCC3 1N-565S CCOC(=O)CSc1nc[nH]n1 1N-566S C=CCSc1nc[nH]n1 1N-567S c1cc(ccc1CSc2nc[nH]n2)Cl 1N-568S c1cc(cc(c1)C(F)(F)F)CSc2nc[nH]n2 1N-569S COc1ccc(cc1)CSc2nc[nH]n2 1N-570S CCOC(=O)/C=C/1\c2ccccc2N(C1=O)Cc3ccc(c(c3)Cl)Cl 1N-571S c1ccc(cc1)c2csc(n2)N3CCSCC3 1N-573S CC(C)(C)c1csc(n1)N2CCSCC2 1N-574S Cc1ccc(cc1)CS(=O)(=O)c2nc[nH]n2 1N-575S CNC(=O)CSc1nc[nH]n1 1N-576S COC(=O)c1cc(n(n1)c2ccc(cc2)F)O 1N-577S c1ccc(cc1)/C=C/c2ccnc(n2)S 1N-700 COC(=O)Cc1c(c(sc1C(=O)OC)N)C(=O)OC 1N-703 c1ccc(cc1)Cc2c(ccn(c2=O)Cc3cccs3)O 1N-704 c1ccc(cc1)/C=C/c2ccnc(n2)SC(F)F 1N-708 COC(=O)Cc1c(c(sc1C(=O)OC)NC(=O)c2cccc(c2)Cl)C(=O)OC 1N-709 CC(=O)Nc1c(c(c(s1)C(=O)OC)CC(=O)OC)C(=O)OC 1N-710 CC(=O)Nc1ccc(cc1[N+](=O)[O-])OC 1N-711 COC(=O)Cc1c(c(sc1C(=O)OC)NC(=O)c2ccccc2)C(=O)OC 1N-713 Cc1ccc(c(c1)C)N/C(=C/C(=O)C(F)(F)F)/C=C/N(C)C 1N-715 CCOC(=O)C(Cc1ccccc1)c2ccnc3n2ncn3 1N-716 C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)F 1N-718 C/C(=C/C(=O)C(F)(F)F)/Nc1ccccn1 1N-719 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)F 1N-721 COc1ccc(cc1)Nc2ccnc(c2)C(F)(F)F 1N-722 COC(=O)c1ccccc1Nc2ccnc(c2)C(F)(F)F 1N-723 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1ccccn1 1N-726 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)Oc3ccc(cn3)[N+](=O)[O-] 1N-727 c1cc(ccc1Nc2ccnc(c2)C(F)(F)F)F 1N-728 C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)Cl 1N-729 C/C(=C/C(=O)C(F)(F)F)/Nc1ccccc1Oc2ccccc2 1N-730 Cc1cccc(c1)C(=O)Nc2c(c(c(s2)C(=O)OC)CC(=O)OC)C(=O)OC 1N-731 Cc1c(c(=O)[nH]c(n1)S)CCO 1N-732 C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)C(F)(F)F 1N-733 CN(C)/C=C\C(=C/C(=O)C(F)(F)F)\Nc1ccccc1Oc2ccccc2 1N-734 Cn1cccc1N2C(=O)CCC2=O 1N-735 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)Cl 1N-736 Cc1c(c(=O)[nH]c(n1)SC(F)F)CCO 1N-742 C=C(c1c[nH]c2c1cccc2)c3c[nH]c4c3cccc4 1N-901 B(c1cc(c(cc1F)Cl)OC)(O)O 1N-902 C=C(c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl)c4cn(c5c4cccc5)c6c(cc(cn6)C(F)(F)F)Cl 1N-904 COc1cc2c(cc1OC)ncnc2NCC(c3ccc4ccccc4c3)O 1P-001 c1cc(c(cc1OCc2cnc(s2)Cl)F)Cl 1P-002 COC(=O)c1cccc(c1)OCc2cnc(s2)Cl 1P-003 COC(=O)c1ccccc1OCc2cnc(s2)Cl 1P-004 CN(C)CCCNc1c2cc(c(cc2ncn1)OC)OC 1P-005 Cn1cnc(c1C#N)C#N 1P-006 COc1cc2c(cc1OC)ncnc2NCc3cccnc3 1P-007 c1ccc(cc1)Oc2ccccc2/C=C\C(=O)N 1P-008 c1ccc(cc1)c2cc(on2)C(=O)C/C=N/OCc3ccc(cc3)Cl 1P-009 c1ccc(cc1)c2cc(on2)C(=O)C/C=N/OCc3ccc(cc3)F 1P-010 c1ccc(c(c1)C=O)OCc2cnc(s2)Cl 1P-012 c1cc(ccc1C=O)OCc2cnc(s2)Cl 1P-013 CCOC(=O)C1CCN(CC1)c2ncc(s2)/C=N/NC(=O)c3ccncc3 1P-015 CCOC(=O)C1CCN(CC1)c2ncc(s2)/C=N/NC(=O)c3ccc(cc3)OCc4ccc(cc4)C 1P-016 CCOC(=O)C1CCN(CC1)c2ncc(s2)/C=N/NC(=O)c3ccc(cc3Cl)Cl 1P-017 CC1CN(CC(O1)C)c2ncc(s2)/C=N/NC(=O)c3ccccc3O 1P-018 c1ccc(cc1)c2cc(on2)C(=O)C/C=N/OCc3ccc(cc3)[N+](=O)[O-] 1P-019 c1ccc(cc1)Oc2ccccc2N/N=C/c3cnc(s3)N4CCOCC4 1P-021 COc1cc2c(cc1OC)ncnc2NCc3cc(ccc3F)F 1P-022 CO/N=C/CC(=O)c1cc(no1)c2ccccc2 1P-023 c1ccc(cc1)c2cc(on2)C(=O)C/C=N/OCc3ccc(cc3Cl)Cl 1P-025 CCOc1ccc(cc1/C=N/NC(=O)c2ccc(cc2Cl)Cl)Br 1P-026 CCOc1ccc(cc1/C=N/NC(=O)c2ccccc2O)Br 1P-027 CCOc1ccc(cc1/C=N/NC(=O)c2ccncc2)Br 1P-028 CCOc1ccc(cc1/C=N/NC(=O)c2cccnc2)Br 1P-029 c1ccc(c(c1)C=O)Oc2ccc(c(c2)F)F 1P-030 COC(=O)c1cccc(c1)OCc2ccc(cc2Cl)Cl 1P-031 c1ccc(c(c1)/C=N/NC(=O)c2ccc(cc2)OCc3c(cccc3Cl)F)O 1P-032 c1cc(ccc1C#N)Oc2ccc(cc2Cl)Cl 1P-033 c1ccc(cc1)Oc2ccccc2/C=C\3/C(=O)NC(=O)S3 1P-034 c1ccc(c(c1)/C=C\2/C(=O)NC(=O)S2)Oc3ccc(cc3)Cl 1P-035 CCOc1ccc(cc1/C=C\2/C(=O)NC(=O)S2)Br 1P-036 c1ccc(c(c1)C=O)Oc2ccc(c(c2)F)Cl 1P-038 c1cc(ccc1/C=N/NC(=O)c2ccc(cc2Cl)Cl)OCc3cnc(s3)Cl 1P-041 c1ccc(c(c1)/C=C\2/C(=O)NC(=O)S2)Oc3ccc(cc3)F 1P-042 CC(C)(C)c1ccc(cc1)Oc2ccccc2/C=C\3/C(=O)NC(=O)S3 1P-043 c1cc(ccc1/C=N/NC(=O)c2ccncc2)OCc3cnc(s3)Cl 1P-044 CC(C)(C)OC(=O)N\1CCOC(=O)/C1=C/C(=O)OC 1P-046 c1ccc(c(c1)C=O)Oc2ccc(cc2F)Br 1P-047 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccc(cc2)F 1P-050 c1ccc(c(c1)/C=C/C(=O)O)Oc2cccc(c2)Cl 1P-051 c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)OCc3cnc(s3)Cl 1P-052 c1ccc(cc1)N2CCN(CC2)c3ncc(s3)/C=N/NC(=O)c4cccnc4 1P-053 Cc1ccn2cc(nc2c1)c3ccccc3 1P-054 CCOC(=O)c1c(c2cccc3c2n(c1=O)CC3)OC(=O)C 1P-055 c1cc(ccc1c2nnco2)OCc3ccc(c(c3)Cl)Cl 1P-057 CCOc1ccc(cc1/C=N/NC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl)Br 1P-058 c1ccc(cc1)N2CCN(CC2)c3ncc(s3)C=C(C#N)C#N 1P-059 c1ccc(cc1)COc2ccc(cc2)Oc3ccccc3C=O 1P-060 Cc1ccc(cc1)COc2ccc(cc2)c3nnco3 1P-061 c1ccc(c(c1)/C=N/NC(=O)c2cccnc2)OCc3cnc(s3)Cl 1P-062 c1ccc(c(c1)C=C(C#N)C#N)OCc2cnc(s2)Cl 1P-063 c1ccc(c(c1)/C=N/NC(=O)c2ccc(cc2)C(F)(F)F)Oc3ccc(cc3)Cl 1P-064 c1ccc(cc1)Oc2ccccc2/C=N/NC(=O)c3ccc(cc3)C(F)(F)F 1P-065 CCOc1ccc(cc1/C=N/NC(=O)c2ccc(cc2)C(F)(F)F)Br 1P-066 CN(C)c1cccc(c1)NC(=S)NC(=O)c2ccccc2 1P-067 COc1ccc(cc1)Oc2ccc(cc2)CN 1P-068 CN1CCN(CC1)c2ncc(s2)/C=N/NC(=O)c3ccc(cc3)C(F)(F)F 1P-070 COc1ccc(cc1)NNC(=S)N 1P-071 Cc1ccccc1NNC(=S)N 1P-072 c1cc(ccc1/C=N/NC(=O)c2ccc(cc2)C(F)(F)F)OCc3cnc(s3)Cl 1P-075 c1ccc2c(c1)C(=O)N(C2=O)CCOc3ccc(cc3Cl)Cl 1P-076 c1ccc2c(c1)c(c[nH]2)/C=N/NC(=O)c3c(c4cccc5c4n(c3=O)CCC5)O 1P-077 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)N/N=C/c4ccc[nH]4)O 1P-078 c1cc(cc(c1)O)/C=N/NC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O 1P-079 c1c(sc(n1)N2CCCCC2)C=C(C#N)C#N 1P-080 c1cc(ccc1C(=O)N/N=C/c2cnc(s2)N3CCCCC3)C(F)(F)F 1P-081 c1ccc(cc1)Oc2ccccc2/C=N/NC(=O)c3c(c4cccc5c4n(c3=O)CCC5)O 1P-082 COC(=O)/C(=C/c1cnc(s1)N2CCCCC2)/C#N 1P-083 Cc1cc(cc(c1)Oc2ccccc2/C=C/C(=O)O)C 1P-084 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccc(c(c2)F)F 1P-085 Cc1ccn2c(c1)nc(c2CO)c3ccccc3 1P-086 CCO/C=N/NC(=O)c1c(c2cccc3c2n(c1=O)CCC3)O 1P-087 Cc1ccc(cc1)Oc2ccccc2/C=N/NC(=O)c3ccc(cc3)C(F)(F)F 1P-089 c1ccc(c(c1)/C=N/NC(=O)c2ccc(cc2)C(F)(F)F)Oc3ccc(cc3)F 1P-090 c1ccc(cc1)c2cn3cc(ccc3n2)Cl 1P-091 CCOC(=O)C=C(C(=O)OCC)C(=O)OCC 1P-093 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccc(c(c2)F)Cl 1P-095 c1ccc(cc1)COc2ccc(cc2)Oc3ccccc3/C=C/C(=O)O 1P-096 c1cc(ccc1C#N)Oc2ccc(c(c2)F)Cl 1P-097 C/C(=N\NC(=O)N)/c1ccccc1 1P-098 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccc(cc2F)Br 1P-099 COc1cc2c(cc1OC)ncnc2NCC3CC3 1P-101 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(c(c2)C(F)(F)F)Cl 1P-102 Cc1ccc(c(c1)C)Oc2ccc(cc2)C#N 1P-103 c1cc(c(cc1NC(=S)N)C(F)(F)F)Cl 1P-104 CCOc1c(cc(cn1)[N+](=O)[O-])C(=O)O 1P-105 c1ccc(c(c1)C=O)Oc2ccc(cc2)I 1P-106 c1ccc2c(c1)NC(=O)CS2(=O)=O 1P-302S C=CCNc1[nH]c(=O)c2ccccc2n1 1P-303S c1ccc(c(c1)CSC2=Nc3ccccc3SC2)Cl 1P-305S CC1=C(C(=O)N(CO1)C(C)(C)C(=O)O)c2ccccc2F 1P-312S Cc1ccc(cc1)C(=O)Nc2ccccc2SCC3CSc4n3c(=O)c5ccccc5n4 1P-321S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccccc4NC(=O)c5ccc(cc5)F 1P-328S c1ccc2c(c1)c(=O)[nH]c(n2)N3CCCC3 1P-330S c1ccc(cc1)CSC2=CS(=O)(=O)c3ccccc3N2 1P-331S CN1CCN(CC1)c2[nH]c(=O)c3ccccc3n2 1P-333S c1ccc(cc1)C(=O)Nc2ccccc2SCC3CSc4n3c(=O)c5ccccc5n4 1P-335S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccccc4NC(=O)c5cccc(c5)Cl 1P-336S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccccc4NC(=O)c5ccccc5Cl 1P-338S COc1ccccc1C(=O)Nc2ccccc2SCC3CSc4n3c(=O)c5ccccc5n4 1P-339S Cc1cccc(c1)C(=O)Nc2ccccc2SCC3CSc4n3c(=O)c5ccccc5n4 1P-340S c1ccc2c(c1)c(=O)n3c(n2)SCC3CSc4ccccc4NC(=O)c5cccc(c5)C(F)(F)F 1P-341S CC(C)Nc1[nH]c(=O)c2ccccc2n1 1P-344S CCCNc1[nH]c(=O)c2ccccc2n1 1P-345S c1ccc2c(c1)NC(=CS2(=O)=O)SCc3cccc(c3)C(F)(F)F 1P-353S COc1ccc(cc1)CSC2=CS(=O)(=O)c3ccccc3N2 1P-354S Cc1cccc(c1)CSC2=CS(=O)(=O)c3ccccc3N2 1P-355S c1ccc2c(c1)NC(=CS2(=O)=O)SCc3cccc(c3)Cl 1P-357S c1ccc2c(c1)NC(=CS2(=O)=O)SCc3cccc(c3)F 1P-358S c1ccc2c(c1)NC(=CS2(=O)=O)SCc3ccc(c(c3)Cl)Cl 1P-359S Cc1ccc(cc1)CSC2=CS(=O)(=O)c3ccccc3N2 1P-360S COc1ccc(cc1)Nc2[nH]c(=O)c3ccccc3n2 1P-363S c1ccc2c(c1)c(=O)[nH]c(n2)Nc3ccc(cc3)Cl 1P-365S c1ccc2c(c1)c(=O)[nH]c(n2)Nc3ccc(cc3F)F 1P-366S CC(C)(C)c1ccc(cc1)CSC2=CS(=O)(=O)c3ccccc3N2 1P-367S c1ccc2c(c1)NC(=CS2(=O)=O)SCc3c(cccc3Cl)F 1P-369S c1ccc2c(c1)NC(=CS2(=O)=O)SCc3ccc(cc3)F 1P-370S c1ccc2c(c1)NC(=CS2(=O)=O)SCc3ccc(cc3Cl)Cl 1P-371S Cc1ccc(cc1C)Nc2[nH]c(=O)c3ccccc3n2 1P-374S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)Cc4cccs4 1P-377S Cn1c2ccccc2c3c1sc(c3)C(=O)NNC(=O)c4cccc(c4)Cl 1P-378S COC(=O)c1ccc2c(c1)N(C(=O)CS2)Cc3ccc(cc3Cl)Cl 1P-501S COC(=O)c1ccc2c(c1)N(C(=O)CS2)Cc3ccccc3 1P-502S CCOC(=O)c1cnc(nc1N(C)CC#N)SC 1P-503S COC(=O)c1c(noc1C(=O)OC)c2ccc(cc2)Cl 1P-510S c1ccc2c(c1)nc(s2)N3CCOCC3 1P-511S Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)c3ccccc3 1P-514S c1ccc(cc1)C(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 1P-515S c1ccc(cc1)C(=O)NC2CCN(CC2)S(=O)(=O)c3cccc(c3)C(F)(F)F 1P-516S COc1ccc(c(c1)S(=O)(=O)N2CCC(CC2)NC(=O)c3ccccc3)OC 1P-517S COC(=O)c1ccccc1S(=O)(=O)N2CCC(CC2)NC(=O)c3ccccc3 1P-518S c1ccc(c(c1)N)SCC(=O)Nc2ccc(cc2Cl)Cl 1P-521S COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)c3ccccc3 1P-522S c1ccc(cc1)C(=O)NC2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)Cl 1P-523S c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)Cl)SCC(=O)Nc3ccc(cc3Cl)Cl 1P-526S Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3ccc(cc3Cl)Cl 1P-527S COc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3ccc(cc3Cl)Cl 1P-528S COC(=O)c1ccc2c(c1)N(C(=O)CS2)Cc3cccc(c3)Cl 1P-529S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2N 1P-531S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NS(=O)(=O)c3ccc(cc3)F 1P-532S COc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3ccsc3C(=O)OC 1P-533S c1ccc(c(c1)NS(=O)(=O)c2cc(ccc2Cl)Cl)SCC(=O)Nc3ccc(cc3Cl)Cl 1P-534S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NS(=O)(=O)c3ccc(cc3)Cl 1P-536S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NS(=O)(=O)c3cc(ccc3Cl)Cl 1P-537S COC(=O)c1ccccc1SCC(=O)Nc2ccsc2C(=O)OC 1P-538S COC(=O)c1c(ccs1)NC(=O)CSc2ccc(cc2)Br 1P-539S COC(=O)c1c(ccs1)NC(=O)COc2ccc(cc2Br)Cl 1P-540S COC(=O)c1c(ccs1)NC(=O)COc2ccsc2C(=O)OC 1P-541S CC(C)(C)OC(=O)N1CCC(=O)CC1 1P-563S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)C=O 1P-565S COc1ccc(cc1)n2c(cc3c2CCC(=C3Sc4ccc(cc4)Br)C=O)c5ccccc5 1P-571S COc1ccc(cc1)n2c(cc3c2CCC(=C3Sc4ccc(cc4)Cl)C=O)c5ccccc5 1P-572S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/c6ccc(cc6)OC 1P-574S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/O 1P-577S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/c6ccc(cc6)Cl 1P-578S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/C6CCCCC6 1P-579S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/C(C)C 1P-580S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/c6ccc(cc6F)F 1P-581S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/c6ccc(cc6)Br 1P-582S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/C6CC6 1P-585S C1CCNC(C1)C(=O)N 1P-588S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/c6ccccc6 1P-589S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/c6cc(cc(c6)C)C 1P-590S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)/C=N/c6ccc(cc6)F 1P-593S COc1ccc(cc1)n2c(cc3c2CCC(=C3Sc4ccc(cc4)F)C=O)c5ccccc5 1P-597S COc1ccc(cc1)n2c(cc3c2CCC(=C3Sc4cccc(c4)OC)C=O)c5ccccc5 1P-598S COc1ccc(cc1)n2c(cc3c2CCC(=C3Sc4cccc(c4Cl)Cl)C=O)c5ccccc5 1P-599S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])COC(=O)Nc4ccc(cc4Cl)Cl 1P-641S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])COC(=O)Nc4cccc(c4)Cl 1P-642S c1ccc(cc1)NC(=O)OCc2ccc(c(c2)[N+](=O)[O-])Sc3nc4ccccc4s3 1P-643S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CN3CCN(CC3)c4cccc(c4)Cl 1P-644S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CN3CCN(CC3)C(c4ccccc4)c5ccccc5 1P-645S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])CN3CCOCC3)Cl 1P-646S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])CN3CCCCC3)Cl 1P-647S c1ccc(c(c1)N2CCN(CC2)Cc3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl)F 1P-649S c1cc(cc(c1)Cl)N2CCN(CC2)Cc3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl 1P-650S c1ccc(cc1)CN2CCN(CC2)Cc3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl 1P-651S c1cnc(nc1)N2CCN(CC2)Cc3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl 1P-652S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])CN3CCCC3)Cl 1P-653S COc1ccc(cc1)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-654S CN1CCN(CC1)Cc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-655S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CN3CCCCC3 1P-656S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CN3CCCC3 1P-657S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)Cc4ccc(c(c4)[N+](=O)[O-])Sc5ccc(cc5)Cl 1P-658S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CN3CCN(CC3)c4ncccn4 1P-659S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CN3CCN(CC3)Cc4ccccc4 1P-660S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])CN4CCOCC4 1P-661S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])CN4CCN(CC4)c5ncccn5 1P-662S c1cc(ccc1OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)F 1P-664S c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])COc3cc(ccc3Cl)Cl)Cl 1P-665S Cc1ccc(cc1)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-666S Cc1cccc(c1C)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-667S c1cc(cc(c1)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)C(F)(F)F 1P-668S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])COc4ccc(cc4F)F 1P-669S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])COc4cc(c(cc4Cl)Cl)Cl 1P-670S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])COc4cccc(c4)C(F)(F)F 1P-671S COC(=O)c1c(ccs1)OCc2ccc(c(c2)[N+](=O)[O-])Sc3nc4ccccc4s3 1P-674S c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])COc4ccc(cc4Cl)Cl 1P-677S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COc3cccc(c3)C(F)(F)F 1P-678S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COc3cccc(c3)Cl 1P-679S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COc3cc(ccc3Cl)Cl 1P-680S Cc1ccc(cc1)OCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)C 1P-681S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COc3ccc(cc3)F 1P-682S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])COc3ccc(cc3Cl)Cl 1P-683S c1cc(c(c(c1)Cl)SCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)Cl 1P-684S COC(=O)c1ccccc1SCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-685S c1ccc(cc1)SCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-686S c1cc(ccc1F)SCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-687S Cc1ccc(cc1)SCc2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl 1P-688S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CSc3ccc(cc3)Cl 1P-689S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CSc3cc(ccc3Cl)Cl 1P-690S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CSc3ccccc3C(=O)OC 1P-691S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CSc3ccc(cc3)F 1P-692S Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CSc3ccc(cc3)Br 1P-693S c1ccc2c(c1)CCC(=C2Cl)/C=N/O 1P-694S CCn1c(nnc1S)c2cc3c(s2)-c4ccccc4CC3 1P-695S c1cc(cc(c1)Cl)Cn2ccc(c(c2=O)Cc3c(cccc3Cl)F)O 1P-700 c1cc(oc1)C(=O)n2c(nc(n2)Br)Br 1P-703 C1=CC(C(C(C1O)Br)Br)O 1P-704 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)Cc3ccc(cc3)S(=O)(=O)N)O)F 1P-705 c1ccc2c(c1)c(c[nH]2)CCn3ccc(c(c3=O)Cc4c(cccc4Cl)F)O 1P-706 CCOC(=O)Cn1c(nc(n1)Br)Br 1P-707 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)CCCn3ccnc3)O)F 1P-709 COc1ccc(c(c1Cc2c(cccc2Cl)F)OC)C=O 1P-710 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)Nc3c(cccn3)[N+](=O)[O-])O)F 1P-712 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)Cc3ccc4c(c3)OCO4)O)F 1P-713 C(C#N)n1c(nc(n1)Br)Br 1P-716 c1cc(ccc1COn2ccnc2)Br 1P-718 COC(=O)CCCCOn1ccnc1 1P-719 CC(C)(Cn1ccc(c(c1=O)Cc2ccccc2)O)SCc3ccc(cc3)F 1P-720 COc1ccc(c(c1Cc2c(cccc2Cl)F)OC)/C=C(/C#N)\C(=O)c3ccccc3 1P-721 c1cc(ccc1C/N=C\c2ccc3c(c2)OCO3)F 1P-723 CCOC(=O)C(Cc1c(cccc1Cl)F)C(=O)C/C=N/OCc2ccc(cc2Cl)Cl 1P-727 c1ccc2c(c1)c(c[nH]2)CCn3cc(c(c(c3=O)Cc4c(cccc4Cl)F)O)/C=N/OCc5ccc(cc5Cl)Cl 1P-729 c1cc(c(c(c1)Cl)Cc2c(c(cn(c2=O)CCc3ccc(cc3)S(=O)(=O)N)/C=N/OCc4ccc(cc4Cl)Cl)O)F 1P-730 CCOC(=O)C(Cc1ccccc1)c2ccnc3n2nc(n3)N 1P-731 CCOC(=O)C(Cc1ccccc1)c2ccnc3n2nc(n3)n4c(ccc4C)C 1P-732 c1cn(cn1)OCCCCC(=O)O 1P-733 c1ccc(cc1)CN2CCCCCC2=O 1P-734 CN(c1ccc(cc1)Cl)c2ccnc(c2)C(F)(F)F 1P-735 c1c(cnc(c1Cl)N2CCCCCC2=O)C(F)(F)F 1P-736 CCOC(=O)C(Cc1ccccc1)c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 1P-737 c1cc(c(c(c1)Cl)Cc2c(ccn(c2=O)C3CCCCCC3)O)F 1P-738 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccc(n2)Nc3c(cc(cn3)C(F)(F)F)Cl 1P-742 c1cc(nc(c1)NC(=O)c2ccc(c(c2)Cl)Cl)Nc3c(cc(cn3)C(F)(F)F)Cl 1P-743 C#CCc1c(ccn(c1=O)Cc2ccc3c(c2)OCO3)O 1P-745 CCOC(=O)C(CC#C)c1ccnc2n1nc(n2)N 1P-746 CCOC(=O)C(Cc1ccccc1)c2ccno2 1P-747 c1ccc(cc1)CCOn2ccnc2 1P-748 CC(C)(C)c1ccc(cc1)COn2ccnc2 1P-749 Cc1cccc(c1)COn2ccnc2 1P-750 Cc1cc(cc(c1)COn2ccnc2)C 1P-751 CN(C)CCCNC1=NC=NC2C1C=CC(=C2)Cl 1P-801 CC(=O)c1ccc(c(c1)F)c2ccccc2 1P-803 c1cc2c(cc1Cl)ncnc2Nc3ccncc3 1P-804 Cc1c(c(nc(n1)C)O)I 1P-805 CN(C(=O)Nc1ccc(cc1)Cl)O 1P-806 c1ccc2cc(ccc2c1)C(CNc3c4ccc(cc4ncn3)Cl)O 1P-808 c1cc(c(cc1F)CNc2c3ccc(cc3ncn2)Cl)F 1P-809 CCOC(=O)c1[nH]c(=O)c2ccccc2n1 1P-813 CC(=O)C(=Cc1ccc(cc1)C(=O)O)C(=O)C 1P-814 CCOC(=O)CC1N(C(=O)N(O1)C)c2ccc(cc2)Cl 1P-815 CN(C(=O)Nc1ccc(cc1Cl)Cl)O 1P-816 c1cc(cnc1)CNc2c3ccc(cc3ncn2)Cl 1P-817 COc1ccc(cc1)S(=O)(=O)NC(Cc2ccc(cc2)C#N)C(=O)O 1P-822 c1ccc(cc1)S(=O)(=O)NC(Cc2ccc(cc2)C#N)C(=O)O 1P-823 CCOC(=O)CC1N(C(=O)N(O1)C)c2ccc(cc2Cl)Cl 1P-827 CC1=C(C(n2c(ncn2)N1)c3ccc(cc3)C(=O)O)C(=O)C 1P-828 Cc1c(c(nc(n1)C)Cl)I 1P-829 CN(C(=O)Nc1ccc(cc1)[N+](=O)[O-])O 1P-830 CN(C(=O)Nc1cccc(c1)Cl)O 1P-831 c1ccc2c(c1)CN(C2=O)C(Cc3ccc(cc3)C#N)C(=O)O 1P-832 c1cc(ccc1CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)Cl)C#N 1P-833 c1cc2c(cc1Cl)ncnc2NCC3CC3 1P-834 CCOC(=O)CC1N(C(=O)N(O1)C)c2ccc(cc2)[N+](=O)[O-] 1P-836 COC(=O)CNC(=O)C1CCN(CC1)C(=O)OCc2ccccc2 1P-915 COc1cnc(o1)C(=O)OC 1P-956 COC(=O)c1c(cnc(c1C(=O)OC)C(=O)OC)O 1P-960 CCOC(=O)c1c2ccccn2cc1c3ccc(cc3)c4ccccc4 1R-0001 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCC(=O)O 1R-0002 c1ccn2cc(c(c2c1)C(=O)O)c3ccc(cc3)Cl 1R-0003 c1ccn2cc(c(c2c1)C(=O)O)C(=O)O 1R-0004 COC(c1ccnc(n1)c2ccc(cc2)O)OC 1R-0008 c1cc(ccc1C#N)Oc2ccc(cc2Br)[N+](=O)[O-] 1R-0010 c1cc(ccc1c2ncc3c(n2)CCCC3=O)O 1R-0011 CCOC(=O)C/C(=N\NC(=O)CC#N)/CCl 1R-0012 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2cccc(c2Cl)Cl 1R-0015 COC(c1ccnc(n1)c2ccc(cc2)OC(=O)c3ccco3)OC 1R-0016 COC(c1ccnc(n1)c2ccc(cc2)OC(=O)c3cccs3)OC 1R-0017 COC(c1ccnc(n1)c2ccc(cc2)OC(=O)c3ccc(cc3)F)OC 1R-0018 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(cc2)OCCCF)Cl 1R-0021 c1cc(c(cc1[N+](=O)[O-])Br)Oc2ccc(c(c2)Cl)Cl 1R-0022 CC(=O)Oc1ccc(cc1)c2nccc(n2)C(OC)OC 1R-0023 c1cc(cc(c1)Cl)Oc2ccc(cc2Br)[N+](=O)[O-] 1R-0024 c1cc(c(c(c1)Cl)Cl)C(=O)c2cc([nH]c2)C(=O)N3CCN(CC3)c4ccc(c(c4)Cl)Cl 1R-0025 c1ccc(c(c1)N2CCN(CC2)C(=O)c3cc(c[nH]3)C(=O)c4cccc(c4Cl)Cl)F 1R-0026 c1ccc(cc1)COc2ccc(cc2)/C=C/C(=O)O 1R-0027 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=C/C(=O)O 1R-0028 c1cc(ccc1COc2ccc(cc2)/C=C/C(=O)O)Br 1R-0029 c1cc(ccc1/C=C/C(=O)O)OCc2ccc(cc2Cl)Cl 1R-0030 COC(c1ccnc(n1)c2ccc(cc2)OC(=O)c3ccc(cc3)[N+](=O)[O-])OC 1R-0031 c1cc(c(c(c1)Cl)Cl)C(=O)c2cc([nH]c2)C(=O)NCc3cccs3 1R-0032 CCCC(=O)Oc1ccc(cc1)c2nccc(n2)C(OC)OC 1R-0033 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2c(cccc2Cl)Cl 1R-0034 c1cc(c(c(c1)Cl)C(=O)c2cc([nH]c2)C(=O)NCc3cccs3)Cl 1R-0035 Cc1cc(n(n1)C(=O)/C(=N/Nc2ccccc2[N+](=O)[O-])/C#N)C 1R-0037 COc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OCCCF 1R-0038 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Cl)OCCCF 1R-0039 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)c4nccc(n4)C(OC)OC 1R-0040 c1cc(c(c(c1)Cl)C(=O)c2cc([nH]c2)C(=O)NC3CCCC3)Cl 1R-0041 c1cc(c(c(c1)Cl)Cl)C(=O)c2cc([nH]c2)C(=O)NCc3ccc(cc3)F 1R-0042 COC(c1ccnc(n1)c2ccc(cc2)OC(=O)c3ccccc3)OC 1R-0043 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)NC3CCCC3)F 1R-0044 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2ccccc2F 1R-0045 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)NCc3cccs3 1R-0046 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)Cc2ccccc2 1R-0047 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)NC3CCCC3 1R-0048 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/C(=O)O)F 1R-0049 CCOC(=O)C/C(=N/NC(=O)/C(=N/Nc1ccccc1[N+](=O)[O-])/C#N)/C 1R-0050 c1cc(c(cc1[N+](=O)[O-])Br)Oc2ccc(cc2Cl)Br 1R-0051 c1cc(c(cc1[N+](=O)[O-])Br)Oc2cc(cc(c2)Cl)Cl 1R-0052 c1cc(ccc1c2nccc(n2)C=O)O 1R-0053 CC1=C(CC(=C(C1)C(=O)O)C(=O)O)C 1R-0056 COCCCNC(=O)c1cc(c[nH]1)C(=O)Cc2ccccc2 1R-0057 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)N4CCOCC4 1R-0060 COCCCNC(=O)COc1ccc(cc1)c2nccc(n2)c3ccccn3 1R-0062 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 1R-0063 Cc1cc(n(n1)C(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/C#N)C 1R-0064 c1cc(oc1)C(=O)Oc2ccc(cc2)c3nccc(n3)C=O 1R-0066 CN(C)CCCNC(=O)/C=C/c1ccc(cc1)OCc2c(cccc2Cl)F 1R-0070 c1cc(ccc1Sc2ccc(cc2Br)[N+](=O)[O-])Br 1R-0071 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)N3CCSCC3 1R-0072 c1ccc2c(c1)C3=NC(=O)CN3C(=S)N2 1R-0073 CN(C)/C=C(/C#N)\C(=O)Nc1cc(cc(c1)Cl)Cl 1R-0076 c1cc(ccc1/C=N/OCc2ccc(cc2Cl)Cl)OCCCF 1R-0078 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NCc3ccc(cc3)Cl)F 1R-0079 CC1(OC(=O)C(=Cc2ccc(cc2)OCCCF)C(=O)O1)C 1R-0082 COCCCNC(=O)/C=C/c1ccc(cc1)OCc2c(cccc2Cl)F 1R-0083 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/C(=O)N3CCOCC3)F 1R-0084 c1cc(ccc1/C=N/NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)OCCCF 1R-0086 CCOC(=O)c1c2ccccn2cc1c3ccc(cc3)F 1R-0087 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NCc3cccs3)F 1R-0090 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NC3CCCCCC3)F 1R-0091 Cc1ccc(cc1)/C=N/Nc2c(nc3ccccc3n2)C 1R-0092 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NC3CCCC3)F 1R-0093 Cc1c(nc2ccccc2n1)N/N=C/c3ccc(cc3)Br 1R-0094 Cc1ccc(cc1)CNC(=O)/C=C/c2ccc(cc2)OCc3c(cccc3Cl)F 1R-0095 Cc1c(nn(c1C)C(=O)/C(=C/N(C)C)/C#N)C 1R-0096 c1ccc(cc1)C(=O)Oc2ccc(cc2)c3nccc(n3)C=O 1R-0097 CC(C)(C)OC(=O)NC(CSc1c(cc(cn1)C(F)(F)F)Cl)C(=O)O 1R-0100 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NCc3ccc(cc3)F)F 1R-0101 CCCc1c(nn(c1C)C(=O)/C(=N/Nc2ccccc2[N+](=O)[O-])/C#N)C 1R-0102 COc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)OCc3c(cccc3Cl)F 1R-0103 CC/C(=N\NC(=O)CC#N)/CC(=O)C(F)(F)F 1R-0104 CC/C(=N\NC(=O)/C(=N/Nc1ccccc1[N+](=O)[O-])/C#N)/CC(=O)C(F)(F)F 1R-0105 c1cc(cc(c1)Cl)CNC(=O)/C=C/c2ccc(cc2)OCc3c(cccc3Cl)F 1R-0106 c1cc(ccc1C(=O)OCC(=O)c2ccc(cc2)F)O 1R-0107 CCC/C(=N\NC(=O)CC#N)/CC(=O)OCC 1R-0108 Cc1cc(n(n1)C(=O)/C(=N/Nc2ccccc2Br)/C#N)C 1R-0109 Cc1ccccc1NC(=O)/C=C/c2ccc(cc2)OCc3c(cccc3Cl)F 1R-0111 CCOC(=O)Cc1cccc[n+]1Cc2ccccc2.[Br-] 1R-0112 CCOC(=O)/C=C/1\C=CC=CN1Cc2ccccc2 1R-0114 CCCCCCCCOc1ccc(cc1)c2nccc(n2)c3ccc(cc3)F 1R-0115 CCOC(=O)Cc1cccc[n+]1Cc2ccc(cc2)C(F)(F)F.[Br-] 1R-0119 Cc1c(nn(c1C)C(=O)/C(=N/Nc2ccccc2[N+](=O)[O-])/C#N)C 1R-0122 c1cc(oc1)c2ccnc(n2)c3ccc(c(c3)F)I 1R-0127 c1cc(c(cc1c2nccc(n2)/C=C\c3ccc(cc3Cl)Cl)F)I 1R-0128 c1ccc(cc1)c2ccc(cc2)c3ccnc(n3)c4ccc(c(c4)F)I 1R-0129 C/C(=N\NC(=O)/C(=N/Nc1ccccc1[N+](=O)[O-])/C#N)/CC(=O)C(F)(F)F 1R-0131 CC(C)(C)OC(=O)NC(CSCC(=O)NCCc1ccccc1)C(=O)O 1R-0133 Cc1cccc(c1C)Oc2c(nc3ccccc3n2)C 1R-0135 Cc1c(nc2ccccc2n1)Oc3ccc(c(c3)F)Cl 1R-0136 CCOC(=O)C(CSCC(=O)c1ccc(cc1)Br)[NH3+].C(=O)(C(F)(F)F)[O-] 1R-0137 COC(=O)c1c(ccs1)n2cccc2 1R-0138 CCOC(=O)/C=C/1\C=CC=CN1Cc2ccc(cc2)C(F)(F)F 1R-0139 c1cc(ccc1Oc2ccc(cc2Br)[N+](=O)[O-])Br 1R-0140 CCOC(=O)Cc1cccc[n+]1Cc2ccc(cc2)Br.[Br-] 1R-0141 COC(=O)/C=C/c1cc2ccccc2nc1 1R-0147 c1cc(ccc1c2nccc(n2)C=O)OC(=O)c3ccc(cc3)F 1R-0150 c1cc(sc1)C(=O)Oc2ccc(cc2)c3nccc(n3)C=O 1R-0151 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(cc1)F 1R-0152 COC(c1ccnc(n1)c2ccc(c(c2)F)I)OC 1R-0154 CC(=O)c1c2ccccn2c(c1OC(=O)C)c3ccc(cc3)C(F)(F)F 1R-0155 CCCCCCCCOc1ccc(cc1)c2nccc(n2)c3ccco3 1R-0156 c1cc(ccc1C(=O)OCC(=O)c2ccc(cc2)Cl)O 1R-0159 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)[N+](=O)[O-])OCCCF 1R-0160 Cc1ccc(n1c2ccccc2N)C 1R-0166 c1ccc(cc1)N2CCN(CC2)Cc3ccc(cc3)OCCCF 1R-0167 CCOC(=O)C(=Cc1ccnc(n1)c2ccc(cc2)OC(=O)c3ccco3)C(=O)OCC 1R-0168 c1ccc(cc1)N/N=C/c2ccnc(n2)c3ccc(cc3)OC(=O)c4ccc(cc4)F 1R-0169 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)Cc4ccc(cc4)OCCCF 1R-0171 CCOC(=O)c1c2ccccn2cc1c3ccccc3Cl 1R-0172 CCCCCCCCOc1ccc(cc1)c2nccc(n2)C(OC)OC 1R-0173 CCC(CC)(/C(=N/NC(=O)CC#N)/C)C(=O)OCC 1R-0174 CCOC(=O)C(Cc1ccccc1)/C(=N/NC(=O)CC#N)/C 1R-0175 c1ccc(c(c1)N2CCN(CC2)Cc3ccc(cc3)OCCCF)F 1R-0180 c1cc(ccc1CNCC#N)F 1R-0185 c1ccn(c1)c2ccsc2C(=O)CC#N 1R-0188 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)/C=C/c4ccc(cc4)OCCCF 1R-0189 CC(=O)c1ccc(cc1)OCc2c(cccc2Cl)F 1R-0190 Cc1ccc(n1c2ccsc2C(=O)OC)C 1R-0192 CCOC(=O)C1Cc2c3ccccc3ccc2O1 1R-0193 c1cc(ccc1CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])OCCCF 1R-0194 COC(=O)/C(=C/c1ccnc(n1)c2ccc(cc2)OC(=O)c3cccs3)/C#N 1R-0195 c1cc(cc(c1)Cl)CNCC#N 1R-0196 c1ccc2c(c1)ccc3c2CC(O3)C(=O)O 1R-0197 c1cc(ccc1CNC(=O)/C=C/c2ccc(cc2)OCCCF)Cl 1R-0198 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCCCF 1R-0199 Cc1ccc(n1c2ccccc2NC(=O)C)C 1R-0201 Cc1ccc(cc1)CNC(=O)/C=C/c2ccc(cc2)OCc3cccc(c3)Cl 1R-0203 CN(C)/C=C/C(=O)c1ccc(cc1)OCc2c(cccc2Cl)F 1R-0204 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NCc3cccs3 1R-0205 c1cc(cc(c1)Cl)CNC(=O)/C=C/c2ccc(cc2)OCc3cccc(c3)Cl 1R-0206 COc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)OCc3c(cccc3Cl)F 1R-0208 c1cc(c(c(c1)Cl)COc2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3)C(F)(F)F)F 1R-0209 COC(=O)/C=C/c1ccc2cc(ccc2c1)OCc3ccccc3 1R-0211 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NCc3ccc(cc3)Cl 1R-0214 c1cc(sc1)CNC(=O)/C=C/c2ccc(cc2)OCCCF 1R-0215 Cc1ccc(c(c1)C)N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCCCF 1R-0216 COc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)OCc3cccc(c3)Cl 1R-0218 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=C/C(=O)NC3CCCC3 1R-0220 c1cc(cc(c1)Cl)COc2ccc(cc2)/C=C/C(=O)N3CCOCC3 1R-0221 c1cc(ccc1/C=C/C(=O)NC2CCCCCC2)OCCCF 1R-0224 c1cc(ccc1/C=C/C(=O)NCc2ccc(c(c2)Cl)Cl)OCCCF 1R-0225 c1cc(ccc1/C=C/C(=O)N2CCOCC2)OCCCF 1R-0226 CN1C(=O)C(C(=O)N(C1=O)C)(Cc2ccc(cc2)C(F)(F)F)Cc3ccc(cc3)C(F)(F)F 1R-0228 Cc1ccc(n1c2ccsc2C(=O)CC#N)C 1R-0233 c1ccn(c1)c2ccsc2C(=O)O 1R-0234 c1cc(c2nnc(n2c1)C(F)(F)Cl)C(F)(F)F 1R-0600 Cc1cccc(c1)C(=O)Nc2ccc(cn2)C#N 1R-0601 c1ccc(cc1)CN2C/C(=C\c3ccccc3)/C(=O)/C(=C/c4ccccc4)/C2 1R-0602 CN1C(C2CN(C/C(=C\c3ccccc3)/C2=N1)Cc4ccccc4)c5ccccc5 1R-0604 c1c(cnc(c1Br)N)C#N 1R-0606 Cc1c(nc2cc(ccc2n1)[N+](=O)[O-])C 1R-0607 CC1CN(CC(O1)C)c2ccc(cc2[N+](=O)[O-])C(=O)OC 1R-0608 Cn1cc2cc(ccc2n1)N 1R-0610 COC(=O)c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)c2ccccc2 1R-0611 c1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccccc3)/CCC2 1R-0613 c1ccc(cc1)CN2C/C(=C\c3ccccc3)/C(/C(=C/c4ccccc4)/C2)O 1R-0614 Cn1cc2cc(ccc2n1)NC(=S)N 1R-0617 CCOC(=O)c1c(nn(c1C)c2ccnc3c2ccc(c3)Cl)C 1R-0618 c1ccc2c(c1)CN(C2=O)C(Cc3ccc(cc3)O)C(=O)NN 1R-0619 c1ccc(cc1)S(=O)(=O)c2c(cccn2)[N+](=O)[O-] 1R-0620 Cc1ccc(cc1)NC(=O)OC(C)c2cc3cccc(c3o2)OC 1R-0621 c1ccc(cc1)CN2CC3(CC3c4ccccc4)C(=O)C5(C2)CC5c6ccccc6 1R-0622 CC(=O)c1nc2ccccc2n1Cc3ccc(cc3)C(F)(F)F 1R-0623 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)N)C 1R-0624 CN1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(=O)OC 1R-0626 Cc1ccc(cc1)S(=O)(=O)c2c(cccn2)[N+](=O)[O-] 1R-0630 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(F)(F)F 1R-0631 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(=O)OC 1R-0633 CN(C)/C=C\C(=O)c1nc2ccccc2n1Cc3ccc(cc3)C(F)(F)F 1R-0635 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)c3cccs3)C 1R-0636 c1ccn(c1)CCNC(=O)C(F)(F)Cl 1R-0638 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)F)C 1R-0639 COc1ccc(cc1)c2cn3cc(ccc3n2)I 1R-0640 c1cc(c2nnc(n2c1)C(F)F)C(F)(F)F 1R-0641 Cc1ccc(n1c2ccc(c(c2)O)C(=O)OC)C 1R-0642 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)c3c(cccc3F)F)C 1R-0643 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)c3ccco3)C 1R-0644 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)c3cccc(c3)C(F)(F)F)C 1R-0645 c1ccc(cc1)C(=O)OC\2C3CCN(/C2=C\c4ccccc4F)CC3 1R-0646 c1cc(sc1)C(=O)Nc2ccc(cn2)C#N 1R-0647 c1ccc2c(c1)CN(C2=O)C(Cc3ccc(cc3)O)C(=O)N/N=C\c4ccc(cc4)Br 1R-0648 c1ccc(c(c1)/C=C\2/C(C3CCN2CC3)OC(=O)c4cccs4)F 1R-0649 c1ccc(c(c1)/C=C\2/C(C3CCN2CC3)OC(=O)c4c(cccc4F)F)F 1R-0650 CC(c1cc2cccc(c2o1)OC)OC(=O)NC3CCCCC3 1R-0651 COC(=O)c1ccc(cc1OC(=O)c2ccccc2Cl)n3cccc3 1R-0652 CC(=O)c1nc2ccccc2n1Cc3ccccc3 1R-0653 c1ccc2c(c1)nc(n2Cc3ccc(cc3)C(F)(F)F)c4cc[nH]n4 1R-0654 CC(c1cc2cccc(c2o1)OC)OC(=O)Nc3ccccc3 1R-0655 c1ccc(c(c1)/C=C\2/C(C3CCN2CC3)OC(=O)c4ccc(cc4)[N+](=O)[O-])F 1R-0656 COC(=O)c1ccc(cc1OC(=O)c2ccc(cc2)F)n3cccc3 1R-0658 CC(c1cc2cccc(c2o1)OC)OC(=O)Nc3cccc(c3)Cl 1R-0659 c1ccc2c(c1)CSCC3C2=NNC3c4cccs4 1R-0661 c1ccc(c(c1)CC2C(=O)C3CCN2CC3)F 1R-0662 COc1cc(c(cc1C(=O)OC)Br)NC(=O)c2cccs2 1R-0663 Cc1c(c(n(n1)c2ccc(cc2)F)C)C(=O)O 1R-0666 CCOC(=O)c1c(nn(c1C)c2ccc(c(c2)Cl)Cl)C 1R-0667 c1ccc(cc1)Cn2c3ccccc3nc2c4cc[nH]n4 1R-0670 c1cc(sc1)C2c3c([nH]cn3)CCN2 1R-0671 CC(=O)c1cc2cc(cc(c2o1)OC)Br 1R-0673 COc1ccccc1/N=C/c2cc(cc(c2O)Br)Br 1R-0674 CCOC(=O)c1c(nn(c1C)C)C 1R-0675 Cc1ccccc1C(=O)Nc2ccc(c(c2)OC)C(=O)OC 1R-0676 c1cc(ccc1C2c3c(nc[nH]3)CCN2)F 1R-0678 CC(=O)c1nc2ccccc2n1Cc3ccc(cc3)F 1R-0679 COc1ccc(cc1)C(=O)C2C(O2)c3ccc(cc3)Cl 1R-0680 c1ccc(cc1)C2c3c([nH]cn3)CCN2 1R-0681 c1ccc2c(c1)CSCC3(C2=O)C(O3)c4cccs4 1R-0683 CCOC(=O)c1c(nn(c1C)c2cccc(c2C)C)C 1R-0684 Cc1cc(cnc1N)I 1R-0685 CN1CCN(CC1)C(=O)/C(=C/N(C)C)/C#N 1R-0686 Cc1c(c(n(n1)c2ccc(c(c2)Cl)Cl)C)C(=O)O 1R-0688 c1ccc2c(c1)C(=O)C3C(C2=O)O3 1R-0689 c1cc(cc(c1)Cl)C2c3c(nc[nH]3)CCN2 1R-0690 c1ccc2c(c1)nc(s2)Sc3ccc4nnc(n4n3)C(F)(F)Cl 1R-0691 COc1cc(ccc1C(=O)OC)NC(=O)c2cccc(c2)C(F)(F)F 1R-0693 CN(C)/C=C\C(=O)c1nc2ccccc2n1Cc3ccc(cc3)F 1R-0695 COc1cc(ccc1C(=O)OC)NC(=O)c2ccc(c(c2)Cl)Cl 1R-0697 c1ccc(cc1)CC(COC(=O)c2ccccc2Cl)N3Cc4ccccc4C3=O 1R-0698 c1cc(ccc1C(F)(F)F)/N=C/c2cc(cc(c2O)Br)Br 1R-0699 c1cc(ncc1I)/N=C/c2cc(cc(c2O)Br)Br 1R-0700 c1ccc(cc1)N2CCN(CC2)C(=O)CC#N 1R-0701 c1ccc(c(c1)CC2C3(CO3)C4CCN2CC4)F 1R-0702 c1cc(ncc1C(F)(F)F)Sc2ccc3nnc(n3n2)C(F)(F)Cl 1R-0703 COc1ccccc1NCc2cc(cc(c2O)Br)Br 1R-0704 c1cc(ccc1/N=C/c2cc(cc(c2O)Br)Br)F 1R-0705 c1ccc(c(c1)/N=C/c2cc(cc(c2O)Br)Br)Cl 1R-0706 c1cc(cc(c1)C(F)(F)F)C2c3c(nc[nH]3)CCN2 1R-0707 c1ccnc(c1)Sc2ccc3nnc(n3n2)C(F)(F)Cl 1R-0708 c1ccc(cc1)CC(=O)c2ccc(s2)Br 1R-0709 c1ccc(c(c1)C2C3(O2)C(=O)C4CC[N+]3(CC4)[O-])F 1R-0711 c1ccc(c(c1)NCc2cc(cc(c2O)Br)Br)Cl 1R-0712 COC(=O)C(Cc1c[nH]c2c1cccc2)N3CCS(=O)(=O)CC3 1R-0714 c1cc(ccc1C(F)(F)F)NCc2cc(cc(c2O)Br)Br 1R-0715 c1ccc(c(c1)COc2ccc3nnc(n3n2)C(F)(F)Cl)Cl 1R-0717 c1cc(ccc1NCc2cc(cc(c2O)Br)Br)F 1R-0719 CCOC(=O)[CH-]C(=O)C(F)(F)F.c1ccc(cc1)N2CC[NH2+]CC2 1R-0720 Cc1c(sc(n1)c2ccccc2)c3ccnn3c4ccc(cc4)Cl 1R-0800 CC(C)NC(=O)C(C)Oc1ccc(cc1)O 1R-0802 Cc1cccc(n1)n2cc(nc2)C(=O)Nc3cccnc3 1R-0804 CCOC(=O)Cc1c(=O)[nH]c2ccccc2n1 1R-0805 COc1ccc(cc1OC)Cn2ccc(c(c2=O)CC(=O)OC)O 1R-0807 Cc1ccc(cc1)Cn2ccc(c(c2=O)CC(=O)OC)O 1R-0808 COC(=O)Cc1c(ccn(c1=O)Cc2ccc(cc2)OC(F)(F)F)O 1R-0809 CC1=C(CC(=O)N1CCc2c[nH]c3c2cccc3)C(=O)OC 1R-0810 COc1ccc(cc1)n2cc(nn2)C(=O)C(CC(=O)OC)C(=O)OC 1R-0811 Cc1c(sc(n1)c2ccccc2)c3cc(c4c(c(sc4n3)C(=O)OC)N)c5ccccc5 1R-0812 CC1=C(CC(=O)N1Cc2ccc3c(c2)OCO3)C(=O)OC 1R-0814 c1c(cnc(c1Cl)CC(=O)NN2CCOCC2)C(F)(F)F 1R-0815 CCC(C)NC(=O)c1cn(cn1)c2cccc(n2)C 1R-0817 Cc1cccc(n1)n2cc(nc2)C(=O)NCC3CCCO3 1R-0818 Cc1c(sc(n1)c2ccccn2)c3ccnc(n3)N 1R-0820 Cc1c(sc(n1)c2ccccn2)c3ccn[nH]3 1R-0821 CCCCN1C(C(CCC1=O)C(=O)O)c2ccccc2 1R-0823 COC(=O)Cc1c(ccn(c1=O)CCc2ccccc2)O 1R-0825 CC1=C(/C(=C/N(C)C)/C(=O)N1CCc2c[nH]c3c2cccc3)C(=O)OC 1R-0826 Cc1c(c(n(n1)c2ccc(cc2)F)O)CC(=O)OC 1R-0827 CCOC(=O)Cc1c(=O)n(c2ccccc2n1)C 1R-0828 Cc1c(c(n2c(n1)ncn2)O)CC(=O)OC 1R-0829 CC1=C(/C(=C/N(C)C)/C(=O)N1Cc2ccc3c(c2)OCO3)C(=O)OC 1R-0830 Cc1c(c(nc(n1)C)OCC(=O)c2ccc(cc2)Cl)I 1R-0834 Cc1c(sc(n1)c2cccnc2)C(=O)/C=C/c3ccc(cc3)Cl 1R-0836 COc1ccc(cc1)N(Cc2ccccc2)C(=O)CSc3ccc(cc3)Cl 1R-1000 COc1ccc(cc1)N(Cc2ccccc2)C(=O)CSc3ccc(cc3)Br 1R-1002 COc1ccc(cc1)N(Cc2ccccc2)C(=O)CSc3cccc(c3Cl)Cl 1R-1003 Cn1cccc1C(=O)C(=O)Nc2ccc(cc2)Cl 1R-1006 Cn1cccc1C(=O)C(=O)Nc2ccccc2 1R-1007 Cn1cccc1C(=O)C(=O)Nc2ccc(cc2Cl)Cl 1R-1008 Cn1cccc1C(=O)C(=O)Nc2cc(cc(c2)Cl)Cl 1R-1009 Cn1cccc1C(=O)C(=O)Nc2cccc(c2)C(F)(F)F 1R-1010 Cn1cccc1C(=O)C(=O)Nc2ccccc2C(F)(F)F 1R-1011 Cn1cccc1C(=O)C(=O)Nc2ccc(cc2)C(=O)OC 1R-1012 Cn1cccc1C(=O)C(=O)Nc2cccc(c2Cl)Cl 1R-1013 c1ccc(cc1)c2c(c3ccccc3[nH]2)C(=O)C(=O)N4CCOCC4 1R-1016 c1ccc(cc1)c2c(c3ccccc3[nH]2)C(=O)C(=O)N4CCCC4 1R-1017 Cn1cccc1C(=O)C(=O)Nc2ccc(cc2OC)[N+](=O)[O-] 1R-1018 Cn1cccc1C(=O)C(=O)Nc2ccc(cc2)Oc3ccccc3 1R-1019 Cn1cccc1C(=O)C(=O)Nc2ccc(c(c2)F)F 1R-1020 Cn1cccc1C(=O)C(=O)Nc2ccc(cc2F)F 1R-1021 CCNC(=O)C(=O)c1c2ccccc2[nH]c1c3ccccc3 1R-1023 c1ccc(cc1)c2c(c3ccccc3[nH]2)C(=O)C(=O)N4CCCCC4 1R-1024 c1cc(ccc1S(=O)(=O)NNC(=O)c2csnn2)Br 1R-1026 c1cc(ccc1/C=N\NC(=O)c2csnn2)F 1R-1028 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(nns2)C 1R-1030 Cc1c(snn1)C(=O)NNS(=O)(=O)c2ccc(cc2)Cl 1R-1031 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2csnn2 1R-1032 Cc1c(snn1)C(=O)NNS(=O)(=O)c2ccc(cc2)Br 1R-1033 Cc1ccc(cc1)/C=N\NC(=O)c2csnn2 1R-1034 CN(C)c1ccc(cc1)/C=N\NC(=O)c2csnn2 1R-1035 Cc1ccccc1/C=N\NC(=O)c2csnn2 1R-1036 Cc1cccc(c1)/C=N\NC(=O)c2csnn2 1R-1037 Cc1c(snn1)C(=O)NNS(=O)(=O)c2ccccc2 1R-1040 Cc1c(snn1)C(=O)NNS(=O)(=O)c2ccc(cc2)F 1R-1041 Cc1c(snn1)C(=O)NNC(=O)Nc2ccccc2 1R-1042 c1ccc(cc1)Oc2ccc(cc2)/C=N\NC(=O)c3csnn3 1R-1043 c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)S(=O)(=O)c4ccccc4 1R-1060 c1ccc(cc1)c2c(cc(=O)[nH]n2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Br 1R-1061 COc1ccc(cc1)NC(=O)c2cc3cccnc3n2S(=O)(=O)c4ccccc4 1R-1063 C1CC(=CC(=O)C1)N 1R-1064 c1ccc(cc1)C2C(=C(C(=O)O2)Cl)Cl 1R-1065 Cc1cc(ccc1NC(=O)c2cc3cccnc3n2S(=O)(=O)c4ccccc4)Cl 1R-1066 c1ccc(cc1)S(=O)(=O)n2c(cc3c2nccc3)C(=O)N4CCOCC4 1R-1067 c1ccc(cc1)c2c(cc(=O)[nH]n2)Cl 1R-1068 c1ccc(cc1)c2c(cc(nn2)Cl)Cl 1R-1069 c1ccc(cc1)S(=O)(=O)n2c(cc3c2nccc3)C(=O)Nc4ccc(cc4)Cl 1R-1070 c1ccc(cc1)c2c(cc(nn2)Sc3ccc(cc3)Cl)Cl 1R-1071 Cc1ccc(cc1)Sc2cc(c(nn2)c3ccccc3)Cl 1R-1073 Cc1ccc(cc1)Oc2cc(c(nn2)c3ccccc3)Cl 1R-1074 c1ccc(cc1)c2c(cc(nn2)Sc3ccc(cc3Cl)Cl)Cl 1R-1075 c1ccc(cc1)c2c(cc(nn2)Sc3ccc(cc3)Br)Cl 1R-1076 c1ccc(cc1)c2c(cc(nn2)Sc3ccc(cc3)F)Cl 1R-1077 c1ccc(cc1)c2c(cc(nn2)Sc3cccc(c3)C(F)(F)F)Cl 1R-1078 c1cc2ccn(c2nc1)S(=O)(=O)c3ccc(cc3Cl)Cl 1R-1080 c1ccc(cc1)c2c(cc(nn2)Oc3ccc(cc3Cl)Cl)Cl 1R-1081 c1ccc(cc1)c2c(cc(nn2)Oc3ccc(cc3)F)Cl 1R-1082 c1cc2ccn(c2nc1)S(=O)(=O)c3ccc(cc3)Br 1R-1086 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/O)/C 1R-1120 c1cc(c(cc1OCC(F)(F)F)C(=O)NNC(=O)C2CC2)OCC(F)(F)F 1R-1122 c1cc(ccc1C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 1R-1124 c1cc(c(cc1C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl)Cl 1R-1125 Cc1ccc(cc1)C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 1R-1126 c1cc(ccc1C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)F 1R-1127 Cc1c(sc(n1)C)/C(=N/OC(=O)c2ccc(c(c2)Cl)Cl)/C 1R-1128 c1ccc(cc1)CN2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 1R-1130 Cc1c(sc(n1)C)/C(=N/OC(=O)c2ccc(cc2)F)/C 1R-1131 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2c(nc(s2)C)C 1R-1133 Cc1c(sc(n1)C)/C(=N/OC(=O)c2cccs2)/C 1R-1134 Cc1c(sc(n1)C)/C(=N/OC(=O)c2cccc(c2)Cl)/C 1R-1135 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 1R-1136 CC(C)(C)OC(=O)N1CCC(CC1)Nc2ccc(cc2)Cl 1R-1139 CC(C)(C)OC(=O)N1CCC(CC1)Nc2ccc(cc2F)F 1R-1140 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)c3ccc(cc3)F)/C 1R-1141 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)c3ccc(cc3)Cl)/C 1R-1142 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2c(nc(s2)c3ccc(cc3)Cl)C 1R-1143 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)c3cccs3)/C 1R-1144 Cc1ccc(cc1)NC(=O)O/N=C(\C)/c2c(nc(s2)c3ccc(cc3)Cl)C 1R-1147 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)NC3CCCCC3)/C 1R-1148 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)Nc3ccccc3)/C 1R-1149 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/C 1R-1150 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)NC(C)C)/C 1R-1151 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)Nc3cccc(c3)Cl)/C 1R-1152 CCNC(=O)O/N=C(\C)/c1c(nc(s1)c2ccc(cc2)Cl)C 1R-1153 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N/OC(=O)C3CC3)/C 1R-1154 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)O 1R-1157 CCOC(=O)N1CCC(CC1)Nc2ccc(cc2)OC 1R-1159 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)c6ccc(cc6F)F 1R-1164 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)c6ccc(cc6)C(=O)O 1R-1165 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)CC(=O)O 1R-1166 COc1cnc(nc1Oc2ccc(cc2)F)c3ccccc3 1R-1180 COc1cnc(nc1Oc2cccc(c2)Cl)c3ccccc3 1R-1182 COc1cnc(nc1Sc2ccccc2)c3ccccc3 1R-1184 COc1cnc(nc1Sc2cccc(c2)Cl)c3ccccc3 1R-1185 COc1ccc(cc1)Sc2c(cnc(n2)c3ccccc3)OC 1R-1186 COc1ccccc1Sc2c(cnc(n2)c3ccccc3)OC 1R-1187 COc1cnc(nc1Sc2cccc(c2Cl)Cl)c3ccccc3 1R-1188 COc1cnc(nc1Sc2ccc(cc2Cl)Cl)c3ccccc3 1R-1189 Cc1c(n2ccccc2n1)C(=O)C 1R-1190 c1ccc(cc1)C(=O)Nn2c(nnc2S)c3cccs3 1R-1240 c1ccc(c(c1)CSc2nnc(n2N)c3cccs3)Cl 1R-1241 c1cc(cc(c1)Cl)CSc2nnc(n2N)c3cccs3 1R-1242 Cc1ccccc1CSc2nnc(n2N)c3cccs3 1R-1243 c1cc(sc1)c2nnc(n2N)SCc3ccc(cc3)Cl 1R-1244 COC(=O)c1ccc(cc1)CSc2nnc(n2N)c3cccs3 1R-1245 c1cc(cc(c1)F)CSc2nnc(n2N)c3cccs3 1R-1246 c1cc(sc1)c2nnc(n2NC(=O)c3ccc(cc3)F)S 1R-1249 c1cc(sc1)c2nnc(n2NC(=O)c3cccs3)S 1R-1250 c1cc(ccc1S(=O)(=O)N2CCC(CC2)C(=O)NN)Cl 1R-1300 CCN(CC)C(=O)C(=O)c1cccn1c2c3ccccc3sc2C(=O)OC 1R-1301 COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)NC4CCCCC4 1R-1302 COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)NC4CC4 1R-1303 CCCNC(=O)C(=O)c1cccn1c2c3ccccc3sc2C(=O)OC 1R-1304 CCCCCCNC(=O)C(=O)c1cccn1c2c3ccccc3sc2C(=O)OC 1R-1306 CC(C)NC(=O)C(=O)c1cccn1c2c3ccccc3sc2C(=O)OC 1R-1307 COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)Nc4ccc(cc4)Cl 1R-1308 Cc1ccc(cc1)NC(=O)C(=O)c2cccn2c3c4ccccc4sc3C(=O)OC 1R-1309 COc1ccc(cc1)NC(=O)C(=O)c2cccn2c3c4ccccc4sc3C(=O)OC 1R-1310 COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)Nc4ccc(cc4)Oc5ccccc5 1R-1311 COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)Nc4ccccc4 1R-1312 COC(=O)c1c(c2ccccc2s1)n3cccc3C(=O)C(=O)Nc4ccc(cc4)F 1R-1313 CSc1nc2c3ccccc3sc2c(n1)N4CCOCC4 1R-1314 CSc1nc2c3ccccc3sc2c(n1)NCC=C 1R-1315 CSc1nc2c3ccccc3sc2c(n1)Oc4ccccc4 1R-1316 CSc1nc2c3ccccc3sc2c(n1)Sc4cccc(c4)C(F)(F)F 1R-1317 Cc1ccc(cc1)C(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 1R-1318 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 1R-1319 c1cc(ccc1C(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)Cl 1R-1320 c1cc(ccc1F)S(=O)(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 1R-1321 c1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 1R-1322 Cc1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 1R-1323 Cc1ccc(cc1)C2N(C(CS2)C(=O)O)C(=O)OC(C)(C)C 1R-1324 CC(C)(C)OC(=O)N1C(CSC1c2ccc(cc2)Cl)C(=O)O 1R-1325 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(cc2)[N+](=O)[O-] 1R-1327 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccccc2 1R-1328 CCOC(=O)Oc1ccc(cc1F)F 1R-1501 CCOC(=O)Oc1cc(c(cc1F)F)[N+](=O)[O-] 1R-1502 c1c(c(cc(c1O)F)F)[N+](=O)[O-] 1R-1504 c1c(c(cc(c1O)F)F)N 1R-1506 CCOC(=O)C(=C1CCN(CC1)Cc2ccccc2)C#N 1R-1507 c1ccc(cc1)CN2CCC3(CC2)CC(=O)NC3=O 1R-1514 COc1cnc(nc1O)c2cccc(c2)C(F)(F)F 1R-1524 COc1ccc(cc1)NC(=O)c2csc(n2)Cc3ccccc3 1R-1525 CCOC(=O)c1csc(n1)Cc2ccccc2 1R-1528 CCOC(=O)c1csc(n1)Cc2ccc(cc2)Cl 1R-1529 c1ccc(cc1)Cc2nc(cs2)C(=O)O 1R-1531 c1cc(ccc1Cc2nc(cs2)C(=O)O)Cl 1R-1532 COc1ccc(cc1)Cc2nc(cs2)C(=O)O 1R-1536 c1ccc2c(c1)[nH]c(n2)C(F)(F)F 1R-1542 CCOC(=O)Cn1c2ccccc2nc1C(F)(F)F 1R-1543 c1ccc2c(c1)nc(n2CC(=O)O)C(F)(F)F 1R-1544 Cc1c(c2nccc(n2n1)C(C)Oc3ccc(cc3Cl)Cl)Cl 1T-0004 Cc1cc2ncc(c(n2n1)N)C(=O)O 1T-0007 c1ccc(cc1)C(=O)C(Sc2ccc(cc2)Cl)Br 1T-0009 Cc1cc(n(n1)c2nc(c(s2)Sc3ccc(cc3)Cl)c4ccccc4)C 1T-0010 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)c5cccc(c5)Cl)C 1T-0011 c1cc(ccc1c2cn[nH]c2N)F 1T-0013 Cc1cc2ncc(c(n2n1)N)c3cccc(c3)Cl 1T-0015 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)C(=O)OC)C 1T-0019 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)CS(=O)(=O)C)C 1T-0021 c1ccc(cc1)N2CCN(CC2)c3nc4nc(cc(n4n3)C(F)(F)F)c5cccs5 1T-0022 c1ccc(cc1)N2CCN(CC2)c3nc4nc(cc(n4n3)C(F)(F)F)c5ccco5 1T-0023 c1ccc(cc1)N2CCN(CC2)c3nc4nc(cc(n4n3)C(F)(F)F)c5cccc(c5)Cl 1T-0024 Cc1cc(n2c(n1)nc(n2)N3CCN(CC3)c4ccccc4)C(F)(F)Cl 1T-0025 Cc1cc2nc(cc(n2n1)O)CS(=O)(=O)C 1T-0027 COCc1cc(n2c(n1)nc(n2)N3CCN(CC3)c4ccccc4)O 1T-0028 c1cc(ccc1c2cnc3cc(nn3c2N)c4ccc(c(c4)Cl)Cl)Cl 1T-0030 CC(C)COCC(=O)O 1T-0032 CC(C)(C)OC(=O)NC(Cc1ccccc1)C=O 1T-0035 c1cc(sc1)c2cc(c(c(n2)O)C#N)C(F)(F)F 1T-0036 c1cc(oc1)c2cc(c(c(n2)O)C#N)C(F)(F)F 1T-0037 Cc1cc(c(c(n1)O)C#N)C(F)(F)Cl 1T-0038 c1ccc(cc1)S(=O)(=O)c2cn[nH]c2N 1T-0041 CCOC(Nc1cc(n[nH]1)c2c(ccs2)n3c(ccc3C)C)OCC 1T-0042 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)C(=O)O)C 1T-0045 Cc1cc(n(n1)c2nc(cs2)c3ccccc3)C 1T-0048 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(c(s2)Sc3ccc(cc3)Cl)c4ccccc4 1T-0051 c1ccc(cc1)c2csc(n2)N/N=C(\CC(=O)C(F)(F)F)/c3ccccc3 1T-0052 Cc1ccc2c(c1)cc(c(n2)Cl)C=O 1T-0053 c1ccc(cc1)c2csc(n2)CC#N 1T-0054 c1ccc(cc1)c2c(sc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F)Sc4ccc(cc4)Cl 1T-0055 Cc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=N2)SC 1T-0200 CCSC1=NC(C2=C(N1)c3ccccc3C2=O)c4ccc(cc4)C 1T-0202 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=C/C(=O)C 1T-0203 Cc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=N2)SCc5c(cccc5Cl)F 1T-0206 Cc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=N2)SCc5cccc(c5)Cl 1T-0207 Cc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=N2)SCc5cccc(c5)F 1T-0208 c1ccc(c(c1)c2c(n3ccsc3n2)C=O)F 1T-0212 CN(C)/C=C/C(=O)c1ccc2c(c1)c(on2)c3cccc(c3)F 1T-0213 c1cc(ccc1CSC2=C(N3C=CSC3N2)/C=C/c4ccn[nH]4)Cl 1T-0214 c1ccc(c(c1)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl 1T-0215 Cc1ccccc1C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 1T-0216 c1ccc(cc1)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 1T-0217 CC(=O)c1ccc2c(c1)c(on2)c3ccc4c(c3)OCO4 1T-0218 COc1ccc(cc1)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 1T-0219 Cc1ccc(cc1)N/C=C/C(=O)c2ccc3c(c2)c(on3)c4cccc(c4)F 1T-0223 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])C\2CCCC/C2=N\OC(=O)c3ccc(cc3Cl)Cl 1T-0225 c1cc(cc(c1)c2c(n3ccsc3n2)C=O)C#N 1T-0227 c1cc(c(cc1Cl)C2C=C(NC(=O)N2)C(=O)O)O 1T-0229 Cc1cc(ccc1N/C=C/C(=O)c2ccc3c(c2)c(on3)c4cccc(c4)F)Cl 1T-0238 c1ccc2c(c1)ccc3c2cc(o3)C(=O)O/N=C/4\CCCCC4c5ccc(cc5[N+](=O)[O-])[N+](=O)[O-] 1T-0239 CC(C)(C)c1ccc(cc1)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 1T-0240 c1cc(cc(c1)Cl)c2[nH]c(=O)c3cc(ccc3n2)N4CCCC4 1T-0242 c1ccc(c(c1)C2C3=C(c4ccccc4C3=O)NC(=S)N2)F 1T-0243 c1ccc(cc1)C(=O)COc2cccc3c2cccc3OCC(=O)c4ccccc4 1T-0244 CC1=C(C(C2=C(N1)c3ccccc3C2=O)c4ccccc4F)C#N 1T-0246 Cc1cc(cc(c1)NC(=O)Cc2ccc(cc2)O)C 1T-0247 c1ccc(cc1)C2=NC(C(=O)O2)c3ccc4ccccc4n3 1T-0248 c1cc(ccc1C2C=C(NC(=O)N2)C(=O)O)O 1T-0254 c1cc(ccc1C#N)O/C=C/C(=O)Oc2ccc(cc2)C#N 1T-0256 Cc1ccc(cc1)CSC2=NC(C3=C(N2)c4ccccc4C3=O)c5ccccc5F 1T-0257 CSC1=NC(C2=C(N1)c3ccccc3C2=O)c4ccccc4F 1T-0259 c1ccc(c(c1)C2C3=C(c4ccccc4C3=O)NC(=N2)SCc5cnc(s5)Cl)F 1T-0261 CCc1c(nc2cc(ccc2n1)N3CCN(CC3)C)CC 1T-0265 Cc1ccc(c(c1)CSC2=NC(C3=C(N2)c4ccccc4C3=O)c5ccccc5F)C 1T-0267 CC(=O)c1ccccc1C#N 1T-0269 c1ccc(cc1)n2c(c(cn2)C(=O)NN)N 1T-0271 CN1CCN(CC1)c2ccc3c(c2)nc(c(n3)c4ccccc4)c5ccccc5 1T-0272 CN1CCN(CC1)c2ccc3c(c2)nccn3 1T-0273 CC(=O)c1ccc2c(c1)c(c3ccccc3n2=O)C#N 1T-0274 c1cc(cc(c1)F)c2c(n3ccsc3n2)C=O 1T-0275 CC1C(NC(=O)N1C)c2ccccc2 1T-0277 CN1CCN(CC1)c2ccc(c(c2)C(=O)N)[N+](=O)[O-] 1T-0278 Cc1c(nc2cc(ccc2n1)N3CCN(CC3)C)C 1T-0280 c1ccc2c(c1)C(=O)C(=Cc3ccco3)C2=O 1T-0281 c1cc(ccc1c2c3cc(ccc3no2)C4OCCO4)F 1T-0284 c1ccc(c(c1)C2C3=C(c4ccccc4C3=O)N=C5N2C(=O)CS5)F 1T-0286 COc1ccc(cc1)O/C=C/C(=O)Oc2ccc(cc2)OC 1T-0287 c1cc(sc1C=O)N2CCC(CC2)O 1T-0289 Cc1ccc(cc1)S(=O)(=O)C(C)N2C(C(N(C2=O)C)C)c3ccccc3 1T-0292 c1cc(ccc1c2c3cc(ccc3no2)C=O)F 1T-0293 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCCC3 1T-0295 c1cc(ccc1CC(=O)Nc2ccc3c(c2)CCC3)O 1T-0297 CC1C(=O)N2C(C3=C(c4ccccc4C3=O)N=C2S1)c5ccccc5F 1T-0301 c1cc2c(cccc2OCC(=O)c3ccc(cc3)Cl)c(c1)OCC(=O)c4ccc(cc4)Cl 1T-0302 CCO/C(=N/NC(=O)c1cnn(c1N)c2ccccc2)/C 1T-0304 c1cc(c(cc1Cl)Cl)C2C=C(NC(=O)N2)C(=O)O 1T-0305 Cc1ccc(cc1)S(=O)(=O)CN2C(C(N(C2=O)C)C)c3ccccc3 1T-0308 c1cc2c(cccc2OCC(=O)c3ccc(c(c3)Cl)Cl)c(c1)OCC(=O)c4ccc(c(c4)Cl)Cl 1T-0309 c1ccc(cc1)c2ccc(cc2)C(=O)COc3cccc4c3cccc4OCC(=O)c5ccc(cc5)c6ccccc6 1T-0314 CCC(N1CCOC1=O)S(=O)(=O)c2ccc(cc2)C 1T-0318 CC(N1CCOC1=O)S(=O)(=O)c2ccccc2 1T-0319 c1ccc(c(c1)C2C3=C(c4ccccc4C3=O)N=C5N2C(=O)CCS5)F 1T-0320 CC1=C(C(C2=C(N1)c3ccccc3C2=O)c4ccco4)C#N 1T-0327 Cc1ccc(cc1)Oc2c(c(nn2C)C(F)(F)F)C=O 1T-0329 CN1CCN(CC1)c2ccc3c(c2)c(=O)[nH]c(n3)c4ccc(cc4)OC 1T-0330 c1ccc2c(c1)NC(=O)CO2 1T-0333 Cc1ccc(cc1)Oc2c(c(nn2C)C(F)(F)F)CO 1T-0334 CCCC(NC(=O)OCc1ccccc1)S(=O)(=O)c2ccccc2 1T-0336 CC(C)C(N1CCOC1=O)S(=O)(=O)c2ccccc2 1T-0337 Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)C=O 1T-0339 c1ccc(c(c1)c2cn3c(n2)ccc4c3nc(cc4C(F)(F)F)C(F)(F)F)F 1T-0341 Cc1nnc(n1c2ccc(cc2)OC)c3cnn(c3N)c4ccccc4 1T-0342 CN1CCN(CC1)c2ccc3c(c2)c(=O)[nH]c(n3)c4ccc(cc4)F 1T-0343 c1ccc2c(c1)C(=O)C=C(C2=O)N3CCC(CC3)C(=O)O 1T-0344 c1cc(n(c1)c2nccs2)/C=N/c3ccc(c(c3)Cl)Cl 1T-0600 c1cc(n(c1)c2ccc(cc2)Br)C(=O)O 1T-0601 c1csc2c1C(CC2=O)NC(=O)C(F)(F)F 1T-0602 c1c2c(cc3c1OCO3)C(=O)CC2N.Cl 1T-0603 COC(=O)CC(c1ccc(cc1)Br)NC(=O)c2ccccc2F 1T-0604 COc1ccc(cc1)S(=O)(=O)NC(CC(=O)OC)c2ccc(cc2)Br 1T-0605 COC(=O)CC(c1ccc(cc1)Br)NS(=O)(=O)c2cccs2 1T-0606 COc1ccc(cc1)C(=O)/C=C/c2ccn(c2)c3ccc(cc3)Br 1T-0607 CCc1ccc(cc1)C(CC(=O)O)NC(=O)C(F)(F)F 1T-0608 COC(=O)CC(c1ccc(cc1)Br)NC(=O)c2ccco2 1T-0609 c1cc(cc(c1)F)C(CC(=O)O)NC(=O)C(F)(F)F 1T-0610 Cc1ccccc1C(CC(=O)O)NC(=O)C(F)(F)F 1T-0611 COC(=O)C1C(=O)CC(NC1=O)c2ccc(cc2)Br 1T-0613 CN1CCN(CC1)c2ccc(c(c2)N)N 1T-0614 CN1C(=O)C(=Cc2cccn2c3ccc(cc3)Br)C(=O)N(C1=O)C 1T-0616 c1cc(n(c1)c2ccc(cc2)Br)C=C(C#N)C#N 1T-0618 CC(C)c1ccc(cc1)C(CC(=O)O)NC(=O)C(F)(F)F 1T-0619 c1cc(n(c1)c2ccc(cc2)Br)/C=N/O 1T-0620 c1ccc2c(c1)/C(=C\c3cccn3c4ccc(cc4)Br)/C(=O)N2 1T-0621 C/C(=C\C(=O)c1cccs1)/N(C)C 1T-0622 COc1ccc(cc1)C/N=C/c2cccn2c3nccs3 1T-0623 c1cc(ccc1C#N)C(CC(=O)O)N 1T-0626 c1ccc2c(c1)/C(=C\c3cccn3c4ccc(cc4)OC(F)(F)F)/C(=O)N2 1T-0627 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccccc3F 1T-0629 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(cc3)C#N 1T-0630 Cc1cc(nc(n1)N)c2cccs2 1T-0631 CN(C)/C=C/C(=O)c1cc2ccccc2s1 1T-0632 CN(C)/C=C/C(=O)c1ccc(s1)Br 1T-0633 CN(C)/C=C/C(=O)c1ccc(s1)Cl 1T-0634 c1ccc2c(c1)C(C(=O)N2)Cc3cccn3c4ccc(cc4)OC(F)(F)F 1T-0636 c1cc(cc(c1)C(F)(F)F)C(CC(=O)O)N2CCS(=O)(=O)CC2 1T-0637 c1ccc(c(c1)C(CC(=O)O)NC(=O)C(F)(F)F)F 1T-0638 COC(=O)CC(c1ccccc1F)N2Cc3ccccc3C2=O 1T-0639 COC(=O)CC(c1ccc(cc1)Br)NC(=S)NC(=O)c2ccccc2 1T-0640 COc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)OC)C(=O)OC 1T-0641 CC1(OC(=O)C2(CCS(=O)(=O)CC2)C(=O)O1)C 1T-0642 CN(C)/C=C\1/C(c2cc(c(cc2C1=O)OC)OC)NC(=O)C(F)(F)F 1T-0645 c1cc(sc1c2ccnc(n2)N)Cl 1T-0646 c1cc(sc1c2ccnc(n2)N)Br 1T-0647 c1ccc2c(c1)cc(s2)c3ccnc(n3)N 1T-0648 C/C(=C\C(=O)c1ccc(s1)Cl)/N(C)C 1T-0650 C/C(=C\C(=O)c1ccc(s1)Br)/N(C)C 1T-0651 C/C(=C\C(=O)c1c(ccs1)Cl)/N(C)C 1T-0652 c1cc(cc(c1)Br)C(CC(=O)O)N2CCS(=O)(=O)CC2 1T-0653 c1cc(cc(c1)[N+](=O)[O-])C(CC(=O)O)NC(=O)C(F)(F)F 1T-0655 COC(=O)c1ccc(cc1)C(CC(=O)O)N 1T-0657 c1cnc(nc1c2c(ccs2)Cl)N 1T-0659 c1cc(sc1C(=O)N)Cl 1T-0800 CN(C)c1ccc(cc1)/C=C/C=N/c2c(c(c(o2)c3ccccc3)c4ccccc4)C#N 1T-0802 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3cccc(c3)N 1T-0803 c1c(cnc(c1Cl)CC(=O)NC2CC2)C(F)(F)F 1T-0804 c1cc(ccc1c2ncc(s2)C(=O)/C=C/Nc3ccc(cc3)S(=O)(=O)NC(=N)N)Cl 1T-0805 c1cc(ccc1c2ncc(s2)c3ccnc(n3)NS(=O)(=O)c4ccc(cc4)N)Cl 1T-0806 c1cc(sc1C(=S)N)Cl 1T-0807 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Cn4cncn4 1T-0808 c1cc(nc(c1)F)NNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 1T-0809 c1c(cnc(c1Cl)CC(=O)NCC2CCCO2)C(F)(F)F 1T-0810 COC(=O)/C(=C\Nc1cc(cc(c1)Cl)Cl)/n2cncn2 1T-0811 COC(=O)/C(=C\Nc1ccc(c(c1)Cl)F)/n2cncn2 1T-0812 COC(=O)/C(=C\Nc1cc(ccc1Cl)C(F)(F)F)/n2cncn2 1T-0821 c1ccnc(c1)CNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 1T-0822 c1c(cnc(c1Cl)Cc2nnc3n2cc(cc3Cl)C(F)(F)F)C(F)(F)F 1T-0823 Cc1ccc(cc1N/C=C(\C(=O)OC)/n2cncn2)F 1T-0824 COC(=O)/C(=C/Nc1ccccc1SC)/n2cncn2 1T-0825 COC(=O)/C(=C\Nc1ccc2c(c1)OCCO2)/n3cncn3 1T-0826 c1cc(cnc1)c2ncc(s2)c3ccnc(n3)NS(=O)(=O)c4ccc(cc4)N 1T-0827 c1ccc(cc1)c2c3c(=N)n(c(=S)[nH]c3oc2c4ccccc4)c5ccccc5 1T-0828 c1ccc(cc1)n2c(=N)c3c(c(oc3[nH]c2=S)c4ccco4)c5ccco5 1T-0829 c1ccc(cc1)c2c(c(oc2c3ccccc3)/N=C/c4ccccc4[N+](=O)[O-])C#N 1T-0830 CN(C)c1ccc(cc1)/C=C/C=N/c2c(c(c(o2)c3ccco3)c4ccco4)C#N 1T-0831 Cc1c(sc(n1)Nc2cccc(c2)C(F)(F)F)c3ccnc(n3)N 1T-0832 CC(=O)/C=C/c1cc(c(c(c1)OC)OC)OC 1T-0833 COc1c(c(cc(c1)/C=C/C(=O)/C=C/c2cc(c(c(c2)OC)OC)OC)OC)OC 1T-0834 c1c(cnc(c1Cl)CC(=O)NC2CCCC2)C(F)(F)F 1T-0835 COC(=O)/C(=C\Nc1nncs1)/n2cncn2 1T-0836 C/C(=N\NC(=S)N)/CC(=O)C(F)(F)F 1T-0837 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)Cl)C(F)(F)F 1T-0838 COc1ccc(cc1OC)CCNC=O 1T-0840 c1cc(cc(c1)N)c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F 1T-0841 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F 1T-0842 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)Br)C(F)(F)F 1T-0843 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)OC)C(F)(F)F 1T-0844 COc1cc2c(cc1OC)N=CCC2 1T-0845 COc1ccc(cc1)C(=O)CSc2ccc(cc2)Cl 1T-0846 COc1cc2c(cc1OC)C3CC(=O)CC(=O)N3CC2 1T-0849 COc1ccc(cc1)C(=O)CS(=O)(=O)c2ccc(cc2)Cl 1T-0850 Cc1cc(n(n1)c2nc(cs2)c3ccccc3)C(F)(F)F 1T-0851 CCOC(=O)c1c(nc(s1)n2c(cc(n2)C)C(F)(F)F)C 1T-0852 Cc1cc(n(n1)c2nc(cs2)C(=O)O)C(F)(F)F 1T-0896 c1cc(sc1)c2ccnc3n2ncc3c4ccc(cc4)Cl 1T-0897 Cc1c(c2nccc(n2n1)c3ccncc3)Br 1T-0898 Cc1cc(n(n1)c2nc(cs2)C(=O)NN)C(F)(F)F 1T-0899 CN(C)c1nc(cc(n1)Cl)Sc2ccccc2C(=O)OC 1T-1003 Cc1cc(nc(n1)C(C)C)N2CC(OC(C2)C)C 1T-1006 CCCCCCNc1cc(nc(n1)C(C)C)C 1T-1007 Cc1cc(n2c(n1)cc(n2)c3ccccc3)O 1T-1010 Cc1cc(nc(n1)C(C)C)NCCCN(C)C 1T-1011 CCN(CC)CCNc1cc(nc(n1)C(C)C)C 1T-1012 Cc1ccc(n1c2ccccc2CNS(=O)(=O)c3ccc(cc3)Cl)C 1T-1014 Cc1ccc(n1c2ccccc2CNS(=O)(=O)c3ccc(cc3)Br)C 1T-1015 Cc1ccc(n1c2ccccc2CNS(=O)(=O)Cc3ccccc3)C 1T-1016 Cc1ccc(n1c2ccccc2CNS(=O)(=O)c3ccc(cc3)NC(=O)C)C 1T-1018 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)C(F)(F)F 1T-1019 Cc1cccc(c1C)Oc2ccc(cc2[N+](=O)[O-])/C=N\OC 1T-1122 C#Cc1ccc(cc1)N 1T-1123 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)C#C 1T-1124 CC(=O)Nc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])/C=N/OC 1T-1130 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Oc2cc(c(cc2Cl)Cl)Cl 1T-1131 C#Cc1ccc(cc1)NC(=O)c2ccc(cc2)F 1T-1136 C#Cc1ccc(cc1)NC(=O)c2cccc(c2)C(F)(F)F 1T-1137 C#Cc1ccc(cc1)NC(=O)c2cccc(c2)Cl 1T-1138 C#Cc1ccc(cc1)NC(=O)c2c(cccc2F)F 1T-1139 C#Cc1ccc(cc1)NC(=O)c2cccs2 1T-1140 Cc1ccccc1C(=O)Nc2ccc(cc2)C#C 1T-1141 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)C#C 1T-1143 C#Cc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)F 1T-1144 C#Cc1ccc(cc1)NS(=O)(=O)c2ccccc2 1T-1145 C#Cc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Cl 1T-1147 C#Cc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Br 1T-1148 C#Cc1ccc(cc1)NS(=O)(=O)c2ccccc2F 1T-1149 CS(=O)(=O)Nc1ccc(cc1)C#C 1T-1150 CCOC(=O)c1cnn(c1n2c(ccc2C)C)c3ccccc3 1T-1151 c1ccc(cc1)c2cc(n(n2)c3ccccc3)O 1T-1152 c1ccc(cc1)C#Cc2ccc(cc2)NC(=O)C(F)(F)F 1T-1153 c1ccc(cc1)C#Cc2ccc(cc2)N 1T-1154 c1ccn(c1)c2ccc(cc2)C(=O)OCC#N 1T-1155 c1ccn(c1)c2ccc(cc2)C(=O)N3CCCC3 1T-1156 c1ccc(cc1)n2c(c(cn2)C(=O)Nc3ccc(cc3)F)C(F)(F)F 1T-1157 Cc1ccc(cc1C)NC(=O)c2cnn(c2C(F)(F)F)c3ccccc3 1T-1159 c1ccc(cc1)n2c(c(cn2)C(=O)Nc3ccc(cc3F)F)C(F)(F)F 1T-1160 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)C#Cc3ccccc3 1T-1161 c1ccc(cc1)C#Cc2ccc(cc2)NC(=O)C3CC3 1T-1162 c1ccc(cc1)C#Cc2ccc(cc2)NC(=O)c3cccs3 1T-1164 c1ccc(cc1)C#Cc2ccc(cc2)NC(=O)c3cccc(c3)C(F)(F)F 1T-1165 CS(=O)(=O)Nc1ccc(cc1)C#Cc2ccccc2 1T-1166 c1ccc(cc1)C#Cc2ccc(cc2)NC(=O)c3ccc(c(c3)Cl)Cl 1T-1167 COc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)N3CCOCC3 1T-1188 c1ccc(cc1)CS(=O)(=O)Nc2ccc(nc2)N3CCOCC3 1T-1189 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCc4ccc(cc4)Cl 1T-1240 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCc4ccc(c(c4)Cl)Cl 1T-1241 Cc1ccc(cc1)CSc2nc3c(c4ccccc4[nH]3)nn2 1T-1242 CCOC(=O)CSc1nc2c(c3ccccc3[nH]2)nn1 1T-1244 C=CCSc1nc2c(c3ccccc3[nH]2)nn1 1T-1245 C#CCSc1nc2c(c3ccccc3[nH]2)nn1 1T-1246 CC(C)Sc1nc2c(c3ccccc3[nH]2)nn1 1T-1247 c1ccc(cc1)C(=O)CSc2nc3c(c4ccccc4[nH]3)nn2 1T-1248 CSc1nc2c(c3ccccc3[nH]2)nn1 1T-1249 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCc4ccc(cc4)F 1T-1252 c1ccc(cc1)CSc2nc3c(c4ccccc4[nH]3)nn2 1T-1253 c1cc(ccc1Sc2c(cc3c(n2)CCCC3)C#N)Cl 1T-1254 COC(=O)c1ccccc1Sc2c(cc3c(n2)CCCC3)C#N 1T-1255 COC(=O)c1ccc(cc1Cl)F 1T-1481 COC(=O)c1ccc(cc1Cl)N2CCCC2 1T-1482 c1cc(c(cc1N2CCCC2)Cl)C(=O)O 1T-1483 COC(=O)c1ccc(cc1Cl)N2CCOCC2 1T-1484 COC(=O)c1ccc(cc1Cl)n2cccn2 1T-1485 c1cc(c(cc1N2CCOCC2)Cl)C(=O)O 1T-1486 c1cnn(c1)c2ccc(c(c2)Cl)C(=O)O 1T-1487 CN(C)c1nc(cc(n1)Cl)N2CCOCC2 1T-1512 c1ccn(c1)c2nccc(n2)c3c(ccs3)Cl 1T-9000 c1ccn(c1)c2nccc(n2)c3ccc(s3)Cl 1T-9002 c1ccn(c1)c2nccc(n2)c3c(ccs3)Br 1T-9003 c1ccn(c1)c2nccc(n2)c3ccc(s3)Br 1T-9004 Cc1ccsc1c2ccnc(n2)n3cccc3 1T-9005 Cc1cc(nc(n1)n2cccc2)c3cccs3 1T-9006 c1ccc2c(c1)cc(s2)c3ccnc(n3)n4cccc4 1T-9007 Cc1cc(nc(n1)n2cccc2)c3c(ccs3)Cl 1T-9008 Cc1cc(nc(n1)n2cccc2)c3ccc(s3)Cl 1T-9009 Cc1ccsc1c2cc(nc(n2)n3cccc3)C 1T-9010 Cc1cc(nc(n1)n2cccc2)c3c(ccs3)Br 1T-9011 Cc1cc(nc(n1)n2cccc2)c3ccc(s3)Br 1T-9012 c1cc(n(c1)c2nccc(n2)c3cccs3)C=O 1T-9014 Cc1ccc(n1c2nc(cc(n2)c3c(ccs3)Cl)C)C 1T-9016 c1cc(n(c1)c2nc(cc(n2)C(F)(F)F)c3cccs3)C=O 1T-9018 Cc1cc(nc(n1)n2cccc2C=O)c3c(ccs3)Cl 1T-9019 c1cc(n(c1)c2nccc(n2)c3cccs3)/C=N/O 1T-9020 c1cc(n(c1)c2nccc(n2)c3cccs3)C#N 1T-9021 c1ccn(c1)c2nc(cc(n2)C(F)(F)F)c3cccs3 1T-9023 CC(=O)O/N=C\c1cccn1c2nccc(n2)c3cccs3 1T-9024 COc1cc2c(cc1OC)C3Cc4c(cnn4c5cccc(c5)Cl)C(=O)N3CC2 1W-0003 Cc1cccc(c1C)n2c3c(cn2)C(=O)N4CCc5cc(c(cc5C4C3)OC)OC 1W-0004 COC(=O)C(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)C(=O)OC 1W-0027 COC(=O)C(c1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])C(=O)OC 1W-0033 COC(=O)C(c1ccc(cn1)n2cccc2)C(=O)OC 1W-0036 Cc1ccc(cc1)C(CCc2cc(c(c(c2)OC)OC)OC)O 1W-0041 Cc1ccc(cc1)n2c(cc(n2)c3cccn3C)C(=O)O 1W-0042 COC(=O)C(CC=C)(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)C(=O)OC 1W-0047 CC(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)(C(=O)OC)C(=O)OC 1W-0048 c1cc(cc(c1)[N+](=O)[O-])/N=C/c2cnc(s2)N3CCCC3 1W-0049 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)Cc4ccccc4 1W-0200 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)Cc4ccccc4 1W-0202 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)CC#N 1W-0203 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)Cc4cccc(c4)C(F)(F)F 1W-0204 c1ccc2c(c1)C(=O)N(C2=O)Cc3ccc(nc3)Cl 1W-0205 Cc1nn(c(=O)n1c2ccccc2F)Cc3ccc(cc3)[N+](=O)[O-] 1W-0206 Cc1nn(c(=O)n1c2ccccc2F)CC3CC3 1W-0208 CCOC(=O)c1c(nc(s1)c2ccc(cc2)C(F)(F)F)C 1W-0211 CCOC(=O)c1cn(c(c1C)c2ccccc2)C(=O)C 1W-0212 CCOC(=O)c1c(c2ccccc2n(c1=O)C)O 1W-0214 c1ccc(cc1)C(C(=O)O)NC=C2C(=O)CCCC2=O 1W-0216 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)c3c(cc(cn3)C(F)(F)F)Cl 1W-0217 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)Cc3ccccc3 1W-0218 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CO 1W-0220 Cc1cccc(c1n2c(nn(c2=O)Cc3ccc(cc3)[N+](=O)[O-])C)C 1W-0221 Cc1cccc(c1n2c(nn(c2=O)Cc3ccc(cc3)OC)C)C 1W-0222 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)Cc3cccc(c3)C(F)(F)F 1W-0224 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)CCOc3ccccc3 1W-0225 CCOC(=O)Cn1c(=O)n(c(n1)C)N(C)c2c(cc(cn2)C(F)(F)F)Cl 1W-0226 Cc1nn(c(=O)n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)CC3CC3 1W-0227 Cc1nnc(n1CCC2=CCCCC2)c3cnn(c3N)C 1W-0228 Cc1cccc(c1n2c(nn(c2=O)c3c(cc(cn3)C(F)(F)F)Cl)C)C 1W-0230 Cc1nn(c(=O)n1c2ccccc2F)C 1W-0231 Cc1cccc(c1n2c(nn(c2=O)CC#N)C)C 1W-0232 CC(=O)c1nc2ccccc2s1 1W-0233 CCOC(=O)c1c(c2ccccc2n(c1=O)C)Cl 1W-0234 C/C(=C(\C=C\C(=O)OC)/C(=O)C)/NCc1ccc(cc1)OC 1W-0235 COC(=O)/C=C/C(=C/NCc1ccccc1)/C(=O)OC 1W-0236 CCOC(=O)c1c(c(c(s1)Nc2ccccc2)C(=O)C)C 1W-0238 c1cc(cc(c1)Oc2ncccn2)C(=O)O 1W-0239 c1cc(cc(c1)OCc2ccc(cc2)F)C(=O)/C=C(/C3CC3)\O 1W-0240 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3ccc(cc3)C(C)(C)C)OC)OC 1W-0242 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)CC4CC4 1W-0244 Cc1cccc(c1n2c(nn(c2=O)CC3CC3)C)C 1W-0245 CCOC(=O)Cn1c(=O)n(c(n1)C)c2c(cccc2C)C 1W-0246 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)Cc4ccc(cc4)OC 1W-0247 c1ccc(cc1)c2ccc(cc2)c3ccn(n3)CCO 1W-0248 C/C(=C\c1cccc(c1)Oc2ncccn2)/[N+](=O)[O-] 1W-0251 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)Oc3ccccc3 1W-0252 Cc1nn(c(=O)n1c2ccc(cc2)Oc3ccccc3)C 1W-0253 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CCl 1W-0254 c1cc2c(cc1[N+](=O)[O-])cc(s2)C(=O)O 1W-0255 CC(C)c1ccc(cc1)NC(=O)CNC(=O)c2c(nn(c2Cl)C)c3ccccc3 1W-0257 c1ccc2c(c1)c(c(c(=O)o2)C=O)Cl 1W-0258 c1ccc(cc1)C(=O)c2coc3c2cc(cc3)O 1W-0264 c1cnc(nc1)Oc2ccc(cc2)C=O 1W-0265 Cc1ccc(cc1)CNC(=O)CNC(=O)c2c(nn(c2Cl)C)c3ccccc3 1W-0267 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3ccc(cc3)C)OC)OC 1W-0269 Cc1c2c(c3cc(cc(c3n1)OC)OC)N(CC2)c4ccccc4OC 1W-0270 CCCCCC1CCC(CC1)C(=O)N/N=C/c2ccc(cc2)Oc3ncccn3 1W-0274 Cc1c2c(c3cc(cc(c3n1)OC)OC)N(CC2)c4ccc(cc4)OC 1W-0275 Cc1c(c(n(n1)C)Cl)NC(=O)OCc2ccc(cc2Cl)Cl 1W-0276 CC(=O)c1c2c(cc(c1Cl)Cl)OCCO2 1W-0279 c1cc(c(cc1N2CCCCC2)C(=O)N)[N+](=O)[O-] 1W-0280 Cc1cccc(c1n2c(nn(c2=O)Cc3ccccc3)C)C 1W-0283 c1cnc(nc1)Oc2ccc(cc2)/C=C/C(=O)c3ccc4c(c3)OCO4 1W-0284 c1cc(ccc1CO/N=C/c2ccc(cc2)O)C(F)(F)F 1W-0285 COc1ccc(cc1)c2nc(cs2)C(=O)O 1W-0286 Cc1c2c(c3cccc(c3n1)C(F)(F)F)N(CC2)c4ccc(cc4OC)OC 1W-0288 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3ccc(cc3)Cl)OC)OC 1W-0289 c1cnc(nc1)Oc2ccc(cc2)/C=C/C(=O)O 1W-0290 Cc1c2c(c3cc(cc(c3n1)OC)OC)N(CC2)c4ccc(cc4)O 1W-0291 c1ccc2c(c1)c(cc(=O)o2)Nc3ccc(cc3)Cl 1W-0293 c1cc(cc(c1)Oc2ncccn2)/C=C\3/C(=O)NC(=S)S3 1W-0295 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)/C=C\4/C(=O)NC(=S)S4 1W-0296 Cc1c2c(c3cc(cc(c3n1)OC)OC)N(CC2)c4ccc(cc4OC)OC 1W-0298 Cc1c2c(c3cc(cc(c3n1)OC)OC)N(CC2)c4ccc(cc4)C(C)C 1W-0299 Cc1c2c(c3cccc(c3n1)OC)N(CC2)c4ccc(cc4)Oc5ccccc5 1W-0300 Cc1c2c(c3cccc(c3n1)OC)N(CC2)c4ccccc4OC 1W-0301 Cc1c2c(c3cccc(c3n1)OC)N(CC2)c4ccc(cc4)OC 1W-0302 CCOC(=O)c1c(c2ccccc2n(c1=O)C)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 1W-0305 CSC1=NC(=O)/C(=C/c2cccc(c2)Oc3ncccn3)/S1 1W-0306 Cc1cccc(c1n2c(nn(c2=O)C)C)C 1W-0307 CCc1ccc(cc1)N2CCc3c2c4cccc(c4nc3C)C(F)(F)F 1W-0309 c1cc(cc(c1)Cl)CNC2=NC(=O)/C(=C\c3cccc(c3)Oc4ncccn4)/S2 1W-0312 c1cnc(nc1)Oc2ccc(cc2)C(=O)O 1W-0313 Cc1c(c(c2cccc(c2n1)OC)Nc3ccc(cc3)O)CCCl 1W-0314 CN(C)/C=C/C(=O)c1c2c(cc(c1Cl)Cl)OCCO2 1W-0315 Cc1cccc(c1n2c(nn(c2=O)Cc3cccc(c3)C(F)(F)F)C)C 1W-0316 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3c(cc(cc3C)C)C)OC)OC 1W-0321 Cc1ccc(n1/C(=C(\C#N)/N)/C#N)C 1W-0324 COc1ccc(cc1)NC(=O)c2ccc(cc2)Oc3ncccn3 1W-0325 Cc1c2c(c3cccc(c3n1)OC)N(CC2)c4ccc(cc4)C(C)C 1W-0326 c1ccc(c(c1)C=O)n2cncn2 1W-0327 COc1ccc(cc1)c2cc(cc(c2)O)c3ccc(cc3)Cl 1W-0328 c1ccc(c(c1)/C=C\2/C(=O)NC(=S)S2)n3cncn3 1W-0329 c1ccc2c(c1)cc([nH]2)c3cccs3 1W-0332 COc1ccc(cc1)N/C=C/C(=O)c2c3c(cc(c2Cl)Cl)OCCO3 1W-0337 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3c(cccc3Cl)F)OC)OC 1W-0341 Cc1c2c(c3cccc(c3n1)OC)N(CC2)c4ccccc4 1W-0343 CCc1ccc(cc1)N2CCc3c2c4cccc(c4nc3C)OC 1W-0344 Cc1c2c(c3cccc(c3n1)OC)N(CC2)c4ccc(cc4OC)OC 1W-0345 Cc1ccc(c(c1)C)N2CCc3c2c4cccc(c4nc3C)OC 1W-0346 c1ccc(cc1)S(=O)(=O)c2cscc2n3cccc3 1W-0347 CC(=O)Nc1cc2c(cc1Cl)OCCO2 1W-0351 CSC1=NC(=O)/C(=C/c2ccccc2n3cncn3)/S1 1W-0352 CC1=NC(=C(NC(C1)c2ccccc2)C#N)C#N 1W-0353 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3ccc(cc3)[N+](=O)[O-])OC)OC 1W-0357 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3cccc(c3)OC)OC)OC 1W-0360 Cc1ccc(n1/C(=C(\C#N)/NC(=O)c2ccc(cc2)F)/C#N)C 1W-0363 Cc1ccc(n1/C(=C(/C#N)\NC(=O)C2CCCCC2)/C#N)C 1W-0365 COc1cccc(c1)/C=C/C(=O)c2ccccc2[N+](=O)[O-] 1W-0366 CCCCCCCCn1c(=N)c2cc(c(cc2nc1SCc3cc(ccc3C)C)OC)OC 1W-0369 CC(C)c1c(nc(s1)N)C(=O)OC 1W-0612 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6cccs6 1W-0615 COc1ccc(cc1)/C=N/NS(=O)(=O)c2ccccc2 1W-0617 CCc1c(nc(s1)N)C(=O)OC 1W-0618 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccccc2F 1W-0622 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccccc6 1W-0625 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccccc6F 1W-0629 c1ccc(cc1)Oc2ccccc2O 1W-0639 c1cc(cc(c1)OCCBr)[N+](=O)[O-] 1W-0640 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/CO2 1W-0647 c1ccc2c(c1)C(=O)/C(=C/c3cccc(c3)Cl)/CO2 1W-0648 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)F)/CO2 1W-0649 c1ccc(c(c1)/C=C/2\COc3ccccc3C2=O)Br 1W-0650 Cc1ccc(cc1)/C=C/2\COc3ccccc3C2=O 1W-0659 c1ccc2c(c1)C(=O)/C(=C/c3cccc(c3)[N+](=O)[O-])/CO2 1W-0660 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccc(cc6)C(F)(F)F 1W-0663 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccccc6Br 1W-0664 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccc(c(c6)Cl)Cl 1W-0665 c1ccc(c(c1)/C=C/2\COc3ccccc3C2=O)Cl 1W-0667 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3Cl)Cl)/CO2 1W-0668 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)C#N)/CO2 1W-0669 c1ccc2c(c1)C(=O)/C(=C/c3ccc(c(c3)[N+](=O)[O-])Cl)/CO2 1W-0670 Cc1c(nc(s1)N)CC(=O)OC 1W-0674 Cc1ccc(cc1)C(c2ccccc2)C(=O)O 1W-0676 Cc1ccc(cc1)n2c(nn(c2=O)c3c(cc(cn3)C(F)(F)F)Cl)C 1W-0800 Cc1ccc(cc1)n2c(nn(c2=O)Cc3ccccc3)C 1W-0802 Cc1ccc(cc1)n2c(nn(c2=O)Cc3cccc(c3)C(F)(F)F)C 1W-0803 Cc1ccc(cc1)n2c(nn(c2=O)Cc3ccc(cc3)OC)C 1W-0804 Cc1c(sc2n1ncn2)c3ccc4ccccc4n3 1W-0805 Cc1ccc(cc1)c2ccc3cc(cc(c3n2)Br)Br 1W-0806 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccc4cc(cc(c4n3)Br)Br 1W-0807 c1ccc(cc1)c2ccc3cc(cc(c3n2)Br)Br 1W-0808 c1ccc(cc1)c2ccc(cc2)c3ccc4cc(cc(c4n3)Br)Br 1W-0809 c1cc(sc1)c2ccc3cc(cc(c3n2)Br)Br 1W-0810 Cc1cc2cc(cc(c2nc1c3ccccc3)Br)Br 1W-0811 c1ccc2cc(ccc2c1)c3ccc4cc(cc(c4n3)Br)Br 1W-0812 Cc1nn(c(=O)n1c2ccccc2)Cc3ccc(cc3)Cl 1W-0813 Cc1nn(c(=O)n1c2ccccc2)c3c(cc(cn3)C(F)(F)F)Cl 1W-0814 COc1ccc(cc1)c2cn3cc(cnc3n2)Br 1W-0815 c1cc(cc(c1)[N+](=O)[O-])c2cn3ccsc3n2 1W-0818 CCc1cc2cc(cc(c2nc1C)Br)Br 1W-0821 Cc1n[nH]c(=O)n1c2cccc(c2)C(F)(F)F 1W-0822 Cc1nn(c(=O)n1c2ccccc2Cl)Cc3ccc(cc3)Cl 1W-0824 Cc1nn(c(=O)n1c2ccccc2Cl)Cc3ccccc3 1W-0825 Cc1nn(c(=O)n1c2ccccc2Cl)c3c(cc(cn3)C(F)(F)F)Cl 1W-0826 Cc1nn(c(=O)n1c2ccccc2Cl)Cc3ccc(cc3)[N+](=O)[O-] 1W-0827 Cc1nn(c(=O)n1c2ccccc2Cl)CCOc3ccccc3 1W-0828 Cc1nn(c(=O)n1c2ccccc2Cl)Cc3cccc(c3)C(F)(F)F 1W-0830 Cc1nn(c(=O)n1c2ccccc2Cl)Cc3ccc(cc3)OC 1W-0831 c1ccc(c(c1)c2nnc3n2CCCCC3)O 1W-0832 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccccc2Cl 1W-0833 CCOC(=O)c1cnc2n(c1=O)CCS2 1W-0834 Cc1c(cccc1n2cccc2)N 1W-0835 Cc1nn(c(=O)n1c2ccccc2)CC3CC3 1W-0838 Cc1nn(c(=O)n1c2ccccc2)Cc3ccc(cc3)OC 1W-0839 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2)OC 1W-0840 Cc1nn(c(=O)n1c2ccccc2)C 1W-0841 Cc1nn(c(=O)n1c2ccc(cc2)OC)C 1W-0842 Cc1ccc(cc1)n2c(nn(c2=O)CCOc3ccccc3)C 1W-0843 Cc1nn(c(=O)n1c2ccc(cc2)OC)CC#N 1W-0846 Cc1nn(c(=O)n1c2ccc(cc2)OC)Cc3ccccc3 1W-0847 Cc1nc2ccc(cc2o1)N 1W-0848 c1cc(ccc1c2cnc3n(c2=O)CCS3)Cl 1W-0849 c1c2cc3c(nc2c(cc1Br)Br)CCCCC3 1W-0850 c1c2cc3c(nc2c(cc1Br)Br)CCCCCC3 1W-0852 c1cc2c(ccc3n2ccc3)c(c1)[N+](=O)[O-] 1W-0853 Cc1c(cc2ccccc2n1)OCc3ccc(cc3)Cl 1W-0854 Cc1nn(c(=O)n1c2ccc(cc2)OC)Cc3ccc(cc3)Cl 1W-0855 Cc1nn(c(=O)n1c2ccc(cc2)OC)c3c(cc(cn3)C(F)(F)F)Cl 1W-0856 Cc1nn(c(=O)n1c2ccc(cc2)OC)Cc3ccc(cc3)[N+](=O)[O-] 1W-0857 c1ccc2c(c1)cc3c(n2)CCCCC3 1W-0858 Cc1nn(c(=O)n1c2ccc(cc2)OC)Cc3cccc(c3)C(F)(F)F 1W-0859 Cc1nn(c(=O)n1c2ccccc2)Cc3cccc(c3)C(F)(F)F 1W-0860 Cc1nn(c(=O)n1c2ccccc2)CCOc3ccccc3 1W-0861 Cc1nn(c(=O)n1c2ccccc2)Cc3ccc(cc3)[N+](=O)[O-] 1W-0862 Cc1nn(c(=O)n1c2ccc(cc2)OC)CC3CC3 1W-0865 Cc1nn(c(=O)n1c2c(cccc2F)F)CC#N 1W-0866 Cc1nn(c(=O)n1c2c(cccc2F)F)Cc3ccccc3 1W-0867 Cc1nn(c(=O)n1c2c(cccc2F)F)Cc3cccc(c3)C(F)(F)F 1W-0868 Cc1nn(c(=O)n1c2ccc(cc2)OC)CCOc3ccccc3 1W-0871 c1c2cc3c(nc2c(cc1Br)Br)CCC3 1W-0872 c1ccn(c1)c2ccc(cc2)c3ccc4cc(cc(c4n3)Br)Br 1W-0873 Cc1nn(c(=O)n1c2ccc(cc2)OC)Cc3ccc(cc3)OC 1W-0876 c1cc(cc(c1)N)c2cn3ccsc3n2 1W-0877 COc1cc(c(cc1C(=O)OC)Br)n2cccc2 1W-0878 Cc1cn2c(nc1c3ccc(c(c3)OC)OC)nnn2 1W-0880 Cc1nn(c(=O)n1c2c(cccc2F)F)C 1W-0881 CCOC(=O)Cn1c(=O)n(c(n1)C)c2c(cccc2F)F 1W-0882 Cc1nn(c(=O)n1c2c(cccc2F)F)Cc3ccc(cc3)Cl 1W-0883 Cc1nn(c(=O)n1c2c(cccc2F)F)c3c(cc(cn3)C(F)(F)F)Cl 1W-0884 Cc1nn(c(=O)n1c2c(cccc2F)F)Cc3ccc(cc3)[N+](=O)[O-] 1W-0885 Cc1nn(c(=O)n1c2c(cccc2F)F)CCOc3ccccc3 1W-08864 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)C 1W-0887 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)CC#N 1W-0888 CCOC(=O)Cn1c(=O)n(c(n1)C)c2ccc(cc2OC)OC 1W-0889 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)Cc3ccccc3 1W-0890 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)Cc3ccc(cc3)Cl 1W-0891 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)c3c(cc(cn3)C(F)(F)F)Cl 1W-0892 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)CC3CC3 1W-0893 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)Cc3cccc(c3)C(F)(F)F 1W-0894 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)Cc3ccc(cc3)[N+](=O)[O-] 1W-0895 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)CCOc3ccccc3 1W-0896 Cc1nn(c(=O)n1c2ccc(cc2OC)OC)Cc3ccc(cc3)OC 1W-0897 c1ccc2c(c1)c(=O)n3c(n2)CCCCC3 1W-0898 CC(=O)c1cn(c2c1cccc2)C(=O)c3ccc(cc3)Cl 1W-0899 Cc1cc(n(n1)c2cc3cc(cc(c3nc2c4ccccc4)Br)Br)C 1W-0900 Cc1c(cc2ccccc2n1)OCc3cccc(c3)OC 1W-0901 Cc1c(cc2ccccc2n1)OCc3ccccc3 1W-0902 Cc1c(cc2ccccc2n1)OCc3ccc(cc3)F 1W-0903 CN1C(=O)C(SC1=O)Cc2ccc(cc2)NC(=O)CCl 1W-0905 C#CCN1CCN(CC1)c2ccc(cc2)F 1W-0906 Cc1cc(nc(n1)n2cc(nn2)c3ccc(cc3)OCc4ccccc4)CC(C)C 1W-0907 Cc1c(c(n2c(n1)c(cn2)c3cccs3)C)Cc4cccc(c4)F 1W-0909 c1ccc2c(c1)c3c([nH]2)C(N(CC3)/C=C\4/c5ccccc5C(=O)O4)C6c7ccccc7C(=O)O6 1W-0910 COC(=O)c1c(ccs1)n2cc(nn2)c3ccc(cc3)OCc4ccccc4 1W-0911 CC1(CN(C1=O)c2cccc(c2)c3ccnc4n3ncc4c5ccc(cc5)OC)C 1W-0912 c1ccc(cc1)c2cc(nc3n2nnn3)C(F)(F)F 1W-0913 c1ccc2c(c1)cc3c(n2)CCCCCC3 1W-0914 CCc1nc2ccc(cc2o1)[N+](=O)[O-] 1W-0916 c1cc(nc2c1cc(cc2Br)Br)c3ccc4c(c3)OCO4 1W-0917 c1c2cc3c(nc2c(cc1Br)Br)CCCC3 1W-0918 Cc1c(n(ccc1=O)CCc2c[nH]c3c2cccc3)C 1W-0921 CC(C)CCC1C(=O)N(C(=O)S1)C 1W-0922 CCc1nc2ccc(cc2o1)N 1W-0924 CN1CCN(CC1)c2ccc(cc2)c3ccc4ccccc4n3 1W-0926 CN1CCN(CC1)c2ccc(cc2)c3ccc4cc(cc(c4n3)Br)Br 1W-0927 Cc1nc2cc(ccc2o1)[N+](=O)[O-] 1W-0929 CCc1nc2cc(ccc2o1)[N+](=O)[O-] 1W-0930 COc1cc2c(cc1OC)nc3n(c2=O)CCCCC3 1W-0932 c1cc2c(cc1Br)c(=O)n3c(n2)CCCCC3 1W-0933 c1ccc2c(c1)C(=O)NN=CO2 1W-0935 c1ccc2c(c1)ccc(n2)c3ccc(cc3)c4ccc(cc4)Br 1W-0936 c1cc(ccc1c2ccc(cc2)Br)c3ccc4cc(cc(c4n3)Br)Br 1W-0937 CNc1ncc(s1)c2ccc3cc(cc(c3n2)Br)Br 1W-0938 Cc1nc2ccc(cc2o1)n3cccc3 1W-0939 CCc1nc2ccc(cc2o1)n3cccc3 1W-0940 c1ccn2cc(nc2c1)c3cccc(c3)n4cccc4 1W-0942 c1ccc2c(c1)C(=O)N(C2=O)n3cccc3 1W-0944 c1cc2c(c(c1)[N+](=O)[O-])[nH]nc2Br 1W-0945 c1ccc2c(c1)ccc(n2)c3ccc(cc3)n4cccc4 1W-0947 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)CC#N 1W-0953 CCOC(=O)Cn1c(=O)n(c(n1)C)c2cccc(c2)C(F)(F)F 1W-0954 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)Cc3ccccc3 1W-0955 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)Cc3ccc(cc3)Cl 1W-0956 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)c3c(cc(cn3)C(F)(F)F)Cl 1W-0957 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)CC3CC3 1W-0958 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)Cc3cccc(c3)C(F)(F)F 1W-0959 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)CCOc3ccccc3 1W-0960 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)Cc3ccc(cc3)OC 1W-0961 Cc1nn(c(=O)n1c2cccc(c2)C(F)(F)F)Cc3ccc(cc3)[N+](=O)[O-] 1W-0962 c1cc(c(nc1)N/N=C(/C=C(/C(F)(F)F)\O)\C(F)(F)F)[N+](=O)[O-] 1W-0963 CN1C(=O)C(SC1=O)Cc2ccc(cc2)NC(=O)C3CCCCC3 1W-0964 CCCc1c(nn(c1C)c2c(cccn2)[N+](=O)[O-])C 1W-0965 Cc1cccc2c1nc3n(c2=O)CCCCC3 1W-0967 Cc1c(cnc(n1)N)c2ccc3c(c2)OCO3 1W-1421 CN(C)c1c(cc(s1)C(=O)c2cccnc2)c3ccccc3 1W-7010 CCN1c2ccccc2CC1=O 1X-0007 CCn1c2c(c(n1)C)c(c(cn2)C(=O)OCC)Oc3ccc(cc3)F 1X-0030 Cc1ccc(cc1)S(=O)(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 1X-0202 c1cc(sc1)S(=O)(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 1X-0203 c1cc2c(cc1C(F)(F)F)N(CC3N2CCC3)S(=O)(=O)c4cc(ccc4Cl)Cl 1X-0204 Cc1ccc(cc1)NC(=S)NNC(=O)Cc2c3ccccc3on2 1X-0205 CC1(C(=O)Nc2ccccc2O1)c3nc(no3)c4ccncc4 1X-0209 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)N 1X-0210 Cc1ccc(cc1)c2csc(n2)/C(=C/c3coc4ccccc4c3=O)/C#N 1X-0211 c1cc(sc1)C(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 1X-0212 c1cc(ccc1C(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F)I 1X-0213 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OCc4ccccc4Cl 1X-0214 Cc1ccc(cc1)n2c(nnc2S)Cc3c4ccccc4on3 1X-0216 c1cc2c(nc1)NC(=O)C(O2)CCN3CCN(CC3)Cc4ccc5c(c4)OCO5 1X-0219 c1ccc(cc1)c2cc(=O)n([nH]2)C(=N)N 1X-0220 Cc1c(nc(s1)Cc2nc(cs2)O)c3ccccc3 1X-0221 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)CBr 1X-0222 c1cc(c(c(c1)F)C(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F)F 1X-0223 COc1ccc(cc1)C(=O)N2CC3CCCN3c4c2cc(cc4)C(F)(F)F 1X-0224 c1cc2c(cc1C(F)(F)F)N(CC3N2CCC3)C(=O)c4ccc(cc4Cl)Cl 1X-0225 c1ccc(cc1)C2C(=C(n3c(c(cn3)C#N)N2)N)C#N 1X-0226 Cc1ccc(cc1)c2nc(cs2)CCN.Br 1X-0227 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)CN3CCOCC3 1X-0230 Cc1ccc(cc1)/C=C(\c2nc(cs2)O)/c3nc(c(s3)C)c4ccccc4 1X-0231 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OC(=O)c4cccc(c4)Br 1X-0234 c1cc2c(cc1/C=C/3\C(=O)NC(=N3)N4CSCC4C(=O)O)OCO2 1X-0235 COC(=O)/C=C/CSC1=N/C(=C/c2ccc3c(c2)OCO3)/C(=O)N1 1X-0236 Cc1c(nc(s1)/C(=C/c2ccccc2C(F)(F)F)/c3nc(cs3)O)c4ccccc4 1X-0239 c1cc(ccc1c2c(cnc(n2)N)CCN3CCOCC3)F 1X-0240 CC1(C(=O)Nc2ccccc2O1)c3nc(no3)c4ccc(cc4)C(F)(F)F 1X-0241 c1cc2c(cc1/C=C/3\C(=O)N4C(=O)C5CSCN5C4=N3)OCO2 1X-0243 c1cc2c(cc1/C=C/3\C(=O)NC(=N3)SCc4cnc(s4)Cl)OCO2 1X-0246 CC(C)(C)c1csc(n1)Cc2nc(cs2)O 1X-0247 Cc1cc2nc(c(cn2n1)CCN3CCOCC3)c4ccc(cc4)F 1X-0248 CC1(C(=O)Nc2ccccc2O1)C(=O)NNC(=O)c3cccc(c3)C(F)(F)F 1X-0249 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3OCc4cccc(c4)C(F)(F)F 1X-0250 c1cc(ccc1c2c(cc3c(nc(nc3n2)N)N)CCN4CCOCC4)F 1X-0253 c1cc(ccc1c2c(cn3c(n2)ncn3)CCN4CCOCC4)F 1X-0254 c1cc(ccc1c2c(cn3c(n2)nc(n3)N)CCN4CCOCC4)F.O 1X-0261 CC1(C(=O)Nc2c(cccn2)O1)C(=O)NCCCN3CCOCC3 1X-0262 Cc1c(c(=O)[nH]c(n1)n2c(=O)cc([nH]2)c3ccccc3)Cc4ccc(cc4)F 1X-0265 c1cc(cc(c1)Cl)c2nc(cs2)CCNc3ccc(cn3)[N+](=O)[O-] 1X-0266 CCCCCC(=O)NNC(=O)C1(C(=O)Nc2ccccc2O1)C 1X-0270 c1ccc(c(c1)C(=O)c2cnn(c2)c3ccc(cc3)Cl)OC(=O)c4ccco4 1X-0271 c1ccc(cc1)c2cnn3c2nc(c(c3)CCN4CCOCC4)c5ccc(cc5)F 1X-0272 Cc1n[nH]c(=O)n1c2cccc(c2)[N+](=O)[O-] 1X-0276 c1cc(ccc1c2c(cn3c(n2)c(cn3)c4ccc(cc4)Cl)CCN5CCOCC5)F 1X-0278 c1cc(cc(c1)Cl)c2nc(cs2)CCNc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 1X-0279 c1cc(cc(c1)Cl)c2nc(cs2)CCNc3ccc(cc3C#N)[N+](=O)[O-] 1X-0281 C/C(=N/OCc1c(cccc1Cl)Cl)/c2cccc(c2)N3Cc4ccccc4C3 1X-0282 c1cc(ccc1c2cnn3c2nc(c(c3)CCN4CCOCC4)c5ccc(cc5)F)F 1X-0283 Cc1cn2c(c(cn2)c3ccc(cc3)Cl)nc1c4ccc(c(c4)F)OC 1X-0285 CC1(C(=O)Nc2c(cccn2)O1)C(=O)NCC3CCCO3 1X-0288 Cc1cn2c(c(cn2)c3ccc(cc3)F)nc1c4ccc(c(c4)F)OC 1X-0289 c1cc(sc1)S(=O)(=O)N2CC3CCCN3c4c2ccc(c4)C(F)(F)F 1X-0290 c1cc2cccnc2c(c1)S(=O)(=O)N3CC4CCCN4c5c3ccc(c5)C(F)(F)F 1X-0291 CCc1cc(=O)[nH]c(n1)n2c(=O)cc([nH]2)c3ccccc3 1X-0292 C/C(=N/OCc1ccc(cc1)C(F)(F)F)/c2cccc(c2)N3Cc4ccccc4C3 1X-0293 C/C(=N/OCc1cccc(c1)C(F)(F)F)/c2cccc(c2)N3Cc4ccccc4C3 1X-0294 Cc1ccc(cc1)CO/N=C(/C)\c2cccc(c2)N3Cc4ccccc4C3 1X-0295 C/C(=N/OCc1c(cccc1Cl)F)/c2cccc(c2)N3Cc4ccccc4C3 1X-0296 C/C(=N/OCc1ccc(cc1Cl)F)/c2cccc(c2)N3Cc4ccccc4C3 1X-0298 C/C(=N/OCc1ccccc1[N+](=O)[O-])/c2cccc(c2)N3Cc4ccccc4C3 1X-0299 C/C(=N\OCc1ccccc1Br)/c2cccc(c2)N3Cc4ccccc4C3 1X-0300 Cc1cn2c(ncn2)nc1c3ccc(c(c3)F)OC 1X-0302 CCC(C)(C)c1ccc(cc1)S(=O)(=O)N2CC3CCCN3c4c2ccc(c4)C(F)(F)F 1X-0303 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CC3CCCN3c4c2ccc(c4)C(F)(F)F 1X-0304 c1cc(ccc1S(=O)(=O)N2CC3CCCN3c4c2ccc(c4)C(F)(F)F)I 1X-0305 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc3c(c2)CN(CC3)C(=O)C(F)(F)F)c4ccccc4)CCO 1X-0306 Cc1c(c(=O)[nH]n1S(=O)(=O)c2cccc3c2nccc3)CCO 1X-0307 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccc(cc2[N+](=O)[O-])OC)CCO 1X-0308 Cc1cn2c(c(cn2)c3ccccc3)nc1c4ccc(c(c4)F)OC 1X-0310 Cc1cn2c(nc1c3ccc(c(c3)F)OC)nc(n2)N 1X-0311 Cc1c(c(c(c(c1C)C)S(=O)(=O)n2c(c(c(=O)[nH]2)CCO)C)C)C 1X-0312 Cc1c2cc(ccc2sc1S(=O)(=O)n3c(c(c(=O)[nH]3)CCO)C)Cl 1X-0313 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)n2c(c(c(=O)[nH]2)CCO)C 1X-0314 Cc1ccc(cc1)c2nc(cs2)CCNc3c(cccn3)[N+](=O)[O-] 1X-0315 Cc1ccc(cc1)c2nc(cs2)CCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F 1X-0316 Cc1ccc(cc1)c2nc(cs2)CCNc3ccc(cc3C)[N+](=O)[O-] 1X-0317 COc1ccc(cc1S(=O)(=O)N2CC3CCCN3c4c2ccc(c4)C(F)(F)F)Cl 1X-0319 COc1ccc(cc1OC)Cl 1X-0320 c1ccc2c(c1)NCCO2 1X-0323 c1cc(ccc1NC(=O)NN)[N+](=O)[O-] 1X-0324 CCOC(=O)N1CCN(CC1)c2ccc(cc2)N 1X-0601 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C=O 1X-0701 CC(c1c(nn(c1Cl)C)C(F)(F)F)O 1X-0702 CS(=O)(=O)c1ccc(cc1)C(=O)CO 1X-0706 CC(C)(C=O)N1CCN(CC1)Cc2ccccc2 1X-0709 CCOC(=O)C1CCN(CC1)C(C)(C)C=O 1X-0710 CS(=O)(=O)c1ccc(cc1)C(=O)CN.Cl 1X-0714 CS(=O)(=O)c1ccc(cc1)c2csc(n2)N 1X-0715 CCOC(=O)c1csc(n1)N 1X-0716 c1nc(c(c(n1)Cl)C=O)Cl 1X-0802 CN(C)/C=C/C=C(C(=O)OC)C(=O)OC 1X-0803 c1nc(c(c(n1)Cl)C=O)N2CCOCC2 1X-0804 c1nc(c(c(n1)Cl)C=O)N 1X-0805 c1ccc(cc1)CC2CCN(CC2)c3c(c(ncn3)Cl)C=O 1X-0806 c1cc(cnc1)C(CC(=O)O)N 1X-0807 CC(C)c1ccc(cc1)C(CC(=O)O)NC(=O)c2cccs2 1X-0808 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC#CCOc4cccc5c4cccc5 1X-0811 COc1ccc(cc1)C(CCO)N2Cc3ccccc3C2=O 1X-0813 CC(C)c1ccc(cc1)C(CC(=O)O)NC(=O)c2cccc(c2)OC 1X-0814 c1ccc2c(c1)OCC(O2)C(=O)N3CCNCC3 1X-0816 Cc1ccc(c2c1c3cc(ccc3[nH]2)OC)C 1X-0817 CSc1ccc(cc1)C(CCO)N 1X-0818 c1ccc2c(c1)ccn2Cc3ccc(nc3)Cl 1X-0819 COC(=O)c1cc2ccccc2n1Cc3ccc(nc3)Cl 1X-0820 c1ccc(cc1)CC2CCN(CC2)Cc3ccc(nc3)Cl 1X-0821 Cc1nccn1Cc2ccc(nc2)Cl 1X-0823 Cc1cc(n(n1)Cc2ccc(nc2)Cl)C 1X-0824 c1cc(ccc1C#N)OCc2ccc(nc2)Cl 1X-0825 CC(C)c1ccc(cc1)C(CC(=O)O)NS(=O)(=O)c2ccccc2 1X-0826 CC(C)c1ccc(cc1)C(CC(=O)O)NC(=O)C2CCCCC2 1X-0827 c1cc(cc(c1)Cl)C(CCO)N 1X-0828 COc1ccc(cc1Cl)CO 1X-0829 COc1ccc(cc1Cl)/C=C/C(=O)c2ccc(cc2)Cl 1X-0830 COc1ccc(cc1Cl)/C=C/C(=O)c2ccc(cc2)F 1X-0831 COc1cccc(c1)C(=O)/C=C/c2ccc(c(c2)Cl)OC 1X-0832 Cc1ccc(cc1)C(=O)/C=C/c2ccc(c(c2)Cl)OC 1X-0833 COc1ccc(cc1Cl)/C=C/C(=O)c2ccc(cc2)[N+](=O)[O-] 1X-0834 COc1ccc(cc1Cl)/C=C/C(=O)c2ccc(cc2)C3CCCCC3 1X-0835 Cc1ccc(c2c1c3cc(ccc3[nH]2)Br)C 1X-0836 CN1C(=O)C(=Cc2ccc(c(c2)OC)OCc3ccc(nc3)Cl)C(=O)N(C1=O)C 1X-0837 CC(=O)/C=C/c1ccc(cc1)OCc2ccc(nc2)Cl 1X-0839 COc1ccc2c(c1)c(c[nH]2)/C=C(/C#N)\S(=O)(=O)c3ccccc3 1X-0840 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)OC 1X-0841 CN1CCN(CC1)Cc2c(nnn2c3ccc(cc3)C(F)(F)F)c4ccccc4 1X-0842 COc1ccc(cc1Cl)/C=N/NS(=O)(=O)c2ccccc2 1X-0843 COc1ccc2c(c1)c(c[nH]2)/C=C(/C#N)\C(=O)c3ccc(cc3)Cl 1X-0845 COc1ccc(cc1Cl)/C=N/O 1X-0847 COc1ccc(cc1Cl)C=C(C#N)C#N 1X-0848 c1cc(ncc1CNc2[nH+]ccs2)Cl.[Cl-] 1X-0849 CC(C)c1ccc(cc1)C(CC(=O)O)NC(=O)CCCl 1X-0852 CC(=O)c1cn(c2c1cccc2)C(=O)C3CCCCC3 1X-0853 CC(=O)c1cn(c2c1cccc2)C(=O)c3ccc(cc3)OC 1X-0854 COc1ccc(cc1Cl)/C=N/NC(=O)c2ccc(cc2Cl)Cl 1X-0859 COc1ccc(cc1Cl)/C=N/NC(=O)c2ccccc2 1X-0860 COc1cc(ccc1OCc2ccc(nc2)Cl)/C=C/3\c4ccccc4NC3=O 1X-0863 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C/N=N/C(=O)CN2Cc3ccccc3C2=O 1X-0864 Cc1ccc(c2c1c3ccccc3n2Cc4ccccc4)C 1X-0865 Cc1ccc(c2c1c3ccccc3n2C=O)C 1X-0866 c1ccc(cc1)CCNC(=O)C2COc3ccccc3O2 1X-0867 COc1cc(ccc1OCc2ccc(nc2)Cl)/C=N/CCc3ccccc3 1X-0868 c1ccc(cc1)N2CCN(CC2)C(=O)C3COc4ccccc4O3 1X-0869 COc1ccc(cc1Cl)/C=N/Cc2ccc(cc2)Cl 1X-0870 COc1ccc(cc1Cl)/C=N/CCO 1X-0871 Cc1ccc(cc1)C(=O)N/N=C/c2ccc(c(c2)Cl)OC 1X-0872 c1cc(ncc1CN2CCCCC2=O)Cl 1X-0873 Cc1cc(n(c(=O)c1C#N)Cc2ccc(nc2)Cl)C 1X-0874 COc1ccn(c(=O)c1C#N)Cc2ccc(nc2)Cl 1X-0875 Cc1cc(c(c(n1)OCc2ccc(nc2)Cl)C#N)C(F)(F)F 1X-0876 c1ccn(c1)Cc2ccc(nc2)Cl 1X-0877 Cc1ccc(c2c1c3ccccc3n2CC=C)C 1X-0879 COc1cc(ccc1OCc2ccc(nc2)Cl)/C=N/CC3CCCO3 1X-0880 Cc1ccc(c2c1c3ccccc3n2CC(=O)OC(C)(C)C)C 1X-0881 Cc1cc(nc(n1)n2cc(nn2)C(=O)c3ccc(cc3)OC)C(F)(F)F 1X-0883 COc1ccc2c(c1)c(c[nH]2)/C=C(/C#N)\C(=O)c3ccccc3 1X-0884 Cc1cc(nc(n1)n2cc(nn2)C(=O)c3ccc4ccccc4c3)C(F)(F)F 1X-0885 COc1ccc2c(c1)c(c[nH]2)/C=C\3/c4ccccc4NC3=O 1X-0886 CN1C(=O)c2ccccc2/C(=C\c3c[nH]c4c3cc(cc4)OC)/C1=O 1X-0887 Cc1ccc(n1C(CC(=O)O)c2cccc(c2)Cl)C 1X-0889 COc1cc(ccc1OCc2ccc(nc2)Cl)/C=N/NC(=S)N 1X-0891 COc1ccc(cc1Cl)/C=C(\C#N)/S(=O)(=O)c2ccccc2 1X-0892 COc1ccc(cc1Cl)/C=C(\C#N)/C(=O)c2ccccc2Cl 1X-0893 Cc1ccc(cc1)/C(=C/c2ccc(c(c2)Cl)OC)/C#N 1X-0894 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(c(c2)Cl)OC)/C#N 1X-0895 CC1(C(=O)Nc2ccccc2O1)C(=O)N/N=C/c3ccccc3F 1X-0897 CN1CCC2(CC1)c3c(c4cc(ccc4[nH]3)OC)CCN2.Cl.Cl 1X-0899 COc1ccc2c(c1)c3c([nH]2)C4(CN5CCC4CC5)NCC3 1X-0900 c1ccc(cc1)COc2ccc(cc2)C(CCO)N 1X-0901 COc1c(c(ncn1)N2CCC(CC2)Cc3ccccc3)C=O 1X-0902 COc1ccc(cc1Cl)/C=C/2\C(=O)OC(=N2)c3ccccc3 1X-0903 Cc1ccc(n1c2ccc(cn2)C#N)C 1X-0904 Cc1ccc(n1C(CC(=O)O)c2ccc(cc2)OCc3ccccc3)C 1X-0905 c1ccc(c(c1)N)NC(=O)c2c(nc3ccccc3n2)C(F)(F)F 1X-0908 CC1(C(=O)Nc2ccccc2O1)C(=O)NCc3ccc(cc3)F 1X-0911 CSc1nc(cc(n1)O)C(=O)O 1X-0921 c1cc2c(cc1/C=C/C(=O)O)CCC2 1X-0923 CCCc1c(cnc(n1)N)C(=O)OCC 1X-0926 c1ccc(cc1)OCCSCC(=O)O 1X-0927 Cc1c(nc(o1)c2ccccc2)CC(=O)O 1X-0928 Cc1csc2c1c(ncn2)Sc3ccccc3N 1X-0929 CCOC(=O)C(C(=O)OCC)Nc1ccc(cc1)Cl 1X-0930 COc1ncc(c(n1)N)C#N 1X-0931 CCN(CC)C(=S)SCC(=O)O 1X-0932 Cc1cc(nc(c1C#N)C)N 1X-0933 c1cc2c(cc1/C=C/C=C/C(=O)O)OCO2 1X-0937 CNCc1ccco1 1X-0939 c1ccc2c(c1)c(c[nH]2)S 1X-5008 c1cc(c(cc1I)N)C(=O)O 1X-5042 c1c(c(n[nH]c1=O)Cl)Cl 1X-7067 c1cc2c(cc1NCC(C(F)(F)F)O)NC(=O)CO2 1Y-0005 c1ccc(cc1)n2cc(c(n2)c3ccc4c(c3)CCC4)CO 1Y-0009 c1cc2c(cc1NS(=O)(=O)Cc3cc(cc(c3)Cl)Cl)NC(=O)CO2 1Y-0012 CS(=O)(=O)c1ccc(cc1)c2csc(n2)NC(=O)Nc3ccccc3 1Y-0082 CS(=O)(=O)c1ccc(cc1)c2csc(n2)NC(=O)c3ccco3 1Y-0096 CS(=O)(=O)c1ccc(cc1)c2csc(n2)NC(=O)c3ccccc3F 1Y-0097 CS(=O)(=O)c1ccc(cc1)c2csc(n2)c3ccccc3 1Y-0234 c1cnccc1CNC(=O)c2cc(c([nH]2)Br)Br 1Y-0242 c1ccc(cc1)c2nc(cs2)c3ccc(cc3)S(=O)(=O)/C=C/c4ccc(cc4)C(F)(F)F 1Y-0244 CS(=O)(=O)c1ccc(cc1)c2csc(n2)c3cccc(c3)C(F)(F)F 1Y-0251 c1cc(ccc1C(=O)Oc2c(c(c(c(c2F)F)F)F)F)C(=O)Oc3c(c(c(c(c3F)F)F)F)F 1Y-0252 c1cc(c(cc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)Cl)Cl 1Y-0263 c1cc(c(c(c1)Cl)Cl)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 1Y-0264 CN(C)c1cccc2c1cccc2S(=O)(=O)Oc3c(c(c(c(c3F)F)F)F)F 1Y-0265 c1ccc(c(c1)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)Cl 1Y-0267 c1cc(ccc1C#N)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 1Y-0268 c1cc(ccc1C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)F 1Y-0270 c1cc(c(cc1Cl)Cl)S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F 1Y-0271 c1cc(ccc1C2c3cc4c(cc3NC5=C2C(=O)OC5)OCCO4)F 1Y-0272 c1cc(ccc1c2c3cc4c(cc3nc5c2C(=O)OC5)OCO4)F 1Y-0274 CS(=O)(=O)Oc1c(c(c(c(c1F)F)F)F)F 1Y-0285 CC(=O)N(C)c1ccc(cc1)[N+](=O)[O-] 1Y-0609 COC(=O)c1cc(n[nH]1)c2ccccc2 1Y-0617 COc1ccc(cc1)c2ccc(s2)C(=O)NN 1Y-0700 c1ccc(cc1)c2ccc(s2)C=O 1Y-0702 c1cc(ccc1c2ccc(s2)C=O)Cl 1Y-0703 c1ccc(cc1)c2nc(cs2)C(=O)NN 1Y-0704 CC(=O)c1ccc(s1)c2ccc(cc2)OC 1Y-0706 c1cc(ccc1C=O)c2ccc(cc2)[N+](=O)[O-] 1Y-0709 CC(=O)c1ccc(s1)c2ccc(cc2)Cl 1Y-0711 CC(=O)c1ccc(s1)c2ccc(cc2)F 1Y-0712 c1ccc(c(c1)C(=O)CBr)Cl 1Y-0714 c1cnc(cc1C#N)Cl 1Y-0715 c1cc(c(nc1)N2CCCCC2)C=O 1Y-0716 c1ccc(cc1)CN2CCN(CC2)c3c(cccn3)C=O 1Y-0717 CCOC(=O)C1CCN(CC1)c2c(cccn2)C=O 1Y-0718 c1cc(c(nc1)N2CCOCC2)C=O 1Y-0719 CCOC(=O)C1CCN(CC1)c2ccc(cn2)[N+](=O)[O-] 1Y-0723 COC(=O)c1ccc(cc1)c2ccc(c(c2)C(F)(F)F)[N+](=O)[O-] 1Y-0728 COC(=O)c1ccc(cc1)c2ccc(cn2)CCl 1Y-0730 COC(=O)c1ccc(cc1)c2cc(ccn2)C#N 1Y-0732 COc1ccc(cc1)c2c(cccn2)C=O 1Y-0733 c1cc(ccc1C(=O)O)N2CCOCC2 1Y-0800 c1c(c[nH]c1C(=O)C(Cl)(Cl)Cl)Br 1Y-0801 CN(C)/C=C/c1cc(ccc1[N+](=O)[O-])C(=O)OC 1Y-0802 Cc1cc(n[nH]1)C(=O)O 1Y-0803 Cc1cc(n2c(n1)nc(n2)SCCCF)C 1Y-0805 Cc1cc(n2c(n1)nc(n2)SCc3ccc(cc3)C(F)(F)F)C 1Y-0806 Cc1cc(n2c(n1)nc(n2)SCc3ccc(cc3)Cl)C 1Y-0807 Cc1cn(c(=O)[nH]c1=O)CC(=O)O 1Y-0808 COC(=O)c1ccc(c(c1)F)N2CCOCC2 1Y-0809 Cc1nn(c(=O)n1c2ccc(c(c2)OC)OC)CC#N 1Y-0810 CC(C)(C)O/N=C(/c1ccc(nc1)C2CC2)\C3CC3 1Y-0812 c1c(c[nH]c1C(=O)N2CCOCC2)Br 1Y-0813 c1ccc2c(c1)CN(C2=O)Cc3ccc(cc3)C(=O)O 1Y-0814 COC(=O)c1cc(c[nH]1)Br 1Y-0815 Cc1cc(n2c(n1)nc(n2)SCc3c(cccc3Cl)F)C 1Y-0819 Cc1cc(n2c(n1)nc(n2)SC3CCCC3)C 1Y-0820 CCOC(=O)c1c(n2cc(ccc2n1)Cl)Br 1Y-0822 Cc1c2cc3c(cc2ncc1/C(=N/OCc4ccccc4)/C5CC5)OCO3 1Y-0823 Cc1cc(nc(n1)n2c(c(nn2)C(=O)OC)C(=O)OC)C 1Y-0824 c1ccc2c(c1)c(=O)n(c3n2ncc3C#N)Cc4cccc(c4)C(F)(F)F 1Y-0826 c1cc(ccc1C(=O)C(CC(=O)O)Br)F 1Y-0827 c1cc(ccc1C(=O)C(CC(=O)O)Br)Cl 1Y-0828 COc1ccc(cc1S(=O)(=O)n2cc(cc2C(=O)OC)Br)Cl 1Y-0829 Cc1ccc(n1c2c(csc2C(=O)OC)C#N)C 1Y-0830 CC(=O)N1CCC(CC1)C(=O)Nc2cccc(c2)C#C 1Y-0833 Cc1cc(n[nH]1)c2ccc(s2)Br 1Y-0835 Cc1cc(n[nH]1)c2c(ccs2)Cl 1Y-0836 Cc1cc(n[nH]1)c2c(ccs2)Br 1Y-0837 Cc1cc(n[nH]1)c2ccc(s2)Cl 1Y-0838 c1cc2nc(c(n2cc1Cl)Cl)C(=O)O 1Y-0839 Cc1cc(cn2c1ncc2)I 1Y-0841 c1cc2nc(c(n2cc1Cl)Br)C(=O)NN 1Y-0842 c1cc2nc(c(n2cc1Cl)Br)C(=O)O 1Y-0843 Cc1cc(nc(n1)n2cc(nn2)C(=O)c3ccccn3)C 1Y-0847 c1ccc2cc3c(cc2c1)C(C(=C(O3)N)C#N)c4cccnc4 1Y-0920 CC(=O)Nc1ccc(cc1)I 1Y-0922 c1cc(ccc1c2c(nc(s2)N)C(=O)NN)Cl 1Y-0925 c1ccc(c(c1)/C=C/2\C(=O)NC(=S)N2)N3CCOCC3 1Y-0928 COc1cc(c(c(c1OC)OC)C=O)OCC#C 1Y-0929 CC(C)(C)c1ccc(cc1)c2c(nc(s2)N)C(=O)NN 1Y-0930 c1cc(ccc1c2c(nc(s2)N)C(=O)NN)F 1Y-0931 CC1(CNc2cc(ccc2S1)N)C 1Y-0933 COc1cc(cc(c1OC)OC)OCC=C 1Y-0934 c1cc(cc(c1)F)c2c(nc(s2)N)C(=O)NN 1Y-0935 c1ccc2cc3c(cc2c1)C(C(=C(O3)N)C#N)c4ccc(cc4)F 1Y-0938 c1ccc2cc3c(cc2c1)C(C(=C(O3)N)C#N)c4cccs4 1Y-0939 c1ccc(cc1)c2c(nc(s2)N)C(=O)NN 1Y-0944 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCc2ccco2 1Y-0946 c1cc(ccc1C2c3cc4cc(ccc4cc3OC(=C2C#N)N)Br)F 1Y-0949 Cc1c2c(c3ccccc3n1)OC(=C(C2c4cccs4)C#N)N 1Y-0954 Cc1c(c2ccccc2nc1c3cccc(c3)Cl)C(=O)O 1Y-0958 COc1cccc(c1)C2c3cc4ccccc4cc3OC(=C2C#N)N 1Y-0959 CCOC(=O)/C(=N\Nc1ccc(cc1[N+](=O)[O-])OC)/Cl 1Y-0960 CCOC(=O)/C(=N\Nc1ccc(cc1[N+](=O)[O-])Cl)/Cl 1Y-0961 Cc1ccc(cc1)C2c3cc4ccccc4cc3OC(=C2C#N)N 1Y-0962 c1ccc(c(c1)C2c3cc4cc(ccc4cc3OC(=C2C#N)N)Br)C(F)(F)F 1Y-0965 c1cc(cc2c1cc3c(c2)C(C(=C(O3)N)C#N)c4ccc(c(c4)[N+](=O)[O-])Cl)Br 1Y-0966 CCOC(=O)/C(=N\Nc1ccc(cc1)C)/Cl 1Y-0967 c1cc2c(cc1Br)c(c[nH]2)CCO 1Y-5033 Cc1ccc(cc1)C(=O)NCCN2CCOCC2 1Y-5036 COc1ccc(c(c1OC)OC)C(=O)NCCN2CCOCC2 1Y-5037 c1cc(sc1)/C(=C/c2ccc3c(c2)OCO3)/C#N 1Y-5051 CC(=O)NCc1ccc(cc1)Br 1Z-0016 COc1ccc(c(c1)C#N)C(F)(F)F 1Z-0027 c1csc2c1nc[nH]c2=O 1Z-0222 c1csc2c1ncnc2Cl 1Z-0226 CC(=C)n1c2ccccc2[nH]c1=O 1Z-0600 CC(=C)n1c2ccccc2n(c1=O)CCCC(=O)O 1Z-0602 c1ccc2c(c1)[nH]c(=O)n2CCCC(=O)O 1Z-0605 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCNCC2 1Z-0807 Cc1c(cccc1[N+](=O)[O-])C(=O)N/N=C/OC 1Z-0811 Cc1ccc2c(c1)nc(o2)CCl 1Z-0812 Cc1cccc(c1)C(=O)NCC(=O)OC 1Z-0816 c1cc(ccc1c2nnc(o2)CN3CCCCC3)I 1Z-0817 CC(C)(C)c1ccc2c(c1)nc(o2)CCl 1Z-0828 Cc1ccc2c(c1)oc(n2)CCl 1Z-0830 Cc1cc(n(n1)c2nc(cs2)CO)C(F)(F)F 1Z-0832 CCCNC(=S)N1CCCN(CC1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F 1Z-0837 c1ccc2c(c1)nc(s2)CCl 1Z-0838 c1cc(ccc1C#N)NC(=S)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F 1Z-0841 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCN(CC2)C(=S)Nc3ccc(cc3Br)F 1Z-0842 c1cc2c(cc1[N+](=O)[O-])C(=O)CC2 1Z-5050 c1cc2c(cc1S(=O)(=O)Cl)C(=O)CCC2 1Z-7003 c1cc2c(cc1S(=O)(=O)Cl)C(=O)CC2 1Z-7004 CN/C(=C\[N+](=O)[O-])/NC(=N)N 2B-001 CS/C(=C/[N+](=O)[O-])/Nc1ccc(cc1F)O 2B-002 CN(C)N/C(=C/[N+](=O)[O-])/SC 2B-003 COc1cccc(c1OCC(=O)O)C=O 2B-004 C1CN(NC1=O)N=O 2B-005 CN(C)N/C(=C/[N+](=O)[O-])/NN 2B-006 COc1cccc(c1OCC(=O)O)/C=N/O 2B-007 C1CSC(=N1)NN.I 2B-008 COc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccc(cc2F)O 2B-009 c1cc(cnc1)/C=C(\C#N)/C(=O)Nc2ccc(cc2F)O 2B-010 c1cc(ccc1N/C(=C/[N+](=O)[O-])/NN)Cl 2B-011 c1cc(c(cc1O)F)N/C(=C/[N+](=O)[O-])/NN 2B-013 COc1cccc(c1OCC(=O)O)C#N 2B-014 CC1=NN(C(=O)C1)C2=NCCS2 2B-016 c1cc(ccc1n2c(nnc2C(F)(F)F)C[N+](=O)[O-])Cl 2B-018 c1ccc(cc1)CNC(=C[N+](=O)[O-])NCc2ccccc2 2B-023 COc1ccc(cc1)N/C(=C/[N+](=O)[O-])/SC 2B-024 COc1ccc(cc1)N/C(=C/[N+](=O)[O-])/NN 2B-025 CONC(=O)N 2B-032 COc1ccc(cc1)n2c(nnc2C(F)(F)F)C[N+](=O)[O-] 2B-037 c1cc(oc1)C(=O)N 2B-052 c1ccc(cc1)NC(=O)CN2CCC(=O)N2 2B-054 CC1=NN(C(=O)C1)C2=NCCN2 2B-057 CC1(OC(=O)C(=Cc2ccc(cc2)Cl)C(=O)O1)C 2B-063 CN(C)/C=N\C(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 2B-064 c1cc(c(cc1OCC(F)(F)F)C(=O)N/C=N/O)OCC(F)(F)F 2B-065 CO/N=C/NC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 2B-066 C1CN(NC1=O)C(=O)CSC(=S)N2CCOCC2 2B-072 c1cc(c(cc1OCC(F)(F)F)c2[nH]ncn2)OCC(F)(F)F 2B-074 COC(=O)N/N=C/NC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 2B-075 c1ccc(cc1)N/N=C/NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 2B-077 CNc1c(cn[nH]1)[N+](=O)[O-] 2B-079 Cc1ccc(cc1)N/C(=C/[N+](=O)[O-])/SC 2B-083 c1ccc(cc1)NC(=O)N2CCN(CC2)C(=O)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F 2B-084 CN1C(=O)C(=CNc2ccccc2)C(=O)N(C1=O)C 2B-089 CN1C(=O)C(=CNc2ccc(cc2)Cl)C(=O)N(C1=O)C 2B-090 CN1C(=O)C(=CNc2ccc(cc2)OC)C(=O)N(C1=O)C 2B-092 CN1C(=O)C(=CNc2cccc(c2)C(F)(F)F)C(=O)N(C1=O)C 2B-093 Cc1ccc(cc1)n2c(nnc2C(F)(F)F)C[N+](=O)[O-] 2B-094 CN1C(=O)C(=CNCc2ccccc2)C(=O)N(C1=O)C 2B-096 C1CCN(C1)C(=S)SCC(=O)N2CCC(=O)N2 2B-099 CN1C(=O)C(=CNNc2ccccc2)C(=O)N(C1=O)C 2B-100 CN1C(=O)C(=CNc2ccccc2C#N)C(=O)N(C1=O)C 2B-101 CN1C(=O)C(=CNc2cccnc2)C(=O)N(C1=O)C 2B-102 C1CCN(CC1)C(=S)SCC(=O)N2CCC(=O)N2 2B-103 c1ccc(cc1)N/C=C/c2c(c(no2)c3c(cccc3Cl)Cl)C#N 2C-003 c1cc(c(c(c1)Cl)c2c(c(on2)/C=C/Nc3ccc(cc3)Cl)C#N)Cl 2C-004 c1ccc2c(c1)c(n[nH]c2=O)CNNC(=O)c3ccc(cc3)Cl 2C-005 Cn1c(nnc1C(F)(F)F)/C(=C(/N(C)C)\Cl)/[N+](=O)[O-] 2C-007 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC 2C-008 CN(C)c1nnnn1c2nccs2 2C-009 c1cc(oc1)/C=C/C(=O)c2ccc(cc2)F 2C-012 c1cc(c(cc1OCC(F)(F)F)C(=O)NN)OCC(F)(F)F 2C-013 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)[N+](=O)[O-])/OC2=O 2C-015 CSc1cccc(c1)N/C=C\2/c3ccccc3C(=O)O2 2C-016 CN(C)/C=C/c1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC 2C-019 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3)[N+](=O)[O-] 2C-021 CSc1cccc(c1)NCc2c3ccccc3c(=O)[nH]n2 2C-022 c1ccc2c(c1)/C(=C/NNC(=O)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F)/OC2=O 2C-026 COC(=O)c1c(onc1c2c(cccc2Cl)Cl)/C=C/Nc3ccccc3 2C-029 CCSC(C(=O)NNC(=S)Nc1ccccc1)SCC 2C-031 CCSC(C(=O)NNC(=S)NC)SCC 2C-032 COC(=O)c1c(onc1c2c(cccc2Cl)Cl)/C=C/Nc3ccc(cc3)Cl 2C-034 CC(=O)Nc1ccc2c(c1)CCC2 2C-035 c1ccc2c(c1)c(=O)c3cc4c(ccn(c4=O)Cc5ccco5)nc3o2 2C-037 c1c2c(cc(c1N)[N+](=O)[O-])CCC2 2C-038 c1cnccc1C(=N)N.Cl 2C-040 CCSC(C(=O)NNC(=S)Nc1ccc(cc1)Cl)SCC 2C-041 CCSC(c1nnc(n1c2ccccc2)S)SCC 2C-043 CCSC(C(=O)NNC(=S)Nc1cccc(c1)C(F)(F)F)SCC 2C-044 CCSC(Cc1nnc(n1C)S)SCC 2C-049 CNc1c(cnc(n1)c2ccncc2)[N+](=O)[O-] 2C-053 Cc1c(cnn1c2ccccc2)CC(=O)NN 2C-060 c1cc(ccc1NC=C2C(=NNC2=O)C(F)(F)F)OC(F)(F)F 2C-086 c1cc(ccc1NC=C2C=NNC2=O)OC(F)(F)F 2C-088 CC1=NNC(=O)C1=CNc2ccc(cc2)OC(F)(F)F 2C-089 COCC1=NNC(=O)C1=CNc2ccc(cc2)OC(F)(F)F 2C-092 c1ccc(cc1)C2=NNC(=O)C2=CNc3ccc(cc3)OC(F)(F)F 2C-093 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N 2C-097 COC(=O)c1c(onc1c2c(cccc2Cl)Cl)/C=C/Nc3ccc(cc3)C(=O)O 2C-098 c1cc(sc1)/C=C/c2ccnc3n2ncc3C#N 2D-001 COc1ccc(cc1)/C=C\c2ccnc3n2ncc3C#N 2D-002 c1cc(ccc1c2cnc3c(cnn3c2N)C#N)F 2D-003 c1cc(ccc1c2cnc3c(cnn3c2N)C#N)Cl 2D-004 COc1ccc(cc1)c2cnc3c(cnn3c2N)C#N 2D-005 c1cc(ccc1/C=C\c2ccnc3n2ncc3C#N)F 2D-006 c1ccc(cc1)Sc2cnc3ccccc3n2 2D-007 c1ccc2c(c1)ncc(n2)Oc3ccc(cc3)Cl 2D-008 c1ccc2c(c1)ncc(n2)Oc3ccc(cc3)F 2D-009 C(C#N)c1c(c([nH]n1)N)C#N 2D-010 CC(c1ccnc2n1ncc2C#N)Oc3ccc(cc3Cl)Cl 2D-011 c1ccc2c(c1)ncc(n2)Sc3ccc(cc3)Br 2D-012 c1ccc2c(c1)ncc(n2)Sc3cccc(c3)C(F)(F)F 2D-013 c1ccc2c(c1)ncc(n2)S(=O)(=O)c3ccc(cc3)Cl 2D-014 c1ccc(cc1)S(=O)(=O)c2cnc3ccccc3n2 2D-015 c1ccc2c(c1)ncc(n2)S(=O)(=O)c3ccc(cc3)Br 2D-016 c1ccc(cc1)Oc2cnc3ccccc3n2 2D-017 c1ccc2c(c1)ncc(n2)Oc3cccc(c3)C(F)(F)F 2D-018 c1ccc(cc1)c2nnc(o2)CC#N 2D-021 c1ccc(cc1)C(=O)NN/C(=C/C#N)/N 2D-022 c1ccc2c(c1)ncc(n2)Oc3cccc(c3)Cl 2D-023 c1ccc2c(c1)ncc(n2)S(=O)(=O)c3cccc(c3)C(F)(F)F 2D-024 c1ccc2c(c1)ncc(n2)Sc3ccccc3Cl 2D-025 Cc1cc(n(n1)CCCl)C 2D-027 c1ccc(cc1)c2ccnc3n2nc(c3C#N)CC#N 2D-029 c1ccc2c(c1)ncc(n2)S(=O)(=O)c3ccc(cc3)F 2D-032 COc1ccc(cc1)Sc2cnc3ccccc3n2 2D-033 Cc1ccc(cc1)Sc2cnc3ccccc3n2 2D-034 COc1ccc(cc1)S(=O)(=O)c2cnc3ccccc3n2 2D-039 c1ccc2c(c1)ncc(n2)Oc3ccccc3Cl 2D-040 COc1ccc(cc1)Oc2cnc3ccccc3n2 2D-041 c1ccc2c(c1)ncc(n2)Oc3ccc(cc3)[N+](=O)[O-] 2D-042 COC(=O)Cc1c(nnn1c2ccccc2C#N)C(=O)OC 2D-043 CNc1c(cnn1c2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] 2D-045 Cc1ccc(cc1)S(=O)(=O)c2cnc3ccccc3n2 2D-046 Cc1cc(cc(c1)S(=O)(=O)c2cnc3ccccc3n2)C 2D-047 Cc1ccc(cc1)Oc2cnc3ccccc3n2 2D-048 c1ccc2c(c1)ncc(n2)Oc3cccc(c3)[N+](=O)[O-] 2D-049 CNc1c(cnn1c2ccc(cc2)C(F)(F)F)[N+](=O)[O-] 2D-052 COC(=O)c1ccccc1Oc2cnc3ccccc3n2 2D-055 COC(=O)c1ccccc1Sc2cnc3ccccc3n2 2D-056 c1cc(c(cc1Cl)Cl)c2ccnc3n2ncc3C#N 2D-061 COC(=O)c1ccccc1S(=O)(=O)c2cnc3ccccc3n2 2D-062 c1ccc(cc1)S(=O)(=O)C(C[NH+]2CCOCC2)Cl.[Cl-] 2D-063 c1ccc2c(c1)ncc(n2)S 2D-065 CC(c1ccnc2n1ncc2C#N)Oc3ccc(cc3)Cl 2D-069 COC(=O)CSc1cnc2ccccc2n1 2D-070 c1ccc2c(c1)ncc(n2)SCC(=O)O 2D-071 c1cc(c(cc1Cl)Cl)c2ccnc3n2ncc3C(=O)N 2D-073 c1cc(ccc1C(=O)c2cc([nH]c2Br)C(=O)C(Cl)(Cl)Cl)Cl 2D-079 COc1ccc(cc1)NC(=O)CC#N 2D-084 CNC(=O)CSc1cnc2ccccc2n1 2D-088 CN(C)C(=O)CSc1cnc2ccccc2n1 2D-089 CC(C(=O)O)Sc1cnc2ccccc2n1 2D-093 c1cc(c(cc1NC(=O)CC#N)Cl)Cl 2D-095 CN(C)/C=N/c1c(cn[nH]1)C#N 2D-101 CNC(=O)c1cc(c([nH]1)Br)C(=O)c2ccc(cc2)Cl 2D-102 c1ccc(cc1)Nn2cnc-3nncc3c2N 2D-105 c1ccc2c(c1)ncc(n2)SCCC(=O)O 2D-111 CSc1nc2nccc(n2n1)c3ccc(c(c3)Cl)Cl 2D-119 CSc1nc2nccc(n2n1)/C=C\c3ccc(cc3)F 2D-120 COc1ccc(cc1)c2cnc3nc(nn3c2N)SC 2D-123 CSc1nc2ncc(c(n2n1)N)c3ccc(cc3)F 2D-124 CSc1nc2ncc(c(n2n1)N)c3ccc(cc3)Cl 2D-125 c1ccc(cc1)S(=O)(=O)C(CS(=O)(=O)c2ccc(cc2)Cl)Cl 2D-129 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 2D-132 Cn1c(nc(n1)NC(=O)/C=C/N(C)C)SC 2E-001 COc1ccc(cc1)c2c(c(nc(n2)c3ccccn3)N4CCOCC4)C#N 2E-002S c1ccc(c(c1)C(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 2E-005S c1cc(c(cc1OCC(F)(F)F)C(=O)NOC(=O)c2ccc(cc2Cl)Cl)OCC(F)(F)F 2E-006S c1cc(c(c(c1)F)C(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)F 2E-007S c1cc(c(cc1OCC(F)(F)F)C(=O)NOCC(=O)O)OCC(F)(F)F 2E-008S Cn1c(nc(n1)NC(=O)C/C=N\OCc2ccc(cc2Cl)Cl)SC 2E-009 Cn1c(nc(n1)NC(=O)C/C=N\OCc2c(cccc2Cl)Cl)SC 2E-010 Cn1c(nc(n1)NC(=O)C/C=N\OCc2ccc(c(c2)Cl)Cl)SC 2E-012 Cn1c(nc(n1)NC(=O)C/C=N\OCc2ccc(cc2)[N+](=O)[O-])SC 2E-013 Cc1cccc2n1c(=O)cc(n2)C(F)(F)F 2E-016S Cc1cccc2n1c(=O)c(c(n2)C)Cl 2E-017S CN1CCN(CC1)c2c(c(nc(n2)c3ccccn3)c4ccc(cc4)OC)C#N 2E-018S COC(CC(=O)N)OC 2E-020 Cn1c(nc(n1)NC(=O)C/C=N\OC)SC 2E-021 c1cc(c(cc1Cl)Cl)OCC(=S)N 2E-022 C#CCONC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 2E-023S C=CCONC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 2E-024S CC(C)Oc1c(c(nc(n1)c2ccccc2)c3ccc(cc3)OC)C#N 2E-025S CCOC(=O)CONC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 2E-026S CNc1c(c(nc(n1)c2ccccc2)c3ccc(cc3)OC)C#N 2E-030S c1ccc(cc1)OC(=O)CC(=O)O 2E-033 COC\1=CC(=O)S/C1=C\Nc2ccc(cc2)Cl 2E-034 COc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)N4CCOCC4)C#N 2E-035S CN1CCN(CC1)c2c(c(nc(n2)c3ccccc3)c4ccc(cc4)OC)C#N 2E-036S CCN(CC)c1c(c(nc(n1)c2ccccc2)c3ccc(cc3)OC)C#N 2E-037S c1cc(ccc1NC(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)OC(F)(F)F 2E-040S COC\1=CC(=O)S/C1=C\Nc2ccc(cc2Cl)Cl 2E-041 COC\1=CC(=O)S/C1=C\Nc2ccc(cc2)Oc3ccccc3 2E-043 c1cc(cc(c1)NC(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)C(F)(F)F 2E-045S c1ccc(cc1)OC(=O)C/C=N\OCc2ccc(cc2Cl)Cl 2E-046 c1cc(ccc1NC(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 2E-046S c1cc(c(cc1Cl)Cl)CONC(=O)N 2E-050 c1ccc(cc1)NC(=O)ONC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 2E-051S c1cc(ccc1S(=O)(=O)CC(=O)O)Cl 2E-054 c1cc(ccc1OC(=O)CC(=O)O)Cl 2E-055 CN(C)/C=C/S(=O)(=O)c1ccc(cc1)Cl 2E-057 CO/N=C/NC(=O)NOCc1ccc(cc1Cl)Cl 2E-058 c1cc(ccc1S(=O)(=O)C/C=N/OCc2ccc(cc2Cl)Cl)Cl 2E-059 c1cc(c(c(c1)Cl)CO/N=C/CS(=O)(=O)c2ccc(cc2)Cl)Cl 2E-061 c1cc(c(c(c1)Cl)CONC(=O)N)Cl 2E-062 c1ccnc(c1)c2nnc(n2N(S(=O)(=O)c3ccc(cc3)Cl)S(=O)(=O)c4ccc(cc4)Cl)c5ccccn5 2E-063 CN(C)/C=C/C(=O)Oc1ccc(cc1)Cl 2E-064 c1cc(c(c(c1)Cl)CO/N=C\CC(=O)Oc2ccc(cc2)Cl)Cl 2E-066 c1cc(ccc1OC(=O)C/C=N\OCc2ccc(cc2Cl)Cl)Cl 2E-067 c1cc(ccc1OC(=O)C/C=N\OCc2ccc(c(c2)Cl)Cl)Cl 2E-068 c1cc(ccc1CO/N=C\CC(=O)Oc2ccc(cc2)Cl)[N+](=O)[O-] 2E-069 c1cc(cc(c1)OCC(=S)N)C(F)(F)F 2E-070 c1cc(c(cc1Cl)Cl)OC(=O)CC(=O)O 2E-072 CN(C)/C=N/C(=O)NOCc1c(cccc1Cl)Cl 2E-073 CO/N=C/NC(=O)NOCc1c(cccc1Cl)Cl 2E-074 c1cc(c(c(c1)Cl)CONC(=O)N/C=N/OCc2ccc(cc2Cl)Cl)Cl 2E-076 CN(C)/C=C/C(=O)Oc1ccc(cc1Cl)Cl 2E-077 c1cc(c(c(c1)Cl)CO/N=C\CC(=O)Oc2ccc(cc2Cl)Cl)Cl 2E-078 c1ccc(cc1)N/C=C/C(=O)Oc2ccc(cc2Cl)Cl 2E-079 CN(C)/C=C(\C=N\OCc1c(cccc1Cl)Cl)/S(=O)(=O)c2ccc(cc2)Cl 2E-080 CO/N=C\C(/C=N/OCc1ccc(cc1Cl)Cl)S(=O)(=O)c2ccc(cc2)Cl 2E-082 c1cc[n+](c(c1)SCC(=O)O)[O-] 2E-083 COc1ccc(cc1)c2c(c(nc(n2)c3ccncc3)NCC=C)C#N 2E-103S COc1ccc(cc1)c2c(c(nc(n2)c3ccncc3)NCc4ccccc4)C#N 2E-104S COc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)Sc4ccccc4)C#N 2E-109S COc1ccc(cc1)c2c(c(nc(n2)c3ccccc3)SCc4ccc(cc4)Cl)C#N 2E-110S CCNC(=O)ONC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 2E-113S c1cc(c(cc1OCC(F)(F)F)C(=O)NOC(=O)NC2CCCCC2)OCC(F)(F)F 2E-114S c1cc(c(cc1OCC(F)(F)F)C(=O)NCC[NH3+])OCC(F)(F)F.[Cl-] 2E-115S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)OCC(F)(F)F 2E-116S c1ccc(cc1)C(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 2E-118S c1cc(ccc1S(=O)(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 2E-119S c1ccnc(c1)c2nc(c(c(n2)N3CCOCC3)C#N)c4cccc(c4)C(F)(F)F 2E-124S c1ccc(cc1)c2cn3ccsc3n2 2E-126S c1ccc(cc1)c2c(n3ccsc3n2)C=O 2E-127S CNc1c(c(nc(n1)c2ccncc2)c3cccc(c3)C(F)(F)F)C#N 2E-132S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl 2E-133S CO/N=C/c1c(nc2n1ccs2)c3ccccc3 2E-134S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/O 2E-135S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4c(cccc4Cl)Cl 2E-141S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4ccc(c(c4)Cl)Cl 2E-142S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4ccc(cc4)[N+](=O)[O-] 2E-143S c1ccc(cc1)c2cn3c(n2)SCC3 2E-144S c1ccc(cc1)c2c(n3ccsc3n2)C#N 2E-146S COC(=O)c1ccccc1Sc2c(n3ccsc3n2)C#N 2E-147S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)c4ccccc4 2E-148S COc1ccc(cc1)C(=O)O/N=C/c2c(nc3n2ccs3)c4ccccc4 2E-149S CO/N=C/c1c(nc2n1CCS2)c3ccccc3 2E-150S c1ccc(cc1)c2c(n3c(n2)SCC3)/C=N/OCc4c(cccc4Cl)Cl 2E-151S COC(=O)c1c(cccn1)O 2E-901 CN(C)/C=C(/C(=O)OC)\NC(=O)c1ccccc1 2E-914 Cc1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(=O)C 2E-915 CCOC(=O)c1cc(c(=O)oc1c2ccccc2)NC(=O)c3ccccc3 2E-917 CC(=O)c1cc(c(=O)oc1/C=C/N(C)C)NC(=O)c2ccccc2 2E-918 c1ccc(c(c1)C(=O)Oc2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl 2F-001 c1ccc(cc1)n2cnc(n2)OCC(=O)NN 2F-004 c1cc(ccc1NC(=O)Nc2cc(c[nH]2)C(=O)c3ccc(cc3Cl)Cl)Cl 2F-005 CNC(=O)/C=C/c1cc(cn1C)C(=O)c2ccc(cc2Cl)Cl 2F-006 Cc1c(c(nc(c1C#N)O)C)Cc2ccc(cc2Cl)Cl 2F-007 c1ccc(cc1)n2cnc(n2)Oc3c(cc(cn3)C(F)(F)F)Cl 2F-012 Cc1cc(nc(c1Cc2ccc(cc2Cl)Cl)C)O 2F-013 c1ccc(cc1)n2cnc(n2)OCC(=O)NNC(=N)Cn3cncn3 2F-015 COC(CC(=O)NNC(=N)Cn1cncn1)OC 2F-016 c1ccc(cc1)n2cnc(n2)OCc3nc([nH]n3)Cn4cncn4 2F-018 c1ccc(cc1)n2cnc(n2)OCC(=O)NNC(=N)COc3cccc(c3)C(F)(F)F 2F-020 c1ccc(cc1)n2cnc(n2)OCc3nc([nH]n3)c4cccnc4 2F-021 c1ccc(cc1)n2cnc(n2)OCc3nc([nH]n3)COc4cccc(c4)C(F)(F)F 2F-022 c1cc(c(cc1Cl)Cl)OC/C(=N\NC(=O)CC#N)/N 2F-023 c1cc(c(cc1Cl)Cl)OCc2nc([nH]n2)CC#N 2F-024 Cn1cccc1C(=O)NN 2F-025 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/c2[nH]nc(n2)COc3ccc(cc3Cl)Cl 2F-027 c1cc(c(cc1Cl)Cl)OC/C(=N/Nc2c(cc(cn2)C(F)(F)F)Cl)/N 2F-028 COc1ccc(cc1)N/N=C(\C(=O)CC(=O)OC)/C(=O)OC 2F-029 CCOC(=O)CC(=N)NNC(=O)c1cccn1C 2F-030 c1cc(cc(c1)n2c(=O)cc(c(n2)C(=O)N)O)C(F)(F)F 2F-031 c1cc(c(cc1Cl)Cl)OCc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl 2F-032 COC(=O)c1c(cc(=O)n(n1)c2cccc(c2)C(F)(F)F)Cl 2F-033 c1cc(ccc1SC/C(=N/NC(=O)c2ccncc2)/N)Cl 2F-035 c1cc(ccc1SC/C(=N/NC(=O)CC#N)/N)Cl 2F-036 Cn1cc(cc1C(=O)NN)C(=O)c2ccc(cc2Cl)Cl 2F-037 c1cc(cc(c1)n2c(=O)cc(c(n2)C#N)Cl)C(F)(F)F 2F-038 Cc1c(c(ns1)SCC(=O)NN)C#N 2F-039 c1cc(ccc1SCc2nc([nH]n2)c3ccncc3)Cl 2F-040 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)O 2F-041 c1ccc2c(c1)c(c[nH]2)c3ccc(nn3)Cl 2F-042 Cc1c(c(ns1)SCC(=O)NNC(=N)COc2ccc(cc2Cl)Cl)C#N 2F-043 Cn1cc(cc1C(=O)NNC(=N)COc2ccc(cc2Cl)Cl)C(=O)c3ccc(cc3Cl)Cl 2F-044 Cn1cc(cc1c2nnc(o2)COc3ccc(cc3Cl)Cl)C(=O)c4ccc(cc4Cl)Cl 2F-045 Cc1c(c(ns1)SCc2nc([nH]n2)COc3ccc(cc3Cl)Cl)C#N 2F-046 c1cc(ccc1SCc2nc([nH]n2)CC#N)Cl 2F-047 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=N)COc3cccc(c3)C(F)(F)F 2F-048 Cc1c(c(no1)c2ccccc2Cl)c3nc([nH]n3)COc4cccc(c4)C(F)(F)F 2F-049 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)O 2F-050 c1cc(ccc1C(=O)N/N=C(/CSc2ccc(cc2)Cl)\N)Cl 2F-051 c1cc(ccc1C(=O)N/N=C(/COc2ccc(cc2Cl)Cl)\N)Cl 2F-052 Cn1c(nnc1COc2ccc(cc2Cl)Cl)C[N+](=O)[O-] 2F-053 Cc1ccc(cc1)Sc2cc(=O)n(nc2C(=O)OC)c3cccc(c3)C(F)(F)F 2F-054 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)C(=O)c2ccccc2C(=O)O 2F-055 c1cc(ccc1c2nnc(o2)COc3ccc(cc3Cl)Cl)Cl 2F-056 CCOC(=O)/C=C/c1ccc(cc1)/C=C/c2c(c(no2)C)[N+](=O)[O-] 2F-057 COc1ccc(cc1)n2c(=O)cc(c(n2)C#N)Cl 2F-058 c1cc(ccc1c2[nH]nc(n2)CSc3ccc(cc3)Cl)Cl 2F-059 COC(=O)CSc1cc(=O)n(nc1C(=O)OC)c2cccc(c2)C(F)(F)F 2F-060 COC(=O)c1c(cc(=O)n(n1)c2cccc(c2)C(F)(F)F)Sc3ccccn3 2F-063 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)Cl 2F-064 Cc1ccc(cc1)Sc2cc(=O)n(nc2C(=O)OC)c3ccc(cc3)OC 2F-065 c1cc(c(cc1Cl)Cl)SC/C(=N/Nc2c(cc(cn2)C(F)(F)F)Cl)/N 2F-066 CN(C)/C=C(/c1nnc(n1c2ccc(cc2)Cl)COc3cccc(c3)C(F)(F)F)\[N+](=O)[O-] 2F-068 COC(=O)c1c(c2c(s1)cc(=O)n(n2)c3cccc(c3)C(F)(F)F)O 2F-069 c1cc(c(cc1Cl)Cl)SCc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl 2F-070 c1ccc2c(c1)cc([nH]2)c3ccc(nn3)NN 2F-071 c1ccc(cc1)SC/C(=N/NC(=O)c2ccncc2)/N 2F-072 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)Sc3ccccn3 2F-073 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)SCC(=O)OC 2F-074 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)C(=O)/C=C/C(=O)O 2F-075 COC(=O)c1c(c2c(s1)cc(=O)n(n2)c3cccc(c3)C(F)(F)F)N 2F-077 COc1ccc(cc1)n2c(=O)cc3c(n2)c(c(s3)C(=O)OC)O 2F-078 CCOC(=O)C(=O)Nc1ccc(cc1)F 2F-079 CCOC(=O)C(=O)Nc1ccc(cc1)OC 2F-080 CCOC(=O)C(=O)Nc1cccc(c1)C(F)(F)F 2F-081 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)Oc3ccccc3 2F-082 c1cc(ccc1NC(=O)C(=O)NN)F 2F-083 COc1ccc(cc1)NC(=O)C(=O)NN 2F-084 c1cc(cc(c1)n2c(=O)cc3c(n2)c(n[nH]3)N)C(F)(F)F 2F-086 c1cc(cc(c1)NC(=O)C(=O)NN)C(F)(F)F 2F-087 c1ccc(cc1)n2cnc(n2)OCC(=N)[NH3+].[Cl-] 2F-088 COc1ccc(cc1)NC(=O)C(=O)NN/C=C\2/c3ccccc3C(=O)O2 2F-090 Cc1ccc(cc1)Sc2cc(=O)n(nc2C(=O)NN)c3ccc(cc3)OC 2F-091 COc1ccc(cc1)n2c(=O)cc3c(n2)c(c(s3)C(=O)OC)N 2F-092 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)O 2F-093 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)Oc3cccc(c3)C(F)(F)F 2F-097 COc1ccc(cc1)n2c(=O)cc3c(n2)c(n[nH]3)N 2F-098 COC(=O)c1c(cc(=O)n(n1)c2cccc(c2)C(F)(F)F)Oc3ccccc3 2F-099 c1ccc2c(c1)c(=O)[nH]c(n2)Cc3cccc(c3)C(F)(F)F 2F-301S Cc1ccc(cc1)CNC2=Nc3ccccc3CS2 2F-302S c1ccc2c(c1)CSC(=N2)NCc3ccccn3 2F-303S c1ccc2c(c1)CSC(=N2)Oc3ccc(cc3)Cl 2F-304S c1ccc2c(c1)CSC(=N2)NCc3ccncc3 2F-306S c1ccc2c(c1)c(=O)[nH]c(n2)Cc3cccc(c3)Cl 2F-310S c1ccc(c(c1)Cc2[nH]c(=O)c3ccccc3n2)Cl 2F-311S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)OC 2F-312S c1cc(ccc1CO/N=C/c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)Cl 2F-313S COc1ccccc1C/N=C/c2c(nc3n2ccs3)Cl 2F-314S c1ccc2c(c1)CSC(=N2)NCc3cccs3 2F-316S COc1cccc(c1)CNC2=Nc3ccccc3CS2 2F-317S COC(=O)c1ccc(nc1)n2cccn2 2F-318S COC(=O)c1ccc(nc1)Cl 2F-320S COC(=O)c1ccc(nc1)n2ccnc2 2F-321S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C4=Nc5ccccc5CS4 2F-323S COc1ccccc1CNC2=Nc3ccccc3CS2 2F-324S c1ccc2c(c1)c(nc(n2)Cc3cccc(c3)C(F)(F)F)OCc4c(cccc4Cl)Cl 2F-325S c1ccc2c(c1)c(nc(n2)Cc3cccc(c3)Cl)OCc4c(cccc4Cl)Cl 2F-326S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2cccc(c2)C(F)(F)F 2F-328S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(cc2)[N+](=O)[O-] 2F-329S c1cnn(c1)c2ccc(cn2)C(=O)O 2F-330S c1cc(ncc1C(=O)O)n2cncn2 2F-331S c1cc(ncc1C(=O)O)n2ccnc2 2F-337S C=CCNC1=Nc2ccccc2CS1 2F-339S COc1c2ccccc2nc(n1)Cc3ccc(cc3)Cl 2F-342S c1ccc2c(c1)c(nc(n2)Cc3cccc(c3)Cl)OCc4ccc(cc4Cl)Cl 2F-343S c1ccc2c(c1)CSC(=N2)N3CCN(CC3)c4ccccn4 2F-344S c1cc(cc(c1)NC(=O)c2ccc(nc2)n3cccn3)C(F)(F)F 2F-347S c1cnn(c1)c2ccc(cn2)C(=O)Nc3ccc(cc3)OC(F)(F)F 2F-348S COc1ccc(cc1)NC(=O)c2ccc(nc2)n3cccn3 2F-349S c1cnn(c1)c2ccc(cn2)C(=O)Nc3ccc(cc3F)F 2F-350S COc1ccc(c(c1)NC(=O)c2ccc(nc2)n3cccn3)OC 2F-351S c1ccc(cc1)Cc2nc3ccccc3c(n2)OCc4c(cccc4Cl)Cl 2F-352S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(cc2F)F 2F-354S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(cc2)OC(F)(F)F 2F-355S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(cc2)Cl 2F-356S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F 2F-357S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2cccc(c2Cl)Cl 2F-358S COC(=O)c1ccc(nc1)n2cnc3c2cccc3 2F-359S Cc1ccc(cc1)NC(=O)c2ccc(nc2)n3cccn3 2F-360S COc1cccc(c1)NC(=O)c2ccc(nc2)n3cccn3 2F-361S COc1ccccc1NC(=O)c2ccc(nc2)n3cccn3 2F-362S CCOc1ccc(cc1)NC(=O)c2ccc(nc2)n3cccn3 2F-363S COc1ccc(cc1OC)NC(=O)c2ccc(nc2)n3cccn3 2F-364S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccccc2Cl 2F-367S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2cccc(c2)Cl 2F-368S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(cc2)F 2F-369S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(c(c2)Cl)Cl 2F-370S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2cc(ccc2Cl)C(F)(F)F 2F-371S c1ccc2c(c1)ncn2c3ccc(cn3)C(=O)O 2F-373S Cn1c(c(c(n1)C(F)(F)F)C(=O)O)Cl 2F-374S Cc1ccc(cc1)NC(=O)c2cccnc2Nc3ccc(cc3)S(=O)(=O)N.Cl 2F-375S c1cc(ccc1NC(=O)c2ccc(nc2)n3cncn3)OC(F)(F)F 2F-376S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(cc2)C(F)(F)F 2F-378S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2cc(ccc2Cl)Cl 2F-379S CN(C)S(=O)(=O)Oc1ccc(cc1)C(=O)Nc2ccc(cc2)OC 2F-380S Cn1c(c(c(n1)C(F)(F)F)C=O)Sc2ccc(cc2)Cl 2F-381S Cc1ccc(cc1)NC(=O)c2ccc(cc2)OS(=O)(=O)N(C)C 2F-382S CN(C)S(=O)(=O)Oc1ccccc1C(=O)OC 2F-383S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccc(cc2)F 2F-384S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccc(cc2F)F 2F-385S COc1ccc(c(c1)OC)NC(=O)c2ccc(nc2)n3cccn3 2F-386S c1cnn(c1)c2ccc(cn2)C(=O)NCc3ccc(cc3)Cl 2F-387S c1cc(cc(c1)C(F)(F)F)CNC(=O)c2ccc(nc2)n3cccn3 2F-388S c1cnn(c1)c2ccc(cn2)C(=O)N3CCOCC3 2F-389S CN1CCN(CC1)C(=O)c2ccc(nc2)n3cccn3 2F-390S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl)Cl 2F-392S Cn1c(c(c(n1)C(F)(F)F)C=O)Sc2ccccc2 2F-393S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(cc2)Cl)Sc3ccc(cc3)Cl 2F-394S CNC(=O)c1ccc(nc1)n2cccn2 2F-395S CN(C)C(=O)c1ccc(nc1)n2cccn2 2F-396S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccc(cc2)OC(F)(F)F 2F-397S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccccc2Cl 2F-398S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2cccc(c2)Cl 2F-399S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2c(cccc2Cl)Cl)Sc3ccc(cc3)Cl 2F-400S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl)Sc3ccc(cc3)Cl 2F-401S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Cl 2F-402S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2cccc(c2)C(F)(F)F)Cl 2F-403S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC(F)(F)F)Cl 2F-404S Cc1ccc(cc1C)NC(=O)c2c(nn(c2Cl)C)C(F)(F)F 2F-405S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2cc(ccc2OC)OC)Cl 2F-406S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(c(c2)Cl)Cl)Cl 2F-407S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2cccc(c2)Cl)Cl 2F-408S Cn1c(c(c(n1)C(F)(F)F)/C=N/O)Sc2ccc(cc2)Cl 2F-409S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccc(cc2)Cl 2F-410S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccc(cc2)OC 2F-411S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)OC 2F-412S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccc(c(c2)Cl)Cl 2F-413S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2cccc(c2)C(F)(F)F 2F-414S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2ccc(cc2)[N+](=O)[O-] 2F-415S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2Cl)Sc3ccc(cc3)Cl 2F-416S Cn1c(c(c(n1)C(F)(F)F)C=O)SCc2ccccc2Cl 2F-417S CNC(=O)c1c(nn(c1Cl)C)C(F)(F)F 2F-418S Cn1c(c(c(n1)C(F)(F)F)C(=O)N(C)C)Cl 2F-419S Cn1c(c(c(n1)C(F)(F)F)C(=O)NCC=C)Cl 2F-420S Cn1c(c(c(n1)C(F)(F)F)C(=O)NCc2ccccc2)Cl 2F-421S Cn1c(c(c(n1)C(F)(F)F)C(=O)NCc2ccc(cc2)Cl)Cl 2F-422S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccc(cc2)Cl 2F-423S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2cccc(c2)Cl 2F-424S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccccc2Cl 2F-425S CN(C)S(=O)(=O)Oc1ccccc1C(=O)Nc2cc(ccc2Cl)C(F)(F)F 2F-426S c1ccc2c(c1)C(C(=O)N(C2=O)OCc3ccc(cc3Cl)Cl)/C=N\OCc4ccc(cc4Cl)Cl 2F-900 c1ccc2c(c1)/C(=C/Nc3cc(ccc3Cl)C(F)(F)F)/C(=O)N(C2=O)OCc4ccc(cc4Cl)Cl 2F-902 COC(=O)c1c(ccs1)NC(=O)CNC(=O)c2ccccc2 2F-903 CCOC(=O)c1cc([nH]c1N2CCCC2)c3ccccc3 2F-905 COc1ccc(cc1)C(=O)NCC(=O)NCCO 2F-906 c1ccc(cc1)/C=C\2/c3ccccc3C(=O)N(C2=O)OCc4ccc(cc4Cl)Cl 2F-907 CCOC(=O)/C=C(\N)/N1CCN(CC1)c2ccccc2 2F-909 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc4c(oc3=O)CCCC4=O 2F-910 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3ccccc3)c4ccccc4 2F-912 CCOC(=O)NC(=O)/C(=C\NN1CCOCC1)/C#N 2F-913 Cc1ccc(cc1)S(=O)(=O)OCCn2cc(c(=O)[nH]c2=O)C#N 2F-914 c1c(c(=O)[nH]c(=O)n1N2CCOCC2)C#N 2F-915 c1c(c(=O)nc2n1CCO2)C#N 2F-916 COc1ccc(cc1)C(=O)NCC(=O)NCCOC(=O)c2ccccc2F 2F-917 CCOC(=O)/C=C(\N)/N1CCN(CC1)c2ccc(cc2)OC 2F-918 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3ccc(cc3)OC)c4ccc(cc4Cl)Cl 2F-919 CCOC(=O)c1cc(c(=O)[nH]c1N2CCCCC2)C(=O)OCC 2F-920 CCOC(=O)NC(=O)/C(=C\NN1CCCCC1)/C(=O)C 2F-921 CCOC(=O)c1cc(c(=O)[nH]c1N2CCN(CC2)c3ccc(cc3)OC)C(=O)OCC 2F-922 CC(=O)c1cn(c(=O)[nH]c1=O)N2CCCCC2 2F-923 CCOC(=O)/C(=C/C(=C(/N)\N1CCN(CC1)c2ccc(cc2)OC)/C(=O)OCC)/C#N 2F-924 CCOC(=O)NC(=O)/C(=C\NN1CCOCC1)/C(=O)C 2F-925 CC(=O)c1cn(c(=O)[nH]c1=O)N2CCOCC2 2F-926 CCOC(=N)CC#N 2F-928 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3ccccc3)c4ccc(cc4)Cl 2F-929 CCOC(=O)/C(=C/C(=C(/N)\N1CCN(CC1)c2ccccc2)/C(=O)OCC)/C#N 2F-930 COc1ccc(cc1)N2CCN(CC2)C(=N)CC#N 2F-932 CCOC(=O)c1cc(c(nc1C)C)C(=O)OCC 2F-933 CCOC(=O)/C(=C\C(=C(\N)/N1CCN(CC1)c2ccc(cc2)OC)\C#N)/C#N 2F-935 COc1ccc(cc1)N2CCN(CC2)c3c(cc([nH]3)c4ccc(cc4)Cl)C#N 2F-936 CCOC(=O)NC(=O)c1cnn(c1C)c2ccccc2 2F-937 CCOC(=O)c1cc(c([nH]c1=O)N2CCN(CC2)c3ccc(cc3)OC)C#N 2F-938 COc1ccc(cc1)N2CCN(CC2)C(=O)CC3(C4CC5CC(C4)CC3C5)c6ccccc6 2F-940 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)N5CCN(CC5)c6ccc(cc6)Cl 2F-941 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)NCCO 2F-942 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)NCCOC(=O)c5cccs5 2F-943 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)NCCOC(=O)c5ccc(cc5)[N+](=O)[O-] 2F-944 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)NCCOC(=O)c5ccc(cc5Cl)Cl 2F-945 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)NCCOC(=O)c5cccc(c5)C(F)(F)F 2F-946 CCOc1c(cc(c(n1)O)C(=O)OCC)C#N 2F-947 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)O 2F-950 c1ccc(cc1)N2CCN(CC2)C(=N)CC#N 2F-952 CN(C)/C=N/C(=O)CC1(C2CC3CC(C2)CC1C3)c4ccccc4 2F-953 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)N/C=N/OCc5ccc(cc5Cl)Cl 2F-954 CCOC(=O)c1c(c[nH]c1N)c2ccccc2 2F-958 c1ccc(cc1)C[N+]23CCCCC2CC(O3)CO.[Br-] 2F-959 COc1ccc(cc1)N2CCN(CC2)CC(=O)c3ccccc3 2F-960 CCOC(=O)c1cc2c(ccn(c2=O)CCO)nc1C 2F-961 COc1ccc(cc1)N2CCN(CC2)C/C(=N\OCc3ccc(cc3)Cl)/c4ccccc4 2F-962 COc1ccc(cc1)N2CCN(CC2)C/C(=N\O)/c3ccccc3 2F-964 CCOC(=O)c1cc(c(=O)[nH]c1N2CCCC2)C(=O)OCC 2F-980 Cc1ccc(cc1)N/N=C(/C(=O)Nc2ccc(cc2)Cl)\N=N\c3ccc(cc3)C 2G-003 c1cc(ccc1/C=C\2/C(=C(C(=O)O2)c3c(cc(cn3)C(F)(F)F)Cl)c4ccc(cc4)Cl)[N+](=O)[O-] 2G-004 CC(c1cc(no1)c2c(cc(cn2)C(F)(F)F)Cl)O 2G-005 CONCCc1c(cc(cn1)C(F)(F)F)Cl 2G-006 c1cc(ccc1Sc2cc(cnc2C#N)C(F)(F)F)Cl 2G-007 COC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)N 2G-009 CCOC(=O)C(c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)C(=O)OCC 2G-010 c1cc(ccc1Oc2cc(cnc2C#N)C(F)(F)F)Cl 2G-013 CC(=O)c1cc(no1)c2c(cc(cn2)C(F)(F)F)Cl 2G-014 C/C(=N\Oc1c(cc(cn1)C(F)(F)F)Cl)/c2ccc(o2)c3ccc(cc3)Cl 2G-015 CC(C)(c1c(cn[nH]1)C#N)n2cncn2 2G-016 Cc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)Cl 2G-017 c1c(cnc(c1Cl)n2cc(cn2)C(=O)N)C(F)(F)F 2G-018 c1c(cnc(c1Cl)CONC(=O)N)C(F)(F)F 2G-019 CN(C)/C=N/C(=O)NOCc1c(cc(cn1)C(F)(F)F)Cl 2G-020 CN(C)/C=C(\C#N)/c1cccc(c1)C(F)(F)F 2G-022 CO/N=C\NC(=O)NOCc1c(cc(cn1)C(F)(F)F)Cl 2G-024 c1ccc(cc1)/C(=C/O)/C#N 2G-025 CN(C)/C=C/C(=O)c1cc(no1)c2c(cc(cn2)C(F)(F)F)Cl 2G-027 c1cn[nH]c1c2cc(no2)c3c(cc(cn3)C(F)(F)F)Cl 2G-030 C/C(=N/O)/c1cc(no1)c2c(cc(cn2)C(F)(F)F)Cl 2G-031 c1cc(c(cc1Cl)Cl)CO/N=C\NC(=O)NOCc2c(cc(cn2)C(F)(F)F)Cl 2G-032 c1cc(ccc1CSc2cc(cnc2C#N)C(F)(F)F)Cl 2G-034 c1c(cnc(c1Cl)n2cc(cn2)C(=S)N)C(F)(F)F 2G-035 c1c(cnc(c1Cl)C(C(=O)N)C(=O)N)C(F)(F)F 2G-036 c1cc(ccc1CS(=O)(=O)c2cc(cnc2C#N)C(F)(F)F)Cl 2G-037 Cc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)Nc2ccccc2 2G-038 c1c(cnc(c1Cl)C(C#N)C(=O)N)C(F)(F)F 2G-039 c1cc(ncc1C(F)(F)F)Sc2cc(cnc2C#N)C(F)(F)F 2G-042 c1cc(ccc1c2ccc(o2)/C=N/O)Cl 2G-046 CN(C)C(=O)Nc1cc2c(s1)cc(cn2)C(F)(F)F 2G-047 C/C(=N\OCc1c(cccc1Cl)Cl)/c2cc(no2)c3c(cc(cn3)C(F)(F)F)Cl 2G-048 CN(C)/C=C(\c1ccc(cc1)Cl)/S(=O)(=O)c2cc(cnc2C#N)C(F)(F)F 2G-049 c1cc(cc(c1)Sc2cc(cnc2C#N)C(F)(F)F)C(F)(F)F 2G-050 c1cc(ccc1NC(=O)n2ccc(n2)/C=C/c3c(cc(cn3)C(F)(F)F)Cl)Cl 2G-051 c1ccc(c(c1)N)Sc2cc(cnc2C#N)C(F)(F)F 2G-052 c1cc(ccc1C(=O)n2ccc(n2)c3cc(no3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 2G-053 CN(C)C(=O)c1csc(n1)c2cccnc2 2G-302S CCOC(=O)c1c(nc(s1)c2ccccn2)C 2G-303S c1cc(c(cc1C(=O)O)[N+](=O)[O-])n2cncn2 2G-304S c1cnccc1c2nc(cs2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 2G-305S COC(=O)c1ccc(cc1)c2nc(cs2)c3ccccc3Cl 2G-306S Cc1c(sc(n1)c2ccccn2)C(=O)O 2G-307S c1ccc2c(c1)N(c3c(cccn3)S2)Cc4c(cccc4Cl)F 2G-308S c1cc2c(cc1[N+](=O)[O-])onc2C(=O)O 2G-311S c1cc(ccc1NC(=O)c2c3ccc(cc3on2)[N+](=O)[O-])Cl 2G-312S c1ccc(c(c1)c2csc(n2)c3ccc(cc3)C(=O)O)Cl 2G-313S Cc1c(sc(n1)c2ccncc2)C(=O)Nc3cccc(c3)C(F)(F)F 2G-318S Cc1c(sc(n1)c2ccncc2)C(=O)Nc3ccc(cc3)OC(F)(F)F 2G-319S c1ccc(c(c1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4)Cl)Cl 2G-322S c1ccc(c(c1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4F)F)Cl 2G-323S c1ccc(c(c1)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4Cl)Cl)Cl 2G-324S c1cc(cc(c1)C(F)(F)F)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4)F 2G-326S c1cc(cc(c1)NC(=O)c2csc(n2)c3cccnc3)C(F)(F)F 2G-327S c1cc(cc(c1)C(F)(F)F)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4F)F 2G-328S CNC(=O)c1ccc(cc1)c2nc(cs2)c3cccc(c3)C(F)(F)F 2G-329S C=CCNC(=O)c1ccc(cc1)c2nc(cs2)c3cccc(c3)C(F)(F)F 2G-330S c1cc(cc(c1)C(F)(F)F)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(c(c4)Cl)Cl 2G-331S c1cnn(c1)c2ccc(cc2[N+](=O)[O-])C(=O)Nc3ccc(cc3)Cl 2G-333S C/N=C(\c1ccccc1)/Nc2cccnc2 2G-335S CC(C)/N=C(\c1ccccc1)/Nc2cccnc2 2G-337S c1ccc(cc1)NC(=O)c2ccc(cc2)c3nc(cs3)c4cccc(c4)C(F)(F)F 2G-338S c1cc(cc(c1)C(F)(F)F)c2csc(n2)c3ccc(cc3)C(=O)Nc4ccc(cc4)Br 2G-339S c1cnn(c1)c2ccc(cc2[N+](=O)[O-])C(=O)Nc3ccc(cc3F)F 2G-340S CN(C)CCCNC(=O)c1ccc(cc1)c2nc(cs2)c3cccc(c3)C(F)(F)F 2G-341S c1cc(cc(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3)C(F)(F)F 2G-342S c1cnn(c1)c2ccc(cc2[N+](=O)[O-])C(=O)Nc3ccc(cc3)F 2G-343S c1cc(c(cc1/C=N/O)[N+](=O)[O-])Cl 2G-344S CC(C)/N=C(\c1cccc(c1)C(F)(F)F)/Nc2cccnc2 2G-345S c1cc(c(nc1)Sc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3F)F 2G-347S COc1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 2G-348S COc1cccc(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 2G-349S c1cc(c(cc1C(=O)N)[N+](=O)[O-])n2cncn2 2G-353S Cc1c(sc(n1)c2ccccn2)C(=O)Nc3ccccc3 2G-354S Cc1c(sc(n1)c2ccccn2)C(=O)Nc3ccc(cc3)F 2G-355S CNC(=O)c1ccc(c(c1)[N+](=O)[O-])n2cccn2 2G-357S c1cc(ccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3)F 2G-360S Cc1c(sc(n1)c2ccccn2)C(=O)Nc3ccc(cc3F)F 2G-361S Cc1c(sc(n1)c2ccccn2)C(=O)Nc3cccc(c3)C(F)(F)F 2G-362S Cc1c(sc(n1)c2ccccn2)C(=O)Nc3cc(cc(c3)Cl)Cl 2G-367S Cc1c(sc(n1)c2ccccn2)C(=O)Nc3ccc(c(c3)Cl)Cl 2G-368S Cc1c(sc(n1)c2ccccn2)C(=O)NCC=C 2G-369S Cc1c(sc(n1)c2ccccn2)C(=O)NC 2G-370S Cc1c(sc(n1)c2ccccn2)C(=O)N 2G-371S c1cc(cc(c1)Cl)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 2G-372S c1ccc(c(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3)Cl 2G-373S CN(C)c1nc(cc(n1)O)O 2G-377S CN(C)c1nc(cc(n1)Cl)Cl 2G-378S CNC(=O)c1c2ccc(cc2on1)[N+](=O)[O-] 2G-379S c1cc(ccc1S(=O)(=O)c2cnns2)Cl 2G-382S c1cc2c(cc1[N+](=O)[O-])onc2C(=O)N 2G-383S CCOC(=O)c1c(nc(s1)c2ccc(cc2)C)C 2G-385S Cc1ccc(cc1)c2nc(c(s2)C(=O)O)C 2G-391S CCOC(=O)c1c(nc(s1)c2ccccc2Cl)C 2G-392S CN(C)c1nc(cc(n1)Cl)OC 2G-393S CN(C)c1nc(c(c(n1)Cl)/C=N/O)OC 2G-395S CCOC(=O)c1csc(n1)c2ccc(cc2)C 2G-397S Cc1c(snn1)Sc2ccccc2 2G-401S Cc1ccc(cc1)c2nc(cs2)C(=O)O 2G-402S CCOC(=O)c1csc(n1)c2ccc(cc2)[N+](=O)[O-] 2G-403S CCOC(=O)c1c(nc(s1)c2ccc(cc2)[N+](=O)[O-])C 2G-404S CN(C)C(=O)c1c2ccc(cc2on1)[N+](=O)[O-] 2G-405S Cc1c(snn1)Sc2cccc(c2)C(F)(F)F 2G-406S c1cc(ccc1Sc2cnns2)Br 2G-407S c1cc(ccc1S(=O)(=O)c2cnns2)Br 2G-409S CCOCCOC(=O)c1ccc(nc1)n2cncn2 2G-411S COc1ccccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3ccnc3 2G-412S c1cc(cc(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3ccnc3)C(F)(F)F 2G-414S c1ccc(cc1)S(=O)(=O)c2cnns2 2G-416S Cc1c(snn1)S(=O)c2cccc(c2)C(F)(F)F 2G-417S c1cc(ccc1S(=O)c2cnns2)Br 2G-419S Cc1ccc(cc1)c2nc(c(s2)C(=O)Nc3ccc(cc3)Cl)C 2G-421S Cc1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc(cc3)F 2G-422S Cc1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc(cc3F)F 2G-423S CCOC(=O)c1c(nc(s1)c2ccc(c(c2)OC)OC)C 2G-424S CCOC(=O)c1csc(n1)c2ccc(c(c2)OC)OC 2G-425S COC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)Cl 2G-429S COC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(c(c3)Cl)Cl 2G-430S Cc1ccc(cc1)c2nc(cs2)C(=O)Nc3cccc(c3)C(F)(F)F 2G-432S Cc1ccc(cc1)c2nc(cs2)C(=O)NC 2G-433S CC(C)(C)CCC(=C)c1ccc(cc1)C2C=CC=C2 2G-435S c1cc(ccc1C(=O)NCC(=O)NNC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 2G-900 CCOC(=O)/C=C(\[NH3+])/Nc1ccc(cc1)OC(F)(F)F.[Cl-] 2G-903 c1ccc(cc1)n2c(nnc2S)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 2G-904 Cc1ccc(cc1)S(=O)(=O)Nc2c(cc(cn2)C(F)(F)F)Cl 2G-906 CN(C)/C=C/C(=O)c1cc(ccc1O)S(=O)(=O)N2CCCCC2 2G-907 c1cc(ccc1CN(Cc2ccc(cc2)Cl)O)Cl 2G-909 CCOC(=O)/C(=N/OCc1ccccc1)/C(=O)C 2G-911 c1ccc(cc1)N/N=C/C=O 2G-912 CCOC(=O)/C(=N\OCc1ccc(cc1Cl)Cl)/C(=O)C 2G-913 CN(C)/C=C/C(=O)c1cc(ccc1O)S(=O)(=O)N2CCOCC2 2G-915 c1ccc(cc1)n2c(=O)c(ccn2)C(=O)O 2G-916 CCOC(=O)/C=C(/N)\NNC(=O)c1ccco1 2G-917 COC(=O)c1ccnn(c1=O)c2ccccc2 2G-920 c1ccc(cc1)n2c(=O)c(ccn2)C(=O)NN 2G-921 COC(=O)CS(=O)(=O)c1c(cc(cn1)C(F)(F)F)Cl 2G-923 c1ccc2c(c1)C(=O)N(C2=O)OCC#N 2G-924 c1cc(ccc1NC(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 2G-926 C=CCOc1ccccc1C=O 2G-928 c1ccc(cc1)C(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 2G-930 Cc1ccc(cc1)n2c(cc3c2CC/C(=C\N(C)C)/C3=O)c4ccccc4 2G-932 C/C(=C\C(=O)Nc1c(cc(cn1)C(F)(F)F)Cl)/N2CCCC2 2G-934 CCOC(=O)C1C(C2CCCCN2O1)(C(F)(F)F)O 2G-935 CCOC(=O)c1c(c(on1)C)C(=O)Nc2c(cc(cn2)C(F)(F)F)Cl 2G-937 Cc1c(c(no1)C(=O)N)C(=O)Nc2c(cc(cn2)C(F)(F)F)Cl 2G-938 Cc1c(c(no1)C(=O)NN)C(=O)Nc2c(cc(cn2)C(F)(F)F)Cl 2G-939 c1ccc(cc1)c2c[nH]cc2[N+](=O)[O-] 2G-941 C1COCCN1/C(=C/C#N)/N 2G-942 c1cc(ccc1C(=O)NCC(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 2G-943 CCOC(=O)c1c(con1)C(=O)c2ccc(cc2)C 2G-944 COc1ccc(cc1)Cn2cc(c(c2/N=C/c3ccc(cc3)Cl)C#N)c4ccccc4 2G-948 Cn1c(=O)c2c3c(sc2nc1SCc4ccc(cc4Cl)Cl)CN(CC3)c5c(cc(cn5)C(F)(F)F)Cl 2G-950 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)O 2H-001 c1ccc(cc1)S(=O)(=O)NNC(=N)COc2ccccc2Cl 2H-002 c1ccc(cc1)S(=O)(=O)C[N+](=O)[O-] 2H-003 c1ccc(cc1)/C(=N/Nc2c(cc(cn2)C(F)(F)F)Cl)/CCC(=O)O 2H-004 CC(C(=O)/C=C/N(C)C)Sc1c(cc(cn1)C(F)(F)F)Cl 2H-006 CN(C)/C=C(\[N+](=O)[O-])/S(=O)(=O)c1ccccc1 2H-007 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N3CCOCC3 2H-009 c1ccc(cc1)C2=NN(C(=O)CC2)c3c(cc(cn3)C(F)(F)F)Cl 2H-010 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)Cl)/[N+](=O)[O-] 2H-012 CN(C)C(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 2H-014 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 2H-015 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Cl 2H-016 c1ccnc(c1)CNC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 2H-017 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)C(F)(F)F)/[N+](=O)[O-] 2H-018 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)/[N+](=O)[O-] 2H-019 CN(C)S(=O)(=O)c1ccc(cc1)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 2H-020 c1ccc(cc1)S(=O)(=O)C(/C=N/OCc2c(cccc2Cl)Cl)[N+](=O)[O-] 2H-021 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 2H-022 COc1ccc(cc1)C(CCC#N)(C#N)c2c(cc(cn2)C(F)(F)F)Cl 2H-023 CC(c1ccc(c(n1)O)C#N)Oc2cccnc2 2H-024 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCc3ccc(cc3)Cl 2H-026 c1cc(ccc1C(=O)c2cc(n(c2)c3c(cc(cn3)C(F)(F)F)Cl)C#N)Cl 2H-027 COc1ccc(cc1)CNC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 2H-028 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)N 2H-029 c1cc(cnc1)CNC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 2H-031 CO/N=C/C([N+](=O)[O-])S(=O)(=O)c1ccccc1 2H-032 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl 2H-033 COC(=O)C(Cc1c(cc(c[nH+]1)C(F)(F)F)Cl)N.[Cl-] 2H-034 COc1ccc(cc1)C2(CCC(=O)NC2=O)c3c(cc(cn3)C(F)(F)F)Cl 2H-038 COCCCNC(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 2H-039 c1ccn(c1)c2ccc(c(c2)Cl)Oc3ccc(cn3)C(F)(F)F 2H-040 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(c(c3)Cl)Oc4ccc(cn4)C(F)(F)F 2H-041 c1ccc(cc1)CC(=O)c2cc([nH]c2)C#N 2H-042 C#CCNC(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 2H-043 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCC#N 2H-045 c1c(cnc(c1Cl)SC2=CCS(=O)(=O)C2)C(F)(F)F 2H-047 c1ccc(cc1)CC(=O)c2cc(n(c2)c3c(cc(cn3)C(F)(F)F)Cl)C#N 2H-048 c1cc(c(cc1n2cc3ccsc3c2)Cl)Oc4ccc(cn4)C(F)(F)F 2H-050 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)Nc3ccc(cc3)Cl 2H-053 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Cl 2H-054 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N 2H-055 CC(c1cccn1c2c(cc(cn2)C(F)(F)F)Cl)O 2H-056 c1ccc(c(c1)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)N 2H-058 c1c(cnc(c1Cl)SC2CC(=O)OC2=O)C(F)(F)F 2H-059 c1cc(ccc1c2ccsc2C(=O)O)Cl 2H-060 CC(c1ccn[nH]1)Sc2c(cc(cn2)C(F)(F)F)Cl 2H-061 CC(/C(=N\OCc1c(cccc1Cl)Cl)/C)Sc2c(cc(cn2)C(F)(F)F)Cl 2H-062 COC(=O)c1c(ccs1)c2ccc(cc2)Cl 2H-063 c1c(c[n+](c(c1Cl)N)[O-])C(F)(F)F 2H-065 c1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccncc3 2H-066 CC(c1ccnc(n1)N)Sc2c(cc(cn2)C(F)(F)F)Cl 2H-067 c1ccc2c(c1)c(=O)n(cn2)Nc3c(cc(cn3)C(F)(F)F)Cl 2H-068 CN(C)S(=O)(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 2H-069 c1cc(ccc1CC(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)Cl 2H-070 c1c(cnc(c1Cl)SN2C(=O)CCC2=O)C(F)(F)F 2H-071 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Nc3ccc(cc3)Cl 2H-072 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Oc3ccc(cc3)Cl 2H-073 c1cc(ccc1CC(=O)c2cc([nH]c2)C(=O)N)Cl 2H-074 CCOC(=O)/C(=N\Nc1ccc(cc1[N+](=O)[O-])Cl)/NC(=O)C 2H-302S Cc1nc(nn1c2ccc(cc2F)F)C(=O)Nc3ccc(cc3Cl)Cl 2H-303S Cc1nc(nn1c2ccc(cc2F)F)C(=O)NC(C)C 2H-304S COC(=O)C(CCSC)NC(=O)CNS(=O)(=O)c1ccc(cc1)Br 2H-305S COc1ccc(cc1)S(=O)(=O)NCC(=O)O 2H-306S COC(=O)C(c1ccccc1)NC(=O)CNS(=O)(=O)c2ccc(cc2)Br 2H-307S COC(=O)C(CCSC)NC(=O)CNS(=O)(=O)c1ccc(cc1)Cl 2H-309S COC(=O)C(Cc1ccccc1)NC(=O)CNS(=O)(=O)c2ccc(cc2)Br 2H-311S Cc1ccc(cc1)S(=O)(=O)c2c(cc([nH]c2=O)c3ccccc3)C 2H-313S Cc1cccc(c1)S(=O)(=O)c2c(cc(n(c2=O)Cc3cccc(c3)C(F)(F)F)C)C 2H-314S Cc1cccc(c1)S(=O)(=O)c2c(cc(n(c2=O)Cc3ccc(cc3)Cl)C)C 2H-315S Cc1nc(nn1c2ccc(cc2)F)C(=O)Nc3ccc(cc3)F 2H-316S Cc1nc(nn1c2ccc(cc2)F)C(=O)Nc3ccc(cc3F)F 2H-317S COC(=O)C(CCSC)NC(=O)CNS(=O)(=O)c1cccc(c1)C(F)(F)F 2H-318S COC(=O)C(CCSC)NC(=O)CNS(=O)(=O)c1ccccc1Cl 2H-319S Cc1nc(nn1c2ccc(cc2)F)C(=O)Nc3cccc(c3)C(F)(F)F 2H-320S Cc1ccc(cc1)S(=O)(=O)c2c(cc(n(c2=O)Cc3ccc(c(c3)Cl)Cl)c4ccccc4)C 2H-322S CCOC(=O)c1nc(n(n1)c2ccc(cc2[N+](=O)[O-])Cl)C 2H-328S Cc1nc(nn1c2ccc(cc2)F)C(=O)Nc3ccc(cc3)Cl 2H-331S Cc1nc(nn1c2ccc(cc2)F)C(=O)Nc3ccc(cc3Cl)Cl 2H-332S CCOC(=O)c1nc(n(n1)c2ccc(cc2Cl)Cl)C 2H-333S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)O 2H-334S Cc1nc(nn1c2ccc(cc2)F)C(=O)Nc3ccc(cc3)OC 2H-336S Cc1nc(nn1c2ccc(cc2)F)C(=O)Nc3ccccc3N4CCN(CC4)C 2H-337S CCOC(=O)/C(=N\Nc1cc(ccc1Cl)Cl)/NC(=O)C 2H-338S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)Nc3ccc(cc3)F 2H-339S c1ccc(cc1)c2c(snn2)Br 2H-341S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)Nc3ccc(cc3)Cl 2H-343S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)NC 2H-344S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)N(C)C 2H-345S CCOC(=O)c1nc(n(n1)c2cc(ccc2Cl)Cl)C 2H-346S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 2H-347S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)NC(C)C 2H-348S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)O 2H-350S Cc1c(c(=O)[nH]c(c1Cl)C)S(=O)(=O)c2ccccc2 2H-354S Cc1c2c([nH]c(=O)c1S(=O)(=O)c3ccccc3)CCCC2 2H-355S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)Cc3ccccc3)c4ccccc4 2H-356S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)CC#C)c3ccccc3 2H-357S CCn1c(cc(c(c1=O)S(=O)(=O)c2ccccc2)C)c3ccccc3 2H-358S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)Nc3ccc(cc3F)F 2H-359S Cc1nc(nn1c2ccc(cc2Cl)Cl)C(=O)Nc3ccc(cc3)OC(F)(F)F 2H-360S c1ccc(cc1)c2c(snn2)Cl 2H-363S c1ccc(cc1)c2c(snn2)Sc3ccc(cc3)Cl 2H-364S c1ccc(cc1)c2c(snn2)Sc3ccc(cc3)F 2H-365S C/C(=C(/C(=O)C)\Sc1ccccc1)/N 2H-367S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3ccc(cc3Cl)Cl 2H-368S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3ccc(cc3)Cl 2H-369S c1ccc(cc1)c2c(snn2)Sc3ccc(cc3)Br 2H-372S c1ccc(cc1)c2c(snn2)Sc3ccc(c(c3)Cl)Cl 2H-373S c1ccc(cc1)c2c(snn2)Sc3cccc(c3)C(F)(F)F 2H-374S c1ccc(cc1)c2c(snn2)S(=O)(=O)c3ccc(cc3)Cl 2H-375S c1ccc(cc1)c2c(snn2)S(=O)(=O)c3ccc(cc3)F 2H-376S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3ccc(cc3)F 2H-377S CCCNC(=O)c1nc(n(n1)c2cc(ccc2Cl)Cl)C 2H-378S c1ccc(cc1)c2c(snn2)S(=O)(=O)c3cccc(c3)C(F)(F)F 2H-379S c1ccc(cc1)c2c(snn2)S(=O)(=O)c3ccc(cc3)Br 2H-380S c1ccc(cc1)c2c(snn2)S(=O)(=O)c3ccc(c(c3)Cl)Cl 2H-381S c1ccc(cc1)c2c(snn2)Sc3ccccc3Cl 2H-382S c1ccc(cc1)c2c(snn2)SCc3ccc(cc3)Cl 2H-383S Cc1ccc(cc1)Sc2c(nns2)c3ccccc3 2H-384S c1ccc(cc1)c2c(snn2)SCc3cccc(c3)C(F)(F)F 2H-385S c1ccc(cc1)c2c(snn2)SCc3ccccc3Cl 2H-386S c1ccc(cc1)c2c(snn2)SCc3ccc(cc3Cl)Cl 2H-387S Cc1ccc(cc1)S(=O)(=O)c2c(nns2)c3ccccc3 2H-388S c1ccc(cc1)c2c(snn2)S(=O)(=O)Cc3ccc(cc3)Cl 2H-389S c1ccc(cc1)c2c(snn2)S(=O)(=O)c3ccccc3Cl 2H-390S c1ccc(cc1)c2c(snn2)S(=O)(=O)Cc3cccc(c3)C(F)(F)F 2H-392S c1ccc(cc1)c2c(snn2)S(=O)(=O)Cc3ccccc3Cl 2H-393S c1ccc(cc1)c2c(snn2)S(=O)(=O)Cc3ccc(cc3Cl)Cl 2H-394S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)NC 2H-397S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)N(C)C 2H-398S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3ccc(c(c3F)Cl)F 2H-399S Cc1ccc(cc1)NC(=O)c2nc(n(n2)c3cc(ccc3Cl)Cl)C 2H-400S c1cc(cc(c1)SCc2ccc(cc2)N)C(F)(F)F 2H-401S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)CSc3cccc(c3)C(F)(F)F 2H-402S c1cc(cc(c1)SCc2ccc(cc2)NC(=O)c3cc(cc(c3)Cl)Cl)C(F)(F)F 2H-403S c1cc(cc(c1)S(=O)(=O)N2CCCC2C(=O)Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F 2H-404S c1cc(cc(c1)S(=O)(=O)N2CCCC2C(=O)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F 2H-405S CC(=O)Nc1ccc(cc1)NC(=O)C2CCCN2S(=O)(=O)c3cccc(c3)C(F)(F)F 2H-406S c1cc(cc(c1)S(=O)(=O)N2CCCC2C(=O)Nc3ccc(cc3)Cl)C(F)(F)F 2H-407S c1ccc(cc1)C(=O)Nc2ccc(cc2)CSc3cccc(c3)C(F)(F)F 2H-408S c1cc(cc(c1)SCc2ccc(cc2)NC(=O)c3ccc(cc3)Cl)C(F)(F)F 2H-409S c1cc(ccc1CSc2ccc(cc2)F)NC(=O)c3cc(cc(c3)Cl)Cl 2H-410S c1cc(cc(c1)SCc2ccc(cc2)NC(=O)c3c(cccc3F)F)C(F)(F)F 2H-411S c1cc(cc(c1)SCc2ccc(cc2)NC(=O)c3ccc(c(c3)Cl)Cl)C(F)(F)F 2H-412S c1cc(cc(c1)SCc2ccc(cc2)NC(=O)c3cccc(c3Cl)Cl)C(F)(F)F 2H-413S c1cc(cc(c1)SCc2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl)C(F)(F)F 2H-414S c1cc(cc(c1)SCc2ccc(cc2)NC(=O)c3cccs3)C(F)(F)F 2H-415S c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)F)F 2H-416S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)F 2H-417S Cc1ccc(cc1)SCc2ccc(cc2)NC(=O)c3ccccc3 2H-419S Cc1ccc(cc1)SCc2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl 2H-420S Cc1ccc(cc1)SCc2ccc(cc2)NC(=O)c3cc(cc(c3)Cl)Cl 2H-421S Cc1ccc(cc1)SCc2ccc(cc2)NC(=O)c3c(cccc3F)F 2H-422S c1ccc(cc1)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)F 2H-424S c1cc(ccc1CSc2ccc(cc2)F)NC(=O)c3ccc(cc3F)F 2H-425S c1cc(c(c(c1)Cl)Cl)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)F 2H-426S c1cc(ccc1CS(=O)(=O)c2ccc(cc2)F)NC(=O)c3cc(cc(c3)Cl)Cl 2H-427S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)CS(=O)c3ccc(cc3)F 2H-428S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)CS(=O)c3ccc(cc3)Br 2H-429S c1cc(ccc1CSc2ccc(cc2)F)NC(=O)c3ccc(c(c3)Cl)Cl 2H-430S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)F 2H-431S c1cc(ccc1CSc2ccc(cc2)F)NC(=O)c3ccc(cc3)Cl 2H-432S c1cc(sc1)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)F 2H-433S c1cc(ccc1CSc2ccc(cc2)Cl)NC(=O)c3ccc(cc3Cl)Cl 2H-435S c1cc(ccc1CSc2ccc(cc2)Cl)NC(=O)c3ccc(cc3F)F 2H-436S c1cc(sc1)C(=O)Nc2ccc(cc2)CSc3ccc(cc3)Cl 2H-437S c1ccc(cc1)S(=O)Cc2ccc(cc2)NC(=O)c3ccc(cc3F)F 2H-440S c1ccc(cc1)S(=O)Cc2ccc(cc2)NC(=O)c3ccc(cc3)C(F)(F)F 2H-441S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)CS(=O)c3cccc(c3)C(F)(F)F 2H-443S c1ccc(cc1)C(=O)Nc2ccc(cc2)CS(=O)(=O)c3ccc(cc3)Cl 2H-444S CN1C(=O)c2ccccc2C1(C#Cc3ccccc3)O 2H-446S c1ccc(cc1)C#CC2(c3ccccc3C(=O)N2c4ccccc4)O 2H-448S c1cc(ccc1C#N)OC(=O)c2ccc(nc2)n3cncn3 2H-449S c1cc(cc(c1)OC(=O)c2ccc(nc2)n3cncn3)C(F)(F)F 2H-450S Cc1c(nc(s1)c2ccncc2)O 2H-451S Cc1c(nc(s1)c2ccncc2)OC(=O)c3ccc(c(c3)Cl)Cl 2H-452S Cc1c(nc(s1)c2ccncc2)OC(=O)c3ccc(cc3Cl)Cl 2H-453S Cc1c(nc(s1)c2ccncc2)OC(=O)c3ccc(cc3)Cl 2H-454S Cc1c(nc(s1)c2ccncc2)OC(=O)c3cc(cc(c3)Cl)Cl 2H-455S Cc1c(nc(s1)c2ccncc2)OC(=O)c3ccc(cc3F)F 2H-456S CCc1cccc(c1NC(=O)C2CCCN2S(=O)(=O)c3cccc(c3)C(F)(F)F)CC 2H-457S Cc1c(nc(s1)c2ccncc2)OC(=O)c3ccccc3 2H-458S Cc1c(nc(s1)c2ccncc2)OC(=O)c3ccc(cc3)C(F)(F)F 2H-459S Cc1c(nc(s1)c2cccnc2)O 2H-460S Cc1c(nc(s1)c2cccnc2)OC(=O)c3ccc(cc3Cl)Cl 2H-461S Cc1c(nc(s1)c2cccnc2)OC(=O)c3ccc(c(c3)Cl)Cl 2H-462S Cc1c(nc(s1)c2cccnc2)OC(=O)c3cc(cc(c3)Cl)Cl 2H-463S c1ccc(c(c1)OC(=O)c2ccc(nc2)n3cncn3)Cl 2H-464S c1cc(ccc1OC(=O)c2ccc(nc2)n3cncn3)Cl 2H-465S Cc1cc(cc(c1)OC(=O)c2ccc(nc2)n3cncn3)C 2H-466S c1cc(c(cc1Cl)Cl)OC(=O)c2ccc(nc2)n3cncn3 2H-469S CC(C)(C)c1ccc(cc1)OC(=O)c2ccc(nc2)n3cncn3 2H-470S Cc1ccc(cc1)OC(=O)c2ccc(nc2)n3cncn3 2H-471S c1cc(ncc1C(=O)Oc2c(c(nc(c2Cl)F)F)Cl)n3cncn3 2H-472S Cc1c(nc(s1)c2cccs2)O 2H-473S Cc1c(nc(s1)c2cccnc2)OC(=O)c3ccccc3 2H-475S Cc1c(nc(s1)c2cccnc2)OC(=O)c3ccc(cc3)Cl 2H-476S Cc1c(nc(s1)c2cccnc2)OC(=O)c3cccc(c3)C(F)(F)F 2H-477S Cc1c(nc(s1)c2cccnc2)OC(=O)c3ccc(cc3Cl)S(=O)(=O)C 2H-478S Cc1c(nc(s1)c2cccnc2)OC(=O)C3CC3 2H-479S Cc1c(nc(s1)c2ccccn2)O 2H-480S Cc1c(nc(s1)c2ccccn2)OC(=O)c3ccc(cc3Cl)Cl 2H-481S Cc1c(nc(s1)c2cccs2)OC(=O)C3CC3 2H-482S Cc1c(nc(s1)c2ccccn2)OC(=O)c3cccc(c3)C(F)(F)F 2H-484S Cc1c(nc(s1)c2ccccn2)OC(=O)c3ccc(cc3F)F 2H-485S Cc1c(nc(s1)c2ccccn2)OC(=O)c3ccc(cc3Cl)S(=O)(=O)C 2H-486S Cc1c(nc(s1)c2ccccn2)OC(=O)c3ccccc3 2H-487S Cc1c(nc(s1)c2ccccn2)OC(=O)c3ccc(c(c3)Cl)Cl 2H-488S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 2H-489S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3ccc(cc3F)F 2H-490S Cc1c(nc(s1)c2ccccn2)OC(=O)c3ccc(cc3)Cl 2H-491S Cc1c(nc(s1)c2ccccn2)OC(=O)c3cccc(c3Cl)Cl 2H-492S Cc1ccc(cc1)C(=O)Oc2c(sc(n2)c3ccccn3)C 2H-493S CCCCC#CC1(c2ccccc2C(=O)N1c3ccccc3)O 2H-494S c1ccc(cc1)C(=O)/C=C/2\c3ccccc3C(=O)N2c4ccccc4 2H-749S c1cc(cc(c1)OCC[NH3+])C(F)(F)F.[Cl-] 2H-900 c1ccc2c(c1)CCC3=C2CCN(C3)CCc4ccc(cc4)S(=O)(=O)N 2H-901 COCc1ccc(cc1)COC 2H-903 CCOC(=O)C1=NOC(C1)CNC(=O)C2=NOC(C2)CNC(=O)c3c(onc3c4ccccc4Cl)C 2H-904 c1cc(ccc1NC(=O)OCCN(CCNc2c(cc(cn2)C(F)(F)F)Cl)c3c(cc(cn3)C(F)(F)F)Cl)Cl 2H-905 CN(c1c(cc(cn1)C(F)(F)F)Cl)N 2H-906 c1cc(ccc1Cn2cc(c(=O)[nH]c2=O)C#N)Cl 2H-907 COCCCn1cc(c(=O)[nH]c1=O)C#N 2H-908 COc1ccc(cc1OC)CCn2cc(c(=O)[nH]c2=O)C#N 2H-909 CC(=O)c1cn(c(=O)[nH]c1=O)N(C)c2c(cc(cn2)C(F)(F)F)Cl 2H-910 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c(=O)[nH]c2=O)C#N 2H-911 c1cc(ccc1Cn2cc(c(=O)n(c2=O)Cc3c(cc(cn3)C(F)(F)F)Cl)C#N)Cl 2H-912 COCCCn1cc(c(=O)n(c1=O)Cc2c(cc(cn2)C(F)(F)F)Cl)C#N 2H-913 COc1ccc(cc1OC)CCn2cc(c(=O)n(c2=O)Cc3c(cc(cn3)C(F)(F)F)Cl)C#N 2H-914 c1cc(ccc1NC(=O)OCCN(CCNc2c(cc(cn2)C(F)(F)F)Cl)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 2H-915 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c(=O)n(c2=O)Cc3ccc(cc3)F)C#N 2H-917 CC(=O)c1cn(c(=O)[nH]c1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl 2H-919 CC(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)F)N3CCN(CC3)C 2H-920 CC(=O)c1cn(c(=O)[nH]c1=O)Cc2ccccc2 2H-921 CC(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)F)Cc3ccccc3 2H-922 c1cc(ccc1NC(=S)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 2H-923 c1ccc(cc1)NC(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 2H-924 c1cc(c(cc1NC(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl 2H-925 CN(C)/C=C/C(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)F)Cc3ccccc3 2H-926 CCOC(=O)C(Cc1ccc(cc1)COC)(C(=O)OCC)NC(=O)C 2H-927 c1cc(ccc1NC(=S)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl 2H-928 c1c(cnc(c1Cl)NCC2CC(=NO2)C(=O)NNC(=O)C3CC3)C(F)(F)F 2H-929 c1cc(c(cc1Cl)Cl)CON/C=N/C(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 2H-930 c1ccc(cc1)CON/C=N/C(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 2H-931 c1ccc(cc1)Cn2cc(c(=O)n(c2=O)Cc3ccc(cc3)F)c4ccnn4c5c(cc(cn5)C(F)(F)F)Cl 2H-932 CC(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)F)N(C)c3c(cc(cn3)C(F)(F)F)Cl 2H-933 CN(C)C=C1C(=O)CC(CC1=O)c2ccc(cc2)Cl 2H-934 COc1ccc(cc1)OCCN2CCC3=C(C2)CCc4c3cccc4.Cl 2H-935 Cc1c(cn(n1)c2ccccc2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 2H-936 C/[N+](=C\C1C(=O)CC(CC1=O)c2ccc(cc2)Cl)/[O-] 2H-937 Cc1c(cnc(n1)c2ccccc2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 2H-938 COc1ccc(cc1)N/C=C/C(=O)c2cn(c(=O)n(c2=O)Cc3ccc(cc3)F)Cc4ccccc4 2H-939 CC1(CC(=O)C(C(=O)C1)/C=[N+](\C)/[O-])C 2H-940 CN(C)/C=C/C(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)F)N(C)c3c(cc(cn3)C(F)(F)F)Cl 2H-941 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c(=O)n(c2=O)CCOc3cccc(c3)C(F)(F)F)C#N 2H-942 CCOC(=O)Cn1c(=O)c(cn(c1=O)N(C)c2c(cc(cn2)C(F)(F)F)Cl)C#N 2H-943 Cn1c(=O)c(cn(c1=O)N(C)c2c(cc(cn2)C(F)(F)F)Cl)C#N 2H-944 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)Nc2ccc(cc2)Cl 2H-945 c1c(cnc(c1Cl)NCCN(CCOc2c(cc(cn2)C(F)(F)F)Cl)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 2H-946 c1ccc2c(c1)CCC3=C2CCN(C3)CCOc4cccc(c4)C(F)(F)F.Cl 2H-948 CN(C=C1C(=O)CC(CC1=O)c2ccc(cc2)Cl)OC(=O)Nc3ccccc3 2H-949 c1c(cnc(c1Cl)NCC2CC(=NO2)C(=O)NC3CC3)C(F)(F)F 2H-950 c1cc(ccc1NC(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 2H-951 CC(C)(C)c1ccc(cc1)NC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 2H-952 c1cc(cnc1)NC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 2H-953 c1cc(sc1)C(=O)NNC(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 2H-954 COc1ccc(cc1)N2CCN(CC2)C(=O)C3=NOC(C3)CNc4c(cc(cn4)C(F)(F)F)Cl 2H-955 C/C(=C\C(=O)N1CCN(CC1)c2ccccc2)/N3CCN(CC3)c4ccc(cc4)Cl 2H-956 c1ccc2c(c1)ccn2c3c(cc(cn3)C(F)(F)F)Cl 2H-958 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c(=O)n(c2=O)Cc3ccc(cc3)F)C(=O)/C=C/Nc4ccc(cc4)Cl 2H-959 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c(=O)n(c2=O)Cc3c(cc(cn3)C(F)(F)F)Cl)C#N 2H-960 CC(=O)c1cn(c(=O)n(c1=O)CCOc2ccc(cc2)OC)N(C)c3c(cc(cn3)C(F)(F)F)Cl 2H-961 CC(=O)c1cn(c(=O)n(c1=O)CC=C)N(C)c2c(cc(cn2)C(F)(F)F)Cl 2H-962 c1ccc(cc1)COc2ccc3c(c2)ccn3c4c(cc(cn4)C(F)(F)F)Cl 2H-963 Cc1c(cn(n1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 2H-964 CC(=O)CC(=O)N1CCN(CC1)c2ccc(cc2)Cl 2H-965 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/c2cn(c(=O)n(c2=O)Cc3ccc(cc3)F)N(C)c4c(cc(cn4)C(F)(F)F)Cl 2H-966 CCOC(=O)NC(=O)/C(=C\Nc1ccc(c(c1)Cl)Oc2ccc(cn2)C(F)(F)F)/C#N 2H-967 Cc1c(n([nH]c1=O)c2c(cc(cn2)C(F)(F)F)Cl)C 2H-968 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c(=O)n(c2=O)CC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C#N 2H-969 CC(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)F)c3ccc(cc3)Cl 2H-970 COc1ccc(cc1)NC(=O)C(=O)c2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl 2H-972 c1cc(c(cc1n2cc(c(=O)[nH]c2=O)C#N)Cl)Oc3ccc(cn3)C(F)(F)F 2H-973 CN(C)/C=C/C(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)F)c3ccc(cc3)Cl 2H-974 c1c(cnc(c1Cl)Sc2nc(sn2)Sc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 2H-975 CN(C)/C=C\1/c2ccccc2NC1=O 2H-976 c1cc(ccc1Cn2c(=O)c(cn(c2=O)c3ccc(cc3)Cl)c4ccnn4c5c(cc(cn5)C(F)(F)F)Cl)F 2H-977 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c(=O)[nH]c2=O)C(=O)/C=C/c3ccc(cc3)Cl 2H-978 Cn1c(=O)c(cn(c1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl)C(=O)/C=C/N(C)C 2H-979 Cn1c(=O)c(cn(c1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl)C#N 2H-980 CCOC(=O)NC(=O)/C(=C\Nc1ccc(c(c1)Cl)Oc2ccc(cn2)C(F)(F)F)/C(=O)C 2H-981 c1c(cnc(c1Cl)NCCCC(=O)O)C(F)(F)F 2H-982 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C(=O)C(=O)Nc4ccc(cc4)Cl 2H-983 CCOC(=O)NC(=O)C(=CNc1ccc(c(c1)Cl)Oc2ccc(cn2)C(F)(F)F)C(=O)NC(=O)OCC 2H-985 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)N(C)c2c(cc(cn2)C(F)(F)F)Cl 2H-987 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)C(F)(F)F 2H-988 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C=O 2H-989 Cn1c(=O)c(cn(c1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl)C(=O)/C=C/Nc3ccc(cc3)C(F)(F)F 2H-991 C/[N+](=C/c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl)/[O-] 2H-992 CN(C)/C=C(\c1ccc(s1)C(=O)/N=C/N(C)C)/c2c(cc(cn2)C(F)(F)F)Cl 2J-001 c1cc(ccc1C(C#N)c2c(cc(cn2)C(F)(F)F)Cl)OC(=O)c3ccc(cc3)Cl 2J-003 CN(C)/C=C(\c1cccs1)/c2c(cc(cn2)C(F)(F)F)Cl 2J-006 c1cc(c(cc1Cl)Cl)/C(=N\NC(=O)N)/c2c(cc(cn2)C(F)(F)F)Cl 2J-007 CCOC(=O)CNC(=O)c1ccc(cc1)Cl 2J-008 c1cc(c(cc1Cl)Cl)c2c3c(cc(cn3)C(F)(F)F)[nH]n2 2J-009 c1cc(c(cc1Cl)Cl)c2c3c(cc(cn3)C(F)(F)F)n(n2)C(=O)Nc4ccc(cc4Cl)Cl 2J-010 c1ccc(c(c1)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)C(=O)O 2J-011 c1cc(cc(c1)C(F)(F)F)C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3 2J-012 c1cc(cc(c1)C(F)(F)F)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 2J-013 CO/N=C/C(c1cccs1)c2c(cc(cn2)C(F)(F)F)Cl 2J-014 c1ccc2c(c1)C(=O)N(C2=O)Nc3c(cc(cn3)C(F)(F)F)Cl 2J-015 c1cc(sc1)C(/C=N/O)c2c(cc(cn2)C(F)(F)F)Cl 2J-016 CCOc1cnc(o1)c2ccc(cc2)Cl 2J-017 c1cc(ccc1C(=O)CSc2ncc(c(n2)C(F)(F)F)C#N)C(F)(F)F 2J-018 c1cc(ccc1C2=CC(=O)OC2=O)Cl 2J-026 c1cc(cc(c1)C(F)(F)F)C(=O)c2cc(cnc2C(=O)c3cccc(c3)C(F)(F)F)C(F)(F)F 2J-028 c1cc(cc(c1)C(F)(F)F)c2c3cc(cnc3c(nn2)c4cccc(c4)C(F)(F)F)C(F)(F)F 2J-029 c1cc(ccc1C(=O)O)n2c(c(cn2)C#N)C(F)(F)F 2J-030 c1cc(ccc1/C(=N\Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F)/c3c(cc(cn3)C(F)(F)F)Cl)Cl 2J-031 CCOC(=O)CNC(=O)C(F)(F)F 2J-033 COc1ccc(cc1)c2c(c(nc(n2)c3cccc(c3)Cl)Cl)C#N 2J-035 CN(C)c1[nH]nc(n1)N(C)C 2J-036 CN1CCN(CC1)c2c(c(nc(n2)c3cccc(c3)Cl)c4ccc(cc4)OC)C#N 2J-037 c1ccc(c(c1)C(=N)N)Cl.Cl 2J-038 c1cc(ccc1C2=CC(=O)N(C2=O)Nc3c(cc(cn3)C(F)(F)F)Cl)Cl 2J-039 c1cc(ccc1c2c3c(cc(cn3)C(F)(F)F)n(n2)c4ccc(cc4[N+](=O)[O-])C(F)(F)F)Cl 2J-041 CN(C)c1nc(n(n1)C(=O)Nc2ccc(cc2)Cl)N(C)C 2J-043 CN(C)c1nc(n(n1)C(=O)c2ccc(cc2)Cl)N(C)C 2J-044 CCOC(=O)/C(=C/c1ccc(cc1)OC)/C#N 2J-048 c1ccc(cc1)C(C#N)(c2cc(cnc2C(=O)c3cccc(c3)C(F)(F)F)C(F)(F)F)N4CCOCC4 2J-049 c1ccc(c(c1)c2[nH]nnn2)Cl 2J-051 COc1ccc(cc1)c2c(c(nc(n2)c3ccc(cc3)Cl)Cl)C#N 2J-052 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)N2CCOCC2 2J-053 c1cc(c(cc1Cl)Cl)c2c3cc(cnc3c(nn2)c4ccc(cc4Cl)Cl)C(F)(F)F 2J-056 c1ccc(cc1)N2CCN(CC2)C(=O)c3ccccc3CC[N+](=O)[O-] 2J-057 CN1CCN(CC1)c2c(c(nc(n2)c3ccc(cc3)Cl)c4ccc(cc4)OC)C#N 2J-059 CN(C)c1nc(n(n1)S(=O)(=O)c2ccc(cc2)Cl)N(C)C 2J-060 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)NCc2cccs2 2J-061 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl 2J-062 c1cc(ccc1CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O)Cl 2J-301S Cc1ccc(cc1)CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O 2J-302S c1ccc(cc1)C(=O)NCc2[nH]c3ccccc3n2 2J-303S c1cc(cc(c1)Cl)C[NH2+]CC(c2ccc(cc2)F)(c3ccc(cc3)F)O.[Cl-] 2J-304S c1ccc(c(c1)C[NH2+]CC(c2ccc(cc2)F)(c3ccc(cc3)F)O)Cl.[Cl-] 2J-305S COc1ccc(cc1)CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O 2J-306S COc1ccccc1CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O 2J-307S COc1cccc(c1)CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O.Cl 2J-308S Cc1cc2c(c(c1C)N)ncn2Cc3ccccc3 2J-309S COc1ccc(cc1OC)CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O 2J-310S c1cc(ccc1CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O)F 2J-311S c1ccc(c(c1)CNCC(c2ccc(cc2)F)(c3ccc(cc3)F)O)F 2J-312S c1cc(cc(c1)C(F)(F)F)C[NH2+]CC(c2ccc(cc2)F)(c3ccc(cc3)F)O.[Cl-] 2J-313S COc1cnc(nc1SCc2ccccc2)c3ccccn3 2J-316S COc1cnc(nc1Sc2cccc(c2)Cl)c3ccccn3 2J-317S COc1cnc(nc1Sc2ccccc2Cl)c3ccccn3 2J-318S COc1cnc(nc1Oc2cccc(c2)C(F)(F)F)c3ccccn3 2J-319S COc1cnc(nc1OC)c2ccccn2 2J-320S c1cc(ccc1C(CNCc2ccc(c(c2)Cl)Cl)(c3ccc(cc3)F)O)F 2J-321S c1ccc(cc1)C(Cn2cncn2)(c3ccccc3)O 2J-322S COc1cnc(nc1Oc2ccccc2)c3ccccn3 2J-323S CC(C)(C)c1ccc(cc1)Oc2c(cnc(n2)c3ccccn3)OC 2J-324S COc1cnc(nc1Oc2ccc(cc2)Cl)c3ccccn3 2J-325S COc1cnc(nc1Oc2ccccc2Cl)c3ccccn3 2J-326S COc1ccc(cc1)Oc2c(cnc(n2)c3ccccn3)OC 2J-327S COc1cnc(nc1Oc2cccc(c2)Cl)c3ccccn3 2J-328S COc1cnc(nc1Oc2ccc(cc2)F)c3ccccn3 2J-329S COc1cnc(nc1Oc2ccccc2C(=O)OC)c3ccccn3 2J-330S c1cc(ccc1C(CNCc2ccc(cc2Cl)Cl)(c3ccc(cc3)F)O)F 2J-331S CN1CCN(CC1)CC(c2ccc(cc2)F)(c3ccc(cc3)F)O.Cl 2J-332S c1cc(cc(c1)Cl)N2CCN(CC2)CC(c3ccc(cc3)F)(c4ccc(cc4)F)O 2J-333S c1ccc(cc1)CNCC(c2ccccc2)(c3ccccc3)O 2J-334S COc1cnc(nc1Oc2cc(cc(c2)Cl)Cl)c3ccccn3 2J-335S c1ccc(cc1)C(CNCc2ccccc2F)(c3ccccc3)O 2J-338S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3)OC)ncn2Cc4ccccc4 2J-339S Cc1ccc(cc1)CNCC(c2ccccc2)(c3ccc(cc3)F)O 2J-340S c1ccc(cc1)C(CNCc2ccc(cc2)Cl)(c3ccc(cc3)F)O 2J-341S COc1ccc(cc1)CNCC(c2ccccc2)(c3ccc(cc3)F)O 2J-342S c1ccc(cc1)C(C[NH2+]Cc2cccc(c2)Cl)(c3ccc(cc3)F)O.[Cl-] 2J-343S c1ccc(cc1)C(CNCc2ccccc2Cl)(c3ccc(cc3)F)O.Cl 2J-344S c1ccc(cc1)C(CNCc2ccc(cc2Cl)Cl)(c3ccc(cc3)F)O 2J-345S c1ccc(cc1)C(CNCc2ccc(c(c2)Cl)Cl)(c3ccc(cc3)F)O 2J-346S COc1ccc(cc1OC)CNCC(c2ccccc2)(c3ccc(cc3)F)O 2J-347S c1ccc(cc1)C(CN2CCOCC2)(c3ccccc3)O 2J-348S COc1ccccc1C[NH2+]CC(c2ccccc2)(c3ccc(cc3)F)O.[Cl-] 2J-349S COc1cccc(c1)CNCC(c2ccccc2)(c3ccc(cc3)F)O.Cl 2J-350S CC(C)Nc1c(cnc(n1)c2ccccn2)OC 2J-352S CCOC(=O)CSc1c(cnc(n1)c2ccccn2)OC 2J-353S COc1cnc(nc1Oc2ccc(cc2F)F)c3ccccn3 2J-355S CN(c1ccccc1)c2c(cnc(n2)c3ccccn3)OC 2J-356S c1ccc(cc1)C(CNCc2cccc(c2)C(F)(F)F)(c3ccc(cc3)F)O.Cl 2J-357S CC(C)[NH2+]CC(c1ccccc1)(c2ccc(cc2)F)O.[Cl-] 2J-358S c1ccc(cc1)C(CNCc2ccccc2F)(c3ccc(cc3)F)O.Cl 2J-359S c1ccc(cc1)C(CNCc2ccc(cc2)F)(c3ccc(cc3)F)O 2J-360S COc1ccccc1Sc2c(cnc(n2)c3ccccn3)OC 2J-361S COc1cnc(nc1Sc2ccc(cc2Cl)Cl)c3ccccn3 2J-362S c1ccc2c(c1)[nH]c(n2)CNC(=O)c3ccc(cc3Cl)Cl 2J-366S c1ccc(cc1)C(CN2CCOCC2)(c3ccc(cc3)F)O 2J-367S c1ccc(cc1)C(CN2CCN(CC2)c3cccc(c3)Cl)(c4ccc(cc4)F)O 2J-368S c1ccc(cc1)CC(C(=O)O)NC(=O)c2ccccc2 2J-369S c1ccc2c(c1)[nH]c(n2)CNC(=O)c3ccc(c(c3)Cl)Cl 2J-371S CCOC(=O)C(C)Sc1c(cnc(n1)c2ccccn2)OC 2J-373S c1ccc(c(c1)C(=O)NCC(=O)O)Cl 2J-374S Cc1ccc2c(c1)nc([nH]2)CNC(=O)c3ccccc3 2J-376S CC(c1[nH]c2ccccc2n1)NC(=O)c3ccccc3 2J-377S c1ccc(cc1)CC(c2[nH]c3ccccc3n2)NC(=O)c4ccccc4 2J-378S c1ccc2c(c1)nc(n2Cc3cc(ccc3Cl)Cl)/C=C/c4ccc(cc4Cl)Cl 2J-503S c1ccc2c(c1)nc(n2Cc3ccc(cc3Cl)Cl)/C=C/c4ccc(cc4Cl)Cl 2J-504S c1ccc(cc1)c2c(cnc(n2)c3ccncc3)C(=O)Nc4cccc(c4)C(F)(F)F 2J-511S CNC(=O)c1cnc(nc1c2ccccc2)c3ccccc3 2J-514S CCNC(=O)c1cnc(nc1c2ccccc2)c3ccccc3 2J-515S C=CCNC(=O)c1cnc(nc1c2ccccc2)c3ccccc3 2J-516S CCCNC(=O)c1cnc(nc1c2ccccc2)c3ccccc3 2J-518S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)N4CCOCC4 2J-519S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)N4CCN(CC4)c5ccccc5F 2J-520S CC(C)NC(=O)c1cnc(nc1c2ccccc2)c3ccccc3 2J-521S CN(C)C(=O)c1cnc(nc1c2ccccc2)c3ccccc3 2J-522S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)N4CCSCC4 2J-523S CC(C)(C#C)NC(=O)c1cnc(nc1c2ccccc2)c3ccccc3 2J-524S c1ccc(cc1)c2c(cnc(n2)c3ccccc3)C(=O)N4CCN(CC4)c5cccc(c5)C(F)(F)F 2J-525S COc1cccc(c1)Cn2c3ccccc3nc2/C=C/c4ccc(cc4)C#N 2J-526S CCOC(=O)Cn1c2ccccc2nc1/C=C/c3ccc(cc3Cl)Cl 2J-527S c1ccc(c(c1)Cn2c3ccccc3nc2/C=C/c4ccc(cc4)C#N)Cl 2J-528S c1ccc2c(c1)nc(n2Cc3ccc(cc3)F)/C=C/c4ccc(cc4)C#N 2J-529S CC1C(=O)Nc2ccccc2N1 2J-532S CC1C(=O)Nc2ccccc2N1C(=O)c3ccccc3 2J-533S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4ccc(cc4)Cl 2J-534S CNC(=O)c1cnc(nc1c2ccccc2)c3cccnc3 2J-535S CCNC(=O)c1cnc(nc1c2ccccc2)c3cccnc3 2J-537S CCCNC(=O)c1cnc(nc1c2ccccc2)c3cccnc3 2J-538S c1ccc2c(c1)nc(n2Cc3ccc(c(c3)Cl)Cl)/C=C/c4ccc(cc4)C#N 2J-540S COc1cccc(c1)Cn2c3ccccc3nc2/C=C/c4ccccc4Cl 2J-541S CC(C)(C)c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccccc4Cl 2J-542S CC1C(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)Cl 2J-543S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4ccc(cc4)C(F)(F)F 2J-544S CCCCNC(=O)c1cnc(nc1c2ccccc2)c3cccnc3 2J-545S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4cccc(c4)Cl 2J-547S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4ccc(c(c4)Cl)Cl 2J-548S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4c(cccc4Cl)F 2J-549S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4c(cccc4Cl)Cl 2J-550S c1ccc2c(c1)nc(n2Cc3cccc(c3)Cl)/C=C/c4ccc(cc4)C#N 2J-551S c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccc(cc4)C#N 2J-552S c1ccc(c(c1)/C=C/c2nc3ccccc3n2Cc4c(cccc4Cl)F)Cl 2J-553S c1ccc(c(c1)/C=C/c2nc3ccccc3n2Cc4c(cccc4Cl)Cl)Cl 2J-554S c1ccc(cc1)Cn2c3ccccc3nc2/C=C/c4ccccc4Cl 2J-555S c1ccc(c(c1)/C=C/c2nc3ccccc3n2Cc4cccc(c4)Cl)Cl 2J-556S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4cccc(c4)F 2J-557S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4cccc(c4)OC 2J-558S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4ccccc4Cl 2J-559S CC(C)(C#C)NC(=O)c1cnc(nc1c2ccccc2)c3cccnc3 2J-560S c1ccc(c(c1)/C=C/c2nc3ccccc3n2Cc4ccc(cc4Cl)Cl)Cl 2J-561S c1ccc(c(c1)/C=C/c2nc3ccccc3n2Cc4cccc(c4)F)Cl 2J-562S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4ccccc4 2J-563S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4ccc(cc4Cl)Cl 2J-564S CC1C(=O)N(c2ccccc2N1C(=O)c3ccccc3)Cc4ccc(cc4)C(C)(C)C 2J-565S CC1C(=O)Nc2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F 2J-566S c1ccc(c(c1)/C=C/c2nc3ccccc3n2Cc4ccc(cc4)Cl)Cl 2J-567S c1ccc(c(c1)/C=C/c2nc3ccccc3n2Cc4cccc(c4)C#N)Cl 2J-568S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)Cl)Cc4ccc(cc4)Cl 2J-569S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)Cl)Cc4ccc(cc4)C(F)(F)F 2J-570S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)Cl)Cc4ccc(c(c4)Cl)Cl 2J-571S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)Cl)Cc4c(cccc4Cl)Cl 2J-572S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)Cl)Cc4c(cccc4Cl)F 2J-573S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)Cl)Cc4cccc(c4)Cl 2J-574S COc1cnc(nc1Sc2c(cccc2Cl)Cl)c3ccccn3 2J-575S Cc1ccc(cc1)Sc2c(cnc(n2)c3ccccn3)OC 2J-576S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4ccc(cc4)C(=O)OC 2J-578S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4ccc(cc4)Cl 2J-579S CC1C(=O)Nc2ccccc2N1C(=O)c3ccc(cc3F)F 2J-580S Cc1ccc(cc1)C(=O)N2c3ccccc3NC(=O)C2C 2J-581S COc1cnc(nc1N2CCOCC2)c3ccccn3 2J-582S CN1CCN(CC1)c2c(cnc(n2)c3ccccn3)OC 2J-583S CNC(=O)c1cnc(nc1c2ccccc2)c3ccncc3 2J-584S CCNC(=O)c1cnc(nc1c2ccccc2)c3ccncc3 2J-585S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4c(cccc4Cl)Cl 2J-589S CN(C)C(=O)c1cnc(nc1c2ccccc2)c3ccncc3 2J-592S COc1cnc(nc1N2CCCC2)c3ccccn3 2J-594S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4ccc(cc4)F 2J-597S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4cccc(c4)Cl 2J-598S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4ccc(c(c4)Cl)Cl 2J-599S Cc1ccc(cc1)C(=O)N2c3ccccc3N(C(=O)C2C)Cc4ccc(cc4)Cl 2J-600S Cc1ccc(cc1)C(=O)N2c3ccccc3N(C(=O)C2C)Cc4c(cccc4Cl)Cl 2J-601S Cc1ccc(cc1)C(=O)N2c3ccccc3N(C(=O)C2C)Cc4ccc(cc4)C(F)(F)F 2J-602S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3F)F)Cc4ccc(cc4)Cl 2J-604S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3F)F)Cc4c(cccc4Cl)Cl 2J-605S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)Cl)Cc4ccc(cc4Cl)Cl 2J-606S c1ccc2c(c1)c3c(n2c4c(cc(cn4)C(F)(F)F)Cl)CCC5(C3)OCCO5 2J-900 Cc1ccc(cc1)SC2C(C(=O)N(C2=O)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl 2J-901 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/c2ccc3c(c2)c(on3)c4ccc(cc4)F 2J-902 c1cc(ccc1CSC2=NCCN2c3ccc(cc3)C(=O)O)Cl 2J-903 c1ccc(cc1)n2c(ccn2)c3c(ccs3)Cl 2J-904 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)CC(C2=O)Sc3ccccc3 2J-905 CC1(CC(=O)C2(C3C(C(=O)N(C3=O)N(C)c4c(cc(cn4)C(F)(F)F)Cl)ON2)C(=O)C1)C 2J-906 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C=C(C2=O)Sc3ccccc3 2J-907 CC1(NC(=O)N(N1)c2ccccc2)C3=NOC4C3C(=O)N(C4=O)CCNc5c(cc(cn5)C(F)(F)F)Cl 2J-908 CC1(NC(=O)N(N1)c2ccc(cc2Cl)Cl)C3=NOC4C3C(=O)N(C4=O)N(C)c5c(cc(cn5)C(F)(F)F)Cl 2J-909 c1cc(ccc1CSc2nc(sn2)SCc3ccc(cc3)F)F 2J-915 c1cc(c(nc1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 2J-916 c1cc(c(nc1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)[NH3+].[Cl-] 2J-917 CCO/C=N/c1cccnc1NCCNc2c(cc(cn2)C(F)(F)F)Cl 2J-918 Cc1ccc(cc1)C(=O)Nc2cccnc2NCCNc3c(cc(cn3)C(F)(F)F)Cl 2J-919 c1cc(c(nc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)[NH3+].[Cl-] 2J-920 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCNc2c(cc(cn2)C(F)(F)F)Cl 2J-922 COc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2)N3CCC(=O)CC3 2J-923 c1cc(c(nc1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)C(F)(F)F 2J-924 c1cc(c(cc1C(F)(F)F)[NH3+])NCCNc2c(cc(cn2)C(F)(F)F)Cl.[Cl-] 2J-925 c1ccc(cc1)c2nccc(n2)c3ccc4c(c3)c(on4)c5ccc(cc5)F 2J-927 c1ccc(cc1)C[NH+]2CCC3(CC2)c4c(c5ccccc5[nH]4)CC[NH2+]3.[Cl-].[Cl-] 2J-928 c1ccc2c(c1)c3c([nH]2)C4(CCN(CC4)c5ccc(cc5)[N+](=O)[O-])[NH2+]CC3.[Cl-] 2J-929 Cc1ccc(cc1)C(=O)N2CCc3c4ccccc4[nH]c3C25CCN(CC5)Cc6ccccc6 2J-931 Cc1ccc(cc1)S(=O)(=O)N2CCc3c4ccccc4[nH]c3C25CCN(CC5)Cc6ccccc6 2J-932 c1cc(c(nc1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)c3ccc(cc3Cl)Cl 2J-934 c1ccc(c(c1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 2J-935 c1c(cnc(c1Cl)OC/C=C\CO)C(F)(F)F 2J-936 c1ccc(c(c1)[NH3+])NCCNc2c(cc(cn2)C(F)(F)F)Cl.[Cl-] 2J-937 CC1(NC(=O)N(N1)c2ccc(cc2Cl)Cl)C3=NOC4C3C(=O)N(C4=O)CCNc5c(cc(cn5)C(F)(F)F)Cl 2J-938 c1ccc(c(c1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)c3ccc(cc3Cl)Cl 2J-940 c1ccc(c(c1)NCCNc2c(cc(cn2)C(F)(F)F)Cl)NS(=O)(=O)c3ccc(cc3)Cl 2J-941 c1cc(cc(c1)NC(=O)Nc2cccnc2NCCNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 2J-942 c1cc(ccc1NC(=O)OC/C=C/COc2c(cc(cn2)C(F)(F)F)Cl)Cl 2J-943 c1cc(ccc1C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)N4CCN=C4Sc5c(cc(cn5)C(F)(F)F)Cl 2J-944 c1ccc(c(c1)c2nccc(n2)c3ccc4c(c3)c(on4)c5ccc(cc5)F)F 2J-946 c1cc(ccc1C(=O)O)N2CCN=C2Sc3ccc(cc3)[N+](=O)[O-] 2J-947 c1ccn(c1)c2cccnc2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 2J-948 c1cc2c(nc1)n(c(=O)c(=O)[nH]2)CCNc3c(cc(cn3)C(F)(F)F)Cl 2J-951 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 2J-952 c1cc(c(cc1C(F)(F)F)N)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 2J-953 c1cc(ccc1NC(=O)Nc2cc(ccc2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F)Cl 2J-954 c1cc(c(cc1C(F)(F)F)n2cc(c(=O)[nH]c2=O)C#N)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 2J-955 c1ccc(cc1)N2C(=O)NC3(N2)CCC4(CC3)OCCO4 2J-956 c1ccc(cc1)N2C(=O)NC3(N2)CCC4(CC3)NC(=O)N(N4)c5ccccc5 2J-957 c1cc(ccc1S(=O)(=O)Nc2cc(ccc2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F)Cl 2J-958 COC(=O)c1c(onc1c2c(cccc2Cl)Cl)/C=C/c3cnc(c4c3onc4c5c(cccc5Cl)Cl)O 2K-001 CCOC(=O)CNC(=S)Nc1ccccc1Oc2c(cc(cn2)C(F)(F)F)Cl 2K-002 CCOC(=C(C#N)C#N)C 2K-004 CN(C)/C=C/C(=C(C#N)C#N)OC 2K-005 c1ccc2c(c1)nc(c(n2)NNC(=O)Nc3ccc(cc3)Cl)C(F)(F)F 2K-007 COC(=O)c1c(onc1c2c(cccc2Cl)Cl)/C=C/c3cnc(c4c3onc4c5c(cccc5Cl)Cl)Cl 2K-008 c1cc(ccc1C(F)(F)F)N2C(=O)CNC2=S 2K-009 CN(c1c(nc2ccccc2n1)C(F)(F)F)NC(=O)Nc3ccc(cc3)Cl 2K-010 c1ccc2c(c1)nc(c(n2)N/N=C/c3ccc(cc3)Cl)C(F)(F)F 2K-011 c1ccc2c(c1)nc(c3n2c(nn3)c4ccc(cc4)Cl)C(F)(F)F 2K-012 Cc1cc(n(n1)c2c(nc3ccccc3n2)C(F)(F)F)C 2K-013 c1ccc2c(c1)nc(c(n2)N/N=C/c3ccc(cc3Cl)Cl)C(F)(F)F 2K-014 COc1ccc(cc1)c2ccnn2c3c(nc4ccccc4n3)C(F)(F)F 2K-015 c1cc(c(cc1Cl)Cl)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 2K-016 c1ccc2c(c1)nc(c3n2c(nn3)c4ccc(cc4Cl)Cl)C(F)(F)F 2K-018 c1ccc(cc1)/C=N\Nc2c(nc3ccccc3n2)C(F)(F)F 2K-019 Cc1ccc(cc1)S(=O)(=O)NNc2c(nc3ccccc3n2)C(F)(F)F 2K-020 COC(=O)c1c(onc1c2c(cccc2Cl)Cl)/C=C/c3cnc(c4c3onc4c5c(cccc5Cl)Cl)Oc6ccc(cc6)Cl 2K-021 COC(=O)c1c(onc1c2c(cccc2Cl)Cl)/C=C/c3cnc(c4c3onc4c5c(cccc5Cl)Cl)Sc6ccc(cc6)Cl 2K-022 c1cc(ccc1/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 2K-024 c1cc(ccc1c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F)Cl 2K-025 c1ccc2c(c1)nc(c(n2)N/N=C/c3cccnc3)C(F)(F)F 2K-026 COc1ccnc(c1C#N)N 2K-027 COc1cc[nH]c(=O)c1C#N 2K-028 Cc1ccccc1C(=O)NN(C)c2c(nc3ccccc3n2)C(F)(F)F 2K-029 Cc1ccc(cc1)S(=O)(=O)NN(C)c2c(nc3ccccc3n2)C(F)(F)F 2K-030 CCOC(=O)CNC(=S)Nc1ccc(cc1)F 2K-031 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)Cl)Sc3c(cc(cn3)C(F)(F)F)Cl 2K-032 c1cc(ccc1N2C(=O)CNC2=S)F 2K-033 c1ccc(cc1)NC(=O)Nc2ccccc2Sc3c(cc(cn3)C(F)(F)F)Cl 2K-034 CN(C)C(=O)CCc1c(cc(cn1)C(F)(F)F)Cl 2K-035 COc1ccc(cc1)C(=O)Nc2ccccc2Sc3c(cc(cn3)C(F)(F)F)Cl 2K-037 COc1ccnc(c1C#N)N2CCN(CC2)c3ccccc3 2K-038 c1c(cn2c(c1Cl)nnc2N)C(F)(F)F 2K-040 CN(C)/C=C/C(=C(C#N)C#N)N(C)C 2K-041 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)Cl 2K-042 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)F 2K-043 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)F 2K-044 COc1ccnc(c1C#N)Cl 2K-045 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)C(F)(F)F 2K-046 CN(C)C(=C(C#N)C#N)/C=C/NOC 2K-047 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)C(F)(F)F 2K-048 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)OC 2K-049 CN(c1c(nc2ccccc2n1)C(F)(F)F)NC(=O)c3ccc(cc3)Cl 2K-050 c1ccc(cc1)c2nnc3n2c4ccccc4nc3C(F)(F)F 2K-051 c1ccc2c(c1)nc(c(n2)n3c(ccn3)c4ccc(cc4)Cl)C(F)(F)F 2K-052 c1cc(c(cc1Cl)Cl)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 2K-053 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)F)Sc3c(cc(cn3)C(F)(F)F)Cl 2K-054 c1ccc2c(c1)nc(c3n2c(nn3)N)C(F)(F)F 2K-055 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)OC 2K-056 c1ccc2c(c1)nc(c(n2)NNC(=O)c3ccc(cc3)Cl)C(F)(F)F 2K-057 CN(C)C(=C(C#N)C#N)C/C=N/Nc1c(cc(cn1)C(F)(F)F)Cl 2K-058 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)OC(F)(F)F 2K-059 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)OC(F)(F)F 2K-060 COc1ccnc(c1C#N)Oc2ccc(cc2)Cl 2K-061 c1ccc2c(c1)nc(c(n2)N/N=C/c3cccn3c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 2K-062 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 2K-063 CN(C)C(=C(C#N)C#N)/C=C/Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F 2K-064 c1cc2nnc(n2c3c1c(cc(n3)C(F)(F)F)C(F)(F)F)N 2K-065 CCOC(=O)CN/C=C/C(=C(C#N)C#N)N(C)C 2K-066 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2K-067 c1ccc(cc1)Oc2c(nc3ccccc3n2)C(F)(F)F 2K-068 c1ccc2c(c1)nc(c(n2)Oc3ccc(cc3)F)C(F)(F)F 2K-069 CC(C)(C)c1ccc(cc1)Oc2c(nc3ccccc3n2)C(F)(F)F 2K-070 CCOC(=O)c1c(c2c(ccnc2s1)OC)N 2K-071 COc1ccc(cc1)Oc2c(nc3ccccc3n2)C(F)(F)F 2K-072 Cc1cc(cc(c1)Oc2c(nc3ccccc3n2)C(F)(F)F)C 2K-073 Cc1cc(ccc1Oc2c(nc3ccccc3n2)C(F)(F)F)Cl 2K-074 c1ccc2c(c1)nc(c(n2)Sc3ccccc3Cl)C(F)(F)F 2K-075 c1ccc2c(c1)nc(c(n2)Sc3cccc(c3)C(F)(F)F)C(F)(F)F 2K-076 c1ccc2c(c1)nc(c(n2)Oc3cccc(c3)Cl)C(F)(F)F 2K-077 c1ccc2c(c1)nc(c(n2)Oc3ccc(cc3)C#N)C(F)(F)F 2K-078 COc1ccnc(c1C#N)Sc2ccc(cc2)Cl 2K-079 c1c(cnc(c1Cl)CCC(=O)N)C(F)(F)F 2K-080 CN(C)C(=C(C#N)C#N)C/C=N/OCc1c(cccc1Cl)F 2K-081 CN(C)C(=C(C#N)C#N)C/C=N/OCc1ccc(cc1Cl)Cl 2K-082 CN(C)S(=O)(=O)c1ccc(cc1)n2cccc2 2K-083 Cc1cccc(c1)C(C#N)c2c(nc3ccccc3n2)C(F)(F)F 2K-084 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)S(=O)(=O)N(C)C 2K-085 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)C#N 2K-086 c1ccn(c1)c2nnc3n2cc(cc3Cl)C(F)(F)F 2K-087 CN(C)c1ccnc(c1C#N)Nn2cnnc2 2K-088 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)Oc2ccccc2 2K-089 COc1ccnc(c1C(=N)NNC(=O)c2ccc(cc2Cl)Cl)N 2K-090 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)Oc3ccccc3 2K-091 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1Cl)Cl 2K-092 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2Cl)Cl 2K-093 CN(C)c1ccnc(c1C#N)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F 2K-094 CCOC(=O)CNC(=S)n1cnc(n1)N 2K-095 CN(C)C(=C(C#N)C#N)/C=C/Nc1c(cccc1F)F 2K-096 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)O 2K-097 CN(C)c1ccn2c3cccc(c3nc2c1C#N)F 2K-098 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)O 2K-099 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1F)F 2K-100 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2F)F 2K-101 CN(C)C(=C(C#N)C#N)/C=C/Nc1cc(ccc1OC)OC 2K-102 CCOC(=O)CNC(=S)n1c(ncn1)N 2K-103 CC(=O)c1ccccc1N/C=C/C(=C(C#N)C#N)N(C)C 2K-105 c1cc(ccc1/C=C\2/C(=O)N(C(=S)N2)c3ccc(cc3)F)Cl 2K-135 c1cc(c(cc1Cn2c3cc(c(cc3nc2c4ccc(=O)[nH]c4)Cl)Cl)Cl)Cl 2K-301S c1cc(c(cc1Cl)Cl)Cn2c3cc(c(cc3nc2c4ccc(=O)[nH]c4)Cl)Cl 2K-302S c1cc(cc(c1)C(F)(F)F)Cn2c3cc(c(cc3nc2c4ccc(nc4)Cl)Cl)Cl 2K-303S c1ccc(cc1)Cn2c3cc(c(cc3nc2c4ccc(nc4)Cl)Cl)Cl 2K-304S c1cc(sc1)c2cc(c(c(=O)[nH]2)C#N)C(F)(F)F 2K-305S Cn1c(c(c(n1)C(F)(F)F)C#N)N(C)NS(=O)(=O)C 2K-307S Cn1c(c(c(n1)C(F)(F)F)C#N)N(C)NS(=O)(=O)c2ccccc2 2K-308S Cc1cc(c(c(=O)[nH]1)C#N)C(F)(F)F 2K-309S c1ccc(cc1)Cn2c3cc(c(cc3nc2c4ccc(=O)[nH]c4)Cl)Cl 2K-311S c1cc(cc(c1)C(F)(F)F)Cn2c3cc(c(cc3nc2c4ccc(=O)[nH]c4)Cl)Cl 2K-312S CCc1ccccc1S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C 2K-313S Cc1ccccc1Cn2c3cc(c(cc3nc2c4ccc(=O)[nH]c4)Cl)Cl 2K-314S c1ccc(c(c1)Cn2c3cc(c(cc3nc2c4ccc(=O)[nH]c4)Cl)Cl)Cl 2K-315S Cc1cc(c(c(=O)n1C)C#N)C(F)(F)F 2K-318S Cn1c2cc(c(cc2nc1c3ccc(=O)[nH]c3)Cl)Cl 2K-320S c1cc(=O)[nH]cc1c2[nH]c3cc(c(cc3n2)Cl)Cl 2K-321S c1cc(c(=O)[nH]c1)c2nc3cc(c(cc3n2Cc4ccc(cc4)Cl)Cl)Cl 2K-322S c1ccc(c(c1)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl)Cl 2K-323S Cc1ccccc1Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 2K-324S CCOC(=O)Cn1c2ccccc2ncc1=O 2K-329S Cc1cccc(c1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 2K-331S c1cc(c(nc1)Cl)c2nc3cc(c(cc3n2Cc4ccc(cc4)F)Cl)Cl 2K-332S c1cc(cc(c1)F)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 2K-333S c1cc(c(c(c1)Cl)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl)F 2K-334S c1cc(c(=O)[nH]c1)c2nc3cc(c(cc3n2Cc4ccc(c(c4)Cl)Cl)Cl)Cl 2K-335S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2C)Cl)Cl)C 2K-337S Cc1ccc(cc1S(=O)(=O)c2c(cc(nc2Cl)C)C)Cl 2K-338S CCCCc1cc(c(c(n1)OCC(C)C)S(=O)(=O)c2ccccc2C)C 2K-339S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2C)Cl)OCC(C)C)C 2K-340S Cc1ccc(cc1S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C)Cl 2K-341S c1ccc(c(c1)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl)F 2K-342S c1cc(cc(c1)Cl)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl 2K-343S CCn1c2cc(c(cc2nc1c3cccnc3Cl)Cl)Cl 2K-344S Cn1c2cc(c(cc2nc1c3cccnc3Cl)Cl)Cl 2K-345S c1cc(c(c(c1)Cl)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl)Cl 2K-351S c1cc(c(nc1)Cl)c2nc3cc(c(cc3n2Cc4ccc(cc4Cl)Cl)Cl)Cl 2K-352S c1cc(cc(c1)F)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl 2K-353S c1cc(c(=O)[nH]c1)c2nc3cc(c(cc3n2Cc4ccc(cc4)F)Cl)Cl 2K-354S Cc1ccccc1Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl 2K-356S CC(C)(C)c1ccc(cc1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 2K-360S Cc1ccc(cc1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 2K-361S CCCn1c2cc(c(cc2nc1c3cccnc3Cl)Cl)Cl 2K-362S C#CCn1c2cc(c(cc2nc1c3cccnc3Cl)Cl)Cl 2K-363S COc1ccc(cc1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)Cl)Cl 2K-364S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccc(cc4)OC 2K-365S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Cl)C)C 2K-366S Cc1cc(nc(c1S(=O)(=O)c2ccccc2Cl)Cl)C 2K-367S Cc1ccccc1S(=O)(=O)c2c(cc(nc2Oc3ccccc3)C)C 2K-368S Cc1ccccc1S(=O)(=O)c2c(cc(nc2N(C)C)C)C 2K-369S c1ccc2c(c1)[nH]c(n2)c3ccc[nH]c3=O 2K-370S c1cc(c(c(c1)Cl)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl)Cl 2K-371S Cn1c(cc(nc1=O)C(=O)Nc2cccc(c2)C(F)(F)F)O 2K-507S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2Cl)Cl)O 2K-508S c1cc(ccc1S(=O)(=O)CC#N)Cl 2K-509S COc1c(cc(c(n1)N)S(=O)(=O)c2ccccc2)C#N 2K-512S Cc1ccc(cc1)S(=O)(=O)c2cc(c(nc2N)OC)C#N 2K-514S COc1c(cc(c(n1)N)S(=O)(=O)c2ccc(cc2)Cl)C#N 2K-515S COc1c(cc(c(n1)N)S(=O)(=O)c2ccc(cc2)F)C#N 2K-516S COc1c(cc(c(n1)N)S(=O)(=O)c2cccc(c2)C(F)(F)F)C#N 2K-517S Cc1ccccc1S(=O)(=O)c2cc(c(nc2N)OC)C#N 2K-524S c1ccc(cc1)S(=O)(=O)c2cc(c(nc2N)O)C#N 2K-525S Cn1c(c(c(n1)c2ccccc2)C=O)Cl 2K-535S Cc1ccc(cc1)S(=O)(=O)c2cc(c(nc2N)O)C#N 2K-536S c1cc(ccc1S(=O)(=O)c2cc(c(nc2N)O)C#N)Cl 2K-537S c1cc(ccc1F)S(=O)(=O)c2cc(c(nc2N)O)C#N 2K-538S c1cc(cc(c1)S(=O)(=O)c2cc(c(nc2N)O)C#N)C(F)(F)F 2K-539S Cc1ccccc1S(=O)(=O)c2cc(c(nc2N)O)C#N 2K-540S Cn1c(c(c(n1)c2ccccc2)CO)Cl 2K-541S Cn1c(c(c(n1)c2ccccc2)CCl)Cl 2K-544S Cc1cc(nc(n1)c2ccccc2)O 2K-547S Cc1cc(nc(n1)c2cccnc2)O 2K-548S Cc1cc(nc(n1)c2ccncc2)O 2K-567S c1cc(c(cc1Cl)Cl)c2nc3c(cc(cc3Cl)Cl)c(=O)n2O 2K-571S Cc1ccc(cc1)c2nc3c(cc(cc3Cl)Cl)c(=O)n2O 2K-573S c1cc(ccc1c2nc3c(cc(cc3Cl)Cl)c(=O)n2O)[N+](=O)[O-] 2K-577S Cn1c2ccccc2nc(c1=O)Cl 2K-579S Cn1c2ccccc2nc(c1=O)Oc3ccc(c(c3)Cl)Cl 2K-580S Cn1c2ccccc2nc(c1=O)Oc3ccc(cc3F)F 2K-581S CNc1c(=O)n(c2ccccc2n1)C 2K-582S Cn1c2ccccc2nc(c1=O)N(C)C 2K-583S Cn1c2ccccc2nc(c1=O)Oc3cc(cc(c3)Cl)Cl 2K-584S Cn1c2ccccc2nc(c1=O)Oc3ccc(cc3)Cl 2K-585S Cc1ccc(cc1)Oc2c(=O)n(c3ccccc3n2)C 2K-586S Cn1c2ccccc2nc(c1=O)Oc3ccc(cc3)OC 2K-587S Cn1c2ccccc2nc(c1=O)Oc3cccc(c3)C(F)(F)F 2K-588S c1ccc(c(c1)c2nc3ccc(cc3c(=O)n2O)Br)Cl 2K-594S c1cc(cc(c1)Cl)c2nc3ccc(cc3c(=O)n2O)Br 2K-595S c1cc(ccc1c2nc3ccc(cc3c(=O)n2O)Br)Cl 2K-596S Cc1ccccc1c2nc3ccc(cc3c(=O)n2O)Br 2K-597S Cn1c(c(c(n1)c2ccccc2)CSc3ccc(cc3)Cl)Cl 2K-598s Cn1c(c(c(n1)c2ccccc2)C=O)Sc3ccccc3C(=O)OC 2K-599S c1cc(ccc1C#N)c2nc3ccc(cc3c(=O)n2O)Br 2K-602S c1cc(ccc1c2nc3ccc(cc3c(=O)n2O)Br)[N+](=O)[O-] 2K-603S Cn1c(cc(nc1=O)C(=O)Nc2cc(ccc2Cl)Cl)O 2K-604S Cn1c(cc(nc1=O)C(=O)Nc2cccc(c2Cl)Cl)O 2K-605S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2)Cl)O 2K-608S Cn1c(cc(n1)c2ccc(c(c2)Cl)Cl)N 2K-611S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2)C(F)(F)F)O 2K-613S Cc1cc(ccc1NC(=O)c2cc(n(c(=O)n2)C)O)Cl 2K-615S Cc1ccc(cc1NC(=O)c2cc(n(c(=O)n2)C)O)Cl 2K-616S Cn1c(cc(nc1=O)C(=O)Nc2ccc(c(c2F)Cl)F)O 2K-617S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2C(F)(F)F)Cl)O 2K-618S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2F)F)O 2K-620S Cn1c(cc(nc1=O)C(=O)Nc2ccc(c(c2)F)F)O 2K-621S Cn1c(cc(nc1=O)C(=O)Nc2ccccc2Br)O 2K-622S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2)Br)O 2K-623S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2)OC(F)(F)F)O 2K-624S Cn1c(cc(nc1=O)C(=O)Nc2ccccc2C(F)(F)F)O 2K-625S Cn1c(cc(nc1=O)C(=O)Nc2ccc(c(c2)Cl)Cl)O 2K-627S Cn1c(cc(nc1=O)C(=O)Nc2ccccc2Cl)O 2K-628S Cn1c(cc(nc1=O)C(=O)Nc2cccc(c2)Cl)O 2K-629S Cn1c(cc(nc1=O)C(=O)Nc2ccccc2F)O 2K-630S Cn1c(cc(nc1=O)C(=O)Nc2ccc(cc2)F)O 2K-631S Cc1ccc(cc1C)NC(=O)c2cc(n(c(=O)n2)C)O 2K-634S CC(CS(=O)(=O)c1ccc(cc1)Br)(c2ccccc2)O 2K-635S Cn1c(cc(nc1=O)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)O 2K-637S Cn1c(cc(nc1=O)C(=O)Nc2ccccc2C(=O)OC)O 2K-638S CCc1cccc(c1NC(=O)c2cc(n(c(=O)n2)C)O)CC 2K-639S CC(CS(=O)(=O)c1ccc(cc1)Cl)(c2ccccc2)O 2K-640S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)O)O 2K-641S COc1ccccc1c2nc3ccccc3c(=O)n2O 2K-642S CC(CS(=O)(=O)c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 2K-645S c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)Nc4cccc(c4)C(F)(F)F 2K-900 CN1C(CC(O1)C(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl)c3ccc(cc3)OC 2K-901 c1csc(c1Cl)c2c[nH]c(c2C#N)N 2K-902 Cc1cc(n2cc(c(c2n1)C(=O)N(C)C)c3c(ccs3)Cl)C 2K-903 c1cc(c(nc1)Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3Cl)Cl 2K-905 c1c(cnc(c1Cl)NC(=S)/N=C/NO)C(F)(F)F 2K-906 CON/C=N/C(=S)Nc1c(cc(cn1)C(F)(F)F)Cl 2K-907 c1cc(cc(c1)C(F)(F)F)CON/C=N/C(=S)Nc2c(cc(cn2)C(F)(F)F)Cl 2K-908 c1c(cnc(c1Cl)NC(=S)/N=C/NOCc2c(snn2)Cl)C(F)(F)F 2K-909 c1c(cnc(c1Cl)NC(=S)/N=C/NOCC(=O)N2CCOCC2)C(F)(F)F 2K-910 CN(/C=N/C(=S)Nc1c(cc(cn1)C(F)(F)F)Cl)O 2K-911 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)C2CC(=NO2)c3c(cccc3Cl)Cl 2K-912 Cc1c(cc(c(=O)n1CC=C)NC(=O)c2ccccc2)C(=O)C 2K-913 Cc1c(cc(c(=O)n1Cc2ccc(cc2)Cl)NC(=O)c3ccc(cc3)Cl)C(=O)C 2K-914 c1cc(c(c(c1)Cl)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl 2K-915 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)c3cccc(c3C2=O)O 2K-916 Cc1c(cc(c(=O)n1Cc2ccc(cc2Cl)Cl)NC(=O)c3cccc(c3)Cl)C(=O)C 2K-917 Cc1c(cc(c(=O)n1CCCOC)NC(=O)c2ccccc2)C(=O)C 2K-918 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C(C2=O)ON=C3c4c(cccc4Cl)Cl 2K-919 CC(c1ccnc2n1ncn2)Oc3cccc(c3)Cl 2L-001 Cc1ccc(cc1)C(=O)N(CCN(Cc2cccc(c2)Cl)C(=O)c3ccc(cc3)C)Cc4cccc(c4)Cl 2L-002 CC(c1ccnc2n1nc(n2)/N=C/N(C)C)Oc3cccc(c3)Cl 2L-003 CC(c1ccnc2n1nc(n2)N/C=N/OC)Oc3cccc(c3)Cl 2L-004 c1cc(ccc1c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl)F 2L-005 c1cc(cc(c1)Cl)CN(CCN(Cc2cccc(c2)Cl)S(=O)(=O)c3ccc(cc3)Cl)S(=O)(=O)c4ccc(cc4)Cl 2L-006 COc1ccc(cc1)S(=O)(=O)N(CCN(Cc2cccc(c2)Cl)S(=O)(=O)c3ccc(cc3)OC)Cc4cccc(c4)Cl 2L-007 c1cc(ccc1c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl)[N+](=O)[O-] 2L-009 c1cc(ccc1/C=C\c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl)Cl 2L-010 COc1ccc(cc1)c2cnc3nc(nn3c2N)Sc4c(cc(cn4)C(F)(F)F)Cl 2L-011 c1ccc(cc1)Oc2ccc(cc2)c3ccnc4n3nc(n4)Sc5c(cc(cn5)C(F)(F)F)Cl 2L-012 c1cc(sc1)CN(CCN(Cc2cccs2)C(=O)Nc3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)Cl 2L-013 COc1ccc(cc1)c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 2L-014 Cc1ccc(cc1)c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 2L-015 c1ccc(cc1)c2ccnc3n2nc(n3)Sc4c(cc(cn4)C(F)(F)F)Cl 2L-016 Cc1ccc(cc1)C(=O)N(CCN(Cc2cccs2)C(=O)c3ccc(cc3)C)Cc4cccs4 2L-017 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/c2nnc(s2)N 2L-018 CN(C)/C=N/c1nnc(s1)/C(=C/c2ccc(cc2Cl)Cl)/C#N 2L-019 c1cc(ccc1CC(=S)N2CCOCC2)Cl 2L-020 Cc1c(cccc1Cl)N/C=C\2/C(=C(NC2=O)C)C(=O)OC 2L-021 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)OC(F)(F)F 2L-022 COc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2L-023 Cc1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)C 2L-025 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl 2L-026 CSc1cccc(c1)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2L-027 CO/N=C/Nc1nnc(s1)/C(=C/c2ccc(cc2Cl)Cl)/C#N 2L-028 c1ccc(cc1)NS(=O)(=O)c2ccc(s2)CCc3c(cc(cn3)C(F)(F)F)Cl 2L-029 CC(C(=O)C)Oc1ccccc1O 2L-030 Cc1cccc(c1C)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2L-032 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Br 2L-033 Cc1cc(ccc1NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl 2L-034 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Nc3ccc(cc3F)F 2L-035 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 2L-036 c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2L-037 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Nc3c(c(c(c(c3F)F)F)F)F 2L-038 CCOC(=O)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2L-039 CC(C)NS(=O)(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 2L-040 CCCNS(=O)(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 2L-041 CC(C)(C)NS(=O)(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 2L-042 Cc1ccc(cc1)CN(CCN(Cc2ccc(cc2)C)C(=O)c3ccccc3Cl)C(=O)c4ccccc4Cl 2L-044 COc1ccc(cc1)/C=C(\C#N)/c2nnc(s2)N 2L-045 CC(C)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2L-046 CN(C)/C=N/c1nnc(s1)/C(=C/c2ccc(cc2)OC)/C#N 2L-047 COc1ccc(cc1)/C=C(\C#N)/c2nnc(s2)N/C=N/OC 2L-050 Cc1c(c(ns1)Sc2c(cc(cn2)C(F)(F)F)Cl)C#N 2L-051 COc1ccccc1Oc2c(cccn2)C(=O)NC3CCSC3=O 2L-301S c1cc(c(nc1)Oc2ccc(cc2)F)C(=O)NC3CCSC3=O 2L-302S Cc1ccccc1C(=O)NC=C2C(=O)OC(OC2=O)(C)C 2L-303S CC1(OC(=O)C(=CNC(=O)c2ccccc2Cl)C(=O)O1)C 2L-304S CC1(OC(=O)C(=CNC(=O)c2ccc(cc2Cl)Cl)C(=O)O1)C 2L-305S CC1(OC(=O)C(=CNC(=O)c2ccc(c(c2)Cl)Cl)C(=O)O1)C 2L-306S CC1(OC(=O)C(=CNC(=O)c2cccc(c2)Cl)C(=O)O1)C 2L-307S CC1(OC(=O)C(=CNC(=O)c2ccc(cc2)Cl)C(=O)O1)C 2L-308S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/NOCc3cccc(c3Cl)Cl 2L-309S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/NOCc3ccc(cc3)F 2L-311S Cc1ccc(cc1)CON/C=C/c2c(nnc(n2)SCc3ccc(cc3)Cl)C 2L-312S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/NOCc3cccc(c3)F 2L-313S Cc1c(nc(nn1)SC)/C=C/NOCc2cccc(c2Cl)Cl 2L-314S Cc1c(nc(nn1)SCc2ccccc2)/C=C/NOCc3cccc(c3Cl)Cl 2L-315S Cc1c(nc(nn1)SCc2ccc(cc2)Cl)/C=C/NOCc3ccc(cc3)C(C)(C)C 2L-317S Cc1c(nc(nn1)SC)/C=C/NOCc2cccc(c2)F 2L-318S CC1(OC(=O)C(=CNC(=O)c2c(cccc2F)F)C(=O)O1)C 2L-320S CC1(OC(=O)C(=CNC(=O)c2ccc(cc2)F)C(=O)O1)C 2L-321S CC(C)CCOC(=O)N/C=C/c1ccco1 2L-322S C=CCOC(=O)N/C=C/c1ccco1 2L-323S CCOCCOC(=O)N/C=C/c1ccco1 2L-324S CC(C)(C)COC(=O)N/C=C/c1ccco1 2L-325S CC1(OC(=O)C(=CNC(=O)c2cccc(c2)C(F)(F)F)C(=O)O1)C 2L-326S CC1(OC(=O)C(=CNC(=O)c2cccc(c2)OC)C(=O)O1)C 2L-327S CC1(OC(=O)C(=CNC(=O)c2cc(cc(c2)Cl)Cl)C(=O)O1)C 2L-329S CCC(=O)NC=C1C(=O)OC(OC1=O)(C)C 2L-330S CC1(OC(=O)C(=CNC(=O)C(C)(C)C)C(=O)O1)C 2L-331S CCCCC(=O)NC=C1C(=O)OC(OC1=O)(C)C 2L-332S c1cc(oc1)/C=C/NC(=O)OCC(Cl)(Cl)Cl 2L-333S C#CCOC(=O)N/C=C/c1ccco1 2L-334S c1cc(oc1)/C=C/NC(=O)OCCCl 2L-335S c1ccc(cc1)COC(=O)N/C=C/c2ccco2 2L-336S c1ccc(c(c1)C#N)Sc2ccccc2C(=O)Nc3ccc(cc3)Cl 2L-337S c1ccc(c(c1)C#N)Sc2ccccc2C(=O)Nc3cccc(c3)C(F)(F)F 2L-340S COc1ccc(cc1)NC(=O)c2ccccc2Sc3ccccc3C#N 2L-341S c1ccc(cc1)NC(=O)c2ccccc2Sc3ccccc3C#N 2L-342S CNC(=O)c1ccccc1Sc2ccccc2C#N 2L-343S c1ccc(c(c1)C#N)S(=O)c2ccccc2C(=O)Nc3ccc(cc3)Cl 2L-345S c1ccc(c(c1)C#N)S(=O)(=O)c2ccccc2C(=O)Nc3ccc(cc3)Cl 2L-346S c1ccc(cc1)C2=NC(=O)N=C2NC(=O)Nc3ccc(cc3)Cl 2L-347S COc1ccc(cc1)NC(=O)c2ccccc2S(=O)c3ccccc3C#N 2L-349S COc1ccc(cc1)NC(=O)c2ccccc2S(=O)(=O)c3ccccc3C#N 2L-350S CNC(=O)c1ccccc1S(=O)c2ccccc2C#N 2L-351S CNC(=O)c1ccccc1S(=O)(=O)c2ccccc2C#N 2L-352S c1cc(oc1)/C=C/NC(=O)OCc2ccc(cc2)Cl 2L-353S COc1ccc(cc1)COC(=O)N/C=C/c2ccco2 2L-354S c1cc(c(c(c1)Cl)COC(=O)N/C=C/c2ccco2)Cl 2L-355S c1cc(oc1)/C=C/NC(=O)OCc2ccc(cc2Cl)Cl 2L-356S c1ccc(c(c1)C#N)S(=O)c2ccccc2C(=O)Nc3cccc(c3)C(F)(F)F 2L-357S c1ccc(cc1)NC(=O)c2ccccc2S(=O)c3ccccc3C#N 2L-358S C=CCNC(=O)c1ccccc1Sc2ccccc2C#N 2L-359S CC(C)NC(=O)c1ccccc1Sc2ccccc2C#N 2L-360S c1cc(oc1)/C=C/NC(=O)OCc2ccc(cc2)Br 2L-361S c1cc(oc1)/C=C/NC(=O)OCc2ccc(cc2)C(F)(F)F 2L-362S c1cc(cc(c1)Cl)COC(=O)N/C=C/c2ccco2 2L-363S CC(C)NC(=O)c1ccccc1S(=O)c2ccccc2C#N 2L-364S CC(C)NC(=O)c1ccccc1S(=O)(=O)c2ccccc2C#N 2L-365S COc1ccccc1COC(=O)N/C=C/c2ccco2 2L-366S c1ccc(c(c1)COC(=O)N/C=C/c2ccco2)Cl 2L-367S CC(C)(C)c1ccc(cc1)COC(=O)N/C=C/c2ccco2 2L-368S CC(C)CC(=O)NC=C1C(=O)OC(OC1=O)(C)C 2L-369S CC1(OC(=O)C(=CNC(=O)C2CC2)C(=O)O1)C 2L-370S CC1(OC(=O)C(=CNC(=O)c2cccnc2Cl)C(=O)O1)C 2L-371S CCCC(=O)NC=C1C(=O)OC(OC1=O)(C)C 2L-372S CC1(OC(=O)C(=CNC(=O)c2ccc(cc2)C(F)(F)F)C(=O)O1)C 2L-373S CC1(OC(=O)C(=CNC(=O)c2ccc(cc2)OC)C(=O)O1)C 2L-374S c1cc(c(nc1)Cl)CO 2L-375S c1cc(c(nc1)Cl)C=O 2L-376S Cc1ccc(cc1)Sc2c(cccn2)C=O 2L-377S Cc1ccc(cc1)Sc2c(cccn2)/C=N/O 2L-378S C=CCNC(=O)c1ccccc1S(=O)c2ccccc2C#N 2L-379S Cc1ccc(cc1)CO/N=C/c2cccnc2Sc3ccc(cc3)C 2L-381S Cc1ccc(cc1)Sc2c(cccn2)/C=N/OCc3cccc(c3)F 2L-382S COC(=O)c1ccccc1S(=O)(=O)NNC(=O)Nc2ccccc2 2L-383S c1ccc(cc1)NC(=O)c2ccccc2S(=O)(=O)c3ccccc3C#N 2L-385S Cc1ccc(cc1)SC(CC(=O)c2ccccc2)C(=O)c3ccccc3 2L-388S COc1ccc(cc1)SC(CC(=O)c2ccccc2)C(=O)c3ccccc3 2L-389S COC(=O)c1ccc(cc1)NS(=O)(=O)c2ccccc2 2L-390S c1ccc(c(c1)C#N)S(=O)(=O)c2ccccc2C(=O)Nc3cccc(c3)C(F)(F)F 2L-391S c1cc(ccc1S(=O)(=O)NC(=O)CCCC(=O)O)Cl 2L-501S Cc1cccc(c1)CC(=O)NCCSc2ccc(cc2)Cl 2L-502S Cc1ccc(cc1)SCCNC(=O)Cc2ccc(cc2)Cl 2L-503S Cc1ccc(cc1)SCCNC(=O)Cc2ccccc2 2L-504S Cc1ccc(cc1)CC(=O)NCCSc2ccc(cc2)C 2L-505S Cc1ccc(cc1)S(=O)CCNC(=O)Cc2ccc(cc2)Cl 2L-510S Cc1ccc(cc1)CC(=O)NCCS(=O)(=O)c2ccc(cc2)C 2L-512S Cc1ccc(cc1)CC(=O)NCCS(=O)c2ccc(cc2)C 2L-513S Cc1ccc(cc1)S(=O)CCNC(=O)Cc2ccccc2 2L-514S Cc1ccc(cc1)S(=O)(=O)CCNC(=O)Cc2ccccc2 2L-515S Cc1ccc(cc1)S(=O)(=O)CCNC(=O)Cc2ccc(cc2)Cl 2L-521S Cc1ccc(cc1)c2cc\3c(nn2)-c4ccccc4/C3=N/OC 2L-523S Cc1ccc(cc1)c2cc\3c(nn2)-c4ccccc4/C3=N/OCc5ccc(cc5)C(C)(C)C 2L-524S Cc1ccc(cc1)CO/N=C\2/c3ccccc3-c4c2cc(nn4)c5ccc(cc5)C 2L-526S Cc1ccc(cc1)c2cc\3c(nn2)-c4ccccc4/C3=N/O 2L-527S Cc1cccc(c1)CC(=O)NCCS(=O)c2ccc(cc2)Cl 2L-532S c1cc(ccc1CC(=O)NCCSc2ccc(cc2)Br)Cl 2L-534S Cc1ccc(cc1)CC(=O)NCCSc2ccc(cc2)Br 2L-535S c1ccc(cc1)CC(=O)NCCSc2ccc(cc2)Br 2L-536S c1cc(ccc1SCCNC(=O)Cc2ccc(c(c2)Cl)Cl)Br 2L-537S CSCc1cc(nc(n1)c2ccccn2)O 2L-539S Cc1nc(cc(n1)O)CSC 2L-540S Cc1ccc(cc1)c2cc\3c(nn2)-c4ccccc4/C3=N/OCc5ccc(cc5Cl)Cl 2L-544S c1ccc(cc1)CC(=O)NCCSc2ccccc2 2L-548S c1ccc(cc1)SCCNC(=O)Cc2ccc(cc2)Cl 2L-549S c1ccc(cc1)SCCNC(=O)Cc2ccc(c(c2)Cl)Cl 2L-550S Cc1ccc(cc1)CC(=O)NCCSc2ccccc2 2L-551S c1ccc(cc1)C(=O)c2c[nH]cc2c3ccc(cc3)Cl 2L-552S c1cc(ccc1CC(=O)NCCS(=O)c2ccc(cc2)Br)Cl 2L-554S c1cc(ccc1CC(=O)NCCS(=O)(=O)c2ccc(cc2)Cl)Cl 2L-555S Cc1ccc(cc1)CC(=O)NCCS(=O)c2ccc(cc2)Br 2L-556S Cc1ccc(cc1)CC(=O)NCCS(=O)(=O)c2ccc(cc2)Br 2L-557S c1cc(ccc1S(=O)CCNC(=O)Cc2ccc(c(c2)Cl)Cl)Br 2L-558S CSCc1cc(nc(n1)c2ccccc2)Sc3ccccc3 2L-559S CSCc1cc(nc(n1)c2ccccc2)Sc3cccc(c3)C(F)(F)F 2L-560S COc1cc(nc(n1)c2ccccc2)CSC 2L-561S Cc1ccc(cc1)S(=O)(=O)NC(=O)CCCC(=O)O 2L-562S CSCc1cc(nc(n1)c2ccccc2)Oc3ccccc3 2L-564S CSCc1cc(nc(n1)c2ccccn2)Oc3ccccc3 2L-565S c1cc(ccc1C(=O)c2c[nH]cc2c3ccc(cc3Cl)Cl)Cl 2L-566S c1cc(c(c(c1)Cl)c2c[nH]cc2C(=O)c3ccc(cc3)Cl)F 2L-567S CCOC(=O)CSc1cc(nc(n1)c2ccccc2)CSC 2L-569S CSCc1cc(nc(n1)c2ccccn2)Sc3ccccc3 2L-570S CCOC(=O)CSc1cc(nc(n1)c2ccccn2)CSC 2L-571S CSCc1cc(nc(n1)c2ccccc2)N3CCOCC3 2L-575S c1cc(c(c(c1)Cl)c2c[nH]cc2C(=O)c3ccc(cc3)Cl)Cl 2L-578S Cc1ccc(cc1)c2c[nH]cc2C(=O)c3ccc(cc3)Cl 2L-579S c1cc(cc(c1)Br)c2c[nH]cc2C(=O)c3ccc(cc3)Cl 2L-580S c1cc(ccc1c2c[nH]cc2C(=O)c3ccc(cc3)Cl)Br 2L-581S c1cc(c(c(c1)Cl)Cl)c2c[nH]cc2C(=O)c3ccc(cc3)Cl 2L-582S c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Cl)Br 2L-583S Cc1ccc(cc1)/C=C/C(=O)c2ccc(c(c2)OC)OC 2L-585S Cc1c(c(on1)C)C(=O)N2CCN(CC2)Cc3ccccc3 2L-587S CSCc1cc(nc(n1)c2ccccn2)N3CCOCC3 2L-589S c1cc(ccc1NC(=O)OC(CC#N)CNc2c(cc(cn2)C(F)(F)F)Cl)Cl 2L-900 Cn1c(=O)c(nn(c1=O)c2ccc(cc2)C(F)(F)F)c3ccn(n3)c4ccccc4 2L-901 Cc1cc(=O)n(c(n1)/N=C/NOCc2ccc(cc2)[N+](=O)[O-])C 2L-902 C=CCn1cc(c(=O)[nH]c1=O)C#N 2L-903 Cn1c(=O)c(cn(c1=O)CC=C)C#N 2L-904 CN(CCO)c1cnn(c(=O)c1Cl)c2c(cc(cn2)C(F)(F)F)Cl 2L-905 c1c(cnc(c1Cl)n2c(=O)c(c(cn2)ON3C(=O)CCC3=O)Cl)C(F)(F)F 2L-906 c1cc(c(c(c1)F)C(=O)OC(CC#N)CNc2c(cc(cn2)C(F)(F)F)Cl)F 2L-907 Cn1c(=O)c(cn(c1=O)CC2CC(N(O2)C)c3ccc(cc3)OC)C#N 2L-908 c1c(cnc(c1Cl)n2c(=O)c(c(cn2)N3CCNCC3)Cl)C(F)(F)F 2L-909 C=CCC1(CCN(CC1)c2ccc(cc2)[N+](=O)[O-])C#N 2L-910 CCOC(=O)C1=NOC(C1)Cn2cc(c(=O)n(c2=O)C)C#N 2L-911 CCOC(=O)NC(=O)/C(=C/N1CCN(CC1)c2cnn(c(=O)c2Cl)c3c(cc(cn3)C(F)(F)F)Cl)/C#N 2L-912 Cn1c(=O)c(cn(c1=O)CC2CC(=NO2)C(=O)NCCOC)C#N 2L-913 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cccc2 2L-914 CN(CCOC(=O)c1c(cccc1F)F)c2cnn(c(=O)c2Cl)c3c(cc(cn3)C(F)(F)F)Cl 2L-915 Cc1cc(=O)[nH]c(n1)/N=C/N(C)C 2L-916 Cc1cc(=O)[nH]c(n1)/N=C/NOCc2c(cccc2Cl)F 2L-917 Cc1cc(=O)[nH]c(n1)/N=C/N(C)O 2L-918 Cc1cc(=O)n(c(n1)/N=C/N(C)C)Cc2ccc(cc2)F 2L-919 Cc1cc(=O)n(c(n1)/N=C/N(C)C)c2c(cc(cn2)C(F)(F)F)Cl 2L-920 c1ccc2c(c1)C(=O)N(C2=O)CCON3C(=O)c4ccccc4C3=O 2L-921 CCOc1cnc(o1)c2ccccc2F 2M-001 c1ccc(cc1)c2nc(cc(=O)s2)O 2M-002 COC(=O)C(C(=O)OC)Oc1ccc(cc1)Cl 2M-003 c1cc(ccc1c2nc(cc(=O)s2)O)Cl 2M-004 COC(=O)C(C(=O)OC)Oc1ccc(cc1Cl)Cl 2M-005 CC(C)c1ccc(cc1)c2nc(cc(=O)s2)O 2M-006 Cc1cccc(c1)CC(C(=O)OC)(C(=O)OC)Oc2ccc(cc2)Cl 2M-008 COc1ccc(cc1)OS(=O)(=O)c2ccc(s2)c3csnn3 2M-009 CC(C)(C)c1ccc(cc1)OS(=O)(=O)c2ccc(s2)c3csnn3 2M-012 c1cc(ccc1OS(=O)(=O)c2ccc(s2)c3csnn3)Cl 2M-013 c1cc(cc(c1)F)OS(=O)(=O)c2ccc(s2)c3csnn3 2M-014 CC(=O)Nc1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2M-015 CCOC(=O)CNC(=O)Cc1ccccc1 2M-016 CNc1ncc(s1)C(=O)/C=C/N(C)C 2M-017 CNc1ncc(s1)C(=O)C/C=N/OCc2ccc(cc2)Cl 2M-019 c1ccc(cc1)N/N=C(\C=O)/C(=O)c2cccs2 2M-021 CCOc1cnc(o1)Cc2ccccc2 2M-022 COc1ccc(cc1)N/N=C(\C=O)/C(=O)c2cccs2 2M-023 Cc1cc(cc(c1)OS(=O)(=O)c2ccc(s2)c3csnn3)C 2M-024 c1cc(c(cc1[N+](=O)[O-])Cl)OS(=O)(=O)c2ccc(s2)c3csnn3 2M-025 c1ccc(cc1)OS(=O)(=O)c2ccc(s2)c3csnn3 2M-026 CC(=O)Nc1cccc(c1)OS(=O)(=O)c2ccc(s2)c3csnn3 2M-027 COc1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2M-028 c1cc(sc1)C(=O)/C(=N/Nc2ccc(cc2)Cl)/C=O 2M-031 Cc1cccc(c1)N/N=C(/C=O)\C(=O)c2cccs2 2M-032 c1ccc(cc1)N/N=C(/C=O)\C(=O)c2ccco2 2M-033 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Oc3ccc(cc3)Cl 2M-034 c1cc(oc1)C(=O)/C(=N/Nc2ccc(cc2)Cl)/C=O 2M-035 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Oc3ccc(cc3Cl)Cl 2M-037 c1cc(ccc1[N+](=O)[O-])OS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 2M-038 Cc1cc(cc(c1)N/N=C(\C=O)/C(=O)c2ccc(cc2)OC)C 2M-039 COc1ccc(cc1)N/N=C(\C=O)/C(=O)c2ccco2 2M-041 CNc1ncc(s1)C(=O)C/C=N/OCc2c(cccc2Cl)Cl 2M-042 CNc1ncc(s1)C(=O)C/C=N/OCc2ccc(cc2)F 2M-043 Cc1cc(cc(c1)N/N=C(\C=N\N)/C(=O)c2ccc(cc2)OC)C 2M-044 Cc1cc(cc(c1)N/N=C/2\C=NN=C2c3ccc(cc3)OC)C 2M-045 Cc1ccc(cc1)C(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/C=O 2M-046 Cc1cccc(c1)N/N=C(\C=O)/C(=O)c2ccco2 2M-047 Cc1ccc(cc1)C(=O)/C(=N/Nc2cccc(c2C)C)/C=O 2M-048 c1cc(ccc1C(=O)/C(=N\Nc2ccc(cc2)Cl)/C=O)Cl 2M-049 Cc1ccc(cc1)C(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/C=N/N 2M-050 c1ccc(cc1)N/N=C(\C=O)/C(=O)c2ccc(cc2)Cl 2M-051 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)F)/C=O)Cl 2M-052 Cc1ccc(cc1)N/N=C(\C=O)/C(=O)c2ccc(cc2)Cl 2M-053 CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)Nc2ccc(c(c2)Cl)Cl 2M-301S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)Nc2ccc(cc2)Br 2M-302S Cc1ccc(cc1)CN/C(=N\c2ccccc2)/NCC(=O)O 2M-303S Cn1c2c(cc(s2)C(=O)Nc3cccc(c3)C(F)(F)F)c(n1)C(F)(F)F 2M-304S Cn1c2c(cc(s2)C(=O)Nc3ccc(cc3F)F)c(n1)C(F)(F)F 2M-305S Cn1c2c(cc(s2)C(=O)Nc3ccc(cc3)Cl)c(n1)C(F)(F)F 2M-306S c1cc(ncc1[N+](=O)[O-])S 2M-307S Cn1c2c(cc(s2)C(=O)N3CCN(CC3)C)c(n1)C(F)(F)F 2M-310S Cn1c2c(cc(s2)C(=O)NCC=C)c(n1)C(F)(F)F 2M-311S CCCNC(=O)c1cc2c(nn(c2s1)C)C(F)(F)F 2M-312S CC(C)NC(=O)c1cc2c(nn(c2s1)C)C(F)(F)F 2M-313S Cn1c2c(cc(s2)C(=O)N3CCOCC3)c(n1)C(F)(F)F 2M-314S Cc1ccc(cc1)CN/C(=N\c2ccccc2)/N3CCN(CC3)C 2M-318S c1ccc(cc1)NC(=S)NCc2cccc(c2)C(F)(F)F 2M-319S Cn1c2c(cc(s2)CO)c(n1)C(F)(F)F 2M-320S CS/C(=N/c1ccccc1)/NCc2cccc(c2)C(F)(F)F 2M-322S CCCN(CCC)/C(=N/c1ccccc1)/NCc2cccc(c2)C(F)(F)F 2M-323S CCCCN/C(=N/c1ccccc1)/NCc2cccc(c2)C(F)(F)F 2M-324S Cc1ccc(cc1)CN/C(=N\c2ccccc2)/NC3CCCCC3 2M-326S Cn1c2c(cc(s2)CBr)c(n1)C(F)(F)F 2M-331S Cc1ccc(cc1)SCc2cc3c(nn(c3s2)C)C(F)(F)F 2M-332S c1ccc(cc1)/N=C(\NCc2cccc(c2)C(F)(F)F)/NC3CC3 2M-333S C=CCN/C(=N/c1ccccc1)/NCc2cccc(c2)C(F)(F)F 2M-334S c1ccc(cc1)NC(=S)NCc2ccc(cc2)Cl 2M-336S c1ccc(cc1)NC(=S)NCc2ccc(cc2Cl)Cl 2M-337S C#CCN1c2ccccc2/C(=N\c3ccc(cc3)Cl)/C1=O 2M-338S COc1ccc(cc1)/N=C\2/c3ccccc3N(C2=O)CC#C 2M-339S Cc1cccc(c1)/N=C\2/c3ccccc3N(C2=O)CC#C 2M-340S c1ccc(c(c1)CN2c3ccccc3C(=O)C2=O)Cl 2M-341S COc1ccc(cc1)Sc2cc3ccccc3nc2c4ccc(cc4)Cl 2M-501S Cn1c2c(cc(s2)C(=O)Nc3ccc(cc3)OC)c(n1)C(F)(F)F 2M-505S Cn1c2c(cc(s2)C(=O)NC3CC3)c(n1)C(F)(F)F 2M-507S CNC(=O)c1c2ccccc2nc(c1Sc3ccc(cc3)Cl)c4ccc(cc4)Cl 2M-508S CN(C)C(=O)c1c2ccccc2nc(c1Sc3ccc(cc3)Cl)c4ccc(cc4)Cl 2M-509S c1ccc(cc1)c2c(c(c3ccccc3n2)C(=O)O)Sc4ccc(cc4)Br 2M-514S c1ccc2c(c1)c(c(c(n2)c3ccc(cc3Cl)Cl)Sc4ccc(cc4)Br)C(=O)O 2M-515S c1ccc(cc1)c2c(cc3ccccc3n2)Sc4ccc(cc4)Br 2M-516S COc1ccc(cc1)N(Cc2ccccc2)C(=O)c3ccc(nc3)Cl 2M-517S COc1ccc(cc1)N(Cc2ccccc2)C(=O)c3cccc(c3)OC 2M-518S COc1ccc(cc1)N(Cc2ccccc2)C(=O)c3ccc(cc3)F 2M-519S COc1ccc(cc1)N(Cc2ccccc2)C(=O)c3cccc(c3)C(F)(F)F 2M-520S c1ccc2c(c1)cc(c(n2)c3ccc(cc3Cl)Cl)Sc4ccc(cc4)Br 2M-522S Cc1ccc(cc1)C(=O)N2CCN3C2(c4ccccc4C3=O)c5ccc(cc5)Cl 2M-523S c1ccc2c(c1)C(=O)N3C2(N(CC3)C(=O)c4ccc(cc4)F)c5ccc(cc5)Cl 2M-524S COc1ccc(cc1)N(Cc2ccccc2)C(=O)c3ccc(cc3)Br 2M-525S CSc1c(c2cc(ccc2nc1c3ccccc3)Cl)C(=O)O 2M-527S c1cc(ccc1c2c(c(c3cc(ccc3n2)Cl)C(=O)O)Sc4ccc(cc4)Cl)Cl 2M-528S COc1ccc(cc1)N(Cc2ccccc2)C(=O)c3ccc(c(c3)Cl)Cl 2M-530S c1cc(cc(c1)C(F)(F)F)c2cc(on2)C(=O)CBr 2M-532S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)CBr 2M-533S COC(=O)c1ccccc1S(=O)C/C(=N/OC)/c2ccc(cc2Cl)Cl 2M-534S COC(=O)c1ccccc1S(=O)(=O)C/C(=N/OC)/c2ccc(cc2Cl)Cl 2M-535S CO/N=C(/CS(=O)(=O)Cc1ccccc1Cl)\c2ccc(cc2Cl)Cl 2M-536S CSc1c(c2ccccc2nc1c3ccccc3)C(=O)O 2M-537S CSc1cc2ccccc2nc1c3ccccc3 2M-538S CSc1cc2cc(ccc2nc1c3ccccc3)Cl 2M-539S c1cc(ccc1c2c(cc3cc(ccc3n2)Cl)Sc4ccc(cc4)Cl)Cl 2M-540S c1ccc(cc1)c2nc(cs2)c3cc(no3)c4cccc(c4)C(F)(F)F 2M-541S c1cc(cc(c1)C(F)(F)F)c2cc(on2)c3csc(n3)c4ccc(cc4)Cl 2M-542S c1ccnc(c1)c2nc(cs2)c3cc(no3)c4cccc(c4)C(F)(F)F 2M-543S c1ccc(cc1)c2cc(on2)c3cn4ccccc4n3 2M-544S c1ccn2cc(nc2c1)c3cc(no3)c4cccc(c4)C(F)(F)F 2M-545S COc1cccc(c1)C(=O)N2CCN3C2(c4ccccc4C3=O)c5ccc(cc5)Cl 2M-546S c1ccc2c(c1)C(=O)N3C2(N(CC3)C(=O)CCl)c4ccc(cc4)Cl 2M-547S CO/N=C(/CS(=O)Cc1ccccc1Cl)\c2ccc(cc2Cl)Cl 2M-551S Cc1cccc(c1C)OCC(=O)c2ccc(cc2)Cl 2M-552S c1ccc(cc1)OCC(=O)c2ccc(cc2)Cl 2M-553S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)/C(=N\OC)/CS(=O)(=O)c2ccc(cc2)F 2M-560S c1ccc(cc1)C23c4ccccc4C(=O)N2CCN3 2M-569S c1cc(cc(c1)OCC(=O)c2ccc(cc2)Cl)C(F)(F)F 2M-570S CC(C)(C)c1ccc(cc1)OCC(=O)c2ccc(cc2)Cl 2M-571S c1ccc(cc1)c2c(c(c3ccccc3n2)C(=O)O)Oc4ccc(cc4)Cl 2M-572S Cc1cccc(c1C)Oc2c(c3ccccc3nc2c4ccccc4)C(=O)O 2M-574S COc1ccc(cc1)/C(=N\OC)/COc2ccc(cc2)F 2M-576S COc1ccc(cc1)/C(=N\OC)/COc2cccc(c2)C(F)(F)F 2M-577S Cc1ccc(cc1)SC/C(=N/OC)/c2ccc(cc2)OC 2M-578S COc1ccc(cc1)/C(=N\OC)/CSc2ccc(cc2)Br 2M-579S c1ccc2c(c1)c(c(c(n2)c3ccc(cc3)Cl)Oc4cccc(c4)C(F)(F)F)C(=O)O 2M-580S CC(C)(C)c1ccc(cc1)Oc2c(c3ccccc3nc2c4ccc(cc4)Cl)C(=O)O 2M-581S c1ccc2c(c1)c(c(c(n2)c3ccc(cc3)Cl)Oc4ccc(cc4)Cl)C(=O)O 2M-582S c1ccc(cc1)c2c(cc3ccccc3n2)Oc4ccc(cc4)Cl 2M-583S Cc1ccc(cc1)S(=O)C/C(=N/OC)/c2ccc(cc2)OC 2M-586S Cc1ccc(cc1)S(=O)(=O)C/C(=N/OC)/c2ccc(cc2)OC 2M-587S COc1ccc(cc1)/C(=N\OC)/CS(=O)c2ccc(cc2)Br 2M-588S COc1ccc(cc1)/C(=N\OC)/CS(=O)(=O)c2ccc(cc2)Br 2M-589S c1ccc2c(c1)c(c(c(n2)c3ccc(cc3)Cl)Oc4ccc(cc4)F)C(=O)O 2M-590S c1ccc2c(c1)c(c(c(n2)c3ccc(cc3)Cl)Oc4ccccc4Cl)C(=O)O 2M-591S Cn1c(c(c(n1)c2ccccc2)COCc3c(cccc3Cl)Cl)Sc4ccc(cc4)Cl 2M-595S c1ccc(cc1)CN2Cc3cc(c4cccnc4c3OC2)Cl 2M-596S c1cc2c(cc3c(c2nc1)OCN(C3)Cc4ccc(c(c4)Cl)Cl)Cl 2M-597S c1ccc(cc1)Oc2ccc(cc2)NC(=O)Cc3cccc(c3)C(F)(F)F 2M-598S c1ccc(cc1)Oc2c(c3ccccc3nc2c4ccc(cc4)Cl)C(=O)O 2M-601S c1ccc2c(c1)cc(c(n2)c3ccc(cc3)Cl)Oc4ccccc4Cl 2M-602S c1ccc2c(c1)c(c(s2)C#N)N3CCOCC3 2M-700 Cc1cc(=O)c(cn1Nc2ccc(cc2)Cl)C(=O)O 2M-701 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(cc4Cl)Cl)C(=O)C1)C 2M-703 CC1=C(C(C(=C(N1)C)C#N)c2c(c3ccccc3s2)Cl)C#N 2M-704 Cc1cc(=O)c(cn1Nc2cccc(c2)Cl)C(=O)O 2M-705 c1cc(c(cc1Cl)Cl)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)C4CCCCC4C3=O 2M-706 Cc1cc(c(c(=O)o1)/C=N/Nc2cccc(c2)[N+](=O)[O-])O 2M-707 Cc1cc(c(c(=O)o1)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)O.CNC 2M-708 Cc1c(c(c(c(n1)C)C#N)c2c(c3ccccc3s2)Cl)C#N 2M-709 c1ccc(c(c1)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)C4CCCCC4C3=O)C(F)(F)F 2M-710 CC(=O)c1c(c2ccccc2[nH]c1=O)OC 2M-711 Cc1c(c(c(c(n1)/C=C/N(C)C)C#N)c2c(c3ccccc3s2)Cl)C#N 2M-713 c1ccc2c(c1)c(c(s2)C=O)Sc3ccccn3 2M-714 Cc1cc(=O)c(cn1Nc2cccc(c2)[N+](=O)[O-])C(=O)O 2M-716 CCOC(=O)C1=C(NC2=C(C1c3ccc(cc3)OC)C(=O)CC(C2)(C)C)C 2M-717 CCOC(=O)C1=C(NC2=C(C1c3ccc(cc3)Cl)C(=O)CC(C2)(C)C)C(F)(F)F 2M-718 CC1(C2CCC(O1)(C(=O)OC2=O)C)C 2M-719 CCOC(=O)c1c(nc2c(c1c3ccc(cc3)OC)C(=O)CC(C2)(C)C)C 2M-723 c1ccc(c(c1)N)NC2=CC(=O)CC(C2)c3c(cccc3Cl)F 2M-726 CCOC(=O)C1=C(NC2=C(C1c3ccc(cc3Cl)Cl)C(=O)C(CC2)c4c(cccc4Cl)F)C 2M-727 c1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)c4c(cccc4Cl)F)c5ccc(cc5)Cl 2M-728 Cc1cc(=O)c(cn1Nc2c(cc(cn2)C(F)(F)F)Cl)C(=O)O 2M-729 c1ccc(c(c1)N)NC2=CC(=O)CC(C2)c3ccc(cc3)F 2M-730 c1cc(ccc1C(=O)COc2ccc(cc2)Cl)Cl 2M-869S CCOC(=O)NC(=O)/C(=N/Nc1cccc(c1)OC)/C(=O)C 2M-900 CCOC(=O)C1=NOC(C1)C(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl 2M-901 CC1(NC(=O)N(N1)c2ccccc2)C3=NOC(C3)C(=O)NN(C)c4c(cc(cn4)C(F)(F)F)Cl 2M-902 CC(=O)c1c(=O)[nH]c(=O)n(n1)c2cccc(c2)OC 2M-903 c1ccc2cc(ccc2c1)c3c[nH]c(c3C#N)N 2M-904 CCOC(=O)c1c(c[nH]c1N)c2ccc3ccccc3c2 2M-905 Cc1cc(n2cc(c(c2n1)C#N)c3ccc4ccccc4c3)C 2M-906 CCOC(=O)C(=O)Nc1ccccc1C(=O)c2ccccc2 2M-907 CN(C)/C=N/C(=O)c1c(c2cc(ccc2[nH]1)Cl)c3ccccc3 2M-908 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cn2)I 2M-909 c1cc(ccc1C(F)(F)F)NC(=O)Nc2ccc(cn2)I 2M-910 CCOC(=O)NC(=O)/C(=C/Nc1ccc(cn1)I)/C#N 2M-911 Cn1c(=O)c(nn(c1=O)c2cccc(c2)OC)C(=O)/C=C/N(C)C 2M-912 c1cc(ncc1I)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl 2M-913 CCOC(=O)NC(=O)/C(=C/Nc1ccc(cn1)I)/C(=O)C 2M-914 Cn1c(=O)c(nn(c1=O)c2cccc(c2)OC)c3ccnn3c4ccccc4 2M-915 Cn1c(=O)c(nn(c1=O)c2cccc(c2)OC)c3ccnn3c4ccc(cc4)OC 2M-916 Cn1c(=O)c(nn(c1=O)c2cccc(c2)OC)c3ccnn3c4cccc(c4)Cl 2M-917 c1cc(c(cc1Cl)Cl)C(=O)/C=C\Nc2ccc(cn2)I 2M-918 Cc1ccc(cc1)n2c(ccn2)c3c(=O)n(c(=O)n(n3)c4cccc(c4)OC)C 2M-919 Cn1c(=O)c(nn(c1=O)c2cccc(c2)OC)c3ccnn3c4ccc(cc4)F 2M-920 CCOC(=O)c1c(c2ccccc2[nH]1)c3ccccc3 2M-922 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)O 2M-923 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3cccs3)Cl 2M-925 c1ccc(cc1)C(=O)c2ccccc2NC(=O)c3cccc(c3)Cl 2M-926 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)N4CCOCC4 2M-928 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)NCc4ccco4 2M-929 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)Nc4ccc(cc4)F 2M-930 c1ccc(cc1)NC2=C(C(=NC(=CS2)c3ccc(cc3)Br)N4CCOCC4)C#N 2M-931 c1ccc(cc1)NC2=C(C(=NC(=CS2)c3ccc(cc3)F)N4CCOCC4)C#N 2M-932 c1ccc(cc1)Nc2c(c(c(s2)C(=O)c3ccc(cc3)Cl)N)C#N 2M-933 c1ccc2c(c1)ccc3c2C(=O)CO3 2M-935 c1ccc2c(c1)cccc2OCC(=O)O 2M-936 c1ccc(cc1)Nc2c(c(c(s2)C(=O)c3ccc(cc3)Cl)n4cccc4)C#N 2M-937 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)NN 2M-938 CN(C)/C=C\1/C(=O)c2c3ccccc3ccc2O1 2M-939 COC(=O)C1CC(CN1C(=O)Nc2ccccc2)O 2M-941 c1ccc2c(c1)ccc3c2OCC3=O 2M-942 CN(C)/C=C/1\C(=O)c2ccc3ccccc3c2O1 2M-943 C/C(=N\O)/C1CC1c2ccc(cc2)F 2N-001 CSc1ccc(cc1)NC(=S)N 2N-002 c1ccc2c(c1)nc(c3n2ccc3)Cl 2N-004 C/C(=N\OC(=O)c1cccs1)/C2CC2c3ccc(cc3)F 2N-005 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)OCO3 2N-006 C/C(=N\OCCOc1ccccc1)/C2CC2c3ccc(cc3)F 2N-007 c1cc2c(cc1NC(=S)N)OCO2 2N-008 c1ccc(cc1)c2ccccc2NC(=S)NC(=O)c3ccccc3 2N-009 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2cccn3 2N-010 C/C(=N\OC(=O)C1CC1)/C2CC2c3ccc(cc3)F 2N-011 c1cc2c(cccn2)c(c1)NC(=S)N 2N-012 c1ccc(cc1)c2ccccc2NC(=S)N 2N-013 c1ccc(cc1)C(=O)NC(=S)NC2CCCCC2 2N-014 C/C(=N\OCCOc1cccc(c1)C(F)(F)F)/C2CC2c3ccc(cc3)F 2N-015 C1CCC(CC1)NC(=S)N 2N-016 C/C(=N\OC(=O)c1cccc(c1)OC)/C2CC2c3ccc(cc3)F 2N-017 COc1ccc(cc1)Oc2c3cccn3c4ccccc4n2 2N-019 c1cc(ccc1C(=O)C2CC2c3ccc(cc3Cl)Cl)Br 2N-022 C/C(=N\OC(=O)c1c(cccc1Cl)Cl)/C2CC2c3ccc(cc3)F 2N-023 Cc1ccc(cc1)Oc2c3cccn3c4ccccc4n2 2N-024 c1ccc(cc1)Oc2c3cccn3c4ccccc4n2 2N-025 c1ccc2c(c1)nc(c3n2ccc3)Oc4cccc(c4)F 2N-026 CC(=O)Nc1ccc(cc1)Oc2c3cccn3c4ccccc4n2 2N-027 c1ccc2c(c1)nc(c3n2ccc3)Oc4ccc(cc4)Cl 2N-028 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)[N+](=O)[O-])Cl 2N-030 c1cc(ccc1C(=O)C2CC2c3ccc(cc3Cl)Cl)Cl 2N-031 c1ccc(cc1)/C=C/C(=O)c2ccccn2 2N-033 COc1cccc(c1)C(=O)/C=C/c2ccc(cc2)Cl 2N-034 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl 2N-035 c1cc(ccc1C2CC2C(=O)c3ccc(cc3)[N+](=O)[O-])Cl 2N-036 c1cc(ccc1/C(=N\O)/C2CC2c3ccc(cc3Cl)Cl)Br 2N-037 c1ccc(cc1)C2CC2C(=O)c3ccccn3 2N-038 c1cc(ccc1/C(=N\O)/C2CC2c3ccc(cc3Cl)Cl)Cl 2N-039 c1cc(ccc1C2CC2/C(=N/OCc3ccc(cc3Cl)Cl)/c4ccc(cc4)[N+](=O)[O-])Cl 2N-040 c1cc(ccc1C2CC2/C(=N/O)/c3ccc(cc3)[N+](=O)[O-])Cl 2N-041 COc1cccc(c1)C(=O)C2CC2c3ccc(cc3)Cl 2N-042 c1cc(c(c(c1)Cl)/C=C/C(=O)c2ccc(cc2)F)F 2N-043 c1cc(ccc1C2CC2C(=O)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)Cl 2N-045 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Br)Cl 2N-046 c1cc(ccc1C2CC2C(=O)c3ccc(cc3)Br)Cl 2N-047 c1ccc(cc1)OCCO/N=C(\c2ccc(cc2)[N+](=O)[O-])/C3CC3c4ccc(cc4)Cl 2N-048 CCCOC(=O)Nc1cc(nc2c1cccc2)c3ccc(cc3)Cl 2N-302S COC(=O)Nc1cc(nc2c1cccc2)c3ccc(cc3)Cl 2N-303S c1ccc(cc1)c2cc(c(c(n2)Cl)C#N)C(F)(F)F 2N-306S c1ccc(cc1)COC(=O)Nc2cc(nc3c2cccc3)c4ccc(cc4)Cl 2N-307S c1ccc2c(c1)c(cc(n2)c3ccc(cc3)Cl)NC(=O)OCc4ccc(cc4)F 2N-308S Cc1c(c(cc(n1)c2ccc(cc2)Cl)C(F)(F)F)C#N 2N-309S C=CCOC(=O)Nc1cc(nc2c1cccc2)c3ccc(cc3)Cl 2N-310S CC(C)(C)c1ccc(cc1)COC(=O)Nc2cc(nc3c2cccc3)c4ccc(cc4)Cl 2N-311S Cn1c2ccccc2cc1O 2N-312S C1CCc2c(c(=O)[nH]c(n2)N)C1 2N-317S CN1c2ccc(cc2CC1=O)[N+](=O)[O-] 2N-318S c1ccc(cc1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 2N-319S c1cc(ccc1C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3)F 2N-321S c1cc(ccc1C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3)Cl 2N-322S Cc1cccc(c1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 2N-323S COc1cccc(c1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 2N-324S c1cc(sc1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 2N-325S Cc1ccc(cc1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 2N-326S Cc1ccc(cc1)Sc2c(c3cc(ccc3n2C)[N+](=O)[O-])C=O 2N-327S Cn1c2ccccc2c(c1Cl)C=O 2N-329S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 2N-331S Cc1[nH]c(=O)n(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl 2N-501S Cc1nn(c(=O)n1C)c2c(cc(cc2Cl)C(F)(F)F)Cl 2N-502S c1cc(c(cc1Cl)Cl)c2csc(n2)N3CCSCC3 2N-503S Cc1cc(c(cc1Cl)F)C(=O)CBr 2N-504S CN(c1ccccc1)C(=O)CCl 2N-505S c1ccc(cc1)C(=O)c2c(cc(=O)n(n2)c3ccccc3)C(F)(F)F 2N-514S C1CC1C(=O)CC(=O)C(F)(F)F 2N-515S Cn1c(c(c(n1)c2ccccc2)/C=N/O)Cl 2N-516S Cn1c(c(c(n1)c2ccccc2)/C=N/OC)Cl 2N-517S Cn1c(c(c(n1)c2ccccc2)/C=N/OCc3ccc(cc3Cl)Cl)Cl 2N-518S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)S 2N-522S c1ccc(cc1)Cn2c(=O)c3ccccc3sc2=O 2N-524S c1ccc2c(c1)c(=O)n(c(=O)s2)Cc3ccc(cc3)Cl 2N-525S CSc1nnc(o1)Cc2c(nc(s2)c3ccccc3)c4ccccc4 2N-527S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)SCc5nc6cc(ccc6s5)F 2N-528S Cn1c(cc(n1)C(F)(F)F)OCC(=O)N(C)c2ccccc2 2N-529S c1ccc(c(c1)Cn2c(=O)c3ccccc3sc2=O)Cl 2N-530S COc1ccc(cc1)Cn2c(=O)c3ccccc3sc2=O 2N-531S Cc1ccc(cc1)Cn2c(=O)c3ccccc3sc2=O 2N-532S c1ccc2c(c1)c(=O)n(c(=O)s2)C3CC3 2N-533S COc1c(c(ncn1)OC)S(=O)(=O)N2CCOCC2 2N-536S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)SCc5cccc(c5)C(F)(F)F 2N-538S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)SCc5ccc(cc5)Cl 2N-539S COc1c(c(ncn1)OC)S(=O)(=O)N2CCSCC2 2N-540S COc1c(c(ncn1)OC)S(=O)(=O)NCc2ccccc2 2N-541S COc1c(c(ncn1)OC)S(=O)(=O)Nc2ccc(cc2)C(F)(F)F 2N-543S CCCSc1nc2ccsc2c(=O)n1CC 2N-545S CN(C)c1ccc(cc1)/C=C/c2nc3ccccc3s2 2N-547S CCOc1ccc(cc1/C=C/c2nc3ccccc3s2)Br 2N-549S c1ccc2c(c1)nc(s2)/C=C/c3ccc(s3)Br 2N-550S CC(C)(C)c1ccc(cc1)/C=C/c2nc3ccccc3s2 2N-551S CCCn1c(=O)c2ccccc2sc1=O 2N-552S C=CCn1c(=O)c2ccccc2sc1=O 2N-553S COCCn1c(=O)c2ccccc2sc1=O 2N-554S Cn1c(cc(n1)c2ccccc2)OCC(=O)N(C)c3ccccc3 2N-555S CN(Cc1ccccc1)Cc2c(nc3n2cccc3)c4ccc(cc4)Cl 2N-557S c1ccn2c(c1)nc(c2CN3CCOCC3)c4ccc(cc4)Cl 2N-558S c1ccn2c(c1)nc(c2CN3CCSCC3)c4ccc(cc4)Cl 2N-561S c1ccc(cc1)CN2CCN(CC2)Cc3c(nc4n3cccc4)c5ccc(cc5)Cl 2N-562S Cc1c(sc2n1ncn2)C(C)OC(=O)c3cccs3 2N-564S Cc1c(sc2n1ncn2)C(C)OC(=O)c3cccc(c3)C(F)(F)F 2N-565S c1ccn2c(c1)nc(c2CN3CCCCC3)c4ccc(cc4)Cl 2N-568S c1ccc(c(c1)N2CCN(CC2)Cc3c(nc4n3cccc4)c5ccc(cc5)Cl)F 2N-569S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)NN 2N-579S CCn1c(=O)c2c(ccs2)nc1S 2N-630S CCn1c(=O)c2c(ccs2)nc1SCC=C 2N-631S Cc1c(c(=O)[nH]c(n1)SC)CCO 2N-700 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)C(F)(F)F 2N-701 c1cc(ccc1Nc2ccnc(c2)C(F)(F)F)Cl 2N-704 Cc1c(c(=O)[nH]c(n1)SC)CCOC(=O)C 2N-705 c1ccnc(c1)Nc2ccnc(c2)C(F)(F)F 2N-706 Cc1c(c(=O)[nH]c(n1)SCc2ccccc2)CCO 2N-707 c1cc(ccc1C(F)(F)F)Nc2ccnc(c2)C(F)(F)F 2N-710 C/C(=C/C(=O)C(F)(F)F)/Nc1ccc(cc1)Br 2N-711 Cc1ccc(cc1)CSc2[nH]c(=O)c(c(n2)C)CCO 2N-712 Cc1c(c(=O)[nH]c(n1)SCc2cccc(c2)Cl)CCO 2N-713 c1ccc(cc1)Oc2ccccc2Nc3ccnc(c3)C(F)(F)F 2N-714 C/C(=C\C(=O)C(F)(F)F)/Nc1ccccc1C(=O)OC 2N-715 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)Br 2N-716 COC(=O)c1ccccc1SCC(=O)c2cc(sc2Cl)Cl 2N-717 CC(=O)N1CC(=O)N/C(=C/c2ccc(cc2)OC)/C1=O 2N-718 c1cc(ccc1Nc2ccnc(c2)C(F)(F)F)Br 2N-719 CC(=O)N1CC(=O)N/C(=C/c2ccco2)/C1=O 2N-721 COC(=O)c1ccccc1SC/C(=N\O)/c2cc(sc2Cl)Cl 2N-722 Cc1ccc(c(c1)C)Nc2ccnc(c2)C(F)(F)F 2N-723 Cc1cccc(c1)C(=O)OCCc2c(nc([nH]c2=O)SC)C 2N-724 CC(=O)N1CC(=O)N/C(=C/c2cccs2)/C1=O 2N-725 Cc1c(c(=O)[nH]c(n1)SC)CCOC(=O)c2cccs2 2N-726 C/C(=C/C(=O)C(F)(F)F)/NC1CCCCC1 2N-727 CC(=O)N1CC(=O)N/C(=C/c2ccccc2)/C1=O 2N-729 Cc1c(c(=O)[nH]c(n1)SC)CCOC(=O)c2cccc(c2)Cl 2N-730 CC(=O)N1CC(=O)N(/C(=C/c2ccc(cc2)OC)/C1=O)Cc3ccccc3 2N-731 Cc1c(c(=O)[nH]c(n1)SC)CCOC(=O)c2ccccc2 2N-732 CC(C(=O)OC)Oc1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 2N-733 C#CCOc1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 2N-734 CC(C(=O)C)Oc1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 2N-735 c1cc(cc(c1)[N+](=O)[O-])N/C=C/C(=O)c2cc(sc2Cl)Cl 2N-736 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/NC1CCCCC1 2N-737 Cc1c(c(nc(n1)SC)Cl)CCCl 2N-738 c1cnc(cc1NC2CCCCC2)C(F)(F)F 2N-739 CCCC(=O)OCCc1c(nc([nH]c1=O)SC)C 2N-740 c1cc[n+](c(c1)SC(F)F)[O-] 2N-743 CC(=O)N1CC(=O)N(/C(=C/c2ccc(cc2)OC)/C1=O)Cc3ccc(cc3)[N+](=O)[O-] 2N-744 Cc1c(c(=O)[nH]c(n1)SC)CCOCc2ccccc2 2N-745 Cc1c(c(=O)[nH]c(n1)SC)CCOCc2ccc(cc2)F 2N-746 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCc3ccc(cc3)[N+](=O)[O-] 2N-747 Cc1c(c(=O)[nH]c(n1)SC)CCOCc2ccc(cc2)[N+](=O)[O-] 2N-750 Cc1c2c(nc(n1)SC)N(CC2)c3ccc(cc3)F 2N-751 c1cc(ccc1N/C=C/C(=O)c2cc(sc2Cl)Cl)F 2N-752 c1cc(c(cc1F)F)N/C=C/C(=O)c2cc(sc2Cl)Cl 2N-753 C/C(=C\C(=O)C(F)(F)F)/Nc1ccccc1Oc2c(cc(cn2)C(F)(F)F)Cl 2N-754 c1cc(ccc1N/C=C/C(=O)c2cc(sc2Cl)Cl)Br 2N-755 C/C(=C/C(=O)C(F)(F)F)/Nc1cccc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl 2N-756 C/C(=C/C(=O)C(F)(F)F)/Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 2N-757 c1cc(ccc1/C=C\2/C(=O)N(C(=N2)SCCC(=C(F)F)F)c3ccc(cc3)F)Cl 2N-758 c1c(cnc(c1Cl)SCCC(=C(F)F)F)C(F)(F)F 2N-760 c1ccc(cc1)n2c(=O)c3c(ccs3)nc2SCCC(=C(F)F)F 2N-761 c1cc(c(cc1Cl)Cl)Cc2c(ccc(c2O)C=O)O 2N-764 Cc1cc(c(c(c1)C)COc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl)C 2N-765 Cc1c(c(=O)[nH]c(n1)SCc2ccccc2)CCOC(=O)c3ccccc3 2N-767 Cc1c2c(nc(n1)SC)N(CC2)c3ccc(cc3)C(F)(F)F 2N-768 Cc1c2c(nc(n1)SC)N(CC2)c3ccccc3 2N-769 CCN\1C(=O)CN(C(=O)/C1=C\c2ccc(cc2)OC)C(=O)C 2N-771 Cc1c(c(=O)[nH]c(n1)NN)CCO 2N-772 Cc1c2c(nc(n1)SC)N(CC2)c3ccc(cc3)OC 2N-773 Cc1c2c(nc(n1)SCc3ccccc3)N(CC2)c4ccc(cc4)Br 2N-774 COc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 2N-775 c1cc(cc(c1)N/C=C/C(=O)c2cc(sc2Cl)Cl)C#N 2N-776 c1cc(ccc1N/C=C/C(=O)c2cc(sc2Cl)Cl)OC(F)(F)F 2N-777 COc1ccc(cc1OC)N/C=C/C(=O)c2cc(sc2Cl)Cl 2N-778 Cn1cccc1/C=N/NC(=S)N 2N-900 c1cc([nH]c1)/C=N/NC(=S)N 2N-901 c1cnc(nc1)Oc2cc(c(cc2Cl)F)N 2N-903 Cc1ccn2c(c1)nc(c2Br)c3ccccc3 2P-001 c1ccc(cc1)c2c(c[nH]n2)C=O 2P-002 COc1cc(cc(c1OC)OC)C(=O)N/N=C/c2ccccc2Oc3ccc(cc3F)Br 2P-003 COc1cc(cc(c1OC)OC)C(=O)N/N=C/c2ccccc2Oc3ccc(cc3)Cl 2P-004 c1ccc(c(c1)/C=N\O)Oc2cccc(c2)Cl 2P-005 c1ccc(cc1)Oc2ccc(cc2)C#N 2P-006 c1ccc(cc1)c2c(c[nH]n2)/C=C/3\C(=O)NC(=O)S3 2P-007 c1ccc(cc1)c2c(c[nH]n2)C=C(C#N)C#N 2P-008 Cc1cc(cc(c1)Oc2ccccc2/C=N\O)C 2P-009 c1ccc(c(c1)/C=N\O)Oc2ccc(cc2Cl)Cl 2P-010 c1ccc(c(c1)/C=N\O)Oc2ccc(cc2)F 2P-011 c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)Br 2P-012 c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)CO 2P-014 c1ccc(c(c1)C=O)Oc2cccc(c2)C(F)(F)F 2P-015 c1ccc(cc1)c2c(c[nH]n2)/C=N/O 2P-016 c1ccc(cc1)c2c(c[nH]n2)/C=C(/C#N)\S(=O)(=O)c3ccccc3 2P-018 c1ccc(cc1)c2c(c[nH]n2)/C=C\C(=O)O 2P-020 c1cc(ccc1c2cn3cc(ccc3n2)Cl)Cl 2P-022 CC1CN(CC(O1)C)c2ncc(s2)/C=N\O 2P-023 c1cnc2nc(cn2c1)c3ccc(cc3)Cl 2P-024 COc1cc(cc(c1OC)OC)C(=O)N/N=C/c2cccc(c2)OCc3cnc(s3)Cl 2P-026 c1cc(ccc1c2nnco2)C(F)(F)F 2P-027 c1cc(cc(c1)OCc2cnc(s2)Cl)/C=N/NC(=S)N 2P-028 c1cc2c(cc1[N+](=O)[O-])ocn2 2P-029 CN(C)/C=C(\c1cnc(s1)Cl)/S(=O)(=O)c2ccccc2 2P-030 c1ccc(c(c1)/C=C/C(=O)O)Oc2ccc(cc2)I 2P-032 c1ccc(c(c1)/C=C/C(=O)O)Oc2cccc(c2)C(F)(F)F 2P-033 CC1CN(CC(O1)C)c2ncc(s2)/C=N/Nc3ccc(cc3)C(F)(F)F 2P-034 c1ccc(cc1)Oc2ccccc2CO 2P-035 c1ccc(c(c1)CO)Oc2ccc(cc2)Cl 2P-036 Cc1ccc(cc1)Oc2ccccc2CO 2P-037 C/C(=N/NC(=S)N)/c1ccccc1OCc2cnc(s2)Cl 2P-038 CCOC(=O)C(=CC(=O)OC(C)(C)C)C(=O)OCC 2P-039 Cc1ccn2c(c1)nc(c2CN3CCOCC3)c4ccccc4 2P-040 c1ccc(cc1)N2CCN(CC2)c3ncc(s3)/C=N\O 2P-041 c1cc2c(cc1N)nc[nH]2 2P-043 Cc1cc(c(cc1N)Cl)C(c2ccc(cc2)Cl)C(=O)N 2P-044 c1cc(c(cc1Cl)Cl)NNC(=S)N 2P-045 c1cc2c(cc1N)ocn2 2P-046 c1cc2c(ccnc2cc1Cl)NNC(=S)N 2P-047 c1cc(ccc1NNC(=S)N)Cl 2P-048 c1cc(c2cc[nH]c2c1)N 2P-050 c1c(cc(c(c1Cl)NNC(=S)N)Cl)Cl 2P-051 Cc1cccc(c1)NNC(=S)N 2P-052 c1ccc(cc1)N(c2ccccc2)NC(=S)N 2P-053 c1c(cc(cc1Cl)Cl)NNC(=S)N 2P-054 c1cc(cc(c1)Cl)NNC(=S)N 2P-056 Cc1ccc(cc1Cl)NNC(=S)N 2P-057 Cc1ccc(c(c1)NNC(=S)N)C 2P-058 c1ccc(c(c1)/C=N/c2ccc(cc2)I)Oc3ccc(c(c3)F)F 2P-060 CN(C)/C=C/C(=O)c1ccccc1OCc2cnc(s2)Cl 2P-061 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2cc[nH]3 2P-062 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)nc[nH]3 2P-063 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)ocn3 2P-064 CCOC(=O)c1ccc(cc1)/N=C/c2cccs2 2P-065 c1ccc(c(c1)CNc2ccc(cc2)I)Oc3ccc(c(c3)F)F 2P-066 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)I)Cl 2P-067 c1cc2c(cc[nH]2)c(c1)NC(=S)N 2P-069 c1cc2c(cc1NC(=S)N)ocn2 2P-070 c1cc(cc(c1)F)COn2cc[n+](c2)[O-] 2P-071 c1ccc(cc1)S(=O)(=O)c2ncc(s2)C=O 2P-073 c1ccc(c(c1)/C=N/c2ccc(cc2)I)Oc3ccc(cc3F)Br 2P-074 CCOc1ccc(cc1/C=N/c2ccc(cc2)I)Br 2P-075 c1cc2c(cc1NC(=S)N)nc[nH]2 2P-076 c1ccc(c(c1)CO)Oc2ccc(cc2Cl)Cl 2P-077 c1ccc(c(c1)CO)Oc2ccc(cc2F)Br 2P-078 c1ccc(c(c1)CO)Oc2ccc(cc2)I 2P-079 c1ccc(cc1)COc2ccc(cc2)Oc3ccccc3CO 2P-080 c1cc(sc1)CNc2ccc(cc2)C(=O)O 2P-081 c1ccc2c(c1)CC(C2Sc3[nH]c4ccccc4n3)O 2P-082 c1ccc2c(c1)CC(C2Sc3nc4ccccc4s3)O 2P-083 c1cc(cc(c1)F)COn2ccnc2 2P-084 CCOC(=O)c1ccc(cc1)/N=C/c2ccccc2Oc3ccc(c(c3)F)F 2P-086 CCOc1ccc(cc1CNc2ccc(cc2)I)Br 2P-087 c1ccc(cc1)COc2ccc(cc2)Oc3ccccc3/C=N/c4ccc(cc4)I 2P-089 c1ccc(c(c1)CO)Oc2ccc(c(c2)F)Cl 2P-090 CCOC(=O)c1ccc(cc1)NCc2ccccc2Oc3ccc(c(c3)F)F 2P-091 c1ccc(cc1)c2c(c[nH]n2)/C=N/NC(=O)c3ccco3 2P-092 c1ccc(cc1)c2c(c[nH]n2)/C=N/NC(=O)c3ccc(cc3)C(F)(F)F 2P-093 c1ccc2c(c1)c(=O)[nH]c(n2)Nc3cccc(c3)C(F)(F)F 2P-301S Cc1cc(cc(c1)Nc2[nH]c(=O)c3ccccc3n2)C 2P-302S COc1cccc(c1)Nc2[nH]c(=O)c3ccccc3n2 2P-303S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Nc4ccc(cc4)OC)CS2 2P-315S CCNC(=O)Nc1ccccc1C#N 2P-317S CC(C)NC(=O)Nc1ccccc1C#N 2P-318S Cn1c2ccccc2c(c1Cl)/C=N/O 2P-319S CC(=O)O/N=C/c1c2ccccc2n(c1Cl)C 2P-320S Cn1c2ccccc2c(c1Cl)C#N 2P-321S c1ccc(cc1)Cn2c(c(c(c2NC(=O)c3ccccc3)C#N)c4ccccc4)c5ccccc5 2P-322S Cc1ccc(cc1)C(=O)Nc2c(c(c(n2Cc3ccccc3)c4ccccc4)c5ccccc5)C#N 2P-323S CCCC(=O)Nc1c(c(c(n1Cc2ccccc2)c3ccccc3)c4ccccc4)C#N 2P-324S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Nc4cc(cc(c4)C)C)CS2 2P-325S Cc1ccc(cc1)S(=O)(=O)N(c2c(c(c(n2Cc3ccccc3)c4ccccc4)c5ccccc5)C#N)S(=O)(=O)c6ccc(cc6)C 2P-326S c1ccc(cc1)Cn2c(c(c(c2/N=C/c3ccc(cc3)Cl)C#N)c4ccccc4)c5ccccc5 2P-327S c1ccc2c(c1)c(=O)n3c(n2)NCC3CBr 2P-328S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Nc4ccc(cc4F)F)CS2 2P-330S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Nc4ccc(cc4)F)CS2 2P-331S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Nc4cccc(c4)Cl)CS2 2P-332S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Nc4ccc(cc4C)Cl)CS2 2P-333S c1ccc(cc1)Cn2c(c(c(c2NC(=O)c3ccc(cc3)F)C#N)c4ccccc4)c5ccccc5 2P-336S c1ccc(cc1)Cn2c(c(c(c2NC(=O)c3cccc(c3)Cl)C#N)c4ccccc4)c5ccccc5 2P-337S Cc1cccc(c1)C(=O)Nc2c(c(c(n2Cc3ccccc3)c4ccccc4)c5ccccc5)C#N 2P-338S c1ccc(cc1)Cn2c(c(c(c2NC(=O)c3cccs3)C#N)c4ccccc4)c5ccccc5 2P-339S CCCCn1c(c(c(c1N)C#N)c2ccccc2)c3ccccc3 2P-341S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Nc4ccc(cc4)OC(F)(F)F)CS2 2P-345S c1ccc(cc1)Cn2c(c(c(c2NC(=O)c3ccccc3Cl)C#N)c4ccccc4)c5ccccc5 2P-348S Cc1ccccc1C(=O)Nc2c(c(c(n2Cc3ccccc3)c4ccccc4)c5ccccc5)C#N 2P-349S Cc1ccc(cc1)SCC2CNc3n2c(=O)c4ccccc4n3 2P-351S CCCCn1c(c(c(c1NC(=O)c2ccccc2OC)C#N)c3ccccc3)c4ccccc4 2P-354S c1ccc2c(c1)c(=O)n3c(n2)NCC3CSc4ccc(cc4)Cl 2P-360S Cc1ccc(c(c1)C)SCC2CNc3n2c(=O)c4ccccc4n3 2P-361S Cc1cccc(c1)C(=O)O/N=C/c2c3ccccc3n(c2Cl)C 2P-362S CCCCn1c(c(c(c1/N=C/c2ccc(cc2)Cl)C#N)c3ccccc3)c4ccccc4 2P-363S CCCCn1c(c(c(c1/N=C/c2ccc(cc2)OC)C#N)c3ccccc3)c4ccccc4 2P-364S Cc1ccc(cc1)C(=O)O/N=C/c2c3ccccc3n(c2Cl)C 2P-365S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)c3cccc(c3)Cl 2P-366S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)c3ccccc3Cl 2P-367S CCCCC(=O)O/N=C/c1c2ccccc2n(c1Cl)C 2P-368S c1csc2n1c(c(n2)Cl)Br 2P-371S CCn1c(=N)c2ccccc2[nH]c1=O 2P-378S CCCCn1c(c(c(c1/N=C/c2ccccc2)C#N)c3ccccc3)c4ccccc4 2P-379S CCCCn1c(c(c(c1/N=C/c2cccc(c2)OC)C#N)c3ccccc3)c4ccccc4 2P-380S CCCCn1c(c(c(c1/N=C/c2ccc(cc2)[N+](=O)[O-])C#N)c3ccccc3)c4ccccc4 2P-381S CCCCn1c(c(c(c1/N=C/c2cccs2)C#N)c3ccccc3)c4ccccc4 2P-382S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)c3cccs3 2P-384S CCn1/c(=N\C(=O)c2ccccc2)/c3ccccc3[nH]c1=O 2P-385S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)c3ccc(cc3)F 2P-386S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)c3ccc(cc3)Cl 2P-387S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)c3ccccc3OC 2P-388S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)Cc3cccs3 2P-389S CC(C)(C)C(=O)O/N=C/c1c2ccccc2n(c1Cl)C 2P-390S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NS(=O)(=O)c3ccc(cc3)Br 2P-502S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NS(=O)(=O)c3cccc(c3)C(F)(F)F 2P-503S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NS(=O)(=O)c3ccccc3Cl 2P-504S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)c3cccs3 2P-505S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)c3cccc(c3)C(F)(F)F 2P-506S Cc1ccc(cc1)C(=O)Nc2ccccc2SCC(=O)Nc3ccsc3C(=O)OC 2P-507S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)c3cccc(c3)Cl 2P-508S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)c3ccc(cc3)F 2P-510S Cc1cccc(c1)C(=O)Nc2ccccc2SCC(=O)Nc3ccsc3C(=O)OC 2P-511S COC(=O)c1c(ccs1)NC(=O)CSc2cccc(c2Cl)Cl 2P-513S COC(=O)c1c(ccs1)NC(=O)CSc2cc(ccc2Cl)Cl 2P-514S COC(=O)c1c(ccs1)NC(=O)CSc2ccc(cc2)Cl 2P-515S CNS(=O)(=O)c1cc(c(cc1CC(=O)OC)OC)OC 2P-517S COc1cc(c(cc1OC)S(=O)(=O)N2CCOCC2)CC(=O)OC 2P-518S CN(C)S(=O)(=O)c1cc(c(cc1CC(=O)OC)OC)OC 2P-519S COc1cc(c(cc1OC)S(=O)(=O)NCc2ccccc2)CC(=O)OC 2P-521S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)CSc3ccc(cc3)Cl 2P-523S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)CSc3ccc(cc3)Br 2P-524S COC(=O)c1c(ccs1)NC(=O)CN2CCOCC2 2P-525S CCOC(=O)c1cnn(c1N)S(=O)(=O)c2ccc(cc2)C 2P-526S c1cc(c(cc1Cl)Cl)C(=O)OCn2c(=O)c(c(cn2)Cl)Cl 2P-528S COC(=O)c1c(ccs1)NC(=O)CN2CCN(CC2)c3ccccc3F 2P-529S COC(=O)c1c(ccs1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F 2P-530S COC(=O)c1c(ccs1)NC(=O)CN2CCN(CC2)CCc3cccc(c3)C(F)(F)F 2P-531S COC(=O)c1c(ccs1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl 2P-532S Cn1c2c(cn1)/C(=N/O)/CCC2 2P-533S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)CSc3cccc(c3)C(F)(F)F 2P-536S COc1ccc(cc1)SCC(=O)Nc2ccccc2SCC(=O)Nc3ccsc3C(=O)OC 2P-537S COC(=O)c1ccccc1SCC(=O)Nc2ccccc2SCC(=O)Nc3ccsc3C(=O)OC 2P-538S COc1ccc(cc1)n2c(cc3c2CCC(=C3Sc4ccccc4Cl)C=O)c5ccccc5 2P-561S Cc1cccc(c1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)C=O 2P-562S COc1ccc(cc1OC)C(C#N)Nc2ccccc2N 2P-565S Cc1c(c(n(n1)C)Oc2ccccc2)C=O 2P-567S Cc1ccc(c(c1)SC2=C(CCc3c2cc(n3c4ccc(cc4)OC)c5ccccc5)C=O)C 2P-568S COc1ccc(cc1)n2c(cc3c2CCC(=C3Sc4ccccc4)C=O)c5ccccc5 2P-570S c1ccc(cc1)c2cc3c(n2c4ccc(cc4)F)CCCC3=O 2P-572S c1ccc(cc1)c2cc3c(n2c4ccc(cc4)Br)CCCC3=O 2P-573S Cc1c(c(n(n1)C)Oc2ccccc2)/C=C/[N+](=O)[O-] 2P-582S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)Cl)c5ccccc5)/C=N/OC(=O)c6ccccc6 2P-583S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)Cl)c5ccccc5)/C=N/OC(=O)c6ccc(cc6)F 2P-585S Cc1ccc(cc1)C(=O)O/N=C/C2=C(c3cc(n(c3CC2)c4ccc(cc4)Cl)c5ccccc5)Sc6ccc(cc6)C 2P-591S CCn1c(nnc1SCc2ccc(cc2)Cl)c3cc4c(s3)-c5ccccc5CC4 2P-641S c1ccc2c(c1)CCC(=C2Cl)/C=N/OC(=O)C3CC3 2P-642S c1ccc2c(c1)CCC(=C2Cl)/C=N/OC(=O)c3cccs3 2P-643S Cc1ccc(cc1)C(=O)O/N=C/C2=C(c3ccccc3CC2)Cl 2P-644S c1ccc2c(c1)CCC(=C2Cl)/C=N/OC(=O)c3ccc(cc3)F 2P-645S CCn1c(nnc1SCc2cccc(c2)C(F)(F)F)c3cc4c(s3)-c5ccccc5CC4 2P-647S CCn1c(nnc1SCc2ccc(cc2)OC)c3cc4c(s3)-c5ccccc5CC4 2P-649S CCn1c(nnc1SCc2cccc(c2)C)c3cc4c(s3)-c5ccccc5CC4 2P-650S c1ccc2c(c1)CCC(=C2Cl)/C=N/OCc3ccc(cc3Cl)Cl 2P-651S c1ccc2c(c1)CCC(=C2Cl)/C=N/OCc3ccc(cc3)F 2P-652S Cc1ccc(cc1)CO/N=C/C2=C(c3ccccc3CC2)Cl 2P-653S c1ccc2c(c1)CCC(=C2Cl)/C=N/c3ccc(cc3F)F 2P-656S c1ccc2c(c1)CCC(=C2Cl)/C=N/c3ccc(cc3)C(F)(F)F 2P-658S c1ccc2c(c1)CCC(=C2Cl)/C=N/c3ccc(cc3Cl)Cl 2P-659S c1ccc(cc1)NC(=O)O/N=C/C2=C(c3ccccc3CC2)Cl 2P-662S Cc1ccc(cc1)NC(=O)O/N=C/C2=C(c3ccccc3CC2)Cl 2P-663S c1ccc2c(c1)CCC(=C2Cl)/C=N/OC(=O)Nc3ccc(c(c3)Cl)Cl 2P-664S c1ccc-2c(c1)CCc3c2sc(c3)c4nnc(o4)S 2P-667S CSc1nnc(o1)c2cc3c(s2)-c4ccccc4CC3 2P-669S c1ccc-2c(c1)CCc3c2sc(c3)c4nnc(o4)c5ccc(cc5)F 2P-671S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)NNS(=O)(=O)c4ccc(cc4)Cl 2P-680S COC(=O)/C(=C\Nc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)Cl 2P-700 c1cc2c(cc1Cl)c(=O)c(c[nH]2)c3c(cc(cn3)C(F)(F)F)Cl 2P-701 COC(=O)/C(=C\Nc1ccccc1N)/c2c(cc(cn2)C(F)(F)F)Cl 2P-703 CCOC(=O)C(C/C=C/c1ccccc1)C(=O)C 2P-704 CCOC(=O)C(Cc1c(cccc1Cl)F)c2ccno2 2P-707 Cc1c(cccc1Cl)N/C=C(/c2c(cc(cn2)C(F)(F)F)Cl)\C(=O)OC 2P-708 Cc1c(ccc2c1[nH]cc(c2=O)c3c(cc(cn3)C(F)(F)F)Cl)Cl 2P-709 COC(=O)/C(=C\Nc1cc(ccc1F)F)/c2c(cc(cn2)C(F)(F)F)Cl 2P-710 c1ccc(c(c1)N/C=C/C(=O)c2ccc(cc2)F)O 2P-711 c1ccc2c(c1)c(=O)ss2 2P-712 Cc1cc(nc(c1C#N)SCCC(=C(F)F)F)C 2P-714 COC(=O)/C(=C\Nc1ccc(cc1)C(F)(F)F)/c2c(cc(cn2)C(F)(F)F)Cl 2P-716 Cc1cc([nH]c(=O)c1C#N)C 2P-717 Cc1cccc[n+]1CC(=O)c2ccccc2.[Br-] 2P-718 c1ccc(cc1)c2cc3ccccn3c2 2P-720 Cc1cc(nc(c1C#N)Cl)C 2P-721 COC(=O)/C(=C\Nc1ccc2c(c1)OCO2)/c3c(cc(cn3)C(F)(F)F)Cl 2P-722 CC(=O)c1c(cc2n1cccc2)c3ccccc3 2P-726 CCOC(=O)C(Cc1ccccc1)C(=O)C/C=N/OCc2cccc(c2)Cl 2P-727 c1ccc(cc1)Cc2c(c(cn(c2=O)CCc3c[nH]c4c3cccc4)/C=N/OCc5cccc(c5)Cl)O 2P-729 c1ccc(cc1)Cc2c(c(cn(c2=O)Cc3ccc(cc3Cl)Cl)/C=N/OCc4cccc(c4)Cl)O 2P-730 c1ccc(cc1)Cc2c(c(cn(c2=O)CCc3c[nH]cn3)/C=N/OCc4cccc(c4)Cl)O 2P-731 CCOC(=O)C(Cc1ccccc1)c2ccnn2c3ccc(cc3F)F 2P-732 CCOC(=O)C(Cc1ccccc1)c2ccnn2c3cccc(c3)[N+](=O)[O-] 2P-733 c1c(cnc(c1Cl)CC(=O)N)C(F)(F)F 2P-736 c1ccc(cc1)S(=O)(=O)NCc2ccco2 2P-738 c1cc2c(cc1Cn3cc(c(=O)nc3)c4c(cc(cn4)C(F)(F)F)Cl)OCO2 2P-740 COc1ccc(cc1OC)Cn2ccc(c(c2=O)C/C=C/c3ccccc3)O 2P-741 c1ccc(cc1)/C=C/Cc2c(ccn(c2=O)Cc3ccc(cc3Cl)Cl)O 2P-742 c1ccc2c(c1)CC(C2O)Br 2P-744 c1ccc(cc1)/C=C/Cc2c(ccn(c2=O)Cc3cccc(c3)Cl)O 2P-745 c1ccc(cc1)/C=C/Cc2c(ccn(c2=O)Cc3cccc(c3)C(F)(F)F)O 2P-746 C/C(=C/C(=O)c1ccc(cc1)OC)/N(C)C 2P-747 Cc1cc(c(c(n1)Cl)C#N)/C=C/N(C)C 2P-748 CC(=NNC=O)C 2P-802 CCOC(=O)CNC=C(C(=O)c1ccccc1)C(=O)c2ccccc2 2P-804 CC(=NN(CC=C)C=O)C 2P-805 CCOC(=O)/C(=C/N(C)C)/NC=C(C(=O)c1ccccc1)C(=O)c2ccccc2 2P-806 Cc1c(c(nc(n1)C)NCc2ccccc2)I 2P-807 CN1C(=O)N(C(O1)CC(=O)O)c2ccc(cc2)Cl 2P-809 CC1(Cc2c(cc(c(=O)o2)NC=C(C(=O)c3ccccc3)C(=O)c4ccccc4)C(=O)C1)C 2P-810 CN1C(=O)N(C(O1)CC(=O)Nc2ccc(cc2)OC)c3ccc(cc3)Cl 2P-811 Cc1c(c(nc(n1)C)NCCCOC)I 2P-812 Cc1c(c(nc(n1)C)Nc2ccc(cc2)OC)I 2P-813 c1cc(ccc1C(=O)/C=C\C(=O)O)O 2P-814 Cc1cc(c(c(c1)C)S(=O)(=O)NC(Cc2ccc(cc2)C#N)C(=O)O)C 2P-822 Cc1cc2c(cc(c(=O)o2)NC=C(C(=O)c3ccccc3)C(=O)c4ccccc4)c(=O)o1 2P-823 c1ccc(cc1)C(=O)C(=CNc2cc3c(c4ccccc4oc3=O)oc2=O)C(=O)c5ccccc5 2P-824 c1ccc(cc1)C(=O)C(=CNc2cc(c3ccccn3c2=O)C#N)C(=O)c4ccccc4 2P-825 c1ccc(cc1)C(=O)C(=CNc2cnc3ccccn3c2=O)C(=O)c4ccccc4 2P-826 c1ccc(cc1)C(=O)C(=CNc2cc3c(oc2=O)CCCC3=O)C(=O)c4ccccc4 2P-827 CC1(CC2=C(C(C3=C(O2)CC(CC3=O)(C)C)c4c5ccccc5ccc4O)C(=O)C1)C 2P-901 COc1ccc(c(c1)OC)C(=O)/C=C/C(=O)O 2P-902 c1ccnc(c1)COc2ccc(cc2)C=O 2P-903 CCOC(=O)C(=Cc1ccc(cc1)OCc2ccccn2)C#N 2P-909 CCOC(=O)/C(=C\c1ccc(cc1)OCc2cccnc2)/C#N 2P-913 c1ccc(cc1)COC(=O)NCC(=O)O 2P-917 COC(=O)c1c2c(c(cn1)O)C(=O)N(C2=O)Cc3ccccc3 2P-922 COc1ccc(c(c1)/C=C/[N+](=O)[O-])OC 2P-923 c1ccc2c(c1)C(=O)N(C2=O)CCCC(=O)O 2P-934 c1cc(cc(c1)Cl)CNC(=O)/C=C/c2ccc(cc2)OCCCF 2R-0001 c1ccc(cc1)COc2ccc(cc2)/C=C/C(=O)NCc3ccc(cc3)Cl 2R-0006 COc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)OCc3ccccc3 2R-0007 CC(C1C(=O)N(C(=O)N(C1=O)C)C)C(=O)OC 2R-0008 c1ccc(cc1)COc2ccc(cc2)/C=C/C(=O)N3CCOCC3 2R-0009 c1cc(cc(c1)N2CCN(CC2)C3CCc4c(cc[nH]4)C3=O)C(F)(F)F 2R-0012 COc1ccc(cc1)N/C=C(\C#N)/c2ccc(cc2)OCCCF 2R-0013 COC(=O)C(CSC1=NCCS1)NC(=O)OCc2ccccc2 2R-0015 c1ccc(cc1)c2ccc(cc2F)Oc3ccc(cc3Br)[N+](=O)[O-] 2R-0016 c1cc(ccc1COc2ccc(cc2)c3ncc4c(n3)CCCC4=O)C(F)(F)F 2R-0017 c1ccc(cc1)CN2CCN(CC2)C(=O)COc3ccc(cc3)c4nccc(n4)c5cccs5 2R-0018 Cc1ccccc1NC(=O)COc2ccc(cc2)c3nccc(n3)c4cccs4 2R-0019 COc1cccc(c1)NC(=O)COc2ccc(cc2)c3nccc(n3)c4cccs4 2R-0020 CC(C)(C)Oc1ccc(cc1)CC(=O)O 2R-0026 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccccc4 2R-0027 c1cc(ccc1/C(=C/Nc2ccc(cc2)F)/C#N)OCCCF 2R-0028 Cc1ccc(c(c1)N/C=C/C(=O)c2ccc(cc2)OCc3c(cccc3Cl)F)C 2R-0029 c1cc(c(c(c1)Cl)COc2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3)F)F 2R-0030 Cc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)OCc3c(cccc3Cl)F 2R-0031 Cc1ccc(cc1)N/C=C/C(=O)C(C)Oc2ccc(c(c2)F)c3ccccc3 2R-0033 c1ccc(cc1)COc2ccc(cc2)/C=C/C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 2R-0034 c1cc(c(c(c1)Cl)COc2ccc(cc2)c3ccnc4n3ncn4)F 2R-0037 COc1ccc(cc1)NC(=O)COc2ccc(cc2)c3nccc(n3)c4cccs4 2R-0038 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCC(=O)N4CCOCC4 2R-0039 c1ccc(cc1)COc2ccc(cc2)/C=C/C(=O)N3CCN(CC3)c4ccccc4F 2R-0042 Cc1ccc(n1c2ccsc2C(=O)O)C 2R-0045 COc1ccccc1N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccccc4 2R-0046 CC(c1ccnc2n1ncn2)Oc3ccc(c(c3)F)c4ccccc4 2R-0047 Cc1cc(ccc1Br)N/C=C/C(=O)C(C)Oc2ccc(c(c2)F)c3ccccc3 2R-0048 c1cc(c(c(c1)Cl)COc2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3C(F)(F)F)Cl)F 2R-0050 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NC4CCCC4 2R-0051 COc1ccc(cc1OC)CNC(=O)COc2ccc(cc2)c3nccc(n3)c4cccs4 2R-0052 c1cc(sc1)CNC(=O)COc2ccc(cc2)c3nccc(n3)c4cccs4 2R-0053 CC(C)(C)OC(=O)NC(CSCCCC(=O)N1CCCCCC1)C(=O)N2CCCCCC2 2R-0054 c1cc(c(c(c1)Cl)COc2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3)OC(F)(F)F)F 2R-0057 Cc1cc(ccc1Br)N/C=C/C(=O)c2ccc(cc2)OCc3c(cccc3Cl)F 2R-0058 c1cc(ccc1/C(=C/Nc2ccc(cc2)OC(F)(F)F)/C#N)OCCCF 2R-0059 Cc1cccc(c1C)N/C=C/C(=O)c2ccc(cc2)OCc3c(cccc3Cl)F 2R-0060 CC(C)(C)c1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)OCc3c(cccc3Cl)F 2R-0061 Cc1ccc(cc1C)N/C=C/C(=O)c2ccc(cc2)OCc3c(cccc3Cl)F 2R-0062 c1cc(c(c(c1)Cl)COc2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3F)Cl)F 2R-0063 CCCCCCCCOc1ccc(cc1)c2nccc(n2)/C=C(/C(=O)C)\C(=O)OC 2R-0064 CN1C(=O)C(C(=O)N(C1=O)C)(CC(=O)c2ccc(cc2)OC)CC(=O)c3ccc(cc3)OC 2R-0067 CC(C(=O)/C=C/Nc1ccc(cc1)C(c2ccccc2)(c3ccccc3)c4ccccc4)Oc5ccc(c(c5)F)c6ccccc6 2R-0068 Cc1cc2nccc(n2n1)C(C)Oc3ccc(c(c3)F)c4ccccc4 2R-0070 c1ccc(cc1)Cc2c(nc3ccccc3n2)Cl 2R-0071 c1ccc(c(c1)N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccc(cc4Cl)Cl)F 2R-0072 CC(C)(C)OC(=O)CC1C(=O)N(C(=O)N(C1=O)C)C 2R-0074 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccc(cc3)OCc4c(cccc4Cl)F 2R-0075 Cc1cc(n2c(n1)cc(n2)c3c(ccs3)n4cccc4)O 2R-0076 c1cc(ccc1C(F)(F)F)NC(=O)C2CC=CCC2C(=O)O 2R-0077 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccc(cc4Cl)Cl 2R-0078 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)/C=C/c4ccc(cc4)OCc5ccc(cc5Cl)Cl 2R-0080 c1ccc(cc1)COc2ccc(cc2)/C=C/C(=O)c3ccccc3Cl 2R-0081 CC(c1ccn(n1)C(=O)/C=C/c2ccc(cc2)OCc3ccccc3)Oc4ccc(c(c4)F)c5ccccc5 2R-0083 c1cc(ccc1/C=C/C(=O)N2CCOCC2)OCc3ccc(cc3Cl)Cl 2R-0084 c1cc(ccc1F)Sc2ccc(cc2Br)[N+](=O)[O-] 2R-0085 Cc1ccccc1NC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0086 COc1cccc(c1)NC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0087 COc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0088 c1cc(c(c(c1)Cl)COc2ccc(cc2)c3ccn(n3)S(=O)(=O)c4ccc(cc4F)F)F 2R-0090 c1cc(ccc1CNC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl)Cl 2R-0092 c1cc(ccc1/C=C/C(=O)NCc2ccc(c(c2)Cl)Cl)OCc3ccc(cc3Cl)Cl 2R-0093 c1cc(sc1)CNC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0094 CCOC(=O)c1c2ccccn2cc1c3ccc(cc3)C 2R-0095 CC(C(=O)/C=C/Nc1ccc(cc1)Cl)Oc2ccc(c(c2)F)c3ccccc3 2R-0096 CC(=O)c1ccc(cc1)OCCCF 2R-0098 Cc1cc(n2c(n1)cc(n2)c3c(ccs3)n4cccc4)C 2R-0099 c1ccc(cc1)Cc2c(nc3ccccc3n2)NN 2R-0102 c1cc(ccc1/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)Cl)OCc4ccc(cc4Cl)Cl 2R-0104 COc1ccc(cc1OC)CNC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0105 CC(c1ccn(n1)C(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl)Oc4ccc(c(c4)F)c5ccccc5 2R-0106 COc1ccccc1N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccc(cc4Cl)Cl 2R-0107 Cc1ccc(cc1)/C=N/Nc2c(nc3ccccc3n2)Cc4ccccc4 2R-0108 c1cc(cc(c1)S(=O)(=O)n2ccc(n2)c3ccc(cc3)OCc4c(cccc4Cl)F)C(F)(F)F 2R-0112 CCC(C)NC(=O)/C=C/c1ccc(cc1)OCc2ccc(cc2Cl)Cl 2R-0117 CN(Cc1ccccc1)C(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0119 CN1C(=O)C(C(=O)N(C1=O)C)CC2CC(=O)OC2=O 2R-0120 CN(C)/C=C/C(=O)c1ccc(cc1)OCCCF 2R-0122 c1cc(ccc1COc2ccc(cc2)c3ncc4c(n3)/C(=N\O)/CCC4)C(F)(F)F 2R-0123 c1cc(c(c(c1)Cl)COc2ccc(cc2)c3ccn(n3)C(=O)c4ccc(c(c4)Cl)Cl)F 2R-0124 COc1ccc(cc1OC)S(=O)(=O)n2ccc(n2)c3ccc(cc3)OCc4c(cccc4Cl)F 2R-0125 COc1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)OCc4c(cccc4Cl)F 2R-0126 COc1cccc(c1)N/C=C/C(=O)c2ccc(cc2)OCCCF 2R-0127 Cc1ccc(cc1)C(=O)COC(=O)c2ccc(cc2)O 2R-0128 CC(c1ccn(n1)S(=O)(=O)c2ccc(cc2)F)Oc3ccc(c(c3)F)c4ccccc4 2R-0129 Cc1cc(nc(n1)NC(=O)/C(=C(\C)/O)/C#N)C 2R-0130 CN1C(=O)C(C(=O)N(C1=O)C)CC(=O)c2ccc(c(c2)Cl)Cl 2R-0132 COc1ccc(c(c1)/C=N/Nc2c(nc3ccccc3n2)Cc4ccccc4)O 2R-0133 c1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)OCc4c(cccc4Cl)F 2R-0136 c1ccn2c(c1)c(c3c2cc(cc3)Oc4ccc(cc4Br)[N+](=O)[O-])C#N 2R-0139 CC(c1ccn(n1)S(=O)(=O)c2ccc(cc2)Cl)Oc3ccc(c(c3)F)c4ccccc4 2R-0140 c1ccc(cc1)c2nccc(n2)c3ccc(cc3)OCCCF 2R-0141 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)/C=C/c4ccc(cc4)OCc5ccc(cc5)Br 2R-0142 c1ccc(c(c1)N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccc(cc4)Br)F 2R-0143 COC(=O)COc1ccc(cc1)O 2R-0144 c1cc(c(c(c1)Cl)Sc2ccc(cc2Br)[N+](=O)[O-])Cl 2R-0145 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccc(cc4)Br 2R-0146 CN1C(=O)C(C(=O)N(C1=O)C)(CC(=O)c2ccc(cc2)Br)CC(=O)c3ccc(cc3)Br 2R-0147 c1cc(ccc1Sc2ccc(cc2Br)[N+](=O)[O-])Cl 2R-0149 c1cc(ccc1/C=N/NC(=O)c2ccc(cc2)C(F)(F)F)OCCCF 2R-0150 c1cc(ccc1CO/N=C/c2ccc(cc2)OCCCF)Cl 2R-0151 c1ccn2cc(c(c2c1)C(=O)O)c3ccc(cc3)F 2R-0152 CCC(C)NC(=O)/C=C/c1ccc(cc1)OCc2ccc(cc2)Br 2R-0153 c1ccc(c(c1)NC(=O)C2CC=CCC2C(=O)O)F 2R-0154 C=CCn1c(=N)c2ccccc2[nH]c1=S 2R-0155 CCOC(=O)Cc1cccc[n+]1Cc2ccc(cc2)C.[Br-] 2R-0156 CN1C(=O)C(C(=O)N(C1=O)C)CC(=O)c2ccc(cc2)Br 2R-0157 CN1C(=O)C(C(=O)N(C1=O)C)(CC(=O)c2ccc(c(c2)Cl)Cl)CC(=O)c3ccc(c(c3)Cl)Cl 2R-0158 CC(c1ccn(n1)C(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br)Oc4ccc(c(c4)F)c5ccccc5 2R-0159 Cc1ccc(c(c1)C)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 2R-0161 c1cc(ccc1COc2ccc(cc2)/C=C/C(=O)NCc3ccc(c(c3)Cl)Cl)Br 2R-0162 c1ccc2c(c1)cc(cn2)/C=C/C(=O)O 2R-0163 C1C=CC[C@H]([C@H]1C(=O)NCCNC(=O)[C@H]2CC=CC[C@H]2C(=O)O)C(=O)O 2R-0164 Cc1ccc(cc1)N/C=C(\C#N)/c2ccc(cc2)OCCCF 2R-0165 CN1C(=O)C(C(=O)N(C1=O)C)C/C=C/C(=O)OC 2R-0166 c1ccc(cc1)NNC(=O)C2CC=CCC2C(=O)O 2R-0172 Cc1cc(ccc1Br)N/C=C/C(=O)c2ccc(cc2)OCCCF 2R-0176 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)F)OCCCF 2R-0177 c1cc(ccc1C(=O)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OCCCF 2R-0178 CCOC(=O)/C(=C\N(C)C)/c1ccccn1 2R-0180 Cc1ccc(cc1Cl)N/C=C(\C#N)/c2ccc(cc2)OCCCF 2R-0183 c1cc(ccc1CO/N=C/C(C#N)c2ccc(cc2)OCCCF)Cl 2R-0184 COc1ccccc1N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OCc4ccc(cc4)Br 2R-0187 CN1C(=O)C(C(=O)N(C1=O)C)(Cc2ccc(cc2)Br)Cc3ccc(cc3)Br 2R-0189 CC(=O)c1ccc(cc1)OCc2ccc(cc2Cl)Cl 2R-0190 CC(c1ccc(cc1)OCc2c(cccc2Cl)F)O 2R-0192 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)Cl)OCCCF 2R-0193 CCOC(=O)Cc1cccc[n+]1Cc2cccc(c2)Cl.[Br-] 2R-0194 c1ccc2c(c1)c(=N)n(c(=S)[nH]2)c3ccc(cc3)Cl 2R-0195 Cc1cccc(c1)N/C=C/C(=O)c2ccc(cc2)OCCCF 2R-0197 c1csc2c1C3=NC(=O)CN3C(=S)N2 2R-0199 CCCCCCCCOc1ccc(cc1)c2nccc(n2)C=O 2R-0203 C=CCSC1=Nc2ccccc2C3=NC(=O)CN31 2R-0208 Cc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0209 Cc1cccc(c1)N/C=C/C(=O)c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0210 COc1ccc(c(c1)N/C=C/C(=O)c2ccc(cc2)OCc3ccc(cc3Cl)Cl)OC 2R-0211 Cc1cccc(c1)C(=O)NNc2c(nc3ccccc3n2)Cc4ccccc4 2R-0213 COc1ccc(cc1OC)/C=N\n2cnnc2 2R-0214 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2ccccc2 2R-0216 c1ccc(cc1)Cc2c(nc3ccccc3n2)NNS(=O)(=O)c4cccc(c4)C(F)(F)F 2R-0217 c1cc(ccc1c2ccnc(n2)N)OCCCF 2R-0218 c1cc(ccc1/C=C/C(=O)n2ccc(n2)c3ccc(cc3)OCCCF)OCCCF 2R-0219 c1cc(ccc1c2ccnc3n2ncn3)OCc4ccc(cc4Cl)Cl 2R-0220 c1cc(ccc1COc2ccc(cc2)/C=C/C(=O)N3CCN(CC3)c4ccc(cc4)Cl)Br 2R-0221 c1cc(ccc1COc2ccc(cc2)/C=C/C(=O)N3CCOCC3)Br 2R-0222 Cc1ccc(cc1)CNC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br 2R-0223 c1cc(sc1)CNC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br 2R-0224 c1cc(ccc1c2ccn(n2)C(=O)c3ccc(cc3)F)OCCCF 2R-0225 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccc(cc3)OCCCF 2R-0226 c1ccc(cc1)/C=C/C=N\n2cnnc2 2R-0227 CC(=C(C#N)C#N)c1ccccc1 2R-0229 CSC1=Nc2ccccc2C3=NC(=O)CN31 2R-0230 Cc1cccc(c1C)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 2R-0232 c1cc(cc(c1)Br)N/C=C/C(=O)c2ccc(cc2)OCc3ccc(cc3Cl)Cl 2R-0233 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)Cl)OCc3ccc(cc3Cl)Cl 2R-0234 c1cc(ccc1c2ccnc(n2)N)OCc3ccc(cc3Cl)Cl 2R-0235 Cc1cc2nccc(n2n1)c3ccc(cc3)OCc4ccc(cc4Cl)Cl 2R-0236 c1cc(sc1)c2ccnc(n2)c3ccc(cc3)OCC(=O)N4CCCCCC4 2R-0238 COC(c1ccnc(n1)c2ccccn2)OC 2R-0239 COc1cccc(c1)NC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br 2R-0242 Cc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br 2R-0243 COc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br 2R-0244 c1cc(ccc1CNC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br)Cl 2R-0245 c1cc(ccc1CO/N=C/CC(=O)c2ccc(cc2)OCc3ccc(cc3Cl)Cl)Cl 2R-0246 COc1cccc(c1)C(=O)n2ccc(n2)c3ccc(cc3)OCCCF 2R-0249 c1cc(oc1)CNC(=O)C2CC=CCC2C(=O)O 2R-0250 c1cc(ccc1/C=N\n2cnnc2)O 2R-0251 c1cc(ccc1/C=N\n2cnnc2)C#N 2R-0252 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)n3ccc(n3)c4ccc(cc4)OCc5c(cccc5Cl)F 2R-0254 c1cscc1/C=N\n2cnnc2 2R-0255 c1ccc2c(c1)C3=NC(=O)CN3C(=N2)SCc4cccc(c4)Cl 2R-0257 Cc1cc(c(c(c1)C)S(=O)(=O)NNc2c(nc3ccccc3n2)Cc4ccccc4)C 2R-0258 c1cc(ccc1c2ccn(n2)S(=O)(=O)c3ccc(cc3)Br)OCCCF 2R-0259 CC(c1ccn(n1)S(=O)(=O)c2ccc(cc2)Br)Oc3ccc(c(c3)F)c4ccccc4 2R-0260 Cc1ccccc1NC(=O)/C=C/c2ccc(cc2)OCc3ccc(cc3)Br 2R-0261 COC(CN1C(=O)CNC1=S)OC 2R-0265 COC(=O)c1ccc(cc1)/C=N\n2cnnc2 2R-0269 c1ccc(cc1)C/N=C/c2cc(cc(c2O)Br)Br 2R-0601 COC(=O)C(Cc1ccc(cc1)OC(=O)c2cccc(c2)C(F)(F)F)N3Cc4ccccc4C3=O 2R-0602 Cc1c(c(n(n1)C)C)C(=O)O 2R-0605 Cc1ccc(cc1)S(=O)(=O)c2ccc(cn2)[N+](=O)[O-] 2R-0608 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3ccccc3 2R-0609 C=CCC(c1nnc2n1cccc2C(F)(F)F)(F)F 2R-0610 COc1cccc(c1)C(=O)OCC(Cc2ccccc2)N3Cc4ccccc4C3=O 2R-0612 CCc1ccc(cc1)NC(=O)/C=C/C(=O)O 2R-0614 c1ccc(cc1)C2C(O2)C(=O)c3cccc[n+]3[O-] 2R-0615 c1cc(c2nnc(n2c1)C(F)(F)Cl)[N+](=O)[O-] 2R-0617 Cc1ccc(cc1)/C=N/NC(=O)C(Cc2ccc(cc2)O)N3Cc4ccccc4C3=O 2R-0618 Cc1cc(nc2c1c(n[nH]2)N)C 2R-0620 COC(=O)C(Cc1ccc(cc1)OC(=O)Nc2ccc(cc2)Cl)N3Cc4ccccc4C3=O 2R-0621 CCOC(=O)c1c(nn(c1C)c2c(cccn2)C(F)(F)F)C 2R-0622 Cc1c(c(n(n1)C)C)C(=O)NN 2R-0625 Cc1ccc(cc1)S(=O)(=O)c2c(cccn2)N 2R-0626 c1cc(c(cc1F)Cl)CON2CCS(=O)(=O)CC2 2R-0627 Cc1cccn2c1nc(c2Br)c3ccc(cc3)OC 2R-0628 Cc1ccccc1C(=O)Oc2ccc(cc2)CC(C(=O)OC)N3Cc4ccccc4C3=O 2R-0629 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)CC(C(=O)OC)N3Cc4ccccc4C3=O 2R-0630 COC(=O)C(Cc1ccc(cc1)OC(=O)c2cccs2)N3Cc4ccccc4C3=O 2R-0631 COc1cc(ccc1C(=O)OC)NC(=O)Nc2ccc(cc2)Cl 2R-0633 c1cc2c(c[nH]c2nc1)Br 2R-0634 c1cc2nnc(n2cc1[N+](=O)[O-])C(F)(F)F 2R-0635 c1ccc2c(c1)c(c[nH]2)CC(C(=O)Nc3ccc(cc3F)Cl)N4CCS(=O)(=O)CC4 2R-0636 c1cc(ccc1CON2CCS(=O)(=O)CC2)Cl 2R-0637 Cc1cc(n(n1)c2ccc(cn2)[N+](=O)[O-])C 2R-0638 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2cc(cc(c2O)Br)Br 2R-0641 COc1cc(ccc1C(=O)OC)NC(=O)Nc2cccc(c2)F 2R-0643 COC(=O)C(Cc1ccc(cc1)OC(=O)c2ccccc2Cl)N3Cc4ccccc4C3=O 2R-0647 CC(C)CC(C(=O)OC)N1Cc2ccccc2C1=O 2R-0648 c1ccc2c(c1)nc(s2)SC(CO)F 2R-0649 CC(c1cc2cc(cc(c2o1)OC)Br)O 2R-0650 c1ccc(cc1)Cn2c3ccccc3nc2c4ccn(n4)C(=O)c5ccc(cc5)I 2R-0653 c1ccc(cc1)Cn2c3ccccc3nc2c4ccn(n4)C(=O)c5ccc(cc5)Cl 2R-0654 c1ccc(cc1)Cn2c3ccccc3nc2c4ccn(n4)C(=O)c5ccccc5C(F)(F)F 2R-0655 COc1cc(ccc1C(=O)OC)NC(=S)NC(=O)c2ccccc2 2R-0656 c1ccc(cc1)CC(CO)NCC(C(F)(F)F)O 2R-0658 CCOC(=O)C(F)(F)S(=O)(=O)c1nc2ccccc2s1 2R-0661 c1ccc(cc1)C(CO)NCC(C(F)(F)F)O 2R-0662 CC(C)CC(C(=O)Nc1ccc(cc1)OC)N2Cc3ccccc3C2=O 2R-0663 c1ccc(cc1)c2cn3cc(ccc3n2)I 2R-0664 COc1cccc(c1)C(=O)Nc2ccc(cn2)I 2R-0665 Cc1cc(cnc1NC(=O)c2cccc(c2)OC)I 2R-0666 COc1c(cccn1)[N+](=O)[O-] 2R-0668 CC(C)CC(C(=O)Nc1ccc(cc1)I)N2Cc3ccccc3C2=O 2R-0670 C1CS(=O)(=O)CCN1CC(=O)NN 2R-0671 Cc1ccccc1C(=O)Nc2c(cc(cn2)I)C 2R-0672 Cc1cc(cnc1NC(=O)c2ccc(cc2)Cl)I 2R-0673 COc1cc(c(cc1C(=O)OC)Br)NC(=O)c2ccco2 2R-0674 COc1ccc(c(c1)NC(=O)C(Cc2c[nH]c3c2cccc3)N4CCS(=O)(=O)CC4)OC 2R-0676 CC(=O)Nc1ccc(c(c1)O)C(=O)OC 2R-0677 CCOC(CNCC(C(F)(F)F)O)OCC 2R-0678 c1cc(nn2c1nnc2C(F)F)Cl 2R-0679 Cc1cc(nc2c1c(n[nH]2)n3cccc3)C 2R-0680 COc1ccc(cc1)/C=N/NC(=O)CN2CCS(=O)(=O)CC2 2R-0681 COc1cc(c(cc1C(=O)O)Br)N 2R-0683 Cc1cc(n(n1)c2c(cccn2)C(F)(F)F)C 2R-0684 Cc1ccc(cc1C)NC(=O)C(Cc2ccccc2)N3CCS(=O)(=O)CC3 2R-0685 Cc1ccc(n1c2ccc(cn2)I)C 2R-0686 CCOC(=O)c1cn2c(cccc2n1)C 2R-0687 c1ccc2c(c1)CN(C2=O)c3ccccc3C(=O)O 2R-0689 Cc1cc(cnc1NC(=O)c2ccc(cc2)C(F)(F)F)I 2R-0690 Cc1cccn2c1nc(c2)c3cccc(c3)C(F)(F)F 2R-0691 Cc1cccc(c1)C(=O)Oc2cc(ccc2C(=O)OC)NC(=O)C 2R-0692 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=O)CN2CCS(=O)(=O)CC2 2R-0693 CC(C)(C)c1ccc(cc1)/C=N/NC(=O)CN2CCS(=O)(=O)CC2 2R-0694 COc1ccc(c(c1)/C=N/NC(=O)CN2CCS(=O)(=O)CC2)O 2R-0695 c1cc(sc1)/C=N/NC(=O)CN2CCS(=O)(=O)CC2 2R-0696 CC(=O)Nc1ccc(c(c1)OC(=O)c2cccs2)C(=O)OC 2R-0698 CCOC(CCNCC(C(F)(F)F)O)OCC 2R-0699 c1ccc(cc1)C(C(F)(F)F)O 2R-0700 c1cc(c(c(c1)Cl)COc2ccc(cc2)c3ccnc(n3)N)F 2R-0701 COC(=O)C(Cc1ccc(cc1)OC(=O)c2ccc(cc2)Cl)N3Cc4ccccc4C3=O 2R-0702 CS(=O)(=O)c1ccccc1 2R-0703 C/C(=C(/CC(=O)OC)\C(=O)OC)/NCc1ccc(c(c1)OC)OC 2R-0800 CC1=C(CC(=O)N1Cc2ccc(c(c2)OC)OC)C(=O)OC 2R-0801 Cc1ccc(cc1Cl)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 2R-0803 COc1cc(cc(c1)OC)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 2R-0804 CCCCCCCn1ccc(c(c1=O)CC(=O)OC)O 2R-0806 CCCCN1C(C(CCC1=O)C(=O)OCC(=O)c2ccc(cc2)Cl)c3ccccc3 2R-0807 COC(=O)c1c(noc1c2cn(nn2)c3ccc(cc3)[N+](=O)[O-])c4ccccc4Cl 2R-0808 c1ccc(cc1)C2C(CCC(=O)N2C3CCCCC3)C(=O)O 2R-0809 COc1ccccc1Cn2ccc(c(c2=O)CC(=O)OC)O 2R-0810 COc1ccn(c(=O)c1CC(=O)OC)CCc2c[nH]c3c2cccc3 2R-0812 c1ccc2c(c1)c(c[nH]2)CCNc3c(cccn3)[N+](=O)[O-] 2R-0813 C/C(=C\[N+](=O)[O-])/N(C)C 2R-0814 Cc1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] 2R-0815 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccc(cc3)Cl 2R-0816 Cc1c(c(n(n1)c2cc(cc(c2)Cl)Cl)O)CC(=O)OC 2R-0817 Cc1cccc(n1)n2cc(nc2)C(=O)N3CCN(CC3)C 2R-0818 Cc1cccc(n1)n2cc(nc2)C(=O)Nc3ccccc3C(=O)N 2R-0819 Cc1cccc(n1)n2cc(nc2)C(=O)Nc3ccc(cc3)C(=O)OC 2R-0820 Cc1cccc(n1)n2cc(nc2)C(=O)Nc3ccc(cc3)N4CCOCC4 2R-0821 CC(=O)C1(C(C1(C#N)C#N)c2ccc(cc2)Cl)C(=O)C 2R-0822 Cc1cc(nc(n1)NCCc2c[nH]c3c2cccc3)C 2R-0827 c1cc(c(cc1C(F)(F)F)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cl 2R-0828 CCCCCC1CCC(CC1)c2ccc(cc2)/N=C/c3ccc4c(c3)OCO4 2R-0830 Cc1cccc(n1)n2cc(nc2)C(=O)N3CCN(CC3)c4cccc(c4)Cl 2R-0831 Cc1cccc(n1)n2cc(nc2)C(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 2R-0832 CCCCCC1CCC(CC1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Br 2R-0833 CCOC(CCNC(=O)c1cn(cn1)c2cccc(n2)C)OCC 2R-0834 Cc1csc(n1)Nc2nccc(n2)c3c(nc(s3)c4ccc(cc4)Cl)C 2R-0838 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)c3ccc(cc3)[N+](=O)[O-] 2R-0839 CCOC(=O)c1ccc(cc1)n2c(c(nn2)[N+](=O)[O-])C 2R-0840 Cc1ccc(cc1Cl)n2c(c(nn2)[N+](=O)[O-])C 2R-0841 Cc1c(nnn1c2cc(cc(c2)Cl)Cl)[N+](=O)[O-] 2R-0842 CC1(CC(=O)C2(C(C2(C#N)C#N)c3ccc(cc3)Cl)C(=O)C1)C 2R-0843 CCCCCC1CCC(CC1)c2ccc(cc2)/N=C/C(C#N)C#N 2R-0844 CC1=C(CC(=O)N1CCc2ccccc2)C(=O)OC 2R-0845 CC1=C(/C(=C/N(C)C)/C(=O)N1CCc2ccccc2)C(=O)OC 2R-0846 c1cc(ccc1C2C(C2(C#N)C#N)(C#N)C#N)Cl 2R-0847 COc1ccc(cc1)N2C(C(CCC2=O)C(=O)O)c3ccccc3 2R-0848 Cc1cccc(n1)n2cc(nc2)C(=O)N3CCN(CC3)c4cccc(c4)C(F)(F)F 2R-0851 Cc1c(c(n2c(n1)ncn2)C)Cc3cccc(c3)F 2R-0852 CC(=O)C1(C(C1(C#N)C#N)c2ccc(cc2)F)C(=O)C 2R-0853 CC(C)(CCl)C(=O)NCCc1c[nH]c2c1cccc2 2R-0855 CN(C)/C=C/c1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] 2R-0856 C/C(=C\C(=O)c1ccc2ccccc2c1)/N(C)C 2R-0857 c1ccc(cc1)C2C(CCC(=O)N2C3CC3)C(=O)O 2R-0859 Cc1c(c(n2cnc(c2n1)C#N)C)Cc3cccc(c3)F 2R-0860 Cc1c(c(n2c(n1)ncn2)C)Cc3c(cccc3Cl)Cl 2R-0861 Cc1csc(n1)Nc2nccc(n2)c3c(nc(s3)c4ccccc4)C 2R-0862 c1ccc(cc1)Oc2ncc(cn2)c3ccc(cc3)Cl 2R-1000 c1cc(ccc1c2cnc(nc2)Oc3ccc(cc3)F)Cl 2R-1001 Cc1cccc(c1C)Oc2ncc(cn2)c3ccc(cc3)Cl 2R-1002 CC(C)(C)c1ccc(cc1)Oc2ncc(cn2)c3ccc(cc3)Cl 2R-1003 c1cc(cc(c1)Oc2ncc(cn2)c3ccc(cc3)Cl)C(F)(F)F 2R-1004 Cc1cccc(c1)Oc2ncc(cn2)c3ccc(cc3)Cl 2R-1005 c1cc(ccc1c2cnc(nc2)Oc3cc(ccc3Cl)Cl)Cl 2R-1006 Cc1ccc(cc1)NC(=O)NNC(=O)c2c(nns2)C 2R-1007 Cc1cc(nc2c1c(c(s2)C(=O)NN)n3cccc3)C 2R-1008 c1ccc(cc1)n2c(=O)ccc(n2)O 2R-1011 Cc1ccc(cc1)/C=N/NC(=O)c2c(c3c(cc(nc3s2)C)C)n4cccc4 2R-1014 Cc1cc(nc2c1c(c(s2)C(=O)NNS(=O)(=O)c3ccc(cc3)Br)n4cccc4)C 2R-1015 Cc1cc(nc2c1c(c(s2)C(=O)NNS(=O)(=O)c3ccc(cc3)F)n4cccc4)C 2R-1016 Cc1cc(nc2c1c(c(s2)C(=O)NNS(=O)(=O)c3ccccc3)n4cccc4)C 2R-1017 Cc1cc(nc2c1c(c(s2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl)n4cccc4)C 2R-1018 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(c3c(cc(nc3s2)C)C)n4cccc4 2R-1019 Cc1cc(nc2c1c(c(s2)C(=O)NNS(=O)(=O)c3ccc(cc3)NC(=O)C)n4cccc4)C 2R-1020 c1ccc(cc1)n2c(=O)ccc(n2)OC(=O)c3ccc(cc3)F 2R-1021 c1ccc2cc(ccc2c1)Oc3ncc(cn3)c4ccc(cc4)Cl 2R-1024 c1ccc2c(c1)cccc2Oc3ncc(cn3)c4ccc(cc4)Cl 2R-1025 c1ccc(cc1)n2c(=O)ccc(n2)Oc3ncc(cn3)c4ccc(cc4)Cl 2R-1026 COC(=O)c1c(ccs1)Oc2ncc(cn2)c3ccc(cc3)Cl 2R-1027 Cc1cc(ccc1Oc2ncc(cn2)c3ccc(cc3)Cl)Cl 2R-1028 c1cc2c(ccc(c2nc1)Oc3ncc(cn3)c4ccc(cc4)Cl)Cl 2R-1029 COc1ccc(cc1)C(=O)Oc2ccc(=O)n(n2)c3ccccc3 2R-1030 c1ccc(cc1)n2c(=O)ccc(n2)OC(=O)c3cccs3 2R-1031 c1ccc(cc1)n2c(=O)ccc(n2)OC(=O)c3cccc(c3)Cl 2R-1032 c1ccc(cc1)n2c(=O)ccc(n2)OC(=O)c3ccc(cc3)Cl 2R-1033 c1ccc(cc1)C(=O)Oc2ccc(=O)n(n2)c3ccccc3 2R-1035 Cc1c(c2ccccc2[nH]1)C(=O)C(=O)N3CCOCC3 2R-1036 Cc1c(c2ccccc2[nH]1)C(=O)C(=O)NC 2R-1037 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3ccc(cc3)Cl)Cl 2R-1060 CCn1c(=O)cc(c(n1)c2ccccc2)Cl 2R-1061 c1ccc(cc1)c2c(cc(nn2)S)N3CCCCC3 2R-1063 c1cc2c(cc1Cl)C(=O)/C(=C/C(=O)O)/CS2 2R-1064 c1ccc(cc1)Cn2c(=O)cc(c(n2)c3ccccc3)N4CCCCC4 2R-1066 c1ccc(cc1)S(=O)(=O)N2CCC3(CC2)CO3 2R-1069 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3ccc(cc3)Cl)N4CCCCC4 2R-1070 Cc1ccccc1Cn2c(=O)cc(c(n2)c3ccccc3)N4CCCCC4 2R-1071 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3c(cccc3Cl)Cl)N4CCCCC4 2R-1072 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3cccc(c3)Cl)N4CCCCC4 2R-1073 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3ccccc3Cl)N4CCCCC4 2R-1074 CC(C)(C)c1ccc(cc1)Cn2c(=O)cc(c(n2)c3ccccc3)N4CCCCC4 2R-1075 COc1ccc(cc1)Cn2c(=O)cc(c(n2)c3ccccc3)N4CCCCC4 2R-1076 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3ccc(cc3Cl)Cl)N4CCCCC4 2R-1077 Cc1ccc(cc1)SCC2(CCN(CC2)S(=O)(=O)c3ccccc3)O 2R-1079 c1ccc-2c(c1)CCc3c2n[nH]c(=O)c3 2R-1080 COC(=O)c1ccc(cc1)Cn2c(=O)cc(c(n2)c3ccccc3)N4CCCCC4 2R-1081 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3ccc(cc3)F)N4CCCCC4 2R-1082 C=CCn1c(=O)cc(c(n1)c2ccccc2)N3CCCCC3 2R-1083 c1ccc(cc1)Cn2c(=O)cc3c(n2)-c4ccccc4CC3 2R-1084 Cc1ccc(cc1)Cn2c(=O)cc(c(n2)c3ccccc3)N4CCCCC4 2R-1085 Cc1cccc(c1)Cn2c(=O)cc(c(n2)c3ccccc3)N4CCCCC4 2R-1086 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3ccc(c(c3)Cl)Cl)N4CCCCC4 2R-1087 c1ccc(cc1)c2c(cc(=O)n(n2)Cc3cccc(c3)F)N4CCCCC4 2R-1090 Cn1c(=O)cc(c(n1)c2ccccc2)N3CCCCC3 2R-1091 CCOC(=O)Cn1c(=O)cc(c(n1)c2ccccc2)N3CCCCC3 2R-1093 C1CCc2c(nc(s2)N)C1.I 2R-1120 Cc1ccc(cc1)C(=O)ON2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1121 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)OC(=O)C6CC6 2R-1126 Cc1ccc(cc1)C(=O)NNC(=O)C(=O)c2c3ccccc3[nH]c2c4ccccc4 2R-1128 c1ccc(cc1)c2c(c3ccccc3[nH]2)C(=O)C(=O)NNC(=O)c4ccccc4 2R-1129 C1CCc2c(nc(s2)N)C1 2R-1130 Cc1cccc(c1)C(=O)ON2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1133 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)c6ccc(cc6)C(=O)NC7CC7 2R-1136 CCNC(=O)c1ccc(cc1)N2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1137 c1cc(c(cc1Cl)Cl)c2cn3c4c(sc3n2)CCCC4 2R-1138 CC(C)NC(=O)c1ccc(cc1)N2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1139 C=CCNC(=O)c1ccc(cc1)N2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1140 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)c6ccc(cc6)C(=O)N7CCOCC7 2R-1141 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)OCc6ccc(cc6)Cl 2R-1142 Cc1ccccc1NC(=O)c2ccc(cc2)N3C(=O)C4C5c6ccccc6C(C4C3=O)c7c5cccc7 2R-1144 COc1ccc(cc1)NC(=O)c2ccc(cc2)N3C(=O)C4C5c6ccccc6C(C4C3=O)c7c5cccc7 2R-1145 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)c6ccc(cc6)C(=O)Nc7cccc(c7)C(F)(F)F 2R-1147 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)CC(=O)N6CCOCC6 2R-1148 C=CCNC(=O)CN1C(=O)C2C3c4ccccc4C(C2C1=O)c5c3cccc5 2R-1150 c1cc(c(cc1Cl)Cl)c2c(n3c4c(sc3n2)CCCC4)C=O 2R-1152 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)OC(=O)c6cccc(c6)Cl 2R-1153 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)OC(=O)c6ccccc6Cl 2R-1154 CC(C)(C)c1ccc(cc1)CON2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1155 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)OCc6ccc(cc6)F 2R-1156 COC(=O)CN1C(=O)C2C3c4ccccc4C(C2C1=O)c5c3cccc5 2R-1157 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)N 2R-1158 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)OCc6ccc(c(c6)Cl)Cl 2R-1159 C=CCON1C(=O)C2C3c4ccccc4C(C2C1=O)c5c3cccc5 2R-1161 CCON1C(=O)C2C3c4ccccc4C(C2C1=O)c5c3cccc5 2R-1162 CCOC(=O)CON1C(=O)C2C3c4ccccc4C(C2C1=O)c5c3cccc5 2R-1163 COc1ccc(cc1)NC(=O)CN2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1164 c1ccc(cc1)C(=O)ON2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 2R-1166 c1cc(ccc1c2cn3c4c(sc3n2)CCCC4)Cl 2R-1168 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)C=O)Cl 2R-1171 Cc1c(n2ccccc2n1)C(=O)CC(c3ccc(cc3)Cl)O 2R-1182 Cc1cccc(c1C)Oc2c(cnc(n2)c3ccccc3)OC 2R-1183 Cc1c(n2ccccc2n1)C(=O)/C=C/c3ccc(cc3)[N+](=O)[O-] 2R-1184 Cc1c(n2ccccc2n1)C(=O)/C=C/c3ccc(cc3)OC 2R-1186 Cc1c(n2ccccc2n1)C(=O)/C=C/c3cccc(c3)[N+](=O)[O-] 2R-1187 CC(C)(C)c1ccc(cc1)Oc2c(cnc(n2)c3ccccc3)OC 2R-1193 Cc1c(n2ccccc2n1)C(=O)CSc3ccc(cc3)Cl 2R-1195 Cc1ccc(cc1)/C=C/C(=O)c2c(nc3n2cccc3)C 2R-1196 Cc1ccc(cc1)SCC(=O)c2c(nc3n2cccc3)C 2R-1197 Cc1c(n2ccccc2n1)C(=O)CSc3ccccc3 2R-1198 Cc1c(n2ccccc2n1)C(=O)CSc3ccc(cc3)Br 2R-1199 Cc1ccccc1Oc2c(cnc(n2)c3ccccc3)OC 2R-1200 Cc1cccc(c1)Oc2c(cnc(n2)c3ccccc3)OC 2R-1201 Cc1cc(ccc1Oc2c(cnc(n2)c3ccccc3)OC)Cl 2R-1202 Cc1c(n2ccccc2n1)C(=O)CSc3cccc(c3)Cl 2R-1204 Cc1c(n2ccccc2n1)C(=O)CSc3ccccc3Cl 2R-1205 Cc1c(n2ccccc2n1)C(=O)CSc3ccc(cc3Cl)Cl 2R-1206 Cc1c(n2ccccc2n1)C(=O)CSc3cccc(c3)C(F)(F)F 2R-1207 COc1cnc(nc1Oc2cccc(c2)[N+](=O)[O-])c3ccccc3 2R-1208 COc1cnc(nc1Oc2ccc(c3c2cccc3)Cl)c4ccccc4 2R-1209 Cc1c(n2ccccc2n1)C(=O)CSc3ccc(cc3)OC 2R-1210 Cc1ccc(cc1)S(=O)(=O)NNC(=O)/C=C/c2ccc(cc2)Cl 2R-1240 c1ccc(cc1)C(=O)NNC(=O)/C=C/c2ccc(cc2)Cl 2R-1242 Cc1cccc(c1)C(=O)NNC(=O)/C=C/c2ccc(cc2)Cl 2R-1243 c1ccc(cc1)CSC\2=Nc3ccccc3/C2=N/Nc4ccccc4 2R-1246 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=O)N2 2R-1251 c1cc(ccc1/C=C/C(=O)NNC(=O)c2ccc(cc2)Cl)Cl 2R-1253 c1cc(ccc1/C=C/C(=O)NNC(=O)c2ccc(c(c2)Cl)Cl)Cl 2R-1254 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=S)N2 2R-1255 C=CCSc1nc2c3ccccc3sc2c(n1)O 2R-1300 c1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)O 2R-1301 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)O 2R-1302 c1ccc2c(c1)c(c(s2)C(=O)NN)n3cccc3 2R-1303 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NN 2R-1304 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NN 2R-1305 C=CCSc1nc2c3ccccc3sc2c(n1)Cl 2R-1306 c1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)Cl 2R-1307 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)Cl 2R-1308 CSc1nc2c3ccccc3sc2c(n1)N4CCCC4 2R-1310 C=CCSc1nc2c3ccccc3sc2c(n1)N4CCOCC4 2R-1313 CC(C)Nc1c2c(c3ccccc3s2)nc(n1)SCC=C 2R-1314 C=CCNc1c2c(c3ccccc3s2)nc(n1)SCC=C 2R-1315 c1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)N5CCCC5 2R-1316 c1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)NC5CCCCC5 2R-1317 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)NCC=C 2R-1319 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)NC5CC5 2R-1320 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)N5CCOCC5 2R-1322 CSc1nc2c3ccccc3sc2c(n1)Sc4ccccc4 2R-1323 CSc1nc2c3ccccc3sc2c(n1)Sc4ccc(cc4)Cl 2R-1324 COc1cccc(c1)Sc2c3c(c4ccccc4s3)nc(n2)SC 2R-1325 COC(=O)c1ccccc1Sc2c3c(c4ccccc4s3)nc(n2)SC 2R-1326 CSc1nc2c3ccccc3sc2c(n1)Sc4ccc(cc4)F 2R-1327 Cc1ccc(cc1)Sc2c3c(c4ccccc4s3)nc(n2)SCc5ccccc5 2R-1328 COc1ccc(cc1)Sc2c3c(c4ccccc4s3)nc(n2)SCc5ccccc5 2R-1329 c1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)Sc5ccccc5 2R-1331 C=CCSc1nc2c3ccccc3sc2c(n1)Sc4ccccc4 2R-1332 C=CCSc1nc2c3ccccc3sc2c(n1)Sc4ccc(cc4)Cl 2R-1333 COC(=O)c1ccccc1Sc2c3c(c4ccccc4s3)nc(n2)SCC=C 2R-1334 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)SCc5cccc(c5)C(F)(F)F 2R-1335 CSc1nc2c3ccccc3sc2c(n1)Oc4ccc(cc4)F 2R-1336 CSc1nc2c3ccccc3sc2c(n1)Oc4ccc5ccccc5c4 2R-1337 C=CCSc1nc2c3ccccc3sc2c(n1)Oc4ccccc4 2R-1340 Cc1ccccc1Oc2c3c(c4ccccc4s3)nc(n2)SCC=C 2R-1341 c1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)Oc5ccc6ccccc6c5 2R-1342 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)Oc5cccc(c5)C(F)(F)F 2R-1343 Cc1ccc(cc1)CSc2nc3c4ccccc4sc3c(n2)Oc5ccccc5 2R-1344 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NNC(=O)c3ccccc3 2R-1345 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NNC(=O)c3ccc(cc3)OC 2R-1347 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NNC(=O)c3ccc(cc3)Cl 2R-1348 Cc1ccc(cc1)C(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)C 2R-1349 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NNC(=O)c3ccc(cc3)F 2R-1350 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N/N=C/c3ccc(cc3)F 2R-1351 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N/N=C/c3ccc(cc3)OC 2R-1353 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N/N=C/c3cccc(c3)Cl 2R-1354 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N/N=C/c3ccc(cc3)OC(F)(F)F 2R-1355 Cc1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)C 2R-1356 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl 2R-1357 c1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccccc3 2R-1358 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NNS(=O)(=O)c3ccc(cc3)F 2R-1359 Cn1c2ccccc2nc1C(F)(F)F 2R-1501 C#CCn1c2ccccc2nc1C(F)(F)F 2R-1502 CCn1c2ccccc2nc1C(F)(F)F 2R-1503 C=CCn1c2ccccc2nc1C(F)(F)F 2R-1504 COc1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccc(cc3)OC 2R-1507 COc1ccc(cc1)NC(=O)c2csc(n2)Cc3ccc(cc3)Cl 2R-1508 c1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccc(cc3)Cl 2R-1509 COc1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccc(cc3)Cl 2R-1510 CC(C)(C)C(=O)Cn1c2ccccc2nc1C(F)(F)F 2R-1511 COc1cnc(nc1Cl)c2cccc(c2)C(F)(F)F 2R-1512 COc1cnc(nc1OC)c2cccc(c2)C(F)(F)F 2R-1513 COc1cnc(nc1SCC(=O)OC)c2cccc(c2)C(F)(F)F 2R-1514 COc1cnc(nc1Sc2ccccc2)c3cccc(c3)C(F)(F)F 2R-1515 COc1cnc(nc1Oc2ccccc2)c3cccc(c3)C(F)(F)F 2R-1516 COc1cnc(nc1Oc2cccc(c2)C(F)(F)F)c3cccc(c3)C(F)(F)F 2R-1517 COc1ccc(cc1)Cc2nc(cs2)C(=O)Nc3cc(cc(c3)Cl)Cl 2R-1526 COc1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccc(cc3)F 2R-1527 c1ccc(cc1)Cn2c3ccccc3nc2C(F)(F)F 2R-1528 COc1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccccc3 2R-1529 COc1ccc(cc1)Cc2nc(cs2)C(=O)N3CCOCC3 2R-1530 CC(C)(C)c1ccc(cc1)Cn2c3ccccc3nc2C(F)(F)F 2R-1531 Cc1ccc(cc1)Cn2c3ccccc3nc2C(F)(F)F 2R-1532 COc1ccc(cc1)Cc2nc(cs2)C(=O)Nc3cccc(c3)C(F)(F)F 2R-1533 c1ccc2c(c1)nc(n2Cc3ccc(cc3)F)C(F)(F)F 2R-1535 Cc1cccc(c1)Cn2c3ccccc3nc2C(F)(F)F 2R-1536 Cc1ccccc1Cn2c3ccccc3nc2C(F)(F)F 2R-1537 COc1ccc(cc1)Cc2nc(cs2)C(=O)NCc3ccc(cc3)OC 2R-1538 c1cc(ccc1Cc2nc(cs2)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl 2R-1541 c1cc(ccc1Cc2nc(cs2)C(=O)Nc3ccc(cc3)F)Cl 2R-1542 c1ccc2c(c1)nc(n2Cc3ccc(cc3)Cl)C(F)(F)F 2R-1544 c1ccc2c(c1)nc(n2Cc3cccc(c3)Cl)C(F)(F)F 2R-1545 c1ccc(c(c1)Cn2c3ccccc3nc2C(F)(F)F)Cl 2R-1546 COC(=O)Cn1c2ccccc2nc1C(F)(F)F 2R-1547 c1cc(ccc1Cc2nc(cs2)C(=O)N3CCOCC3)Cl 2R-1548 c1cc(ccc1Cc2nc(cs2)C(=O)NCc3ccc(cc3)Cl)Cl 2R-1550 CCOC(=O)c1nc(no1)c2cccc(c2)Cl 2R-1551 c1cc(ccc1c2nc(on2)CC(=O)O)Cl 2R-1555 c1ccc2c(c1)nc(n2Cc3c(cccc3Cl)Cl)C(F)(F)F 2R-1556 c1ccc2c(c1)nc(n2Cc3cccc(c3)[N+](=O)[O-])C(F)(F)F 2R-1557 COc1ccc(cc1)CNC(=O)c2csc(n2)Cc3ccc(cc3)Cl 2R-1558 COc1ccccc1CNC(=O)c2csc(n2)Cc3ccc(cc3)Cl 2R-1559 c1cc(ccc1Cc2nc(cs2)C(=O)N3CCCCC3)Cl 2R-1560 c1ccc2c(c1)nc(n2CC(=O)c3ccc(cc3)Cl)C(F)(F)F 2R-1561 CC(=O)Cn1c2ccccc2nc1C(F)(F)F 2R-1562 c1ccc2c(c1)nc(n2Cc3ccc(c(c3)Cl)Cl)C(F)(F)F 2R-1563 CCOC(=O)c1nc(no1)c2cccc(c2)C(F)(F)F 2R-1565 CCOC(=O)Cc1nc(no1)c2cccc(c2)C(F)(F)F 2R-1566 c1ccc2c(c1)nc(n2Cc3ccc(cc3Cl)Cl)C(F)(F)F 2R-1567 CC(C(=O)O)n1c2ccccc2nc1C(F)(F)F 2R-1568 c1ccc2c(c1)nc(n2CC(=O)c3ccc(cc3)F)C(F)(F)F 2R-1569 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NNC(=O)c3cccc(c3)C(F)(F)F 2R-1570 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N/N=C/c3ccc(cc3)Cl 2R-1571 Cc1ccc(cc1)/C=N/NC(=O)C2CCN(CC2)S(=O)(=O)c3ccccc3 2R-1572 c1cc(cc(c1)C(F)(F)F)CC(=S)N 2R-1573 COc1ccc(cc1)Cc2nc(cs2)C(=O)NCc3ccccc3OC 2R-1574 COc1ccc(cc1)Cc2nc(cs2)C(=O)N3CCCCC3 2R-1575 c1cc(cc(c1)C(F)(F)F)Cc2nc(cs2)C(=O)O 2R-1577 c1cc(cc(c1)C(F)(F)F)c2nc(on2)CC(=O)O 2R-1579 COc1ccc(cc1)NC(=O)Cc2nc(no2)c3cccc(c3)C(F)(F)F 2R-1580 COc1ccc(cc1)NC(=O)Cn2c3ccccc3nc2C(F)(F)F 2R-1581 Cc1ccc(cc1)NC(=O)Cn2c3ccccc3nc2C(F)(F)F 2R-1584 Cc1cccc(c1)NC(=O)Cn2c3ccccc3nc2C(F)(F)F 2R-1585 Cc1ccccc1NC(=O)Cn2c3ccccc3nc2C(F)(F)F 2R-1586 c1cc(cc(c1)C(F)(F)F)Cc2nc(cs2)C(=O)Nc3cc(cc(c3)Cl)Cl 2R-1589 Cc1ccc(cc1)/C=N/NC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 2R-1591 CC/C=N/NC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 2R-1592 COc1ccc(cc1OC)/C=N/NC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 2R-1593 c1ccc(cc1)Oc2ccc(cc2)/C=N/NC(=O)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 2R-1594 c1cc(ccc1/C=N/NC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)F 2R-1595 c1cc(oc1)/C=N/NC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 2R-1596 c1ccc(c(c1)/C=N/NC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O 2R-1597 COc1cc(ccc1O)/C=N/NC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 2R-1598 c1ccc(cc1)C(=O)NNC(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 2R-1599 c1ccc(cc1)c2csc(n2)n3c(ccn3)c4ccc(cc4Cl)Cl 2T-0001 c1ccc(cc1)c2cc(n(n2)c3nc(cs3)c4ccccc4)C(F)(F)F 2T-0002 Cc1cc(n2c(n1)c(cn2)S(=O)(=O)c3ccccc3)C 2T-0003 COC(=O)c1cnc(c(c1N)C#N)O 2T-0004 CN(C)/C=C(/C#N)\c1nc(cs1)c2ccccc2 2T-0005 c1cc(ccc1c2cc(n3c(n2)cc(n3)c4ccc(c(c4)Cl)Cl)C(F)(F)Cl)C(F)(F)F 2T-0006 c1cc(c(cc1c2cc3nccc(n3n2)c4cnc5n(c4=O)CCS5)Cl)Cl 2T-0007 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccco5)C 2T-0008 c1ccc(cc1)c2c(sc(n2)n3c(c(cn3)S(=O)(=O)c4ccc(cc4)Cl)c5ccccc5)Sc6ccc(cc6)Cl 2T-0009 c1ccc(cc1)N2CCN(CC2)c3nc4nc(cc(n4n3)C(F)(F)Cl)c5ccc(cc5)C(F)(F)F 2T-0010 Cc1c(c(ccc1OCC(=O)c2ccc(cc2)Cl)Br)C 2T-0011 CCOC(=O)C1=C(NC(=S)C(C1c2ccccc2)C#N)c3ccccc3 2T-0014 c1cc(sc1)c2ccnn2c3nc(c(s3)Sc4ccc(cc4)Cl)c5ccc(cc5Cl)Cl 2T-0015 c1ccc(cc1)c2c(cnn2c3nc(c(s3)Sc4ccc(cc4)Cl)c5ccc(cc5Cl)Cl)S(=O)(=O)c6ccc(cc6)Cl 2T-0017 c1ccc(cc1)c2c(sc(n2)n3c(ccn3)c4cccs4)Sc5ccc(cc5)Cl 2T-0020 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)c5ccccc5)S(=O)(=O)c6ccc(cc6)Cl)C 2T-0024 Cc1c(c(n2c(n1)c(cn2)c3ccc(cc3)F)N)c4ccccc4 2T-0027 c1cc(cc(c1)Cl)c2cc(n3c(n2)c(cn3)c4ccc(cc4)F)C(F)(F)F 2T-0029 c1cc(cc(c1)n2c(ccn2)c3cnc4n(c3=O)CCS4)C(F)(F)F 2T-0030 c1ccc(cc1)c2csc(n2)n3c(c(cn3)c4ccc(cc4)Cl)N 2T-0033 CCOC(=O)/C(=N\O)/C(=O)C(F)(F)F.O 2T-0036 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3cccc(c3)F 2T-0037 c1cc(ccc1c2cnn(c2N)c3nc(cs3)c4ccc(c(c4)Cl)Cl)Cl 2T-0046 c1ccc(c(c1)c2csc(n2)n3c(c(cn3)c4ccc(cc4)Cl)N)F 2T-0047 c1cc(cc(c1)F)c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F 2T-0048 c1cc(cc(c1)F)c2csc(n2)n3c(c(cn3)c4ccc(cc4)F)N 2T-0049 CCOC(=O)/C(=N/OC)/C(=O)C(F)(F)F 2T-0050 c1cc(ccc1Sc2c(nc(s2)NN/C=C(/C#N)\C(=O)C(F)(F)F)c3ccc(cc3Cl)Cl)Cl 2T-0054 c1cc(c(c(c1)Cl)CN2CCC(=O)CC2)Cl 2T-0055 CCOC(=O)CC1CCN(CC1)c2ccc(cc2)N 2T-0058 CC1(CC(=O)c2ccc(cc2O1)O)C 2T-0063 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)C(F)(F)F 2T-0068 Cc1ccc(cc1)S(=O)(=O)NC(C)C(=O)O 2T-0200 Cc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=O)N2C 2T-0201 CCCCCCC(N1CCOC1=O)S(=O)(=O)c2ccccc2 2T-0203 Cc1ccc(cc1)S(=O)(=O)C(C2CCCCC2)NC(=O)OCc3ccccc3 2T-0204 Cc1ccc(cc1)S(=O)(=O)C(C2CCCCC2)N3C(C(N(C3=O)C)C)c4ccccc4 2T-0205 Cc1nnc(n1Cc2ccccc2)c3cnn(c3N)c4ccccc4 2T-0209 c1ccc(c(c1)C(=O)c2ccc3c(c2)NC(=O)CO3)C(=O)O 2T-0210 COC(=O)c1cccc(c1)Oc2ccc(cc2[N+](=O)[O-])C=O 2T-0212 c1ccc2c(c1)c(n[nH]c2=O)c3ccc4c(c3)NC(=O)CO4 2T-0213 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4ccc5c(c4)NC(=O)CO5 2T-0215 Cc1nnc(n1CCc2ccccc2)c3cnn(c3N)c4ccccc4 2T-0216 Cc1nnc(n1CCNc2ccc(cc2Cl)C(F)(F)F)c3cnn(c3N)c4ccccc4 2T-0217 CCN1C(C2=C(c3ccccc3C2=O)NC1=O)c4ccccc4F 2T-0220 Cc1nnc(n1Cc2ccc(cc2)F)c3cnn(c3N)c4ccccc4 2T-0221 Cc1nnc(n1CCCN(C)C)c2cnn(c2N)c3ccccc3 2T-0222 Cc1nnc(n1Cc2ccncc2)c3cnn(c3N)c4ccccc4 2T-0224 c1cc2c(cc1C(=O)/C=C/C(=O)O)NC(=O)CO2 2T-0225 Cc1nnc(n1CC2CCCO2)c3cnn(c3N)c4ccccc4 2T-0229 COC(=O)c1c(c2c3c(c(nc2s1)c4ccccc4)CCC3)N 2T-0233 CCCCCCC(N1CCOC1=O)S(=O)(=O)c2ccc(cc2)C 2T-0234 Cc1nnc(n1Cc2cccc(c2)C(F)(F)F)c3cnn(c3N)c4ccccc4 2T-0235 CC(c1ccccc1)(c2ccccc2)c3cccnc3 2T-0237 COC(=O)c1ccc(c(c1)N)n2cncn2 2T-0238 COC(=O)c1c(c2c3c(c(nc2s1)c4ccc(cc4)Cl)CCCC3)N 2T-0239 Cc1nnc(n1CCCOC)c2cnn(c2N)c3ccccc3 2T-0240 Cc1ccc(cc1)c2c3c(c(c(n2)SCC(=O)OC)C#N)CCCC3 2T-0243 COC(=O)CSc1c(c2c(c(n1)c3ccc(cc3)Br)CCC2)C#N 2T-0244 c1ccc(cc1)c2c3c(c4c(c(sc4n2)C#N)N)CCC3 2T-0245 c1ccc(cc1)CNC(=O)c2ccccc2C(=O)c3ccc4c(c3)NC(=O)CO4 2T-0246 c1ccc(cc1)c2c3c(c4c5c(c(ncn5)N)sc4n2)CCC3 2T-0247 c1cc(c(cc1CN2CCC(CC2)C(=O)O)Cl)Cl.Cl 2T-0248 c1cc(cc(c1)F)CN2CCC(CC2)C(=O)O.Cl 2T-0249 c1cc(ccc1F)S(=O)(=O)O/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 2T-0250 c1cc(ccc1S(=O)(=O)O/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl 2T-0251 CC(C)(C)c1ccc(cc1)S(=O)(=O)O/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 2T-0252 CC(c1ccccc1)(c2ccccc2)c3ccncc3 2T-0253 COc1cc(cc(c1OC)OC)C(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 2T-0256 Cc1ccccc1CSc2c(c3c(c(n2)c4ccccc4)CCC3)C#N 2T-0258 CCOC(=O)c1c(nc(s1)c2cccnc2)C 2T-0259 Cc1ccc(cc1)c2c3c(c(c(n2)SCC#N)C#N)CCCC3 2T-0260 c1ccc(cc1)c2c3c(c(c(n2)SCc4c(cccc4Cl)F)C#N)CCC3 2T-0261 Cn1c(c(cn1)C(=O)NN)N 2T-0263 COC(=O)CC1COc2ccccc2N1C(=O)c3cccc(c3)Cl 2T-0264 COC(=O)CC1COc2ccccc2N1C(=O)c3ccc(cc3)Cl 2T-0265 c1ccc(c(c1)C2C3=C(c4ccccc4C3=O)NC(=N2)SCc5ccc(cc5)F)F 2T-0267 c1cc(ncc1[N+](=O)[O-])N2CCCC2 2T-0268 CC(C)(C)c1ccc(cc1)CSc2c(c3c(c(n2)c4ccccc4)CCC3)C#N 2T-0269 c1ccc(cc1)c2c3c(c(c(n2)SCc4cccc(c4)Cl)C#N)CCC3 2T-0271 c1ccc(c(c1)C(=O)N2c3ccccc3OCC2CC(=O)O)Cl 2T-0272 COC(=O)CC1COc2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F 2T-0275 CC(C)(C)c1ccc(cc1)C(=O)N2c3ccccc3OCC2CC(=O)OC 2T-0276 COc1cc(cc(c1OC)OC)C(=O)N2c3ccccc3OCC2CC(=O)OC 2T-0277 COC(=O)CC1COc2ccccc2N1C(=O)/C=C/c3ccccc3 2T-0279 COC(=O)CC1COc2ccccc2N1C(=O)c3ccc(cc3)Br 2T-0280 c1cc2c(cc1N)NC(=O)CO2 2T-0281 c1ccc(cc1)c2c3c(c(c(n2)SC4CCCC4)C#N)CCC3 2T-0282 CCO/C(=N/NC(=O)c1cnn(c1N)C)/C 2T-0283 CC(C)(C)OC(=O)N1CCC(CC1)(c2ccccc2)C(=O)O 2T-0284 Cc1ccc(cc1)c2c3c(c(c(n2)SCc4ccc(c(c4)Cl)Cl)C#N)CCCC3 2T-0285 Cc1ccc(cc1)c2c3c(c4c(c(sc4n2)C#N)N)CCCC3 2T-0287 Cc1ccc(cc1)c2c3c(c(c(n2)SCc4cccc(c4)C)C#N)CCCC3 2T-0288 CC1CC(CC(C1)(CC(=O)Nc2cccc(c2)C(F)(F)F)C(=O)O)(C)C 2T-0289 Cc1nnc(n1CCCn2ccnc2)c3cnn(c3N)C 2T-0290 Cc1nnc(n1CCCN(C)C)c2cnn(c2N)C 2T-0293 Cc1nnc(n1Cc2ccc(cc2)OC)c3cnn(c3N)C 2T-0295 Cc1nnc(n1CCc2ccccc2)c3cnn(c3N)C 2T-0296 Cc1ccc(cc1)c2c3c(c4c5c(c(ncn5)N)sc4n2)CCCC3 2T-0297 c1cc2c(cc1[N+](=O)[O-])NC(=O)CO2 2T-0299 c1ccc(cc1)c2c3c(c(c(n2)Sc4c(cc(cn4)C(F)(F)F)Cl)C#N)CCC3 2T-0300 Cc1nnc(n1CCCOC)c2cnn(c2N)C 2T-0302 CC(C)(C)c1ccc(cc1)c2c3c(c(c(n2)SCC(=O)OC)C#N)CCC3 2T-0303 CC(C)(C)c1ccc(cc1)c2c3c(c(c(n2)SCc4ccc(cc4)F)C#N)CCC3 2T-0304 CCCCCCCn1c(nnc1c2cnn(c2N)C)C 2T-0305 Cc1nnc(n1Cc2cccc(c2)C(F)(F)F)c3cnn(c3N)C 2T-0307 Cc1nnc(n1Cc2cccc(c2)Cl)c3cnn(c3N)C 2T-0308 Cc1cc(n2cc(nc2n1)c3ccccc3)N4CCN(CC4)c5ccccc5 2T-0309 CC(C)(C)c1ccc(cc1)c2c3c(c(c(n2)SCc4ccccc4)C#N)CCC3 2T-0311 c1ccc(cc1)CSc2c(c3c(c(n2)c4ccc(cc4)Br)CCC3)C#N 2T-0312 c1ccc(c(c1)C(=O)Nc2cccn3c2ncc3c4ccc(cc4)Cl)F 2T-0313 c1cc(c2ncc(n2c1)c3ccc(cc3)Cl)NC(=O)c4ccc(cc4Cl)Cl 2T-0315 Cc1nnc(n1Cc2ccncc2)c3cnn(c3N)C 2T-0320 c1cc(cc(c1)C(F)(F)F)CSc2c(c3c(c(n2)c4ccc(cc4)Br)CCC3)C#N 2T-0322 Cc1ccccc1c2c3c(c(c(=S)[nH]2)C#N)CCC3 2T-0323 Cc1cc(n2cc(nc2n1)c3ccccc3)N(C)N 2T-0324 Cc1cc(n2cc(nc2n1)c3ccccc3)NNc4ccccc4 2T-0325 Cc1cc(n2cc(nc2n1)c3ccccc3)N4CCOCC4 2T-0328 Cc1cc(n2cc(nc2n1)c3ccccc3)N4CCN(CC4)c5ccccn5 2T-0330 Cc1cc(n2cc(nc2n1)c3ccccc3)N4CC(OC(C4)C)C 2T-0331 Cc1cc(n2cc(nc2n1)c3ccccc3)N4CCN(CC4)c5ccccc5Cl 2T-0332 CCCCCCC(NC(=O)OCc1ccccc1)S(=O)(=O)c2ccc(cc2)C 2T-0333 Cc1ccccc1c2c3c(c(c(n2)SCC#N)C#N)CCC3 2T-0334 c1cc(c(c(c1)Cl)CSc2c(c3c(c(n2)c4ccc(cc4)Cl)CCCC3)C#N)Cl 2T-0339 Cc1ccccc1C(=O)Oc2ccc(cc2)CC(=O)Nc3cc(cc(c3)C)C 2T-0341 Cc1ccc(cc1)S(=O)(=O)C(C)NC(=O)OCc2ccccc2 2T-0342 Cc1ccccc1c2c3c(c(c(n2)SCc4ccccc4)C#N)CCC3 2T-0345 Cc1cc(cc(c1)NC(=O)Cc2ccc(cc2)OC(=O)c3c(onc3c4ccccc4Cl)C)C 2T-0346 Cc1cc(cc(c1)NC(=O)Cc2ccc(cc2)OC(=O)C3CCCCC3)C 2T-0347 c1ccc(cc1)CSc2c(c3c(c(n2)c4ccccc4F)CCCC3)C#N 2T-0349 COC(=O)c1ccccc1Sc2c(n3ccsc3n2)/C=C/c4ccn[nH]4 2T-0350 COc1ccc(cc1)C(=O)Oc2ccc(cc2)CC(=O)Nc3ccc4c(c3)CCC4 2T-0351 c1ccc(cc1)CSc2c(c3c(c(n2)c4ccc(cc4)Cl)CCCC3)C#N 2T-0353 c1cc(cc(c1)F)CSc2c(c3c(c(n2)c4ccc(cc4)Cl)CCCC3)C#N 2T-0354 Cc1ccccc1c2c3c(c(c(n2)SCc4cccc(c4)F)C#N)CCC3 2T-0356 CC1=NN(C(=O)C1C(=O)C)C(=O)C 2T-0357 c1ccc2c(c1)c(nn(c2=O)c3cc(cc(c3)Cl)Cl)c4ccc5c(c4)NC(=O)CO5 2T-0358 Cn1c(=O)c2ccccc2c(n1)c3ccc4c(c3)NC(=O)CO4 2T-0359 Cc1ccccc1c2c3c(c(c(n2)SCc4ccc(cc4Cl)Cl)C#N)CCC3 2T-0362 CC(C)(C)c1ccc(cc1)c2c3c(c(c(n2)SCC(=O)N)C#N)CCC3 2T-0364 Cc1cccc(c1)n2c(=O)c3ccccc3c(n2)c4ccc5c(c4)NC(=O)CO5 2T-0365 COC(=O)c1ccccc1C(=O)c2ccc3c(c2)NC(=O)CO3 2T-0366 c1ccc(c(c1)C(=O)c2ccc3c(c2)NC(=O)CO3)C(=O)NCc4cccc(c4)C(F)(F)F 2T-0367 COc1ccc(cc1)CNC(=O)c2ccccc2C(=O)c3ccc4c(c3)NC(=O)CO4 2T-0368 CN1CCN(CC1)C(=O)CC(c2cccs2)NC(=O)C(F)(F)F 2T-0601 c1cc(c(cc1C(CC(=O)O)N)O)O 2T-0602 CN(C)/C=C\1/C(c2cc3c(cc2C1=O)OCO3)NC(=O)C(F)(F)F 2T-0605 COC(=O)c1ccc(cc1)NC(=O)CC(c2cccs2)NC(=O)C(F)(F)F 2T-0606 c1cc2c(cc1C=O)OCCO2 2T-0607 Cc1cc(nc(n1)N)c2ccc(s2)Cl 2T-0609 Cc1cc(nc(n1)N)c2c(ccs2)Cl 2T-0610 c1cc(c(cc1C(CC(=O)O)N2CCS(=O)(=O)CC2)Cl)Cl 2T-0611 COc1cc2c(cc1OC)C(=O)C(C2NC(=O)C(F)(F)F)Br 2T-0613 Cc1ccsc1C(=O)/C=C/N(C)C 2T-0614 Cc1cc(nc(n1)N)c2ccc(s2)Br 2T-0615 Cc1ccsc1c2ccnc(n2)N 2T-0617 c1cc(ccc1C(=O)NC2CC(=O)c3c2cc4c(c3)OCO4)F 2T-0620 c1cc(sc1)C(CC(=O)N)NC(=O)C(F)(F)F 2T-0623 c1cc(sc1)C(=O)NC2CC(=O)c3c2cc4c(c3)OCO4 2T-0626 c1c2c(cc3c1OCO3)C(=O)CC2NC(=O)C4CC4 2T-0627 c1cc(oc1)C(=O)NC2CC(=O)c3c2cc4c(c3)OCO4 2T-0628 c1c2c(cc3c1OCO3)/C(=N\O)/CC2NC(=O)C(F)(F)F 2T-0631 COc1ccc2c(c1)C(CC2=O)NC(=O)C(F)(F)F 2T-0633 c1cc(sc1)S(=O)(=O)NC2CC(=O)c3c2cc4c(c3)OCO4 2T-0636 c1cc2c(cc1C(CC(=O)O)N)OCCO2 2T-0637 Cc1ccsc1C(=O)/C=C(\C)/N(C)C 2T-0638 c1cc(sc1)c2cc(nc(n2)N)C(F)(F)F 2T-0639 COc1cccc2c1C(=O)CC2NC(=O)C(F)(F)F 2T-0642 COC(=O)c1ccc(cc1)/C=C/C(=O)O 2T-0643 COc1ccc2c(c1)C(CC2=O)[NH3+].[Cl-] 2T-0644 COc1cc2c(cc1OC)/C(=N/O)/CC2NC(=O)C(F)(F)F 2T-0646 C(/C(=N/NC(=S)N)/C(F)(F)F)C(=O)C(F)(F)F 2T-0800 Cc1cc(n(n1)c2nc(cs2)c3cccc(c3)[N+](=O)[O-])C(F)(F)F 2T-0801 c1c(c(n2c(n1)ncn2)O)n3cncn3 2T-0802 COC(=O)/C(=C\Nc1ccc(cc1)OCc2ccccc2)/n3cncn3 2T-0803 Cc1c(c(n2c(n1)nc(n2)N)C)Cc3ncc(s3)Cl 2T-0804 Cc1cc(n(n1)c2nc(cs2)CCl)C(F)(F)F 2T-0805 Cc1cc2nccc(n2n1)c3ccc(cc3)c4ccccc4 2T-0806 Cc1c(c2nccc(n2n1)c3ccc(cc3)c4ccccc4)Br 2T-0807 c1cc(ccc1SC(C(=O)c2ccc(cc2Cl)Cl)Br)Cl 2T-0808 C1CCc2c(c(c(s2)N)C#N)C1 2T-0811 c1ccc(cc1)c2c3c(=N)n(c(=S)[nH]c3oc2c4ccccc4)c5ccc(cc5)O 2T-0812 c1cc(oc1)c2c3c(=N)n(c(=S)[nH]c3oc2c4ccco4)c5ccc(cc5)Cl 2T-0813 c1cc(ccc1c2cnc3[n+](c2)[C@@H](CS3)CBr)Cl.[Br-] 2T-0816 Cc1cc(n(n1)c2nc(c(s2)CC(=O)OC)c3ccccc3)C(F)(F)F 2T-0817 c1ccc(cc1)c2csc(n2)N/N=C(/CC(=O)C(F)(F)F)\C(F)(F)F 2T-0818 CCOC(=O)c1c(nc(s1)N/N=C(/C)\CC(=O)C(F)(F)F)C(F)(F)F 2T-0819 Cc1cc2nc(cc(n2n1)O)CC(=O)OC 2T-0820 c1c(cnc(c1Cl)CC(=O)NCCCCCCCN)C(F)(F)F 2T-0822 Cc1cc2ncc(c(n2n1)O)n3cncn3 2T-0823 COC(=O)Cc1cc(n2c(n1)ncn2)O 2T-0824 Cc1c(c2nccc(n2n1)c3ccc(cc3)c4ccccc4)Cl 2T-0825 Cc1cc(n(n1)c2nc(c(s2)Sc3ccc(cc3)Cl)c4ccc(cc4)OC)C(F)(F)F 2T-0826 COc1cc2c(cc1OC)C3Cc4c(cncn4)C(=O)N3CC2 2T-0827 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3cccc(c3)OC 2T-0829 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)OC)Cl 2T-0830 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)OC 2T-0831 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)F 2T-0832 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3cccc(c3)OC)Cl 2T-0833 Cc1cc(n(n1)c2nc(c(s2)Sc3ccc(cc3)Cl)c4ccc(cc4)OC)C 2T-0834 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)F)Cl 2T-0835 Cc1cc(n(n1)c2nc(c(s2)CC(=O)O)c3ccccc3)C(F)(F)F 2T-0836 c1cc(ccc1C(=O)CC(=O)C(F)(F)F)F 2T-0837 COc1cccc(c1)C(=O)CC(=O)C(F)(F)F 2T-0838 COc1ccc(cc1)C(=O)CC(=O)C(F)(F)F 2T-0839 COc1cc2c(cc1OC)C3Cc4c(cnc5n4ncn5)C(=O)N3CC2 2T-0840 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5ccc(cc5)F)C 2T-0841 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5ccc(cc5)OC)C 2T-0842 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5cccc(c5)OC)C 2T-0843 Cc1cc(n(n1)c2nc(c(s2)CC(=O)NN)c3ccccc3)C(F)(F)F 2T-0844 COc1cc2c(cc1OC)C3Cc4c(cnc(n4)N)C(=O)N3CC2 2T-0846 Cc1cc2ncc3c(n2n1)CC4c5cc(c(cc5CCN4C3=O)OC)OC 2T-0847 Cc1cc2nc(cc(n2n1)C(F)(F)Cl)c3ccc(cc3)C(F)(F)F 2T-0848 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])n2c(c(cn2)n3cncn3)O 2T-0849 Cc1c(c2nc(cc(n2n1)C(F)(F)Cl)c3ccc(cc3)C(F)(F)F)Cl 2T-0850 Cc1c(c2nc(cc(n2n1)C(F)(F)Cl)c3ccc(cc3)C(F)(F)F)Br 2T-0851 CN(C)/C=C/C(=O)c1c(cc(cn1)C(F)(F)F)Cl 2T-0854 COc1ccccc1C(=O)CC(=O)C(F)(F)F 2T-0855 Cc1cc(n(n1)c2nc(c(s2)C(=O)O)C)C(F)(F)F 2T-0856 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccccc3OC 2T-0862 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5ccccc5OC)C 2T-0864 c1cc(ccc1c2cc(c(c(n2)O)C#N)C(F)(F)F)F 2T-0865 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)Cl)c5ccc(cc5)C(F)(F)F)C 2T-0866 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccccc3OC)Cl 2T-0870 COc1cccc(c1)c2cc(c(c(n2)O)C#N)C(F)(F)F 2T-0871 Cc1cc2nccc(n2n1)c3ccncc3 2T-0872 COc1ccc(cc1)c2cc(c(c(n2)O)C#N)C(F)(F)F 2T-0873 COC(=O)Cc1c(nc(s1)c2ccc(cc2)C(=O)OC)c3ccccc3 2T-0874 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccncc5)C 2T-0876 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccccc3F 2T-0877 CC(=O)c1cnc(s1)Nc2cccc(c2)C(F)(F)F 2T-0885 c1ccc(c(c1)c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F)F 2T-0886 COc1ccccc1c2cc(c(c(n2)O)C#N)C(F)(F)F 2T-0889 c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)C(=O)O)CC(=O)O 2T-0890 c1cc(ccc1c2cc(c(c(n2)O)C#N)C(F)(F)Cl)C(F)(F)F 2T-0891 CCOC(=O)c1csc(n1)n2c(cc(n2)C)C(F)(F)F 2T-0892 COC(=O)Cc1c(nc(s1)c2ccccn2)c3ccccc3 2T-0893 Cc1c(c2nccc(n2n1)c3ccncc3)Cl 2T-0894 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)c4ccccc4 2T-0895 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5cccs5)C 2T-0896 CN1CCN(CC1)C(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 2T-0899 c1csc(c1C(=O)N)N 2T-0905 c1cc(ccc1C(=S)N)F 2T-0908 Cc1cc2nccc(n2n1)c3cccs3 2T-0910 Cc1cc([nH]n1)N/C=C/C(=O)c2cccs2 2T-0911 c1cc(ccc1c2cc(n3c(n2)c(cn3)c4ccc(cc4)Cl)C(F)(F)Cl)C(F)(F)F 2T-0912 c1cc(ccc1c2cnn3c2nccc3c4ccncc4)F 2T-0913 c1cc(sc1)c2ccnc3n2ncc3c4ccc(cc4)F 2T-0914 c1c(cnc(c1Cl)/C=C/c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 2T-0915 c1cc(ccc1c2cnn3c2nccc3c4ccncc4)Cl 2T-0916 c1ccc(cc1)c2ccc(cc2)c3csc(n3)n4c(c(cn4)C(=O)O)C(F)(F)F 2T-0919 Cc1cc2nccc(n2n1)c3ccc(o3)c4ccc(cc4Cl)Cl 2T-0920 COc1ccc(cc1)c2csc(n2)n3c(c(cn3)c4ccc(cc4)F)N 2T-0922 c1ccc(cc1)c2csc(n2)n3c(c(cn3)c4ccc(cc4)F)N 2T-0923 c1cc(ccc1c2cnn(c2N)c3nc(cs3)c4ccc(cc4)F)F 2T-0924 Cc1c(c2nccc(n2n1)c3ccc(o3)c4ccc(cc4Cl)Cl)Cl 2T-0925 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc(o5)c6ccc(cc6Cl)Cl)C 2T-0926 c1ccc(cc1)C#Cc2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl 2T-1120 c1ccc(cc1)C#Cc2ccc(cc2)NS(=O)(=O)c3ccccc3 2T-1121 c1ccc(cc1)C#Cc2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Br 2T-1122 c1ccc(cc1)C#Cc2ccc(cc2)NS(=O)(=O)c3ccc(cc3)F 2T-1123 c1ccc(cc1)CS(=O)(=O)Nc2ccc(cc2)C#Cc3ccccc3 2T-1124 Cc1ccc(n1c2c(cnn2c3ccccc3)C(=O)NN)C 2T-1125 CCCCC#Cc1ccc(cc1)NC(=O)c2ccc(cc2)C 2T-1128 CCCC(=O)Nc1ccc(cc1)C#Cc2ccccc2 2T-1131 c1ccc(cc1)C#Cc2ccc(cc2)NC(=O)C(Cl)(Cl)Cl 2T-1132 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Cl)C=O 2T-1133 CCCCC#Cc1cccc(c1)NC(=O)c2cccs2 2T-1135 CCCCC#Cc1cccc(c1)NC(=O)c2cccc(c2)Cl 2T-1136 CCCCC#Cc1cccc(c1)NC(=O)c2ccc(c(c2)Cl)Cl 2T-1137 CCCCC#Cc1ccc(cc1)NC(=O)c2ccc(cc2)F 2T-1138 CCCCC#Cc1cccc(c1)NC(=O)C2CC2 2T-1139 CCCCC#Cc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)C 2T-1140 CCCCC#Cc1ccc(cc1)NS(=O)(=O)Cc2ccccc2 2T-1141 CCCCC#Cc1ccc(cc1)NS(=O)(=O)C 2T-1142 Cc1ccc(cc1)Sc2c(c(nn2c3ccccc3)c4ccccc4)C=O 2T-1143 CCCCC#Cc1cccc(c1)NS(=O)(=O)c2ccc(cc2)Cl 2T-1144 c1ccn(c1)c2ccc(cc2)C(=O)N3CCOCC3 2T-1145 c1ccn(c1)c2ccc(cc2)C(=O)N3CCCCC3 2T-1146 c1ccc(cc1)N2CCN(CC2)C(=O)c3ccc(cc3)n4cccc4 2T-1147 c1ccc(cc1)C\2=NN(C(=O)/C2=C\c3ccc(cc3)Cl)c4ccccc4 2T-1149 c1ccc(cc1)C\2=NN(C(=O)/C2=C\c3ccc(cc3)F)c4ccccc4 2T-1150 Cc1ccc(cc1)/C=C\2/C(=NN(C2=O)c3ccccc3)c4ccccc4 2T-1151 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Sc4ccc(cc4)F)C=O 2T-1152 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Sc4ccc(cc4)Cl)C=O 2T-1153 c1ccn(c1)c2ccc(cc2)C(=O)NC3CC3 2T-1154 CN1CCN(CC1)C(=O)c2ccc(cc2)n3cccc3 2T-1157 c1ccc(cc1)CN2CCN(CC2)C(=O)c3ccc(cc3)n4cccc4 2T-1158 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Sc4c(cccc4Cl)Cl)C=O 2T-1160 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Sc4ccc(cc4)Br)C=O 2T-1161 Cc1ccc(c(c1)C)Sc2c(c(nn2c3ccccc3)c4ccccc4)C=O 2T-1162 CSc1[nH]cnn1 2T-1506 CC(=O)c1ccc(c(c1)n2cccc2)C#N 2T-1515 COC(=O)C(Cc1cnc(s1)Cl)(c2ccc(cc2[N+](=O)[O-])C(F)(F)F)C(=O)OC 2W-0002 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(nc2)C(C(=O)OC)C(=O)OC 2W-0005 CC(c1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])(C(=O)OC)C(=O)OC 2W-0010 COC(=O)C(CC=C)(c1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])C(=O)OC 2W-0014 Cc1ccc(cc1)C(CCc2cc(c(c(c2)OC)OC)OC)OC(=O)c3ccc(cc3)Cl 2W-0016 C1CCC2(CC1)NCCO2 2W-0018 COc1ccccc1C/C=C/c2cccs2 2W-0019 Cc1ccc(cc1[N+](=O)[O-])C(F)(F)F 2W-0021 c1cc(ccc1S(=O)(=O)N2CCOC23CCCCC3)I 2W-0022 c1cc(ccc1C(=O)N2CCOC23CCCCC3)I 2W-0023 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCOC34CCCCC4 2W-0024 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCOC23CCCCC3 2W-0025 c1cc(ccc1NC(=O)N2CCOC23CCCCC3)Cl 2W-0027 c1cc(ccc1NC(=O)N2CCOC23CCC4(CC3)OCCO4)Cl 2W-0029 CCc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] 2W-0035 COc1ccc(cc1)c2csc(n2)c3nc(cs3)c4ccc(cc4)OC 2W-0037 c1ccc(c(c1)CCc2cnc(s2)Cl)[N+](=O)[O-] 2W-0039 COC(=O)C(Cc1cnc(s1)Cl)(c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])C(=O)OC 2W-0047 C1CCC2(CC1)C3CCCCC3=NC(=C(N2)C#N)C#N 2W-0200 CN1/C(=C\c2ccccc2OC)/C(=O)N=C1N 2W-0201 CC1=NC(=C(NC(C1)c2c(cccc2Cl)F)C#N)C#N 2W-0204 CC1=NC(=C(NC(C1)c2ccc(cc2)Cl)C#N)C#N 2W-0205 Cc1c2c(c3cccc(c3n1)OC)SCC2 2W-0209 c1ccc(cc1)S(=O)(=O)c2cscc2NC(=O)c3ccco3 2W-0210 c1ccc(c(c1)/C=C\2/C(=O)N=C(S2)NC(=N)N)n3cncn3 2W-0215 c1ccc(c(c1)/C=C\2/C(=O)NC(=S)S2)n3cccn3 2W-0216 CC(=O)c1c2c(c(c(c1Cl)Cl)[N+](=O)[O-])OCCO2 2W-0219 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3cccnc3 2W-0220 Cc1c(c(n(n1)C)Cl)NC(=O)OCc2ccccc2 2W-0221 Cc1c(c(n(n1)C)Cl)NC(=O)OCc2ccc(cc2)F 2W-0222 Cc1ccc(n1/C(=C(\C#N)/NC(=O)c2cccs2)/C#N)C 2W-0226 CSC1=NC(=O)/C(=C/c2ccccc2n3cccn3)/S1 2W-0228 c1cc2c(cc1/C=C/3\C(=O)NC(=S)S3)OCO2 2W-0230 Cc1c(c(n(n1)C)Cl)NC(=O)OCc2cccnc2 2W-0234 Cc1c(c(c2cc(ccc2n1)Oc3ccccc3)Cl)CCCl 2W-0237 Cc1ccc(cc1)NC(=O)c2ccc(cc2)Oc3ncccn3 2W-0238 Cc1ccc(n1/C(=C(\C#N)/NC(=O)c2cccc(c2)C(F)(F)F)/C#N)C 2W-0240 c1ccc(c(c1)/C=C\2/C(=O)N=C(S2)NC(=N)N)n3cccn3 2W-0242 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)C=O 2W-0244 Cc1c(c(=O)n([nH]1)C)CCO 2W-0245 CSC1=NC(=O)/C(=C\c2ccc3c(c2)OCO3)/S1 2W-0246 Cc1c(c(=O)[nH][nH]1)CCO 2W-0248 Cc1ccc(n1/C(=C(\C#N)/NC(=O)c2c(onc2c3ccccc3Cl)C)/C#N)C 2W-0252 CC1=NC(=C(NC(C1)(C)C)C#N)C#N 2W-0256 Cc1c(c(c2cc(ccc2n1)Oc3ccccc3)Nc4ccc(cc4)O)CCCl 2W-0257 CN(C)/C=C/C(=O)c1ccc(cc1)C2CCCCC2 2W-0259 Cc1c2c(c3cc(ccc3n1)Oc4ccccc4)SCC2 2W-0262 CCOC(=O)C1=C(C(=O)N(C1)Cc2cccs2)O 2W-0263 Cc1c([nH]c(c1C#N)N)C 2W-0265 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)/C=C(\C#N)/c5cccs5 2W-0267 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)/C=C(\C#N)/c5ccc(cc5)Cl 2W-0268 Cc1ccc(cc1)S(=O)(=O)/C(=C\c2cn(nc2c3ccc4ccccc4c3)c5ccccc5)/C#N 2W-0269 c1cc(cc(c1)Oc2ncccn2)/C=C(\C#N)/c3ccc4c(c3)OCO4 2W-0271 Cc1cc2nc(ccn2n1)c3ccc(cc3)C4CCCCC4 2W-0273 Cc1c(c2ncc(c(n2n1)N)C(=O)O)c3cccc(c3)C(F)(F)F 2W-0276 Cc1c(c(=O)n([nH]1)C(C)(C)C)CCO 2W-0277 c1cc(ccc1CN)N2CCC(CC2)CO 2W-0279 Cc1c(c(=O)n([nH]1)c2ccccc2)CCO 2W-0281 c1cc(cc(c1)Oc2ncccn2)/C=C(\C#N)/c3cccs3 2W-0282 Cc1cccc(c1N2CCN(CC2)C3=NC(=O)/C(=C\c4ccc5c(c4)OCO5)/S3)C 2W-0283 c1cc(cc(c1)Oc2ncccn2)/C=C(/C#N)\c3ccc(cc3)O 2W-0284 CC1=NC(=C(N=C(C1)C)C#N)C#N 2W-0285 Cc1cn2c(nc1c3ccc(c(c3)F)OC)nc(n2)SC 2W-0286 COc1ccc(cc1OC)/C(=C/c2cccc(c2)Oc3ncccn3)/C#N 2W-0288 Cc1ccc(n1/C(=C(\C#N)/NC(=O)C(C)(C)CCl)/C#N)C 2W-0289 c1cc(c(cc1N2CCOCC2)C(=O)N)[N+](=O)[O-] 2W-0291 Cc1c(sc(n1)c2ccc(cc2)Cl)CO 2W-0294 COC(=O)COc1ccccc1C#N 2W-0299 c1ccc(c(c1)/C(=C\c2cccc(c2)Oc3ncccn3)/C#N)F 2W-0300 Cc1cn2c(c(cn2)C#N)nc1c3ccc(c(c3)F)OC 2W-0301 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5ccccc5[N+](=O)[O-])CCS4 2W-0303 COC(=O)c1ccc(cc1)c2ccc(cc2)Br 2W-0305 COC(=O)c1c(c2ccccc2o1)N 2W-0306 Cc1cc2nc(c(cn2n1)C)c3ccc(c(c3)F)OC 2W-0308 Cc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)N3CCC(CC3)CO 2W-0309 c1cc(cc(c1)Oc2ncccn2)/C=C(\C#N)/C(=O)c3ccc(cc3)Cl 2W-0310 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2cccc(c2)Oc3ncccn3)/C#N 2W-0311 CCOC(=O)c1c([nH]c(=O)nc1c2ccccc2)C 2W-0312 CCN1C(=C(N=C(CC1(C)C)C)C#N)C#N 2W-0315 Cc1c(sc(n1)c2ccc(cc2)Cl)CCl 2W-0316 Cc1c2c(c3cc(ccc3n1)Oc4ccccc4)N(CC2)c5ccc(cc5)C(C)C 2W-0321 c1ccc(cc1)OC(=O)NO 2W-0324 c1cc(ccc1c2ccn3c(n2)c(cn3)C#N)C4CCCCC4 2W-0327 CSc1nc2nc(ccn2n1)c3ccc(cc3)C4CCCCC4 2W-0329 c1ccc(c(c1)/C=C\2/C(=O)N=C(S2)NO)n3cccn3 2W-0330 c1cc2c(nc1)NC(=O)C(O2)CCO 2W-0332 Cc1c2c(c3cccc(c3n1)C(F)(F)F)SCC2 2W-0336 C[C@H](c1ccccc1)N2CC(CC2=O)C(=O)O 2W-0339 Cc1c(c(=O)n([nH]1)c2ccc(c(c2)Cl)Cl)CCO 2W-0340 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)C#N 2W-0343 Cc1c(c(=O)n([nH]1)c2ccc(cc2)C(=O)O)CCO 2W-0346 COC(=O)CO/C=C(/C#N)\c1ccc(cc1Cl)Cl 2W-0348 CSc1nc2nc(ccn2n1)c3c4c(cc(c3Cl)Cl)OCCO4 2W-0349 CCOC(=O)C1=C(NC(=O)N(C1c2ccc(cc2)[N+](=O)[O-])C=O)C 2W-0350 c1cc(ccc1c2c3c(nn2c4ccc(cc4)C(=O)O)CCCC3)Cl 2W-0353 C(=O)(NN)NO 2W-0354 Cc1c(c2ncc(c(n2n1)N)C#N)c3cccc(c3)C(F)(F)F 2W-0357 Cc1c(c(=O)n([nH]1)c2ccc(cc2)F)CCO 2W-0359 Cc1ccc(cc1)C2CN(C3(C24COc5ccccc5C4=O)c6ccccc6NC3=O)C 2W-0600 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)Cl)/CO2 2W-0607 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccc(cc6Cl)Cl 2W-0608 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccccc6Cl 2W-0609 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccc(c(c6)[N+](=O)[O-])Cl 2W-0610 c1ccc2c(c1)C(=O)/C(=C/c3cccc(c3)F)/CO2 2W-0612 c1ccc2c(c1)C(=O)/C(=C/c3c(cccc3Cl)Cl)/CO2 2W-0613 c1ccc2c(c1)C(=O)/C(=C/c3c(cccc3Cl)F)/CO2 2W-0614 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6ccc(cc6)C#N 2W-0618 c1ccc(cc1)Sc2ccc(cc2)c3ccc4cc(cc(c4n3)Br)Br 2W-0800 c1ccc(c(c1)NC(=O)Nc2cccc(c2)c3cn4cccnc4n3)F 2W-0802 c1cc(cc(c1)NC(=O)c2ccc(cc2Cl)Cl)c3cn4cccnc4n3 2W-0803 c1ccc(cc1)Sc2ccc(cc2)c3ccc4ccccc4n3 2W-0804 c1ccc2c(c1)ccc(n2)c3ccc(cc3)n4ccnc4 2W-0805 c1cc(ccc1c2ccc3cc(cc(c3n2)Br)Br)n4ccnc4 2W-0806 Cc1c(n(ccc1=O)CCc2c[nH]cn2)C 2W-0807 Cc1c2c(nc(n1)n3cc(nn3)C(=O)NCCN4CCOCC4)CCC2 2W-0808 CCOC(=O)c1c(n(nn1)c2nc(cc(n2)C(F)(F)F)c3ccccc3)C(=O)OCC 2W-0809 CC1(CN(C1=O)c2cccc(c2)c3ccnc4n3ncc4c5ccc(cc5)Cl)C 2W-0810 CCCCCCc1c(nnn1c2nc(cc(n2)C(F)(F)F)c3ccccc3)C(=O)OC 2W-0811 CC1=NN(C(=O)c2ccccc2O1)Cc3cccc(c3)C(F)(F)F 2W-0813 CC(C)(C)NC(=S)NCc1ccc(cc1)OC 2W-0814 CC1(CN(C1=O)c2cccc(c2)c3ccnc4n3ncc4c5cccs5)C 2W-0819 Cc1c2ccccc2nc(c1C(=O)OC)C(=O)OC 2W-0820 COC(=O)c1c(n(nn1)c2ccsc2C(=O)OC)C(=O)OC 2W-0822 CC(=O)c1ccc(cc1)N2CCOCC2 2W-0823 Cc1c2cc3c(cc2nc(c1C(=O)OC)C(=O)OC)OCO3 2W-0824 Cc1c(cc2cc(cc(c2n1)Br)Br)O 2W-0825 c1ccc2c(c1)ccc(n2)c3cnccn3 2W-0826 c1cc(nc2c1cc(cc2Br)Br)c3cnccn3 2W-0827 c1ccc2c(c1)ccc(n2)c3ccc(cc3)N4CCOCC4 2W-0828 c1cc(ccc1c2ccc3cc(cc(c3n2)Br)Br)N4CCOCC4 2W-0829 c1cc2c(nc1)nc3n(c2=O)CCCCC3 2W-0830 c1ccc(cc1)S(=O)(=O)c2ccc(cc2)c3ccc4cc(cc(c4n3)Br)Br 2W-0832 c1ccc(cc1)c2cc(nc(n2)n3c(c(nn3)CO)CO)C(F)(F)F 2W-0835 Cc1c(c(n2c(n1)nnn2)C)Cc3ccc(cc3)Cl 2W-0836 c1cc(c(nc1)n2c(cc(n2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] 2W-0837 CCc1nc2cc(ccc2o1)N 2W-0838 Cc1c(cc2cc(cc(c2n1)Br)Br)OCc3ccc(cc3)Cl 2W-0840 C/C(=N/O)/c1cnccn1 2W-0841 c1cc2c(cc1[N+](=O)[O-])c(=O)n3c(n2)CCCCC3 2W-0842 CCCc1c(nn(c1C)c2c(cccn2)N)C 2W-0844 Cc1c(c(nn2c1nnc2)C)Cc3ccc(cc3)Cl 2W-0845 CN(C)/C=C/C(=O)C1CCCCC1=O 2W-0847 Cc1c(n(ccc1=O)c2cccc(c2)SC)C 2W-0848 C/C(=N\OC(=O)c1ccc(cc1)F)/c2cnccn2 2W-0851 C/C(=N\OC(=O)c1ccccc1F)/c2cnccn2 2W-0852 C/C(=N/OC(=O)c1ccc(cc1)Cl)/c2cnccn2 2W-0853 CN(C)/C=C/C(=O)c1ccc(cc1)N2CCOCC2 2W-0854 Cc1nc2ccc(cc2o1)NC(=O)c3cccs3 2W-0855 CCCCCC(=O)Nc1ccc2c(c1)oc(n2)C 2W-0856 Cc1nc2ccc(cc2o1)NC(=O)c3cccc(c3)C(F)(F)F 2W-0857 Cc1nc2ccc(cc2o1)NS(=O)(=O)C 2W-0858 Cc1ccc(cc1)NC(=O)Nc2ccc3c(c2)oc(n3)C 2W-0859 Cc1nc2ccc(cc2o1)NC(=S)NC 2W-0860 Cc1nc2ccc(cc2o1)NC(=S)NCC=C 2W-0861 CC1=NN(C(=O)c2ccccc2O1)Cc3cnc(s3)Cl 2W-0864 CCOC(=O)CN1C(=O)c2ccccc2OC(=N1)C 2W-0866 CC1=NN(C(=O)c2ccccc2O1)c3c(cc(cn3)C(F)(F)F)Cl 2W-0867 CC1=NN(C(=O)c2ccccc2O1)c3c(cccn3)[N+](=O)[O-] 2W-0868 Cc1nc2ccc(cc2o1)NC(=O)NC(C)(C)C 2W-0869 c1cc2c(cc1I)c(=O)n3c(n2)CCCCC3 2W-0870 Cc1cc(nc(n1)n2cccc2C=C(C#N)C#N)c3c(ccs3)Cl 2W-0871 c1cc(n(c1)c2nccc(n2)c3cccs3)C=C(C#N)C#N 2W-0872 c1cc(ccc1c2ccnn2c3ccc(cc3)F)N4CCOCC4 2W-0873 c1ccc2c(c1)ccc(n2)c3nccs3 2W-0874 Cc1ccccc1S(=O)(=O)c2cc3ccccc3nc2N 2W-0875 Cc1c(cc2cc(cc(c2n1)Br)Br)OC 2W-0876 Cc1c(cc2cc(cc(c2n1)Br)Br)Oc3c(cc(cn3)C(F)(F)F)Cl 2W-0878 C/C(=N\OC(=O)c1ccc(cc1)OC)/c2cnccn2 2W-0880 C/C(=N\OC(=O)C1CCCCC1)/c2cnccn2 2W-0881 CCCCCC(=O)O/N=C(\C)/c1cnccn1 2W-0882 c1cc(nc2c1cc(cc2Br)Br)c3nccs3 2W-0883 C/C(=N\OC(=O)c1ccco1)/c2cnccn2 2W-0884 c1ccc2c(c1)C(=O)N(C2=O)n3cccc3C=O 2W-0885 Cc1nc2ccc(cc2o1)NC(=O)C(F)(F)F 2W-0886 Cc1nc2ccc(cc2o1)NC(=O)C 2W-0887 CCCCc1c(n(nn1)c2nc(cc(n2)c3ccccc3)C)CCCC 2W-0888 c1ccc2c(c1)c(c[nH]2)CCn3ccc(=O)c4c3CCCC4 2W-0889 c1cc(c(nc1)n2c(cc(n2)C(F)(F)F)C(F)(F)F)N 2W-0890 CC1=NN(C(=O)c2ccccc2O1)S(=O)(=O)c3ccc(cc3)OC 2W-0891 Cc1nc2ccc(cc2o1)NC=C(C#N)C#N 2W-0893 Cc1ccccc1S(=O)(=O)c2cc3cc(cc(c3nc2N)Br)Br 2W-0895 Cc1c(nc2cc(ccc2n1)NC(=S)NC)C 2W-0897 COc1ccc(cc1OC)c2ccc3cc(cc(c3n2)Br)Br 2W-0898 CCOC(=O)C(=CNc1ccc(cn1)Cl)C(=O)OCC 2W-0899 CCOC(=O)C(=CNc1ccc2c(c1)nc(c(n2)C)C)C(=O)OCC 2W-0902 Cc1c(nc2cc(ccc2n1)NC(=S)NCC=C)C 2W-0903 C/C(=N\OC(=O)N(C)C)/c1c(cc(cn1)C(F)(F)F)N2CCCC2 2W-0904 C/C(=N\OC(=O)C)/c1c(cc(cn1)C(F)(F)F)N2CCCC2 2W-0905 c1cc(ccc1C2CCNCC2)[N+](=O)[O-] 2W-1308 CCOC(=O)c1ccccc1NC(=O)C(c2ccccc2)Cl 2W-1360 c1cc(c(cc1F)F)NC(=O)N 2X-0017 COc1cccc(c1)NC(=O)N 2X-0019 Cc1cnc(nc1c2ccc(c(c2)F)OC)N 2X-0201 COc1cc(c(c(c1OC)[N+](=O)[O-])Cl)[N+](=O)[O-] 2X-0202 Cc1ccc(cc1)c2nc(cs2)CCNc3ccc(cc3[N+](=O)[O-])C(=O)OC 2X-0204 c1ccnc(c1)c2nc(cs2)CCN.Br 2X-0208 C/C(=N\OCc1ccccc1)/c2cccc(c2)N3Cc4ccccc4C3 2X-0211 c1ccnc(c1)c2nc(cs2)CCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F 2X-0215 COc1cc(c(c(c1OC)[N+](=O)[O-])N2CCOCC2)[N+](=O)[O-] 2X-0217 c1ccc(cc1)c2c(c(n(c(=O)c2C#N)N)N)C#N 2X-0221 COc1cccc(c1)CN2c3cc(ccc3N4CSCC4C2=O)C(F)(F)F 2X-0224 c1cc(cc(c1)F)CN2c3cc(ccc3N4CSCC4C2=O)C(F)(F)F 2X-0225 c1cc(cc(c1)C(F)(F)F)CN2c3cc(ccc3N4CSCC4C2=O)C(F)(F)F 2X-0226 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2)N3CCN(CC3)C(=O)OC(C)(C)C)\N 2X-0235 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)c3nc(on3)C4CCCCC4 2X-0236 c1cc(c(cc1C#N)[N+](=O)[O-])N2CCCC2C(=O)O 2X-0238 Cc1ccc(cc1)CN2c3cc(ccc3N4CSCC4C2=O)C(F)(F)F 2X-0240 c1cc2c(cc1C=C(C#N)C#N)OCO2 2X-0244 c1cc2c(cc1C#N)NC(=O)C3N2CCC3 2X-0246 Cc1cccc(c1CN2c3cc(ccc3N4CSCC4C2=O)C(F)(F)F)C 2X-0247 c1ccnc(c1)c2nc(cs2)CCNc3ccc(cc3[N+](=O)[O-])C=O 2X-0248 CC(=O)c1ccc(c(c1)[N+](=O)[O-])NCCc2csc(n2)c3ccccn3 2X-0249 c1cc2c(cc1c3c(c(n(c(=O)c3C#N)N)N)C#N)OCO2 2X-0251 COc1ccc(cc1)S(=O)(=O)N2CCOc3c2cccc3 2X-0254 Cc1ccc(cc1)c2nc(cs2)CCNc3ccc(cc3[N+](=O)[O-])C(=O)O 2X-0259 Cc1ccc(cc1)c2nc(cs2)CCNc3ccc(cc3/C=C/C(=O)O)[N+](=O)[O-] 2X-0267 Cc1ccc(cc1)c2nc(cs2)CCNc3ccc(cc3C=O)[N+](=O)[O-] 2X-0268 Cc1ccc(cc1)c2nc(cs2)CCNc3ccc(cc3C(=O)O)[N+](=O)[O-] 2X-0269 CC(C)CC(=O)N1CCC(CC1)(CS(=O)(=O)Cc2ccc(cc2)Cl)O 2X-0272 c1cc(cc(c1)Cl)CN2c3cc(ccc3N4CSCC4C2=O)C(F)(F)F 2X-0273 c1cc(c(c(c1)Cl)CN2c3cc(ccc3N4CSCC4C2=O)C(F)(F)F)F 2X-0274 c1ccc(c(c1)CSC2=NC(C3=C(N2)c4ccccc4C3=O)c5ccc6c(c5)OCO6)Cl 2X-0276 c1ccc(c(c1)CSC2=NC(C3=C(N2)c4ccccc4C3=O)c5ccc6c(c5)OCO6)F 2X-0277 c1ccc(cc1)Nc2nc(cs2)CCN3C(=O)c4ccccc4C3=O 2X-0279 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)c3nc(on3)c4ccc(c(c4)Cl)Cl 2X-0284 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)c3nc(on3)c4ccc(cc4)F 2X-0285 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)c3nc(on3)c4ccc(cc4Cl)Cl 2X-0286 CC(=O)Nc1nc(cs1)CCN2C(=O)c3ccccc3C2=O 2X-0287 CNc1nc(cs1)CCN2C(=O)c3ccccc3C2=O 2X-0288 COc1cccc(c1)CSC2=NC(C3=C(N2)c4ccccc4C3=O)c5ccc6c(c5)OCO6 2X-0289 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2ccc3c(c2)OCO3)C(=O)OC 2X-0292 COc1ccc(c(c1)/C=N/NC(=S)N)OC 2X-0293 COc1ccc(c(c1)/C=N/Nc2nc(cs2)CCN3C(=O)c4ccccc4C3=O)OC 2X-0295 CN(C)/C=N/c1ncc(s1)C(=O)c2ccc(cc2)OC 2X-0296 CN(CC(=O)O)c1ccc(cc1[N+](=O)[O-])C(F)(F)F 2X-0297 c1ccnc(c1)c2nc(cs2)CCNC(=O)c3ccc(cc3)[N+](=O)[O-] 2X-0301 CCOC(=O)c1csc(n1)Nc2ncc(c(n2)c3ccc(c(c3)F)OC)C 2X-0302 c1cc(ccc1C(=O)C2CC2)Br 2X-0304 c1cc(cc(c1)C(F)(F)F)COc2ccc(cc2)C=O 2X-0306 Cc1ccc(cc1)C2C(C(=C(C(C2(C#N)C#N)c3ccc(cc3)C)C(=O)OC)O)C(=O)OC 2X-0310 Cc1ccc(cc1)C2C(=C(OC(=C2C(=O)OC)CC(=O)OC)N)C#N 2X-0311 Cc1ccc(cc1)c2nc(cs2)CCNC(=O)c3cccnc3 2X-0312 CCC(=O)c1cnc([nH]c1=O)NC(=S)N 2X-0315 c1c(nc([nH]c1=O)NC(=S)N)C(F)(F)F 2X-0318 CCOC(=O)c1cnc([nH]c1=O)Nc2nc(cs2)c3ccc(cc3)OC 2X-0319 Cc1ccc(cc1)CN2c3cc(ccc3N4CCCC4C2=O)C#N 2X-0321 c1ccc2c(c1)-c3c(c(c(c(n3)/C=C/c4ccc(cc4)O)C#N)c5ccc6c(c5)OCO6)C2=O 2X-0324 CCN(CC)c1ccc(cc1)C(=O)c2cnc(s2)/N=C/N(C)C 2X-0327 CN(C)/C=N/c1ncc(s1)C(=O)c2ccc(cc2)c3ccccc3 2X-0328 Cc1cnc(nc1c2ccc(c(c2)F)OC)NC(=S)N 2X-0330 CCOC(=O)c1csc(n1)Nc2[nH]c(=O)cc(n2)C(F)(F)F 2X-0332 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)Nc4ccc(c(c4)Cl)Cl 2X-0336 COC(=O)c1ccc(cc1)c2ccc(cc2)Cl 2X-0700 c1cc(ccc1c2ccc(cc2)Cl)C(=O)O 2X-0702 c1cc2c(n[nH]c2nc1)N 2X-0703 CC(=O)c1c(nn(c1Cl)C)C(F)(F)F 2X-0704 COC(=O)c1c(c2cccnc2s1)N 2X-0705 Cn1c2c(cccn2)c(n1)N 2X-0707 COC(=O)c1ccc(cc1)c2ccc(cc2)[N+](=O)[O-] 2X-0709 c1cc2c(noc2nc1)N 2X-0710 c1ccc(cc1)COC(=O)NC(c2ccc(cc2)Cl)C(=O)O 2X-0711 COC(=O)C(c1ccc(cc1)Cl)N.Cl 2X-0715 COC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] 2X-0716 Cc1cc(cc(c1O)C)c2csc(n2)N 2X-0717 c1cc(c(nc1)N)C=O 2X-0724 CCOC(=O)C(c1ccccc1)N2CCN(CC2)Cc3ccccc3 2X-0725 CCOC(=O)C(c1ccccc1)n2cccn2 2X-0726 COC(=O)c1c(ccs1)Oc2ccc(cc2N)N 2X-0727 COC(=O)c1c(ccs1)Oc2ccc(cc2)N 2X-0728 c1ccc(cc1)c2ncc(s2)C=O 2X-0730 COC(=O)c1ccc(cc1)c2ccc(cc2)N 2X-0732 Cc1ccc(c2c1c3cc(ccc3n2C=O)OC)C 2X-0802 Cc1ccc(c2c1c3cc(ccc3n2CC(=O)OC(C)(C)C)[N+](=O)[O-])C 2X-0803 COc1ccc(cc1Cl)/C=C/2\C(=O)OC(=N2)c3ccccc3I 2X-0804 CC1(C(=O)Nc2c(cccn2)O1)C(=O)NCc3ccccc3OC 2X-0805 CN1CC(C(C1)C(=O)c2ccc(cc2)F)c3ccc(c(c3)Cl)OC 2X-0806 c1cc(c(cc1CC(=O)O)[N+](=O)[O-])O 2X-0807 c1ccc2c(c1)OCC(O2)C(=O)Nc3ccc(cc3)C(=O)O 2X-0808 CC1(C(=O)Nc2c(cccn2)O1)C(=O)NCc3ccc(c(c3)Cl)Cl 2X-0809 CC1(C(=O)Nc2ccccc2O1)C(=O)NC(c3ccccc3)C(=O)OC 2X-0810 c1ccc2c(c1)OCC(O2)C(=O)N3CCN(CC3)C(=O)c4cccs4 2X-0811 COC(=O)c1c(c2ccccc2[nH]1)/C=N/O 2X-0817 CC(=O)N1CCN(CC1)Cc2ccc(nc2)Cl 2X-0818 Cc1cccc(c1N2CCN(CC2)Cc3ccc(nc3)Cl)C 2X-0819 c1ccc2c(c1)c(=O)c(co2)/C=C(\C#N)/c3nc(cs3)c4ccccc4F 2X-0822 c1ccc(cc1)CNC(=O)c2cn[nH]c2C(F)(F)F 2X-0823 CCOC(=O)COc1ccccc1C(=O)c2cnn(c2)c3ccccc3 2X-0824 CC1(C(=O)Nc2ccccc2O1)C(=O)NCc3ccc(c(c3)Cl)Cl 2X-0826 Cc1ccc(cc1)CNC(=O)C2(C(=O)Nc3ccccc3O2)C 2X-0827 Cc1cc(n(n1)c2nc(cs2)C(=O)NNC(=S)NCCC3=CCCCC3)C(F)(F)F 2X-0830 c1ccc(cc1)c2ccc(cc2)c3csc(n3)/C(=C/c4coc5ccccc5c4=O)/C#N 2X-0832 CC1CCCN(C1)Cc2ccc(nc2)Cl 2X-0833 c1c(c([nH]n1)C(F)(F)F)C(=O)O 2X-0834 CN(Cc1ccccc1)Cc2ccc(nc2)Cl 2X-0835 CC1CCN(CC1)Cc2ccc(nc2)Cl 2X-0836 c1cc2cccnc2c(c1)OCc3ccc(nc3)Cl 2X-0838 c1ccc(cc1)c2c(c3ccccc3n2Cc4ccc(nc4)Cl)Cc5ccc(nc5)Cl 2X-0839 CC1CCCCN1Cc2ccc(nc2)Cl 2X-0841 COC(=O)C1(C2C(C(N1)c3ccc(cc3)Cl)C(=O)OC2=O)Cc4ccccc4 2X-0844 COc1ccc(cc1Cl)/C=N/C(Cc2ccccc2)C(=O)OC 2X-0845 CN1CC(C(C1)C(=O)c2ccc(cc2)C3CCCCC3)c4ccc(c(c4)Cl)OC 2X-0846 c1ccc2c(c1)nc(s2)SCc3ccc(nc3)Cl 2X-0847 c1cc(ncc1Cn2cncn2)Cl 2X-0848 c1ccnc(c1)N2CCN(CC2)Cc3ccc(nc3)Cl 2X-0850 c1cc2c(cc1CN3CCN(CC3)Cc4ccc(nc4)Cl)OCO2 2X-0852 CN(CCC#N)Cc1ccc(nc1)Cl 2X-0853 COC(=O)c1cccc(c1CN2CCCC(C2)C(=O)N)[N+](=O)[O-] 2X-0854 Cc1cc(nc(n1)n2cc(nn2)C(=O)c3ccco3)C(F)(F)F 2X-0857 Cn1c2c(cn1)c(ncn2)N3CCC(CC3)Cc4ccccc4 2X-0859 c1cc(c(cc1CC(=O)O)N)O 2X-0862 CC1(C(=O)Nc2ccccc2O1)C(=O)NCCCN3CCOCC3 2X-0865 Cc1ccc(n1C(CCO)c2cccc(c2)Cl)C 2X-0866 Cc1cc(nc(n1)n2cc(nn2)C(=O)c3ccc(cc3)F)C(F)(F)F 2X-0867 Cc1cc(nc(n1)n2cc(nn2)C(=O)/C=C/c3cccs3)C(F)(F)F 2X-0868 c1cc2c(cc1CC(=O)O)nco2 2X-0870 CC1(C(=O)Nc2ccccc2O1)C(=O)NCc3ccccc3 2X-0872 CC1(C(=O)Nc2ccccc2O1)C(=O)NCCOC 2X-0873 COC(=O)Cc1ccc(c(c1)[N+](=O)[O-])O 2X-0875 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2ccccc2)C(=O)OC 2X-0878 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2ccc(cc2)F)C(=O)OC 2X-0879 COc1ccc(cc1Cl)C2C3C(C(=O)OC3=O)C(N2)(Cc4ccccc4)C(=O)OC 2X-0880 c1ccc(cc1)COc2ccc(cc2)C(CCO)/N=C/c3ccc(cc3)[N+](=O)[O-] 2X-0881 COc1cc(c(c(c1)OC)OC)OC 2X-5005 c1cnccc1NC(=O)C2CC2 2X-5009 c1cc(cnc1)NC(=O)C2CC2 2X-5013 c1ccc2c(c1)C(=O)N(C2=O)CCc3cccc(c3)Br 2X-5027 Cc1cc(n2c(n1)nc(n2)S)C 2X-5046 Cc1cc(n2c(n1)nc(n2)SCC(=O)Nc3ccc(cc3)Cl)C 2X-5069 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCCCC2CCO 2X-7008 c1cc(cc(c1)F)C(=NC#N)N 2X-9008 CS(=O)(=O)c1ccc(cc1)c2csc(n2)NC(=O)Nc3ccccc3F 2Y-0001 c1ccc(c(c1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)C(=O)O 2Y-0005 c1cc(c(cc1C(F)(F)F)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)F 2Y-0006 c1ccc(c(c1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCCO4)[N+](=O)[O-] 2Y-0052 CC(=O)NNC(=O)c1cccnc1 2Y-0058 c1cc(c(cc1Cl)Cl)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 2Y-0092 c1ccc(c(c1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCCO4)C(F)(F)F 2Y-0093 COC(=O)C(CC=C)(c1c(cccc1Cl)[N+](=O)[O-])C(=O)OC 2Y-0222 Cn1c(c(c(n1)C(F)(F)F)C#N)OC(=O)c2ccc(cc2)F 2Y-0237 Cn1c(c(c(n1)C(F)(F)F)C#N)OS(=O)(=O)c2ccccc2 2Y-0248 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Oc3c(c(nn3C)C(F)(F)F)C#N 2Y-0249 Cn1c(c(c(n1)C(F)(F)F)C#N)OC(=O)c2c(cccc2F)F 2Y-0253 COC(=O)C(CC#C)(c1cc(ccc1[N+](=O)[O-])C(F)(F)F)C(=O)OC 2Y-0256 COC(=O)C(CC=C)(c1cc(ccc1[N+](=O)[O-])C(F)(F)F)C(=O)OC 2Y-0257 c1c(c2c([nH]1)ncnc2Cl)I 2Y-0261 CC(=O)OCCCc1cnc2nc(nn2c1)N 2Y-0700 c1cc(ncc1[N+](=O)[O-])N2CCC(CC2)C(=O)O 2Y-0705 COC(=O)C1CCN(CC1)S(=O)(=O)C 2Y-0706 c1cc(ncc1C(=O)O)N2CCOCC2 2Y-0709 CCOC(=O)c1ccc(cc1)CN2Cc3ccccc3C2=O 2Y-0800 c1ccc2c(c1)c(cs2)C(=O)CBr 2Y-0801 CCOC(=O)c1c(nn(c1C)S(=O)(=O)c2ccccc2[N+](=O)[O-])C 2Y-0802 CC(c1ccc(cc1)NC(=O)OC(C)(C)C)C(=O)O 2Y-0803 CCCS(=O)(=O)Nc1cc2c(cc1OC)c3ccccc3o2 2Y-0804 COc1ccc(cc1S(=O)(=O)Nc2cc3c(cc2OC)c4ccccc4o3)Cl 2Y-0805 COc1cc2c3ccccc3oc2cc1NS(=O)(=O)c4ccc(cc4)I 2Y-0806 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(cc3)I 2Y-0808 CN(C)/C=C/C(=O)c1ccsc1 2Y-0809 c1c(cn2c(cnc2c1Cl)Br)C(F)(F)F 2Y-0810 COC(=O)c1ccc2nc(cn2c1)c3ccc(cc3)C4CCCCC4 2Y-0811 CC(C)(CCl)C(=O)Nc1cccc(c1)C#C 2Y-0813 CCOC(=O)c1cc2cc(ccc2o1)Br 2Y-0815 COc1ccc(cc1OC)S(=O)(=O)NCCc2c[nH]c3c2cccc3 2Y-0816 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3cccc4c3nccc4 2Y-0817 c1cc(c(cc1C(=O)CC#N)F)N2CCOCC2 2Y-0818 COC(=O)Cc1ccc2c(c1)nco2 2Y-0819 c1cc(ccc1c2cn3cc(ccc3n2)C(=O)O)C4CCCCC4 2Y-0821 CCCc1nc2cc(ccc2o1)N 2Y-0822 c1cc2c(cc1Br)cc(o2)C(=O)O 2Y-0823 CC1(CN(C1=O)c2cccc(c2)C#C)C 2Y-0824 c1ccc(c(c1)n2cccc2)Br 2Y-0825 Cc1cc(ccc1n2cccc2)Br 2Y-0826 Cc1cc(nc(n1)n2c(c(nn2)CO)CO)C 2Y-0827 Cc1c2cc(ccc2sc1S(=O)(=O)NCCc3c[nH]c4c3cccc4)Cl 2Y-0828 COc1ccc(cc1)c2cc[nH]n2 2Y-0829 COc1ccc(cc1)c2ccnc(n2)N 2Y-0830 c1cc(ccc1/C=C(/C#N)\C(=O)c2ccc(c(c2)F)N3CCOCC3)F 2Y-0831 CCCCS(=O)(=O)NCCc1c[nH]c2c1cccc2 2Y-0832 COc1cccc(c1)/C=C(/C#N)\C(=O)c2ccc(c(c2)F)N3CCOCC3 2Y-0834 c1ccc2c(c1)c(c[nH]2)/C=C(\C#N)/C(=O)c3ccc(c(c3)F)N4CCOCC4 2Y-0835 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CCCCl 2Y-0836 c1cc(cc(c1)[N+](=O)[O-])N2CCCC2=O 2Y-0837 COC(=O)Cc1c(nc(s1)c2ccccc2)c3ccc(cc3)F 2Y-0840 COC(=O)Cc1c(nc(s1)c2ccccc2)c3ccc(cc3)Cl 2Y-0841 Cc1cc(nc(n1)n2cc(nn2)C(=O)OC)C 2Y-0842 c1ccn(c1)c2cccc(c2)Br 2Y-0843 Cc1c(c2ccccc2nc1c3ccc(cc3)O)C(=O)O 2Y-0922 COc1cccc(c1)C2c3cc4cc(ccc4cc3OC(=C2C#N)N)Br 2Y-0924 c1cc(cnc1)C2c3cc4cc(ccc4cc3OC(=C2C#N)N)Br 2Y-0929 c1cc(sc1)C2c3cc4cc(ccc4cc3OC(=C2C#N)N)Br 2Y-0930 Cc1c(c2cc(ccc2nc1c3ccccc3)Cl)C(=O)O 2Y-0931 Cc1c(c2cc(ccc2nc1c3ccc(cc3)O)Cl)C(=O)O 2Y-0933 CC(C)(C)c1ccc(cc1)C2c3cc4cc(ccc4cc3OC(=C2C#N)N)Br 2Y-0935 CCOC(=O)/C(=C/c1cccnc1)/C#N 2Y-0936 Cc1c(c2cc(ccc2nc1c3ccccc3)Cl)C(=O)OC 2Y-0940 CCOC(=O)/C(=C/c1ccc2c(c1)OCO2)/C#N 2Y-0941 c1cc2c(cc1/C=C(\C#N)/C(=O)O)OCO2 2Y-0942 CCOC(=O)/C(=C/c1cccs1)/C#N 2Y-0943 Cc1c(c2cc(ccc2nc1c3cccc(c3)Cl)Cl)C(=O)O 2Y-0944 CCOC(=O)/C(=C/c1ccc(cc1)C)/C#N 2Y-0946 c1cc(sc1)/C=C(\C#N)/C(=O)O 2Y-0947 c1cc(cnc1)/C=C(\C#N)/C(=O)O 2Y-0953 Cc1ccc(cc1)/C=C(\C#N)/C(=O)O 2Y-0954 c1cc(cnc1)/C=C(\C#N)/C(=O)N 2Y-0956 COc1cccc(c1)/C=C(\C#N)/C(=O)N 2Y-0957 CCCc1nc2cc(c(cc2o1)[N+](=O)[O-])Cl 2Y-5006 COc1ccc(cc1Cl)/C=C(\C#N)/c2cccs2 2Y-5008 CCCc1nc2cc(ccc2o1)[N+](=O)[O-] 2Y-5016 Cc1ccc(c2c1c3cc(ccc3[nH]2)c4ccc(cc4)F)C 2Y-5025 Cc1ccc(c2c1c3cc(ccc3[nH]2)c4ccc(cc4)OC)C 2Y-5029 CCCc1nc2cc(ccc2o1)CC(=O)OC 2Y-5030 CCCc1nc2cc(ccc2o1)S(=O)(=O)CC 2Y-5048 CCCc1nc2ccc(cc2o1)[N+](=O)[O-] 2Y-5061 CCc1nc2cc(ccc2o1)S(=O)(=O)CC 2Y-5062 CCS(=O)(=O)c1ccc2c(c1)nco2 2Y-5065 CCCC(=O)Nc1cc(ccc1O)CC(=O)OC 2Y-5071 CCCc1[nH]c(c(n1)C#N)C#N 2Y-5073 c1c2c(c(nc(n2)Cl)Cl)[nH]c1C(=O)O 2Y-7035 CC(C)(c1cccc2c1sc3c2cccc3)O 2Z-0008 Cc1ccccc1Nc2ccccc2C 2Z-0033 c1cc2c(c3c1cc(cc3)Br)C(C(=C(O2)N)C#N)c4ccncc4 2Z-0208 c1cc(cnc1)C=C(C#N)C#N 2Z-0210 COc1ccc2c(c1)OC(=C(C2c3cccnc3)C#N)N 2Z-0211 c1ccc2c(c1)c(cc3c2OC(=C(C3c4cccnc4)C#N)N)Cl 2Z-0218 c1ccc2c(c1)c(cc3c2OC(=C(C3c4ccncc4)C#N)N)Cl 2Z-0219 COc1cccc(c1)C2c3cc(c4ccccc4c3OC(=C2C#N)N)Cl 2Z-0221 c1ccc2c(c1)ccc3c2OC(=C(C3c4ccncc4)C#N)N 2Z-0223 COc1ccc(cc1)C2c3ccc4ccccc4c3OC(=C2C#N)N 2Z-0224 COc1cccc(c1)C2c3ccc4ccccc4c3OC(=C2C#N)N 2Z-0225 c1ccc2cc3c(cc2c1)C(C(=C(O3)N)C#N)c4ccncc4 2Z-0227 CCOC(=O)C1=C(Oc2c3ccccc3ccc2C1c4cccnc4)N 2Z-0235 CC(C)(C)OC(=O)C1=C(Oc2c3ccccc3ccc2C1c4cccnc4)N 2Z-0236 c1cc(sc1C=O)N2CCCC2 2Z-0702 c1cnc(cc1C=O)Cl 2Z-0705 CC1CN(CC(O1)C)C(C)(C)C=O 2Z-0707 c1cc(ccc1Sc2ccc(o2)C=O)Br 2Z-0709 c1cc(c(cc1C(=O)CO)Cl)Cl 2Z-0712 c1cc(ccc1Sc2ccc(o2)C=O)Cl 2Z-0715 c1cc(ccc1Sc2ccc(s2)C=O)Cl 2Z-0716 c1cc(ccc1Sc2ccc(s2)C=O)Br 2Z-0717 c1cc(c(=O)[nH]c1)C=O 2Z-0720 c1cc(=O)[nH]cc1C#N 2Z-0721 c1ccc(cc1)Sc2ccc(o2)C=O 2Z-0722 CCOC(=O)c1cnc(s1)N 2Z-0725 c1cc2nc(cn2cc1Cl)C(=O)NCCO 2Z-0800 CC(=O)Nc1ccc(cc1)OCc2ccccc2C#N 2Z-0804 CCOC(=O)c1c(nn(c1C)c2cccc(c2)C(F)(F)F)C 2Z-0811 Cn1c(c(cnc1=S)C(=O)c2ccccc2)N 2Z-0812 Cc1c(c(n(n1)c2cccc(c2)C(F)(F)F)C)C(=O)O 2Z-0813 c1cc2c(cc1Br)c(c[nH]2)C3=CCNCC3 2Z-0814 Cc1cccc[n+]1CC(=O)c2ccc(cc2)[N+](=O)[O-].[Br-] 2Z-0821 CCOC(=O)c1c2ccccn2cc1c3ccc(cc3)Br 2Z-0822 COc1ccc2c(c1)c(c[nH]2)/C=C\3/c4c(cccc4Cl)NC3=O 2Z-0823 c1cc(ccc1c2cc(on2)N)Br 2Z-0824 COC(=O)Cc1c(cc(cn1)C(F)(F)F)Cl 2Z-0829 c1cc2c(cc1N)C(=O)CCC2 2Z-5003 c1cc2c(cc1N)C(=O)CC2 2Z-5014 Cn1c(nnc1C(F)(F)F)/C(=C/Nc2ccccc2)/[N+](=O)[O-] 3B-001 c1ccc(cc1)N/C=C(/c2nnc(n2c3ccc(cc3)Cl)C(F)(F)F)\[N+](=O)[O-] 3B-002 COc1ccc(cc1)N/C=C(/c2nnc(n2c3ccc(cc3)Cl)C(F)(F)F)\[N+](=O)[O-] 3B-003 CS/C(=C\[N+](=O)[O-])/Nc1cccc(c1)Cl 3B-004 COc1ccc(cc1)n2c(nnc2C(F)(F)F)/C(=C/Nc3ccc(cc3)Cl)/[N+](=O)[O-] 3B-006 c1cc(cc(c1)Cl)Nc2c(cn[nH]2)[N+](=O)[O-] 3B-008 COc1ccc(cc1)n2c(nnc2C(F)(F)F)/C(=C/Nc3cccc(c3)C(F)(F)F)/[N+](=O)[O-] 3B-009 Cc1ccc(cc1)N/C=C(/c2nnc(n2c3ccc(cc3)C)C(F)(F)F)\[N+](=O)[O-] 3B-010 Cc1ccc(cc1)n2c(nnc2C(F)(F)F)/C(=C\Nc3cccc(c3)Cl)/[N+](=O)[O-] 3B-011 CNc1c(cnc(n1)N)[N+](=O)[O-] 3B-012 CC(C)(C)c1cc[nH]n1 3B-013 c1ccc(cc1)n2c(ncn2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F 3B-014 CC(C)(C)c1ccn(n1)CC(=O)c2ccc(cc2)Cl 3B-015 CC(C)(C)c1c(c[nH]n1)Br 3B-016 CS/C(=C\[N+](=O)[O-])/Nc1ccc(cc1)F 3B-017 c1cc(ccc1N/C(=C/[N+](=O)[O-])/NN)F 3B-018 CC(C)(C)c1c(c[nH]n1)[N+](=O)[O-] 3B-019 c1cc(ccc1n2c(nnc2C(F)(F)F)C[N+](=O)[O-])F 3B-020 COc1cccc(c1)N/C=C(/c2nnc(n2c3ccc(cc3)F)C(F)(F)F)\[N+](=O)[O-] 3B-023 CN/C(=N\NC(=O)C(Cl)(Cl)Cl)/C[N+](=O)[O-] 3B-024 C/N=C(/C[N+](=O)[O-])\NN=C(SC)SC 3B-027 CN(C)c1c(cnc(n1)NC(=O)Nc2ccccc2)c3ccccc3 3B-028 c1cc(c(cc1OCC(F)(F)F)c2ncno2)OCC(F)(F)F 3B-029 c1cc(ccc1n2c(nnn2)N)Cl 3B-030 c1cc(ccc1Nc2c(cn[nH]2)[N+](=O)[O-])F 3B-031 c1ccc(cc1)CN(Cc2ccccc2)C#N 3B-036 CC(C)(C)N1C(CC(=O)CC1=O)c2ccc(cc2)Cl 3B-037 c1ccc(c(c1)CN(Cc2ccccc2Cl)C#N)Cl 3B-038 COC(c1ccc(c(n1)O)C#N)OC 3B-040 C=CCN(CC=C)C#N 3B-041 c1cc2c(cc1Cl)SCC(=O)N2 3B-045 c1cnn2c1C(n3c(ccn3)C2O)O 3B-048 c1ccc2c(c1)c([n+](cn2)[O-])N 3B-051 c1cc(nc(c1)Cl)NN 3B-055 CC\1=NNC(=O)/C1=N\Nc2ccccc2 3B-057 CC\1=NNC(=O)/C1=N\Nc2cccc(c2)C(F)(F)F 3B-058 CN(C)c1c(cn(n1)C(=O)Nc2ccccc2)c3ccccc3 3B-059 CC\1=NN(C(=O)/C1=N\Nc2ccccc2)C3=NCCS3 3B-061 CC\1=NN(C(=O)/C1=N\Nc2cccc(c2)C(F)(F)F)C3=NCCS3 3B-062 c1cc(nc(c1)Cl)NN/C=N/C(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 3B-063 CN(C)c1c(cn(n1)C(=O)Nc2ccc(cc2)Cl)c3ccccc3 3B-064 CN(C)c1c(cn(n1)C(=O)Nc2ccc(cc2Cl)Cl)c3ccccc3 3B-065 CN(C)c1c(cn(n1)C(=S)Nc2ccccc2)c3ccccc3 3B-067 CS(=O)c1ccccc1O 3B-068 CN(C)c1c(cn(n1)C(=O)Nc2cccc(c2)C(F)(F)F)c3ccccc3 3B-069 CC(C)(C)NC(=O)n1cc(c(n1)N(C)C)c2ccccc2 3B-070 CN(C)c1c(cn(n1)C(=S)Nc2ccc(cc2)Cl)c3ccccc3 3B-072 CN(C)c1c(cn(n1)C(=S)Nc2cccc(c2)C(F)(F)F)c3ccccc3 3B-073 CC1=NN(C(=O)C1)C2=NCCCN2 3B-075 CC\1=NN(C(=O)/C1=N\Nc2ccccc2)C3=NCCCN3 3B-077 CC(C)(C)N1C(CC(=O)/C(=C/N(C)C)/C1=O)c2ccc(cc2)OC 3B-084 C1CN=C(N1)C[N+](=O)[O-] 3B-086 Cc1c(c(on1)/C=C/Nc2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] 3C-003 c1cc(c(c(c1)Cl)c2c(c(on2)/C=C/Nc3ccc(cc3F)F)C#N)Cl 3C-004 CN(C)c1c(cn(n1)C(=O)Nc2ccccc2)c3ccc(cc3)Oc4ccccc4 3C-005 c1cc(c(c(c1)Cl)c2c(c(on2)/C=C/Nc3ccc(cc3Cl)Cl)C#N)Cl 3C-006 CN(C)c1c(cn(n1)C(=O)Nc2ccc(cc2Cl)Cl)c3ccc(cc3)Oc4ccccc4 3C-007 c1cc(c(c(c1)Cl)c2c(c(on2)/C=C/Nc3ccc(cc3)C(=O)O)C#N)Cl 3C-009 c1cc(c(c(c1)Cl)c2c(c(on2)/C=C/Nc3cc(cc(c3)Cl)Cl)C#N)Cl 3C-011 COc1ccccc1N/C=C/c2c(c(no2)c3c(cccc3Cl)Cl)C#N 3C-012 c1ccc(c(c1)C(F)(F)F)N/C=C/c2c(c(no2)c3c(cccc3Cl)Cl)C#N 3C-013 COc1ccc(cc1)N/C=C/c2c(c(no2)c3c(cccc3Cl)Cl)C#N 3C-016 COc1ccc(c(c1)OC)N/C=C/c2c(c(no2)c3c(cccc3Cl)Cl)C#N 3C-017 Cc1c(c(n(n1)C)/C=C/Nc2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] 3C-018 CN(C)c1c(cn(n1)C(=O)c2ccccc2)c3ccc(cc3)Oc4ccccc4 3C-027 c1ccc(cc1)c2ccccc2N/C=C/c3c(c(no3)c4c(cccc4Cl)Cl)C#N 3C-030 Cc1ccc(cc1)N/C=C/c2c(c(no2)c3c(cccc3Cl)Cl)C#N 3C-033 Cc1cc(ccc1N/C=C/c2c(c(no2)c3c(cccc3Cl)Cl)C#N)O 3C-035 CN(C)c1c(cnc(n1)N)c2ccc(cc2)Oc3ccccc3 3C-047 CC(=O)C(Cc1ccc(cc1)O)C(=O)C 3C-059 Cc1c(c(n[nH]1)C)Cc2ccc(cc2)O 3C-062 Cc1c(c(ns1)SC)C#N 3C-072 CN(C)/C=C/c1c(c(ns1)SC)C#N 3C-075 CN(C)/C=C(\C#N)/c1ccc(cc1)Cl 3C-083 Cc1c(c(no1)c2c(cccc2Cl)F)C#N 3C-084 c1ccc(cc1)N/C=C(/C#N)\c2ccc(cc2)Cl 3C-086 COc1ccccc1N/C=C(/C#N)\c2ccc(cc2)Cl 3C-087 COc1cccc(c1)N/C=C(/C#N)\c2ccc(cc2)Cl 3C-088 COc1ccc(cc1)N/C=C(/C#N)\c2ccc(cc2)Cl 3C-089 Cc1ccc(cc1)N/C=C(/C#N)\c2ccc(cc2)Cl 3C-090 c1cc(c(c(c1)Cl)C(=O)NNc2ccc(cc2)OC(F)(F)F)Cl 3C-091 c1cc(ccc1/C(=C/Nc2cc(ccc2O)Cl)/C#N)Cl 3C-093 c1cc(ccc1/C(=C\Nc2ccc(cc2)Cl)/C#N)Cl 3C-094 c1cc(ccc1/C(=C\Nc2cc(cc(c2)Cl)Cl)/C#N)Cl 3C-095 CN(C)/C=C/c1c(c(no1)c2c(cccc2Cl)F)C#N 3C-096 c1cc(ccc1NNC(=O)c2ccc(cc2Cl)Cl)OC(F)(F)F 3C-097 CCOC(=O)c1cnc2nc(nn2c1N)SC 3C-098 c1ccc(c(c1)N/C=C(/C#N)\c2ccc(cc2)Cl)O 3C-099 c1ccc(c(c1)C(=O)NNc2ccc(cc2)OC(F)(F)F)C(F)(F)F 3C-101 Cc1ccccc1N/C=C(/C#N)\c2ccc(cc2)Cl 3C-104 Cc1cccc(c1)N/C=C(/C#N)\c2ccc(cc2)Cl 3C-105 c1cc(cc(c1)Cl)N/C=C(/C#N)\c2ccc(cc2)Cl 3C-106 c1cc(cc(c1)N/C=C(\C#N)/c2ccc(cc2)Cl)C(F)(F)F 3C-108 c1ccc(c(c1)N/C=C(/C#N)\c2ccc(cc2)Cl)Cl 3C-109 c1ccc(cc1)N/C=C/c2c(c(no2)c3c(cccc3Cl)F)C#N 3C-112 Cc1c(c(n(n1)C)C)Cc2ccc(cc2)O 3C-113 CSc1nc2ncc(c(n2n1)N)C(=O)O 3C-114 c1cc(c(c(c1)Cl)c2c(c(on2)/C=C/Nc3ccc(cc3)C(=O)O)C#N)F 3C-115 c1ccc(cc1)CNC(=O)c2ccccc2N 3C-117 c1cc(ccc1/C(=C\NNC(=O)c2ccc(cc2)Cl)/C#N)Cl 3C-131 c1cc(ccc1N2C(=O)CC(=N2)C(F)(F)F)OC(F)(F)F 3C-133 c1cc(c(c(c1)Cl)c2c(c(on2)/C=C/Nc3ccc(cc3)Cl)C#N)F 3C-134 CSc1nc2nccc(n2n1)N 3C-136 Cc1csc(n1)NC(=N)N 3C-137 CN(C)/C=C/1\C(=NN(C1=O)c2ccc(cc2)OC(F)(F)F)C(F)(F)F 3C-138 CCOC(=O)c1c(c2c(snc2s1)C)N 3C-140 c1cc(ccc1N/C=C/2\C(=NN(C2=O)c3ccc(cc3)OC(F)(F)F)C(F)(F)F)Cl 3C-141 COC(=O)c1ccc(cc1)N/C=C/2\C(=NN(C2=O)c3ccc(cc3)OC(F)(F)F)C(F)(F)F 3C-142 c1cc(ccc1N2C(=O)/C(=C/Nc3cc(cc(c3)Cl)Cl)/C(=N2)C(F)(F)F)OC(F)(F)F 3C-143 COC(=O)c1c(ccs1)N/C=C/2\C(=NN(C2=O)c3ccc(cc3)OC(F)(F)F)C(F)(F)F 3C-144 Cc1cc(ccc1NC=C2C(=NNC2=O)C(F)(F)F)O 3C-149 CN(C)C(=O)c1cc(c[nH]1)C(=O)Cc2ccccc2 3D-002 c1ccc(cc1)NNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)Cl 3D-013 c1cc(ccc1C(=O)CSc2ccc(cc2)Cl)Cl 3D-014 c1cc(ccc1C(=O)CS(=O)(=O)c2ccc(cc2)Cl)Cl 3D-018 CN(C)/C=C(\c1ccccc1)/C(=O)c2cc([nH]c2)C(=O)N(C)C 3D-019 c1ccc(c(c1)Oc2ccc(cc2[N+](=O)[O-])C=O)Cl 3D-026 c1cc(ccc1Nn2cnc-3nncc3c2N)Cl 3D-032 c1cc(c(cc1Cl)Cl)Nn2cnc-3nncc3c2N 3D-033 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl)Cl 3D-034 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 3D-035 c1ccc(c(c1)Nn2cnc-3nncc3c2N)F 3D-037 c1cc(nc(c1)Cl)NNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)Cl 3D-038 c1cc(nc(c1)Cl)NNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3Cl)Cl 3D-040 c1ccc(c(c1)Oc2ccc(cc2[N+](=O)[O-])/C=N/O)Cl 3D-041 CO/N=C/c1ccc(c(c1)[N+](=O)[O-])Oc2ccccc2Cl 3D-042 CC(=O)Nc1ccc(cc1)Oc2cnc3ccccc3n2 3D-043 CC(=O)Nc1cccc(c1)Oc2cnc3ccccc3n2 3D-044 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 3D-045 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NNc3cccc(n3)Cl 3D-046 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NNc3ccccc3 3D-047 c1ccc(cc1)NNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3Cl)Cl 3D-048 COC(=O)c1cc(c[nH]1)/C(=N\Nc2ccccc2)/Cc3ccccc3 3D-049 CN(C)/C=C(\c1ccc(cc1)Cl)/S(=O)(=O)/C=C/c2ccc(cc2)Cl 3D-053 c1cc(c(cc1c2ccnc3n2nc(n3)N4CCOCC4)Cl)Cl 3D-055 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])/C=C/C(=O)O)Cl 3D-056 c1cc(cc(c1)Cl)Oc2ccc(cc2[N+](=O)[O-])/C=C/C(=O)O 3D-057 c1ccc(c(c1)Oc2ccc(cc2[N+](=O)[O-])/C=C/C(=O)O)Cl 3D-058 CC1(Cc2c(cnc3n2nc(n3)SC)C(=O)C1)C 3D-059 CC(c1ccnc2n1nc(n2)SC)Oc3ccc(cc3Cl)Cl 3D-060 CC(c1ccnc2n1nc(n2)N3CCOCC3)Oc4ccc(cc4Cl)Cl 3D-061 CC(c1ccnc2n1nc(n2)N3CCOCC3)Oc4ccccc4 3D-062 c1ccc(cc1)c2ccnc3n2nc(n3)N4CCN(CC4)c5ccccc5 3D-063 COc1ccc(cc1)c2ccnc3n2nc(n3)N4CCN(CC4)c5ccccc5 3D-070 c1ccc(cc1)N2CCN(CC2)c3nc4nccc(n4n3)c5ccc(cc5)F 3D-072 CN(C)C(=O)c1cc(c[nH]1)c2c(cnc(n2)N)c3ccccc3 3D-073 COc1ccc(cc1)c2cnc3nc(nn3c2N)N4CCN(CC4)c5ccccc5 3D-075 c1ccc(cc1)N2CCN(CC2)c3nc4nccc(n4n3)c5ccc(cc5)Oc6ccccc6 3D-076 c1ccc(cc1)N2CCN(CC2)c3nc4ncc(c(n4n3)N)c5ccc(cc5)F 3D-077 c1cc(c(c(c1)Cl)CSc2nc([nH]n2)N)Cl 3D-079 Cc1ccc(c(c1)F)NC(=S)NC(=O)/C=C/c2ccc(c(c2)OC)OC 3D-081 Cc1cc(ccc1NC(=S)NC(=O)/C=C/c2ccc(c(c2)OC)OC)F 3D-082 COc1ccc(cc1OC)C2CC(=O)N/C(=N\c3ccc(cc3F)Cl)/S2 3D-084 c1cc(c(c(c1)Cl)CSc2nc3ncc(c(n3n2)N)c4ccc(cc4)F)Cl 3D-087 c1ccc(cc1)N2CCN(CC2)c3nc4nccc(n4n3)c5ccc(cc5)n6ccnc6 3D-088 c1ccc(cc1)c2ccnc3n2nc(n3)SCc4c(cccc4Cl)Cl 3D-089 CN(C)C(=O)c1cc(c[nH]1)c2c(c[nH]n2)c3ccccc3 3D-090 c1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3cnc4ccccc4n3 3D-091 c1ccc2c(c1)ncc(n2)Oc3ccc(cc3)NC(=O)c4ccc(cc4)Cl 3D-092 c1ccc2c(c1)ncc(n2)Oc3ccc(cc3)NC(=O)CCl 3D-095 COc1ccc(cc1)c2ccnc3n2nc(n3)SCc4c(cccc4Cl)Cl 3D-096 c1ccnc(c1)c2ccnc3n2nc(n3)SCc4c(cccc4Cl)Cl 3D-097 c1cc(c(c(c1)Cl)CSc2nc3ncc(c(n3n2)N)c4ccc(cc4)Cl)Cl 3D-098 COc1ccc(cc1)c2cnc3nc(nn3c2N)SCc4c(cccc4Cl)Cl 3D-099 c1ccc2c(c1)ncc(n2)Oc3ccc(cc3)NC(=O)C(Cl)Cl 3D-100 c1ccc2c(c1)ncc(n2)Oc3ccc(cc3)NS(=O)(=O)c4ccc(cc4)Cl 3D-102 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3cnc4ccccc4n3 3D-103 c1cc(c(c(c1)Cl)CSc2nc([nH]n2)N)F 3D-104 COc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3cnc4ccccc4n3 3D-105 c1ccc2c(c1)ncc(n2)Oc3ccccc3[N+](=O)[O-] 3D-106 CSc1nc2nccc(n2n1)c3ccc(cc3Cl)Cl 3D-107 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)F 3E-001 CO/N=C/CS(=O)(=O)c1ccc(cc1)Cl 3E-002 CN(C)/C=C(\C=N\OC)/S(=O)(=O)c1ccc(cc1)Cl 3E-003 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)Cl 3E-005 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 3e-006 c1cc(c(cc1F)F)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 3E-007 c1cc(c(c(c1)F)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)F 3E-008 c1cc(c(cc1Cl)Cl)CO/N=C(/c2ccncc2)\N 3E-010 c1cc(c(c(c1)Cl)CONC(=O)N/C=N/OCc2c(cccc2Cl)Cl)Cl 3E-011 c1ccc(cc1)Cc2c3ccccc3c(nn2)Sc4ccc(cc4)Cl 3E-012 c1cc(c(c(c1)Cl)CONC(=O)N/C=N/O)Cl 3E-014 c1cc(ccc1OC(=O)CC(=O)O)F 3E-015 COc1ccc(cc1)OC(=O)CC(=O)O 3E-016 c1ccc(cc1)Cc2c3ccccc3c(nn2)NCc4ccc(cc4)Cl 3E-018 CN(C)/C=C/C(=O)Oc1ccc(cc1)OC 3E-021 CN(C)/C=N/C(=O)NOCc1ccc(c(c1)Cl)Cl 3E-023 c1ccc(cc1)Cc2c3ccccc3c(nn2)NCc4ccccc4 3E-024 COc1ccc(cc1)OC(=O)C/C=N\OCc2c(cccc2Cl)Cl 3E-025 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccccc2Cl 3E-026 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2F)F 3E-027 CCC(=O)c1cc([nH]c1)C(=O)N(C)C 3E-029 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2ccccc2F 3E-030 c1cc(ccc1n2c(c(nn2)C(=O)O)CC(=O)O)Cl 3E-032 CN(C)C(=O)c1cc(c[nH]1)C(=O)c2c(cccc2F)F 3E-033 c1cc(ccc1n2c(c(nn2)C(=O)O)CC(=O)O)OC(F)(F)F 3E-034 COc1ccc(cc1)n2c(c(nn2)C(=O)O)CC(=O)O 3E-035 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)N(C)C 3E-036 c1ccc(cc1)Cc2c3ccccc3c(nn2)Sc4ccccn4 3E-037 c1cc(c(cc1CONC(=O)N)Cl)Cl 3E-038 COc1ccc(cc1)CNc2c3ccccc3c(nn2)Cc4ccccc4 3E-039 CN(C)/C=C/C(=O)Oc1ccc(cc1)F 3E-040 c1cc(c(c(c1)Cl)CO/N=C\CC(=O)Oc2ccc(cc2)F)Cl 3E-041 c1ccc(cc1)Cc2c3ccccc3c(nn2)NCc4cccc(c4)C(F)(F)F 3E-043 c1ccc(cc1)Cc2c3ccccc3c(nn2)Oc4ccccc4 3E-045 c1ccc2c(c1)C(OC2=O)NC(=O)N 3E-046 c1cc(cc(c1)n2c(c(nn2)C(=O)O)CC(=O)O)C(F)(F)F 3E-048 CN(C)CCCNc1c2ccccc2c(nn1)Cc3ccccc3 3E-049 c1ccc(cc1)Cc2c3ccccc3c(nn2)Oc4ccc(cc4)F 3E-051 CCOC(=O)C(=C(c1ccccc1)c2ccccc2)CC(=O)O 3E-052 COc1ccc(cc1)Oc2c3ccccc3c(nn2)Cc4ccccc4 3E-053 c1cc(ccc1CONC(=O)N)[N+](=O)[O-] 3E-054 Cc1ccc(cc1)Oc2c3ccccc3c(nn2)Cc4ccccc4 3E-055 CO/N=C/NC(=O)NOCc1ccc(c(c1)Cl)Cl 3E-058 c1cc(c(cc1CONC(=O)N/C=N/OCc2ccc(cc2Cl)Cl)Cl)Cl 3E-059 COCCCNc1c2ccccc2c(nn1)Cc3ccccc3 3E-060 c1cc(c(cc1CONC(=O)N/C=N/O)Cl)Cl 3E-061 CN(C)/C=N/C(=O)NOCc1ccc(cc1)[N+](=O)[O-] 3E-063 c1cc(ccc1CONC(=O)N/C=N\O)[N+](=O)[O-] 3E-064 CO/N=C\NC(=O)NOCc1ccc(cc1)[N+](=O)[O-] 3E-065 c1ccc(cc1)Cc2c3ccccc3c(nn2)Oc4cccc(c4)C(F)(F)F 3E-066 Cc1cc(ns1)O 3E-067 c1ccc(cc1)Cc2c3ccccc3c(nn2)Oc4ccc(cc4)C#N 3E-068 Cc1c(c(ns1)O)Br 3E-070 c1cc(c(cc1Cl)Cl)CONC(=O)N/C=N/O 3E-071 CC(C)(C#N)N1CCN(CC1)c2ccccc2 3E-073 CN(C)/C=C(\C#N)/C(=O)N/C=N/OCc1ccc(cc1Cl)Cl 3E-074 c1ccc(cc1)Cc2c3ccccc3c(nn2)SCc4ccccc4 3E-075 c1ccc(cc1)c2c(n3c(n2)SCC3)/C=N/OCc4ccc(cc4Cl)Cl 3E-301S c1ccc(cc1)c2c(n3c(n2)SCC3)C#N 3E-303S c1ccc(cc1)c2c(n3ccsc3n2)/C=C/[N+](=O)[O-] 3E-305S c1cc(ccc1c2cn3ccsc3n2)Cl 3E-306S c1cc(ccc1c2c(n3ccsc3n2)C=O)Cl 3E-307S c1cc(ccc1c2cn3c(n2)SCC3)Cl 3E-308S CO/N=C/c1c(nc2n1ccs2)c3ccc(cc3)Cl 3E-309S c1cc(cc(c1)Sc2c(n3ccsc3n2)C#N)C(F)(F)F 3E-310S c1cc(ccc1C(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 3E-311S COc1ccc(cc1)C(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 3E-312S c1cc(cc(c1)C(F)(F)F)C(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 3E-313S CC(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-314S CC(C)(C)C(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-315S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCNC(=O)c2ccc(cc2Cl)Cl)OCC(F)(F)F 3E-316S c1cc(c(cc1C(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl)Cl 3E-317S CCCCC(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-318S CC(C)CC(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-319S Cc1ccc(cc1)S(=O)(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 3E-320S COCCNc1c(c(nc(n1)c2ccccn2)c3cccc(c3)C(F)(F)F)C#N 3E-321S c1ccc(cc1)CNc2c(c(nc(n2)c3ccccn3)c4cccc(c4)C(F)(F)F)C#N 3E-322S c1cc(c(c(c1)Cl)CO/N=C/c2c(nc3n2ccs3)c4ccc(cc4)Cl)Cl 3E-324S c1cc(ccc1c2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl)Cl 3E-325S c1cc(ccc1CO/N=C/c2c(nc3n2ccs3)c4ccc(cc4)Cl)[N+](=O)[O-] 3E-326S c1cc(ccc1c2c(n3ccsc3n2)/C=N/O)Cl 3E-327S c1ccc(cc1)S(=O)(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 3E-328S CS(=O)(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-329S c1cc(cc(c1)S(=O)(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)C(F)(F)F 3E-330S c1cc(ccc1c2c(n3ccsc3n2)C#N)Cl 3E-331S c1cc(cc(c1)Sc2c(n3ccsc3n2)C(=O)N)C(F)(F)F 3E-332S c1ccc(c(c1)S(=O)(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 3E-333S CCN(CC)CCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-334S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCNC(=O)CCl)OCC(F)(F)F 3E-335S c1cc(c(cc1OCC(F)(F)F)C(=O)NCC[NH+]2CCOCC2)OCC(F)(F)F.[Cl-] 3E-336S c1cc(ccc1c2c(n3ccsc3n2)/C=C/[N+](=O)[O-])Cl 3E-337S c1cc(ccc1c2c(n3ccsc3n2)/C=N/c4ccc(cc4)C(F)(F)F)Cl 3E-338S CCNC(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-339S c1ccc(cc1)NC(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 3E-340S c1cc(ccc1NC(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 3E-342S CN(C)S(=O)(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 3E-343S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCN2CCCCC2)OCC(F)(F)F 3E-344S c1cc(ccc1NC(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)OC(F)(F)F 3E-345S c1ccc(cc1)/C(=C/c2c(nc3n2ccs3)c4ccc(cc4)Cl)/C#N 3E-346S c1ccnc(c1)c2nc(c(c(n2)Nc3ccc(cc3)OC(F)(F)F)C#N)c4cccc(c4)C(F)(F)F 3E-347S c1cc(cc(c1)NC(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)C(F)(F)F 3E-348S c1csc2n1c(c(n2)S)C=O 3E-349S c1cc(cc(c1)Cl)CSc2c(n3ccsc3n2)C=O 3E-350S c1cc(cc(c1)Cl)CSc2c(n3ccsc3n2)/C=N/O 3E-351S c1cc(cc(c1)Cl)CSc2c(n3ccsc3n2)C#N 3E-352S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCNC(=O)C(Cl)Cl)OCC(F)(F)F 3E-354S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCNC(=O)C(Cl)(Cl)Cl)OCC(F)(F)F 3E-355S c1cc(cc(c1)C(F)(F)F)CSc2c(n3ccsc3n2)C(=O)O 3E-356S c1ccc(cc1)c2c(n3ccsc3n2)/C=C(\C#N)/c4ccccc4 3E-357S c1ccnc(c1)c2nc(cc(n2)O)C(F)(F)F 3E-358S c1csc2n1c(c(n2)SCc3cc(cc(c3)C(F)(F)F)C(F)(F)F)/C=N/O 3E-360S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)c4ccc(cc4Cl)Cl 3E-361S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)c4cccc(c4)C(F)(F)F 3E-362S c1csc2n1c(c(n2)SCc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C#N 3E-363S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)c4ccc(cc4)Cl 3E-365S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)Nc4ccccc4 3E-366S c1ccnc(c1)c2nc(cc(n2)Cl)C(F)(F)F 3E-367S c1ccc(cc1)Sc2cc(nc(n2)c3ccccn3)C(F)(F)F 3E-369S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)CCl 3E-370S CC(C)(C)C(=O)O/N=C/c1c(nc2n1ccs2)c3ccccc3 3E-371S Cc1ccc(cc1)C(=O)O/N=C/c2c(nc3n2ccs3)c4ccccc4 3E-372S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)c4ccc(c(c4)Cl)Cl 3E-373S c1ccnc(c1)c2nc(cc(n2)SCc3cccc(c3)C(F)(F)F)C(F)(F)F 3E-375S CCOC(=O)c1c(nc2n1cccc2)c3ccccc3 3E-706 CCOC(=O)c1c(nc2n1cc(cc2)C)c3ccccc3 3E-707 CCOC(=O)c1c(nc2n1ccc(c2)C)c3ccccc3 3E-708 CCOC(=O)c1c(nc2n1cccc2C)c3ccccc3 3E-709 CCOC(=O)c1c(nc2n1cc(cc2)Cl)c3ccccc3 3E-715 CCOC(=O)NC(=O)CC(=O)C 3E-900 CCO/C=C(/C(=O)C)\C(=O)NC(=O)OCC 3E-901 CC(=O)c1c[nH]c(=O)[nH]c1=O 3E-902 c1ccc2c(c1)CCC(C2=O)(CO)CO 3E-903 c1ccc2c(c1)CCC3(C2=O)CC3C#N 3E-906 c1ccc(cc1)C2OCC3(CCc4ccccc4C3=O)CO2 3E-907 c1ccc2c(c1)C3(C4CC5CC(C4)CC3C5)C(=N2)[NH3+].[Cl-] 3E-911 c1cc2c(ccnc2cc1Cl)NN 3E-912 CCOC(=O)Cc1c(cccn1)C(=O)O 3E-920 CC(=O)c1cn(c(=O)[nH]c1=O)CCO 3E-923 c1ccc(cc1)C(=O)Nc2cc3c(oc2=O)CCCC3=O 3E-924 Cc1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(=O)OC 3E-925 CC1(OC(=O)C(C(=O)O1)C2(C3CC4CC(C3)CC2C4)C)C 3E-927 CSc1c(c(ns1)O)C#N 3E-928 c1cc(ccc1C(=O)NCC(=O)O)Cl 3E-929 c1cc(ccc1C(=O)Nc2cc3c(oc2=O)CCCC3=O)Cl 3E-930 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)Cl)C(=O)OC 3E-931 CCOC(=O)c1cc(c(=O)oc1c2ccccc2)NC(=O)c3ccc(cc3)Cl 3E-932 COc1ccc(cc1)C(=O)NCC(=O)O 3E-933 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)Cl)C(=O)C 3E-934 CC(=O)c1cc(c(=O)oc1/C=C/N(C)C)NC(=O)c2ccc(cc2)Cl 3E-935 c1cc(cc(c1)C(F)(F)F)C(=O)NCC(=O)O 3E-936 CCOC(=O)c1cc(c(=O)oc1c2ccccc2)NC(=O)c3ccc(cc3)OC 3E-937 Cc1ccc(cc1)S(=O)(=O)NC(=O)n2c(=O)c(c(s2)SC)C#N 3E-940 Cc1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(=O)c3ccccc3 3E-941 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)OC)C(=O)c3ccccc3 3E-942 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)Cl)C(=O)c3ccccc3 3E-943 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)OC)C(=O)C 3E-945 COc1ccc(cc1)C(=O)Nc2cc3c(oc2=O)CCCC3=O 3E-946 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)OC)C(=O)OC 3E-947 CC(=O)c1cc(c(=O)oc1/C=C/N(C)C)NC(=O)c2ccc(cc2)OC 3E-948 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc3c(oc2=O)CCCC3=O 3E-949 Cc1c(c2ccccc2[nH]1)c3ccc(nn3)Cl 3F-001 c1cc(ccc1n2c(=O)cc(c(n2)C(=O)N)O)Cl 3F-003 C1COCCN1C(=O)C(=O)NN 3F-004 CCOC(=O)CC(=N)NNS(=O)(=O)c1ccccc1 3F-006 COC(=O)c1c(cc(=O)n(n1)c2ccccc2)Oc3ccccc3 3F-008 c1ccc(cc1)S(=O)(=O)NNC(=N)COc2ccc(cc2Cl)Cl 3F-009 c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)NN)Oc3ccccc3 3F-010 c1ccc(cc1)n2c(=O)cc(c(n2)C#N)Cl 3F-011 c1cc(ccc1n2c(=O)cc(c(n2)C#N)Cl)Cl 3F-012 c1cc(c(cc1Cl)Cl)CO/N=C/CC(=O)NNC(=N)COc2ccc(cc2Cl)Cl 3F-014 c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)Oc3ccccc3 3F-016 CO/N=C\NC(=O)c1c(cc(=O)n(n1)c2ccccc2)Oc3ccccc3 3F-022 COC(=O)c1c(c2c(s1)cc(=O)n(n2)c3ccc(cc3)Cl)N 3F-023 c1cc(cnc1)C(=N)NNC(=O)C/C=N/OCc2ccc(cc2Cl)Cl 3F-024 c1cc(c(cc1Cl)Cl)OCC(=N)NNC(=O)C(=O)N 3F-025 c1ccc(cc1)C(=O)NNC(=N)Cn2cncn2 3F-026 c1cc(cc(c1)NC(=O)C(=O)NNC(=N)Cn2cncn2)C(F)(F)F 3F-027 c1cc(c(cc1Cl)Cl)C(=O)NNC(=N)Cn2cncn2 3F-028 c1cc(cc(c1)NC(=O)c2[nH]nc(n2)Cn3cncn3)C(F)(F)F 3F-029 c1cc(c(cc1Cl)Cl)c2[nH]nc(n2)Cn3cncn3 3F-030 c1ccc(cc1)c2nnc(o2)Cn3cncn3 3F-032 CCOC(=O)C(=O)Nc1ccc(cc1)OC(F)(F)F 3F-034 c1cc(ccc1NC(=O)C(=O)NN)OC(F)(F)F 3F-035 c1ncn(n1)CC(=N)NNC(=O)C(=O)N 3F-036 c1ncn(n1)Cc2nc([nH]n2)C(=O)N 3F-037 c1cc(ccc1NC(=O)C(=O)NNC(=N)Cn2cncn2)OC(F)(F)F 3F-038 COc1ccc(cc1)NC(=O)C(=O)NNC(=N)Cn2cncn2 3F-039 c1cc(ccc1NC(=O)c2[nH]nc(n2)Cn3cncn3)OC(F)(F)F 3F-040 c1ccc(cc1)NNC(=N)COc2ncn(n2)c3ccccc3 3F-041 c1ccc(cc1)C(=O)NNC(=N)COc2ncn(n2)c3ccccc3 3F-042 COC(=O)c1c(c(c(=O)n(n1)c2ccccc2)N=Nc3cccc(c3)C(F)(F)F)O 3F-043 c1ccc(cc1)n2c(=O)cc(c(n2)c3nc[nH]n3)Oc4ccccc4 3F-045 c1ccc(cc1)n2cnc(n2)OCC(=N)NS(=O)(=O)c3ccccc3 3F-046 c1ccc(cc1)c2[nH]nc(n2)COc3ncn(n3)c4ccccc4 3F-047 c1cc(cnc1)c2nc([nH]n2)C/C=N/OCc3ccc(cc3Cl)Cl 3F-048 CCOC(=O)C(=O)Nc1ccccc1 3F-049 c1cc(c(cc1Cl)Cl)OCc2nc([nH]n2)C(=O)N 3F-050 COC(=O)c1c(c(c(=O)n(n1)c2ccccc2)N=Nc3cccc(c3)C(F)(F)F)Cl 3F-051 c1ccc(cc1)n2cnc(n2)OCC(=N)NS(=O)(=O)c3ccc(cc3Cl)Cl 3F-052 c1ccc(cc1)NC(=O)C(=O)NN 3F-053 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)Oc3cccc(c3)C(F)(F)F 3F-054 COC(=O)CSc1cc(=O)n(nc1C(=O)OC)c2ccc(cc2)Cl 3F-055 COC(=O)c1c(c2c(s1)cc(=O)n(n2)c3ccc(cc3)Cl)O 3F-056 Cn1cc(cc1/C=N\OC)C(=O)c2ccc(cc2Cl)Cl 3F-059 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)Cl 3F-060 c1cc([nH]c1)C(=O)NN 3F-061 c1cc(ccc1Nc2cc(=O)n(nc2C#N)c3ccc(cc3)Cl)Cl 3F-063 Cc1ccc(cc1)Oc2cc(=O)n(nc2C(=O)OC)c3ccc(cc3)Cl 3F-065 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN 3F-066 Cc1c(c(no1)c2ccccc2)C(=O)NN 3F-067 c1cc([nH]c1)C(=O)NNC(=N)COc2ccc(cc2Cl)Cl 3F-068 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)Oc3cccc(c3)Cl 3F-069 c1ccc(cc1)NC(=O)C(=O)NNC(=N)Cn2cncn2 3F-070 c1ccc(cc1)NC(=O)c2[nH]nc(n2)Cn3cncn3 3F-072 c1cc(c(cc1Cl)Cl)CO/N=C/CC(=O)NNC(=N)Cn2cncn2 3F-073 CC1(OC(=O)C(=C(Cn2cncn2)N)C(=O)O1)C 3F-074 c1cc(c(cc1Cl)Cl)CO/N=C/Cc2[nH]nc(n2)Cn3cncn3 3F-075 c1cc(ccc1c2ccnc(n2)Cn3cncn3)Cl 3F-076 c1ccc(cc1)S(=O)(=O)NNC(=N)Cn2cncn2 3F-077 CN(C)/C=C/C(=O)/C(=C/c1ccccc1)/Oc2ccc(cc2)C#N 3F-078 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)Sc3ccccn3 3F-080 c1ccc(cc1)Oc2cc(=O)n(nc2C#N)c3ccc(cc3Cl)Cl 3F-081 c1ccc(cc1)n2cnc(n2)OCC(=N)NNc3ccc(cc3Cl)Cl 3F-082 c1ccc(c(c1)C(C#N)c2ccc(nn2)Cl)Br 3F-083 Cc1c(c(no1)c2ccccc2)C(=O)NNC(=N)COc3ccc(cc3)Cl 3F-084 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=N)COc3ccc(cc3)Cl 3F-085 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNC(=N)COc3ccc(cc3)Cl 3F-086 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nnc(o3)COc4ccc(cc4)Cl 3F-087 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)NN 3F-088 c1ccc2c(c1)ncc(n2)NCCO 3F-089 c1ccnc(c1)SC/C(=N/Nc2cccc(n2)F)/N 3F-090 c1cc(ccc1n2c(=O)cc3c(n2)c(n[nH]3)N)Cl 3F-091 Cc1c(c(no1)c2ccccc2Cl)c3nnc(o3)COc4ccc(cc4)Cl 3F-092 Cc1c(c(no1)c2ccccc2)c3[nH]c(nn3)COc4ccc(cc4)Cl 3F-093 c1ccnc(c1)SC/C(=N/NC(=O)c2ccncc2)/N 3F-094 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)Oc3ccccc3Cl 3F-095 c1ccnc(c1)SCc2nc([nH]n2)c3ccncc3 3F-096 c1ccc(c(c1)Cc2ccc(nn2)O)Br 3F-098 Cc1ccc(cc1)Sc2cc(=O)n(nc2C(=O)OC)c3ccc(cc3)Cl 3F-099 COC(=O)/C=C(/Cn1cncn1)\N 3F-100 c1ccc(c(c1)C(c2ccc(nn2)O)C(=O)N)Br 3F-101 COc1ccc(cc1)n2c(=O)cc3c(n2)c(n[nH]3)O 3F-104 CC(C)C(=O)O/N=C/c1c(nn(c1Sc2ccc(cc2)Cl)C)C(F)(F)F 3F-301S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2)Sc3ccc(cc3)Cl 3F-302S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Sc3ccc(cc3)Cl 3F-303S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2cccc(c2)C(F)(F)F)Sc3ccc(cc3)Cl 3F-304S c1cc(c(nc1)NN)[N+](=O)[O-] 3F-306S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2cccc(c2)C(F)(F)F 3F-307S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccc(cc2)OC(F)(F)F 3F-308S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccc(cc2F)F 3F-309S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccc(cc2)OC 3F-310S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccc(cc2)F 3F-311S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F 3F-312S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccc(c(c2)Cl)Cl 3F-313S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)SCc3cccc(c3)C(F)(F)F 3F-314S Cc1ccc(cc1C)NC(=O)c2c(nn(c2SCc3cccc(c3)C(F)(F)F)C)C(F)(F)F 3F-315S c1cc(ccc1NC(=O)c2ccc(nc2)n3ccnc3)OC(F)(F)F 3F-316S c1cc(c(cc1F)F)NC(=O)c2ccc(nc2)n3ccnc3 3F-318S Cc1cccc(c1)NC(=O)c2ccc(nc2)n3ccnc3 3F-320S Cc1c(cccc1Cl)NC(=O)c2ccc(nc2)n3ccnc3 3F-321S Cc1ccc(cc1)Sc2c(c(nn2C)C(F)(F)F)C(=O)Nc3ccc(cc3F)F 3F-322S Cc1ccc(cc1)Sc2c(c(nn2C)C(F)(F)F)C(=O)Nc3cccc(c3)C(F)(F)F 3F-323S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(cc2Cl)Cl)Sc3ccc(cc3)Cl 3F-324S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC)Cl 3F-325S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(cc2Cl)Cl)Sc3ccccc3 3F-326S Cn1c(c(c(n1)C(F)(F)F)/C=N/O)SCc2ccccc2Cl 3F-327S CN(C)S(=O)(=O)Oc1cccc(c1)C(=O)Nc2ccc(cc2)[N+](=O)[O-] 3F-328S CN(C)S(=O)(=O)Oc1ccc(cc1Cl)C(=O)OC 3F-330S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2cccc(c2)C(F)(F)F)SCc3ccc(cc3)Cl 3F-331S Cc1ccc(cc1C)NC(=O)c2c(nn(c2SCc3ccc(cc3)Cl)C)C(F)(F)F 3F-332S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC)Sc3ccc(cc3)Cl 3F-333S c1cc(ccc1NC(=O)c2ccc(nc2)n3ccnc3)F 3F-334S Cn1c(c(c(n1)C(F)(F)F)C=O)SCc2ccc(cc2)Cl 3F-335S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)CCl)Sc2ccc(cc2)Cl 3F-336S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)CCl)SCc2ccccc2Cl 3F-337S Cn1c(c(c(n1)C(F)(F)F)/C=N/O)Sc2ccccc2 3F-338S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2)Sc3ccccc3 3F-339S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC)Sc3ccccc3 3F-340S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC)SCc3ccccc3 3F-341S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC)SCc3ccccc3Cl 3F-342S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)OC)Sc3ccccc3Cl 3F-343S CN(C)S(=O)(=O)Oc1c(cc(cc1Cl)Cl)C(=O)OC 3F-345S CN(C)S(=O)(=O)Oc1ccc(cc1Cl)C(=O)Nc2ccc(cc2)Cl 3F-346S CN(C)S(=O)(=O)Oc1ccc(cc1Cl)C(=O)Nc2cccc(c2)Cl 3F-347S CN(C)S(=O)(=O)Oc1ccc(cc1Cl)C(=O)Nc2ccccc2Cl 3F-348S CN(C)S(=O)(=O)Oc1ccc(cc1Cl)C(=O)Nc2ccc(cc2)OC(F)(F)F 3F-349S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccc(cc2)OC)SCc3ccccc3Cl 3F-351S c1cc(c2ncnn2c1)[N+](=O)[O-] 3F-355S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)CCl)Sc2ccccc2 3F-356S CN(C)S(=O)(=O)Oc1cc(ccc1C(=O)OC)Cl 3F-364S CN(C)S(=O)(=O)Oc1ccc(cc1C(=O)OC)Cl 3F-365S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)C(Cl)Cl)Sc2ccc(cc2)Cl 3F-366S Cn1c(c(c(n1)C(F)(F)F)C(=O)OC)Cl 3F-368S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccc(cc2Cl)Cl)Sc3ccc(cc3)Cl 3F-369S Cc1ccc(cc1)C(=O)O/N=C/c2c(nn(c2Sc3ccc(cc3)Cl)C)C(F)(F)F 3F-370S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(c(c2)Cl)Cl)Sc3ccc(cc3)Cl 3F-371S CN(C)S(=O)(=O)Oc1cc(ccc1C(=O)Nc2ccccc2Cl)Cl 3F-372S CN(C)S(=O)(=O)Oc1cc(ccc1C(=O)Nc2ccc(cc2F)F)Cl 3F-373S CN(C)S(=O)(=O)Oc1cc(ccc1C(=O)Nc2cccc(c2)C(F)(F)F)Cl 3F-374S c1cc(c2ncnn2c1)N 3F-375S CN(C)S(=O)(=O)Oc1ccc(cc1C(=O)Nc2cccc(c2)C(F)(F)F)Cl 3F-376S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC)Sc2ccc(cc2)Cl 3F-377S CN(C)S(=O)(=O)Oc1ccc(cc1C(=O)Nc2ccccc2Cl)Cl 3F-378S CN(C)S(=O)(=O)Oc1ccc(cc1C(=O)Nc2ccc(cc2F)F)Cl 3F-379S Cn1c(c(c(n1)C(F)(F)F)/C=N/O)SCc2ccc(cc2)Cl 3F-381S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2)SCc3ccc(cc3)Cl 3F-382S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2Cl)SCc3ccc(cc3)Cl 3F-383S Cn1c(c(c(n1)C(F)(F)F)C=O)Sc2ccccc2C(=O)OC 3F-384S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)CCl)SCc2ccc(cc2)Cl 3F-385S CN(C)S(=O)(=O)Oc1cc(ccc1C(=O)Nc2ccc(cc2)Cl)Cl 3F-387S CN(C)S(=O)(=O)Oc1cc(ccc1C(=O)Nc2ccc(c(c2)Cl)Cl)Cl 3F-388S CN(C)S(=O)(=O)Oc1cc(ccc1C(=O)Nc2ccc(cc2)[N+](=O)[O-])Cl 3F-390S c1ccc(cc1)C(=O)Nc2cccn3c2ncn3 3F-391S COc1ccc(cc1)C(=O)Nc2cccn3c2ncn3 3F-392S c1cc(c2ncnn2c1)NC(=O)c3ccc(cc3Cl)Cl 3F-393S c1cc(c2ncnn2c1)NC(=O)c3ccc(cc3)Cl 3F-394S c1ccc(c(c1)C(=O)Nc2cccn3c2ncn3)Cl 3F-395S CC(C)(C)C(=O)Nc1cccn2c1ncn2 3F-396S Cc1ccc(cc1)c2nc(on2)c3c(nn(c3Cl)C)C(F)(F)F 3F-397S CC(C)(C)c1ccc(cc1)CSc2c(c(nn2C)C(F)(F)F)C=O 3F-398S c1ccc2c(c1)C3(C(=O)N2)N(C(=O)CS3)c4ccc(c(c4)Cl)Cl 3F-399S c1ccc(c(c1)S(=O)(=O)Nc2cccn3c2ncn3)Cl 3F-400S CC(C)(C)c1ccc(cc1)CSc2c(c(nn2C)C(F)(F)F)/C=N/O 3F-402S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2)SCc3ccccc3Cl 3F-403S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2Cl)SCc3ccccc3Cl 3F-404S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC)Sc2ccccc2C(=O)OC 3F-405S c1ccc(cc1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5ccc(c(c5)Cl)Cl 3F-406S c1ccc2c(c1)C3(C(=O)N2Cc4ccc(cc4Cl)Cl)N(C(=O)CS3)c5ccc(c(c5)Cl)Cl 3F-407S c1ccc(cc1)N2C(=O)CSC23c4ccccc4NC3=O 3F-408S c1ccc(c(c1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5ccc(c(c5)Cl)Cl)Cl 3F-409S c1ccc2c(c1)C3(C(=O)N2Cc4cccc(c4)Cl)N(C(=O)CS3)c5ccc(c(c5)Cl)Cl 3F-410S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)C2CC2)SCc3ccccc3Cl 3F-411S c1cc(ccc1C(=O)CN)Cl.Cl 3F-900 CCOC(=O)c1c(c[nH]c1N)c2ccc(cc2)Cl 3F-903 CCOC(=O)c1c(cn2c1nc(cc2C)C)c3ccc(cc3)Cl 3F-904 Cc1c(c2c3ccccc3oc(=O)c2c(n1)C)C#N 3F-906 COc1ccc(cc1)N2CCN(CC2)C/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/c4ccccc4 3F-907 CCOC(=O)c1cc2c(ccn(c2=O)CCOC(=O)c3cccc(c3)C(F)(F)F)nc1C 3F-908 COc1ccc(cc1)N2CCN(CC2)C/C(=N\OC(=O)c3ccc(cc3)Cl)/c4ccccc4 3F-909 c1ccc(cc1)C(=O)NCC(=O)NOC(=O)c2ccccc2 3F-910 C/[N+](=C/c1ccccc1)/[O-] 3F-912 CCOC(=O)/C=C(\N)/N1CCN(CC1)c2c(cccc2C)C 3F-913 CCOC(=O)/C=C(\N)/N1CCN(CC1)c2cccc(c2)Cl 3F-914 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3c(cccc3C)C)c4ccc(cc4)C 3F-915 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3cccc(c3)Cl)c4ccc(cc4)F 3F-916 CN1C(CC(O1)CO)c2ccccc2 3F-918 CCOC(=O)c1cc([nH]c1N2CCOCC2)c3ccc(c(c3)Cl)Cl 3F-922 CCOC(=O)c1cc([nH]c1N2CCCCC2)c3ccc(cc3)[N+](=O)[O-] 3F-923 C/[N+](=C/c1ccc(cc1)OC)/[O-] 3F-926 CCOC(=O)/C=C(\N)/N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 3F-928 CCOC(=O)/C=C(\N)/N1CCN(CC1)c2ccc(cc2)Cl 3F-929 CCOC(=O)/C(=C/C(=C(/N)\N1CCN(CC1)c2c(cccc2C)C)/C(=O)OCC)/C#N 3F-932 CCOC(=O)/C(=C/C(=C(/N)\N1CCN(CC1)c2ccc(cc2)Cl)/C(=O)OCC)/C#N 3F-933 CCOC(=O)/C(=C/C(=C(/N)\N1CCN(CC1)c2ccccn2)/C(=O)OCC)/C#N 3F-934 c1ccc(cc1)OCCON2C(=O)c3ccccc3C2=O 3F-935 c1ccc(cc1)OCCON.Cl 3F-936 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])c4ccc(c(c4)Cl)Cl 3F-937 c1ccc2c(c1)C(=O)N(C2=O)OCc3ccc(cc3)F 3F-939 c1cc(ccc1CON)F.Cl 3F-940 c1ccc(cc1)OCCONC(=O)c2ccc(cc2Cl)Cl 3F-941 c1cc(cc(c1)OCCBr)C(F)(F)F 3F-943 c1cc(c(cc1Cl)Cl)CONC(=O)CCCCl 3F-946 c1cc(c(cc1Cl)Cl)OCCBr 3F-947 Cc1c(c(no1)c2ccccc2Cl)C(=O)NOCCOc3ccccc3 3F-948 CC1(OC(=O)C(=C(CC#N)N)C(=O)O1)C 3F-949 CC1(OC(=O)C(=C(Cc2ccc(cc2)Cl)N)C(=O)O1)C 3F-951 Cc1cc(n2cc(c(c2n1)C(=O)O)c3ccc(cc3)Cl)C 3F-952 C(C(=NNC(=O)N)CCl)Cl 3F-953 CN1C(CC(O1)COC(=O)c2ccc(cc2)Cl)c3ccccc3 3F-954 Cc1cc(n2cc(c(c2n1)C(=O)NC)c3ccc(cc3)Cl)C 3F-955 CN1C(CC(O1)COC(=O)Nc2ccccc2)c3ccccc3 3F-956 c1cc(ccc1SCc2c(snn2)Cl)Cl 3F-958 COC(=O)/C=C(\Cc1ccc(cc1)Cl)/N 3F-959 COc1ccc(cc1)N2CCN(CC2)Cc3c(snn3)Cl 3F-960 c1ccc(cc1)NCc2c(snn2)Cl 3F-961 C1CCN(CC1)Cc2c(snn2)Cl 3F-963 c1ccc(cc1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-002 c1cc(ccc1Sc2cc(cnc2C(=O)N)C(F)(F)F)Cl 3G-003 c1cc(ccc1S(=O)(=O)c2cc(cnc2C#N)C(F)(F)F)Cl 3G-004 CCOC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)N(C)C 3G-006 CN(C)C(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)N(C)C 3G-007 c1cc(ccc1S(=O)(=O)c2cc(cnc2C(=O)N)C(F)(F)F)Cl 3G-010 c1cc(ccc1CSc2cc(cnc2C(=O)N)C(F)(F)F)Cl 3G-011 c1cc(ccc1CS(=O)(=O)c2cc(cnc2C(=O)N)C(F)(F)F)Cl 3G-012 c1ccc(cc1)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-013 CN(C)/C=N/C(=O)C(c1ccccc1)c2c(cc(cn2)C(F)(F)F)Cl 3G-014 CN(C)/C=N/C(=O)c1c(cc(cn1)C(F)(F)F)Sc2ccc(cc2)Cl 3G-015 c1cc(ncc1C(F)(F)F)S(=O)(=O)c2cc(cnc2C#N)C(F)(F)F 3G-016 c1ccc(cc1)C(=O)c2cc(no2)c3c(cc(cn3)C(F)(F)F)Cl 3G-021 CO/N=C/NC(=O)C(c1ccccc1)c2c(cc(cn2)C(F)(F)F)Cl 3G-022 c1cc(c(c(c1)Cl)CO/N=C/C(c2ccc(cc2)Cl)S(=O)(=O)c3cc(cnc3C#N)C(F)(F)F)Cl 3G-023 c1ccc(cc1)C(c2c(cc(cn2)C(F)(F)F)Cl)c3nc[nH]n3 3G-024 CN(C)/C=N/C(=O)c1c(cc(cn1)C(F)(F)F)S(=O)(=O)c2ccc(cc2)Cl 3G-025 c1ccc(cc1)/C(=N\O)/c2cc(no2)c3c(cc(cn3)C(F)(F)F)Cl 3G-026 c1c(cnc(c1Cl)c2c(noc2O)O)C(F)(F)F 3G-027 c1cc(c(c(c1)Cl)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-029 c1cc(ccc1C(C#N)c2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-030 c1cc(ncc1C(F)(F)F)S(=O)(=O)c2cc(cnc2C(=O)N)C(F)(F)F 3G-031 COc1ccc(cc1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-032 c1cc(ccc1C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N)Cl 3G-033 CN(C)c1ccc(cc1)/C=C/C=[N+]\2/C(=C(C(=O)O2)c3c(cc(cn3)C(F)(F)F)Cl)[O-] 3G-034 CN(C)/C=N/C(=O)C(c1ccc(cc1)Cl)c2c(cc(cn2)C(F)(F)F)Cl 3G-035 c1c(cnc(c1Cl)CC(=O)NO)C(F)(F)F 3G-036 c1ccc(cc1)/C(=N\OCc2c(cccc2Cl)Cl)/c3cc(no3)c4c(cc(cn4)C(F)(F)F)Cl 3G-037 c1cc(ccc1C(C#N)c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 3G-038 CO/N=C(\c1ccccc1)/c2cc(no2)c3c(cc(cn3)C(F)(F)F)Cl 3G-039 c1c(cnc(c1Cl)c2nc(on2)NC(=N)N)C(F)(F)F 3G-040 COc1ccc(cc1OC)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-041 CN(C)/C=C(\c1ccc(cc1)Cl)/S(=O)(=O)c2cc(cnc2C(=O)/N=C/N(C)C)C(F)(F)F 3G-043 c1cc(cc(c1)C(F)(F)F)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-045 c1ccc(cc1)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N/C=N/O 3G-046 c1cscc1C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-047 c1cc(c(c(c1)Cl)CO/N=C/NC(=O)C(c2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl)Cl 3G-048 c1cc(ccc1C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N/C=N/O)Cl 3G-049 c1cc(cc(c1)C(F)(F)F)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-051 c1ccc(c(c1)NN/C=N/C(=O)C(c2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl)Cl 3G-052 c1ccnc(c1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-053 Cn1cccc1C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-055 c1cc(ccc1N)Sc2cc(cnc2C#N)C(F)(F)F 3G-057 c1ccnc(c1)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-058 CO/N=C/NC(=O)c1c(cc(cn1)C(F)(F)F)SCc2ccc(cc2)Cl 3G-059 CN(C)/C=N/C(=O)C(c1ccccn1)c2c(cc(cn2)C(F)(F)F)Cl 3G-060 COc1ccc(cc1OC)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-064 c1c(cnc2c1nc(nc2N)N)C(F)(F)F 3G-065 c1ccnc(c1)C(c2c(cc(cn2)C(F)(F)F)Cl)c3nc[nH]n3 3G-068 COc1ccc(cc1OC)C(c2c(cc(cn2)C(F)(F)F)Cl)c3nc[nH]n3 3G-070 c1cc(ccc1C(c2c(cc(cn2)C(F)(F)F)Cl)c3nc[nH]n3)Cl 3G-071 CC(c1cc(no1)c2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-074 c1cc(sc1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-077 CC(=O)OC(c1ccccc1)c2cc(no2)c3c(cc(cn3)C(F)(F)F)Cl 3G-079 C/C(=C\N(C)C)/C(=O)c1ccc2c(c1)ccc(c2Br)OC 3G-081 c1cc(c(c(c1)Cl)CO/N=C/C(=C\NNc2c(cc(cn2)C(F)(F)F)Cl)/S(=O)(=O)c3ccc(cc3)Cl)Cl 3G-083 CNC(=S)NNC(=O)C/C=N/OCc1ccc(cc1Cl)Cl 3G-084 c1c(cnc(c1Cl)/C(=N/OC(=O)CCCC(=O)O)/N)C(F)(F)F 3G-085 c1cc(sc1)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-086 Cc1cccc(c1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-087 c1cc(c(cc1Cl)Cl)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-088 Cc1cccc(c1)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-089 c1cc(c(c(c1)Cl)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N)Cl 3G-090 CN(C)/C=N/C(=O)C(c1c(cccc1Cl)Cl)c2c(cc(cn2)C(F)(F)F)Cl 3G-091 c1cc(cc(c1)Cl)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3G-092 c1cc(cc(c1)Cl)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-093 c1cc(c(cc1Cl)Cl)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 3G-095 Cc1c(sc(n1)c2ccc(cc2)[N+](=O)[O-])C(=O)O 3G-301S c1cc(cc(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3)C(F)(F)F 3G-303S C=CCOC(=O)c1ccc(nc1)n2cncn2 3G-305S Cc1c(sc(n1)c2ccc(c(c2)OC)OC)C(=O)O 3G-308S C#CCOC(=O)c1ccc(nc1)n2cncn2 3G-310S COC(=O)c1c2ccc(cc2on1)NC(=O)c3cccc(c3)C(F)(F)F 3G-311S c1cc(ccc1c2nc(cs2)c3ccc(cc3)Cl)C(=O)O 3G-313S c1cc(ccc1c2nc(cs2)c3ccc(c(c3)Cl)Cl)C(=O)O 3G-314S c1cc(ccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3)Cl 3G-316S c1cc(c(cc1C(=O)Nc2ccc(cc2F)F)[N+](=O)[O-])n3cncn3 3G-317S CC(C)NC(=O)c1c2ccc(cc2on1)[N+](=O)[O-] 3G-318S Cc1c(sc(n1)c2ccc(c(c2)OC)OC)C(=O)Nc3ccc(cc3)Cl 3G-319S Cc1c(sc(n1)c2ccc(c(c2)OC)OC)C(=O)Nc3ccc(c(c3)Cl)Cl 3G-320S Cc1c(sc(n1)c2ccc(c(c2)OC)OC)C(=O)Nc3cccc(c3)C(F)(F)F 3G-321S Cc1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-323S COc1ccc(cc1OC)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-324S COc1ccccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-325S c1ccc(cc1)c2nc(cs2)c3ccc(cc3)C(=O)O 3G-326S c1cc(cc(c1)S(=O)(=O)c2cnns2)C(F)(F)F 3G-329S c1cc(c(cc1Sc2cnns2)Cl)Cl 3G-330S CCOC(=O)/C(=N\NC(=O)N)/CSc1ccc(cc1)Cl 3G-332S CCOC(=O)/C(=N\NC(=O)N)/CS(=O)(=O)c1ccc(cc1)Cl 3G-334S COc1cccc(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-335S COc1ccc(cc1OC)c2nc(cs2)C(=O)Nc3ccc(cc3)F 3G-336S COc1ccc(cc1OC)c2nc(cs2)C(=O)Nc3ccc(cc3F)F 3G-337S Cc1c(cccc1Cl)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-338S COc1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-342S COc1ccc(cc1Cl)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-343S CC(C)NC(=O)c1ccc(c(c1)[N+](=O)[O-])n2cncn2 3G-344S c1cc(ccc1c2nc(cs2)c3ccc(cc3)Cl)O 3G-345S c1cc(cc(c1)NC(=O)c2ccc(cc2)c3nc(cs3)c4ccc(cc4)Cl)C(F)(F)F 3G-346S c1cc(ccc1c2nc(cs2)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)OC(F)(F)F 3G-347S Cc1ccccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cncn3 3G-348S COc1ccccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-349S c1cc(cc(c1)Cl)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-350S c1ccc(cc1)COC(=O)c2ccc(nc2)n3cncn3 3G-351S COC(=O)c1ccc(c(c1)[N+](=O)[O-])n2ccnc2 3G-355S c1ccc(cc1)NC(=O)c2ccc(cc2)c3nc(cs3)c4ccc(cc4)Cl 3G-356S CN(C)CCCNC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)Cl 3G-357S Cc1c(cccc1Cl)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-358S c1ccc(c(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3)Cl 3G-359S COc1ccc(cc1OC)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-360S c1cc(cnc1)C(=O)Nc2ccc(cc2)Cl 3G-363S c1ccc(cc1)OC(=O)c2ccc(nc2)n3cncn3 3G-364S C/N=C(\c1cccnc1)/Nc2ccc(cc2)Cl 3G-365S c1cc(ccc1c2nc(cs2)C(=O)O)[N+](=O)[O-] 3G-366S c1ccc(c(c1)NC(=O)c2ccc(cc2)c3nc(cs3)c4ccc(c(c4)Cl)Cl)Cl 3G-368S c1cc(cc(c1)Cl)NC(=O)c2ccc(cc2)c3nc(cs3)c4ccc(c(c4)Cl)Cl 3G-369S Cc1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-371S Cc1ccccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-372S Cc1cccc(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-373S Cc1c(snn1)Sc2ccccn2 3G-376S c1cc(ccc1c2nc(cs2)c3ccc(c(c3)Cl)Cl)C(=O)Nc4ccc(cc4)Cl 3G-377S CNC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(c(c3)Cl)Cl 3G-378S C=CCNC(=O)c1ccc(cc1)c2nc(cs2)c3ccc(c(c3)Cl)Cl 3G-379S COc1ccc(cc1Cl)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-380S Cc1ccc(cc1C)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccn3 3G-382S CC(C)/N=C(\c1cccnc1)/Nc2ccc(cc2)Cl 3G-383S CCOC(=O)c1csc(n1)c2cccs2 3G-384S Cc1[nH]nc(n1)Sc2ccc(cn2)C(=O)Oc3ccccc3 3G-386S c1cc(sc1)c2nc(cs2)C(=O)O 3G-388S c1ccc(cc1)NC(=O)c2csc(n2)c3ccc(cc3)[N+](=O)[O-] 3G-389S c1cc(ccc1c2nc(cs2)C(=O)Nc3ccc(cc3)F)[N+](=O)[O-] 3G-390S c1cc(ccc1c2nc(cs2)C(=O)Nc3ccc(cc3F)F)[N+](=O)[O-] 3G-391S CCOC(=O)CSc1c(nns1)C 3G-393S Cc1c(snn1)Sc2ccccc2Cl 3G-395S Cc1c(cccc1Cl)NC(=O)c2ccc(c(c2)[N+](=O)[O-])n3ccnc3 3G-396S CCCC/N=C(\c1cccnc1)/Nc2ccc(cc2)Cl 3G-399S CCOCCOC(=O)c1ccc(nc1)Sc2nc([nH]n2)C 3G-401S Cc1c(snn1)SCC(=O)O 3G-403S Cc1c(snn1)S(=O)c2ccccn2 3G-404S Cc1c(snn1)S(=O)Cc2ccc(cc2)C(C)(C)C 3G-406S COC(=O)c1c2ccc(cc2on1)NC(=O)c3ccccc3Cl 3G-407S c1cc(sc1)c2nc(cs2)C(=O)Nc3ccc(cc3)F 3G-408S c1cc(sc1)c2nc(cs2)C(=O)Nc3ccc(cc3F)F 3G-409S c1cc(cc(c1)NC(=O)c2csc(n2)c3cccs3)C(F)(F)F 3G-410S CCC/N=C(\c1cccnc1)/Nc2ccc(cc2)Cl 3G-412S CCOC(=O)c1c(nc(s1)c2cccs2)C 3G-414S Cc1c(snn1)S(=O)(=O)c2ccccc2Cl 3G-416S CCOC(=O)C(C)Sc1c(nns1)C 3G-417S CC/N=C(\c1cccnc1)/Nc2ccc(cc2)Cl 3G-418S CNC(=O)c1csc(n1)c2cccs2 3G-419S Cc1c(snn1)SC(C)C(=O)O 3G-420S Cc1c(sc(n1)c2cccs2)C(=O)O 3G-423S COc1ccc(cc1)COC(=O)c2ccc(nc2)n3cncn3 3G-424S CCOC(=O)C(C)S(=O)(=O)c1c(nns1)C 3G-426S c1ccc(cc1)c2nc(c(s2)C(=O)Nc3ccc(cc3)F)C(F)(F)F 3G-428S c1ccc(cc1)c2nc(c(s2)C(=O)Nc3ccc(cc3F)F)C(F)(F)F 3G-429S c1ccc(cc1)c2nc(c(s2)C(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F 3G-430S c1ccc(cc1)C(=O)Nc2ccc(cc2)Cl 3G-432S Cc1c(sc(n1)c2cccs2)C(=O)Nc3ccc(c(c3)Cl)Cl 3G-434S Cc1c(sc(n1)c2cccs2)C(=O)Nc3ccc(cc3)Cl 3G-435S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)NCc2ccc(cc2)Cl 3G-436S c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)Cl 3G-439S c1cc(ccc1CNC(=O)c2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl 3G-440S CN(c1ccc(cc1)Cl)C(=O)c2ccc(cc2Cl)S(=O)(=O)C 3G-441S Cc1c(snn1)Sc2ccc3ccccc3c2 3G-443S Cc1c(snn1)SC(C)C 3G-444S Cc1c(snn1)SC(C)(C)C 3G-445S Cc1c(snn1)SC2CCCCC2 3G-446S Cc1c(snn1)S(=O)(=O)c2ccc3ccccc3c2 3G-448S Cc1c(snn1)S(=O)c2ccc3ccccc3c2 3G-451S Cc1c(snn1)S(=O)(=O)C2CCCCC2 3G-452S Cc1c(snn1)S(=O)(=O)C(C)C 3G-453S Cc1c(snn1)S(=O)(=O)C(C)(C)C 3G-454S CCOCCOC(=O)c1ccc(nc1)n2cnc(n2)C 3G-457S c1c(cnc(c1Cl)N2CCC3(CC2)C(=O)NC(=O)N3)C(F)(F)F 3G-900 Cc1c(c(no1)C(=O)NN)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 3G-901 c1ccc(c(c1)C=O)OCCBr 3G-902 Cc1c(c(no1)C(=O)NNC(=O)Nc2ccc(cc2)Cl)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 3G-903 Cc1c(c(no1)C(=O)NNC(=S)NC)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 3G-904 CCOC(=O)c1c(con1)C(=O)c2ccc(cc2)Br 3G-905 C/C(=C\C(=O)Nc1nccs1)/N2CCCC2 3G-906 CCOC(=O)c1c(noc1C(F)(F)F)C(=O)OCC 3G-907 COC(=O)C(=NO)C(=O)OC 3G-908 CCOC(=O)c1c(c(on1)C)C(=O)Nc2nccs2 3G-909 c1ccc(c(c1)C=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3G-910 COC(=O)C1C(C2CCCCN2O1)(C(F)(F)F)O 3G-911 Cc1c(c(no1)C(=O)N2CCN(CC2)C)C(=O)Nc3nccs3 3G-912 Cc1c(c(no1)CO)C(=O)Nc2nccs2 3G-913 Cc1c(c(no1)C(=O)N)C(=O)Nc2nccs2 3G-914 COC(=O)C1(C2C(C(=O)N(C2=O)c3ccccc3)ON1)C(=O)OC 3G-916 C/C(=C/C(=O)N1CCN(CC1)c2ccccc2)/N3CCCC3 3G-917 c1ccc(cc1)C(=O)N2[C@H]3c4c5ccccc5ccc4OC[C@H]3CO2 3G-918 CC(=O)N1[C@H]2c3c4ccccc4ccc3OC[C@H]2CO1 3G-919 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4C(=O)c5cccs5 3G-920 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4C(=O)c5ccc(c(c5)Cl)Cl 3G-921 CCOC(=O)N1[C@H]2c3c4ccccc4ccc3OC[C@H]2CO1 3G-922 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3[C@H]4c5c6ccccc6ccc5OC[C@H]4CO3 3G-923 Cc1c(c(no1)c2ccccc2)C(=O)N3[C@H]4c5c6ccccc6ccc5OC[C@H]4CO3 3G-924 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4S(=O)(=O)c5ccc(cc5)Cl 3G-925 CN(C)/C=N/C(=O)N1[C@H]2c3c4ccccc4ccc3OC[C@H]2CO1 3G-926 Cc1ccc(cc1)CON/C=N/C(=O)N2[C@H]3c4c5ccccc5ccc4OC[C@H]3CO2 3G-927 CON/C=N/C(=O)N1[C@H]2c3c4ccccc4ccc3OC[C@H]2CO1 3G-928 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4C(=O)/N=C/NOCc5ccc(cc5Cl)Cl 3G-929 c1c(cnc(c1Cl)NCCN)C(F)(F)F 3G-930 c1cc(ccc1NC(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-931 c1c(cnc(c1Cl)NC(=O)CCl)C(F)(F)F 3G-932 c1ccc(c(c1)/C=N/OCc2ccc(cc2)Cl)OCCN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 3G-934 c1cc(cc(c1)OCCBr)C=O 3G-935 CCOC(=O)c1cc(c(=O)[nH]c1N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)OCC 3G-936 CCOC(=O)/C(=C\C(=C(/N)\N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)\C(=O)OCC)/C#N 3G-937 c1cc(ccc1C=O)OCCBr 3G-938 CCOC(=O)c1cc(c([nH]c1=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C#N 3G-939 c1c(cnc(c1Cl)NCCn2cc(c(=O)[nH]c2=O)C#N)C(F)(F)F 3G-940 CN(C)c1ccc(cc1)/C=N\CCNc2c(cc(cn2)C(F)(F)F)Cl 3G-941 c1cc(cc(c1)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C=O 3G-942 c1cc(ccc1C=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3G-943 CCOC(=O)/C(=C/C(=C(\N)/N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)/C#N)/C#N 3G-944 c1cc(cc(c1)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)/C=N\Nc4c(cc(cn4)C(F)(F)F)Cl 3G-946 c1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OCCN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 3G-947 c1cc(cc(c1)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)/C=C\C(=O)c4ccc(cc4)Cl 3G-948 c1cc(cc(c1)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)CO 3G-949 c1cc(ccc1c2csc(n2)Nc3c(cc(cn3)C(F)(F)F)Cl)Cl 3G-950 c1cc(ccc1C(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-951 Cc1c(c(no1)c2ccccc2)C(=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl 3G-952 c1cc(ccc1CO)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3G-953 c1ccc(c(c1)S(=O)(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-954 C=CCNC(=S)NCCNc1c(cc(cn1)C(F)(F)F)Cl 3G-955 CC(C)(C)c1csc(n1)Nc2c(cc(cn2)C(F)(F)F)Cl 3G-956 c1c(cnc(c1Cl)NC(=O)CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 3G-959 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl 3G-960 CN1CCN(CC1)CC(=O)Nc2c(cc(cn2)C(F)(F)F)Cl 3G-961 CCOC(=O)NC(=O)/C(=C\NNc1c(cc(cn1)C(F)(F)F)Cl)/C#N 3G-962 c1cc(ccc1COCCO)Cl 3G-963 c1cc(ccc1[N+](=O)[O-])OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3G-964 c1cc(ccc1COCCCl)Cl 3G-965 CN(C)c1ccc(cc1)CN(CCNc2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Cl 3G-966 CN(C)CCN(C)c1c(cc(cn1)C(F)(F)F)Cl 3G-967 c1cc(ccc1COCC[NH+]2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl.[Cl-] 3G-968 Cc1c(cnc(n1)c2ccccc2)C(=O)Nc3c(cc(cn3)C(F)(F)F)Cl 3G-969 CCOC(=O)NC(=O)c1cnn(c1N)c2c(cc(cn2)C(F)(F)F)Cl 3G-970 CN(C)CCCNc1c(cc(cn1)C(F)(F)F)Cl 3G-971 CN(C)CCNc1c(cc(cn1)C(F)(F)F)Cl 3G-972 c1cc(ccc1/C=N\CCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-973 c1c(cnc(c1Cl)NCCNS(=O)(=O)C(F)(F)F)C(F)(F)F 3G-974 COCCCNc1c(cc(cn1)C(F)(F)F)Cl 3G-975 COCCNc1c(cc(cn1)C(F)(F)F)Cl 3G-976 c1cc(ccc1CNCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 3G-978 c1cc(ccc1CN(CCNc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)c3ccc(cc3)Cl)Cl 3G-981 Cc1c(c(no1)c2ccccc2)C(=O)N(CCNc3c(cc(cn3)C(F)(F)F)Cl)Cc4ccc(cc4)Cl 3G-982 COC(CNc1c(cc(cn1)C(F)(F)F)Cl)OC 3G-983 c1cc(ccc1/C=C\C(=O)c2ccncc2)OCCN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 3G-984 CNC(=S)N(CCNc1c(cc(cn1)C(F)(F)F)Cl)Cc2ccc(cc2)Cl 3G-985 CC(=O)N(CCNc1c(cc(cn1)C(F)(F)F)Cl)Cc2ccc(cc2)Cl 3G-986 c1cc(c(cc1Cl)Cl)NC(=O)C(=CNOCc2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3Cl)Cl 3G-987 CCCNCCOc1c(cc(cc1Cl)Cl)Cl.Cl 3G-989 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4C(=O)/N=C/NOCc5cccc(c5)C(F)(F)F 3G-991 CC(=O)/C(=C\Nc1ncccn1)/C(=O)Nc2ncccn2 3G-992 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4C(=O)CN5CCOCC5 3G-993 c1ccc2c(c1)ccc3c2[C@H]4[C@@H](CO3)CON4C(=O)CN5CCCCC5 3G-994 CN(C)/C=N/S(=O)(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 3H-001 c1cc(c(cc1Cl)Cl)S(=O)(=O)n2cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 3H-002 c1ccc(cc1)S(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 3H-003 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 3H-004 c1cc(ccc1CC(=O)c2cc([nH]c2)C#N)Cl 3H-005 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 3H-007 c1cc(cnc1)CNS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 3H-008 c1c(cc(c(c1[N+](=O)[O-])Sc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-])C(F)(F)F 3H-009 c1ccc(c(c1)N)Sc2c(cc(cn2)C(F)(F)F)Cl 3H-010 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NCc3ccc(cc3)Cl 3H-011 c1ccc(c(c1)n2cccc2)Sc3c(cc(cn3)C(F)(F)F)Cl 3H-012 c1ccc(cc1)S(=O)(=O)C(CCC#N)c2c(cc(cn2)C(F)(F)F)Cl 3H-014 c1ccc(cc1)S(=O)(=O)c2cc(ccc2O)Oc3c(cc(cn3)C(F)(F)F)Cl 3H-015 c1ccc(cc1)S(=O)(=O)c2cc(ccc2Oc3c(cc(cn3)C(F)(F)F)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 3H-016 COC(=O)CCC(c1c(cc(cn1)C(F)(F)F)Cl)S(=O)(=O)c2ccccc2 3H-017 c1cc(c(nc1)Sc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 3H-018 CN(C)/C=N/C(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 3H-019 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 3H-020 CC(=O)Nc1ccc(cc1)OS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 3H-021 c1cc(cc(c1)OS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 3H-022 c1ccc(cc1)S(=O)(=O)C(CCC(=O)N)c2c(cc(cn2)C(F)(F)F)Cl 3H-023 c1ccc(c(c1)NC(=O)Nc2ccc(c(c2)Cl)Cl)Sc3c(cc(cn3)C(F)(F)F)Cl 3H-024 c1cc(ccc1CC(=O)c2cc(n(c2)c3c(cc(cn3)C(F)(F)F)Cl)C#N)Cl 3H-025 c1c(cnc(c1Cl)S(=O)(=O)C2=CCS(=O)(=O)C2)C(F)(F)F 3H-026 c1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3c(cc(cc3F)F)F 3H-027 c1cc2c(cc1[N+](=O)[O-])cnn2c3c(cc(cn3)C(F)(F)F)Cl 3H-028 CCC(=O)Oc1cc(ccc1S(=O)(=O)c2ccccc2)Oc3c(cc(cn3)C(F)(F)F)Cl 3H-029 CO/N=C/NC(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 3H-030 CS(=O)(=O)c1ccccc1Oc2c(cc(cn2)C(F)(F)F)Cl 3H-031 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Nc3ccc(c(c3)Cl)Oc4ccc(cn4)C(F)(F)F 3H-033 CCOC(=O)c1cccc(c1)NS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 3H-034 CCOC(=O)C(C)Oc1ccc(cc1S(=O)(=O)c2ccccc2)Oc3c(cc(cn3)C(F)(F)F)Cl 3H-035 Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2)S(=O)(=O)Nc3ccc(c(c3)Cl)Oc4ccc(cn4)C(F)(F)F 3H-036 CCC(=O)Nc1ccccc1Sc2c(cc(cn2)C(F)(F)F)Cl 3H-037 c1ccc(cc1)S(=O)(=O)C(CCC(=O)O)c2c(cc(cn2)C(F)(F)F)Cl 3H-038 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)Nc3ccc(c(c3)Cl)Oc4ccc(cn4)C(F)(F)F 3H-042 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 3H-043 CC(=O)C(=O)Nc1ccccc1 3H-044 c1cc(cnc1)OS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 3H-045 CC1(CC(=CC(=O)C1)Nc2ccccc2[N+](=O)[O-])C 3H-046 c1cc(ccc1C(=O)c2cc([nH]c2)C#N)Cl 3H-047 c1ccc(c(c1)NC(=O)NC2CCCCC2)Sc3c(cc(cn3)C(F)(F)F)Cl 3H-048 CC(=O)C(=O)Nc1ccc(cc1)Cl 3H-049 COC(=O)Nc1cccn1c2c(cc(cn2)C(F)(F)F)Cl 3H-051 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)Sc3c(cc(cn3)C(F)(F)F)Cl 3H-052 CC(C)(CCOO)Cc1c[n+](c2ccccc2n1)[O-] 3H-053 CN(C)/C=C/C(=O)C(=O)Nc1ccc(cc1)Cl 3H-054 CCNC(=O)Nc1ccccc1Sc2c(cc(cn2)C(F)(F)F)Cl 3H-056 C#CCNS(=O)(=O)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 3H-057 c1c(cnc(c1Cl)SCC2CC2(Cl)Cl)C(F)(F)F 3H-060 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)c3nc[nH]n3 3H-061 c1ccc(cc1)S(=O)(=O)C(CCC(=O)Nc2ccc(c(c2)Cl)Oc3ccc(cn3)C(F)(F)F)c4c(cc(cn4)C(F)(F)F)Cl 3H-067 c1ccc(cc1)S(=O)(=O)c2cc(ccc2OC(=O)c3ccc(cc3)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 3H-068 c1ccc(cc1)S(=O)(=O)c2cc(ccc2OS(=O)(=O)c3ccc(cc3)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 3H-069 c1ccc(cc1)S(=O)(=O)c2cc(ccc2OC(=O)Nc3ccc(cc3)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 3H-070 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2cccc(c2)Cl)/[N+](=O)[O-] 3H-071 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccccc2Cl)/[N+](=O)[O-] 3H-072 c1ccc(cc1)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccccc2 3H-073 c1ccc(c(c1)NC(=O)CCl)Sc2c(cc(cn2)C(F)(F)F)Cl 3H-074 c1ccc(cc1)S(=O)(=O)C(CCC(=O)Nc2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl 3H-075 c1ccc(cc1)S(=O)(=O)C(CCC(=O)Nc2cccc(c2)C(F)(F)F)c3c(cc(cn3)C(F)(F)F)Cl 3H-076 c1cc(ccc1C(CC#N)(C#N)c2c(cc(cn2)C(F)(F)F)Cl)Cl 3H-077 c1ccc(cc1)/C=C\c2ccnc(n2)[S-].[K+] 3H-079 c1ccc(cc1)/C=C/c2ccnc(n2)SCc3c(cccc3Cl)Cl 3H-081 c1ccc(cc1)/C=C/c2ccnc(n2)SCc3c(cc(cn3)C(F)(F)F)Cl 3H-082 CS(=O)(=O)Nc1ccccc1Sc2c(cc(cn2)C(F)(F)F)Cl 3H-083 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)N3CCOCC3 3H-084 C1C(C1(Cl)Cl)CSc2nnc(s2)N 3H-085 c1ccc(c(c1)NC2=CC(=O)CCC2)[N+](=O)[O-] 3H-086 c1ccc(cc1)/C=C/c2ccnc(n2)Sc3c(cc(cn3)C(F)(F)F)Cl 3H-087 c1ccc(cc1)/C=C/c2ccnc(n2)SCC#N 3H-088 c1ccc(c(c1)NS(=O)(=O)C(F)(F)F)Sc2c(cc(cn2)C(F)(F)F)Cl 3H-090 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)Cl)Sc3c(cc(cn3)C(F)(F)F)Cl 3H-091 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)Oc3ccc(cc3)Cl 3H-092 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=S)N 3H-095 CN(C)/C=N\C(=S)c1cccn1c2c(cc(cn2)C(F)(F)F)Cl 3H-096 CS/C(=N\S(=O)(=O)c1ccccc1)/NNc2ccccc2 3H-099 CS/C(=N\S(=O)(=O)c1ccccc1)/NNc2c(cc(cn2)C(F)(F)F)Cl 3H-100 c1ccc(cc1)NN/C(=N/S(=O)(=O)c2ccccc2)/NN 3H-101 c1cc(c(cc1Cl)Cl)c2c(snn2)Cl 3H-301S c1cc(ccc1c2c(snn2)Cl)Cl 3H-302S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)NC(C)C 3H-303S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3cc(cc(c3)Cl)Cl 3H-304S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3ccc(c(c3)F)F 3H-305S Cc1nc(nn1c2cc(ccc2Cl)Cl)C(=O)Nc3ccccc3Cl 3H-306S c1ccc(cc1)Sc2c(nns2)c3ccc(cc3Cl)Cl 3H-307S c1cc(ccc1F)Sc2c(nns2)c3ccc(cc3Cl)Cl 3H-308S CCOC(=O)c1nc(n(n1)c2cc(cc(c2)Cl)Cl)C 3H-310S Cc1ccc(cc1)n2c(nc(n2)C(=O)Nc3ccc(cc3)Cl)C 3H-312S c1ccc(cc1)CSc2c(nns2)c3ccc(cc3Cl)Cl 3H-313S c1cc(ccc1c2c(snn2)Sc3ccc(cc3)Br)Cl 3H-314S c1cc(ccc1c2c(snn2)Sc3ccc(cc3)F)Cl 3H-315S c1ccc(c(c1)NC(=O)C(=C(Cl)Cl)Cl)Cl 3H-316S c1ccc(cc1)CS/C(=C(/C(=O)Nc2ccccc2Cl)\Cl)/Cl 3H-319S CCOC(=O)CSc1c(nns1)c2ccccc2 3H-321S CC(C(=O)OC)Sc1c(nns1)c2ccccc2 3H-322S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)O 3H-323S Cc1ccc(cc1)n2c(nc(n2)C(=O)Nc3ccc(cc3)F)C 3H-325S Cc1ccc(cc1)n2c(nc(n2)C(=O)Nc3ccc(cc3F)F)C 3H-326S c1ccc(cc1)Sc2c(nns2)c3ccc(cc3)Cl 3H-327S c1ccc(cc1)CSc2c(nns2)c3ccc(cc3)Cl 3H-328S Cc1ccc(cc1)n2c(nc(n2)C(=O)Nc3cccc(c3)C(F)(F)F)C 3H-329S c1cc(ccc1c2c(snn2)SC3CCCCC3)Cl 3H-330S c1ccc(cc1)S(=O)/C(=C(/C(=O)Nc2ccccc2Cl)\Cl)/Cl 3H-332S CC(C)Sc1c(nns1)c2ccccc2 3H-333S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccc(cc3)F 3H-334S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccc(cc3Cl)Cl 3H-335S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccc(cc3)Cl 3H-336S c1ccc(c(c1)Sc2c(nns2)c3ccc(cc3Cl)Cl)Cl 3H-337S CC(C)(C)Sc1c(nns1)c2ccccc2 3H-339S CN(c1ccccc1)C(=O)C(=C(Cl)Cl)Cl 3H-340S c1ccc(cc1)c2c(snn2)Sc3ccccc3 3H-341S c1ccc(cc1)CSc2c(nns2)c3ccccc3 3H-342S CC(C)(C)c1ccc(cc1)CSc2c(nns2)c3ccccc3 3H-343S c1ccc(cc1)c2c(snn2)Sc3ccccn3 3H-344S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)NC 3H-346S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)N(C)C 3H-347S CCCNC(=O)c1nc(n(n1)c2cc(cc(c2)Cl)Cl)C 3H-348S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 3H-349S c1ccc(cc1)S(=O)(=O)/C(=C(/C(=O)Nc2ccccc2Cl)\Cl)/Cl 3H-350S c1cc(ccc1c2c(snn2)Cl)F 3H-353S c1cc(ccc1c2c(snn2)Sc3ccc(cc3)Cl)Cl 3H-354S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccc(cc3F)F 3H-355S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccccc3N4CCOCC4 3H-356S c1cc(ccc1c2c(snn2)Sc3ccc(cc3)F)F 3H-358S c1ccc(cc1)Sc2c(nns2)c3ccc(cc3)F 3H-359S Cc1ccc(cc1)Sc2c(nns2)c3ccc(cc3)Cl 3H-360S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccc(cc3)OC 3H-361S Cc1ccc(cc1)NC(=O)c2nc(n(n2)c3cc(cc(c3)Cl)Cl)C 3H-362S c1cc(ccc1CSc2c(nns2)c3ccc(cc3)F)Cl 3H-363S c1ccc(cc1)CSc2c(nns2)c3ccc(cc3)F 3H-364S CC(C)S(=O)(=O)/C(=C(/C(=O)Nc1ccccc1Cl)\Cl)/Cl 3H-367S c1cc(ccc1c2c(snn2)SC3CCCCC3)F 3H-368S COC(=O)CSc1c(nns1)c2ccc(cc2)F 3H-369S c1ccc(c(c1)Sc2c(nns2)c3ccc(cc3)F)Cl 3H-370S Cc1ccc(cc1)S(=O)c2c(nns2)c3ccc(cc3)Cl 3H-371S c1ccc(cc1)c2c(snn2)S 3H-372S CSc1c(nns1)c2ccccc2 3H-373S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccc(cc3)OC(F)(F)F 3H-374S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)NC(C)C 3H-375S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccccc3Cl 3H-376S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3cccc(c3)Cl 3H-377S Cc1cccc(c1)Sc2c(nns2)c3ccc(cc3)F 3H-378S c1cc(ccc1c2c(snn2)Sc3ccc(cc3)Br)F 3H-379S c1ccnc(c1)Sc2c(nns2)c3ccc(cc3)F 3H-380S c1cc(ccc1c2c(snn2)S(=O)C3CCCCC3)F 3H-381S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3cccc(c3Cl)Cl 3H-382S Cc1nc(nn1c2cc(cc(c2)Cl)Cl)C(=O)Nc3ccccc3C(F)(F)F 3H-383S CS(=O)c1c(nns1)c2ccccc2 3H-384S c1cc(ccc1c2c(snn2)Sc3ccc(c(c3)Cl)Cl)F 3H-385S c1cc(c(cc1Cl)Cl)c2c(snn2)S 3H-386S c1cc(ccc1c2c(snn2)S)Cl 3H-387S C=CCSc1c(nns1)c2ccccc2 3H-388S Cc1cccc(c1NC(=O)C(=C(Cl)Cl)Cl)C 3H-389S CSc1c(nns1)c2ccc(cc2Cl)Cl 3H-391S Cc1ccccc1NC(=O)C(=C(Cl)Cl)Cl 3H-393S c1cc(ccc1NC(=O)CSCC(=O)O)Cl 3H-394S c1ccc(cc1)NC(=O)CSCC(=O)O 3H-395S c1cc(ccc1N2C(=O)CSCC2=O)Cl 3H-396S COC(=O)CSc1c(nns1)c2ccc(cc2Cl)Cl 3H-397S C=CCSc1c(nns1)c2ccc(cc2Cl)Cl 3H-399S c1ccc(cc1)N2C(=O)CSCC2=O 3H-400S Cc1c(nc(s1)c2ccccn2)OC(=O)C3CC3 3H-401S Cc1c(nc(s1)c2ccncc2)OC(=O)C3CC3 3H-402S Cc1c(nc(s1)c2cccnc2)OC(=O)c3cccc(c3Cl)Cl 3H-403S Cc1c(nc(s1)c2cccnc2)OC(=O)C(C)(C)C 3H-404S Cc1c(nc(s1)c2cccs2)OC(=O)c3ccccc3 3H-406S Cc1c(nc(s1)c2cccs2)OC(=O)c3cccc(c3)C(F)(F)F 3H-407S CCCCC(=O)/C=C/1\c2ccccc2C(=O)N1c3ccccc3 3H-408S CCCC(=O)/C=C/1\c2ccccc2C(=O)N1c3ccccc3 3H-409S CCCCCC#CC1(c2ccccc2C(=O)N1c3ccccc3)O 3H-410S Cc1c(nc(s1)c2cnccn2)O 3H-411S CCCCCC(=O)/C=C\1/c2ccccc2C(=O)N1c3ccccc3 3H-412S CCCC(=O)/C=C\1/c2ccccc2C(=O)N1C 3H-413S Cc1c(nc(s1)c2cnccn2)OC(=O)c3ccc(cc3F)F 3H-414S Cc1c(nc(s1)c2cnccn2)OC(=O)c3cccs3 3H-415S Cc1c(nc(s1)c2cnccn2)OC(=O)c3cccc(c3)OC 3H-416S Cc1c(nc(s1)c2cnccn2)OC(=O)c3ccc(cc3Cl)S(=O)(=O)C 3H-417S Cc1c(nc(s1)c2cnccn2)OC(=O)C3CC3 3H-418S Cc1c(nc(s1)c2cccc(c2)C(F)(F)F)OC(=O)C3CC3 3H-419S Cc1c(nc(s1)c2cnccn2)OC 3H-420S c1cc(ccc1SCC(CSc2ccc(cc2)Cl)O)Cl 3H-422S c1ccc(cc1)SCC(=O)CSc2ccc(cc2)Cl 3H-423S Cc1c(nc(s1)c2ccc(cc2)Cl)OC(=O)Nc3cccc(c3)C(F)(F)F 3H-425S Cc1c(nc(s1)c2ccc(cc2)Cl)OCc3ccc(cc3)Cl 3H-426S Cc1c(nc(s1)c2ccc(cc2)C(=O)OC)O 3H-429S Cc1c(nc(s1)c2ccc(cc2)C(=O)OC)OC(=O)CCCl 3H-431S Cc1c(nc(s1)c2ccc(cc2)C(=O)OC)OC 3H-432S Cc1c(nc(s1)c2ccc(cc2)C(=O)OC)OCc3ccc(c(c3)Cl)Cl 3H-433S c1ccc(cc1)S(=O)(=O)CC(CSc2ccc(cc2)Cl)O 3H-442S c1ccc(cc1)S(=O)(=O)CC(CSc2cccc(c2)C(F)(F)F)O 3H-444S c1ccc(cc1)S(=O)(=O)CC(=O)CSc2ccc3ccccc3c2 3H-447S Cc1c(nc(s1)c2ccc(cc2)C(=O)OC)OCc3ccc(cc3)Cl 3H-452S Cc1c(nc(s1)c2ccc(nc2)Cl)OC(=O)C3CC3 3H-453S Cc1c(nc(s1)c2ccc(nc2)Cl)OC(=O)C(=C(Cl)Cl)Cl 3H-454S Cc1c(nc(s1)c2ccc(nc2)Cl)OC(=O)c3cccs3 3H-455S Cc1c(nc(s1)c2ccc(nc2)Cl)OC(=O)c3ccc(cc3F)F 3H-456S c1ccc(cc1)S(=O)(=O)CC(CSc2cccc(c2)Cl)O 3H-459S Cc1ccc(cc1)SCC(CS(=O)(=O)c2ccccc2)O 3H-460S Cc1ccc(cc1)SCC(=O)CSc2ccc(cc2)C 3H-462S Cn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)Cl 3H-465S c1cc(ccc1F)SCC(CSc2ccc(cc2)F)O 3H-467S c1cc(ccc1SCC(=O)CSc2ccc(cc2)Br)Br 3H-468S c1cc(ccc1SCC(CSc2ccc(cc2)Br)O)Br 3H-470S c1cc(cc(c1)Cl)SCC(CSc2cccc(c2)Cl)O 3H-472S c1ccc(c(c1)SCC(CSc2ccccc2Cl)O)Cl 3H-474S Cc1ccc(cc1)S(=O)(=O)CC(=O)CSc2ccc(cc2)Br 3H-479S c1ccc(cc1)SCC(CS(=O)(=O)c2ccccc2)O 3H-482S Cc1ccc(cc1)NC(=O)CSCC(=O)O 3H-501S c1cc(ccc1Sc2c(nns2)c3ccc(cc3Cl)Cl)Cl 3H-506S c1cc(ccc1CSc2c(nns2)c3ccc(cc3Cl)Cl)Cl 3H-507S COc1ccc(cc1)NC(=O)CSCC(=O)O 3H-508S CC(C)S(=O)c1c(nns1)c2ccc(cc2Cl)Cl 3H-509S Cc1ccc(cc1)Sc2c(nns2)c3ccc(cc3Cl)Cl 3H-510S c1ccnc(c1)Sc2c(nns2)c3ccc(cc3Cl)Cl 3H-511S Cc1ccccc1NC(=O)/C(=C(/S(=O)(=O)C(C)C)\Cl)/Cl 3H-515S Cc1ccc(cc1)N2C(=O)CSCC2=O 3H-516S COc1ccc(cc1)N2C(=O)CSCC2=O 3H-517S c1cc(ccc1C#N)NC(=O)CSCC(=O)O 3H-518S c1cc(c(cc1NC(=O)CSCC(=O)O)Cl)Cl 3H-519S c1cc(ccc1CS(=O)c2c(nns2)c3ccc(cc3Cl)Cl)Cl 3H-520S CSc1c(nns1)c2ccc(cc2)Cl 3H-521S C=CCSc1c(nns1)c2ccc(cc2)Cl 3H-522S c1cc(ccc1N2C(=O)CS(=O)CC2=O)Cl 3H-523S c1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)O 3H-524S COc1ccc(cc1OC)NC(=O)CSCC(=O)O 3H-525S c1cc(ccc1C#N)N2C(=O)CSCC2=O 3H-526S c1cc(ccc1N2C(=O)CS(=O)(=O)CC2=O)Cl 3H-527S Cc1ccc(cc1)S(=O)c2c(nns2)c3ccc(cc3Cl)Cl 3H-528S c1cc(cc(c1)Cl)Sc2c(nns2)c3ccc(cc3Cl)Cl 3H-529S c1cc(c(cc1N2C(=O)CSCC2=O)Cl)Cl 3H-530S c1cc(c(cc1Cl)Cl)N2C(=O)CSCC2=O 3H-531S COc1ccc(cc1OC)N2C(=O)CSCC2=O 3H-532S c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2c(nns2)c3ccc(cc3Cl)Cl 3H-533S COc1ccc(cc1)Oc2cnns2 3H-544S c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2cnns2 3H-549S c1ccc(cc1)S(=O)(=O)CC(CSc2ccc(cc2)F)O 3H-852S c1c(cnc(c1Cl)N2CCN(CC2)CCNS(=O)(=O)C(F)(F)F)C(F)(F)F 3H-900 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C(=O)C(=O)N4CCOCC4 3H-901 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C(=O)C(=O)N 3H-903 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)C(=O)c2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl 3H-904 COC(=O)CCCNc1c(cc(cn1)C(F)(F)F)Cl 3H-905 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C(=O)C(=O)N4CCN(CC4)c5ccc(cc5)Cl 3H-906 c1c(cnc(c1Cl)NCCCC(=O)NN)C(F)(F)F 3H-908 c1ccc(cc1)CN2CCN(CC2)C(=O)C(=O)c3cn(c4c3cccc4)c5c(cc(cn5)C(F)(F)F)Cl 3H-909 c1cc(ccc1C(=O)NCC(=O)NNC(=O)CCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl 3H-910 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)/C=N\Nc4c(cc(cn4)C(F)(F)F)Cl 3H-911 CN1C(=O)C(=CC2=NC(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl)C(=O)N(C1=O)C 3H-912 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C=C(C#N)C#N 3H-913 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)CO 3H-914 c1ccc(cc1)COc2ccc3c(c2)c(cn3c4c(cc(cn4)C(F)(F)F)Cl)C=O 3H-915 CC1(OC(=O)C(=Cc2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl)C(=O)O1)C 3H-916 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C4OCCO4 3H-917 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)/C=N\OCc4ccc(cc4)Cl 3H-918 CO/N=C\c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 3H-919 CCOC(=O)/C=C\c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 3H-920 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)/C=N\OCc4c(cc(cn4)C(F)(F)F)Cl 3H-922 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)/C=N\O 3H-923 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C#N 3H-924 CC(=O)/C=C\c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 3H-925 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)/C=C\[N+](=O)[O-] 3H-926 c1ccc(cc1)COc2ccc3c(c2)c(cn3c4c(cc(cn4)C(F)(F)F)Cl)C=C(C#N)C#N 3H-927 c1c(cnc(c1Cl)NCCCC(=O)NNC(=N)CC#N)C(F)(F)F 3H-928 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C(=O)C(=O)NCCN4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 3H-929 CCOC(=O)NC(=O)C(/C=N\NC(=O)CCCNc1c(cc(cn1)C(F)(F)F)Cl)C#N 3H-930 c1ccc2c(c1)C(=O)N(C2=O)OCc3ccc(cc3)Cl 3H-931 C/C(=N\Nc1ccc(cc1)Cl)/c2cn(c(=O)n(c2=O)Cc3ccc(cc3)F)N(C)c4c(cc(cn4)C(F)(F)F)Cl 3H-933 c1ccc(cc1)C2=N/C(=C/c3cn(c4c3cccc4)c5c(cc(cn5)C(F)(F)F)Cl)/C(=O)O2 3H-934 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)/C=C/C(=O)O 3H-935 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)C4SCCCS4 3H-936 CNC(=S)/C(=C(\N)/N1CCN(CC1)c2ccc(cc2)OC)/C#N 3H-937 CCOC(=O)c1cc(c(nc1NN=C2CCN(CC2)C)O)C(=O)OCC 3H-938 CCOC(=O)c1cc(c(nc1NN=C2CCN(CC2)c3cccc(n3)F)O)C(=O)OCC 3H-939 CCOC(=O)c1cc(c(nc1NN=C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])O)C(=O)OCC 3H-940 CNC(=S)/C(=C(\N)/N1CCN(CC1)c2ccccn2)/C#N 3H-943 CNc1c(c(ns1)N2CCN(CC2)c3ccc(cc3)OC)C#N 3H-944 CCOC(=O)c1cc(c(nc1NN=C2CCN(CC2)Cc3ccccc3)O)C(=O)OCC 3H-946 CN1C(C2C(O1)C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)c4ccc(cc4)OC 3H-947 CCOC(=O)/C(=C(/N)\N1CCN(CC1)c2ccc(cc2)OC)/SC#N 3H-948 c1c(cnc(c1Cl)CO/N=C/c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 3H-949 CCOC(=O)c1cc(c(nc1n2c(cc(n2)C)C)O)C(=O)OCC 3H-950 CN1C(C2C(O1)C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)c4ccccc4 3H-951 c1c(cnc(c1Cl)N2CCN(CC2)c3c(cc(c(n3)N)C#N)C#N)C(F)(F)F 3H-952 c1c(cnc(c1Cl)N2CCN(CC2)/C(=C(\C=C(C#N)C#N)/C#N)/N)C(F)(F)F 3H-954 c1c(cnc(c1Cl)NCC2CC(=NO2)C(=O)/N=C/NO)C(F)(F)F 3H-956 CCOC(=O)c1cc(c(=O)n(c1N)NC(=O)c2ccccc2)C(=O)OCC 3H-957 CCOC(=O)c1cc(c(nc1NN=C2CCN(CC2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])O)C(=O)OCC 3H-958 CON/C=N/C(=O)C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 3H-959 c1c(cnc(c1Cl)N2CCN(CC2)c3c(cc4c(ncnc4n3)N)C#N)C(F)(F)F 3H-960 CC1(CC(=O)C2(C3C(C(=O)N(C3=O)CCNc4c(cc(cn4)C(F)(F)F)Cl)ON2)C(=O)C1)C 3H-961 c1cc(ccc1C(=O)N2CC(CC2C(=O)O)O)F 3H-962 c1c(cnc(c1Cl)NCC2CC(=NO2)CO)C(F)(F)F 3H-964 CNC(=S)NNC(=O)C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 3H-965 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)NNc2cccc(n2)Cl 3J-001 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)NNc2ccccn2 3J-002 c1ccc(c(c1)CC[N+](=O)[O-])NC(=O)Nc2ccc(cc2)Cl 3J-005 COC(=O)c1ccccc1CC[N+](=O)[O-] 3J-006 CCOC(=O)/C(=C/c1c(cc(cn1)C(F)(F)F)Cl)/O 3J-007 c1ccc2c(c1)N/C(=C/c3c(cc(cn3)C(F)(F)F)Cl)/C(=O)N2 3J-010 CCOC(=O)/C(=C/c1c(cc(cn1)C(F)(F)F)Cl)/N 3J-012 CCOC(=O)/C(=C(\C#N)/c1cccs1)/O 3J-013 COC(=O)c1ccccc1CSC(=[NH2+])N.[Br-] 3J-015 c1ccc2c(c1)CSC2=O 3J-016 CC(=O)Oc1ccc(cc1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3J-019 CN(C)/C=C\1/c2ccccc2C(=O)S1 3J-020 c1ccc(cc1)N/C=C\2/c3ccccc3C(=O)S2 3J-021 Cc1ccc(cc1)c2nc(c(c(n2)Cl)C#N)c3ccc(cc3)OC 3J-022 Cc1ccc(cc1)c2nc(c(c(n2)N3CCN(CC3)C)C#N)c4ccc(cc4)OC 3J-023 CS(=O)(=O)Oc1ccc(cc1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl 3J-025 CCOC(=O)/C(=C/c1c(cc(cn1)C(F)(F)F)Cl)/N/C=N/OC 3J-027 CC(=O)OCc1ccc(cc1)Cl 3J-029 Cc1c(c(n(n1)C)Cl)S(=O)(=O)N(C)C 3J-032 c1ccc(cc1)CC(=O)C(C#N)c2ccc(cc2)Cl 3J-041 CC(C)(CNc1c(cc(cn1)C(F)(F)F)Cl)SCC(=O)c2ccc(cc2)Cl 3J-042 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 3J-043 CC(=O)Oc1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 3J-044 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCc3ccc(cc3)Cl 3J-045 c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 3J-048 CS(=O)(=O)Oc1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 3J-052 Cc1cc2c(cc1C)nc([nH]2)C(Cc3ccccc3)NC(=O)c4ccccc4 3J-301S CC(C)CC(c1[nH]c2ccccc2n1)NC(=O)c3ccccc3 3J-302S Cc1ccc2c(c1)nc([nH]2)CNC(=O)c3ccc(cc3Cl)Cl 3J-303S COc1cccc(c1)C(=O)NC(Cc2ccccc2)C(=O)O 3J-304S c1ccc(cc1)CC(C(=O)O)NC(=O)c2ccc(c(c2)Cl)Cl 3J-305S c1ccc(c(c1)C(=O)NCc2[nH]c3ccccc3n2)Cl 3J-306S CC(c1[nH]c2ccccc2n1)NC(=O)c3ccc(cc3)Cl 3J-307S CC(C)C(C(=O)O)NC(=O)c1ccccc1 3J-309S COc1cccc(c1)C(=O)NC(Cc2ccccc2)c3[nH]c4ccccc4n3 3J-310S Cc1ccc2c(c1)nc([nH]2)C(Cc3ccccc3)NC(=O)c4cccc(c4)OC 3J-311S Cc1ccc2c(c1)nc([nH]2)C(CC(C)C)NC(=O)c3ccccc3 3J-312S CN(C)c1c(cnc(n1)c2ccccn2)OC 3J-313S c1ccc(cc1)CC(c2[nH]c3ccccc3n2)NC(=O)c4ccc(c(c4)Cl)Cl 3J-315S CC(C)C(c1[nH]c2ccccc2n1)NC(=O)c3ccccc3 3J-316S Cc1cc2c(cc1C)nc([nH]2)CNC(=O)c3ccccc3Cl 3J-317S CC(C(=O)O)NC(=O)c1ccccc1F 3J-318S c1ccc(cc1)C(C(=O)O)NC(=O)c2ccccc2 3J-319S CC(C)Oc1c(cnc(n1)c2ccccn2)OC 3J-320S COc1cnc(nc1Oc2ccc(c3c2cccc3)Cl)c4ccccn4 3J-321S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)Cl)ncn2Cc4ccccc4 3J-322S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)F)ncn2Cc4ccccc4 3J-323S CC(c1[nH]c2ccccc2n1)NC(=O)c3ccccc3F 3J-324S Cc1ccc2c(c1)nc([nH]2)C(C)NC(=O)c3ccccc3F 3J-325S Cc1cccc(c1Oc2c(cnc(n2)c3ccccn3)OC)C 3J-326S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)ncn2Cc4ccccc4 3J-328S Cc1cc2c(c(c1C)NS(=O)(=O)C)ncn2Cc3ccccc3 3J-329S c1cc(ccc1C(=O)NCC(=O)O)F 3J-330S CC(C(=O)O)NC(=O)c1cccc(c1)Cl 3J-334S CC(C)C(C(=O)O)NC(=O)c1ccc(cc1)F 3J-335S CC(C)C(C(=O)O)NC(=O)c1ccc(cc1Cl)Cl 3J-337S CC(C(=O)O)NC(=O)c1ccc(cc1Cl)Cl 3J-338S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3)C(F)(F)F)ncn2Cc4ccccc4 3J-339S c1ccc2c(c1)[nH]c(n2)CNC(=O)c3ccc(cc3)F 3J-340S c1ccc(cc1)CC(c2[nH]c3ccccc3n2)NC(=O)c4ccccc4F 3J-341S CC(C)CC(c1[nH]c2ccccc2n1)NC(=O)c3ccccc3Cl 3J-342S CC(c1[nH]c2ccccc2n1)NC(=O)c3cccc(c3)Cl 3J-343S Cc1cc2c(c(c1C)[N+](=O)[O-])ncn2C 3J-344S Cc1cc2c(c(c1C)N)ncn2C 3J-345S Cc1cc2c(cc1C)nc([nH]2)C(Cc3ccccc3)NC(=O)c4ccccc4F 3J-346S c1ccc2c(c1)[nH]c(n2)CNC(=O)c3cccc(c3)Cl 3J-347S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(ccc3Cl)Cl)ncn2Cc4ccccc4 3J-348S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(cc(c3)Cl)Cl)ncn2Cc4ccccc4 3J-349S CC(C)C(c1[nH]c2ccccc2n1)NC(=O)c3ccc(cc3)F 3J-350S CC(C)C(c1[nH]c2ccccc2n1)NC(=O)c3ccc(cc3Cl)Cl 3J-351S CC(c1[nH]c2ccccc2n1)NC(=O)c3ccc(cc3Cl)Cl 3J-352S Cc1ccc2c(c1)nc([nH]2)C(C(C)C)NC(=O)c3ccc(cc3)F 3J-353S c1cc2nnc(n2nc1)Cl 3J-354S COc1cnc(nc1O)S 3J-355S CC1COc2ccccc2N1 3J-356S CC1COc2ccccc2N1C(=O)C(Cl)Cl 3J-357S Cc1ccc2c(c1)nc([nH]2)C(C)NC(=O)c3ccc(cc3Cl)Cl 3J-358S Cc1ccc(cc1)S(=O)(=O)Nc2c(c(cc3c2ncn3Cc4ccccc4)C)C 3J-360S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)Cl)ncn2C 3J-361S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)F)ncn2C 3J-362S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)OC)ncn2C 3J-363S CC(C)CC(C(=O)O)NC(=O)c1cccc(c1)Cl 3J-364S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(ccc3Cl)Cl)ncn2C 3J-365S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)ncn2C 3J-366S Cc1cc2c(cc1C)nc([nH]2)CNC(=O)c3ccc(cc3)F 3J-367S Cc1cc2c(c(c1C)NS(=O)(=O)C)ncn2C 3J-368S Cc1ccc(cc1)Cn2cnc3c2cc(c(c3N(=O)=O)C)C 3J-370S Cc1ccc(cc1)Cn2cnc3c2cc(c(c3N)C)C 3J-371S Cc1ccc(cc1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)Cl)C)C 3J-372S CN(C)c1ncc(c(n1)O)OC 3J-373S COc1cnc(nc1O)SC 3J-374S COc1cnc(nc1O)SCc2ccc(cc2)Cl 3J-375S COc1cnc(nc1O)SCc2ccccc2 3J-376S COc1cnc(nc1O)SCc2cccc(c2)C(F)(F)F 3J-377S CCOC(=O)CSc1ncc(c(n1)O)OC 3J-378S COc1cnc(nc1O)SCc2ccc(cc2Cl)Cl 3J-379S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3)C(F)(F)F)ncn2C 3J-380S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3Cl)Cl)ncn2C 3J-381S CCOC(=O)C(C)Sc1ncc(c(n1)O)OC 3J-383S CC(C)Sc1ncc(c(n1)O)OC 3J-384S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)C(C)(C)C)ncn2C 3J-385S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccccc3Cl)ncn2C 3J-386S Cc1cc2c(c(c1C)NS(=O)(=O)c3c(cc(cc3Cl)Cl)Cl)ncn2C 3J-387S Cc1cc2c(cc1C)nc([nH]2)CNC(=O)c3ccccc3 3J-389S CC1C(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)F 3J-501S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4ccc(cc4Cl)Cl 3J-502S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4c(cccc4Cl)F 3J-504S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4c(cccc4Cl)Cl 3J-505S Cc1ccc(cc1C)NC(=O)Cn2c3ccccc3nc2/C=C/c4ccccc4 3J-506S c1ccc(cc1)/C=C/c2nc3ccccc3n2CC(=O)Nc4ccc(cc4)Cl 3J-507S c1ccc(cc1)/C=C/c2nc3ccccc3n2CC(=O)Nc4ccc(cc4)OC(F)(F)F 3J-508S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4ccc(cc4)C#N 3J-509S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4ccc(c(c4)Cl)Cl 3J-510S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4ccc(cc4)C(F)(F)F 3J-511S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4ccc(cc4)C(=O)OC 3J-512S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4ccccc4F 3J-513S CC1C(=O)N(c2ccccc2N1C(=O)c3ccc(cc3)F)Cc4ccc(cc4)F 3J-514S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4cccc(c4)C#N 3J-515S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4ccc(cc4)[N+](=O)[O-] 3J-516S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4ccccc4F 3J-518S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4ccc(cc4)F 3J-519S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4ccc(cc4)C(=O)OC 3J-520S CC1C(=O)Nc2ccccc2N1C(=O)c3c(cccc3F)F 3J-521S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4c(cccc4Cl)Cl 3J-522S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4cccc(c4)OC 3J-524S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4cccc(c4)OC 3J-525S CC1C(=O)Nc2ccccc2N1C(=O)C3CC3 3J-526S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4ccc(cc4)OC 3J-539S CC1C(=O)N(c2ccccc2N1C(=O)c3c(cccc3F)F)Cc4ccc(cc4)C(C)(C)C 3J-540S CC(=O)COc1ccccc1[N+](=O)[O-] 3J-542S c1ccc2c(c1)[nH]c(n2)c3cccnc3Cl 3J-543S c1cc(cc(c1)Cl)n2c(nnn2)c3ccc(c(c3)Cl)Cl 3J-545S CC1C(=O)N(c2ccccc2N1C(=O)C3CC3)Cc4ccc(cc4)[N+](=O)[O-] 3J-546S CC1C(=O)N(c2ccccc2N1C(=O)C3CC3)Cc4ccc(cc4)C(=O)OC 3J-547S c1ccc(cc1)Cn2c3ccccc3nc2c4cccnc4Cl 3J-548S c1ccc2c(c1)nc(n2Cc3ccc(cc3Cl)Cl)c4cccnc4Cl 3J-549S c1ccc2c(c1)nc(n2Cc3ccc(c(c3)Cl)Cl)c4cccnc4Cl 3J-550S COc1cccc(c1)Cn2c3ccccc3nc2c4cccnc4Cl 3J-551S c1ccc2c(c1)nc(n2Cc3c(cccc3Cl)Cl)c4cccnc4Cl 3J-552S CN(C)/C=C(\C=O)/c1ccc(cc1)Cl 3J-553S c1cc(cc(c1)Cl)c2nnnn2c3cccc(c3)Cl 3J-554S c1cc(c(cc1c2nnnn2c3ccc(c(c3)Cl)Cl)Cl)Cl 3J-555S CC1C(=O)N(c2ccccc2N1C(=O)C(C)(C)C)Cc3ccc(c(c3)Cl)Cl 3J-556S c1ccc(c(c1)Cn2c3ccccc3nc2c4cccnc4Cl)F 3J-557S c1ccc2c(c1)nc(n2Cc3cccc(c3)F)c4cccnc4Cl 3J-558S c1ccc2c(c1)nc(n2Cc3ccc(cc3)F)c4cccnc4Cl 3J-559S c1ccc2c(c1)nc(n2Cc3c(cccc3Cl)F)c4cccnc4Cl 3J-560S c1cc(cc(c1)Cl)c2nnnn2c3ccc(c(c3)Cl)Cl 3J-561S CC1C(=O)N(c2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F)Cc4ccc(cc4)C(F)(F)F 3J-562S c1ccc(c(c1)Cn2c3ccccc3nc2c4cccnc4Cl)Cl 3J-563S c1ccc2c(c1)nc(n2Cc3cccc(c3)Cl)c4cccnc4Cl 3J-564S c1ccc2c(c1)nc(n2Cc3ccc(cc3)Cl)c4cccnc4Cl 3J-565S c1cc(cc(c1)C(F)(F)F)c2nnnn2c3ccc(c(c3)Cl)Cl 3J-566S Cc1cccc(c1)c2nnnn2c3cccc(c3)C 3J-567S Cc1cccc(c1)c2nnnn2c3ccc(c(c3)Cl)Cl 3J-570S COc1cnc(nc1Oc2cccc(c2)[N+](=O)[O-])c3ccccn3 3J-574S Cc1cccc(c1)n2c(nnn2)c3cccc(c3)Cl 3J-575S Cc1cccc(c1)n2c(nnn2)c3cccc(c3)C(F)(F)F 3J-576S Cc1c2ccccc2oc1C(=O)c3ccc(cc3)Cl 3J-577S Cc1c2ccccc2oc1C(=O)c3ccccc3 3J-578S Cc1cccc(c1)Cn2c3ccccc3nc2c4cccnc4Cl 3J-579S Cc1ccc(cc1)Cn2c3ccccc3nc2c4cccnc4Cl 3J-580S c1ccc2c(c1)C(=O)N(C2=O)CCSc3ccc(cc3)Br 3J-581S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CBr 3J-583S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CBr 3J-584S c1cc(cc(c1)C(F)(F)F)c2nnnn2c3cccc(c3)Cl 3J-586S c1ccc(cc1)SCc2c3ccccc3oc2C(=O)c4ccc(cc4)Cl 3J-587S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CSc4ccc(cc4)Cl 3J-588S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CSc4ccc(cc4Cl)Cl 3J-589S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CSc4cccc(c4)C(F)(F)F 3J-590S COc1ccc(cc1)SCc2c3ccccc3oc2C(=O)c4ccc(cc4)Cl 3J-591S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)c4cccc(c4)C(F)(F)F 3J-592S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)(=O)c4cccc(c4)C(F)(F)F 3J-593S Cc1ccccc1Cn2c3ccccc3nc2c4cccnc4Cl 3J-594S c1ccc2c(c1)nc(n2Cc3cccc(c3)C(F)(F)F)c4cccnc4Cl 3J-595S c1ccc2c(c1)nc(n2Cc3ccc(cc3)C(F)(F)F)c4cccnc4Cl 3J-596S c1ccc(cc1)S(=O)(=O)Cc2c3ccccc3oc2C(=O)c4ccc(cc4)Cl 3J-597S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)(=O)c4ccc(cc4Cl)Cl 3J-598S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)(=O)c4ccc(cc4)Cl 3J-599S Cn1c2ccccc2nc1c3cccnc3Cl 3J-600S CCn1c2ccccc2nc1c3cccnc3Cl 3J-601S CCOC(=O)Cn1c2ccccc2nc1c3cccnc3Cl 3J-602S C=CCn1c2ccccc2nc1c3cccnc3Cl 3J-603S Cc1cccc(c1)n2c(nnn2)c3ccc(c(c3)Cl)Cl 3J-604S Cc1cccc(c1)c2nnnn2c3cccc(c3)C(F)(F)F 3J-605S c1cc(cc(c1)n2c(nnn2)c3ccc(c(c3)Cl)Cl)C(F)(F)F 3J-606S c1cc(cc(c1)Cl)c2nnnn2c3cccc(c3)C(F)(F)F 3J-607S c1ccc2c(c1)C(=O)N(C2=O)CCSc3ccc(cc3)Cl 3J-608S c1cc(ccc1SCCN)Cl 3J-609S c1cc(ccc1C(=O)NCCSc2ccc(cc2)Cl)F 3J-610S c1cc(cc(c1)Cl)C(=O)NCCSc2ccc(cc2)Cl 3J-611S c1ccc(cc1)CN2CC3CN(CC(C2)C3=O)Cc4ccccc4 3J-901 c1ccc(cc1)N2C(=O)NC3(N2)CCC(=O)CC3 3J-902 c1cc(c(nc1)N2CCC(=O)CC2)[N+](=O)[O-] 3J-903 c1cnn(c1c2c(ccs2)Cl)c3c(cc(cn3)C(F)(F)F)Cl 3J-905 c1ccc(cc1)N2C(=O)NC3(N2)CCC4(CC3)NC(=O)N(N4)C5CCS(=O)(=O)C5 3J-907 c1cc(sc1)S(=O)(=O)Nc2cc(ccc2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 3J-909 c1cc(c(nc1)N2CCC(CC2)O)[N+](=O)[O-] 3J-910 c1cc(cc(c1)F)c2nccc(n2)c3ccc4c(c3)c(on4)c5ccc(cc5)F 3J-911 c1cc(c(nc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)NS(=O)(=O)c4cccs4 3J-912 c1cc(c(nc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)NS(=O)(=O)C(F)(F)F 3J-913 c1cc(ccc1c2c3cc(ccc3no2)c4cc[nH]n4)F 3J-914 c1cc(ccc1c2c3cc(ccc3no2)c4ccn(n4)c5c(cc(cn5)C(F)(F)F)Cl)F 3J-915 c1cc(c(cc1C(F)(F)F)NS(=O)(=O)C(F)(F)F)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3J-917 COC(CNC(=S)Nc1ccccc1)OC 3J-918 c1ccc(cc1)n2ccnc2S 3J-919 c1cc(c(nc1)N2CCC(CC2)Oc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 3J-922 c1ccc(cc1)n2ccnc2Sc3c(cc(cn3)C(F)(F)F)Cl 3J-923 c1ccc(cc1)Oc2ccc(cc2)C(=O)c3conc3c4c(cccc4Cl)Cl 3J-924 c1ccnc(c1)C(=O)c2conc2c3c(cccc3Cl)Cl 3J-925 c1cc2c(nc1)n(c(=O)c(n2)Cl)CCNc3c(cc(cn3)C(F)(F)F)Cl 3J-928 CCOC(=O)c1c[nH]c2c(cnn2c1=O)C#N 3J-930 c1cc2c(nc1)n(c(=O)c(n2)NN)CCNc3c(cc(cn3)C(F)(F)F)Cl 3J-931 c1cc2c(nc1)n(c(=O)c(n2)N3CCOCC3)CCNc4c(cc(cn4)C(F)(F)F)Cl 3J-932 CN1CCN(CC1)c2c(=O)n(c3c(n2)cccn3)CCNc4c(cc(cn4)C(F)(F)F)Cl 3J-933 c1cc2c(nc1)n(c(=O)c3n2cnn3)CCNc4c(cc(cn4)C(F)(F)F)Cl 3J-934 COc1ccc(cc1)/C=N/Nc2c(=O)n(c3c(n2)cccn3)CCNc4c(cc(cn4)C(F)(F)F)Cl 3J-935 c1ccc2c(c1)C3C(C(=NO3)c4c(cccc4Cl)Cl)C(=O)O2 3J-936 CCOC(=O)c1cn[nH]c1N/C=C(\C#N)/C(=O)OCC 3J-937 C1C(NC(S1)C(=O)O)C(=O)O 3J-939 c1ccc2c(c1)c3c([nH]2)C4(CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl)NCC3.Cl 3J-941 c1cc(ccc1C(=O)O)N2CCN=C2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 3J-942 COC(=O)C1CSC([NH2+]1)C(=O)OC.[Cl-] 3J-943 COC(=O)C1CSC(N1)C(=O)OC 3J-945 COC(=O)C1CSC(N1C(=O)CCl)C(=O)OC 3J-946 c1cc(ccc1Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)S(=O)(=O)Cl 3K-002 CCN(CC)S(=O)(=O)c1ccc(cc1)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 3K-004 c1cc(cnc1)CNS(=O)(=O)c2ccc(cc2)Oc3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 3K-005 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(C#N)c3ccc(cc3)Cl 3K-006 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(c3ccc(cc3)Cl)C(=O)N 3K-007 COc1ccnc(c1C#N)n2cccc2 3K-008 c1ccn(c1)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 3K-009 COc1ccnc(c1C#N)NCc2ccc(cc2)Cl 3K-011 c1cc(ccc1Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)S(=O)(=O)N4CCOCC4 3K-012 CN(C)/C=N/C(=O)C(c1ccc(cc1)Cl)c2c(nc3ccccc3n2)C(F)(F)F 3K-014 CO/N=C/NC(=O)C(c1ccc(cc1)Cl)c2c(nc3ccccc3n2)C(F)(F)F 3K-015 Cc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 3K-016 COc1ccnc(c1C#N)n2cccc2C=O 3K-017 CN(C)/C=N/c1c(c(ccn1)OC)C#N 3K-020 CN(c1c(c(ccn1)OC)C#N)N 3K-021 COc1ccnc(c1C(=O)N)Oc2ccc(cc2)Cl 3K-022 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)C(=O)CCl 3K-023 Cc1ccc(cc1)SCC(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl 3K-025 c1cc(c(cc1F)F)N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N 3K-026 c1cc(ccc1N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N)OC(F)(F)F 3K-027 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)N/C=C\c3c4cnc5c(cnn5c4ccn3)C#N 3K-028 CN(C)S(=O)(=O)c1ccc(cc1)N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N 3K-029 c1ccc(c(c1)C#N)N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N 3K-030 Cc1c(c(nc(c1C#N)Cl)N)C#N 3K-032 COc1ccnc(c1C#N)n2cccc2/C=N/O 3K-034 COc1ccnc(c1C#N)n2cccc2CO 3K-035 COc1ccnc(c1C#N)n2cccc2C#N 3K-036 C/C(=C/1\C(C(=O)O1)(C)c2c(cc(cn2)C(F)(F)F)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 3K-037 COC(=O)c1ccccc1N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N 3K-039 CCOC(=O)C(=O)c1ccc(s1)Cc2c(cc(cn2)C(F)(F)F)Cl 3K-041 COc1ccnc(c1C#N)n2cccc2/C=N/OC 3K-043 CCOC(=O)c1cnc2c(c1Oc3ccc(cc3)Cl)c(nn2C)C 3K-045 Cc1c2ccccc2sc1C(=O)/C=C/N(C)C 3K-048 Cc1c2ccccc2sc1c3ccn[nH]3 3K-049 c1ccc(c(c1)c2c3c(c(cnc3N4CCOCC4)/C=C/c5c(c(no5)c6ccccc6Cl)C(=O)N7CCOCC7)on2)Cl 3K-050 c1c(cnc(c1Cl)CCc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 3K-051 COc1ccnc(c1C#N)S(=O)(=O)c2ccc(cc2)Cl 3K-056 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)C(c3ccc(s3)Cc4c(cc(cn4)C(F)(F)F)Cl)C(c5ccc(s5)Cc6c(cc(cn6)C(F)(F)F)Cl)c7ccc(s7)Cc8c(cc(cn8)C(F)(F)F)Cl 3K-058 Cc1c(c(no1)c2c(cccc2Cl)F)C(=S)N 3K-060 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(cs3)c4cccc(c4)[N+](=O)[O-] 3K-061 Cc1c2ccccc2sc1c3ccnn3S(=O)(=O)c4ccccc4F 3K-062 CCOCCOc1c(c(cc(n1)C)C)S(=O)(=O)c2ccccc2C 3K-301S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OCCO)C)C 3K-302S Cc1ccc(cc1)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl 3K-303S c1ccc2c(c1)nc(n2Cc3ccc(cc3)F)c4ccc[nH]c4=O 3K-304S CC(C)(C)c1ccc(cc1)Cn2c3ccccc3nc2c4ccc[nH]c4=O 3K-307S CC(C)(C)c1ccc(cc1)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl 3K-308S Cn1c2cc(c(cc2nc1c3ccc[nH]c3=O)Cl)Cl 3K-309S c1cc(c(=O)[nH]c1)c2nc3cc(c(cc3n2Cc4ccc(cc4Cl)Cl)Cl)Cl 3K-311S CCCn1c2cc(c(cc2nc1c3ccc[nH]c3=O)Cl)Cl 3K-312S Cc1cccc(c1)Cn2c3ccccc3nc2c4ccc[nH]c4=O 3K-319S CC(C)(C)c1ccc(cc1)Cn2c3ccccc3nc2c4cccnc4Cl 3K-320S Cc1ccccc1S(=O)(=O)c2c(cc(nc2NCc3ccccc3)C)C 3K-322S CCCn1c2ccccc2nc1c3ccc[nH]c3=O 3K-326S Cc1ccccc1S(=O)(=O)c2c(c(c(nc2Cl)C)c3ccccc3)C 3K-327S CCn1c2ccccc2nc1c3ccc[nH]c3=O 3K-329S c1cc(cc(c1)C(F)(F)F)Cn2c3cc(c(cc3nc2c4ccc[nH]c4=O)Cl)Cl 3K-332S Cc1ccccc1S(=O)(=O)c2c(c(c(nc2OCC(C)C)C)c3ccccc3)C 3K-334S Cc1cc(nc(c1S(=O)(=O)c2cccc(c2C)Cl)OCC(C)C)C 3K-335S Cc1cc([nH]c(=O)c1S(=O)(=O)C)C 3K-336S Cc1cc(nc(c1S(=O)(=O)C)Cl)C 3K-342S c1ccc(c(c1)Cn2c3ccccc3nc2c4ccc[nH]c4=O)F 3K-343S c1ccc2c(c1)nc(n2Cc3cccc(c3)F)c4ccc[nH]c4=O 3K-344S CN(c1cnns1)N 3K-345S Cc1cc2c(cc1C)n(c(n2)c3ccc[nH]c3=O)Cc4ccc(cc4)F 3K-346S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)C=O 3K-347S Cc1cc(cc(c1)S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C)C 3K-348S Cc1cc(nc(c1S(=O)(=O)C)OC(C)C)C 3K-349S Cc1cc([nH]c(=O)c1S(=O)(=O)c2cccc(c2)C(F)(F)F)C 3K-350S Cc1ccccc1S(=O)(=O)c2c(cc(nc2NC)C)C 3K-354S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)CO 3K-355S CC(CS(=O)(=O)Cc1ccc(cc1)Cl)(c2ccccc2)O 3K-358S CC(CS(=O)(=O)Cc1ccc(cc1)Cl)(c2ccc(cc2)Cl)O 3K-359S CC(CS(=O)(=O)Cc1ccc(cc1)OC)(c2ccccc2)O 3K-360S CC(CS(=O)(=O)Cc1ccc(cc1)OC)(c2ccc(cc2)Cl)O 3K-361S Cc1ccc(cc1)S(=O)(=O)c2c(c(nn2C)c3ccccc3)CO 3K-362S Cc1cc(nc(c1S(=O)(=O)c2cccc(c2)C(F)(F)F)Cl)C 3K-364S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)C(C)(C)C)Cl)C 3K-365S Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)CO 3K-366S CC(CS(=O)(=O)Cc1ccc(cc1Cl)Cl)(c2ccccc2)O 3K-367S Cc1ccc(cc1)CS(=O)(=O)CC(C)(c2ccccc2)O 3K-368S Cc1ccc(cc1)CS(=O)(=O)CC(C)(c2ccc(cc2)Cl)O 3K-369S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)COC(=O)Nc4ccc(cc4)Cl 3K-370S CC(CS(=O)(=O)Cc1ccc(cc1Cl)Cl)(c2ccc(cc2)Cl)O 3K-371S CC(CS(=O)(=O)Cc1ccccc1)(c2ccc(cc2)Cl)O 3K-372S CC(CS(=O)(=O)Cc1ccccc1)(c2ccccc2)O 3K-373S c1ccc(cc1)c2nc3ccc(cc3c(=O)n2O)Cl 3K-505S c1ccc(c(c1)c2nc3ccc(cc3c(=O)n2O)Cl)Cl 3K-506S c1cc(cc(c1)Cl)c2nc3ccc(cc3c(=O)n2O)Cl 3K-507S c1cc(ccc1c2nc3ccc(cc3c(=O)n2O)Cl)Cl 3K-508S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(cc3)Cl)O 3K-509S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(cc3Cl)Cl)O 3K-510S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3cccc(c3Cl)Cl)O 3K-511S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3cc(cc(c3)Cl)Cl)O 3K-512S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(cc3)Br)O 3K-513S Cc1ccc(cc1C)NC(=O)c2cc(n(c(=O)n2)Cc3ccccc3)O 3K-514S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3c(cccc3Cl)Cl)O 3K-515S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(c(c3)Cl)Cl)O 3K-516S c1ccc(cc1)c2nnc(o2)c3ccc(nc3)Cl 3K-518S c1cc(c(cc1Cl)Cl)c2nc3ccc(cc3c(=O)n2O)Cl 3K-520S c1cc(c(cc1c2nc3ccc(cc3c(=O)n2O)Cl)Cl)Cl 3K-521S Cc1ccccc1c2nc3ccc(cc3c(=O)n2O)Cl 3K-523S CCOC(=O)COc1cc(nc(n1)c2ccccc2)C 3K-524S Cc1ccc(cc1)c2nc3ccc(cc3c(=O)n2O)Cl 3K-525S c1cc(ccc1C#N)c2nc3ccc(cc3c(=O)n2O)Cl 3K-527S Cn1c(c(c(n1)c2ccccc2)C(=O)O)Cl 3K-528S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(cc3)C(F)(F)F)O 3K-529S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3cccc(c3)C(F)(F)F)O 3K-530S COc1cccc(c1)NC(=O)c2cc(n(c(=O)n2)Cc3ccccc3)O 3K-531S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(cc3)OC(F)(F)F)O 3K-532S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccccc3)O 3K-533S Cc1c(cccc1Cl)NC(=O)c2cc(n(c(=O)n2)Cc3ccccc3)O 3K-534S c1cc(ccc1c2nc3ccc(cc3c(=O)n2O)Cl)[N+](=O)[O-] 3K-537S COc1ccccc1c2nc3ccc(cc3c(=O)n2O)Cl 3K-538S Cc1cc(nc(n1)c2ccccc2)OCC(=O)N 3K-542S COc1ccccc1c2nc3cc(ccc3c(=O)n2O)Cl 3K-544S c1cc(cc(c1)C(F)(F)F)c2nc3cc(ccc3c(=O)n2O)Cl 3K-545S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccccc3F)O 3K-546S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(cc3)F)O 3K-547S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(cc3F)F)O 3K-548S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(c(c3)F)F)O 3K-549S Cc1cccc(c1)NC(=O)c2cc(n(c(=O)n2)Cc3ccccc3)O 3K-561S c1ccc(cc1)Cn2c(cc(nc2=O)C(=O)Nc3ccc(c(c3F)Cl)F)O 3K-562S c1ccc(cc1)n2c(cc(nc2=O)C(=O)Nc3ccc(cc3)Br)O 3K-565S c1ccc(cc1)n2c(cc(nc2=O)C(=O)Nc3ccc(cc3)OC(F)(F)F)O 3K-566S c1ccc(cc1)n2c(cc(nc2=O)C(=O)Nc3ccc(cc3F)F)O 3K-567S c1ccc(cc1)n2c(cc(nc2=O)C(=O)Nc3ccc(c(c3)F)F)O 3K-568S Cn1c(c(c(n1)c2ccccc2)CSc3c(cccc3Cl)Cl)Cl 3K-571S Cc1ccc(cc1)SCc2c(nn(c2Cl)C)c3ccccc3 3K-574S Cn1c(c(c(n1)c2ccccc2)COC)Cl 3K-578S Cn1c(c(c(n1)c2ccccc2)CO)Sc3ccccc3C(=O)OC 3K-579S CCOC(=O)C(C)Oc1cc(nc(n1)c2ccccc2)C 3K-583S c1ccc(cc1)c2c(nc([nH]2)S)c3ccccc3 3K-584S c1ccc(cc1)CSc2[nH]c(c(n2)c3ccccc3)c4ccccc4 3K-585S c1ccc(cc1)c2c(nc([nH]2)SCc3ccc(cc3)Cl)c4ccccc4 3K-587S Cn1c(c(c(n1)c2ccccc2)CSc3ccccc3Cl)Cl 3K-589S Cn1c(c(c(n1)c2ccccc2)CSc3cccc(c3)Cl)Cl 3K-590S Cn1c(c(c(n1)c2ccccc2)CSc3ccccc3)Cl 3K-591S Cn1c(c(c(n1)c2ccccc2)CSc3ccc(cc3)Br)Cl 3K-592S Cn1c(c(c(n1)c2ccccc2)CSc3ccc(cc3)F)Cl 3K-593S Cn1c(c(c(n1)c2ccccc2)CSc3ccccc3C(=O)OC)Cl 3K-594S Cc1ccc(c(c1)SCc2c(nn(c2Cl)C)c3ccccc3)C 3K-595S Cc1ccc(c(c1)C)SCc2c(nn(c2Cl)C)c3ccccc3 3K-596S Cc1cccc(c1)SCc2c(nn(c2Cl)C)c3ccccc3 3K-597S Cn1c(c(c(n1)c2ccccc2)CSc3cccc(c3)C(F)(F)F)Cl 3K-598S COc1ccc(cc1)NC(=O)c2cc(n(c(=O)n2)Cc3ccccc3)O 3K-601S c1ccc(cc1)c2c(nc([nH]2)SCc3nc4cc(ccc4s3)F)c5ccccc5 3K-602S Cc1cc(nc(n1)c2ccccc2)OC(C)C(=O)O 3K-603S Cc1ccc(cc1)S(=O)(=O)Cc2c(nn(c2Cl)C)c3ccccc3 3K-610S Cc1cc(nc(n1)c2ccccc2)OC(C)C(=O)N 3K-611S Cn1c(c(nc1SCc2ccccc2)c3ccccc3)c4ccccc4 3K-616S CCCn1c(c(nc1SCc2ccccc2)c3ccccc3)c4ccccc4 3K-617S C=CCn1c(c(nc1SCc2ccccc2)c3ccccc3)c4ccccc4 3K-623S C#CCn1c(c(nc1SCc2ccccc2)c3ccccc3)c4ccccc4 3K-624S c1cc(ccc1n2c(cc(nc2=O)C(=O)Nc3ccc(cc3Cl)Cl)O)Cl 3K-632S c1cc(ccc1n2c(cc(nc2=O)C(=O)Nc3ccc(c(c3)Cl)Cl)O)Cl 3K-633S Cn1c(c(c(n1)c2ccccc2)CSc3ccccc3C(=O)O)Cl 3K-634S CCc1ccccc1SCc2c(nn(c2Cl)C)c3ccccc3 3K-636S c1cc(cc(c1)NC(=O)c2cc(n(c(=O)n2)c3ccc(cc3)Cl)O)C(F)(F)F 3K-638S CC(C)c1ccc(cc1)SCc2c(nn(c2Cl)C)c3ccccc3 3K-641S Cn1c(c(c(n1)c2ccccc2)CSc3c(c(c(c(c3F)F)F)F)F)Cl 3K-642S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(c(c3)Cl)Cl)Cl 3K-643S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3Cl)Cl)Cl 3K-644S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)[N+](=O)[O-])Cl 3K-645S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)F)Cl 3K-646S Cn1c(c(nc1SCc2ccc(cc2)Cl)c3ccccc3)c4ccccc4 3K-650S CCCn1c(c(nc1SCc2ccc(cc2)Cl)c3ccccc3)c4ccccc4 3K-651S c1ccc(cc1)c2c(nc([nH]2)SCc3ccc(c(c3)Cl)Cl)c4ccccc4 3K-745S Cc1cc(c(c(=O)o1)C(=O)/C=C(\C)/N(C)C)O 3K-901 Cc1c/c(=N\O)/c-2c(cc(oc2[n+]1[O-])C)O 3K-902 c1ccc2c(c1)[nH]c(=O)c(n2)NN=C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 3K-903 c1ccc2c(c1)[nH]c(=O)c(n2)NN=C3CCN(CC3)c4ccc(cc4)[N+](=O)[O-] 3K-904 c1ccc2c(c1)[nH]c(=O)c(n2)NN=C3CCN(CC3)c4c(cccn4)[N+](=O)[O-] 3K-905 CN(/C=N/C(=S)Nc1ccc(cc1Cl)Cl)O 3K-906 Cc1ccc(cc1)NC(=O)ON(C)/C=N/C(=S)Nc2c(cc(cn2)C(F)(F)F)Cl 3K-907 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)c3cccc(c3C2=O)OCc4ccc(cc4)Br 3K-909 c1cc(c(nc1)Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Cl 3K-910 c1ccc(cc1)CCNC(=O)c2cccnc2Sc3c(cc(cn3)C(F)(F)F)Cl 3K-911 COc1ccc(cc1)/C=C(\C#N)/c2nnc(s2)/N=C/Nc3ccc(cc3)Cl 3L-001 CN(C)/C=C/c1c(c(ns1)Sc2c(cc(cn2)C(F)(F)F)Cl)C#N 3L-002 COc1ccc(cc1)N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N 3L-003 c1cc(c(cc1N)Cl)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 3L-004 c1ccc(cc1)N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N 3L-005 c1cc(ccc1N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N)Br 3L-006 Cc1ccc(cc1C)N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N 3L-007 c1cc(ccc1N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N)OC(F)(F)F 3L-008 CC(C)c1ccc(cc1)N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N 3L-009 c1cc(cc(c1)N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N)C(F)(F)F 3L-010 c1cc(ccc1N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N)Cl 3L-011 c1cc(ccc1N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N)F 3L-012 Cc1ccc(c(c1)C)N/C=C/c2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N 3L-013 c1cc(ccc1N/C=C/C#N)Cl 3L-014 CO/N=C\Cc1c(c(ns1)Sc2c(cc(cn2)C(F)(F)F)Cl)C#N 3L-015 c1cc(c(c(c1)Cl)CO/N=C\Cc2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N)F 3L-016 Cc1ccc(cc1)CO/N=C\Cc2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N 3L-017 c1ccc(c(c1)CO/N=C\Cc2c(c(ns2)Sc3c(cc(cn3)C(F)(F)F)Cl)C#N)Br 3L-018 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)Cl)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 3L-019 c1cnc(nc1)Oc2ccc(cc2Cl)N 3L-021 CC(=O)Nc1ccc(c(c1)Cl)Oc2ncccn2 3L-022 CC(=O)Nc1ccc(c(c1)Cl)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 3L-023 COc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)Cl)Oc3ncccn3 3L-024 c1cc(ccc1S(=O)(=O)Nc2ccc(c(c2)Cl)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl 3L-025 COc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)Cl)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 3L-026 CC1=C(C(C(=O)N1)/C=N/OCc2ccccc2F)C(=O)OC 3L-027 Cc1c(c(ns1)Sc2ncccn2)C#N 3L-028 CC(C)(C)c1ccc(cc1)Oc2cc(cnc2C#N)C(F)(F)F 3L-029 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)Cl)Oc3ncccn3 3L-033 CC1=C(/C(=C/Nc2ccc(cc2)OC(F)(F)F)/C(=O)N1)C(=O)OC 3L-034 c1cnc(nc1)Oc2ccc(cc2Cl)NS(=O)(=O)c3ccc(cc3)Cl 3L-037 c1cnc(nc1)Oc2ccc(cc2Cl)NS(=O)(=O)c3ccc(cc3)F 3L-038 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)Cl)Oc3ncccn3 3L-039 c1ccc(c(c1)C(=O)Nc2ccc(c(c2)Cl)Oc3ncccn3)F 3L-040 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(c(c2)Cl)Oc3ncccn3 3L-041 c1cnc(nc1)Oc2ccc(cc2Cl)NC(=O)C3CC3 3L-042 Cc1ccc(cc1)Sc2c(cccn2)CO 3L-302S c1cc(c(nc1)Sc2ccc(cc2)Cl)C=O 3L-303S c1cc(c(nc1)Sc2ccc(cc2Cl)Cl)C=O 3L-304S c1cc(c(nc1)Sc2ccc(cc2)Br)C=O 3L-305S c1ccc(cc1)Sc2c(cccn2)C=O 3L-306S c1ccc(c(c1)Sc2c(cccn2)C=O)Cl 3L-307S Cc1ccc(cc1)Oc2c(cccn2)C=O 3L-311S Cc1ccc(cc1)Oc2c(cccn2)/C=N/O 3L-312S Cc1ccc(cc1)Oc2c(cccn2)/C=N/OCc3ccc(cc3Cl)Cl 3L-313S Cc1ccc(cc1)Oc2c(cccn2)/C=N/OCc3ccc(c(c3)Cl)Cl 3L-314S c1ccc(cc1)CNC(=O)N/C=C/c2ccco2 3L-315S CNC(=O)N/C=C/c1ccco1 3L-316S CC(C)NC(=O)N/C=C/c1ccco1 3L-318S c1ccc(cc1)COC(=O)N/C=C/c2ccccc2 3L-320S c1cc(c(nc1)Sc2ccc(cc2)Cl)/C=N/O 3L-321S CO/N=C/c1cccnc1Sc2ccc(cc2)Cl 3L-322S c1ccc(cc1)/C=C/NC(=O)OCc2ccc(cc2)Cl 3L-323S COc1ccc(cc1)COC(=O)N/C=C/c2ccccc2 3L-324S c1ccc(cc1)/C=C/NC(=O)OCc2c(cccc2Cl)Cl 3L-325S c1cc(c(nc1)Sc2ccc(cc2)Cl)/C=N/OCc3ccc(cc3Cl)Cl 3L-327S c1cc(c(nc1)Sc2ccc(cc2)Cl)/C=N/OCc3ccc(c(c3)Cl)Cl 3L-328S c1cc(c(nc1)Sc2ccc(cc2)Cl)/C=N/OCc3ccc(cc3)F 3L-329S c1cc(oc1)/C=C/NC(=O)NCc2ccc(cc2)Cl 3L-330S COc1ccc(cc1)NC(=O)N/C=C/c2ccco2 3L-333S Cc1cccc(c1NC(=O)N/C=C/c2ccco2)C 3L-335S c1cc(c(nc1)Oc2ccc(cc2)Cl)C=O 3L-338S c1cc(c(nc1)Sc2ccc(cc2)Br)CO 3L-339S c1cc(cc(c1)F)CO/N=C/c2cccnc2Sc3ccc(cc3)Cl 3L-340S Cc1ccc(cc1)CO/N=C/c2cccnc2Sc3ccc(cc3)Cl 3L-341S c1ccc(cc1)Sc2c(cccn2)/C=N/O 3L-342S COc1ccc(cc1)COC(=O)N/C=C/c2ccc(cc2)Cl 3L-343S c1cc(ccc1COC(=O)N/C=C/c2ccc(cc2)Cl)Cl 3L-344S c1ccc(cc1)COC(=O)N/C=C/c2ccc(cc2)Cl 3L-345S CC(C)(C)c1ccc(cc1)COC(=O)N/C=C/c2ccc(cc2)Cl 3L-346S c1ccc(c(c1)COC(=O)N/C=C/c2ccc(cc2)Cl)Cl 3L-347S c1ccc(cc1)Sc2c(cccn2)/C=N/OCc3ccc(cc3Cl)Cl 3L-348S c1ccc(cc1)Sc2c(cccn2)/C=N/OCc3ccc(c(c3)Cl)Cl 3L-349S Cc1ccc(cc1)CO/N=C/c2cccnc2Sc3ccccc3 3L-350S c1ccc(cc1)NC(=O)OCc2cccnc2Sc3ccc(cc3)Br 3L-351S c1ccc(cc1)Sc2c(cccn2)/C=N/OCc3cccc(c3)F 3L-352S c1ccc(c(c1)Sc2c(cccn2)/C=N/OCc3ccc(cc3Cl)Cl)Cl 3L-353S c1cc(c(nc1)Sc2ccc(cc2Cl)Cl)/C=N/OCc3ccc(cc3Cl)Cl 3L-354S c1ccc(c(c1)Sc2c(cccn2)CO)Cl 3L-357S c1cc(c(nc1)Sc2ccc(cc2)Cl)CO 3L-358S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3ccccc3 3L-360S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3cccc(c3)Cl 3L-361S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)NC3CCCCC3 3L-362S COc1ccc(cc1)COC(=O)N/C=C/c2ccccc2Cl 3L-364S c1ccc(c(c1)/C=C/NC(=O)OCc2ccc(cc2)Cl)Cl 3L-365S c1ccc(c(c1)COC(=O)N/C=C/c2ccccc2Cl)Cl 3L-367S c1ccc(c(c1)/C=C/NC(=O)OCc2ccc(cc2)Br)Cl 3L-368S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3ccc(cc3)Cl 3L-371S c1cc(c(nc1)Sc2ccc(cc2)Br)COC(=O)Nc3cc(cc(c3)Cl)Cl 3L-372S c1cc(c(nc1)Sc2ccc(cc2)Br)COC(=O)Nc3ccc(cc3)Cl 3L-373S Cc1ccccc1NC(=O)OCc2cccnc2Sc3ccc(cc3)Br 3L-374S COc1ccccc1COC(=O)N/C=C/c2ccc(cc2)Cl 3L-375S c1cc(ccc1/C=C/NC(=O)Nc2ccc(cc2)Cl)Cl 3L-376S COc1ccc(cc1)NC(=O)N/C=C/c2ccc(cc2)Cl 3L-377S Cc1ccc(cc1)NC(=O)N/C=C/c2ccc(cc2)Cl 3L-378S c1cc(ccc1CNC(=O)N/C=C/c2ccc(cc2)Cl)Cl 3L-379S COc1ccccc1CNC(=O)N/C=C/c2ccc(cc2)Cl 3L-380S c1ccc(cc1)N/C=C/C=N/c2ccccc2 3L-381S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3c(cccc3C)C 3L-386S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3cc(cc(c3)Cl)Cl 3L-387S CCCNC(=O)OCc1cccnc1Sc2ccc(cc2)C 3L-388S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)NC(C)C 3L-389S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3ccccc3C 3L-390S Cc1ccc(cc1)Oc2c(cccn2)CO 3L-391S c1cc(c(nc1)Oc2ccc(cc2)Cl)CO 3L-392S Cc1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3cccc(c3)C(F)(F)F 3L-393S c1cc(ccc1COC(=O)N/C=C/c2ccc(cc2Cl)Cl)Cl 3L-394S COc1ccc(cc1)COC(=O)N/C=C/c2ccc(cc2Cl)Cl 3L-395S c1ccc(c(c1)Sc2c(cccn2)COC(=O)Nc3cc(cc(c3)Cl)Cl)Cl 3L-399S c1ccc(c(c1)Sc2c(cccn2)COC(=O)Nc3ccc(cc3)Cl)Cl 3L-400S Cc1ccccc1NC(=O)OCc2cccnc2Sc3ccc(cc3)Cl 3L-401S Cc1ccc(cc1)Oc2c(cccn2)COC(=O)Nc3ccccc3C 3L-402S Cc1ccccc1NC(=O)OCc2cccnc2Oc3ccc(cc3)Cl 3L-403S c1cc(c(nc1)Oc2ccc(cc2)Cl)COC(=O)Nc3ccc(cc3)Cl 3L-404S c1cc(c(nc1)Sc2ccc(cc2Cl)Cl)CO 3L-407S c1ccc(cc1)Sc2c(cccn2)CO 3L-408S Cc1c(c(on1)C)C(=O)N2CCCC2 3L-501S Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)Cl 3L-502S Cc1c(c(on1)C)C(=O)Nc2ccc(c(c2)Cl)Cl 3L-503S c1cc(cc(c1)C(F)(F)F)C(=O)c2c[nH]cc2c3c(cccc3Cl)F 3L-504S c1ccc(cc1)C(=O)c2c[nH]cc2c3ccc(cc3)Br 3L-506S CN(c1ccccc1)c2cc(nc(n2)c3ccccn3)CSC 3L-507S Cc1nc(cc(n1)Oc2ccccc2)CSC 3L-508S Cc1nc(cc(n1)Sc2cccc(c2)C(F)(F)F)CSC 3L-509S Cc1nc(cc(n1)NCC=C)CSC 3L-510S Cc1ccc(cc1)c2c[nH]cc2C(=O)c3ccc(c(c3)OC)OC 3L-511S c1cc(ccc1c2c[nH]cc2C(=O)c3ccc(cc3)Cl)Cl 3L-512S Cc1nc(cc(n1)Sc2ccccc2)CSC 3L-513S CSCc1cc(nc(n1)c2cccnc2)O 3L-514S CSCc1cc(nc(n1)c2ccncc2)O 3L-515S Cc1c(c(on1)C)C(=O)Nc2cc(cc(c2)Cl)Cl 3L-516S Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)Br 3L-517S Cc1c(c(on1)C)C(=O)NCC=C 3L-518S Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)F 3L-519S Cc1c(c(on1)C)C(=O)Nc2ccc(c(c2)F)F 3L-520S Cc1nc(cc(n1)N2CCOCC2)CSC 3L-521S Cc1c(c(on1)C)C(=O)Nc2cccc(c2Cl)Cl 3L-522S Cc1c(c(on1)C)C(=O)NC 3L-523S CSCc1cc(nc(n1)c2ccncc2)Cl 3L-524S COc1ccc(cc1OC)C(=O)c2c[nH]cc2c3ccc(cc3)Br 3L-525S Cc1ccc(cc1)C(=O)c2c[nH]cc2c3ccc(cc3)Br 3L-526S c1cc(cc(c1)F)c2c[nH]cc2C(=O)c3ccc(c(c3)Cl)Cl 3L-528S CSCc1cc(nc(n1)c2ccncc2)Sc3ccc(cc3)Cl 3L-530S CSCc1cc(nc(n1)c2ccncc2)Oc3ccc(cc3)Cl 3L-531S c1cc(ccc1c2c[nH]cc2C(=O)c3ccc(cc3)Cl)F 3L-533S Cc1ccc(cc1)C(=O)c2c[nH]cc2c3ccc(cc3Cl)Cl 3L-534S Cc1ccc(cc1)c2c[nH]cc2C(=O)c3ccc(cc3)Br 3L-535S CSCc1cc(nc(n1)c2ccncc2)N3CCCC3 3L-537S Cc1c(c(on1)C)C(=O)NCc2ccccc2 3L-538S CC(C)c1ccc(cc1)c2c[nH]cc2C(=O)c3ccc(cc3)Cl 3L-541S c1ccc(cc1)c2c[nH]cc2C(=O)c3ccc(cc3)Cl 3L-542S c1ccc(cc1)C(=O)c2c[nH]cc2c3cccc(c3Cl)Cl 3L-543S CSCc1cc(nc(n1)c2ccncc2)NC3CCCCC3 3L-548S CSCc1cc(nc(n1)c2ccncc2)NCc3ccccc3 3L-549S Cc1c(c(on1)C)C(=O)N(C)C 3L-550S Cc1c(c(on1)C)C(=O)N2CCN(CC2)c3ccccc3 3L-551S CSCc1cc(nc(n1)c2cccnc2)SC 3L-552S CS(=O)(=O)Cc1cc(nc(n1)c2ccccc2)Sc3ccc(cc3)Cl 3L-554S CCOC(=O)CSc1cc(nc(n1)c2ccccn2)CS(=O)(=O)C 3L-555S CS(=O)Cc1cc(nc(n1)c2ccncc2)Sc3ccccc3 3L-556S Cc1ccc(cc1)c2c[nH]cc2C(c3ccc(cc3)Cl)O 3L-560S c1ccc(cc1)C(c2c[nH]cc2c3ccc(cc3)Br)O 3L-562S c1cc(c(c(c1)Cl)c2c[nH]cc2C(c3ccc(cc3)Cl)O)Cl 3L-567S Cc1ccc(cc1)NC(=O)c2c(noc2C)C 3L-570S Cc1c(c(on1)C)C(=O)Nc2ccc(cc2Cl)Cl 3L-571S Cc1c(c(on1)C)C(=O)N2CCN(CC2)c3cccc(c3)Cl 3L-572S Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)OC 3L-573S Cc1c(c(on1)C)C(=O)Nc2ccc(cc2F)F 3L-575S Cn1c(cc(n1)CSc2ccccc2)O 3L-576S Cn1c(cc(n1)CSc2ccc(cc2)Cl)O 3L-577S Cn1c(c(c(n1)CSc2ccccc2)C=O)Cl 3L-578S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)C=O)Cl 3L-579S COC(=O)c1ccccc1Sc2cc(nc(n2)c3ccccc3)CS(=O)(=O)C 3L-582S CS(=O)Cc1cc(nc(n1)c2ccncc2)Oc3ccccc3 3L-583S CS(=O)Cc1cc(nc(n1)c2cccnc2)Cl 3L-584S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CO)Cl 3L-586S Cc1c(c(on1)C)C(=O)Nc2ccc(c(c2F)Cl)F 3L-589S Cc1c(c(on1)C)C(=O)Nc2cc(ccc2OC)OC 3L-590S Cc1ccc(cc1C)NC(=O)c2c(noc2C)C 3L-591S Cc1ccc(c(c1)C)NC(=O)c2c(noc2C)C 3L-592S Cc1cccc(c1C)NC(=O)c2c(noc2C)C 3L-593S Cc1cccc(c1NC(=O)c2c(noc2C)C)C 3L-594S Cc1c(c(on1)C)C(=O)N2CC(OC(C2)C)C 3L-595S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3ccc(cc3)Cl)Cl 3L-598S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3c(cccc3Cl)Cl)Cl 3L-599S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3ccc(cc3)Br)Cl 3L-600S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3ccc(cc3)OC)Cl 3L-601S CN(c1ccccc1)c2cc(nc(n2)c3ccccc3)CSC 3L-602S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3cccc(c3)Cl)Cl 3L-603S CS(=O)Cc1cc(nc(n1)c2cccnc2)Sc3ccccc3 3L-605S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3ccccc3Cl)Cl 3L-611S Cc1ccc(cc1)SCc2c(nn(c2Cl)C)CSc3ccc(cc3)Cl 3L-612S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3ccc(cc3Cl)Cl)Cl 3L-613S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3cccc(c3Cl)Cl)Cl 3L-614S CC(C)(C)c1ccc(cc1)SCc2c(nn(c2Cl)C)CSc3ccc(cc3)Cl 3L-615S Cc1ccccc1SCc2c(nn(c2Cl)C)CSc3ccc(cc3)Cl 3L-617S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3ccccc3)Cl 3L-618S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3ccc(cc3)F)Cl 3L-620S c1cc(cc(c1)F)c2c[nH]cc2C(=O)c3ccc(cc3)Cl 3L-621S Cc1ccc(cc1)c2c[nH]cc2C(=O)c3ccc(c(c3)Cl)Cl 3L-622S Cn1c(c(c(n1)CSc2ccc(cc2)Cl)CSc3cccc(c3)C(F)(F)F)Cl 3L-625S Cc1c(c(on1)C)C(=O)NS(=O)(=O)c2ccc(cc2)OC 3L-628S Cc1c(c(on1)C)C(=O)NS(=O)(=O)c2ccc(c(c2Cl)Cl)Cl 3L-629S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CO 3L-630S CCn1c(cc(c(c1=O)C#N)SC)c2ccccc2 3L-632S CSc1cc(n(c(=O)c1C#N)Cc2ccc(c(c2)Cl)Cl)c3ccccc3 3L-633S COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCC(=O)CC3)Cl 3L-901 C(CON)N.Cl.Cl 3L-902 c1cc(c(cc1Cl)Cl)n2c(=O)c(c(cn2)Cl)Cl 3L-903 c1cc(c(cc1Cl)Cl)n2c(=O)c(c(cn2)N3CCC(=O)CC3)Cl 3L-904 c1cc(nnc1N2CCC(CC2)C(=O)NN)Cl 3L-905 CCOC(=O)/C(=C\N)/C#N 3L-906 c1cc(c(c(c1)F)C(=O)NCCONC(=O)c2c(cccc2F)F)F 3L-907 c1cc(c(cc1Cl)Cl)n2c(=O)c(c(cn2)N3CCC(=NNC(=O)C4CCN(CC4)c5ccc(nn5)Cl)CC3)Cl 3L-908 c1cc(nnc1N2CCC(CC2)C(=O)NN=C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 3L-909 c1cc(ccc1N2CCc3c(sc(c3C#N)N)C2)[N+](=O)[O-] 3L-910 COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCc4c(sc(c4C#N)N)C3)Cl 3L-911 c1cc(nc(c1)F)N2CCc3c(sc(c3C#N)N)C2 3L-912 C(CONC(=O)N)NC(=O)N 3L-913 c1cc(ccc1N2C(=O)NC3(N2)CCN(CC3)c4cnn(c(=O)c4Cl)c5ccc(cc5Cl)Cl)Cl 3L-914 COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCC(CC3)C(=O)N)Cl 3L-915 CCOC(=O)CNC(=S)NNC(=O)C1CCN(CC1)c2ccc(nn2)Cl 3L-916 CC(=O)c1cn(c(=O)[nH]c1=O)c2cccnc2Cl 3L-917 CN(C)/C=C\1/c2ccccc2N(C1=O)c3c(cc(cn3)C(F)(F)F)Cl 3L-918 c1ccc(cc1)N2C(=O)NC3(N2)CCN(CC3)c4cnn(c(=O)c4Cl)c5ccc(cc5Cl)Cl 3L-919 c1ccn(c1)c2c(c3c(s2)CN(CC3)c4ccc(cc4)[N+](=O)[O-])C#N 3L-921 c1ccc(cc1)N2C(=O)NC3(N2)CCN(CC3)C(=O)N 3L-922 c1cc(ccc1C(=O)NCCONC(=O)c2ccc(cc2)Cl)Cl 3L-923 c1csc2n1c(c(c(=O)n2)N=O)N 3L-924 CNc1ncc(s1)C(=O)C/C=N/OC 3M-001 Cc1ccc(cc1)C\2=NN=C/C2=N\Nc3cc(cc(c3)Cl)Cl 3M-002 CNc1ncc(s1)C(=O)C/C=N/OCc2ccccc2F 3M-003 c1cc(ccc1N/N=C(\C=O)/C(=O)c2ccncc2)F 3M-005 c1cc(ccc1N/N=C(\C=O)/C(=O)c2ccncc2)Cl 3M-006 c1ccc(cc1)N/N=C(\C=O)/C(=O)c2ccncc2 3M-007 Cc1ccc(cc1)N/N=C(\C=O)/C(=O)c2ccncc2 3M-008 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)Cl)/C=O)Br 3M-009 c1cc(ccc1C(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/C=O)Br 3M-010 c1cc(ccc1C#N)OS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 3M-011 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Oc3ccc(c(c3)Cl)Cl 3M-012 Cc1cccc(c1)N/N=C(\C=O)/C(=O)c2ccc(cc2)Br 3M-013 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/C=O)Br 3M-015 CC(=O)Nc1cccc(c1)OS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 3M-016 COc1ccc(cc1)C(=O)/C(=N\Nc2ccc(cc2)C(F)(F)F)/C=O 3M-017 c1cc(ccc1C(=O)/C(=N\Nc2ccc(cc2)Cl)/C=N/N)Cl 3M-018 c1cc(sc1)C(=O)/C(=N/Nc2ccc(cc2)Cl)/C=N/N 3M-019 C/C(=N\O)/c1cnc(s1)Nc2ccccc2 3M-020 c1ccc(cc1)N/N=C(\C=N\N)/C(=O)c2ccc(cc2)Cl 3M-021 Cc1cccc(c1)N/N=C(\C=N\N)/C(=O)c2ccco2 3M-022 COc1ccc(cc1)C(=O)/C(=N/Nc2ccccc2)/C=O 3M-023 Cc1ccc(cc1)c2c(cnc(n2)N)/N=N\c3cccc(c3C)C 3M-024 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/C=N/N 3M-025 Cc1ccc(cc1)/N=N\c2cnc(nc2c3ccc(cc3)Cl)N 3M-026 c1cc(ccc1C(=O)/C(=N\Nc2ccc(cc2)F)/C=N/N)Cl 3M-027 c1ccc(cc1)N/N=C/2\C=NN=C2c3ccco3 3M-028 Cc1ccc(cc1)c2c(cnc(n2)c3ccncc3)/N=N\c4cccc(c4C)C 3M-029 Cc1ccc(cc1)C(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/C=N/O 3M-030 Cc1cccc(c1)N/N=C/2\C=NN=C2c3ccco3 3M-031 COc1ccc(cc1)C\2=NN=C/C2=N\Nc3ccc(cc3)C(F)(F)F 3M-032 COc1ccc(cc1)/N=N\c2cnc(nc2c3ccco3)N 3M-033 COc1ccc(cc1)c2c(cnc(n2)c3ccccc3)/N=N\c4ccc(cc4)C(F)(F)F 3M-034 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)F)/C=O 3M-035 c1cc(ccc1N/N=C/2\C=NN=C2c3ccncc3)Cl 3M-036 COc1ccc(cc1)C\2=NN=C/C2=N\Nc3ccccc3 3M-037 CN(C)/C=C/C(=O)c1cnc(s1)c2ccccc2 3M-038 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)OC)/C=O 3M-039 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)OC(F)(F)F)/C=O 3M-040 C/C(=N\O)/c1cnc(s1)c2ccccc2 3M-041 Cc1cccc(c1)N/N=C/2\C=NN=C2c3ccc(cc3)Br 3M-043 c1ccc(cc1)c2ncc(s2)C(=O)C/C=N/OCc3ccc(cc3)Cl 3M-044 CO/N=C/CC(=O)c1cnc(s1)c2ccccc2 3M-045 Cc1ccc(cc1)CO/N=C/CC(=O)c2cnc(s2)c3ccccc3 3M-046 c1ccc(cc1)c2ncc(s2)C(=O)C/C=N/OCc3c(cccc3Cl)Cl 3M-047 c1ccc(cc1)c2ncc(s2)C(=O)C/C=N/OCc3ccccc3Br 3M-048 c1ccc(cc1)c2ncc(s2)C(=O)C/C=N/OCc3ccc(cc3Cl)F 3M-049 Cc1ncc(c(n1)c2ccc(cc2)OC)/N=N\c3ccccc3 3M-050 Cc1cccc(c1)N/N=C(\C=N\N)/C(=O)c2ccc(cc2)Br 3M-051 c1ccc(cc1)C(=O)/C(=N/Nc2ccccc2)/C=O 3M-052 Cc1ccc(cc1)N/N=C(\C=N\N)/C(=O)c2ccc(cc2)Cl 3M-053 c1ccc(cc1)N/N=C(\C=O)/C(=O)c2ccc(cc2Cl)Cl 3M-054 c1ccc(cc1)c2ncc(s2)C(=O)/C=C/Nc3ccccc3 3M-055 Cc1ccc(c(c1)C)N/C=C/C(=O)c2cnc(s2)c3ccccc3 3M-056 c1ccc(cc1)c2ncc(s2)C(=O)/C=C/Nc3ccc(cc3)F 3M-057 c1ccc(cc1)c2ncc(s2)C(=O)/C=C/Nc3cccc(c3)C(F)(F)F 3M-058 c1ccc(cc1)c2ncc(s2)C(=O)/C=C/Nc3ccc(cc3)I 3M-059 c1ccc(cc1)c2ncc(s2)c3cc[nH]n3 3M-061 c1cc(ccc1N/N=C(\C=N\N)/C(=O)c2ccncc2)Cl 3M-062 c1ccc(cc1)c2ncc(s2)c3ccno3 3M-063 Cc1ncc(c(n1)c2ccccc2)/N=N\c3ccccc3 3M-064 c1ccc(cc1)c2ncc(s2)c3ccnc(n3)N 3M-065 c1ccc(cc1)N/N=C/2\C=NN=C2c3ccc(cc3)Cl 3M-066 c1cc(ccc1C\2=NN=C/C2=N\Nc3ccc(cc3)Cl)Cl 3M-067 CN(C)/C=C/C(=O)c1cnc(s1)c2ccc(cc2)Cl 3M-068 c1cc(ccc1C(=O)/C(=N\Nc2ccc(cc2)Cl)/C=N/N)Br 3M-069 CS/C(=N/c1ccccc1)/NCc2ccc(cc2)Cl 3M-301S CS/C(=N/c1ccccc1)/NCc2ccc(cc2Cl)Cl 3M-302S COc1cccc(c1)CN/C(=N/c2ccccc2)/NCc3cccc(c3)C(F)(F)F 3M-304S Cc1ccc(cc1)/N=C\2/c3ccccc3N(C2=O)CC=C 3M-305S C=CCN1c2ccccc2/C(=N/c3cc(cc(c3)Cl)Cl)/C1=O 3M-306S C=CCN1c2ccccc2/C(=N/c3ccc(c(c3)Cl)Cl)/C1=O 3M-308S Cc1ccc(cc1Cl)/N=C\2/c3ccccc3N(C2=O)CC=C 3M-309S C=CCN1c2ccccc2/C(=N/c3cccc(c3)[N+](=O)[O-])/C1=O 3M-310S c1ccc2c(c1)C(=O)C(=O)N2Cc3c(cccc3Cl)Cl 3M-311S Cc1ccc2c(c1)C(=O)C(=O)N2Cc3c(cccc3Cl)Cl 3M-312S C#CCN1c2ccccc2/C(=N\c3ccc(cc3F)F)/C1=O 3M-313S CN1c2ccccc2/C(=N\c3ccc(cc3)F)/C1=O 3M-314S CN1c2ccccc2/C(=N\c3ccc(cc3)Oc4ccccc4)/C1=O 3M-315S CCN(CC)/C(=N/c1ccccc1)/NCc2ccc(cc2)Cl 3M-317S c1ccc(cc1)/N=C(\NCc2ccc(cc2)Cl)/NC3CCCCC3 3M-318S CN1CCN(CC1)/C(=N/c2ccccc2)/NCc3ccc(cc3)Cl 3M-319S Cc1ccc(cc1)/N=C/2\c3ccccc3N(C2=O)C 3M-320S Cc1ccc(cc1Cl)/N=C/2\c3ccccc3N(C2=O)C 3M-321S CN1c2ccccc2/C(=N\c3ccc(cc3)OC)/C1=O 3M-322S CC(C)N1c2ccccc2/C(=N\c3ccc(cc3)OC)/C1=O 3M-323S c1ccc(cc1)/N=C(\NCc2ccc(cc2Cl)Cl)/NC3CCCCC3 3M-324S CC(C)N/C(=N/c1ccccc1)/NCc2ccc(cc2Cl)Cl 3M-325S c1ccc(cc1)/N=C(/NCc2ccc(cc2Cl)Cl)\NC3CC3 3M-327S CC(C)N1c2ccccc2/C(=N\c3ccc(cc3)Br)/C1=O 3M-328S Cc1cc(cc(c1)/N=C/2\c3ccccc3N(C2=O)C(C)C)C 3M-329S Cc1ccc(cc1C)/N=C/2\c3ccccc3N(C2=O)C(C)C 3M-330S Cc1cc(cc(c1)/N=C/2\c3ccccc3N(C2=O)Cc4ccccc4Cl)C 3M-331S c1ccc(c(c1)CN2c3ccccc3/C(=N\c4ccc(cc4)F)/C2=O)Cl 3M-335S c1ccc(c(c1)CN2c3ccccc3/C(=N\c4cccc(c4)C(F)(F)F)/C2=O)Cl 3M-336S Cn1c2c(cc(s2)c3nnc(n3c4ccccc4)S)c(n1)C(F)(F)F 3M-337S c1cc(ccc1NC(=S)Nc2ccc(cc2)Cl)F 3M-338S CS/C(=N\c1ccc(cc1)Cl)/Nc2ccc(cc2)F 3M-340S Cn1c2c(cc(s2)CSc3c(cccc3Cl)Cl)c(n1)C(F)(F)F 3M-343S Cn1c2c(cc(s2)CSc3ccc(cc3)Br)c(n1)C(F)(F)F 3M-344S Cn1c2c(cc(s2)c3nnc(n3c4ccccc4)SC)c(n1)C(F)(F)F 3M-346S Cn1c2c(cc(s2)c3nnc(n3c4ccccc4)SCC=C)c(n1)C(F)(F)F 3M-347S Cn1c2c(cc(s2)COc3ccc(cc3Cl)Cl)c(n1)C(F)(F)F 3M-348S CC(C)(C)c1ccc(cc1)OCc2cc3c(nn(c3s2)C)C(F)(F)F 3M-349S Cn1c2c(cc(s2)COc3ccc(cc3)OC)c(n1)C(F)(F)F 3M-350S Cn1c2c(cc(s2)COc3ccc(cc3)F)c(n1)C(F)(F)F 3M-351S CC(C)n1cc(c(=O)c2c1cccc2)C(=O)O 3M-352S c1ccc2c(c1)/C(=N\c3ccc(cc3)Cl)/C(=O)N2Cc4ccc(cc4)Cl 3M-353S COc1ccc(cc1)/N=C/2\c3ccccc3N(C2=O)Cc4ccc(cc4)Cl 3M-354S c1ccc2c(c1)/C(=N\c3ccc(cc3)Cl)/C(=O)N2Cc4c(cccc4Cl)Cl 3M-355S c1ccc2c(c1)/C(=N\c3ccc(cc3)C(F)(F)F)/C(=O)N2Cc4c(cccc4Cl)Cl 3M-356S c1ccc2c(c1)/C(=N\c3ccc(cc3)F)/C(=O)N2Cc4c(cccc4Cl)Cl 3M-357S c1ccc(cc1)C(=O)COc2ccccc2[N+](=O)[O-] 3M-358S c1ccc(cc1)C23c4ccccc4C(=O)N2CCN3C(=O)c5ccc(cc5)F 3M-501S Cc1ccc(cc1)C(=O)N2CCN3C2(c4ccccc4C3=O)c5ccccc5 3M-502S Cn1c(cnc1SCc2ccccc2)CO 3M-504S c1ccc(cc1)Cn2c(cnc2SCc3ccc(cc3)Cl)CO 3M-505S c1ccc(cc1)Cn2c(cnc2SCc3ccccc3)CO 3M-506S CSc1ncc(n1Cc2ccccc2)CO 3M-507S C=CCSc1ncc(n1Cc2ccccc2)CO 3M-508S CCOC(=O)CSc1ncc(n1Cc2ccccc2)CO 3M-509S Cc1cccc(c1)CSc2ncc(n2C)CO 3M-511S Cn1c(cnc1SCc2ccc(cc2)[N+](=O)[O-])CO 3M-512S c1ccc(cc1)C23c4ccccc4C(=O)N2CCN3C(=O)C5CC5 3M-513S c1ccc(cc1)C(=O)Nc2nc(ns2)O 3M-519S c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)Cl 3M-520S c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)Br 3M-521S c1cc2c(cc3c(c2nc1)OCN(C3)Cc4ccc(cc4)Cl)Cl 3M-524S c1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)c3ccccc3 3M-527S c1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)C3CC3 3M-528S c1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)c3cccc(c3)C(F)(F)F 3M-529S c1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)c3cccs3 3M-530S CC(C)CC(=O)n1c(=O)nc(s1)NC(=O)c2ccccc2 3M-531S Cn1c(c(c(n1)c2ccccc2)C(=O)N3CCOCC3)Cl 3M-532S CNC(=O)c1c(nn(c1Cl)C)c2ccccc2 3M-533S Cn1c(c(c(n1)c2ccccc2)C(=O)Nc3ccc(cc3)C(F)(F)F)Cl 3M-541S Cn1c(c(c(n1)c2ccccc2)C(=O)Nc3ccc(c(c3)Cl)Cl)Cl 3M-542S Cc1nc(cc(n1)O)COC 3M-543S COCc1cc(nc(n1)S)O 3M-544S Cc1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)C3CC3 3M-545S Cc1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)CC(C)C 3M-546S Cc1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)c3ccccc3Cl 3M-547S Cc1ccc(cc1)C(=O)Nc2nc(=O)n(s2)C(=O)c3ccccc3C 3M-548S Cc1nc(cs1)CSc2ccccc2C(=O)OC 3M-550S Cc1nc(cs1)CSc2ccc(cc2)Br 3M-551S Cc1nc(cs1)CSc2cccc(c2Cl)Cl 3M-552S Cn1c(c(c(n1)c2ccccc2)C(=O)N(C)C)Cl 3M-563S COC(=O)c1c(ccs1)NC(=S)NC(=O)c2ccccc2 3M-564S Cc1nc(cs1)CSc2c(cccc2Cl)Cl 3M-565S Cc1nc(cs1)COC 3M-566S COCc1cc(nc(n1)SCc2ccc(cc2)Cl)Cl 3M-570S CC1COc2ccccc2N1S(=O)(=O)c3ccccc3 3M-575S CC1COc2ccccc2N1C(=O)c3ccc(nc3)Cl 3M-576S CN(C)c1nc(n(n1)C(=O)c2ccc(cc2)[N+](=O)[O-])N(C)C 3M-700 CN(C)c1nc(n(n1)C(=O)c2ccccc2Cl)N(C)C 3M-701 CN(C)c1nc(n(n1)C(=O)c2ccc(cc2)C(F)(F)F)N(C)C 3M-702 Cc1ccc(cc1)C(=O)n2cc(c(n2)C(F)(F)F)CCCOC(=O)c3ccc(cc3)C 3M-703 CN(C)c1nc(n(n1)C(=O)c2cccs2)N(C)C 3M-704 CN(C)c1nc(n(n1)C(=O)c2c(cccc2Cl)Cl)N(C)C 3M-705 CN(C)c1nc(n(n1)S(=O)(=O)c2ccc(cc2)OC)N(C)C 3M-706 Cc1ccc(cc1)C(=O)n2c(nc(n2)N(C)C)N(C)C 3M-707 CN(C)c1nc(n(n1)C(=O)c2ccc(cc2Cl)Cl)N(C)C 3M-708 CC1(CN(C1=O)c2cccc(c2)OCc3ccc(cc3)[N+](=O)[O-])C 3M-709 COc1ccc(cc1)C2C3=C(CC(CC3=O)c4c(cccc4Cl)F)Nc5ccccc5N2 3M-710 CCOC(=O)C1=C(NC2=C(C1c3ccc(cc3)F)C(=O)CCC2)C(F)(F)F 3M-713 CCOC(=O)C1=C(NC2=C(C1c3ccccc3C(F)(F)F)C(=O)CC(C2)c4ccc(cc4)F)C 3M-714 CN(C)c1nc(n(n1)C(=O)c2ccc(cc2)OC)N(C)C 3M-715 CN(C)c1nc(n(n1)C(=O)c2ccccc2F)N(C)C 3M-716 CN(C)c1nc(n(n1)C(=O)c2ccc(cc2)F)N(C)C 3M-717 CC1(CC2=C(C(Nc3ccccc3N2)c4cccs4)C(=O)C1)C 3M-718 CN(C)c1nc(n(n1)S(=O)(=O)c2ccc(cc2)Br)N(C)C 3M-720 CC1(CC2=C(CNc3ccccc3N2)C(=O)C1)C 3M-721 Cc1ccc(cc1)S(=O)(=O)n2c(nc(n2)N(C)C)N(C)C 3M-722 CN(C)c1nc(n(n1)S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)N(C)C 3M-723 Cc1ccc(cc1)S(=O)(=O)N/N=C\2/CCCc3c2cco3 3M-724 CC1(CC2=C(C(Nc3ccccc3N2)c4ccco4)C(=O)C1)C 3M-726 CN(C)c1nc(n(n1)S(=O)(=O)c2cccs2)N(C)C 3M-727 CN(C)c1nc(n(n1)S(=O)(=O)c2ccc(cc2)F)N(C)C 3M-728 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)[N+](=O)[O-])C(=O)C1)C 3M-729 CN(C)c1nc(n(n1)S(=O)(=O)c2ccc(cc2Cl)Cl)N(C)C 3M-731 CN(C)c1nc(n(n1)S(=O)(=O)c2ccc3ccccc3c2)N(C)C 3M-732 CN(C)c1nc(n(n1)S(=O)(=O)c2cc(ccc2Cl)Cl)N(C)C 3M-733 CCOC(=O)C1=C(NC2=C(C1c3ccco3)C(=O)CCC2)C 3M-734 CN1C(=O)c2ccccc2/C(=N/Nc3ccc(cc3)/N=N/c4ccccc4)/C1=O 3M-735 CCOC(=O)C(Cc1ccccc1)N2CC(C2=O)(C)C 3M-737 c1ccc2c(c1)NCC3=C(N2)CC(CC3=O)c4ccc(cc4)F 3M-740 CC(=O)/C(=N/O)/C(=O)Nc1ccccc1 3M-742 C/C(=N\Nc1ccccc1)/C(=N/O)/C(=O)Nc2ccccc2 3M-743 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccc(cc4)Cl)C(=O)CCC3 3M-744 Cc1nnc2n1nc(cc2)Cl 3M-746 C/C(=N\Nc1ccc(cc1)Cl)/C(=N/O)/C(=O)Nc2ccccc2 3M-747 CCO.Cc1cc2c(cc1C)NC3=C(C(N2)c4ccc(cc4)Br)C(=O)CCC3 3M-748 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)N/N=C/c4ccccc4C(F)(F)F 3M-900 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)NNC(=O)Nc4cccc(c4)C(F)(F)F 3M-901 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)NNC(=S)Nc4cccc(c4)C(F)(F)F 3M-902 c1cc(c2ncc(n2c1)c3ccc(cc3)Cl)N 3M-903 Cc1ccc(cc1)C(=O)Nc2cccn3c2ncc3c4ccc(cc4)Cl 3M-904 Cc1ccc(cc1)CN2C(=C(CCC2=O)C#N)C 3M-906 CC1=C(C(CC(=O)N1)/C=N/OCc2ccc(cc2)Cl)C#N 3M-907 CC1=C(C(CC(=O)N1)/C=N/N(C)c2c(cc(cn2)C(F)(F)F)Cl)C#N 3M-908 CC1=C(C(CC(=O)N1)/C=N/OC)C#N 3M-909 CN(C)/C=N/C(=O)c1c(c2cc(ccc2n1Cc3ccc(cc3)[N+](=O)[O-])Cl)c4ccccc4 3M-910 c1ccc2c(c1)ccc3c2/C(=N\OCc4ccc(cc4)Cl)/CO3 3M-911 CC1=C(/C(=C/Nc2cc(c(c(c2)OC)OC)OC)/CC(=O)N1)C#N 3M-912 CC1=C(C(CC(=O)N1)/C=N/O)C#N 3M-913 CC1=C(/C(=C/Nc2cccc(c2)Cl)/CC(=O)N1)C#N 3M-914 c1ccc2c(c1)ccc3c2/C(=N\OCc4cccc(c4)C(F)(F)F)/CO3 3M-915 c1ccc2c(c1)ccc3c2/C(=N\OCCOc4cccc(c4)C(F)(F)F)/CO3 3M-916 c1cc(c2ncc(n2c1)c3ccc(c(c3)Cl)Cl)N 3M-917 CCOC(=O)C1=NN(C2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F)C(=O)Nc4ccccc4 3M-918 Cc1c(c(cc(=O)[nH]1)C#N)C#N 3M-919 CCOC(=O)C1C2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F 3M-920 c1cc(c2ncc(n2c1)c3ccc(c(c3)Cl)Cl)NC(=O)c4cccs4 3M-921 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccn3c2ncc3c4ccc(c(c4)Cl)Cl 3M-922 c1cc(cc(c1)NC(=O)Nc2cccn3c2ncc3c4ccc(c(c4)Cl)Cl)C(F)(F)F 3M-923 CCOC(=O)C1C2C1C(=O)N(C2=O)c3ccc(cc3)Cl 3M-924 c1ccc2c(c1)ccc3c2C(=O)/C(=C/Nc4cccc(c4)C(F)(F)F)/O3 3M-926 CCOC(=O)C1=NN(C2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F)C(=O)Nc4cccc(c4)C(F)(F)F 3M-927 COc1ccc(cc1)C(=O)/C=C/Nc2cccn3c2ncc3c4ccc(c(c4)Cl)Cl 3M-928 COc1ccc(cc1)S(=O)(=O)Nc2cccn3c2ncc3c4ccc(c(c4)Cl)Cl 3M-929 CCOC(=O)C1=NN(C2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F)C(=O)Nc4ccc(cc4)OC 3M-930 COc1ccc(cc1)N/C=C\2/C(=O)c3c4ccccc4ccc3O2 3M-931 c1ccc2c(c1)ccc3c2c4c(o3)cno4 3M-933 c1ccc2c(c1)ccc3c2C(=O)C(O3)/C=N\OCc4ccc(cc4)Cl 3M-934 CCOC(=O)C1C(C1C(=O)NN)C(=O)Nc2cccc(c2)C(F)(F)F 3M-935 CCOC(=O)C1C(C1C(=O)NN)C(=O)Nc2ccc(cc2)Cl 3M-936 CCOC(=O)C1C2C1C(=O)N(C2=O)N(C)c3c(cc(cn3)C(F)(F)F)Cl 3M-937 CCOC(=O)C1=NN(C2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F)C(=O)NC4CCCCC4 3M-938 CCOC(=O)C1C(C1C(=O)N2CCCC2)C(=O)Nc3cccc(c3)C(F)(F)F 3M-939 Cc1cc(n2cc(c(c2n1)C#N)c3c(ccs3)Cl)C 3M-940 CCOC(=O)C1C(C1C(=O)OCC)C(=O)Nc2cccc(c2)C(F)(F)F 3M-941 COC(=O)c1ccncc1C(=O)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 3M-942 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2cnccc2C(=O)OC 3M-943 CCOC(=O)NC(=O)/C(=C/Nc1cc(ccc1N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F)/C#N 3M-944 c1c(cnc(c1Cl)N2CCN(CC2)CCO)C(F)(F)F 3M-945 CCOC(=O)C1C(C1C(=O)NC(C)C)C(=O)Nc2cccc(c2)C(F)(F)F 3M-946 Cc1ccc(cc1)C(=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3M-949 c1cc(ccc1C(=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 3M-950 c1cc(ccc1C(=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)F 3M-951 c1cc(cc(c1)C(F)(F)F)C(=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3M-952 c1cc(sc1)C(=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 3M-953 c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Cl 3N-001 C/C(=N\NC(=O)N)/c1ccc(cc1)OC 3N-002 c1cc(c(c(c1)Cl)C2CC2C(=O)c3ccc(cc3)F)F 3N-003 C/C(=N\NC(=O)N)/c1ccc(cc1)Cl 3N-004 C/C(=N\NC(=O)N)/c1ccccn1 3N-005 c1cc(ccc1C2CC2/C(=N/O)/c3ccc(cc3)Br)Cl 3N-006 Cc1c(ccc(=O)[nH]1)C(=O)C 3N-007 c1cc(ccc1CO/N=C(\c2ccc(cc2)Br)/C3CC3c4ccc(cc4)Cl)[N+](=O)[O-] 3N-008 CC(=O)c1ccc(=O)[nH]c1/C=C/N(C)C 3N-009 C/C(=N\NC(=O)N)/c1ccc(cc1)F 3N-010 c1cc(ccc1C2CC2/C(=N/OC(=O)C3CC3)/c4ccc(cc4)Br)Cl 3N-011 Cc1c2ccc(=O)[nH]c2ccn1 3N-012 c1cc(ccc1C2CC2/C(=N/OC(=O)c3ccc(cc3)F)/c4ccc(cc4)Br)Cl 3N-013 c1cc(ccc1C2CC2/C(=N/OC(=O)c3ccc(c(c3)Cl)Cl)/c4ccc(cc4)Br)Cl 3N-014 Cc1ccc(cc1)C(=O)O/N=C(\c2ccc(cc2)Br)/C3CC3c4ccc(cc4)Cl 3N-015 Cc1ccc(cc1)CNS(=O)(=O)C 3N-017 c1ccc(cc1)C(=O)O/N=C(\c2ccc(cc2)Br)/C3CC3c4ccc(cc4)Cl 3N-018 c1ccc(cc1)C2CC2/C(=N/O)/c3ccccn3 3N-019 Cc1ccc(cc1)CN(C(=O)OC(C)(C)C)S(=O)(=O)C 3N-020 c1cc(ccc1C(=O)/C=C/c2ccncc2)Oc3c(cc(cn3)C(F)(F)F)Cl 3N-023 c1ccn(c1)c2c(cccc2F)F 3N-024 c1cc(cc(c1)[N+](=O)[O-])C(=O)O/N=C(\c2ccc(cc2)Br)/C3CC3c4ccc(cc4)Cl 3N-026 CCOC(=O)c1ccc(=O)[nH]c1C 3N-028 c1cc(c(c(c1)Cl)C2CC2/C(=N\O)/c3ccc(cc3)F)F 3N-029 COc1ccc(cc1)/C=C/C(=O)c2ccccn2 3N-030 Cc1ccc(cc1)CNS(=O)(=O)/C=C/c2ccc(cc2)Cl 3N-031 Cc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)F 3N-032 c1ccc(cc1)C2CC2C(=O)c3ccc(cc3)Cl 3N-033 Cc1ccc(cc1)CNS(=O)(=O)/C=C/c2ccc(cc2)C(C)C 3N-034 Cc1ccc(cc1)CNS(=O)(=O)/C=C/c2ccncc2 3N-035 CCOC(c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Br)OCC 3N-036 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Br)C=O 3N-037 Cc1ccc(cc1)C2CC2C(=O)c3ccc(cc3)F 3N-038 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)F)/C=C/C(=O)c3ccc(cc3)Br 3N-039 c1cc(ccc1NC(=O)/C=C/C(=O)O)Br 3N-040 Cc1c2ccc(nc2ccn1)Cl 3N-041 c1cc2c(cc1/C=C/C(=O)c3ccc(c(c3)[N+](=O)[O-])Cl)OCO2 3N-042 c1cc(ccc1N2C(=O)C=CC2=O)Br 3N-043 c1cc2c(cc1C3CC3C(=O)c4ccc(c(c4)[N+](=O)[O-])Cl)OCO2 3N-044 c1ccc2c(c1)nc(c3n2ccc3)N4CCOCC4 3N-045 c1cc2c(c(c1)F)n3cccc3c(=O)[nH]2 3N-046 COc1ccc(cc1)C2CC2C(=O)c3ccccn3 3N-047 Cc1c2ccc(nc2ccn1)N3CCCCC3 3N-048 c1ccc2c(c1)nc(c3n2ccc3)Oc4ccc(c(c4)Cl)Cl 3N-050 c1cc2c(c(c1)F)n3cccc3c(n2)Cl 3N-051 CN(C)c1ccc(cc1)/C=N/NC(=S)N 3N-052 Cc1c2ccc(nc2ccn1)Oc3ccc(cc3)OC 3N-054 c1cc(ccc1C2CC2C(=O)c3ccc(cc3)F)C4CC4C(=O)c5ccc(cc5)Br 3N-055 c1cc(c(c(c1)Cl)C2CC2/C(=N/OCc3ccc(cc3Cl)Cl)/c4ccc(cc4)F)F 3N-056 CCCO/N=C(\c1ccc(cc1)[N+](=O)[O-])/C2CC2c3ccc(cc3)Cl 3N-058 c1ccc2c(c1)nc(c3n2ccc3)Oc4cccc(c4)C(F)(F)F 3N-059 COc1cccc(c1)/C(=N/O)/C2CC2c3ccc(cc3)Cl 3N-060 c1cc(c(c(c1)Cl)CO/N=C(\c2ccc(cc2)Br)/C3CC3c4ccc(cc4)Cl)F 3N-063 Cc1ccc(cc1)C2CC2/C(=N/O)/c3ccc(cc3)F 3N-064 COc1ccc(cc1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 3N-301S c1ccc(c(c1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3)C(F)(F)F 3N-302S c1cc(c(cc1Cl)Cl)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 3N-304S Cn1c2ccc(cc2c(c1Sc3ccc(cc3)Br)C=O)[N+](=O)[O-] 3N-305S CC(C)c1ccc(cc1)Sc2c(c3cc(ccc3n2C)[N+](=O)[O-])C=O 3N-306S Cn1c2ccccc2c(c1Sc3ccc(cc3)Br)C=O 3N-308S Cn1c2ccccc2c(c1Sc3ccc(cc3)Cl)C=O 3N-309S Cc1ccc(cc1)Sc2c(c3ccccc3n2C)C=O 3N-310S Cc1ccc(cc1)Oc2c(c3ccccc3n2C)C=O 3N-311S Cc1ccccc1C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 3N-312S c1ccc(c(c1)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3)Cl 3N-313S c1cc(cc(c1)Cl)C(=O)Nc2[nH]c(=O)c3c(n2)CCCC3 3N-315S Cc1ccc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C 3N-316S Cn1c2ccccc2c(c1Sc3c(cccc3Cl)Cl)C=O 3N-317S Cn1c2ccccc2c(c1Sc3ccccc3Cl)C=O 3N-318S Cn1c2ccccc2c(c1SCc3cccc(c3)C(F)(F)F)C=O 3N-319S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)C=O 3N-320S CC(C)C(=O)Nc1[nH]c(=O)c2c(n1)CCCC2 3N-323S CC(=O)Nc1[nH]c(=O)c2c(n1)CCCC2 3N-324S Cn1c2ccccc2c(c1Sc3cccc(c3)C(F)(F)F)C=O 3N-325S Cn1c2ccccc2c(c1Sc3ccc(cc3)OC)C=O 3N-326S Cc1cccc(c1)Sc2c(c3ccccc3n2C)C=O 3N-327S Cn1c2ccccc2c(c1SCc3ccc(cc3)Cl)C=O 3N-328S CCCC(=O)Nc1[nH]c(=O)c2c(n1)CCCC2 3N-329S CC(C)CC(=O)Nc1[nH]c(=O)c2c(n1)CCCC2 3N-330S CC(C)(C)C(=O)Nc1[nH]c(=O)c2c(n1)CCCC2 3N-331S CC(=O)CCC(=O)c1ccc(cc1)Cl 3N-332S Cn1c2ccccc2c(c1Oc3ccc(cc3)Cl)C=O 3N-333S Cn1c2ccccc2c(c1Oc3ccc(cc3)OC)C=O 3N-334S Cn1c2ccccc2c(c1Oc3ccc(cc3)F)C=O 3N-335S Cn1c2ccccc2c(c1Oc3cccc(c3)C(F)(F)F)C=O 3N-336S c1csc2c1C(=O)CCS2(=O)=O 3N-337S Cc1ccc(n1c2cc(ccc2OC)OC)c3ccc(cc3)S(=O)(=O)C 3N-338S Cc1c(cc(n1c2cc(ccc2OC)OC)c3ccc(cc3)S(=O)(=O)C)C(=O)C(F)(F)F 3N-339S C1CCc2c(c(=O)[nH]c(n2)NC(=O)C3CC3)C1 3N-340S CCC(=O)Nc1[nH]c(=O)c2c(n1)CCCC2 3N-341S CCCCC(=O)Nc1[nH]c(=O)c2c(n1)CCCC2 3N-342S Cc1c(cc(n1c2cc(ccc2OC)OC)c3ccc(cc3)S(=O)(=O)C)C=O 3N-344S Cc1c(cc(n1c2cc(ccc2OC)OC)c3ccc(cc3)S(=O)(=O)C)/C=N/c4ccc(cc4)OC 3N-345S Cn1c2ccccc2c(c1Oc3ccccc3)C=O 3N-348S Cc1cccc(c1C)Oc2c(c3ccccc3n2C)C=O 3N-349S Cc1cccc(c1)Oc2c(c3ccccc3n2C)C=O 3N-350S Cn1c2ccccc2c(c1Oc3ccc(cc3F)F)C=O 3N-351S Cn1c2ccccc2c(c1Oc3cc(c(cc3Cl)Cl)Cl)C=O 3N-352S Cc1ccc(c(c1)[N+](=O)[O-])Oc2c(c3ccccc3n2C)C=O 3N-353S c1ccc(cc1)N/N=C/2\CCS(=O)(=O)c3c2ccs3 3N-355S Cn1c2ccccc2c(c1OC)C=O 3N-356S CCSc1c(c2ccccc2n1C)C=O 3N-358S Cc1c(nc(c(c1c2ccccc2)C(=O)N)N)C 3N-359S Cc1cccc2c1nc(cc2C)O 3N-501S c1ccn2c(c1)nc(c2CN3CCN(CC3)c4ccc(c(c4)Cl)Cl)c5ccc(cc5)Cl 3N-503S c1ccn2c(c1)nc(c2CN3CCN(CC3)c4cccc(c4)Cl)c5ccc(cc5)Cl 3N-504S Cc1cccc2c1nc(cc2C)Cl 3N-508S Cc1cccc2c1nc(cc2C)Sc3ccc(cc3)Cl 3N-509S Cc1cccc2c1nc(cc2C)Oc3cccc(c3)C(F)(F)F 3N-510S Cc1cccc2c1nc(cc2C)N3CCOCC3 3N-511S c1cc(ccc1c2c(n3cc(ccc3n2)Cl)CN4CCOCC4)Cl 3N-512S c1cc(ccc1c2c(n3cc(ccc3n2)Cl)CN4CCSCC4)Cl 3N-513S c1ccc(c(c1)N2CCN(CC2)Cc3c(nc4n3cc(cc4)Cl)c5ccc(cc5)Cl)F 3N-514S c1cc(ccc1c2c(n3cc(ccc3n2)Cl)CN4CCCCC4)Cl 3N-515S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3Cl)Cl 3N-519S Cc1cccc2c1nc(cc2C(F)(F)F)O 3N-521S Cn1c(cc(n1)c2ccccc2)OCC(=O)N(Cc3ccccc3)c4ccc(cc4)OC 3N-522S Cc1cccc2c1nc(cc2C(F)(F)F)Cl 3N-523S CCOC(=O)C1CSC2(N1)CCC(CC2)c3ccccc3 3N-524S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3)F 3N-525S c1ccc(c(c1)/C=C/c2nc3ccccc3s2)Cl 3N-526S COc1ccc(cc1)/C=C/c2nc3ccccc3s2 3N-527S c1c(c(c(=O)[nH]c1C2CC2)C#N)C(F)(F)F 3N-528S c1ccc2c(c1)nc(s2)/C=C/c3cccc(c3)C(F)(F)F 3N-529S c1ccc2c(c1)nc(s2)/C=C/c3cccc(c3Cl)Cl 3N-530S COc1ccc(cc1)Sc2c(c(nn2c3ccccc3)C(=O)OC)/C=N/O 3N-531S CN(C)Cc1c(nc2n1cccc2)c3ccc(cc3)Cl 3N-532S c1ccc(c(c1)Cn2c(=O)c3ccccc3sc2=O)F 3N-533S c1ccc2c(c1)c(=O)n(c(=O)s2)Cc3cccc(c3)Cl 3N-534S COc1cccc(c1)Cn2c(=O)c3ccccc3sc2=O 3N-535S CC(COC)n1c(=O)c2ccccc2sc1=O 3N-536S c1ccc2c(c1)c(=O)n(c(=O)s2)CCN3CCOCC3 3N-537S c1ccc(c(c1)Cn2c(=O)c3ccccc3sc2=O)C(F)(F)F 3N-538S c1ccc2c(c1)c(=O)n(c(=O)s2)Cc3cccc(c3)C(F)(F)F 3N-539S Cc1ccccc1Cn2c(=O)c3ccccc3sc2=O 3N-540S Cc1ccc2nc(c(n2c1)CN3CCOCC3)c4ccccc4 3N-544S Cc1ccc2nc(c(n2c1)CN3CCSCC3)c4ccccc4 3N-545S Cc1ccc2nc(c(n2c1)CN3CCN(CC3)c4ccccc4F)c5ccccc5 3N-546S Cc1ccc2nc(c(n2c1)CN3CCN(CC3)c4cccc(c4)Cl)c5ccccc5 3N-547S c1ccc(cc1)CN2CCN(CC2)Cc3c(nc4n3cc(cc4)Cl)c5ccc(cc5)Cl 3N-548S COc1ccc(cc1)c2c(n3ccccc3n2)CN4CCN(CC4)c5ccccc5F 3N-550S CN(C)Cc1c(nc2n1cc(cc2)Cl)c3ccc(cc3)Cl 3N-551S COC(=O)c1c(c(n(n1)c2ccccc2)Sc3ccc(cc3)Cl)/C=N/O 3N-552S COC(=O)c1ccccc1Sc2c(c(nn2c3ccccc3)C(=O)OC)/C=N/O 3N-553S Cc1ccc(cc1)Sc2c(c(nn2c3ccccc3)C(=O)OC)/C=N/O 3N-554S c1ccc2c(c1)nc(o2)/C=C/c3cccc(c3)C(F)(F)F 3N-556S Cc1cc(nc2c1cc(cc2)Cl)O 3N-560S Cc1cc(nc2c1cc(cc2)Cl)Cl 3N-561S COC(=O)c1c(c(n(n1)c2ccccc2)Sc3ccc(cc3)Cl)C#N 3N-562S CCOC(=O)C1CSC2(N1C(=O)c3ccc(cc3)Cl)CCC(CC2)c4ccccc4 3N-565S c1ccc2c(c1)nc(o2)/C=C/c3ccc(cc3)F 3N-566S COc1ccc(cc1)/C=C/c2nc3ccccc3o2 3N-567S CN(C)c1ccc(cc1)/C=C/c2nc3ccccc3o2 3N-568S c1ccc2c(c1)nc(o2)/C=C/c3ccc(cc3Cl)Cl 3N-569S Cc1cc(ccc1O/C(=C/OC)/C(=O)OC)Cl 3N-570S c1ccc2c(c1)nc(o2)/C=C/c3cccc(c3)Cl 3N-573S Cc1cccc2c1nc(cc2C(F)(F)F)Sc3ccc(cc3)Cl 3N-576S Cc1cccc2c1nc(cc2C)Sc3cccc(c3)C(F)(F)F 3N-577S Cc1cccc2c1nc(cc2C)Oc3ccc(cc3)OC 3N-580S Cc1cccc2c1nc(cc2C)N3CCN(CC3)C 3N-581S CC(C)(C)c1ccc(cc1)/C=C/c2nc3ccccc3o2 3N-586S c1ccc2c(c1)nc(o2)/C=C/c3c(cccc3Cl)F 3N-587S c1ccc2c(c1)nc(o2)/C=C/c3cccc(c3)Br 3N-588S c1ccc2c(c1)nc(o2)/C=C/c3ccccn3 3N-589S c1cc(ccc1C(=O)CC(=O)C(F)(F)F)Cl 3N-590S COC(=O)c1c(c(n(n1)c2ccccc2)Sc3ccccc3)/C=N/O 3N-592S Cc1cccc2c1nc(cc2C)Oc3ccc(cc3F)F 3N-593S Cc1cccc2c1nc(cc2C)N3CCCC3 3N-594S COC(=O)c1c(c(n(n1)c2ccccc2)Sc3ccc(cc3)Br)/C=N/O 3N-595S COC(=O)c1c(c(n(n1)c2ccccc2)Sc3cccc(c3)C(F)(F)F)/C=N/O 3N-596S c1ccc(cc1)C(=O)c2c(cc(=O)n(n2)c3ccc(cc3)Cl)C(F)(F)F 3N-600S Cc1cc(nc2c1cccc2)O 3N-601S COC(=O)C(=O)CC(=O)c1ccc(cc1)Cl 3N-606S COC(=O)c1cc(n(n1)c2ccc(cc2)S(=O)(=O)N)c3ccc(cc3)Cl 3N-607S COC(=O)c1cc(n(n1)c2ccc(cc2)Cl)c3ccc(cc3)Cl 3N-608S COC(=O)c1cc(n(n1)c2ccccc2)c3ccc(cc3)Cl 3N-609S COC(=O)c1ccc(cc1)COc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 3N-700 c1ccc2cc(ccc2c1)S(=O)(=O)Oc3ccc(cc3)Cc4c(cc(cn4)C(F)(F)F)Cl 3N-702 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 3N-703 Cc1c2c(nc(n1)SC)N(CC2)c3ccc(cc3)C(C)C 3N-704 COc1ccc(cc1)/C=C/2\C(=O)NCC(=O)N2 3N-705 c1cnc(nc1c2cc(sc2Cl)Cl)S 3N-706 C/C(=C/C(=O)C(F)(F)F)/Nc1ccc(cc1)OC(F)(F)F 3N-708 C/C(=C\C(=O)C(F)(F)F)/Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F 3N-709 Cc1c2c(nc(n1)SCc3ccccc3)N(CC2)c4ccccc4 3N-710 CC(=O)N1CC(=O)N/C(=C/c2ccc(cc2)N(C)C)/C1=O 3N-711 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1)OC(F)(F)F 3N-712 COc1ccc(cc1)/C=C/2\C(=O)NCC(=O)N2Cc3ccccc3 3N-713 Cc1cccc(c1)N2CCc3c2nc(nc3C)SC 3N-715 Cc1c2c(nc(n1)SCc3ccccc3)N(CC2)c4cccc(c4)OC 3N-716 CC(=O)N1CC(=O)N/C(=C/c2ccc(cc2)F)/C1=O 3N-718 c1ccc(cc1)/C=C/2\C(=O)NCC(=O)N2 3N-719 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCC3CC3(Cl)Cl 3N-723 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 3N-724 c1cc(oc1)/C=C\2/C(=O)NCC(=O)N2 3N-725 CN(C)c1ccc(cc1)/C=C/2\C(=O)NCC(=O)N2 3N-728 c1cc(sc1)/C=C\2/C(=O)NCC(=O)N2 3N-729 Cc1c2c(nc(n1)SC)N(CC2)c3ccc(cc3)O 3N-731 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F 3N-732 c1cc(ccc1/C=C/2\C(=O)NCC(=O)N2)F 3N-733 COC(=O)CSCCC(=C(F)F)F 3N-734 CCOc1ccc(cc1)N2CCc3c2nc(nc3C)SC 3N-735 Cc1c2c(nc(n1)SC)N(CC2)c3cccc(c3)SC 3N-736 Cc1c(c(=O)[nH]c(=O)[nH]1)CCO 3N-737 Cc1c2c(nc(n1)SC)N(CC2)c3ccc(c(c3)Cl)Cl 3N-738 Cc1c2c(nc(n1)SC)N(CC2)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl 3N-739 CC(=O)N1CC(=O)N(/C(=C/c2ccc(cc2)OC)/C1=O)C 3N-740 CCCCOc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 3N-741 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OS(=O)(=O)c3ccc(cc3)Br 3N-742 c1ccc(c(c1)S(=O)(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl 3N-743 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 3N-744 CC(C)(C)NC(=O)C1CC2CCCCC2CN1 3N-745 CC(C)(C)NC(=O)C1Cc2ccccc2CN1 3N-746 CN\1C(=O)CNC(=O)/C1=C\c2ccc(cc2)OC 3N-747 CC(=O)N1CC(=O)N(/C(=C/c2ccc(cc2)OC)/C1=O)Cc3ccc(cc3)F 3N-748 c1ccc(cc1)S(=O)(=O)c2c(cc(cn2)C(F)(F)F)OCCC(=C(F)F)F 3N-749 c1cc(ccc1CSc2nccc(n2)c3cc(sc3Cl)Cl)Br 3N-751 c1ccc(cc1)COC(=O)NCC(=O)N2CCOCC2 3P-001 CCCc1ccc(cc1)OCc2cnc(s2)Cl 3P-002 Cc1ccc(cc1)S(=O)(=O)c2ncc(s2)C=O 3P-005 Cc1cc(cc(c1)Oc2ccccc2CO)C 3P-006 CC(C)(C)c1ccc(cc1)Oc2ccccc2CO 3P-007 C/C(=N\NC(=O)N)/c1cccc(c1)OC 3P-008 CC1(OC(=O)C(=Cc2c[nH]nc2c3ccccc3)C(=O)O1)C 3P-009 c1ccc(c(c1)CO)Oc2cccc(c2)Cl 3P-010 Cc1ccc(cc1)S(=O)(=O)c2ncc(s2)/C=N\NC(=O)c3ccc(cc3)C(F)(F)F 3P-012 c1ccc(cc1)S(=O)(=O)c2ncc(s2)/C=N/NC(=O)c3ccco3 3P-013 CCOc1ccc(cc1)NC(=S)NC(=O)c2ccccc2 3P-015 Cc1ccc(cc1)S(=O)(=O)Cc2cnc(s2)Cl 3P-016 CCc1ccc(cc1)COn2ccnc2 3P-018 c1cc(ccc1c2c(c[nH]n2)/C=N\OCc3ccc(cc3Cl)Cl)F 3P-020 COC(=O)c1ccc(cc1)/N=C/c2cnc(s2)Cl 3P-021 COC(=O)c1ccc(cc1)/N=C/c2cnc(s2)S(=O)(=O)c3ccccc3 3P-022 CC(=O)CS(=O)(=O)c1ccccc1 3P-024 c1cc(ccc1CO/N=C/c2c[nH]nc2c3ccc(cc3)F)F 3P-025 Cc1ccccc1COn2ccnc2 3P-026 c1ccc(c(c1)CO)Oc2cccc(c2)C(F)(F)F 3P-027 c1ccc(c(c1)CO)Oc2ccc(cc2)F 3p-029 c1cc(cc(c1)OCc2cnc(s2)Cl)/C=N/O 3P-030 c1ccc(cc1)CCNC(=O)C2CC2 3P-033 c1cc(ccc1CO/N=C/c2c[nH]nc2c3ccc(cc3)F)Cl 3P-034 c1cc(ccc1/C=N/O)OCc2cnc(s2)Cl 3P-036 CC(=O)OCc1ccccc1Oc2ccc(cc2F)Br 3P-038 CC(=O)OCc1ccccc1Oc2ccc(cc2)I 3P-040 CS(=O)(=O)/C(=C\c1cnc(s1)S(=O)(=O)c2ccccc2)/C#N 3P-041 CC(=O)OCc1ccccc1Oc2ccc(c(c2)F)Cl 3P-044 c1cc(ccc1c2cn3cc(ccc3n2)Cl)F 3P-045 c1ccc(c(c1)CO)Oc2ccc(c(c2)F)F 3P-048 COc1ccc(cc1)c2cn3cc(ccc3n2)Cl 3P-050 CCCc1ccc(c(c1)F)c2ccc(cc2)C(=O)/C(=C/N(C)C)/c3ccc(cc3)Cl 3P-052 CCOc1ccc(cc1)Nc2nc(cs2)c3ccsc3 3P-054 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(con3)c4ccc(cc4)Cl 3P-055 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnc(n3)S)c4ccc(cc4)Cl 3P-057 Cc1cc(c(c(c1)O)C(=O)O)O 3P-058 c1cc(oc1)C(=O)N/N=C/c2cnc(s2)N3CCCC3 3P-059 Cc1cccn2c1nc(c2)c3ccc(cc3)Cl 3P-060 c1cc(ccc1c2c(c[nH]n2)/C=N/Nc3ccc(cc3)Cl)F 3P-062 Cc1cc(c(c(c1)O)C(=O)OC)O 3P-063 CC(=O)OCc1ccccc1Oc2cccc(c2)Cl 3P-064 c1cc(ccc1c2c(c[nH]n2)/C=N\Nc3ccnc4c3ccc(c4)Cl)F 3P-066 c1ccc(cc1)CSCC(=O)O 3P-067 c1ccc(c(c1)CCl)Oc2cccc(c2)C(F)(F)F 3P-068 c1ccc(c(c1)CCl)Oc2ccc(cc2Cl)Cl 3P-069 CCOC(=O)C(C(C(=O)OC(C)(C)C)Nc1ccc(c(c1)C)C)C(=O)OCC 3P-075 c1cc(ccc1c2c(c[nH]n2)/C=N/NC(=O)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)F 3P-080 COc1ccc(cc1)N/C=N\C(=C(\C#N)/N)\C#N 3P-082 CC(=O)OCc1ccccc1Oc2ccccc2 3p-084 c1cc(cnc1)/C=C\2/C(=O)C3CCN2CC3 3P-086 Cn1cccc1C(=O)N/N=C/c2c[nH]nc2c3ccc(cc3)F 3P-087 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=O)c2cccc(c2)OCc3ccc(cc3Cl)Cl 3P-088 c1cc2cn[nH]c2c(c1)N 3P-091 CCOC(=O)C(C(C(=O)OC(C)(C)C)NCc1ccc(cc1)Oc2ccc(cc2)OC)C(=O)OCC 3P-095 c1cc(ccc1c2cn3cc(ccc3n2)Cl)Br 3P-096 c1ccc2c(c1)CC(C2Sc3ncccn3)O 3P-098 COC(=O)c1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl 3P-099 CCOC(=O)C=C1CCCCC1 3P-100 c1cc(ccc1c2c(c[nH]n2)/C=N/NC(=O)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F)F 3P-104 CC(C)(C(=O)N/N=C/c1c[nH]nc1c2ccc(cc2)F)n3cncn3 3P-105 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2[nH]cc3 3P-106 Cc1ccc(cc1)S(=O)(=O)Oc2ccsc2C(=O)OC 3P-108 c1cc(sc1)c2cn3cc(ccc3n2)Cl 3P-109 Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Oc4ccc(cc4)Cl)CS2 3P-302S c1ccc2c(c1)c(=O)n3c(n2)NCC3CSc4ccc(cc4Cl)Cl 3P-304S COc1ccc(cc1)SCC2CNc3n2c(=O)c4ccccc4n3 3P-305S c1ccc2c(c1)c(=O)n3c(n2)NCC3CSc4ccc(cc4)Br 3P-306S CCCCn1c(c(c(c1NC(=O)C(C)C)C#N)c2ccccc2)c3ccccc3 3P-307S CCCCn1c(c(c(c1N(S(=O)(=O)c2ccc(cc2)C)S(=O)(=O)c3ccc(cc3)C)C#N)c4ccccc4)c5ccccc5 3P-308S Cc1ccc2c(c1)-c3c(cc(s3)C(=O)Oc4ccc(cc4)F)CS2 3P-309S CCCCn1c(c(c(c1/N=C/c2c(cccc2Cl)Cl)C#N)c3ccccc3)c4ccccc4 3P-310S CCCCn1c(c(c(c1/N=C/c2ccccc2F)C#N)c3ccccc3)c4ccccc4 3P-311S c1ccc(cc1)P2(=O)C3(CCCCC3)Nc4ccccc4O2 3P-312S c1ccc2c(c1)c(=O)n3c(n2)NCC3CSc4ccc(cc4)F 3P-314S c1ccc2c(c1)C(=O)N3C(CNC3N2)CSc4ccccc4N 3P-315S c1ccc2c(c1)c(=O)n3c(n2)NCC3CSc4cccc(c4)C(F)(F)F 3P-316S Cn1c2ccccc2c(c1Cl)/C=N/OC(=O)C3CC3 3P-317S CC(C)C(=O)O/N=C/c1c2ccccc2n(c1Cl)C 3P-318S Cn1c2ccccc2c(c1N3CCOCC3)C=O 3P-319S Cn1c2ccccc2c(c1N3CCOCC3)/C=N/O 3P-320S CC(=O)O/N=C/c1c2ccccc2n(c1N3CCOCC3)C 3P-321S Cn1c2ccccc2c(c1N3CCOCC3)C#N 3P-322S Cn1c2ccccc2c(c1N3CCOCC3)/C=N/c4ccc(cc4)OC 3P-323S CCCCn1c(c(c(c1/N=C/c2cccc(c2Cl)Cl)C#N)c3ccccc3)c4ccccc4 3P-324S CCCCn1c(c(c(c1/N=C/c2ccc(c(c2)F)F)C#N)c3ccccc3)c4ccccc4 3P-325S CCCCn1c(c(c(c1/N=C/c2ccccc2Cl)C#N)c3ccccc3)c4ccccc4 3P-326S CCCCn1c(c(c(c1/N=C/c2ccc(c(c2)[N+](=O)[O-])Cl)C#N)c3ccccc3)c4ccccc4 3P-327S CCCCn1c(c(c(c1/N=C/c2cccc(c2)C)C#N)c3ccccc3)c4ccccc4 3P-328S CCCCn1c(c(c(c1/N=C/c2cccc(c2)C(F)(F)F)C#N)c3ccccc3)c4ccccc4 3P-329S CCCCn1c(c(c(c1/N=C/c2cccc(c2O)OC)C#N)c3ccccc3)c4ccccc4 3P-330S CCCCn1c(c(c(c1/N=C/c2ccccc2C)C#N)c3ccccc3)c4ccccc4 3P-331S CCCCn1c(c(c(c1/N=C/c2ccc(cc2)C(=O)O)C#N)c3ccccc3)c4ccccc4 3P-332S CCCCn1c(c(c(c1/N=C/c2ccc(cc2)N(C)C)C#N)c3ccccc3)c4ccccc4 3P-333S CCCCn1c(c(c(c1/N=C/c2ccc(o2)C)C#N)c3ccccc3)c4ccccc4 3P-334S Cn1c2ccccc2c(c1N3CCN(CC3)C)C=O 3P-335S Cn1c2ccccc2c(c1N3CCN(CC3)C)/C=N/O 3P-336S Cc1c(n(c(c1C#N)NC(=O)c2ccccc2)Cc3ccccc3)C 3P-341S Cc1ccc(cc1)C(=O)Nc2c(c(c(n2Cc3ccccc3)C)C)C#N 3P-342S CCn1/c(=N\C(=O)c2ccc(cc2)C)/c3ccccc3[nH]c1=O 3P-343S CCn1/c(=N\C(=O)c2ccc(cc2)F)/c3ccccc3[nH]c1=O 3P-344S CC1(Nc2ccccc2OP1(=O)c3ccccc3)C 3P-345S Cc1cc(cc(c1)Oc2c(c3ccccc3n2C)/C=N/O)C(C)C 3P-346S Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)F)Cc3ccccc3)C 3P-352S Cc1c(n(c(c1C#N)NC(=O)c2ccccc2OC)Cc3ccccc3)C 3P-353S Cc1c(n(c(c1C#N)NC(=O)c2ccccc2Cl)Cc3ccccc3)C 3P-354S Cc1c(n(c(c1C#N)NC(=O)c2cccs2)Cc3ccccc3)C 3P-355S Cc1c(n(c(c1C#N)NC(=O)c2cccc(c2)Cl)Cc3ccccc3)C 3P-356S Cc1cccc(c1)C(=O)Nc2c(c(c(n2Cc3ccccc3)C)C)C#N 3P-357S Cc1c(n(c(c1C#N)NC(=O)Cc2cccs2)Cc3ccccc3)C 3P-358S Cc1c(n(c(c1C#N)NC(=O)C(C)C)Cc2ccccc2)C 3P-359S CCCC(=O)Nc1c(c(c(n1Cc2ccccc2)C)C)C#N 3P-360S Cc1c(n(c(c1C#N)NC(=O)C(C)(C)C)Cc2ccccc2)C 3P-361S Cc1c(n(c(c1C#N)N(S(=O)(=O)c2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)OC)Cc4ccccc4)C 3P-363S Cc1c(n(c(c1C#N)N(S(=O)(=O)c2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)F)Cc4ccccc4)C 3P-364S Cc1c(n(c(c1C#N)N(S(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl)Cc4ccccc4)C 3P-366S Cc1c(n(c(c1C#N)N(S(=O)(=O)c2ccccc2)S(=O)(=O)c3ccccc3)Cc4ccccc4)C 3P-367S CCn1/c(=N\C(=O)c2cccc(c2)Cl)/c3ccccc3[nH]c1=O 3P-372S CCn1/c(=N\C(=O)c2cccs2)/c3ccccc3[nH]c1=O 3P-373S CCn1/c(=N\C(=O)C(C)C)/c2ccccc2[nH]c1=O 3P-374S CCn1/c(=N\S(=O)(=O)c2ccc(cc2)C)/c3ccccc3[nH]c1=O 3P-376S c1ccc(cc1)n2c(=N)c3ccccc3[nH]c2=O 3P-377S Cc1c(n(c(c1C#N)N(S(=O)(=O)C)S(=O)(=O)C)Cc2ccccc2)C 3P-380S Cc1c(c(on1)N)C#N 3P-382S CCCC(=O)/N=c/1\c2ccccc2[nH]c(=O)n1CC 3P-387S Cc1ccc(cc1)CSC\2=Nc3ccccc3/C2=N\Nc4ccccc4 3P-388S Cc1c(c(on1)NC(=O)c2ccccc2)C#N 3P-392S Cc1c(c(on1)NC(=O)c2ccc(cc2)F)C#N 3P-393S Cc1cccc(c1)C(=O)Nc2c(c(no2)C)C#N 3P-394S Cc1c(c(on1)NC(=O)c2ccccc2C(F)(F)F)C#N 3P-395S Cc1c(c(on1)NC(=O)c2ccccc2Cl)C#N 3P-397S Cc1c(c(on1)NC(=O)c2ccccc2OC)C#N 3P-398S COC(=O)c1c(ccs1)NC(=O)COc2ccc(c3c2cccc3)Cl 3P-502S COC(=O)c1c(ccs1)NC(=O)COc2ccc(cc2Cl)[N+](=O)[O-] 3P-504S Cc1ccc(cc1)OCC(=O)Nc2ccsc2C(=O)OC 3P-505S Cc1cccc(c1)SCC(=O)Nc2ccccc2SCC(=O)Nc3ccsc3C(=O)OC 3P-508S CC(C)(C)c1ccc(cc1)SCC(=O)Nc2ccccc2SCC(=O)Nc3ccsc3C(=O)OC 3P-509S CN(CC(=O)Nc1ccsc1C(=O)OC)NS(=O)(=O)c2ccc(cc2)F 3P-514S CN(CC(=O)Nc1ccsc1C(=O)OC)NS(=O)(=O)c2ccc(cc2)Cl 3P-515S CN(CC(=O)Nc1ccsc1C(=O)OC)NS(=O)(=O)c2ccc(cc2)OC 3P-516S COC(=O)c1ccc(nc1)Sc2ccccc2N 3P-519S COc1ccc(cc1)S(=O)(=O)Nc2ccccc2Sc3ccc(cn3)C(=O)OC 3P-520S Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2Sc3ccc(cn3)C(=O)OC 3P-521S COC(=O)c1ccc(nc1)Sc2ccccc2NS(=O)(=O)c3ccc(cc3)Cl 3P-522S CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccccc2Sc3ccc(cn3)C(=O)OC 3P-523S CN(CC(=O)Nc1ccsc1C(=O)OC)NC(=O)c2cccs2 3P-524S COC(=O)c1ccc(nc1)Sc2ccccc2NC(=O)c3cccs3 3P-526S COC(=O)c1ccc(nc1)Sc2ccccc2NC(=O)c3cccc(c3Cl)Cl 3P-527S CN(CC(=O)Nc1ccsc1C(=O)OC)NS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] 3P-532S c1ccc2c(c1)C(=O)N(C2=O)COc3ccc(cc3Br)Cl 3P-536S Cc1c(c(n(n1)C)Oc2ccccc2)CCNC(=O)CCl 3P-563S Cc1c(c(n(n1)C)Oc2ccccc2)CCNC(=O)c3ccc(cc3)Cl 3P-564S Cc1c(c(n(n1)C)Oc2ccccc2)CCNS(=O)(=O)c3ccccc3 3P-565S Cc1c(c(n(n1)C)Oc2ccccc2)CCNC(=O)Nc3ccccc3 3P-566S Cc1c(c(n(n1)C)Oc2ccccc2)CCNC(=O)c3ccccc3 3P-567S Cc1c(c(n(n1)C)Oc2ccccc2)CCNC(=O)c3cccc(c3)Cl 3P-568S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)Cl)c5ccccc5)/C=N/OC(=O)c6ccc(cc6)Cl 3P-574S Cc1c(c(n(n1)C)Oc2ccccc2)CCNC(=O)C(C)(C)C 3P-577S Cc1c(c(n(n1)C)Oc2ccccc2)CCNS(=O)(=O)c3ccc(cc3)F 3P-578S Cc1c(c(n(n1)C)Oc2ccccc2)CCNS(=O)(=O)c3ccc(cc3)Cl 3P-579S Cc1c(c(n(n1)C)Oc2ccccc2)CCNS(=O)(=O)c3ccc(cc3)OC 3P-580S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)Cl)c5ccccc5)/C=N/OC(=O)c6cccc(c6)C 3P-581S Cc1ccc(cc1)SC2=C(CCc3c2cc(n3c4ccc(cc4)Cl)c5ccccc5)/C=N/OC(=O)c6cccc(c6Cl)Cl 3P-582S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccc(cc3)Cl)C#N 3P-583S COc1ccc(cc1)/C=N/c2c(cc(o2)c3ccccc3)C#N 3P-584S Cc1c(c(n(n1)C)Oc2ccccc2)CCNC(=O)CC(C)C 3P-585S Cc1cccc(c1)/C=N/c2c(cc(o2)c3ccccc3)C#N 3P-587S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccccc3F)C#N 3P-589S CN(C)c1ccc(cc1)/C=N/c2c(cc(o2)c3ccccc3)C#N 3P-592S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccc(cc3Cl)F)C#N 3P-593S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccc(cc3)Oc4ccccc4)C#N 3P-594S COc1cccc(c1O)/C=N/c2c(cc(o2)c3ccccc3)C#N 3P-595S COc1ccc(cc1OC)/C=N/c2c(cc(o2)c3ccccc3)C#N 3P-596S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccc(cc3)[N+](=O)[O-])C#N 3P-598S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccc(cc3Cl)Cl)C#N 3P-599S c1ccc(cc1)c2cc(c(o2)/N=C/c3c(cccc3Cl)F)C#N 3P-600S Cc1ccc(o1)/C=N/c2c(cc(o2)c3ccccc3)C#N 3P-601S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccccc3Cl)C#N 3P-602S c1ccc(cc1)c2cc(c(o2)/N=C/c3cccs3)C#N 3P-603S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccc(s3)Br)C#N 3P-604S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccccc3O)C#N 3P-605S c1ccc(cc1)c2cc(c(o2)/N=C/c3ccoc3)C#N 3P-606S COc1cc(ccc1O)/C=N/c2c(cc(o2)c3ccccc3)C#N 3P-607S c1ccc(cc1)c2cc(c(o2)NC(=O)c3ccc(cc3)Cl)C#N 3P-609S COc1cccc(c1)C(=O)Nc2c(cc(o2)c3ccccc3)C#N 3P-610S c1ccc(cc1)c2cc(c(o2)NC(=O)c3ccccc3C(F)(F)F)C#N 3P-611S c1ccc(cc1)c2cc(c(o2)NC(=O)c3cccc(c3)Cl)C#N 3P-612S Cc1cccc(c1)C(=O)Nc2c(cc(o2)c3ccccc3)C#N 3P-613S COc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc3c(s2)-c4ccccc4CC3 3P-640S CS(=O)(=O)NNC(=O)c1cc2c(s1)-c3ccccc3CC2 3P-642S Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc3c(s2)-c4ccccc4CC3 3P-643S COc1ccc(cc1)/C=N/NC(=O)c2cc3c(s2)-c4ccccc4CC3 3P-644S Cc1ccc(cc1)C2=NN(C(=O)CO2)CCC#N 3P-645S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)N/N=C/c4ccc(cc4)Cl 3P-646S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)N/N=C/c4cccc(c4)C(F)(F)F 3P-648S Cc1cccc(c1)/C=N/NC(=O)c2cc3c(s2)-c4ccccc4CC3 3P-649S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)N/N=C/c4ccc(c(c4)F)F 3P-650S c1ccc-2c(c1)CCc3c2sc(c3)C(=O)N/N=C/c4ccc(cc4)[N+](=O)[O-] 3P-652S Cc1ccc(cc1)c2nnc(o2)c3cc4c(s3)-c5ccccc5CC4 3P-676S c1ccc-2c(c1)CCc3c2sc(c3)c4nnc(o4)c5ccccc5C(F)(F)F 3P-677S c1ccc-2c(c1)CCc3c2sc(c3)c4nnc(o4)SCc5ccc(cc5)Cl 3P-679S c1ccc-2c(c1)CCc3c2sc(c3)c4nnc(o4)SCc5ccc(cc5)F 3P-680S Cc1ccc(cc1)CSc2nnc(o2)c3cc4c(s3)-c5ccccc5CC4 3P-681S c1ccc-2c(c1)CCc3c2sc(c3)c4nnc(o4)SCc5cccc(c5)C(F)(F)F 3P-682S CCSc1nnc(o1)c2cc3c(s2)-c4ccccc4CC3 3P-683S C=CCSc1nnc(o1)c2cc3c(s2)-c4ccccc4CC3 3P-684S Cc1cc(nc(c1C#N)Sc2ccccc2N)C 3P-686S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)C(=O)O 3P-687S Cc1cc(nc(c1C#N)Sc2ccccc2NS(=O)(=O)c3ccc(cc3)OC)C 3P-691S Cc1cc(nc(c1C#N)Sc2ccccc2NS(=O)(=O)c3cc(ccc3Cl)Cl)C 3P-692S Cc1ccc(o1)Cn2ccc(c(c2=O)C/C=C/c3ccccc3)O 3P-700 c1ccc(cc1)/C=C/Cc2c(ccn(c2=O)Cc3cccnc3)O 3P-701 C(#N)C1=C(Oc2c(c(=O)[nH]c(=O)[nH]2)C1(C#N)C#N)N 3P-702 Cn1c(=O)c2c(n(c1=O)C)OC(=C(C2(C#N)C#N)C#N)N 3P-703 CN1C(=O)N(C(O1)CC(=O)NCc2ccc(cc2)F)c3ccc(cc3)Cl 3P-705 c1cc2c(cc1C(F)(F)F)c(=O)c(c[nH]2)c3c(cc(cn3)C(F)(F)F)Cl 3P-706 c1cc(c2c(c1F)c(=O)c(c[nH]2)c3c(cc(cn3)C(F)(F)F)Cl)F 3P-707 c1c(cnc(c1Cl)c2c[nH]c3cc4c(cc3c2=O)OCO4)C(F)(F)F 3P-708 CC1(CC2=C(C(=O)C1)C(C(=C(O2)N)C#N)(C#N)C#N)C 3P-709 CCOC(=O)CNC=C(C(=O)C)C(=O)C 3P-710 CN1C(=O)N(C(O1)CC(=O)Nc2ccc(cc2)Br)c3ccc(cc3)Cl 3P-711 CN1C(=O)N(C(O1)CC(=O)NCc2ccc3c(c2)OCO3)c4ccc(cc4)Cl 3P-712 CN1C(=O)N(C(O1)CC(=O)Nc2ccccn2)c3ccc(cc3)Cl 3P-713 Cc1ccc(cc1)CNC(=O)CC2N(C(=O)N(O2)C)c3ccc(cc3)Cl 3P-714 c1cc(cc(c1)C(F)(F)F)Cn2cc(c(=O)nc2)c3c(cc(cn3)C(F)(F)F)Cl 3P-716 c1ccc2c(c1)c(c[nH]2)CCn3cc(c(=O)nc3)c4c(cc(cn4)C(F)(F)F)Cl 3P-718 c1ccc(cc1)/C=C/Cc2c(ccn(c2=O)CCc3c[nH]c4c3cccc4)O 3P-720 C=CCN(C=O)NC=O 3P-721 CN(C(=O)Nc1ccccc1F)O 3P-722 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)(C#N)C#N 3P-723 c1ccc(cc1)/C=C/Cc2c(ccn(c2=O)CC3CC3)O 3P-724 COC(=O)/C(=N/O)/c1c(cc(cn1)C(F)(F)F)Cl 3P-726 COC(=O)/C(=N\OC(=O)Nc1ccc(c(c1)Cl)Cl)/c2c(cc(cn2)C(F)(F)F)Cl 3P-727 COC(=O)/C(=N\OC(=O)Nc1cccc(c1)C(F)(F)F)/c2c(cc(cn2)C(F)(F)F)Cl 3P-728 COC(=O)/C(=N\OC(=O)Nc1ccccc1F)/c2c(cc(cn2)C(F)(F)F)Cl 3P-729 CCOC(=O)C(Cc1ccc(cc1Cl)Cl)C(=O)C 3P-730 CCOC(=O)C(Cc1ccc(cc1Cl)Cl)(Cc2ccc(cc2Cl)Cl)C(=O)C 3P-731 CCOC(=O)C(Cc1ccc(cc1Cl)Cl)(Cc2ccc(cc2Cl)Cl)C(=O)/C=C\N(C)C 3P-732 c1ccc(cc1)/N=N/c2ccc3c(c2)c(=O)c(c[nH]3)c4c(cc(cn4)C(F)(F)F)Cl 3P-734 COC(=O)/C(=C\Nc1ccc(cc1F)Cl)/c2c(cc(cn2)C(F)(F)F)Cl 3P-735 c1c(cc(c2c1c(=O)c(c[nH]2)c3c(cc(cn3)C(F)(F)F)Cl)F)Cl 3P-736 C1CC2=C(C(=O)C1)C(C(=C(O2)N)C#N)(C#N)C#N 3P-737 CC(=O)c1cccc2c1[nH]cc(c2=O)c3c(cc(cn3)C(F)(F)F)Cl 3P-740 COC(=O)/C(=C\Nc1ccc(c2c1cccc2)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 3P-741 c1ccc2c(c1)c(cc3c2[nH]cc(c3=O)c4c(cc(cn4)C(F)(F)F)Cl)Cl 3P-742 c1cc(c(cc1Cl)Cl)OCCOc2ccc(cc2Cl)Cl 3P-743 c1ccn(c1)c2ccsc2c3cc4nccc(n4n3)c5ccc(cc5)OCc6ccc(cc6Cl)Cl 3R-0001 CC(c1ccc(cc1)OCc2ccc(cc2Cl)Cl)O 3R-0002 CC(C1C(=O)N(C(=O)N(C1=O)C)C)C(=O)O 3R-0003 c1cc(ccc1C(=O)C/C=N/OCc2ccc(cc2Cl)Cl)OCc3ccc(cc3Cl)Cl 3R-0005 Cc1cc(c2nncn2n1)O 3R-0006 CC(=O)NC1=NC(CS1)CC(=O)OC 3R-0007 c1cnccc1c2nccc(n2)N 3R-0009 c1ccc2c(c1)CC(CC2O)c3ccc(cc3)c4ccc(cc4)Br 3R-0012 c1cc(ccc1C(=O)/C=C/Nc2ccc(c(c2)[N+](=O)[O-])Cl)OCCCF 3R-0013 c1ccc(cc1)Oc2ccc(cc2)N/C=C/C(=O)c3ccc(cc3)OCCCF 3R-0014 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)OC(F)(F)F)OCc3ccc(cc3Cl)Cl 3R-0015 c1ccc(cc1)Cc2c(nc3ccccc3n2)NNC(=O)c4cccc(c4)Cl 3R-0016 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(c(c2)[N+](=O)[O-])F 3R-0019 c1ccc(cc1)c2cc(c3nncn3n2)O 3R-0020 CCOC(=O)c1c2ccccn2cc1c3cccc(c3)[N+](=O)[O-] 3R-0023 CN(CCO)c1c(cc(cn1)C(F)(F)F)Cl 3R-0025 C1C=CCC2C1C(=O)N(C2=O)CCC#N 3R-0028 Cc1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl 3R-0030 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)F)OCc3ccc(cc3Cl)Cl 3R-0031 COc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)OCCCF 3R-0032 c1cc(ccc1c2ccn(n2)C(=O)C3CCCCC3)OCc4ccc(cc4Cl)Cl 3R-0033 c1cc(ccc1C(=O)/C=C/Nc2ccc(c(c2)Cl)Cl)OCc3ccc(cc3Cl)Cl 3R-0034 CCOC(=O)C(CSCC(=O)NCCc1ccccc1)[NH3+].C(=O)(C(F)(F)F)[O-] 3R-0035 COc1ccc(cc1)CNC(=O)/C=C/c2ccc(cc2)OCCCF 3R-0036 c1cc(ccc1/C=C/C(=O)NCc2ccc3c(c2)OCO3)OCCCF 3R-0037 CC(C)(C)c1ccccc1N/C=C/C(=O)c2ccc(cc2)OCc3ccc(cc3Cl)Cl 3R-0038 COC(CNc1ccc(cc1Br)[N+](=O)[O-])OC 3R-0041 c1cnc(nc1)NC(=O)C2CC=CCC2C(=O)Nc3ncccn3 3R-0042 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NC4CCCCC4 3R-0043 c1ccc(cc1)CNC(=O)COc2ccc(cc2)c3nccc(n3)c4ccccn4 3R-0044 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NCc4ccco4 3R-0045 COc1ccccc1NC(=O)C2CC=CCC2C(=O)O 3R-0046 c1ccc(cc1)S(=O)(=O)NNC(=O)C2CC=CCC2C(=O)O 3R-0048 Cc1cc(nn2c1nnc2)C(F)(F)F 3R-0049 C=CCSC1=Nc2c(ccs2)C3=NC(=O)CN31 3R-0050 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NCc4ccc5c(c4)OCO5 3R-0051 c1c(cc(cc1Cl)Cl)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 3R-0052 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NCc4cccs4 3R-0053 c1cc(c(cc1NS(=O)(=O)c2cc(ccc2Cl)Cl)[N+](=O)[O-])F 3R-0054 c1cc(ccc1OCCOCCNn2cnnc2)Br 3R-0055 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)NNC(=O)C3CC=CCC3C(=O)O 3R-0057 COc1ccc(cc1OC)CNC(=O)/C=C/c2ccc(cc2)OCCCF 3R-0058 Cc1ccc(o1)CNC(=O)/C=C/c2ccc(cc2)OCCCF 3R-0059 c1ccc(c(c1)N/C=C/C(=O)c2ccc(cc2)OCc3ccc(cc3Cl)Cl)N4CCOCC4 3R-0060 c1ccc2cc(ccc2c1)c3ccc(cc3)c4ccc(cc4)Br 3R-0061 COC(=O)CSC1=Nc2ccccc2C3=NC(=O)CN31 3R-0062 CN1C(=O)C(=Cc2ccccc2Oc3ccc(c(c3)F)Cl)C(=O)N(C1=O)C 3R-0064 c1cc(c(cc1CNC(=O)c2cc(cc(c2O)I)I)Cl)Cl 3R-0066 c1ccc(c(c1)c2cc(n3c(n2)cc(n3)c4c(ccs4)n5cccc5)C(F)(F)F)Cl 3R-0069 c1cc(ccc1c2ccnc3n2ncn3)OCCCF 3R-0070 COC(=O)CSc1nc2ccccc2c(=N)n1c3ccc(cc3)Cl 3R-0071 c1cc(ccc1/C=C/C(=O)n2ccc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl)OCCCF 3R-0073 c1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)Oc3ccc(c(c3)F)Cl 3R-0074 c1ccc(cc1)C(=O)NC(=S)N2CCOCC2 3R-0075 c1cc(ccc1c2ccn(n2)C(=O)c3ccc(cc3)F)OCc4ccc(cc4Cl)Cl 3R-0078 c1cc(sc1)C(=O)n2ccc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl 3R-0079 c1ccc(c(c1)/C=N/OCc2c(cccc2Cl)Cl)Oc3ccc(c(c3)F)Cl 3R-0081 c1ccc(c(c1)/C=N/OCc2ccc(cc2Cl)Cl)Oc3ccc(c(c3)F)Cl 3R-0083 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])C2CCCCC2=O 3R-0086 CCC(C)c1ccc(c(c1)C=O)O 3R-0089 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl 3R-0090 COc1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl 3R-0091 c1cc(cc(c1)Cl)Cn2ccc(n2)c3ccc(cc3)OCc4c(cccc4Cl)F 3R-0093 CC(=O)c1cccc(c1)OCc2c(cccc2Cl)F 3R-0094 c1cc(ccc1c2ccnc(n2)c3ccncc3)OCc4ccc(cc4Cl)Cl 3R-0097 c1cc(ccc1c2ccn(n2)S(=O)(=O)c3ccc(c(c3)Cl)Cl)OCc4ccc(cc4Cl)Cl 3R-0098 Cc1cc2nccc(n2n1)c3ccc(cc3)OCCCF 3R-0100 CN(C)/C=C/C(=O)c1ccc(cc1)OCCN(C)c2ccccn2 3R-0102 c1ccn(c1)c2ccsc2c3cc4nccc(n4n3)c5ccc(cc5)OCCCF 3R-0103 CCC(C)c1ccc(c(c1)/C=N/O)O 3R-0104 CCOC(=O)CNc1ccc(cc1[N+](=O)[O-])NS(=O)(=O)c2cc(ccc2Cl)Cl 3R-0105 CC1=C(C(C(=C(N1)CCl)C(=O)OC)c2cccc(c2)[N+](=O)[O-])C(=O)OC 3R-0108 CN(C1CCCCC1)C(=O)/C=C/c2cc3ccccc3nc2 3R-0110 CC(C)CCN(CCC(C)C)C(=O)/C=C/c1cc2ccccc2nc1 3R-0111 CCOc1ccc(cc1)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 3R-0113 c1cc(c(cc1Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F)Cl)Br 3R-0114 c1cc(c(cc1Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F)Cl)Cl 3R-0115 c1cc(ccc1/C=N\n2cnnc2)c3[nH]nnn3 3R-0121 c1ccc2c(c1)cc(cn2)/C=C/C(=O)N3CCCCC3 3R-0124 c1ccc(cc1)CNC(=O)/C=C/c2cc3ccccc3nc2 3R-0125 c1ccc2c(c1)cc(cn2)/C=C/C(=O)NCc3ccco3 3R-0128 Cc1c(nc2cc(nn2c1C)c3c(ccs3)n4cccc4)C 3R-0129 Cc1cccc(c1)C(=O)Nc2ccnc(n2)c3ccncc3 3R-0130 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NN 3R-0134 c1cc(oc1)CNC(=O)c2ccc(cc2)N3CCCC3=O 3R-0135 COc1ccc(cc1)N/C=C/C(=O)c2cccc(c2)OCc3c(cccc3Cl)F 3R-0137 c1c2c(cc(c1Cl)Cl)nc(c(n2)C(F)(F)F)NN 3R-0138 c1(nnc(n1N)N)N 3R-0139 Cc1ccc(cc1)N/C=C/C(=O)c2cccc(c2)OCc3c(cccc3Cl)F 3R-0141 c1ccc2c(c1)cc(cn2)/C=C/C(=O)NCc3ccc(c(c3)Cl)Cl 3R-0142 CCN(C)C(=O)/C=C/c1cc2ccccc2nc1 3R-0143 c1cc(sc1)C(=O)Nc2ccnc(n2)c3ccncc3 3R-0144 c1ccc(c(c1)C(=O)Nc2ccnc(n2)c3ccncc3)Cl 3R-0145 c1ccc(cc1)Oc2ccc(cc2)N/C=C(\C#N)/c3ccc(cc3)OCCCF 3R-0146 c1cc(ccc1/C(=C/Nc2cc(cc(c2)Cl)Cl)/C#N)OCCCF 3R-0147 COc1cc(cc(c1)OC)N/C=C(\C#N)/c2ccc(cc2)OCCCF 3R-0148 Cc1ccccc1C(=O)Nc2ccnc(n2)c3ccncc3 3R-0149 c1cc(cc(c1)OCc2c(cccc2Cl)F)C(=O)/C=C/Nc3ccc(cc3)OC(F)(F)F 3R-0150 COc1ccc(cc1Cl)N/C=C/C(=O)c2cccc(c2)OCc3c(cccc3Cl)F 3R-0151 c1cc(c(cc1Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F)F)Cl 3R-0152 CN(C)/C=C\1/C(=O)N(C(=S)N1)CC(OC)OC 3R-0155 CCOC(=O)CNC(=S)Nc1cc(c(cc1C#N)OC)OC 3R-0158 c1cc(ccc1C(=O)NCc2ccc(c(c2)Cl)Cl)N3CCCC3=O 3R-0161 c1ccc(cc1)NN2C(=O)C3CC=CCC3C2=O 3R-0163 c1ccc2c(c1)cc(cn2)/C=C/C(=O)NO 3R-0164 c1ccc2c(c1)cc(cn2)/C=C/C(=O)NNc3ccc(cc3)Cl 3R-0165 c1ccc2c(c1)cc(cn2)/C=C/C(=O)NNc3ccccc3F 3R-0166 c1cc(cc(c1)N/C=C(\C#N)/c2ccc(cc2)OCCCF)C(F)(F)F 3R-0168 COc1cccc(c1)N/C=C(\C#N)/c2ccc(cc2)OCCCF 3R-0169 c1ccc2c(c1)cc(cn2)/C=C/C(=O)NNC(=O)N 3R-0170 Cc1ccc(cc1)Cn2ccc(n2)c3ccc(cc3)OCc4c(cccc4Cl)F 3R-0172 Cc1cc(ccc1Br)N/C=C/C(=O)c2cccc(c2)OCc3c(cccc3Cl)F 3R-0173 c1cc(ccc1C(=O)N2CCOCC2)N3CCCC3=O 3R-0175 CCC(C)NC(=O)c1ccc(cc1)N2CCCC2=O 3R-0177 COc1cccc(c1)C(=O)Nn2cnnc2 3R-0178 c1cc(c(c(c1)Cl)COc2ccc(cc2)c3ccn(n3)Cc4ccc(cc4)C(F)(F)F)F 3R-0179 c1cc(cc(c1)OCc2c(cccc2Cl)F)C(=O)C/C=N/OCc3ccc(cc3Cl)Cl 3R-0180 c1cc(c(c(c1)Cl)COc2ccc(cc2)c3ccn(n3)c4c(cc(cn4)C(F)(F)F)Cl)F 3R-0181 CC(C)(CCl)C(=O)Nc1ccnc(n1)c2ccncc2 3R-0182 c1cc(ccc1C(=O)N2CCN(CC2)c3ccc(cc3)Cl)N4CCCC4=O 3R-0183 CCOC(=O)c1c(c(nnc1C(=O)OCC)c2ccccc2)c3ccccc3 3R-0184 CC(c1ccc(cc1)OCCN(C)c2ccccn2)O 3R-0189 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccnc(n2)c3ccncc3 3R-0190 Cc1cc(c2nncn2n1)OC(=O)c3ccc(cc3)OC 3R-0191 c1ccc(cc1)Oc2ccc(cc2)N/C=C/C(=O)c3cccc(c3)OCc4c(cccc4Cl)F 3R-0193 Cc1c(c(nn2c1nnc2)C)Cl 3R-0195 c1ccc(cc1)C2=NOC3C2CC(C3)C(=O)O 3R-0196 c1ccc(cc1)n2ccnc2SCC(=O)c3ccc(cc3)Br 3R-0197 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NN 3R-0198 c1cc(cnc1)c2nccc(n2)N 3R-0199 COc1cc(c(cc1OC)N2C(=O)CNC2=S)C#N 3R-0201 Cc1cc(c2nncn2n1)OC(=O)c3cccc(c3)C(F)(F)F 3R-0202 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nn2cnnc2 3R-0203 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccnc(n3)N 3R-0205 c1ccc(cc1)COc2ccc(cc2F)Oc3ccc(cc3Br)[N+](=O)[O-] 3R-0206 c1cc(cc(c1)OCc2c(cccc2Cl)F)C(=O)/C=C/Nc3ccc(c(c3)Cl)Cl 3R-0207 c1cc(ccc1Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F)Cl 3R-0209 COC(=O)CSc1nccn1c2ccccc2 3R-0211 c1cc(ccc1/C=C/C(=O)Nc2ccnc(n2)c3ccncc3)OCCCF 3R-0213 c1cc(ccc1c2nc[nH]n2)N3CCCC3=O 3R-0214 CC(=O)c1cccc(c1)OCc2ccc(cc2Cl)Cl 3R-0215 c1ccnc(c1)c2ccnc(n2)c3ccc(cc3)OCC(=O)NCc4ccc(c(c4)Cl)Cl 3R-0216 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3cc[nH]n3 3R-0217 c1cc(cc(c1)OCc2c(cccc2Cl)F)C(=O)/C=C/Nc3ccc(cc3)F 3R-0219 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccnc(n3)c4ccncc4 3R-0220 c1cc(cc(c1)OCc2c(cccc2Cl)F)C(=O)/C=C/Nc3ccc(cc3)Cl 3R-0221 c1cc(ccc1C(=O)Nc2ccnc(n2)c3ccncc3)F 3R-0223 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NNC(=O)Nc3ccccc3 3R-0224 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NNC(=O)NC3CCCCC3 3R-0225 CCNC(=O)NNC(=O)c1ccc(cc1Cl)OCc2ccccc2 3R-0226 CCNC(=S)NNC(=O)c1ccc(cc1Cl)OCc2ccccc2 3R-0228 Cc1ccc(cc1)S(=O)(=O)NC(=O)NNC(=O)c2ccc(cc2Cl)OCc3ccccc3 3R-0229 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NNC(=O)Nc3cccc(c3)Cl 3R-0230 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NNC(=O)Nc3ccc(cc3)Cl 3R-0231 C=CCNC(=S)NNC(=O)c1ccc(cc1Cl)OCc2ccccc2 3R-0232 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)/C=C/Nc3ccc(cc3)OC(F)(F)F 3R-0234 c1ccc(cc1)Oc2ccc(cc2)N/C=C/C(=O)c3cccc(c3)OCc4ccc(cc4Cl)Cl 3R-0235 Cc1ccc(cc1)N/C=C/C(=O)c2cccc(c2)OCc3ccc(cc3Cl)Cl 3R-0236 Cc1cc(c2nncn2n1)Cl 3R-0237 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NNC(=S)Nc3cccc(c3)C(F)(F)F 3R-0238 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NCc3ccccc3Cl 3R-0239 c1ccc(cc1)n2ccnc2SCC(=O)c3ccc(cc3)Cl 3R-0240 c1ccc(cc1)n2ccnc2SCc3ccc(cc3)C(F)(F)F 3R-0242 c1ccc2c(c1)cc(cn2)/C=C/C(=O)N3CCOCC3 3R-0245 Cc1ccc(cc1)C(=O)CSc2nccn2c3ccccc3 3R-0246 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccn(n3)C(=O)c4ccc(cc4)F 3R-0250 COc1ccc(cc1Cl)N/C=C/C(=O)c2cccc(c2)OCc3ccc(cc3Cl)Cl 3R-0251 CC1(C(=O)NC(CS1)C(=O)O)C 3R-0252 c1cc(ccc1C(=O)NNC(=O)C2CC=CCC2C(=O)O)Cl 3R-0254 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 3R-0255 c1cc(ccc1CC(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3)Cl 3R-0256 c1cc(c(c(c1)Cl)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F)Cl 3R-0257 Cc1cccc(c1Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F)C 3R-0258 c1c(cc(c(c1Cl)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F)Cl)Cl 3R-0259 CC1=C(C(C=C(N1)CSc2nccn2c3ccccc3)c4cccc(c4)[N+](=O)[O-])C(=O)OC 3R-0260 CCOC(CCNC(=O)c1ccc(cc1Cl)OCc2ccccc2)OCC 3R-0261 c1cc(c(c(c1)Cl)COc2ccc(cc2)c3ccn(n3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])F 3R-0262 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NCCCl 3R-0263 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCCOCCSc4nnc(s4)N 3R-0264 c1c(cc(c(c1Cl)NNC(=O)C2CC=CCC2C(=O)O)Cl)Cl 3R-0267 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)/C=C/Nc3ccc(cc3)Cl 3R-0269 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccn(n3)C(=O)c4ccc(cc4)I 3R-0270 c1cc(ccc1C(=O)NN2C(=O)C3CC=CCC3C2=O)Cl 3R-0272 c1c(cc(c(c1Cl)NN2C(=O)C3CC=CCC3C2=O)Cl)Cl 3R-0275 c1ccc(cc1)n2ccnc2SCCN3C(=O)c4ccccc4C3=O 3R-0278 C1COCCN1C(=O)C2CC=CCC2C(=O)O 3R-0280 Cc1ccc(cc1)C(=O)n2ccc(n2)c3cccc(c3)OCc4c(cccc4Cl)F 3R-0281 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)/C=C/Nc3ccc(c(c3)[N+](=O)[O-])Cl 3R-0282 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccn(n3)C(=O)c4ccc(c(c4)Cl)Cl 3R-0283 Cc1cccc(c1)C(=O)n2ccc(n2)c3cccc(c3)OCc4c(cccc4Cl)F 3R-0284 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccn(n3)C(=O)/C=C/c4ccc(cc4)OCCCF 3R-0285 COCCCNC(=O)c1cc(c[nH]1)C(=O)c2ccccc2 3R-0286 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)c2ccccc2 3R-0287 c1ccc(cc1)c2c(c(nnc2c3ccccc3)C(=O)O)C(=O)O 3R-0293 c1ccc(cc1)n2ccnc2SCCCN3C(=O)c4ccccc4C3=O 3R-0294 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)Cc2ccc(cc2)Cl 3R-0297 CC(C)N(C(C)C)C(=O)c1cc(c[nH]1)C(=O)c2ccccc2 3R-0298 c1cc(cnc1)CNC(=O)c2cc(c[nH]2)C(=O)Cc3ccc(cc3)Cl 3R-0299 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccnc3 3R-0300 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)/C=C/Nc3cccc(c3)[N+](=O)[O-] 3R-0301 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)/C=C/Nc3ccc(cc3)I 3R-0302 c1cc(c(cc1Cl)Cl)C(=O)NNC(=O)[C@H]2CC=CC[C@H]2C(=O)O 3R-0303 c1cc(ccc1CC(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3)Cl 3R-0304 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3 3R-0307 c1ccc(c(c1)CSC2=Nc3ccccc3C4=NC(=O)CN42)Cl 3R-0311 c1ccc(cc1)N2CCN(CC2)C(=O)C3CC=CCC3C(=O)O 3R-0312 COC(=O)C(Cc1ccc(cc1)OC(=O)c2ccc(cc2)C(F)(F)F)N3Cc4ccccc4C3=O 3R-0600 Cc1cc(cnc1NC(=O)c2cccs2)I 3R-0601 CC(C)CC(C(=O)N1CCN(CC1)C)N2Cc3ccccc3C2=O 3R-0602 Cc1cc(cn2c1nc(c2)c3ccc(cc3)F)I 3R-0606 CC(C)CC(C(=O)Nc1cc(cc(c1)Cl)Cl)N2Cc3ccccc3C2=O 3R-0607 c1cc(ccc1c2cn3cc(ccc3n2)I)F 3R-0610 CCOC(=O)c1cn2cc(ccc2n1)I 3R-0613 Cc1c(c(n(n1)C)C)C(=O)N/N=C/c2ccc(c(c2)OC)OC 3R-0614 CCOC(=O)C(F)Sc1nc[nH]n1 3R-0616 C=CCN(CC(C(F)(F)F)O)CC(C(F)(F)F)O 3R-0617 c1ccc2c(c1)c(c[nH]2)CC(C(=O)Nc3ccc(cc3F)F)N4CCS(=O)(=O)CC4 3R-0618 Cc1ccc(o1)CN2CCS(=O)(=O)CC2 3R-0619 C=CCCOC(c1ccccc1)C(F)(F)F 3R-0620 COC(=O)C(Cc1ccccc1)N2CCS(=O)(=O)CC2 3R-0621 c1ccc(cc1)CC(CO)NC(=O)c2cccc(c2)[N+](=O)[O-] 3R-0622 c1ccc(cc1)CC(CO)NC(=O)c2ccc(cc2)Cl 3R-0624 c1ccc(cc1)CC(CO)NC(=O)c2c(cccc2F)F 3R-0625 c1ccc(cc1)CC(CO)NC(=O)c2ccc(cc2)I 3R-0627 c1ccc(cc1)C(CO)NC(=O)c2cccc(c2)[N+](=O)[O-] 3R-0628 c1ccc2c(c1)c(c[nH]2)CC(C(=O)NCc3ccccn3)N4CCS(=O)(=O)CC4 3R-0629 c1ccc2c(c1)c(c[nH]2)CC(C(=O)NCc3ccco3)N4CCS(=O)(=O)CC4 3R-0630 c1ccc(cc1)N2CCN(CC2)C(=O)C(Cc3c[nH]c4c3cccc4)N5CCS(=O)(=O)CC5 3R-0632 c1ccc2c(c1)c(c[nH]2)CC(C(=O)Nc3cccc(c3)Br)N4CCS(=O)(=O)CC4 3R-0633 c1ccc(cc1)C(CO)NC(=O)c2ccc(cc2)I 3R-0635 c1cc2nc(cn2cc1I)C(=O)O 3R-0636 Cc1cc(cn2c1nc(c2)c3cccc(c3)C(F)(F)F)I 3R-0639 c1cc(cc(c1)C(F)(F)F)c2cn3cc(ccc3n2)I 3R-0640 c1ccc(cc1)C(CO)NC(=O)Nc2cccc(c2)F 3R-0641 c1ccc(cc1)CC(CO)NC(=O)Nc2cccc(c2)F 3R-0642 c1ccn(c1)CCN 3R-0643 c1ccc(cc1)C(CO)NC(=S)Nc2ccc(cc2)Cl 3R-0646 Cc1cccn2c1nc(c2)c3ccc(cc3)F 3R-0648 Cc1c(c(n(n1)C)C)C(=O)NNC(=O)c2ccc(cc2)Cl 3R-0649 COc1ccc(cc1)CNC(=O)C(Cc2c[nH]c3c2cccc3)N4CCS(=O)(=O)CC4 3R-0650 c1ccc2c(c1)c(c[nH]2)CC(C(=O)NCc3cccs3)N4CCS(=O)(=O)CC4 3R-0651 c1ccc(cc1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 3R-0652 c1ccc(cc1)CCNC(=O)C(Cc2c[nH]c3c2cccc3)N4CCS(=O)(=O)CC4 3R-0654 CCOC(=O)c1cn2ccc(cc2n1)C 3R-0655 Cc1c(c(n(n1)C)C)C(=O)NNC(=O)c2cccs2 3R-0657 c1ccc(cc1)CCN/C=C/C(=O)C(F)(F)F 3R-0658 c1cc(cnc1)N/C=C/C(=O)C(F)(F)F 3R-0662 c1ccc(cc1)C(CO)N/C=C/C(=O)C(F)(F)F 3R-0663 CCOC(=O)c1cn2cccnc2n1 3R-0666 CCOC(=O)c1c(n2cc(ccc2n1)I)Br 3R-0667 c1cc(ccc1C(=O)O)N2CCS(=O)(=O)CC2 3R-0668 c1ccnc(c1)N/C=C/C(C(F)(F)F)O 3R-0669 c1cc(ccc1C(F)(F)F)N/C=C/C(=O)C(F)(F)F 3R-0670 c1ccc2c(c1)CCN(C2)/C=C/C(=O)C(F)(F)F 3R-0671 c1ccc2c(c1)c(c[nH]2)CC(C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F)N4CCS(=O)(=O)CC4 3R-0672 c1ccc2c(c1)CCN2/C=C/C(=O)C(F)(F)F 3R-0674 Cc1ccn2cc(nc2c1)c3cccc(c3)C(F)(F)F 3R-0676 CCOC(=O)c1cn2cc(ccc2n1)Cl 3R-0683 CCOC(=O)c1c(n2cccnc2n1)Br 3R-0684 CCO/C=C\C(=O)C(F)(F)Cl 3R-0685 c1ccc2c(c1)nc(s2)N/C=C/C(=O)C(F)(F)F 3R-0686 c1ccc2c(c1)c(c[nH]2)CCN/C=C/C(=O)C(F)(F)F 3R-0687 C1CN(CCN1CCO)/C=C\C(=O)C(F)(F)F 3R-0688 c1ccc2c(c1)nc(s2)NCCC(C(F)(F)F)O 3R-0690 COc1cccc(c1)NC(=O)C(c2ccccc2)N3Cc4ccccc4C3=O 3R-0691 c1ccc2c(c1)CCN2/C=C/C(=O)C(F)(F)Cl 3R-0692 C1CN=C(C=CN1)C(F)(F)F 3R-0693 c1ccc2c(c1)c(c[nH]2)/C=C/C(=O)C(F)(F)F 3R-0695 CC(C)CC(C(=O)N1CCOCC1)N2Cc3ccccc3C2=O 3R-0699 c1ccc2c(c1)c(c[nH]2)CC(C(=O)N3CCOCC3)N4CCS(=O)(=O)CC4 3R-0700 c1ccc2c(c1)c(c[nH]2)/C=C/C(C(F)(F)F)O 3R-0704 CC(=O)c1nc2ccccc2n1CCc3ccccc3 3R-0705 C1CCN(CC1)/C=C\C(=O)C(F)(F)F 3R-0706 c1ccc2c(c1)c(cn2Cc3ccc(cc3)F)CCN4CCS(=O)(=O)CC4 3R-0707 c1ccc(cc1)CNCc2cc(cc(c2O)Br)Br 3R-0708 c1cc(ccc1N2Cc3cc(cc(c3OC2)Br)Br)F 3R-0709 c1cc(cc(c1)C(F)(F)F)CN2CCS(=O)(=O)CC2 3R-0710 CCOC(=O)c1c(n2cc(ccc2n1)Cl)Cl 3R-0711 c1ccc2c(c1)CCN2/C=C\C(=O)C(F)F 3R-0713 c1cc(ccc1CON2CCS(=O)(=O)CC2)C(F)(F)F 3R-0714 c1ccc2c(c1)c(c[nH]2)CC(C(=O)NCc3cccc(c3)C(F)(F)F)N4CCS(=O)(=O)CC4 3R-0716 Cc1cc(nc2c1c(n[nH]2)NC(=O)C)C 3R-0721 c1ccc(c(c1)N/C=C/C(=O)C(F)(F)F)OC(F)(F)F 3R-0722 c1cc(ccc1N/C=C/C(=O)C(F)(F)F)OC(F)(F)F 3R-0725 c1ccc(c(c1)N/C=C/C(=O)C(F)(F)F)F 3R-0726 CC(C)CC(C(=O)NCc1cccc(c1)C(F)(F)F)N2Cc3ccccc3C2=O 3R-0728 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 3R-0729 c1cc(cc(c1)C(F)(F)F)CN/C=C/C(=O)C(F)(F)F 3R-0733 c1ccc2c(c1)c(n[nH]c2=O)CC#N 3R-0801 CCCCN1C(C(CCC1=O)C(=O)O)c2ccc(cc2)[N+](=O)[O-] 3R-0802 CC1(CN(C1=O)CCc2c[nH]c3c2cccc3)C 3R-0804 C/C(=C\C(=O)c1ccc2ccccc2c1)/Nc3ccc(cc3)OC(F)(F)F 3R-0806 Cc1cc(n2c(n1)ncn2)c3ccc4ccccc4c3 3R-0808 Cc1ccc(n1CCc2c[nH]c3c2cccc3)C 3R-0811 c1ccc2c(c1)c(c[nH]2)CCNc3c(cccn3)C(F)(F)F 3R-0812 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/Nc3ccc(cc3)OC 3R-0813 Cc1c(nnn1c2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] 3R-0814 Cc1ccc(cc1)N/C=C/C(=O)c2c(nc(s2)c3ccc(cc3)Cl)C 3R-0815 Cc1c(sc(n1)c2ccccc2)C(=O)C3C(C3(C#N)C#N)c4ccccc4 3R-0816 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3cccnc3 3R-0818 Cc1c(nnn1c2ccc(cc2)[N+](=O)[O-])C(=O)c3ccc4ccccc4c3 3R-0819 CN(C)/C=C/c1c(nnn1c2ccc(cc2)[N+](=O)[O-])C(=O)c3ccc4ccccc4c3 3R-0820 CCOC(=O)Cc1c(=O)n(c2ccccc2n1)Cc3cccc(c3)C 3R-0825 CCOC(=O)Cc1c(=O)n(c2ccccc2n1)CC(=O)c3ccc(cc3)Br 3R-0826 CCOC(=O)Cc1c(=O)n(c2ccccc2n1)CC3CC3 3R-0827 CCOC(=O)Cc1c(=O)n(c2ccccc2n1)CC#N 3R-0829 CCOC(=O)C(=O)NCc1ccccc1 3R-0833 Cc1c(sc(n1)c2ccccc2)c3cc(c(c(n3)Br)C#N)c4ccccc4 3R-0834 CC(=O)C1(C(C1(C#N)C#N)c2ccc(cc2)[N+](=O)[O-])C(=O)C 3R-0835 CC(=O)C1(C(C1(C#N)C#N)c2ccccc2[N+](=O)[O-])C(=O)C 3R-0836 CNC(=O)C(=O)NCc1ccccc1 3R-0837 CC(C(=O)c1cn(nn1)c2ccsc2C(=O)OC)n3cncn3 3R-0838 Cc1c(sc(n1)c2ccccc2)c3ccnc(n3)NCCC[C@@H](C(=O)O)N 3R-0839 CC1(CC(=O)C2(C(C2(C#N)C#N)c3ccccc3[N+](=O)[O-])C(=O)C1)C 3R-0840 COC(=O)CS(=O)(=O)C 3R-0841 Cn1c(cnc1c2ccccc2)Cl 3R-0842 CCCCN1C(C(CCC1=O)C(=O)O)c2cccs2 3R-0844 CCCCN1C(C(CCC1=O)C(=O)O)c2cccc3c2OCO3 3R-0846 CC(C(=O)c1cn(nn1)c2ccc(cc2)C(=O)C)n3cncn3 3R-0848 CC(=O)c1ccc(cc1)n2cc(nn2)c3c(cc(cn3)C(F)(F)F)Cl 3R-0849 CC(C(=O)c1cn(nn1)c2ccc(cc2)C(=O)C)Oc3ccc(cc3Cl)Cl 3R-0850 CC(=O)c1ccc(cc1)n2cc(nn2)[N+](=O)[O-] 3R-0851 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)c3cccs3 3R-0853 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)C(C)(C)C 3R-0854 CCCCCC1CCC(CC1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C 3R-0855 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)Cc3ccccc3 3R-0856 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl 3R-0857 C/C(=C\C(=O)c1ccc(cc1Cl)Cl)/N(C)C 3R-0859 CC1(CC(=O)C2(C(C2(C#N)C#N)c3ccc(cc3)OC)C(=O)C1)C 3R-0860 Cc1c(sc(n1)c2cccnc2)C(=O)/C=C/Nc3ccc(cc3)OC 3R-0861 Cc1c(sc(n1)c2cccnc2)C(=O)/C=C/Nc3ccc(cc3)Cl 3R-0862 C/C(=C(\c1ccccc1)/C(=O)OC)/Nc2ccc(cc2F)Cl 3R-0864 CC1(CC(=O)C2(C(C2(C#N)C#N)c3ccc(cc3Cl)Cl)C(=O)C1)C 3R-0866 CC1(CC(=O)C2(C(C2(C#N)C#N)c3ccc(cc3)[N+](=O)[O-])C(=O)C1)C 3R-0867 CCCCCC1CCC(CC1)c2ccc3c(c2)c(c(cn3)C(=O)OCC)O 3R-0869 c1ccc2c(c1)c(nn(c2=O)Cc3ccc(cc3)F)CC#N 3R-0870 CCCCCC1CCC(CC1)c2ccc(cc2)NS(=O)(=O)c3ccc4ccccc4c3 3R-0872 CCCCCC1CCC(CC1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C(C)(C)C 3R-0873 COC(=O)Cc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 3R-0875 CN(C)/C=C(\C(=O)OC)/n1cncn1 3R-0876 Cc1c(c(=O)c2cc(cc(c2[nH]1)F)Cl)c3ccccc3 3R-0877 Cc1c(nnn1c2ccc(cc2)C(=O)C)C(=O)c3ccc(cc3Cl)Cl 3R-0878 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C 3R-0879 CCCCCC1CCC(CC1)c2ccc(cc2)NS(=O)(=O)c3cc(ccc3Cl)Cl 3R-0880 Cc1c(nnn1c2ccccc2C(F)(F)F)[N+](=O)[O-] 3R-0888 Cn1c(cc(n1)Oc2ccc(cn2)C(F)(F)F)C(F)(F)F 3R-1000 Cn1c(cc(n1)Oc2ncc(cn2)c3ccc(cc3)Cl)C(F)(F)F 3R-1002 COCc1cc(nc(n1)SCc2ccc(cc2)Cl)N3CCOCC3 3R-1003 COCc1cc(nc(n1)S(=O)(=O)Cc2ccc(cc2)Cl)N3CCOCC3 3R-1004 Cc1c(c2ccccc2[nH]1)C(=O)C(=O)N3CCCCC3 3R-1005 CCNC(=O)C(=O)c1c([nH]c2c1cccc2)C 3R-1006 Cc1c(cnc(n1)SC)C(=O)OC 3R-1007 Cc1c(cnc(n1)S(=O)C)C(=O)OC 3R-1008 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)O 3R-1011 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N3CCOCC3 3R-1015 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N3CCC4(CC3)OCCO4 3R-1016 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N3CCCCC3 3R-1018 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N3CCCCCC3 3R-1019 c1ccc(cc1)N2CCN(CC2)C(=O)C3CCN(CC3)S(=O)(=O)c4ccccc4 3R-1020 CC1CN(CC(O1)C)C(=O)C2CCN(CC2)S(=O)(=O)c3ccccc3 3R-1021 CN1CCN(CC1)C(=O)C2CCN(CC2)S(=O)(=O)c3ccccc3 3R-1022 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3)Cl 3R-1023 COc1ccc(cc1)NC(=O)C2CCN(CC2)S(=O)(=O)c3ccccc3 3R-1024 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)C3C(=O)CCCC3=O 3R-1025 CC(C)(C)NC(=O)C1CCN(CC1)S(=O)(=O)c2ccccc2 3R-1026 CC(COC)NC(=O)C1CCN(CC1)S(=O)(=O)c2ccccc2 3R-1027 CC1(CC(=O)C(C(=O)C1)C(=O)C2CCN(CC2)S(=O)(=O)c3ccccc3)C 3R-1028 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3)C(F)(F)F 3R-1029 CCOC(=O)c1cnn(c1c2ccccc2)c3ccccc3 3R-1030 c1ccc(cc1)c2c(cnn2c3ccccc3)C(=O)O 3R-1031 c1ccn(c1)c2ccsc2C(=O)Nc3ccc(cc3)Cl 3R-1032 COc1ccc(cc1)NC(=O)c2c(ccs2)n3cccc3 3R-1033 c1ccc(cc1)c2c(cnn2c3ccccc3)C(=O)N4CCOCC4 3R-1036 c1ccc(cc1)c2c(cnn2c3ccccc3)C(=O)N4CCCC4 3R-1037 CCNC(=O)c1cnn(c1c2ccccc2)c3ccccc3 3R-1038 C=CCNC(=O)c1cnn(c1c2ccccc2)c3ccccc3 3R-1039 c1ccc(cc1)c2c(cnn2c3ccccc3)C(=O)N4CCCCCC4 3R-1040 c1ccc(cc1)c2c(cnn2c3ccccc3)C(=O)Nc4ccc(cc4)Cl 3R-1041 c1ccc(cc1)c2c(cnn2c3ccccc3)C(=O)Nc4ccccc4 3R-1042 Cc1cccc(c1C)NC(=O)c2cnn(c2c3ccccc3)c4ccccc4 3R-1043 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3)Br 3R-1044 C=CCNC(=O)C1CCN(CC1)S(=O)(=O)c2ccccc2 3R-1045 c1ccc(cc1)SCC2(CCN(CC2)S(=O)(=O)c3ccccc3)O 3R-1061 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)(CSc3ccc(cc3)F)O 3R-1062 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)(CSc3ccc(cc3)Cl)O 3R-1063 c1ccc(cc1)N2CCN(CC2)CC3(CCN(CC3)S(=O)(=O)c4ccccc4)O 3R-1064 c1cc(ccc1S(=O)(=O)N2CCC3(CC2)CO3)Cl 3R-1065 c1cc(ccc1SCC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O)Cl 3R-1066 Cc1ccc(cc1)SCC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O 3R-1067 c1ccc(cc1)N2CCN(CC2)CC3(CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl)O 3R-1068 c1cc(ccc1S(=O)(=O)N2CCC(CC2)(CN3CCOCC3)O)Cl 3R-1069 c1cc(c(cc1Cl)Cl)/C=C/C(=O)OCC#N 3R-1070 c1cc(c(cc1Cl)Cl)/C=C/C(=O)NN 3R-1072 c1cc(ccc1S(=O)(=O)N2CCC(CC2)(CN3CCCC3)O)Cl 3R-1073 c1cc(ccc1S(=O)(=O)N2CCC(CC2)(CN3CCCCC3)O)Cl 3R-1074 CN1CCN(CC1)CC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O 3R-1075 c1cc(ccc1N2CCN(CC2)CC3(CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl)O)F 3R-1076 CCN(CC)CC1(CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl)O 3R-1077 c1ccc(cc1)CN2CCN(CC2)CC3(CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl)O 3R-1078 c1cc(ccc1S(=O)(=O)N2CCC(CC2)(CN3CCCCCC3)O)Cl 3R-1079 COC(=O)C1CCN(CC1)CC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O 3R-1080 c1cc(ccc1S(=O)(=O)N2CCC(CC2)(CN3CCC(=O)CC3)O)Cl 3R-1082 Cc1ccc(cc1)S(=O)(=O)N2CCC(=O)CC2 3R-1084 c1cc(ccc1SCC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O)Br 3R-1086 c1cc(ccc1F)SCC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O 3R-1087 COc1ccccc1SCC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)O 3R-1088 Cc1ccc(cc1)C(=O)Nn2ccc3c2nccc3 3R-1089 Cc1ccc(cc1)/C=N/n2ccc3c2nccc3 3R-1090 c1cc(c(cc1Cl)Cl)/C=C/c2nnc(o2)S 3R-1091 Cc1ccc(cc1)C(=O)NNC(=O)/C=C/c2ccc(cc2Cl)Cl 3R-1092 Cc1ccc(cc1)S(=O)(=O)NNC(=O)/C=C/c2ccc(cc2Cl)Cl 3R-1093 c1ccc(cc1)/C=C\C(=O)OCC#N 3R-1096 c1cc(cc(c1)Cl)/C(=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5Cl)Cl)/C#N 3R-1126 c1cc(cc(c1)C(F)(F)F)/C(=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5Cl)Cl)/C#N 3R-1127 Cc1cccc(c1)/C(=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5Cl)Cl)/C#N 3R-1128 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/O)Cl 3R-1132 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/OC(=O)C5CC5)Cl 3R-1134 Cc1ccc(cc1)C(=O)O/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl 3R-1135 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl 3R-1136 Cc1cccc(c1)CO/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl 3R-1144 c1cc(ccc1CO/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl)F 3R-1145 c1cc(cc(c1)F)CO/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl 3R-1146 CO/N=C/c1c(nc2n1c3c(s2)CCCC3)c4ccc(cc4)Cl 3R-1147 c1cc(cc(c1)C(F)(F)F)CO/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl 3R-1148 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/OCc5ccc(cc5Cl)Cl)Cl 3R-1149 Cc1c(cnc(n1)SC)C(=O)C 3R-1150 CC(=O)N(C(=O)C)N1C(=O)C2C3c4ccccc4C(C2C1=O)c5c3cccc5 3R-1152 CC(=O)/C(=C\N(C)C)/C(=O)OC 3R-1153 COc1cccc(c1)/C(=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl)/C#N 3R-1154 c1cc(cc(c1)Cl)/C(=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl)/C#N 3R-1155 Cc1c(cnc(n1)NC(C)C)C(=O)NC(C)C 3R-1157 c1cc(sc1)C(=O)O/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl 3R-1159 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/OC(=O)c5ccc(cc5)Cl)Cl 3R-1160 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/OC(=O)c5ccc(cc5)F)Cl 3R-1161 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/OC(=O)c5ccc(c(c5)Cl)Cl)Cl 3R-1162 c1ccc(c(c1)C(=O)O/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl)Cl 3R-1163 c1cc(cc(c1)C(F)(F)F)/C(=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl)/C#N 3R-1164 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=C(\C#N)/c5ccc(c(c5)Cl)Cl)Cl 3R-1165 COc1ccc(cc1OC)/C(=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl)/C#N 3R-1166 Cc1c(cnc(n1)SC)C(=O)O 3R-1168 Cc1c(cnc(n1)SCc2c(cccc2Cl)Cl)C(=O)C 3R-1169 Cc1c(cnc(n1)S)C(=O)O 3R-1172 Cc1c(cnc(n1)SCc2ccc(cc2)Cl)C(=O)C 3R-1174 Cc1c(cnc(n1)SCc2ccc(c(c2)Cl)Cl)C(=O)C 3R-1175 Cc1c(cnc(n1)SCCN2C(=O)c3ccccc3C2=O)C(=O)C 3R-1176 Cc1c(cnc(n1)SCN2C(=O)c3ccccc3C2=O)C(=O)C 3R-1177 COc1ncc(cn1)c2ccc(cc2)Cl 3R-1179 Cc1c(n2ccccc2n1)C(=O)CN3CCOCC3 3R-1181 Cc1c(n2ccccc2n1)C(=O)/C=C/c3c(cccc3Cl)Cl 3R-1182 Cc1c(n2ccccc2n1)C(=O)/C=C/c3ccc(cc3)F 3R-1183 Cc1c(n2cc(ccc2n1)Cl)C(=O)C 3R-1184 Cc1ccn2c(c1)nc(c2C(=O)C)C 3R-1187 Cc1c(n2ccccc2n1)C(=O)CN3CCN(CC3)C(c4ccccc4)c5ccccc5 3R-1188 Cc1ccn2c(c1)nc(c2C(=O)CSc3ccc(cc3)Cl)C 3R-1192 Cc1ccn2c(c1)nc(c2C(=O)CSc3ccc(cc3)Br)C 3R-1193 Cc1ccc(cc1)SCC(=O)c2c(nc3n2ccc(c3)C)C 3R-1194 Cc1ccn2c(c1)nc(c2C(=O)CSc3cccc(c3)Cl)C 3R-1195 Cc1ccn2c(c1)nc(c2C(=O)CSc3ccccc3Cl)C 3R-1196 Cc1ccn2c(c1)nc(c2C(=O)CSc3ccccc3)C 3R-1197 Cc1ccn2c(c1)nc(c2C(=O)CSc3cccc(c3Cl)Cl)C 3R-1198 Cc1ccn2c(c1)nc(c2C(=O)CSc3ccc(cc3)F)C 3R-1199 Cc1ccn2c(c1)nc(c2C(=O)CSc3ccccc3C)C 3R-1200 Cc1ccn2c(c1)nc(c2C(=O)CSc3ccc(cc3Cl)Cl)C 3R-1201 Cc1ccn2c(c1)nc(c2C(=O)CSc3cccc(c3)C(F)(F)F)C 3R-1202 Cc1ccn2c(c1)nc(c2/C(=N/O)/C)C 3R-1203 Cc1ccn2c(c1)nc(c2/C(=N/O)/CSc3ccc(cc3)Cl)C 3R-1207 c1ccc(cc1)CSC\2=Nc3ccccc3/C2=N/Nc4c(cc(cc4Cl)Cl)Cl 3R-1240 c1ccc(c(c1)CSC\2=Nc3ccccc3/C2=N/Nc4c(cc(cc4Cl)Cl)Cl)Cl 3R-1242 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=N2)SCc4ccc(c(c4)Cl)Cl 3R-1243 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=N2)SCc4ccc(cc4)F 3R-1244 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=N2)SCc4cccc(c4)Cl 3R-1245 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=N2)SCc4ccc(cc4Cl)Cl 3R-1246 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=N2)SCc4c(cccc4Cl)Cl 3R-1247 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4ccc(cc4)Cl 3R-1249 Cc1ccc(cc1)Cn2c(=O)cc3c(n2)-c4ccccc4CC3 3R-1250 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4ccc(c(c4)Cl)Cl 3R-1252 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4c(cccc4Cl)Cl 3R-1253 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4ccccc4Cl 3R-1254 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4ccc(cc4Cl)Cl 3R-1255 c1ccc2c(c1)/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C(=N2)SCc4cccc(c4)[N+](=O)[O-] 3R-1257 CCSC\1=Nc2ccccc2/C1=N/Nc3c(cc(cc3Cl)Cl)Cl 3R-1261 Cc1ccc(cc1)CSc2cc3c(nn2)-c4ccccc4CC3 3R-1262 CCCSC\1=Nc2ccccc2/C1=N/Nc3c(cc(cc3Cl)Cl)Cl 3R-1263 CC(C)SC\1=Nc2ccccc2/C1=N/Nc3c(cc(cc3Cl)Cl)Cl 3R-1264 CC(C)CSC\1=Nc2ccccc2/C1=N/Nc3c(cc(cc3Cl)Cl)Cl 3R-1265 CCC(C)SC\1=Nc2ccccc2/C1=N/Nc3c(cc(cc3Cl)Cl)Cl 3R-1266 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4ccc(cc4)F 3R-1272 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4cccc(c4)Cl 3R-1273 c1ccc-2c(c1)CCc3c2nn(c(=O)c3)Cc4cccc(c4)[N+](=O)[O-] 3R-1274 c1cc(cc(c1)n2c(nnc2S)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl)C(F)(F)F 3R-1300 CSc1nnc(n1c2cccc(c2)C(F)(F)F)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 3R-1301 C=CCSc1nnc(n1c2cccc(c2)C(F)(F)F)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 3R-1302 COc1ccc(cc1)CSc2nnc(n2c3cccc(c3)C(F)(F)F)C4CCN(CC4)S(=O)(=O)c5ccc(cc5)Cl 3R-1303 c1ccc(cc1)CSc2nnc(n2c3cccc(c3)C(F)(F)F)C4CCN(CC4)S(=O)(=O)c5ccc(cc5)Cl 3R-1304 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)OC 3R-1306 COC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 3R-1307 COC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(cc2)F 3R-1308 COC(=O)C1CCN(CC1)S(=O)(=O)c2ccccc2 3R-1309 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)OC 3R-1310 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NN 3R-1312 c1coc2c1/C(=N\O)/CCC2 3R-1314 c1coc2c1C(=O)NCCC2 3R-1315 c1cc(ccc1C(=O)O/N=C\2/CCCc3c2cco3)F 3R-1317 c1ccc(cc1)NC(=O)c2csc(n2)Cc3cccc(c3)C(F)(F)F 3R-1501 CNC(=O)Cc1ccccc1 3R-1505 COc1ccc(cc1)NC(=O)Cc2nc(no2)c3ccc(cc3)Cl 3R-1514 Cc1ccc(c(c1)C)NC(=O)Cc2nc(no2)c3ccc(cc3)Cl 3R-1515 COc1ccc(cc1)NC(=O)Cc2nc(no2)c3cccc(c3)Cl 3R-1516 Cc1ccc(c(c1)C)NC(=O)Cc2nc(no2)c3cccc(c3)C(F)(F)F 3R-1517 c1cc(cc(c1)C(F)(F)F)Cc2nc(cs2)C(=O)Nc3cccc(c3)C(F)(F)F 3R-1518 COc1ccccc1CNC(=O)c2csc(n2)Cc3cccc(c3)C(F)(F)F 3R-1520 c1ccc2c(c1)nc(n2CC#N)C(F)(F)F 3R-1522 c1cc(cc(c1)C(F)(F)F)Cc2nc(cs2)C(=O)Nc3ccc(cc3Cl)Cl 3R-1524 c1cc(cc(c1)C(F)(F)F)Cc2nc(cs2)C(=O)Nc3ccc(c(c3)Cl)Cl 3R-1525 C/C(=N/NC(=O)N)/Cn1c2ccccc2nc1C(F)(F)F 3R-1526 COc1ccccc1NC(=O)Cn2c3ccccc3nc2C(F)(F)F 3R-1527 COc1cccc(c1)NC(=O)Cn2c3ccccc3nc2C(F)(F)F 3R-1528 c1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccc(cc3Cl)Cl 3R-1529 c1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccc(c(c3)Cl)Cl 3R-1530 c1ccc(cc1)Cc2nc(cs2)C(=O)Nc3cc(cc(c3)Cl)Cl 3R-1531 c1ccc(cc1)Cc2nc(cs2)C(=O)Nc3ccc(cc3)F 3R-1532 COC(=O)CCNC(=O)Nc1cccc(c1)Cl 3R-1533 c1cc(cc(c1)Cl)NC(=O)NCCC(=O)O 3r-1534 COc1ccc(cc1)CNC(=O)c2csc(n2)Cc3ccccc3 3R-1544 c1cc(cc(c1)C(F)(F)F)Cc2nc(cs2)C(=O)Nc3cc(ccc3Cl)Cl 3R-1545 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)O 3R-1549 Cc1c(cnc(n1)SCc2ccc(c(c2)Cl)Cl)C(=O)O 3R-1552 Cc1c(cnc(n1)SCc2ccc(cc2)Cl)C(=O)O 3R-1555 Cc1ccc(cc1)Sc2c(nnc(n2)c3ccccc3)C(F)(F)F 3R-1561 CCOc1ccc(cc1)NC(=O)Cn2c3ccccc3nc2C(F)(F)F 3R-1565 CCOc1ccccc1NC(=O)Cn2c3ccccc3nc2C(F)(F)F 3R-1566 c1ccc2c(c1)nc(n2CC(=O)Nc3ccccc3Cl)C(F)(F)F 3R-1567 c1ccc2c(c1)nc(n2CC(=O)Nc3cccc(c3)Cl)C(F)(F)F 3R-1568 c1ccc2c(c1)nc(n2CC(=O)Nc3ccc(cc3)Cl)C(F)(F)F 3R-1569 c1ccc2c(c1)nc(n2CC(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F 3R-1570 c1ccc(c(c1)C(F)(F)F)NC(=O)Cn2c3ccccc3nc2C(F)(F)F 3R-1571 c1ccc2c(c1)nc(n2CC(=O)Nc3cc(ccc3Cl)C(F)(F)F)C(F)(F)F 3R-1574 c1ccc(cc1)c2csc(n2)n3cc(cn3)c4ccc(cc4)Cl 3T-0001 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(c(s2)S(=O)(=O)c3ccc(cc3)Cl)c4ccccc4 3T-0005 c1cc(ccc1Sc2c(nc(s2)n3c(ccn3)c4ccc(cc4Cl)Cl)c5ccc(cc5Cl)Cl)Cl 3T-0007 c1ccc(cc1)COc2ccc3ccc(cc3c2)O 3T-0008 Cc1c2c([nH]n1)NC3=C(C2c4ccccc4)C(=O)CC(C3)(C)C 3T-0010 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(o3)c4ccc(cc4Cl)Cl 3T-0011 c1cc(c(c(c1)Cl)CN2CCC(CC2)CC(=O)O)Cl 3T-0012 c1cc(ccc1C(=O)N2CCC(=O)CC2)[N+](=O)[O-] 3T-0014 c1ccc(cc1)C(=O)C(c2ccccc2)(Br)Br 3T-0015 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCC(=O)CC2 3T-0017 c1ccc(cc1)C(=O)CSc2nc[nH]n2 3T-0019 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(s3)Cl 3T-0020 CCOc1nc(c(s1)S(=O)(=O)c2ccc(cc2)Cl)c3ccccc3 3T-0021 c1cc(c(cc1Cl)Cl)c2ccc(o2)c3csc(n3)n4c(c(cn4)C(=O)O)C(F)(F)F 3T-0023 c1c(c(n(n1)c2nc(cs2)C(F)(F)F)C(F)(F)F)C(=O)O 3T-0024 CCN(CC)c1ccc(c(c1)O)C(=O)C(F)(F)F 3T-0029 Cc1cc(n(n1)c2nc(c(s2)Sc3ccc(cc3)Cl)c4ccc(cc4Cl)Cl)C 3T-0031 Cn1c(c(cn1)C(=O)CC#N)C(F)(F)F 3T-0032 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(c(s2)Sc3ccc(cc3)Cl)c4ccc(cc4Cl)Cl 3T-0033 CCOC(=O)C/C(=N\Nc1nc(cs1)c2ccccc2)/C 3T-0038 CCO/C=C(\C#N)/S(=O)(=O)C(C)(C)C 3T-0039 Cc1c2c([nH]n1)NC3=C(C2c4ccoc4)C(=O)CC(C3)(C)C 3T-0040 CC(C)(C)S(=O)(=O)c1cnn(c1N)c2nc(cs2)c3ccccc3 3T-0041 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)S(=O)(=O)C(C)(C)C)C 3T-0045 c1cc(ccc1C(=O)N2CCC(CC2)O)[N+](=O)[O-] 3T-0049 CCOC(=O)/C(=N\OC)/C(C(F)(F)F)O 3T-0051 CCOC(=O)C=C1CCN(CC1)C(=O)c2cccc(c2)C(F)(F)F 3T-0054 COC(=O)c1cnn(c1N)c2nc(cs2)c3ccccc3 3T-0055 Cn1c(c(cn1)c2cc([nH]n2)N)C(F)(F)F 3T-0058 Cc1ccc(n1c2c(cnn2c3nc(cs3)c4ccccc4)c5ccc(cc5)Cl)C 3T-0060 Cc1cc(n2c(n1)cc(n2)c3cnn(c3C(F)(F)F)C)C 3T-0061 c1cc2c(cc1[N+](=O)[O-])[nH]c(=O)o2 3T-0063 CCN(CC)c1ccc2c(c1)oc(=O)c(c2C(F)(F)F)C(=O)O 3T-0064 Cc1cc(n2c(n1)c(c(n2)c3cnn(c3C(F)(F)F)C)Cl)C 3T-0067 COC(=O)c1ccc(cc1)N2CCOCC2 3T-0068 CCO/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)C 3T-0076 c1ccc(cc1)C2(Nc3ccccc3C(=O)N2)CO 3T-0081 c1cc(c(cc1[N+](=O)[O-])F)N2CCC(=O)CC2 3T-0082 CCO/C=C(\C#N)/S(=O)(=O)C 3T-0083 Cc1c(c(n(n1)c2nc(c(s2)Cl)c3ccc(cc3)Cl)C)Cl 3T-0084 Cc1c(c(n(n1)c2nc(c(s2)Cl)c3ccc(cc3)F)C)Cl 3T-0085 c1cc(nnc1Cl)I 3T-0088 COc1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C=O)C(=O)OC 3T-0206 CN(C)/C=C\1/C(=Nc2ccccc2O1)Cl 3T-0209 c1ccc(c(c1)C(=O)c2ccc3c(c2)NC(=O)CO3)C(=O)NCc4ccc(cc4)F 3T-0212 c1ccc(c(c1)C(=O)c2ccc3c(c2)NC(=O)CO3)C(=O)NC4CCCCC4 3T-0213 c1cc(c(cc1[N+](=O)[O-])CO)O 3T-0215 Cc1nnc(n1Cc2ccc(c(c2)OC)OC)c3cnn(c3N)C 3T-0217 c1ccc(c(c1)C(=O)c2ccc3c(c2)NC(=O)CO3)C(=O)NCc4cccc(c4)Cl 3T-0218 c1ccc(cc1)c2c3c(c(c(n2)SCC#N)C#N)CCCC3 3T-0219 c1c(cnc(c1C(F)(F)F)N2CCNCC2)C(F)(F)F 3T-0220 COC(=O)CSc1c(c2c(c(n1)c3ccccc3)CCCC2)C#N 3T-0221 CN1CCN(CC1)c2c(cccn2)N 3T-0223 Cc1ccccc1c2c3c(c(c(n2)SCc4ccc(cc4)F)C#N)CCC3 3T-0224 Cc1ccc(cc1)CSc2c(c3c(c(n2)c4ccccc4C)CCC3)C#N 3T-0225 COc1ccc(cc1)C(=O)N2c3ccccc3OCC2CC(=O)OC 3T-0226 COC(=O)CC1COc2ccccc2N1C(=O)c3ccco3 3T-0227 COC(=O)c1c(c2c3c(c(nc2s1)c4ccccc4)CCCC3)N 3T-0228 Cc1cc(ccc1N/C(=C\C(=O)c2ccc3c(c2)c(on3)c4ccc(cc4)F)/C)F 3T-0229 CC(C)(C)c1ccc(cc1)CSc2c(c3c(c(n2)c4ccc(cc4)C(C)(C)C)CCC3)C#N 3T-0231 c1cc(c(cc1C(=O)O)F)N 3T-0232 c1ccc(cc1)n2cc3c(n2)Nc4ccccc4O3 3T-0237 COc1ccc(cc1)C(=O)N2c3ccccc3OCC2CC(=O)O 3T-0238 Cc1ccc(cc1)C(=O)Nc2cccnc2N3CCN(CC3)C 3T-0239 CN1C(C2=C(c3ccccc3C2=O)NC1=O)c4ccccc4F 3T-0244 c1ccc(cc1)c2c3c(c4c(c(sc4n2)C#N)N)CCCC3 3T-0249 c1cc(ccc1c2cn3ccsc3n2)Br 3T-0252 CN1CCN(CC1)c2c(cccn2)NC(=O)C3CC3 3T-0255 CC(=O)C(C/C=C/c1ccccc1)C(=O)C 3T-0261 c1cc(ccc1CNC(=O)c2cc(cc(c2O)I)I)F 3T-0263 Cc1ccc(c(c1)CN2c3cc(ccc3OCC2=O)C(=O)c4ccccc4C(=O)O)C 3T-0266 c1ccc(c(c1)C(=O)c2ccc3c(c2)N(C(=O)CO3)Cc4ccc(c(c4)Cl)Cl)C(=O)O 3T-0267 c1c(cc(c2c1[nH]c(=O)o2)I)I 3T-0269 c1cc(ccc1C=O)n2cncn2 3T-0275 COC(=O)CC1COc2ccccc2N1Cc3ccccc3 3T-0276 CC(=O)OC(c1ccc(c(c1)N)Oc2ccc(cc2)C(=O)OC)OC(=O)C 3T-0277 Cc1ccc(cc1)c2c(n3ccsc3n2)C=C4C(=O)NC(=O)NC4=O 3T-0283 Cc1ccc(cc1)c2c(n3ccsc3n2)C=C4C(=O)OC(OC4=O)(C)C 3T-0284 c1cc(ccc1c2c(n3ccsc3n2)C=O)Br 3T-0286 c1cc(ccc1C=O)n2ccnc2 3T-0287 c1cc(c(cc1N)CO)O 3T-0288 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4ccc(cc4)Cl 3T-0291 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl 3T-0292 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=C/C(=O)c4ccc(cc4)Cl 3T-0293 COc1ccc(cc1)C(=O)n2c3cc(cc(c3oc2=O)I)I 3T-0294 c1cc(ccc1c2ccc(cc2)Br)C(=O)O 3T-0295 Cc1ccc(cc1)c2c(n3ccsc3n2)C=C4C(=O)N(C(=O)N(C4=O)C)C 3T-0297 Cc1ccc(cc1)c2c(n3ccsc3n2)C=C4C(=O)c5ccccc5C4=O 3T-0298 c1cc(ccc1CO)n2cncn2 3T-0299 CN1CCN(CC1)c2ccc(cc2)C=O 3T-0301 COC(=O)CC1COc2ccccc2N1S(=O)(=O)c3ccc(cc3)Br 3T-0302 c1ccc(c(c1)C(=O)c2ccc3c(c2)NC(=O)CO3)C(=O)NC4CC4 3T-0303 CN1C(=O)C(=Cc2ccc(cc2)n3cncn3)C(=O)N(C1=O)C 3T-0304 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4c(cccc4Cl)F 3T-0305 C1CC1C(=O)N/C(=C(/C#N)\[NH3+])/C#N.[Cl-] 3T-0307 c1ccc(c(c1)C(=O)c2ccc3c(c2)NC(=O)CO3)C(=O)NCc4ccco4 3T-0308 c1cnn(c1)c2ccc(cc2)C=O 3T-0309 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=N/OCc4ccc(cc4)C(C)(C)C 3T-0311 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=C(\C#N)/S(=O)(=O)c4ccccc4 3T-0312 COc1ccc(cc1)S(=O)(=O)N2c3ccccc3OCC2CC(=O)OC 3T-0315 c1ccc2c(c1)N(C(CO2)CC(=O)O)S(=O)(=O)c3ccc(cc3)Br 3T-0316 COC(=O)CC1COc2ccccc2N1S(=O)(=O)c3ccc4ccccc4c3 3T-0317 c1cc(ccc1CO)n2ccnc2 3T-0318 Cc1ccc(cc1)c2c(n3ccsc3n2)CO 3T-0319 COc1cc(cc(c1OC)OC)C=C2C(=O)c3ccccc3C2=O 3T-0321 c1ccc2c(c1)ncn2c3ccc(cc3)C=O 3T-0322 c1ccc(cc1)C(=O)COC(=O)c2ccccc2N 3T-0323 Cc1cccc(c1)c2c3c(c(c(n2)SCC#N)C#N)CCCC3 3T-0325 Cc1cccc(c1)c2c3c(c(c(n2)SCc4ccc(c(c4)Cl)Cl)C#N)CCCC3 3T-0326 Cc1cccc(c1)CSc2c(c3c(c(n2)c4cccc(c4)C)CCCC3)C#N 3T-0327 Cc1cccc(c1)c2c3c(c(c(n2)SCc4cccc(c4)F)C#N)CCCC3 3T-0328 CN1CCN(CC1)c2ccc3c(c2)[nH]c(n3)c4cccc(c4)OC 3T-0330 Cc1ccc(cc1)c2c(n3ccsc3n2)/C=C(\C#N)/S(=O)(=O)C 3T-0331 c1ccc2c(c1)ncn2c3ccc(cc3)CO 3T-0332 c1ccc(c(c1)C(=O)c2ccc3c(c2)N(C(=O)CO3)Cc4cccc(c4)F)C(=O)O 3T-0335 Cc1cccc(c1)c2c3c(c(c(n2)SCC(=O)OC)C#N)CCCC3 3T-0336 c1cc(c(c(c1)Cl)CO/N=C/c2c(nc3n2ccs3)c4ccc(cc4)Br)F 3T-0338 c1cc(ccc1c2c(n3ccsc3n2)CO)Br 3T-0339 Cc1ccc(cc1)C(=O)/C=C/c2c(nc3n2ccs3)c4ccc(cc4)Br 3T-0340 c1ccc2cc(ccc2c1)S(=O)(=O)N3c4ccccc4OCC3CC(=O)O 3T-0341 COc1ccc(cc1)S(=O)(=O)N2c3ccccc3OCC2CC(=O)O 3T-0342 c1cc(ccc1C(=O)n2c3cc(cc(c3oc2=O)I)I)C(F)(F)F 3T-0343 c1cc(ccc1C(=O)n2c3cc(cc(c3oc2=O)I)I)F 3T-0344 c1cc(c(c(c1)Cl)C(C#N)c2ccc(nn2)Sc3ccc(cc3F)F)Cl 3T-0345 c1cc(ccc1CO/N=C/c2c(nc3n2ccs3)c4ccc(cc4)Br)C(F)(F)F 3T-0346 CN1c2ccccc2OCC1=O 3T-0348 CN1CCN(CC1)c2ccc(c(c2)N)NC(=O)c3cccc(c3)Cl 3T-0349 c1cc(c(cc1N2CCOCC2)N)[N+](=O)[O-] 3T-0352 c1ccc(cc1)C(=O)N/N=C/c2c(nc3n2ccs3)c4ccc(cc4)Br 3T-0354 CC1(OC(=O)C(=Cc2c(nc3n2ccs3)c4ccc(cc4)Br)C(=O)O1)C 3T-0356 CN1C(C2=C(c3ccccc3C2=O)NC1=S)c4cc(c(c(c4)OC)OC)OC 3T-0358 CNC(=S)Nc1ccccc1N 3T-0361 c1cc2c(cc1[N+](=O)[O-])OCC(=O)N2 3T-0362 CN1CCN(CC1)c2ccc3c(c2)[nH]c(n3)C4CCCCC4 3T-0363 CN1C(=O)C(=Cc2c(nc3n2ccs3)c4ccc(cc4)Br)C(=O)N(C1=O)C 3T-0364 COc1ccc(cc1)c2c[nH]cn2 3T-0366 Cc1cc(c(cc1N2CCN(CC2)c3ccccc3)NC(=O)C)[N+](=O)[O-] 3T-0600 Cc1ccc(cc1)C(=O)NC2CC(=O)c3c2cc(c(c3)OC)OC 3T-0601 CN(C)/C=C/C(=O)c1c(ccs1)Br 3T-0603 C/C(=C\C(=O)c1c(ccs1)Br)/N(C)C 3T-0604 Cc1ccsc1c2cc(nc(n2)N)C 3T-0607 c1cnc(nc1c2c(ccs2)Br)N 3T-0608 c1ccc(cc1)N2CCN(CC2)C(=O)CC(c3cccs3)NC(=O)C(F)(F)F 3T-0609 Cc1cc(nc(n1)N)c2c(ccs2)Br 3T-0610 COC(=O)C1CCN(CC1)C(=O)CC(c2cccs2)NC(=O)C(F)(F)F 3T-0613 c1cc2nc(cn2cc1Cl)c3ccc(s3)Br 3T-0615 COc1cc2c(cc1OC)C(=O)/C(=C/c3ccc(cc3)Cl)/C2NC(=O)C(F)(F)F 3T-0619 c1cnc2nc(cn2c1)c3ccc(s3)Br 3T-0620 COc1cccc2c1oc(=O)c(c2)C(=O)O 3T-0621 CCc1ccc(cc1)C(CC(=O)NCc2ccc(cc2)OC)NC(=O)C(F)(F)F 3T-0622 c1cc(ccc1C(CC(=O)O)N)Cl 3T-0623 CCc1ccc(cc1)C(CC(=O)Nc2ccc3c(c2)OCO3)NC(=O)C(F)(F)F 3T-0624 COC(=O)c1ccc(cc1)C(CC(=O)O)NC(=O)C(F)(F)F 3T-0625 Cc1c(nc2c(n1)cccn2)C 3T-0629 c1cc(sc1)c2ccnc(n2)S 3T-0630 CCOc1ccc(cc1)C(CC(=O)O)NC(=O)C(F)(F)F 3T-0633 c1cc(ccc1C(CC(=O)O)NC(=O)C(F)(F)F)Cl 3T-0634 COc1cc2c(cc1OC)C(=O)/C(=C\c3cccs3)/C2NC(=O)C(F)(F)F 3T-0640 c1ccc2c(c1)ncc(n2)c3ccc(cc3)Cl 3T-0641 COC(=O)c1ccc(cc1)C(CC(=O)N)NC(=O)C(F)(F)F 3T-0646 c1ccn2cc(nc2c1)c3cccc(c3)[N+](=O)[O-] 3T-0650 c1ccc2c(c1)ncc(n2)c3cccc(c3)[N+](=O)[O-] 3T-0651 c1cc(cc(c1)[N+](=O)[O-])c2cn3cccnc3n2 3T-0652 c1cc(cc(c1)[N+](=O)[O-])c2cn3cc(ccc3n2)I 3T-0653 c1cc(sc1)/C=C/C(=O)O 3T-0655 c1ccc(c(c1)C(CC(=O)O)NC(=O)C(F)(F)F)Br 3T-0659 c1cc(ccc1C(CC(=O)O)NC(=O)C(F)(F)F)F 3T-0660 Cc1c(c2nccc(n2n1)c3ccc(o3)c4ccc(cc4Cl)Cl)Br 3T-0803 c1cc(ccc1c2cnn(c2N)c3nc(cs3)c4ccc(cc4)Cl)F 3T-0804 c1ccc(cc1)c2ccc(cc2)c3csc(n3)n4c(c(cn4)c5ccc(cc5)F)N 3T-0805 c1cc(ccc1c2cnn(c2N)c3nc(cs3)c4ccc(cc4Cl)Cl)F 3T-0806 Cc1c(sc(n1)N(c2ccccc2)C(=O)c3ccccc3)C(=O)C 3T-0807 Cc1c(c(n2c(n1)c(cn2)c3ccc(cc3)Cl)N)c4ccc(cc4)F 3T-0810 c1ccc(cc1)S(=O)(=O)c2cnn3c2nc(cc3C(F)(F)Cl)c4ccc(cc4)C(F)(F)F 3T-0811 COc1ccc(cc1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4Cl)Cl 3T-0812 c1cc(ccc1c2cc(c(c(=S)[nH]2)C#N)C(F)(F)F)F 3T-0813 COc1ccc(cc1)c2cnn(c2N)c3nc(cs3)c4ccccc4 3T-0814 COc1ccc(cc1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4)Cl 3T-0815 COc1ccc(cc1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4)F 3T-0816 COc1ccccc1c2cc(c(c(=S)[nH]2)C#N)C(F)(F)F 3T-0817 COc1cccc(c1)c2cc(c(c(=S)[nH]2)C#N)C(F)(F)F 3T-0818 COC(=O)C(/C=N/Nc1c(cc(cn1)C(F)(F)F)Cl)n2cncn2 3T-0819 c1cc(nc(c1)F)n2c(c(cn2)n3cncn3)O 3T-0820 COC(=O)Cc1cc(n2c(n1)nc(n2)SC)O 3T-0823 CC(C(=O)OC)Oc1ccc(cc1)O 3T-0825 CC(C(=O)OC)Oc1ccc(cc1)OC(C)C(=O)OC 3T-0826 c1c(cnc(c1Cl)C#CCO)C(F)(F)F 3T-0828 CC(C)(C#Cc1c(cc(cn1)C(F)(F)F)Cl)O 3T-0829 CCOC(=O)C(=O)Nc1c(ccs1)C(=O)N 3T-0832 c1cc(sc1)c2ccnc(n2)NS(=O)(=O)c3ccc(cc3)N 3T-0836 COc1ccc(cc1)c2csc(n2)n3c(c(cn3)c4cccs4)N 3T-0839 COc1ccc(cc1)c2csc(n2)n3c(c(cn3)c4ccsc4)N 3T-0840 COc1ccc(cc1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4)OC 3T-0841 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)c4ccccc4)C(F)(F)F 3T-0843 Cc1c(sc(n1)c2ccc(cc2)F)C(=O)C 3T-0845 Cc1c(sc(n1)c2cccc(c2)F)C(=O)C 3T-0846 COc1ccc(cc1)c2cc(c(c(=S)[nH]2)C#N)C(F)(F)F 3T-0848 c1ccc(c(c1)c2ncc(s2)c3c(cnc(n3)N)Br)Cl 3T-0849 c1cc(sc1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4)F 3T-0850 c1cc(sc1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4Cl)Cl 3T-0851 c1cc(sc1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4)Br 3T-0852 COc1ccc(cc1)NC(=O)OCC#Cc2c(cc(cn2)C(F)(F)F)Cl 3T-0854 COc1ccc(cc1)c2cnn(c2N)c3nc-4c(s3)COc5c4cccc5 3T-0856 COc1ccc(cc1)c2cnn(c2N)c3nc(c(s3)Sc4ccc(cc4)Cl)c5ccc(cc5)OC 3T-0857 COc1ccc(cc1)c2cnn(c2N)c3nc(c(s3)CC(=O)O)c4ccccc4 3T-0858 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)N)c5ccc(cc5)F)C)C 3T-0859 Cc1cc2nc(c(c(n2n1)N)c3ccc(cc3)F)C 3T-0861 Cc1c(c2nccc(n2n1)c3cccs3)Cl 3T-0862 Cc1c(c2nccc(n2n1)c3cccs3)Br 3T-0863 CC(=O)c1c(cc(cn1)C(F)(F)F)OCC(C(C(C(F)F)(F)F)(F)F)(F)F 3T-0864 Cc1c(c(n2c(n1)ncn2)O)C/C=C/c3ccccc3 3T-0865 CC(c1c(cc(cn1)C(F)(F)F)Cl)Oc2ccc(cc2Cl)Cl 3T-0866 COc1ccc(cc1)c2cnn(c2N)c3nc(cs3)c4ccccc4F 3T-0867 c1ccc(c(c1)c2csc(n2)n3c(c(cn3)c4ccsc4)N)F 3T-0868 Cc1cc2ncc(cn2n1)c3ccc(cc3)Cl 3T-0871 CN(C)/C=C(\C#N)/c1ccccn1 3T-0872 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3cccs3 3T-0874 Cc1c(c2ncc(cn2n1)c3ccc(cc3)Cl)Cl 3T-0877 Cc1c(c2ncc(cn2n1)c3ccc(cc3)Cl)Br 3T-0878 Cc1ccc(n1c2ccsc2c3cc4ncc(cn4n3)c5ccc(cc5)Cl)C 3T-0880 Cc1c(sc(n1)c2ccc(cc2)F)C(=O)/C=C/N(C)C 3T-0881 Cc1c(sc(n1)c2cccc(c2)F)C(=O)/C=C/N(C)C 3T-0882 Cc1ccc(cc1)c2cnc3cc(nn3c2)c4c(ccs4)n5c(ccc5C)C 3T-0884 c1cc(cc(c1)Cl)N2CCN(CC2)c3nc([nH]n3)N 3T-0887 Cc1ccc(cc1)c2cnc3cc(nn3c2)C 3T-0888 Cc1ccc(cc1)c2cnc3c(c(nn3c2)C)Cl 3T-0889 CC1=Nc2ccccc2Oc3c1ncc(c3)C(F)(F)F 3T-0890 Cc1ccc(cc1)c2cnc3c(c(nn3c2)C)Br 3T-0891 c1cc(cc(c1)Cl)N2CCN(CC2)c3nc4nc(cc(n4n3)C(F)(F)F)c5ccc(cc5)F 3T-0892 CC(C)(C)NC(=S)N1CCN(CC1)c2ccc(cc2)OC 3T-0893 CCOC(=O)C(Cc1ccc(cc1)F)(Cc2ccc(cc2)F)C(=O)C 3T-0894 c1ccnc(c1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4)F 3T-0895 COc1ccc(cc1)c2csc(n2)n3c(c(cn3)c4ccccn4)N 3T-0896 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)c5ccc(cc5)OC)C 3T-0897 c1cc(sc1)c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F 3T-0900 c1c(cnc(c1Cl)CC(=O)NCCCNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 3T-0903 c1cc(cc(c1)Br)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 3T-0904 COc1ccc(cc1)c2cnc3c(cnn3c2N)c4ccc(cc4)F 3T-0905 COc1ccc(cc1)c2c(sc(n2)c3ccccn3)Sc4ccc(cc4)Cl 3T-0906 Cc1cc2nc(c(c(n2n1)O)C/C=C/c3ccccc3)C 3T-0910 CC1(OCCO1)c2cnc(s2)c3ccc(cc3)Cl 3T-0911 Cc1cc2ncc(c(n2n1)N)c3cccs3 3T-0913 COc1ccc(cc1)N2CCN(CC2)C(=O)Cn3cncn3 3T-0914 c1ccc(cc1)S(=O)(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F 3T-0919 c1cc(sc1)c2cnc3c(cnn3c2N)c4ccc(cc4)F 3T-0920 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)c5cccs5)C 3T-0921 CC(C)(C)S(=O)(=O)c1cnc2c(cnn2c1N)c3ccc(cc3)F 3T-0922 Cc1cc2ncc(c(n2n1)N)S(=O)(=O)C(C)(C)C 3T-0923 c1c(cnc(c1Cl)CC(=O)NC23CC4CC(C2)CC(C4)C3)C(F)(F)F 3T-0926 Cc1ccc(cc1NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)F 3T-0928 CSc1nc2nc(cc(n2n1)c3ccccc3)C(F)(F)F 3T-0929 Cc1cc(nc2n1nc(n2)SC)C(F)(F)Cl 3T-0930 c1cc(ccc1c2cnn3c2ncc(c3N)c4ccc(cc4)Cl)F 3T-0931 Cc1cc(n2c(n1)c(cn2)c3ccc(cc3)F)C 3T-0932 Cc1c(c(n2c(n1)c(cn2)c3ccc(cc3)F)N)c4ccc(cc4)F 3T-0934 c1cc(ccc1c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)F 3T-0935 Cc1cc(n2c(n1)c(cn2)c3ccc(cc3)F)C(F)(F)F 3T-0936 COc1ccc(cc1)c2c(sc(n2)c3ccccc3)Sc4ccc(cc4)Cl 3T-0937 COc1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl 3T-0938 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)c5ccsc5)C 3T-0940 Cc1cc(n2c(n1)c(cn2)c3ccc(cc3)F)N 3T-0941 c1ccc(c(c1)C(=O)OCn2c(=O)c(c(cn2)Cl)Cl)Cl 3T-1000 c1cc(ccc1C(=O)OCn2c(=O)c(c(cn2)Cl)Cl)F 3T-1001 c1cc(cc(c1)C(F)(F)F)C(=O)OCn2c(=O)c(c(cn2)Cl)Cl 3T-1002 c1cc(ccc1C(=O)OCn2c(=O)c(c(cn2)Cl)Cl)C(F)(F)F 3T-1003 Cc1ccc(cc1)C(=O)OCn2c(=O)c(c(cn2)Cl)Cl 3T-1004 c1cc(sc1)C(=O)OCn2c(=O)c(c(cn2)Cl)Cl 3T-1005 Cc1ccc(cc1)Oc2c(c(nn2c3ccccc3)c4ccccc4)C=O 3T-1120 CC(C)(C)C1CCC(=NO)CC1 3T-1121 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Oc4cccnc4)C=O 3T-1122 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Oc4cccc(c4)Cl)C=O 3T-1123 c1ccc(cc1)c2c(c(n(n2)c3ccccc3)Oc4cc(ccc4Cl)Cl)C=O 3T-1124 COc1ccc(cc1OC)/C(=C/c2c(nn(c2Cl)c3ccccc3)c4ccccc4)/C#N 3T-1125 C=CCNC(=O)c1ccc(cc1)n2cccc2 3T-1130 Cc1ccc(cc1)C(=O)ON=C2CCC(CC2)C(C)(C)C 3T-1132 CC(C)(C)C1CCC(=NOC(=O)C2CC2)CC1 3T-1138 CC(C)(C)C1CCC(=NOC(=O)c2cccs2)CC1 3T-1139 CC(C)(C)C1CCC(=NOC(=O)c2ccc(cc2)F)CC1 3T-1140 CC(C)(C)C1CCC(=NOC(=O)c2ccc(c(c2)Cl)Cl)CC1 3T-1143 c1cc2c(cc1Br)cc(s2)C(=O)O 3T-1185 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(C(=O)OC)OC 3T-1240 CCOC(=O)CSc1c(cc2c(n1)CCCC2)C#N 3T-1241 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(C(=O)OCC#C)OCC#C 3T-1246 CN(C)C(=O)c1cc2cc(ccc2s1)Br 3T-1251 CNC(=O)c1cc2cc(ccc2s1)Br 3T-1252 c1cc2c(cc1Br)cc(s2)C(=O)N3CCOCC3 3T-1253 c1cc2c(cc1Br)cc(s2)C(=O)N3CCCC3 3T-1254 c1ccc(cc1)CNC(=O)c2cc3cc(ccc3s2)Br 3T-1255 c1ccc(cc1)NC(=O)c2cc3cc(ccc3s2)Br 3T-1256 Cc1ccc(cc1)C2N=C(C(=N2)c3ccccc3OC)C 3T-1258 CC1=NC(N=C1c2ccccc2OC)c3ccc(cc3)F 3T-1259 CC1=NC(N=C1c2ccccc2OC)c3c(cc(cc3Cl)Cl)Cl 3T-1260 Cc1c(cn(n1)C(C)(C)C)c2ccccc2OC 3T-1261 c1ccc(c(c1)C(=O)OCn2c(=O)c(c(cn2)Br)Br)Cl 3T-1482 c1cc(c(cc1C(=O)OCn2c(=O)c(c(cn2)Br)Br)Cl)Cl 3T-1483 c1cc(ccc1C(=O)OCn2c(=O)c(c(cn2)Br)Br)F 3T-1484 c1cc(c(c(c1)F)C(=O)OCn2c(=O)c(c(cn2)Br)Br)F 3T-1485 c1cc(cc(c1)C(F)(F)F)C(=O)OCn2c(=O)c(c(cn2)Br)Br 3T-1486 c1(nnc(s1)NN)C(F)(F)F 3T-1490 CC(=O)OCn1c(=O)c(c(cn1)Br)Br 3T-1493 CCN(CC)CCNC(=O)c1cc2cc(ccc2s1)Br 3T-1532 c1cc2c(cc1Br)cc(s2)C(=O)NC3CC3 3T-1533 COC(=O)c1cc(cc(c1)OCc2ccccc2)OCc3ccccc3 3W-0014 COC(=O)c1cc(cc(c1)OCC#C)OCC#C 3W-0015 COC(=O)C(Cc1cccc(c1)C(F)(F)F)(c2ccc(cc2[N+](=O)[O-])C(F)(F)F)C(=O)OC 3W-0016 Cc1c(c(cc(n1)c2cccs2)c3cccc(c3)Cl)C#N 3W-0017 Cc1ccc(cc1)c2cc(c(c(n2)C)C#N)c3cc(c(c(c3)OC)OC)OC 3W-0022 Cc1c(c(cc(n1)c2cccs2)c3ccccc3OC)C#N 3W-0025 c1c(c(cnc1Cl)Cl)C(=O)O 3W-0027 COC(=O)C(c1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C(=O)OC 3W-0036 c1ccc(cc1)c2cn3cc(ccc3n2)C#N 3W-0042 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])CC(=O)O 3W-0048 COc1cc(ccc1OCc2ccc(cc2)C#N)CC=C 3W-0054 c1cc(c(c(c1)[N+](=O)[O-])CC(=O)O)[N+](=O)[O-] 3W-0056 c1ccc(cc1)c2cn3cc(ccc3n2)C=O 3W-0059 c1ccc2c(c1)C(CCC2=O)c3ccc(c(c3)Cl)Cl 3W-0200 c1cc(ccc1OCCCN)OCCCN 3W-0201 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)CO 3W-0202 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)CO 3W-0203 Cc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)n3c(ccc3C)C 3W-0204 Cc1ccc(n1c2ccc(cc2)c3cc[nH]n3)C 3W-0208 Cc1ccc(n1c2ccc(cc2)c3ccnc(n3)N)C 3W-0209 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)CO 3W-0210 c1cc(ccc1c2ccn3c(n2)ncn3)C4CCCCC4 3W-0214 Cc1c(sc(n1)c2ccc(cc2)Cl)CN 3W-0217 c1ccc(c(c1)/C=C/2\C(=O)N=C(S2)NCCCn3ccnc3)n4cccn4 3W-0218 c1cc(cc(c1)n2cc(cn2)O)C(F)(F)F 3W-0219 CN(C)/C=C/1\CC(c2ccccc2C1=O)c3ccc(c(c3)Cl)Cl 3W-0220 c1cc2c(cc1Cl)NC(=O)C(O2)CCOC(=O)C3CCCCC3 3W-0224 Cc1cn2c(c(c(n2)CC#N)C#N)nc1c3ccc(c(c3)F)OC 3W-0226 c1cc2c(cc1Cl)NC(=O)CO2 3W-0227 Cc1c(sc(n1)c2ccc(cc2)Cl)CNS(=O)(=O)c3ccccc3 3W-0228 c1cc2cc(ccc2nc1)c3nnc(n3c4ccc5c(c4)OCCO5)S 3W-0229 COC(=O)C1=C(C(=O)N(C1)Cc2ccccn2)O 3W-0231 Cc1c(sc(n1)c2ccc(cc2)Cl)COc3ccc(cc3)OC 3W-0232 c1ccc(c(c1)/C=C/c2c3c(c4cccc(c4n2)C(F)(F)F)SCC3)[N+](=O)[O-] 3W-0233 Cc1c2c(c3cc(ccc3n1)Oc4ccccc4)N(CC2)c5ccc(cc5)Oc6ccccc6 3W-0235 COC(=O)c1cc(c(nc1)Sc2ccccc2)Cl 3W-0238 Cc1c(sc(n1)c2ccc(cc2)Cl)CNC(=O)c3cccc(c3)OC 3W-0239 Cc1c(c(=O)n(n1C(=O)C)c2ccc(c(c2)Cl)Cl)CCOC(=O)C 3W-0241 c1ccc(c(c1)/C=C/c2c3c(c4cccc(c4n2)C(F)(F)F)SCC3)Cl 3W-0242 Cc1c2c(c3cc(ccc3n1)Oc4ccccc4)N(CC2)c5ccc(cc5)OC 3W-0243 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)/C=N/O 3W-0245 c1cc2c(cc1Cl)NC(=O)C(O2)CCCl 3W-0252 COC(=O)c1c(c2ccccc2o1)n3cccc3 3W-0254 CC(=O)OCCC1C(=O)Nc2cc(ccc2O1)Cl 3W-0255 CC(=O)N(c1ccccc1/C=C/c2c3c(c4cccc(c4n2)C(F)(F)F)SCC3)C(=O)C 3W-0256 COc1cccc(c1)CONC(=O)NN 3W-0260 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)/C=C/C(=O)O 3W-0261 c1ccc(cc1)n2cc(cn2)C(=O)c3cc(ccc3O)F 3W-0262 Cc1ccc2c(c1)NC(=O)CO2 3W-0266 c1cc(ccc1C2CCCCC2)C(=O)c3cc(cc(c3)C(=O)c4ccc(cc4)C5CCCCC5)C(=O)c6ccc(cc6)C7CCCCC7 3W-0267 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)/C(=N/O)/N 3W-0269 COC(=O)c1cc(c(nc1)Cl)Cl 3W-0272 c1cc(ccc1C(CC(=O)N)NC(=O)C(F)(F)F)Cl 3W-0273 Cc1c(sc(n1)c2ccc(cc2)Cl)CNC(=O)c3ccc(cc3)Cl 3W-0274 c1cc2c(c(c1)C(F)(F)F)nc(c3c2SCC3)/C=C/c4ccc(cc4)[N+](=O)[O-] 3W-0276 COC(=O)c1c(c2ccccc2o1)N(C(=O)Oc3ccccc3)C(=O)Oc4ccccc4 3W-0279 COC(=O)c1c(c2ccccc2o1)N3Cc4ccccc4C3 3W-0280 COC(=O)c1c(ccs1)Oc2ccc(cc2N)F 3W-0282 CSc1ncc(c(n1)C(=O)O)Br 3W-0283 c1cc2c(cc1/C=C/3\C(=O)N=C(S3)NCC(=O)O)OCO2 3W-0294 Cc1c(c(=O)n2c([nH]1)c(cn2)C#N)CCOC(=O)C 3W-0298 COC(=O)c1ccc(cc1)n2c(c3c(n2)CCCC3)c4ccccc4F 3W-0300 c1ccc2c(c1)c(c(o2)C(=O)O)n3cccc3 3W-0301 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)CN 3W-0305 Cc1ccc(cc1)C(=O)OCCc2c([nH]n(c2=O)c3ccccc3)C 3W-0308 c1ccc(c(c1)c2c3c(nn2c4ccc(cc4)C(=O)NC5CCCC5)CCCC3)F 3W-0312 c1ccc(c(c1)c2c3c(nn2c4ccc(cc4)C(=O)NCc5ccc(cc5)F)CCCC3)F 3W-0313 c1ccc(c(c1)c2c3c(nn2c4ccc(cc4)C(=O)NCC5CCCO5)CCCC3)F 3W-0314 c1ccc(c(c1)c2c3c(nn2c4ccc(cc4)C(=O)NC5CCCCCC5)CCCC3)F 3W-0316 CC1(OC(=O)C2(Cc3ccccc3C2)C(=O)O1)C 3W-0317 Cc1c(c(n2c(n1)c(cn2)C#N)Cl)CCOC(=O)C 3W-0318 COc1ccc(cc1)CNC(=O)c2ccc(cc2)n3c(c4c(n3)CCCC4)c5ccccc5F 3W-0321 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)/C=C\5/C(=O)NC(=S)S5 3W-0324 Cc1c(c(n2c(n1)c(cn2)C#N)N3CCCC3)CCOC(=O)C 3W-0325 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5ccc(cc5)Cl)CCS4 3W-0326 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5ccccc5Cl)CCS4 3W-0327 COc1ccc(cc1)CNC(=O)c2c(c3ccccc3o2)n4cccc4 3W-0328 C1CC(=CNC1)C(=O)N 3W-0332 CC(=O)c1cc(ccc1[N+](=O)[O-])Cl 3W-0333 COC(=O)c1c(ccs1)Oc2ccccc2N 3W-0336 CC(=O)c1cc2c(cc1NC(=O)c3cccc(c3)Cl)OCO2 3W-0341 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5ccc(cc5Cl)Cl)CCS4 3W-0343 C1=NNC(=O)C1CCCN 3W-0345 C1COCc2c1c(c(s2)N)C#N 3W-0346 c1ccc2c(c1)-c3c(cnc(n3)N)CC2c4ccc(c(c4)Cl)Cl 3W-0352 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5ccc(cc5)F)CCS4 3W-0353 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5ccccc5F)CCS4 3W-0354 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCOCC2 3W-0356 Cc1ccc(n1c2ccc(cc2)c3ccnc4n3ncc4C#N)C 3W-0400 Cc1ccc(n1c2ccc(cc2)c3ccnc4n3ncn4)C 3W-0401 Cc1ccc(n1c2ccc(cc2)c3ccnc4n3nc(c4)C)C 3W-0403 Cc1ccc(n1c2ccc(cc2)c3ccnc(n3)c4ccncc4)C 3W-0409 Cc1ccc(n1c2ccc(cc2)c3ccnc(n3)c4ccccn4)C 3W-0410 COc1ccc(cc1)NC(=O)CCl 3W-0415 c1ccc(c(c1)CN2C(=O)c3ccccc3C2=O)CN4C(=O)c5ccccc5C4=O 3W-0417 Cc1ccc(n1c2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3)Br)C 3W-0424 Cc1ccc(n1c2ccc(cc2)c3ccn(n3)CCO)C 3W-0425 Cc1ccc(n1c2ccc(cc2)c3ccnc(n3)C)C 3W-0427 CCOC(=O)c1cnn(c1N)C(=O)c2ccc3c(c2)cccn3 3W-0430 Cc1ccc(cc1)C2c3c([nH]nc3NC4=C2C(=O)CC(C4)(C)C)C 3W-0438 Cc1ccc(n1c2ccc(cc2)c3ccnc4n3nc(c4c5cccc(c5)C(F)(F)F)C)C 3W-0439 Cc1c2c(n[nH]1)NC3=C(C2c4ccc(cc4)Cl)C(=O)CC(C3)(C)C 3W-0443 Cc1c2c(n[nH]1)NC3=C(C2c4ccccc4)C(=O)CC(C3)(C)C 3W-0444 Cc1c2c(n[nH]1)NC3=C(C2c4ccc(cc4)F)C(=O)CC(C3)(C)C 3W-0445 Cc1c2c(n[nH]1)NC3=C(C2c4ccc(cc4)OC)C(=O)CC(C3)(C)C 3W-0447 Cc1c2c(n[nH]1)NC3=C(C2c4ccc5c(c4)OCO5)C(=O)CC(C3)(C)C 3W-0448 Cc1c2c(n[nH]1)NC3=C(C2c4ccncc4)C(=O)CC(C3)(C)C 3W-0449 Cc1c2c(n[nH]1)NC3=C(C2c4ccc(cc4)[N+](=O)[O-])C(=O)CC(C3)(C)C 3W-0451 Cc1c2c(n[nH]1)NC3=C(C2c4cccs4)C(=O)CC(C3)(C)C 3W-0453 Cc1c2c(n[nH]1)NC3=C(C2c4ccc(cc4)O)C(=O)CC(C3)(C)C 3W-0454 CN1CC(C2(C13c4ccccc4NC3=O)COc5ccccc5C2=O)c6cccc(c6)[N+](=O)[O-] 3W-0605 c1ccc(cc1)/C=N/NS(=O)(=O)c2ccccc2 3W-0610 c1ccc(cc1)S(=O)(=O)N/N=C/c2cccc(c2)Cl 3W-0611 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)F 3W-0612 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)Cl 3W-0613 Cc1ccc(cc1)/C=N/NS(=O)(=O)c2ccccc2 3W-0615 c1ccc(cc1)S(=O)(=O)N/N=C/c2cccc(c2)[N+](=O)[O-] 3W-0625 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)C#N 3W-0626 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2Cl)Cl 3W-0627 c1ccc(cc1)NC(=O)N/C(=C(/C#N)\N)/C#N 3W-0628 c1ccc(cc1)c2cc(nc(n2)N)O 3W-0631 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccccc2Cl 3W-0632 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccccc2[N+](=O)[O-] 3W-0633 COc1ccccc1/C=N/NS(=O)(=O)c2ccccc2 3W-0634 COc1cccc(c1)/C=N/NS(=O)(=O)c2ccccc2 3W-0635 c1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)[N+](=O)[O-] 3W-0637 c1ccc(cc1)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccccc4 3W-0650 c1cc(ccc1NC(=O)N/C(=C(/C#N)\N)/C#N)Cl 3W-0654 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4ccc(cc4)Cl)[nH]c2=O 3W-0656 COc1ccc(cc1OC)c2ccc3ccccc3n2 3W-0800 CC1=NN(C(=O)c2ccccc2O1)S(=O)(=O)c3ccc(cc3)F 3W-0802 Cc1ccc(cc1)S(=O)(=O)N2C(=O)c3ccccc3OC(=N2)C 3W-0803 CC1=NN(C(=O)c2ccccc2O1)S(=O)(=O)c3ccc(cc3Cl)Cl 3W-0804 c1cc(c(nc1)n2c(cc(n2)C(F)(F)F)C(F)(F)F)NO 3W-0805 c1ccc2c(c1)cc3c(n2)-c4ccccc4C3 3W-0807 c1ccc-2c(c1)Cc3c2nc4c(c3)cc(cc4Br)Br 3W-0808 CN1C(=O)/C(=C/c2ccc3c(c2)OCO3)/SC1=O 3W-0809 CCOC(=O)C(=CNc1c2ccccc2[nH]n1)C(=O)OCC 3W-0811 CN1C(=O)/C(=C/c2ccc(cc2)C#N)/SC1=O 3W-0812 CC(=O)c1c(cc(cn1)C(F)(F)F)S(=O)(=O)c2ccccc2 3W-0814 CC(=O)c1c(cc(cn1)C(F)(F)F)S(=O)(=O)C 3W-0815 CCNC(=O)O/N=C(\C)/c1c(cc(cn1)C(F)(F)F)N2CCCC2 3W-0816 CCOC(=O)C(=CNc1ncccn1)C(=O)OCC 3W-0817 CCOC(=O)c1cnc2c3ccccc3[nH]n2c1=O 3W-0818 CCOC(=O)C(=CNc1ccc(cn1)I)C(=O)OCC 3W-0819 CN1C(=O)/C(=C\c2cccnc2)/SC1=O 3W-0820 CN1C(=O)C(SC1=O)Cc2ccc3c(c2)OCO3 3W-0821 Cc1ccc(cc1)COc2coc(cc2=O)CO 3W-0822 c1cc(ccc1N2CCN(CC2)CC#Cc3cncnc3)F 3W-0824 CC(=O)C(Cc1ccc(nc1)Cl)(Cc2ccc(nc2)Cl)C(=O)C 3W-0826 CC(=O)C(Cc1ccc(nc1)Cl)Cc2ccc(nc2)Cl 3W-0827 CN1C(=O)/C(=C\NCc2ccc(cc2)OC)/SC1=O 3W-0828 c1cnccc1CC2C(=O)NC(=O)S2 3W-0829 c1cc(c2ccc3cccn3c2c1)N 3W-0830 CCOc1ccc(cc1OC)C(CC(=O)O)N 3W-0831 CSc1nncn1c2ccccc2 3W-0832 CN1C(=O)/C(=C/NC2CCCCC2)/SC1=O 3W-0833 c1ccc-2c(c1)CCc3c2nc4c(c3)cc(cc4Br)Br 3W-0835 COc1cccc-2c1CCc3c2nc4c(c3)cc(cc4Br)Br 3W-0836 Cc1cc2c(cc(=O)[nH]c2cc1N)COC 3W-0839 CS(=O)(=O)NC1CC(=O)c2c1ccs2 3W-0840 c1cc(cc(c1)C(F)(F)F)C(=O)NC2CC(=O)c3c2ccs3 3W-0841 c1cc(sc1)S(=O)(=O)NC2CC(=O)c3c2ccs3 3W-0842 COc1ccc(cc1)S(=O)(=O)NC2CC(=O)c3c2ccs3 3W-0843 COC(=O)c1c(c2ccccc2nc1C(=O)OC)c3cn(nn3)c4ccc(cc4)C(F)(F)F 3W-0845 c1cc(ccc1C(F)(F)F)n2cc(nn2)C(=O)c3c(cc(cn3)C(F)(F)F)Cl 3W-0846 CCOc1ccc(cc1OC)C(CC(=O)O)N2Cc3ccccc3C2=O 3W-0848 CCOc1cc2c(cc1OC)C(CC2=O)NC(=O)C(F)(F)F 3W-0849 c1cc(oc1)C(=O)NC2CC(=O)c3c2ccs3 3W-0850 c1csc2c1C(CC2=O)NC(=O)C3CCCCC3 3W-0851 c1cc(c(cc1Cl)Cl)C(=O)NC2CC(=O)c3c2ccs3 3W-0852 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NC2CC(=O)c3c2ccs3 3W-0853 Cc1ccc(cc1)C(=O)OCc2coc(cc2=O)OC(=O)c3ccc(cc3)C 3W-0854 c1cc(ccc1N2CCN(CC2)CC#CC#CCN3CCN(CC3)c4ccc(cc4)F)F 3W-0855 c1ccc2c(c1)ccc(n2)c3cccc(c3)C(F)(F)F 3W-0856 c1cc(cc(c1)C(F)(F)F)c2ccc3cc(cc(c3n2)Br)Br 3W-0857 Cc1cc2ccccc2nc1c3ccc(cc3)F 3W-0858 Cc1cc2cc(cc(c2nc1c3ccc(cc3)F)Br)Br 3W-0859 CCCC(C)C(CC(=O)O)N 3W-0865 c1csc2c1C(CC2O)NC(=O)C(F)(F)F 3W-0866 CC(=O)CN1C(=O)c2ccccc2C1=O 3W-0868 CC1(CN(C1=O)c2cccc(c2)C(=O)c3cn(nn3)c4ccc(cc4)C(F)(F)F)C 3W-0870 c1csc2c1C(C(C2=O)Br)NC(=O)C(F)(F)F 3W-0871 CN(C)/C=C\1/C(c2ccsc2C1=O)NC(=O)C(F)(F)F 3W-0872 CN(C)/C=C/C(=O)c1cnccn1 3W-0873 Cc1cc(nc(c1C#N)N2CCOCC2)C 3W-0874 c1cc(sc1c2ccn[nH]2)Br 3W-0876 c1cc(sc1c2ccn[nH]2)Cl 3W-0877 Cc1cc([nH]n1)c2cccs2 3W-0878 Cc1c(c(=O)[nH]c(c1Br)C)C#N 3W-0879 CCOc1cc2c(cc1OC)C(CC2=O)N.Cl 3W-0880 Cc1cc2c(cc(=O)[nH]c2cc1NC(=O)C(F)(F)F)COC 3W-0881 COc1cc(cc(c1)OC)N/C=C\2/C(c3ccsc3C2=O)NC(=O)C(F)(F)F 3W-0882 CCOC(=O)C1CCN(CC1)c2c(c(cc(n2)C)C)C#N 3W-0883 Cc1c(c[nH]n1)c2ccc(cc2)Cl 3W-0884 CC1=CC(=O)Nc2cccc3c2n1nc3 3W-0885 c1cc(cc(c1)Cl)n2ccc(n2)c3cnccn3 3W-0886 c1cc(cc(c1)C(F)(F)F)COc2coc(cc2=O)CO 3W-0887 c1cc(cc(c1)F)COc2coc(cc2=O)CO 3W-0888 CCOc1cc2c(cc1OC)C(CC2=O)NC(=O)c3ccco3 3W-0889 CCOc1cc2c(cc1OC)C(CC2=O)NS(=O)(=O)c3ccc(cc3)C(C)(C)C 3W-0890 c1cc(c2ccc3cccn3c2c1)NC(=O)c4ccco4 3W-0891 COc1cccc(c1)C(=O)Nc2cccc3c2ccc4n3ccc4 3W-0892 c1cc(c2ccc3cccn3c2c1)NS(=O)(=O)c4cccs4 3W-0893 COc1ccc(cc1)S(=O)(=O)Nc2cccc3c2ccc4n3ccc4 3W-0894 c1cc(c(cc1Cl)F)C#CCO 3W-0897 Cc1c(c(nc(c1Br)C)Cl)C#N 3W-0900 c1cc(ccc1NC(=O)OCc2cc(=O)c(co2)O)Cl 3W-0901 CN(C)/C=N/c1ncc(s1)C(=O)c2c(ccs2)Br 3X-0200 CN(C)/C=N/c1ncc(s1)C(=O)c2ccc(cc2)S(=O)(=O)C 3X-0201 Cc1cc(cc(c1O)C)C(=O)c2cnc(s2)/N=C/N(C)C 3X-0202 C1CCc2c(c(=O)[nH]c(n2)NC(=S)N)C1 3X-0206 CN(C)/C=N/c1ncc(s1)C(=O)c2ccc3ccccc3c2 3X-0208 CN(C)/C=N/c1[n+](cc(s1)C(=O)c2ccc(cc2)OC)CC(=O)c3ccc(cc3)OC.[Br-] 3X-0209 c1ccc2c(c1)cccc2C3C4=C(c5ccccc5C4=O)NC(=S)N3 3X-0210 CC(C)(C)C(=O)N1CCC(CC1)(CS(=O)(=O)Cc2ccc(cc2)Cl)O 3X-0212 c1ccc(cc1)OC(=O)Nc2ccc3c(c2)OCCO3 3X-0213 c1c(nc(s1)c2nc(cs2)CCN)CCN 3X-0214 Cc1cc(c(cc1Cl)F)C(=O)c2cnc(s2)/N=C/N(C)C 3X-0215 Cc1c(sc2n1ncn2)C(=O)c3cnc(s3)/N=C/N(C)C 3X-0216 c1cc2cc(ccc2nc1)C(=O)NNC(=S)Nc3ccc4c(c3)OCCO4 3X-0217 CC(C)(C)C(=O)N1CCC(CC1)(CS(=O)(=O)Cc2ccccc2Cl)O 3X-0218 CC(C)CC(=O)N1CCC(CC1)(CS(=O)(=O)Cc2ccccc2Cl)O 3X-0219 c1cc2c(cc1NC(=O)N3CCOCC3)OCCO2 3X-0220 Cc1c(c(c2c(n1)-c3ccccc3C2=O)c4cccc5c4cccc5)C#N 3X-0226 c1cc(cc(c1)C(F)(F)F)COc2ccc(cc2)/C=C\3/C(=O)C4CCN3CC4 3X-0227 COC(=O)/C=C/c1ccc(cc1)C(=O)C2CC2 3X-0230 CC(C)CC(=O)N1CCC(CC1)(CS(=O)(=O)Cc2ccccc2)O 3X-0231 CC(C)(C)C(=O)N1CCC(CC1)(CS(=O)(=O)Cc2ccccc2)O 3X-0232 COc1ccc(cc1OC)NC(=O)Oc2ccccc2 3X-0233 c1cc2c(cc1/C=C/3\C(=O)NC(=N3)N4CCCCC4)OCO2 3X-0234 CCOC(=O)c1cnc(s1)/N=C/N(C)C 3X-0235 CN(C)/C=N/c1ncc(s1)C(=O)c2ccc(cc2Cl)Cl 3X-0236 c1cc(c(c(c1)Cl)CN2c3cc(ccc3N4CCCC4C2=O)C#N)F 3X-0240 c1cc(ccc1CN2c3cc(ccc3N4CCCC4C2=O)C#N)F 3X-0241 CN(C)/C=N/c1ncc(s1)C(=O)c2ccccc2 3X-0242 CCOC(=O)C1CSC2([NH2+]1)CCCCC2.[Cl-] 3X-0243 CC(C)CC(=O)N1CCC(CC1)(CS(=O)(=O)c2ccc(cc2)OC)O 3X-0244 CC(C)(C)C(=O)N1CCC(CC1)(CS(=O)(=O)c2ccc(cc2)OC)O 3X-0245 c1cc(cc(c1)C(F)(F)F)COc2ccc(cc2)c3cc(n[nH]3)C4CCNCC4 3X-0246 COc1ccc(cc1OC)NC(=O)N2CCOCC2 3X-0250 c1cc2c(cc1N3C(=O)C4CCCN4C3=O)OCCO2 3X-0252 c1cc2c(cc1/C=C/3\C(=O)NC(=N3)N4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl)OCO2 3X-0253 c1ccc(c(c1)CN2c3cc(ccc3N4CCCC4C2=O)C#N)F 3X-0254 CN(C)/C=N/c1ncc(s1)C(=O)c2cc([nH]c2)C=O 3X-0255 CCOC(=O)C(=O)c1cnc(s1)/N=C/N(C)C 3X-0256 Cc1cccc(c1)CN2c3cc(ccc3N4CCCC4C2=O)C#N 3X-0257 CC1CN(CC(O1)C)C(=O)Nc2ccc(c(c2)OC)OC 3X-0258 CC1CN(CC(O1)C)C(=O)Nc2ccc3c(c2)OCCO3 3X-0261 CN(C)/C=N/c1ncc(s1)C(=O)C(F)(F)F 3X-0265 c1cc2c(cc1/C=C/3\C(=O)N(C(=S)N3)CN4CCOCC4)OCO2 3X-0266 COc1ccc(cc1OC)NC(=O)N2CCN(CC2)c3ccccc3 3X-0271 CC1CCCCN1C(=O)Nc2ccc(c(c2)OC)OC 3X-0272 Cc1cccc(c1N2CCN(CC2)C(=O)Nc3ccc(c(c3)OC)OC)C 3X-0273 COc1ccc(cc1)c2ccc(cc2)C(=O)C3CC3 3X-0274 CC1CN(CC(O1)C)CN2C(=O)/C(=C\c3ccc4c(c3)OCO4)/NC2=S 3X-0275 CC(C)CC(=O)N1CCC(CC1)(CS(=O)(=O)c2ccc(c(c2)Cl)Cl)O 3X-0276 CC(C)(C)C(=O)N1CCC(CC1)(CS(=O)(=O)c2ccc(c(c2)Cl)Cl)O 3X-0277 c1cc2c(cc1/C=C/3\C(=O)N(C(=S)N3)CN4CCCCC4)OCO2 3X-0279 CN1CCN(CC1)C(=O)Nc2ccc3c(c2)OCCO3 3X-0280 Cc1cccc(c1N2CCN(CC2)CN3C(=O)/C(=C\c4ccc5c(c4)OCO5)/NC3=S)C 3X-0281 CN(C)/C=N/c1ncc(s1)C(=O)c2ccc(cc2)Cl 3X-0284 CN1CCN(CC1)CN2C(=O)/C(=C\c3ccc4c(c3)OCO4)/N=C2SC 3X-0286 COc1ccc(cc1)N2CCN(CC2)CN3C(=O)/C(=C\c4ccc5c(c4)OCO5)/NC3=S 3X-0288 CC(C)(C)OC(=O)N1CCN(CC1)CN2C(=O)/C(=C\c3ccc4c(c3)OCO4)/NC2=S 3X-0290 c1cc(cc(c1)N2CCN(CC2)CN3C(=O)/C(=C\c4ccc5c(c4)OCO5)/NC3=S)C(F)(F)F 3X-0293 c1cc2c(=O)[nH]cnc2nc1 3X-0294 c1ccc(cc1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCCO4 3X-0295 CC1CCCCN1C(=O)Nc2ccc3c(c2)OCCO3 3X-0296 Cc1cccc(c1N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCCO4)C 3X-0297 Cc1cccc(c1N2CCN(CC2)CN3C(=O)/C(=C\c4ccc5c(c4)OCO5)/N=C3SCC(=O)OC)C 3X-0300 Cc1cccc(c1N2CCN(CC2)CN3C(=O)/C(=C\c4ccc5c(c4)OCO5)/N=C3SCCC(=C(F)F)F)C 3X-0301 c1ccc(cc1)CN2CCN(CC2)C(=O)Nc3ccc4c(c3)OCCO4 3X-0302 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)Nc2ccc3c(c2)OCCO3 3X-0303 CCOC(=O)C1CSC2(N1)CCC(CC2)c3ccccc3.Cl 3X-0305 c1cc(ccc1N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCCO4)F 3X-0308 c1cc2c(cc1NC(=O)N3CCN(CC3)c4ccncc4)OCCO2 3X-0309 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccc5c(c4)OCCO5 3X-0310 COc1ccc(cc1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCCO4 3X-0311 CSC1=N/C(=C/c2ccc3c(c2)OCO3)/C(=O)N1CN4CCN(CC4)c5ccccc5 3X-0314 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)c3nc(on3)c4cccc(c4)C(F)(F)F 3X-0316 Cc1ccc(c(c1)CN2c3cc(ccc3N4CCCC4C2=O)C#N)C 3X-0320 Cc1cc(c(c(c1)C)CN2c3cc(ccc3N4CCCC4C2=O)C#N)C 3X-0321 c1ccc2c(c1)C(=O)/C(=C/c3ccc4c(c3)OCO4)/CO2 3X-0322 Cn1c2c(cc(s2)C(=O)N/N=C/c3ccc4c(c3)OCO4)c(n1)C(F)(F)F 3X-0324 CCNC(=S)NNC(=O)c1cc2c(nn(c2s1)C)C(F)(F)F 3X-0325 CCCCc1ccc(cc1)NC(=S)NNC(=O)c2cc3c(nn(c3s2)C)C(F)(F)F 3X-0326 CSC1=N/C(=C/c2ccc3c(c2)OCO3)/C(=O)N1CN4CCOCC4 3X-0328 Cc1cccc(c1N2CCN(CC2)CN3C(=O)/C(=C\c4ccc5c(c4)OCO5)/N=C3SCCC(C)CCC=C(C)C)C 3X-0329 c1cc2c(cc1CN3CCN(CC3)CN4C(=O)/C(=C\c5ccc6c(c5)OCO6)/NC4=S)OCO2 3X-0330 Cn1c2c(cc(s2)C(=O)N/N=C/c3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl)c(n1)C(F)(F)F 3X-0331 c1ccc2c(c1)c(=O)c(co2)/C=C\3/C(=O)NC(=S)N3 3X-0332 c1cc(ccc1N2CCN(CC2)CN3C(=O)/C(=C\c4ccc5c(c4)OCO5)/NC3=S)[N+](=O)[O-] 3X-0333 CCCCc1ccc(cc1)n2c(nnc2S)c3cc4c(nn(c4s3)C)C(F)(F)F 3X-0334 c1ccc(c(c1)COc2ccc(cc2)C=O)Cl 3X-0335 C#CCOc1ccc(cc1)C=O 3X-0336 CCCN(CC1CC1)C(=O)Nc2ccc3c(c2)OCCO3 3X-0339 C#CCOc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O 3X-0341 CCCN(CC1CC1)CN2C(=O)/C(=C/c3coc4ccccc4c3=O)/NC2=S 3X-0343 c1c(nc(s1)Nc2[nH]c(=O)c3c(n2)CCCC3)C(F)(F)F 3X-0346 c1ccc2c(c1)c(=O)c(co2)/C=C\3/C(=O)N(C(=S)N3)CN4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 3X-0348 CN(CC1OCCO1)CN2C(=O)/C(=C/c3coc4ccccc4c3=O)/NC2=S 3X-0350 CN(C)/C=N/c1ncc(s1)C(=O)c2ccc(o2)c3ccc(cc3Cl)Cl 3X-0352 CC(=CNC(=O)Nc1ccc2c(c1)OCCO2)C 3X-0356 COc1ccc(cc1OC)NC(=O)NN 3X-0357 c1ccc2c(c1)-c3c(cn4c(n3)c(cn4)C#N)CO2 3X-0362 CN(C)/C=C/C(=O)c1cccc(c1)C(F)(F)F 3X-0365 CCOC(=O)CC(=O)c1cnc(s1)/N=C/N(C)C 3X-0366 CCn1c(nnc1S)c2cc3c(nn(c3s2)C)C(F)(F)F 3X-0369 c1ccc2c(c1)c(=O)c(co2)/C=C\3/C(=O)N(C(=S)N3)CN4CCCCC4 3X-0370 c1ccc2c(c1)c(=O)c(co2)/C=C\3/C(=O)N(C(=S)N3)CN4CCSCC4 3X-0372 CC(C)(C)OC(=O)c1cnc(s1)/N=C/N(C)C 3X-0379 c1cc(cc(c1)C(F)(F)F)c2cc[nH]n2 3X-0381 c1c(oc(c(c1=O)O)CN2CCOCC2)CO 3X-0382 c1c(oc(c(c1=O)O)CN2CCSCC2)CO 3X-0383 c1ccc(cc1)CN(CCC#N)Cc2c(c(=O)cc(o2)CO)O 3X-0384 c1ccc(c(c1)COc2ccc(cc2)/C=C\3/C(=O)C4CCN3CC4)Cl 3X-0385 Cc1cc(c(c(c1)C)COc2ccc(cc2)C=O)C 3X-0387 c1c(cnc(c1CO)Cl)Cl 3X-0704 COC(=O)c1ccccc1Oc2ccc(cc2)[N+](=O)[O-] 3X-0705 c1cc(c(cc1C=O)[N+](=O)[O-])N2CCOCC2 3X-0707 COC(=O)c1ccccc1Oc2ccc(cc2[N+](=O)[O-])C=O 3X-0709 CCOC(=O)C1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C=O 3X-0710 COC(=O)c1ccccc1Oc2ccc(cc2)N 3X-0711 CCOC(=O)C(C)Oc1ccc(cc1)OCc2ccccc2 3X-0713 c1ccc(c(c1)C(=O)O)Oc2ccc(cc2)[N+](=O)[O-] 3X-0714 Cn1c2c(cc(s2)C=O)c(n1)C(F)(F)F 3X-0715 c1cc(ccc1c2ccc(cc2)[N+](=O)[O-])C(=O)O 3X-0716 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C=O)Cl 3X-0717 c1cc(c(nc1)Sc2ccc(cc2)Cl)C#N 3X-0718 Cn1c2c(cc(s2)C(=O)NN)c(n1)C(F)(F)F 3X-0720 c1cc(c(nc1)Sc2ccc(cc2)Cl)/C(=N/O)/N 3X-0721 CC(C)(C)OC(=O)N1CCCC(C1)CO 3X-0724 c1cc(c(nc1)N2CCOCC2)C#N 3X-0726 CC(C)(C)OC(=O)N1CCCCC1CO 3X-0727 c1cc(cc(c1)[N+](=O)[O-])C(=O)CO 3X-0728 COC(=O)c1ccc(cc1)c2c(cc(cn2)C(F)(F)F)Cl 3X-0730 c1cc(c(cc1N)Cl)Oc2c(cc(cn2)C(F)(F)F)Cl 3X-0731 CCOC(=O)C(c1ccccc1)N2CCCCC2 3X-0732 COC(=O)c1ccc(cc1)c2c(cccn2)C#N 3X-0733 c1cc(c(cc1/C=N/O)[N+](=O)[O-])N2CCOCC2 3X-0737 c1ccc(cc1)Sc2c(cccn2)C#N 3X-0738 CCOC(=O)c1ccc[nH]1 3X-0740 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2ccccc2)(C#N)C#N)c3ccc(cc3)F 3X-0800 Cc1ccc(cc1)C2C(=C(C(C(C2(C#N)C#N)c3ccccc3)C(=O)OC)O)C(=O)OC 3X-0801 Cc1ccc(cc1)C2C(=C(C(C(C2(C#N)C#N)c3ccccc3F)C(=O)OC)O)C(=O)OC 3X-0802 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2cccc3c2cccc3)C(=O)OC 3X-0803 COc1ccc(cc1Cl)C2C(=C(OC(=C2C(=O)OC)CC(=O)OC)N)C#N 3X-0805 Cc1ccc(cc1)C2C(=C(C(C(C2(C#N)C#N)c3ccc(cc3)C#N)C(=O)OC)O)C(=O)OC 3X-0806 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2cccc(c2)C(F)(F)F)C(=O)OC 3X-0808 CCOc1ccc(cc1)C2C(=C(OC(=C2C(=O)OC)CC(=O)OC)N)C#N 3X-0809 COC(=O)c1ccc(cc1)OCc2ccc(nc2)Cl 3X-0810 c1ccnc(c1)N2CCN(CC2)Cc3cnc(s3)Cl 3X-0812 c1ccc2c(c1)OCC(O2)C(=O)Nc3nnc(s3)C(F)(F)F 3X-0813 Cc1ccc(cc1)C2C(=C(C(C(C2(C#N)C#N)c3cccc(c3)C(F)(F)F)C(=O)OC)O)C(=O)OC 3X-0815 CCOc1ccc(cc1)C2C(C(=C(C(C2(C#N)C#N)c3ccc(cc3)C)C(=O)OC)O)C(=O)OC 3X-0816 Cc1ccc(cc1)C2C(C(=C(C(C2(C#N)C#N)c3cccc4c3cccc4)C(=O)OC)O)C(=O)OC 3X-0817 c1ccc2c(c1)OCC(O2)C(=O)NCCc3ccccn3 3X-0818 c1ccc2c(c1)OCC(O2)C(=O)Nc3nccc(n3)c4cccs4 3X-0819 COc1ccc(cc1Cl)c2c(c(n(c(=O)c2C#N)N)N)C#N 3X-0821 C=CCN1CCN(CC1)Cc2cnc(s2)Cl 3X-0823 c1cc(ncc1CC#N)Cl 3X-0825 c1c(sc(n1)Cl)CC#N 3X-0826 CC(CCc1ccccc1)NCc2cnc(s2)Cl 3X-0827 COc1ccc(cc1Cl)CNC=O 3X-0833 CN(C)/C=N/c1nccc(n1)c2cccs2 3X-0837 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2cccc3c2cccc3)(C#N)C#N)c4cccc5c4cccc5 3X-0838 COC(=O)c1c(c2ccccc2[nH]1)CN 3X-0839 Cc1cccc(c1N2CCN(CC2)Cc3c(cccc3N)C(=O)OC)C 3X-0842 Cc1ccc(cc1)C2C(C(=C(C(C2(C#N)C#N)c3ccc(cc3)F)C(=O)OC)O)C(=O)OC 3X-0843 COC(=O)Cc1ccc(c(c1)N)O 3X-0844 Cc1cccc(c1)N2CCN(CC2C)Cc3cnc(s3)Cl 3X-0845 COC(=O)c1cccc(c1CN2CCN(CC2)c3ccccc3)N 3X-0846 Cc1ccc(cc1)C(=O)NCc2c3ccccc3[nH]c2C(=O)OC 3X-0850 c1ccc(c(c1)C2=NCCCN2)S 3X-0852 CCOC(=O)c1ccc2c(c1)sc(n2)N 3X-0853 c1cc(sc1)c2ccnc(n2)N/C=N/O 3X-0854 CC(=O)N1CCN(CC1)Cc2cnc(s2)Cl 3X-0855 Cc1cc(nc(c1C#N)OCc2ccc(nc2)Cl)C 3X-0856 COc1ccc(cc1Cl)/C=N/CC(OC)OC 3X-0857 CN(C)/C=N/C(=O)C1CCCN(C1)Cc2c(cccc2[N+](=O)[O-])C(=O)OC 3X-0859 COC(=O)c1cccc(c1CN2CCN(CC2)c3ccccc3)NC(=O)Nc4ccccc4 3X-0860 CO/N=C/Nc1nccc(n1)c2cccs2 3X-0861 CC(=O)c1ccc(c(c1)F)O 3X-0862 CC(=O)c1ccc(c(c1)F)OCc2ccccc2 3X-0863 c1cc(sc1)c2ccnc(n2)N/C=N/OCc3ccc(cc3Cl)Cl 3X-0865 Cc1ccc(cc1)CO/N=C/Nc2nccc(n2)c3cccs3 3X-0866 COc1ccc(cc1Cl)CNCC(OC)OC 3X-0867 CCCCCOc1ccc(cc1)C(=O)Nc2ccc3c(c2)ncn3C(=O)c4ccc(cc4)OCCCCC 3X-0868 c1ccc(cc1)C2=N/C(=C/Nc3nccc(n3)c4cccs4)/C(=O)O2 3X-0869 CC(C)c1cccc(c1NC(=O)Nc2cccc(c2CN3CCC(CC3)Cc4ccccc4)C(=O)OC)C(C)C 3X-0870 c1ccc(cc1)N2CCN(CC2)/C=N/c3nccc(n3)c4cccs4 3X-0872 CCOc1ccccc1NC(=O)Nc2cccc(c2CN3CCC(CC3)Cc4ccccc4)C(=O)OC 3X-0877 Cc1ccc(cc1)CNC(=O)c2cnc(nc2C(F)(F)F)c3ccccn3 3X-0878 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2ccc(cc2)F)(C#N)C#N)c3ccc(cc3)C#N 3X-0880 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2ccc(cc2)C#N)C(=O)OC 3X-0881 CN(Cc1ccccc1)c2c(c(nc(n2)N)Cl)C=O 3X-0882 Cc1cc(c(c(=O)n1Cc2ccc(nc2)Cl)C#N)C(F)(F)F 3X-0883 Cc1c(c(n2c(n1)c(cn2)c3ccsc3)C)C/C=C/c4ccccc4 3X-0889 c1ccc(cc1)CNC(=O)c2cnc(nc2C(F)(F)F)c3ccccn3 3X-0893 c1ccnc(c1)c2ncc(c(n2)C(F)(F)F)C(=O)NCc3ccc(cc3)F 3X-0894 c1ccc2c(c1)NC(=O)c3cccc(c3CO2)[N+](=O)[O-] 3X-0895 c1ccc2c(c1)OCC(O2)C(=O)Nc3ccc(cc3)I 3X-0896 CN1C(=O)C(=Cc2cc(c[nH]2)C(=O)CCl)C(=O)N(C1=O)C 3X-0902 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2ccc(cc2)C#N)(C#N)C#N)c3ccccc3F 3X-0903 CCOc1ccc(cc1)C2C(C(=C(C(C2(C#N)C#N)c3ccc(cc3)C#N)C(=O)OC)O)C(=O)OC 3X-0904 CN(Cc1ccccc1)c2c3cc(sc3nc(n2)N)C(=O)OC 3X-0906 COC(=O)c1ccccc1Oc2ccc(cc2)NC(=O)Nc3ccc(cc3)Cl 3X-0907 C1CCN(CC1)c2c(c(nc(n2)N)Cl)C=O 3X-0908 C1CCN(CC1)c2c(c(nc(n2)N)N3CCCCC3)C=O 3X-0910 CC(C)(CCl)C(=O)Nc1ccc(cc1)Oc2ccccc2C(=O)OC 3X-0911 c1ccc(cc1)CN2CCN(CC2)C(=O)CN3CCOCC3 3X-0912 COC(=O)c1ccccc1Oc2ccc(cc2)NC(=O)c3ccccc3 3X-0913 CN(Cc1ccccc1)c2c(c(nc(n2)N)N(C)Cc3ccccc3)C=O 3X-0916 CN1CCN(CC1)c2c(c(nc(n2)N)N3CCN(CC3)C)C=O 3X-0917 Cc1ccc(n1c2ccc(cc2)Oc3ccccc3C(=O)OC)C 3X-0918 Cc1ccc(cc1)C(=O)C2CN(CC2c3ccc(c(c3)Cl)OC)C 3X-0919 CC1(C(=O)CN1c2ccc(cc2)Oc3ccccc3C(=O)OC)C 3X-0920 CC(=O)Nc1ccc(cc1)OC(=O)C2COc3ccccc3O2 3X-0921 CCOc1ccc(cc1)C(CCO)NC(=S)Nc2ccc(cc2C)Cl 3X-0922 c1cnccc1NCC2CC2 3X-5001 COc1cc(c(c(c1C=O)OC)OC)OC 3X-5002 c1cc(cc(c1)Cl)C(=NC#N)N 3X-5053 CC1(OC(=O)C(C(=O)O1)C(=O)CCl)C 3X-5070 CC1(OC(=O)C(C(=O)O1)c2csc(n2)N)C 3X-5080 c1ccc(c(c1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)[N+](=O)[O-] 3Y-0026 c1ccc(c(c1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)C(F)(F)F 3Y-0028 COc1cc2c(cc1OC)NC3=C(C2c4ccccc4[N+](=O)[O-])C(=O)OC3 3Y-0037 COc1cc2c(cc1OC)NC3=C(C2c4ccccc4C(F)(F)F)C(=O)OC3 3Y-0038 COc1cc2c(cc1OC)NC3=C(C2c4ccc(cc4Cl)Cl)C(=O)OC3 3Y-0052 COc1cc2c(cc1OC)NC3=C(C2c4cc(ccc4F)C(F)(F)F)C(=O)OC3 3Y-0053 Cc1c([nH]c(c1C(=O)O)C)C=O 3Y-0054 CCOC(=O)c1c(c2c(s1)cccc2I)N 3Y-0085 COc1cc2c(cc1OC)NC3=C(C2c4cccc(c4)Br)C(=O)OC3 3Y-0088 c1cc(cc(c1)Br)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 3Y-0090 c1ccc2c(c1)c(c[nH]2)C3=CCC4(CC3)OCCO4 3Y-0246 C1CC2(CCC13NC(CS3)C(=O)O)OCCO2 3Y-0252 c1ccc(cc1)CN2CCC3(CC2)NC(CS3)C(=O)O 3Y-0253 CC(C)(C)OC(=O)Nc1ccc(cn1)C(=O)O 3Y-0608 CC(C)(C)OC(=O)N1CCc2c(sc(c2C(=O)OC)N)C1 3Y-0700 CC(C)(C)OC(=O)N1CCc2c(sc(c2C#N)N)C1 3Y-0701 CS(=O)(=O)N1CCC(CC1)C(=O)O 3Y-0704 c1ccc(cc1)c2ccc(cn2)CCl 3Y-0706 COc1ccc(cc1)c2ccc(cn2)CCl 3Y-0708 c1cc(ccc1c2ccc(cn2)[N+](=O)[O-])Cl 3Y-0712 c1cc(c(nc1)c2ccc(cc2)Cl)[N+](=O)[O-] 3Y-0713 c1ccc(cc1)c2cc(ccn2)C#N 3Y-0714 COc1ccc(cc1)c2cc(ccn2)C#N 3Y-0715 c1cc(ccc1C=O)c2cc(ccn2)C#N 3Y-0716 c1ccc(cc1)c2ccc(cn2)[N+](=O)[O-] 3Y-0717 COc1ccc(cc1)c2ccc(cn2)[N+](=O)[O-] 3Y-0718 COC(=O)c1ccc(cc1)c2ccc(cn2)[N+](=O)[O-] 3Y-0719 Cc1[nH]nc(n1)C(F)(F)F 3Y-0800 CCOC(=O)c1c(nn(c1C)S(=O)(=O)c2cccc(c2)[N+](=O)[O-])C 3Y-0801 CCOC(=O)c1c(nn(c1C)S(=O)(=O)c2cc(ccc2C)[N+](=O)[O-])C 3Y-0802 CCOC(=O)c1c(nn(c1C)S(=O)(=O)c2ccccc2)C 3Y-0803 c1c(cc(c(c1Cl)N)Br)C(F)(F)F 3Y-0805 c1cc(cc(c1)N2CCCC2=O)N 3Y-0809 c1cc(ccc1C#N)C(=O)CC#N 3Y-0811 Cc1c(c(nn2c1nnc2)C)Cc3c(cccc3Cl)F 3Y-0812 c1cnc2ncc(n2c1)Br 3Y-0813 COC(=O)c1ccc2ncc(n2c1)I 3Y-0815 CCOC(=O)c1c(nn(c1C)S(=O)(=O)CC)C 3Y-0816 CCOC(=O)c1c(nn(c1C)S(=O)(=O)c2ccc(cc2)C(C)(C)C)C 3Y-0817 CCS(=O)(=O)n1cc(cc1C(=O)OC)Br 3Y-0818 COC(=O)c1cc(cn1S(=O)(=O)c2ccccc2)Br 3Y-0821 C/C(=C\C(=O)c1ccc(cc1)c2ccccc2)/N(C)C 3Y-0823 C/C(=C\C(=O)c1cccc(c1)C(F)(F)F)/N(C)C 3Y-0824 c1cc2c([nH]cn2)nc1 3Y-0826 CCCc1nc2c(o1)cccn2 3Y-0827 CCCc1nc2ccc(cc2o1)N 3Y-0828 CCOC(=O)c1c(nn(c1C)c2ccccc2C(=O)O)C 3Y-0830 Cc1c(c(n(n1)c2ccccc2C(=O)O)C)C(=O)O 3Y-0835 CCOC(=O)c1c(nn(c1C)c2cccc(c2)F)C 3Y-0836 CC(=O)Nc1ccccc1OC(F)(F)F 3Y-0839 CCOc1c(ccc(n1)c2ccc3c(c2)OCO3)C#N 3Y-0841 c1ccc2c(c1)C(C(=O)N2)Cc3ccc(cc3)OC(F)(F)F 3Y-0843 c1cc(ccc1c2cc([nH]n2)N)Cl 3Y-0844 c1ccc(c(c1)/C=C(\C#N)/C(=O)c2ccc(cc2)C#N)C(F)(F)F 3Y-0845 c1cc(c2c(c1)OCO2)/C=C(\C#N)/C(=O)c3ccc(cc3)C#N 3Y-0846 Cc1cc(cc(c1O)OC)CC2c3ccccc3NC2=O 3Y-0848 COc1ccc(cc1)n2c(c(cn2)C#N)N 3Y-0920 c1cc(ccc1/C=C(\C#N)/C(=O)O)Cl 3Y-0922 c1cc(ccc1/C=C(\C#N)/C(=O)N)Br 3Y-0925 c1cc(cc(c1)n2c(c(cn2)C#N)N)C(F)(F)F 3Y-0926 CCOC(=O)c1c(n2cc(ccc2n1)Cl)[N+](=O)[O-] 3Y-0931 c1ccc2c(c1)c(cc(n2)c3cccc(c3)Cl)C(=O)O 3Y-0933 c1ccc2c(c1)c(cc(n2)c3ccccc3F)C(=O)O 3Y-0936 COc1ccc(cc1)c2cc(c3ccccc3n2)C(=O)O 3Y-0940 c1ccc2c(c1)[nH]c(n2)NN 3Y-0941 c1cc(c(cc1n2c(c(cn2)C#N)N)Cl)Cl 3Y-0942 c1cc(ccc1n2c(c(cn2)C#N)N)[N+](=O)[O-] 3Y-0943 CN(C)/C=N/c1c(cnn1c2ccc(cc2)OC)C#N 3Y-0947 Cc1ccc(cc1)n2c(c(cn2)C#N)N/C=N/O 3Y-0948 CN(C)/C=N/c1c(cnn1c2ccc(c(c2)Cl)Cl)C#N 3Y-0953 c1ccc2c(c1)c(cc(n2)c3ccccc3Cl)C(=O)O 3Y-0954 Cc1ccc(cc1)c2cc(c3ccccc3n2)C(=O)O 3Y-0955 COc1ccc(cc1)n2c(c(cn2)C#N)N/C=N\O 3Y-0959 c1cc(sc1)C(=O)C(=O)O 3Y-0962 CCS(=O)(=O)c1ccc2c(c1)nc(o2)C 3Y-5001 c1cc2c(cc1[N+](=O)[O-])c(n[nH]2)N 3Y-5005 c1cc(ccc1Oc2ccc(cn2)C#N)Cl 3Y-5009 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)C#N 3Y-5016 COc1ccc2c(c1)c(c[nH]2)C=C(C#N)C#N 3Y-5021 COc1ccc(cc1OC)CCN2Cc3c(cccc3[N+](=O)[O-])C2=O 3Y-5023 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)C(=O)N 3Y-5026 CCCOc1ccc(cc1)Oc2ccc(cn2)C#N 3Y-5030 COc1ccc2c(c1)c(c[nH]2)CCO 3Y-5037 COc1ccc(cc1OC)CCNC(=O)c2cc(ccc2O)[N+](=O)[O-] 3Y-5042 COc1ccc(cc1OC)CCN2Cc3c(cccc3N)C2=O 3Y-5044 c1cc2c(c(c1)[N+](=O)[O-])CN(C2=O)C3CCCCC3 3Y-5048 COc1ccc(cc1OC)CCn2c(=O)c3cc(ccc3oc2=O)[N+](=O)[O-] 3Y-5051 c1ccnc(c1)CCN2Cc3c(cccc3[N+](=O)[O-])C2=O 3Y-5053 Cc1c(scn1)CCOc2ccc(cn2)C#N 3Y-5070 COc1ccc(cc1OC)CCn2c(=O)c3cc(ccc3oc2=O)N 3Y-5076 COc1ccc2c(c1)cc([nH]2)/C=C(\C#N)/S(=O)(=O)C 3Y-5079 c1ccnc(c1)CCN2Cc3c(cccc3N)C2=O 3Y-5081 COc1ccc(cc1OC)CCN2Cc3c(cccc3/N=C/c4ccc(cc4O)O)C2=O 3Y-5086 c1cc2c(c(c1)N)CN(C2=O)C3CCCCC3 3Y-5087 COC(=O)c1c(ccs1)Oc2ccccc2NC(=O)c3ccccc3F 3Y-5151 COC(=O)c1c(ccs1)Oc2ccccc2NC(=O)CCc3ccccc3 3Y-5152 CC(C)CC(=O)Nc1ccccc1Oc2ccsc2C(=O)OC 3Y-5153 CC(C)(C)C(=O)Nc1ccccc1Oc2ccsc2C(=O)OC 3Y-5154 COC(=O)c1c(ccs1)Oc2ccccc2NC(=O)c3cccs3 3Y-5155 CC(=O)Nc1ccccc1Oc2ccsc2C(=O)OC 3Y-5156 COCC(=O)Nc1ccccc1Oc2ccsc2C(=O)OC 3Y-5157 COC(=O)c1c(ccs1)Oc2ccccc2NC(=O)C3CC3 3Y-5158 COC(=O)c1c(ccs1)Oc2ccccc2NC(=O)c3ccccc3 3Y-5159 COC(=O)c1c(ccs1)Oc2ccccc2NC(=O)COCc3ccccc3 3Y-5160 COC(=O)c1c(ccs1)Oc2ccccc2NS(=O)(=O)c3ccccc3 3Y-5161 COC(=O)c1c(ccs1)Oc2ccccc2NS(=O)(=O)C 3Y-5162 COC(=O)c1c(ccs1)Oc2ccccc2NS(=O)(=O)c3ccc(cc3)Cl 3Y-5167 COC(=O)c1c(ccs1)Oc2ccccc2NS(=O)(=O)CC(F)(F)F 3Y-5170 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCCOC 3Y-5171 CCN(CC)C(=O)C1CCN(CC1)c2ccc(cc2)C(=O)C 3Y-5172 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCCN(C)C 3Y-5173 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)N3CCOCC3 3Y-5174 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCC3CC3 3Y-5175 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCc3ccncc3 3Y-5176 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCCN3CCOCC3 3Y-5178 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCc3ccccc3 3Y-5179 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)N3CCCC3 3Y-5181 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)N3CCN(CC3)C 3Y-5182 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)N3CCCCC3 3Y-5183 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCc3ccc(cc3)OC 3Y-5185 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCCN3CCCC3 3Y-5186 CC(=O)c1ccc(cc1)N2CCC(CC2)C(=O)NCc3cccs3 3Y-5187 c1ccc(c(c1)C(=O)Nc2ccccc2Oc3ccsc3C(=O)O)F 3Y-5190 c1ccc(cc1)CCC(=O)Nc2ccccc2Oc3ccsc3C(=O)O 3Y-5191 CC(C)CC(=O)Nc1ccccc1Oc2ccsc2C(=O)O 3Y-5192 CC(C)(C)C(=O)Nc1ccccc1Oc2ccsc2C(=O)O 3Y-5193 c1ccc(c(c1)NC(=O)c2cccs2)Oc3ccsc3C(=O)O 3Y-5194 CC(=O)Nc1ccccc1Oc2ccsc2C(=O)O 3Y-5195 COCC(=O)Nc1ccccc1Oc2ccsc2C(=O)O 3Y-5196 c1ccc(c(c1)NC(=O)C2CC2)Oc3ccsc3C(=O)O 3Y-5197 c1ccc(cc1)C(=O)Nc2ccccc2Oc3ccsc3C(=O)O 3Y-5198 c1ccc(cc1)COCC(=O)Nc2ccccc2Oc3ccsc3C(=O)O 3Y-5199 c1ccc(cc1)S(=O)(=O)Nc2ccccc2Oc3ccsc3C(=O)O 3Y-5200 CS(=O)(=O)Nc1ccccc1Oc2ccsc2C(=O)O 3Y-5201 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)Cl)Oc3ccsc3C(=O)O 3Y-5206 c1cc(cc(c1)F)COc2ccc(cc2Br)N 3Y-7010 c1cc(cc(c1)F)Oc2ccc(cc2F)N 3Y-7016 COc1cc(c(c(c1)OC)C(c2cccnc2)C3=C(COC3=O)O)N 3Z-0206 COc1cc2c(c(c1)OC)C(C3=C(N2)COC3=O)c4cccs4 3Z-0208 COc1ccc(cc1)C2c3c(cc(cc3OC)OC)NC4=C2C(=O)OC4 3Z-0209 c1cc2c(ccc3c2OC(=C(C3c4cccnc4)C#N)N)c(c1)N 3Z-0210 c1cc(ccc1c2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl)Cl 3Z-0227 c1cc(ccc1n2ccc(=O)c(n2)c3ccnc(n3)N)Cl 3Z-0228 CN1C(=O)N(C(O1)CC(=O)O)c2ccc(cc2)OC 3Z-0242 c1c[nH]c2c1c(ncn2)Cl 3Z-0603 CC(C(=O)C)NC(=O)C 3Z-0703 c1cc(sc1C=O)c2ccsc2 3Z-0704 COC(=O)c1ccc2nc(cn2c1)c3ccccc3 3Z-0809 CCOC(=O)COc1ccc(cc1)[N+](=O)[O-] 3Z-0931 c1cc2c(cc1[N+](=O)[O-])NCCO2 3Z-5010 c1ccc(c(c1)CN(Cc2ccccc2Cl)c3[nH]nnn3)Cl 4B-002 C=CCN(CC=C)c1[nH]nnn1 4B-003 c1ccc(c(c1)CN(Cc2ccccc2Cl)/C(=N/O)/N)Cl 4B-005 CC(C)(C)N1C(CC(=O)CC1=O)c2cccs2 4B-006 Cc1ccc(cc1)n2c(ncn2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F 4B-011 CC(C)(C)N1C(CC(=O)CC1=O)/C=C/c2ccccc2 4B-012 c1cc(ccc1n2c(ncn2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F)F 4B-013 Cn1c(c(c(n1)Cl)Cl)Cl 4B-014 c1ccc(c(c1)NN/C=N/C(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl 4B-016 c1ccc(c(c1)NN/C=N/C(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)F 4B-018 c1ccc2c(c1)c(ncn2)N 4B-019 CN(C)/C=N/c1c(cnn1c2ccccc2)C#N 4B-022 CC(C)(C)N1C(C/C(=N/O)/CC1=O)/C=C/c2ccccc2 4B-023 CC(C)(C#Cc1ccccn1)O 4B-025 CC(C)(C)N1C(CC(=O)/C(=C/N(C)C)/C1=O)/C=C/c2ccccc2 4B-026 CCOC(=O)COc1c(cc(cc1OC)Br)C=O 4B-028 CC(C)(C)N1C(CC(=O)CC1=O)c2ccc(cc2)F 4B-030 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N/O 4B-031 CCOC(=O)COc1c(cccc1OC)/C=N/OC 4B-033 COc1cc(cc(c1O)/C=N\OC)Br 4B-034 CNc1c(cnn1c2ccccc2)[N+](=O)[O-] 4B-037 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N\OC 4B-038 CC(C)(C)N1C(C/C(=N\O)/CC1=O)c2ccc(cc2)F 4B-039 Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2Cl)Cl 4B-041 CNc1c(cnn1c2ccc(cc2)F)[N+](=O)[O-] 4B-043 CNc1c(cnn1c2cccc(n2)Cl)[N+](=O)[O-] 4B-044 CNc1c(cnn1c2ccccc2Cl)[N+](=O)[O-] 4B-045 CNc1c(cnn1c2ccccc2F)[N+](=O)[O-] 4B-047 Cc1ccc(cc1)n2c(c(cn2)[N+](=O)[O-])NC 4B-048 CC(C)(C)N1C(CC(=O)CC1=O)c2ccc(cc2Cl)Cl 4B-050 CNc1c(cnn1c2ccc(cc2Cl)Cl)[N+](=O)[O-] 4B-051 Cc1ccc(cc1)C2CC(=O)CC(=O)N2C(C)(C)C 4B-052 CNc1c(cn(n1)C(=O)Nc2ccccc2)[N+](=O)[O-] 4B-053 c1cc(ccc1N/N=C\2/C=NNC2=O)Cl 4B-054 CN/C(=C/[N+](=O)[O-])/N1CCCC1 4B-055 CN(C)/C=C/1\C(=O)Nc2ccccc2S1 4B-057 c1ccc2c(c1)NC(=O)CS2 4B-058 CC(C)(C)N1C(C/C(=N\O)/CC1=O)c2ccc(cc2Cl)Cl 4B-062 Cc1ccc(cc1)C2C/C(=N\O)/CC(=O)N2C(C)(C)C 4B-063 C/N=C(/C(=N\Nc1ccc(cc1)Cl)/[N+](=O)[O-])\N2CCCC2 4B-064 c1ccc2c(c1)NC(=O)/C(=C\Nc3ccc(cc3)Cl)/S2 4B-065 c1ccc2c(c1)NC(=O)/C(=C\Nc3ccccc3Cl)/S2 4B-067 c1ccc2c(c1)NC(=O)/C(=C\Nc3cccc(c3)Cl)/S2 4B-068 Cc1ccc(cc1)N/C=C/2\C(=O)Nc3ccccc3S2 4B-069 COc1ccc(cc1)N/C=C/2\C(=O)Nc3ccccc3S2 4B-070 c1ccc2c(c1)NC(=O)/C(=C\Nc3cccc(c3)C(F)(F)F)/S2 4B-071 c1ccc(c(c1)CN/C=C/2\C(=O)Nc3ccccc3S2)Cl 4B-073 c1ccc2c(c1)NC(=O)/C(=C\NCc3ccc(cc3)Cl)/S2 4B-074 COc1ccc(cc1)CN/C=C/2\C(=O)Nc3ccccc3S2 4B-075 c1cc(cc(c1)Cl)N/N=C\2/C=NNC2=O 4B-076 c1ccc(c(c1)N/N=C\2/C=NNC2=O)Cl 4B-078 c1ccc(c(c1)C(F)(F)F)N/N=C\2/C=NNC2=O 4B-079 COc1cccc(c1)N/N=C\2/C=NNC2=O 4B-080 Cn1c(c(c(n1)Cl)Cl)Oc2ccccc2 4B-082 C/N=C(/C(=N/Nc1cccc(c1)C(F)(F)F)/[N+](=O)[O-])\N2CCCC2 4B-088 CCOC(=O)COc1c(cc(cc1OC)Cl)C=O 4B-094 C/N=C(/C[N+](=O)[O-])\NCC(OC)OC 4B-095 CN(C)/C=C/1\C(=O)Nc2ccc(cc2S1)Cl 4B-097 c1cc2c(cc1Cl)nc(o2)S 4B-098 CCOC(=O)COc1c(cc(cc1OC)Cl)/C=N\O 4B-099 CCOC(=O)COc1c(cc(cc1OC)Cl)/C=N\OC 4B-100 c1ccc(cc1)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl 4B-101 c1ccc(c(c1)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl)O 4B-102 c1cc2c(cc1Cl)S/C(=C/Nc3cc(ccc3O)Cl)/C(=O)N2 4B-103 C(#N)/C(=N\O)/C(=O)N 4B-107 c1ccc(cc1)C(=O)O/N=C(\C#N)/C(=O)N 4B-109 COc1cc(cc(c1O)/C=N/c2ccc(cc2)Cl)Br 4B-110 c1ccc(c(c1)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl)Cl 4B-111 c1cc(cc(c1)Cl)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl 4B-112 c1ccc(c(c1)C(F)(F)F)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl 4B-113 COc1ccc(cc1)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl 4B-115 COc1ccccc1N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl 4B-116 c1cc(cc(c1)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl)C(F)(F)F 4B-117 c1cc(ccc1N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl)Cl 4B-118 Cc1ccc(cc1)N/C=C/2\C(=O)Nc3ccc(cc3S2)Cl 4B-119 c1ccc(c(c1)CSc2nc3cc(ccc3o2)Cl)Cl 4B-120 c1cc(cc(c1)Cl)CSc2nc3cc(ccc3o2)Cl 4B-121 c1cc(ccc1C(=O)CSc2nc3cc(ccc3o2)Cl)Cl 4B-123 CCOC(=O)CSc1nc2cc(ccc2o1)Cl 4B-124 c1cc2c(cc1Cl)nc(o2)Sc3ccc(cn3)[N+](=O)[O-] 4B-126 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N\c2ccc(cc2)Cl 4B-127 CN(C)c1nnnn1c2ccc(cc2Cl)Cl 4C-001 COc1cccc(c1)N/C=C/c2c(c(no2)c3c(cccc3Cl)F)C#N 4C-004 CN(C)c1nnnn1c2ccc(cc2F)F 4C-005 CN(C)c1nnnn1c2cccc(c2)C(F)(F)F 4C-006 CNc1c(cnc(n1)c2cccnc2)[N+](=O)[O-] 4C-007 CN(C)c1nnnn1c2ccc(cc2)OC(F)(F)F 4C-008 COc1ccccc1N/C=C/c2c(c(no2)c3c(cccc3Cl)F)C#N 4C-013 CN(C)c1nnnn1c2ccc(cc2)C#N 4C-014 CN(C)c1nnnn1c2ccsc2C(=O)OC 4C-017 CN(C)c1nnnn1Cc2ccccc2 4C-018 CN(C)c1nnnn1N(C)C 4C-019 CN(C)c1nnnn1Cc2cccs2 4C-020 CN(C)c1nnnn1Cc2ccc(cc2Cl)Cl 4C-021 CN\1C(=O)CS/C1=C/[N+](=O)[O-] 4C-023 Cc1csc(n1)Nc2ncc(c(n2)NC)[N+](=O)[O-] 4C-024 CN(C)c1nnnn1c2cccnc2 4C-025 Cc1nnc(n1N)C 4C-026 CN(C)c1nnnn1c2ccncc2 4C-029 COc1ccc(cc1)S(=O)(=O)N 4C-033 CN(C)c1nnnn1S(=O)(=O)c2ccc(cc2)OC 4C-036 Cn1c(nc(n1)N)SC 4C-037 CN(C)c1nnnn1S(=O)(=O)c2ccc(cc2Cl)Cl 4C-039 COCc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)OC 4C-041 CCc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)OC 4C-042 CN(C)c1nnnn1S(=O)(=O)c2ccccc2 4C-043 c1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)Cl 4C-044 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)OC 4C-045 Cc1ccnc(c1)n2c(nnn2)N(C)C 4C-047 Cn1/c(=C\[N+](=O)[O-])/s/c(=C/c2cccc(c2)Cl)/c1=O 4C-048 CSc1c(c(sn1)/C=C/Nc2ccccc2)C#N 4C-049 Cn1/c(=C\[N+](=O)[O-])/s/c(=C/c2cccc(c2)OC)/c1=O 4C-050 CN(C)c1nnnn1c2ccc(cn2)Cl 4C-051 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)Cl)Cl 4C-052 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)O 4C-056 c1cc(ccc1N\2C(=O)CS/C2=C\[N+](=O)[O-])Cl 4C-059 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)OC 4C-062 c1cc(ccc1N\2C(=O)CS/C2=C\[N+](=O)[O-])F 4C-064 CN(C)/C=C/c1c(c(no1)c2c(cccc2Cl)F)C(=O)OC 4C-068 c1ccc(cc1)N\2C(=O)CS/C2=C\[N+](=O)[O-] 4C-073 COc1ccc(cc1)N\2C(=O)CS/C2=C\[N+](=O)[O-] 4C-077 CN(C)c1nnnn1Cc2cccnc2 4C-079 Cn1/c(=C\[N+](=O)[O-])/s/c(=C/N(C)C)/c1=O 4C-081 COC(=O)c1c(onc1c2c(cccc2Cl)F)/C=C/Nc3ccc(cc3)Cl 4C-083 COC(=O)c1c(onc1c2c(cccc2Cl)F)/C=C/Nc3ccccc3 4C-084 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)Nc4ccc(cc4)Cl 4C-085 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)Nc4cccc(c4)C(F)(F)F 4C-086 COC(=O)c1c(onc1c2c(cccc2Cl)F)/C=C/Nc3ccc(cc3Cl)Cl 4C-087 Cn1c(nnc1C(F)(F)F)CN(O)S(=O)(=O)c2ccc(cc2)Cl 4C-088 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)NCc4ccccc4 4C-089 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)NCc4ccc(cc4)Cl 4C-090 Cn1c(nnc1C(F)(F)F)CN(O)S(=O)(=O)C 4C-091 Cc1c(cnn1c2ccccc2)CC(=O)NNC(=S)NCC=C 4C-093 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)NC(C)(C)C 4C-099 Cc1c(cc2c(=O)c3ccccc3oc2n1)C(=O)NCC=C 4C-100 COc1ccc(cc1)N/C=C/c2c(c(no2)c3c(cccc3Cl)F)C(=O)OC 4C-104 Cc1ccc(cc1)N/C=C/c2c(c(no2)c3c(cccc3Cl)F)C(=O)OC 4C-106 COc1ccc(cc1)N/C(=C\[N+](=O)[O-])/NC(=N)N 4C-108 c1cc(c(cc1Cl)Cl)OCC(=C(C#N)C#N)N 4C-111 c1cc2cccc3c2c(c1)COC3=O 4C-112 c1ccc(cc1)C2CC(=O)Oc3c2c(cc(c3)O)O 4D-002 c1cc(c(c(c1)Cl)CSc2nc3nccc(n3n2)c4ccc(cc4Cl)Cl)Cl 4D-003 CCOC(=O)COc1ccccc1[N+](=O)[O-] 4D-011 c1ccc2c(c1)N(C(=O)CO2)O 4D-012 CN(C)/C=C(/C(=O)c1ccc(cc1)Cl)\S(=O)(=O)c2ccc(cc2)Cl 4D-015 c1cc(ccc1c2c(cnc(n2)N)S(=O)(=O)c3ccc(cc3)Cl)Cl 4D-016 c1cc(ccc1c2c(c[nH]n2)S(=O)(=O)c3ccc(cc3)Cl)Cl 4D-017 CC(c1ccnc2n1nc(n2)SCc3c(cccc3Cl)Cl)Oc4ccc(cc4Cl)Cl 4D-019 Cc1ccc(cc1)SCC(=O)c2ccc(cc2)Cl 4D-020 c1cc(c(c(c1)Cl)CSc2nc3nccc(n3n2)c4ccc(cc4)F)F 4D-023 c1cc(ccc1C2CC(=O)Oc3c2c(cc(c3)O)O)Cl 4D-025 CN(C)/C=C(/C(=O)c1ccc(cc1)Cl)\Sc2ccc(cc2)Cl 4D-028 c1cc(ccc1c2c(cnc(n2)N)Sc3ccc(cc3)Cl)Cl 4D-031 c1cc(ccc1c2c(c[nH]n2)Sc3ccc(cc3)Cl)Cl 4D-032 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)Cl 4D-033 Cc1ccc(cc1)S/C(=C\N(C)C)/C(=O)c2ccc(cc2)Cl 4D-037 c1ccc2c(c1)ncc(n2)Oc3ccccc3NS(=O)(=O)c4ccc(cc4)Cl 4D-038 Cc1ccc(cc1)Sc2cnc(nc2c3ccc(cc3)Cl)N 4D-039 Cc1ccc(cc1)Sc2c[nH]nc2c3ccc(cc3)Cl 4D-040 c1cc(ccc1N2CSCC2=O)Cl 4D-045 CCOC(=O)c1cc2cccnc2nc1C 4D-046 CC(=O)/C(=C/N(C)C)/Sc1ccc(cc1)Cl 4D-051 Cc1c(cnc(n1)N)Sc2ccc(cc2)Cl 4D-054 c1cc(ccc1N2CS(=O)(=O)CC2=O)Cl 4D-055 Cc1c(c[nH]n1)Sc2ccc(cc2)Cl 4D-056 Cc1ccc(cc1)S(=O)(=O)/C(=C\N(C)C)/C(=O)c2ccc(cc2)Cl 4D-060 CCOC(=O)C1CC(=NNC1=O)c2ccccc2 4D-063 Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2c3ccc(cc3)Cl)N 4D-069 COC(=O)CC(=O)/C(=N/Nc1ccccc1)/C(=O)OC 4D-072 Cc1ccc(cc1)S/C(=C\N(C)C)/C(=O)C 4D-073 Cc1ccc(cc1)S(=O)(=O)c2c[nH]nc2c3ccc(cc3)Cl 4D-074 Cc1ccc(cc1)Sc2cnc(nc2C)N 4D-075 c1ccc(cc1)CSc2nc3ccsc3c(=O)n2c4ccccc4 4D-076 CCOC(=O)c1cc(n[nH]c1=O)c2ccccc2 4D-077 CN(C)/C=C/1\C(=O)N(CS1(=O)=O)c2ccc(cc2)Cl 4D-078 Cc1ccc(cc1)Sc2c[nH]nc2C 4D-080 c1ccc(cc1)c2cc(c(=O)[nH]n2)C(=O)N 4D-083 COC(=O)CC(=O)/C(=N/Nc1ccc(cc1Cl)Cl)/C(=O)OC 4D-085 c1ccc(cc1)/C=[N+]/2\CCC(=O)[N-]2 4D-087 c1ccc(cc1)CN2CCC(=O)N2 4D-090 c1ccc(cc1)c2cc(c(nn2)Cl)C#N 4D-091 c1ccc(cc1)/C=C/CSc2nc([nH]n2)N 4D-093 c1cc(c(c(c1)Cl)CSc2nc3ncc(c(n3n2)N)c4ccc(cc4)Cl)F 4D-095 c1ccc(cc1)c2cc(c(nn2)Sc3ccc(cc3)Cl)C#N 4D-096 c1ccc(cc1)c2cc(c(nn2)SCc3ccc(cc3)Cl)C#N 4D-097 Cc1ccc(cc1)Sc2c(cc(nn2)c3ccccc3)C#N 4D-098 COc1ccc(cc1)Sc2c(cc(nn2)c3ccccc3)C#N 4D-099 c1ccc(cc1)c2cc(c(nn2)Sc3cccc(c3)C(F)(F)F)C#N 4D-100 c1ccc(cc1)c2cc(c(nn2)Sc3ccccc3)C#N 4D-101 COC(=O)c1ccccc1Sc2c(cc(nn2)c3ccccc3)C#N 4D-102 COC(=O)c1ccc(cc1)Sc2c(cc(nn2)c3ccccc3)C#N 4D-103 c1ccc(cc1)c2cc(c(nn2)Sc3ccc(cc3)F)C#N 4D-104 c1ccc(cc1)CSc2c(cc(nn2)c3ccccc3)C#N 4D-105 COC(=O)c1c(ccs1)OCc2ccc(cc2)F 4D-106 CC(C)(C(=O)N)N1CCN(CC1)c2ccccc2 4E-001 c1ccc(cc1)Cc2c3ccccc3c(nn2)SCc4ccc(cc4)Cl 4E-002 c1ccc(cc1)C(=O)NC(=O)CC(=O)NC(=O)c2ccccc2 4E-017 C1C(=CNC(=O)N1)C#N 4E-021 COC(=O)CSc1c2ccccc2c(nn1)Cc3ccccc3 4E-025 Cc1cc(n(n1)c2cc(nc(c2)C(F)(F)F)C(F)(F)F)C 4E-026 c1ccc(cc1)Cc2c3ccccc3c(nn2)Sc4cccc[n+]4[O-] 4E-029 c1cc(ccc1CONC(=O)N/C=N/OCc2ccc(cc2)[N+](=O)[O-])[N+](=O)[O-] 4E-030 c1cc(c(c(c1)Cl)CO/N=C(/c2ccncc2)\N)Cl 4E-031 c1c(cnc(n1)Cl)C#N 4E-036 c1cc(nc(c1)F)NN 4E-037 Cc1c(c(ns1)SCC(=O)c2ccccc2)C#N 4E-040 COc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-301S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCNC(=O)/C=C/C(=O)O)OCC(F)(F)F 4E-302S c1ccnc(c1)c2nc(cc(n2)Sc3cccc(c3)C(F)(F)F)C(F)(F)F 4E-304S COc1ccc(cc1)Sc2cc(nc(n2)c3ccccn3)C(F)(F)F 4E-305S c1ccnc(c1)c2nc(cc(n2)Sc3ccc(cc3)Cl)C(F)(F)F 4E-306S CCCN1CC(=C(C1=O)C#N)O 4E-307S c1ccc(cc1)c2c(n3ccsc3n2)/C=N/OC(=O)C4CC4 4E-308S CC(C)CC(=O)O/N=C/c1c(nc2n1ccs2)c3ccccc3 4E-309S CNc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-310S CN(C)c1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-311S CN1CCN(CC1)c2cc(nc(n2)c3ccccn3)C(F)(F)F 4E-312S CCCCC(=O)O/N=C/c1c(nc2n1ccs2)c3ccccc3 4E-314S CC(C)N1CC(=C(C1=O)C#N)O 4E-315S COC(=O)CSc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-317S c1ccc(cc1)CNc2cc(nc(n2)c3ccccn3)C(F)(F)F 4E-319S c1ccnc(c1)c2nc(cc(n2)S)C(F)(F)F 4E-321S CSc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-322S CN(C)C(=O)NCCNC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F 4E-323S Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 4E-324S c1cc(c(cc1OCC(F)(F)F)C(=O)NCCNC(=O)C(F)(F)F)OCC(F)(F)F 4E-326S CCN(CC)c1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-327S CC(C)Nc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-328S C=CCNc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-329S c1ccnc(c1)c2nc(cc(n2)N3CCOCC3)C(F)(F)F 4E-330S C#CCSc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-333S c1ccnc(c1)c2nc(cc(n2)SCC(=O)O)C(F)(F)F 4E-334S CNC(=O)CSc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-335S c1ccc(cc1)Oc2cc(nc(n2)c3ccccn3)C(F)(F)F 4E-336S c1ccnc(c1)c2nc(cc(n2)Oc3cccc(c3)C(F)(F)F)C(F)(F)F 4E-337S c1ccnc(c1)c2nc(cc(n2)Oc3ccc(cc3)Cl)C(F)(F)F 4E-338S CCOC(=O)CSc1cc(nc(n1)c2ccccn2)C(F)(F)F 4E-340S CC1=NN(C(=O)C1)c2ccccc2 4E-901 Cn1c(=O)c2cc(c(=O)oc2n(c1=O)C)NC(=O)c3ccccc3 4E-902 c1ccc(cc1)C(=O)Nc2cc3ccc(cc3oc2=O)O 4E-904 c1ccc(cc1)C2=NOC(=O)C2 4E-905 Cc1c(cc(c(=O)o1)NC(=O)c2cccc(c2)C(F)(F)F)C(=O)C 4E-906 CCOC(=O)c1cc(c(=O)oc1c2ccccc2)NC(=O)c3cccc(c3)C(F)(F)F 4E-907 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)[N+](=O)[O-])C(=O)C 4E-908 Cc1c(cc(c(=O)o1)NC(=O)c2cccc(c2)C(F)(F)F)C(=O)OC 4E-910 CCOC(=O)c1cc(c(=O)oc1c2ccccc2)NC(=O)c3ccc(cc3)[N+](=O)[O-] 4E-911 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)[N+](=O)[O-])C(=O)c3ccccc3 4E-912 Cc1c(cc(c(=O)o1)NC(=O)c2ccc(cc2)[N+](=O)[O-])C(=O)OC 4E-913 CCOC(=O)c1cc(c(=O)oc1C(F)(F)F)NC(=O)c2ccccc2 4E-914 CC(=O)c1cc(c(=O)oc1/C=C/N(C)C)NC(=O)c2cccc(c2)C(F)(F)F 4E-915 c1ccc(cc1)c2c3cc(c(=O)oc3n(n2)c4ccccc4)NC(=O)c5ccccc5 4E-916 CC(=O)c1cn2c(nc1=O)OCC2 4E-920 COC(=O)C(/C=N/OCc1ccc(cc1Cl)Cl)NC(=O)c2ccccc2 4E-921 c1ccc(cc1)C(=O)OCC2(CCc3ccccc3C2=O)COC(=O)c4ccccc4 4E-923 c1ccc2c(c1)CCC(C2=O)(COC(=O)c3cccc(c3)C(F)(F)F)COC(=O)c4cccc(c4)C(F)(F)F 4E-924 c1ccc2c(c1)CCC3(C2=O)COC(OC3)c4ccc(cc4)Cl 4E-926 c1ccc(c(c1)Cc2ccc(nn2)Cl)Br 4F-001 C/C(=N\O)/c1ccc(cc1)Cl 4F-002 Cc1cc(n2c(n1)c(c(n2)/C(=C/c3ccccc3)/C#N)C#N)C 4F-003 Cc1cc(n2c(n1)c(c(n2)/C(=C/c3ccccn3)/C#N)C#N)C 4F-004 Cc1ccc(cc1)/C=C(\C#N)/c2c(c3nc(cc(n3n2)C)C)C#N 4F-005 Cc1cc(n2c(n1)c(c(n2)/C(=C/c3ccco3)/C#N)C#N)C 4F-006 Cn1cc(cc1C(=O)NNC(=N)COc2cccc(c2)C(F)(F)F)C(=O)c3ccc(cc3Cl)Cl 4F-007 C/C(=N\Oc1cccc(n1)F)/c2ccc(cc2)Cl 4F-008 c1cc(ccc1c2ccnc(n2)Cn3cncn3)F 4F-011 CCOC(=O)/C(=C/N(C)C)/C(=O)C 4F-012 CCOC(=O)c1c(c2c(snc2s1)C)/N=C/N(C)C 4F-013 Cn1cc(cc1c2nnc(o2)COc3cccc(c3)C(F)(F)F)C(=O)c4ccc(cc4Cl)Cl 4F-014 c1ncn(n1)CC(=N)NC(=O)N 4F-016 c1ccc(cc1)Nc2cc(=O)n(nc2C#N)c3ccc(cc3)Cl 4F-018 CC1(OC(=O)C(=C(COc2ccc(cc2Cl)Cl)N)C(=O)O1)C 4F-020 CCO/C(=N/C(=O)Nc1ccccc1)/Cn2cncn2 4F-022 c1ccc2c(c1)[nH]c(n2)Cn3cncn3 4F-023 CN1C(=O)C(=C(Cn2cncn2)N)C(=O)N(C1=O)C 4F-024 Cc1c(c(ns1)SCC(=O)NNC(=N)COc2cccc(c2)C(F)(F)F)C#N 4F-025 Cc1c(c(ns1)SCC(=O)NNC(=N)COc2ccccc2)C#N 4F-026 Cn1cc(cc1C(=O)NNC(=N)COc2ccccc2)C(=O)c3ccc(cc3Cl)Cl 4F-027 c1ccc(cc1)n2c(c(c(nc2=O)Cn3cncn3)C#N)N 4F-028 Cc1c(c(ns1)SCC(=O)NNC(=N)COc2ccc(cc2)F)C#N 4F-029 c1ccc(cc1)NC(=O)/N=C(/Cn2cncn2)\NNc3cccc(n3)Cl 4F-030 Cn1cc(cc1C(=O)NNC(=N)COc2ccc(cc2)F)C(=O)c3ccc(cc3Cl)Cl 4F-033 Cn1cc(cc1c2nnc(o2)COc3ccccc3)C(=O)c4ccc(cc4Cl)Cl 4F-035 c1ccc(cc1)NC(=O)/N=C(\COc2ccc(cc2Cl)Cl)/NNc3cccc(n3)Cl 4F-036 Cc1c(c(ns1)SCc2nc([nH]n2)COc3cccc(c3)C(F)(F)F)C#N 4F-038 c1ccc(cc1)n2c(c(c(nc2=O)COc3ccc(cc3Cl)Cl)C#N)N 4F-039 Cc1c(c(ns1)SCc2nc([nH]n2)COc3ccccc3)C#N 4F-040 c1ccnc(c1)SC/C(=N/NC(=O)CC#N)/N 4F-041 c1ccnc(c1)SC/C(=N/NC(=O)c2ccc(cc2)Cl)/N 4F-042 Cn1cc(cc1c2nnc(o2)COc3ccc(cc3)F)C(=O)c4ccc(cc4Cl)Cl 4F-044 Cc1c(c(ns1)SCc2nnc(o2)COc3ccccc3)C#N 4F-045 c1ccnc(c1)SC/C(=N/Nc2c(cc(cn2)C(F)(F)F)Cl)/N 4F-046 c1ccc(cc1)Nc2nc(nn2c3cccc(n3)Cl)Cn4cncn4 4F-047 COC(=O)c1ccccc1OCC#N 4F-048 c1ccnc(c1)SCc2ncn(n2)c3c(cc(cn3)C(F)(F)F)Cl 4F-049 CCO/C(=N/C(=O)Nc1ccc(cc1)Cl)/Cn2cncn2 4F-050 Cc1c(c(ns1)SCC(=O)NNC(=N)Cn2cncn2)C#N 4F-051 c1cc[n+](c(c1)SC/C(=N/NC(=O)c2ccncc2)/N)[O-] 4F-052 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)NN 4F-054 c1cc(ccc1n2c(=O)cc3c(n2)c(n[nH]3)O)Cl 4F-055 c1cc(ccc1n2c(c(c(nc2=O)Cn3cncn3)C#N)N)Cl 4F-056 c1cc[n+](c(c1)SCc2nc([nH]n2)c3ccncc3)[O-] 4F-057 CCOC(=O)c1cnn(c1C)c2c(cc(cn2)C(F)(F)F)Cl 4F-058 c1cc(ccc1COc2ccsc2C(=O)NNC(=N)COc3ccc(cc3Cl)Cl)F 4F-059 c1ccc(cc1)NN/C(=N\C(=O)Nc2ccc(cc2)Cl)/Cn3cncn3 4F-060 COC(=O)c1c(cc(=O)n(n1)c2cccc(c2)C(F)(F)F)NN 4F-061 Cn1cc(cc1C(=O)NNC(=N)COc2ccc(cc2)Cl)C(=O)c3ccc(cc3Cl)Cl 4F-062 Cn1cc(cc1c2nnc(o2)COc3ccc(cc3)Cl)C(=O)c4ccc(cc4Cl)Cl 4F-063 c1ccc(cc1)n2c(nc(n2)Cn3cncn3)Nc4ccc(cc4)Cl 4F-064 c1cc(ccc1COc2ccsc2c3nc([nH]n3)COc4ccc(cc4Cl)Cl)F 4F-065 c1ccc2c(c1)C3(C(=O)N2Cc4cccc(c4)C(F)(F)F)N(C(=O)CS3)c5ccc(c(c5)Cl)Cl 4F-301S c1ccc2c(c1)C3(C(=O)N2Cc4ccc(c(c4)Cl)Cl)N(C(=O)CS3)c5ccc(c(c5)Cl)Cl 4F-302S c1ccc2c(c1)C3(C(=O)N2)N(C(=O)CS3)c4cccc(c4)C(F)(F)F 4F-303S c1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5ccc(cc5Cl)Cl 4F-305S c1ccc(cc1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5ccccc5 4F-306S c1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5cccc(c5)C(F)(F)F 4F-308S c1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5ccc(c(c5)Cl)Cl 4F-309S c1cc(cc(c1)NC(=O)c2ccc(nc2)n3cncn3)C(F)(F)F 4F-310S c1cc(c(cc1F)F)NC(=O)c2ccc(nc2)n3cncn3 4F-311S COc1ccc(cc1)N2C(=O)CSC23c4ccccc4NC3=O 4F-313S c1ccc(c(c1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5cccc(c5)C(F)(F)F)Cl 4F-314S c1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5ccccc5Cl 4F-315S c1ccc(cc1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5cccc(c5)C(F)(F)F 4F-317S c1ccc2c(c1)C3(C(=O)N2Cc4ccc(cc4Cl)Cl)N(C(=O)CS3)c5cccc(c5)C(F)(F)F 4F-318S c1cc(c2ncnn2c1)NC(=O)CCl 4F-319S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccn3c2ncn3 4F-320S CCCCC(=O)Nc1cccn2c1ncn2 4F-321S CS(=O)(=O)Nc1cccn2c1ncn2 4F-323S c1cc(c2ncnn2c1)NC(=O)C3CC3 4F-324S c1ccc2c(c1)C3(C(=O)N2Cc4cccc(c4)C(F)(F)F)N(C(=O)CS3)c5cccc(c5)C(F)(F)F 4F-326S c1ccc2c(c1)C3(C(=O)N2Cc4c(cccc4Cl)Cl)N(C(=O)CS3)c5cccc(c5)C(F)(F)F 4F-327S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)C(Cl)Cl)SCc2ccccc2Cl 4F-328S c1cc(ccc1n2cc(nn2)CO)Cl 4F-329S Cn1c(c(c(n1)C(F)(F)F)/C=N/O)Sc2ccccc2C(=O)OC 4F-330S CC(C)C(=O)O/N=C/c1c(nn(c1SCc2ccccc2Cl)C)C(F)(F)F 4F-331S c1ccc2c(c1)C3(C(=O)N2Cc4ccc(cc4)C(F)(F)F)N(C(=O)CS3)c5cccc(c5)C(F)(F)F 4F-333S c1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5ccc(cc5)Cl 4F-335S COc1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5ccc(cc5)Cl 4F-336S c1ccc2c(c1)C3(C(=O)N2Cc4ccc(cc4)Cl)N(C(=O)CS3)c5ccc(c(c5)Cl)Cl 4F-337S c1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5cccc(c5)Cl 4F-338S c1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5c(cccc5Cl)Cl 4F-339S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2)Sc3ccccc3C(=O)OC 4F-341S CC(C)(C)c1ccc(cc1)CSc2c(c(nn2C)C(F)(F)F)/C=N/OC(=O)c3ccccc3 4F-342S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(cc2Cl)Cl)Sc3ccccc3C(=O)OC 4F-343S c1ccc(cc1)NC(=O)OCc2cn(nn2)c3ccc(cc3)Cl 4F-344S c1cc(c2ncnn2c1)NC(=O)C(Cl)Cl 4F-345S c1cc(c2ncnn2c1)NC(=O)C(Cl)(Cl)Cl 4F-346S c1cc(c2ncnn2c1)NC(=O)C(F)(F)F 4F-347S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccc(cc2Cl)Cl)Sc3ccccc3C(=O)OC 4F-349S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)CCl)Sc2ccccc2C(=O)OC 4F-350S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)C2CC2)Sc3ccccc3C(=O)OC 4F-351S COc1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5ccccc5 4F-352S COc1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5ccc(c(c5)Cl)Cl 4F-354S COc1ccc(cc1)N2C(=O)CSC23c4ccccc4N(C3=O)Cc5c(cccc5Cl)Cl 4F-355S CC(C)(C)c1ccc(cc1)CSc2c(c(nn2C)C(F)(F)F)/C=N/OC(=O)c3ccc(cc3)OC 4F-356S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(cc2)Cl)Sc3ccccc3C(=O)OC 4F-357S c1cc(c(cc1n2cc(nn2)CO)Cl)Cl 4F-359S c1ccc2c(c1)C3(C(=O)N2Cc4cccc(c4)C(F)(F)F)N(C(=O)CS3)c5ccc(cc5)Cl 4F-360S c1ccc2c(c1)C3(C(=O)N2Cc4c(cccc4Cl)Cl)N(C(=O)CS3)c5ccc(cc5)Cl 4F-361S COc1ccc(cc1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5ccc(cc5)Cl 4F-362S COc1ccc(cc1)CN2c3ccccc3C4(C2=O)N(C(=O)CS4)c5ccc(cc5)OC 4F-363S c1cc(cc(c1)Cl)NC(=O)OCc2cn(nn2)c3ccc(cc3)Cl 4F-364S c1cc(cc(c1)NC(=O)OCc2cn(nn2)c3ccc(cc3)Cl)C(F)(F)F 4F-365S c1cc(ccc1NC(=O)OCc2cn(nn2)c3ccc(cc3)Cl)Cl 4F-366S CCNC(=O)OCc1cn(nn1)c2ccc(cc2)Cl 4F-367S c1ccc(cc1)C(=O)OCc2cn(nn2)c3ccc(cc3)Cl 4F-368S c1ccc(cc1)COCc2cn(nn2)c3ccc(cc3)Cl 4F-369S CO/N=C/c1cn(nn1)c2ccc(cc2)Cl 4F-370S c1cc(ccc1n2cc(nn2)/C=N/O)Cl 4F-372S Cc1ccccc1NC(=O)OCc2cn(nn2)c3ccc(cc3)Cl 4F-373S Cc1ccc(cc1)NC(=O)OCc2cn(nn2)c3ccc(cc3)Cl 4F-374S c1cc(ccc1n2cc(nn2)C=O)Cl 4F-375S c1cc(ccc1n2cc(nn2)COC(=O)CCl)Cl 4F-376S CCCCC(=O)OCc1cn(nn1)c2ccc(cc2)Cl 4F-377S c1cc(ccc1n2cc(nn2)COC(=O)C(Cl)(Cl)Cl)Cl 4F-378S c1cc(ccc1C(=O)OCc2cn(nn2)c3ccc(cc3)Cl)Cl 4F-379S c1cc(ccc1n2cc(nn2)COC(=O)c3ccc(cc3Cl)Cl)Cl 4F-380S c1cc(cc(c1)C(F)(F)F)C(=O)OCc2cn(nn2)c3ccc(cc3)Cl 4F-381S CC(C)(C)c1ccc(cc1)CSc2c(c(nn2C)C(F)(F)F)/C=N/OC(=O)c3ccc(cc3Cl)Cl 4F-382S CC(C)(C)C(=O)OCc1cn(nn1)c2ccc(cc2)Cl 4F-383S c1cc(ccc1n2cc(nn2)COC(=O)CCCCl)Cl 4F-384S c1ccc(cc1)NC(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl 4F-387S CS(=O)(=O)OCc1cn(nn1)c2ccc(cc2)Cl 4F-388S c1ccc(cc1)C(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl 4F-389S COC(=O)c1c(c2cccnc2s1)O 4F-390S Cn1c(c(c(n1)C(F)(F)F)C#N)Cl 4F-391S Cn1c(c(c(n1)C(F)(F)F)C#N)Sc2ccccc2C(=O)OC 4F-392S c1ccc(c(c1)C(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl)Cl 4F-393S c1cc(cc(c1)NC(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl)C(F)(F)F 4F-394S COC(=O)c1c(c2cccnc2s1)OCc3ccc(c(c3)Cl)Cl 4F-395S c1ccc2c(c1)nc(c(=O)n2Cc3ccc(cc3Cl)Cl)C(=O)Nc4ccc(cc4)F 4F-401S COC(=O)c1c(c2cccnc2s1)OCc3ccccc3 4F-402S COC(=O)c1c(c2cccnc2s1)OCc3cccc(c3)C(F)(F)F 4F-403S COC(=O)c1c(c2cccnc2s1)OCc3ccc(cc3Cl)Cl 4F-404S Cn1c(c(c(n1)C(F)(F)F)C#N)Sc2ccccc2Cl 4F-406S COC(=O)c1c(c2cccnc2s1)OCc3ccccc3Cl 4F-407S COC(=O)c1c(c2cccnc2s1)OCc3cccc(c3)Cl 4F-408S COC(=O)c1c(c2cccnc2s1)OCc3ccc(cc3)Cl 4F-409S COC(=O)c1c(c2cccnc2s1)OCc3c(cccc3Cl)Cl 4F-410S c1ccc(cc1)n2cc(nn2)CO 4F-411S c1cc(ccc1C(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl)Cl 4F-412S c1cc(cc(c1)NC(=O)c2cc(cc(c2)Cl)Cl)C(F)(F)F 4F-413S c1cc(ccc1NC(=O)c2cc(cc(c2)Cl)Cl)[N+](=O)[O-] 4F-414S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)c2ccccc2Cl 4F-415S Cn1c(c(c(n1)C(F)(F)F)C#N)Sc2ccc(cc2)Cl 4F-416S c1cc(c(cc1n2cc(nn2)COC(=O)c3ccc(cc3Cl)Cl)Cl)Cl 4F-417S c1ccc(cc1)n2cc(nn2)COC(=O)c3ccc(cc3Cl)Cl 4F-418S CC(C)C(=O)OCc1cn(nn1)c2ccc(c(c2)Cl)Cl 4F-419S Cc1ccc(cc1)NC(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl 4F-420S c1cc2c(c(sc2nc1)C(=O)O)OCc3ccc(c(c3)Cl)Cl 4F-421S c1cc(cc(c1)Cl)NC(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl 4F-422S COc1ccc(cc1)C(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl 4F-423S c1cc(c(cc1n2cc(nn2)COC(=O)C(Cl)(Cl)Cl)Cl)Cl 4F-424S CN(c1cccc(c1)C(F)(F)F)C(=O)c2cc(cc(c2)Cl)Cl 4F-425S CN(c1ccc(cc1)[N+](=O)[O-])C(=O)c2cc(cc(c2)Cl)Cl 4F-426S c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4ccc(cc4)Cl 4F-427S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)c2ccc(cc2)Cl 4F-428S COc1ccc(cc1)CON2C(=O)c3ccccc3C2=O 4F-900 c1ccc(cc1)C(=O)NCC(=O)NCCOC(=O)c2ccccc2 4F-901 COc1ccc(cc1)CON.Cl 4F-903 c1cc(c(cc1C(=O)NCC(=O)O)Cl)Cl 4F-904 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)Cl)/C(=O)N(C2=O)OCc4ccc(cc4)Cl 4F-905 CO/N=C/C1c2ccccc2C(=O)N(C1=O)OCc3ccc(cc3Cl)Cl 4F-906 c1cc(c(cc1C(=O)NCC(=O)NCCO)Cl)Cl 4F-909 Cc1cccc(c1)C(=O)NCC(=O)NCCO 4F-910 c1cc(ccc1C(=O)NCC(=O)NCCO)F 4F-911 c1ccc2c(c1)/C(=C/Nc3cccc(c3)C(F)(F)F)/C(=O)N(C2=O)OCc4ccc(cc4)Cl 4F-912 Cc1ccc(cc1)N/C=C\2/c3ccccc3C(=O)N(C2=O)OCc4ccc(cc4)Cl 4F-913 Cc1cccc(c1)C(=O)NCC(=O)N2CCN(CC2)c3ccc(cc3)Cl 4F-916 COc1cccc(c1)CON2C(=O)c3ccccc3C2=O 4F-917 COc1ccc(cc1)C(=O)NCC(=O)N2CCN(CC2)c3ccc(cc3)Cl 4F-918 c1cc(ccc1N2CCN(CC2)C(=O)CNC(=O)c3ccc(c(c3)Cl)Cl)Cl 4F-919 Cc1cccc(c1)C(=O)NCC(=O)NCCOC(=O)c2c(onc2c3c(cccc3Cl)F)C 4F-921 COc1cccc(c1)CON.Cl 4F-922 c1cc(ccc1C2(C3CC4CC(C3)CC2C4)CC(=O)O)F 4F-923 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)OCCNC(=O)CNC(=O)c3ccc(cc3)OC 4F-924 c1ccc2c(c1)C(=O)N(C2=O)OCCOc3cccc(c3)C(F)(F)F 4F-925 c1cc(ccc1C2(C3CC4CC(C3)CC2C4)CC(=O)O)Cl 4F-927 c1ccc2c(c1)c3c([nH]2)c(ncn3)N4CCN(CC4)c5ccc(cc5)Cl 4F-928 COc1ccc(cc1)N2CCN(CC2)c3c4c(c5ccccc5[nH]4)ncn3 4F-929 CCOC(=O)/C=C(\N)/NNC(=O)c1ccccc1 4F-930 c1ccc2c(c1)c3c([nH]2)c(ncn3)N4CCCCC4 4F-931 c1ccc2c(c1)c3c([nH]2)c(ncn3)N4CCCC4 4F-932 CNc1c2c(c3ccccc3[nH]2)ncn1 4F-934 c1ccc(c(c1)CON2C(=O)c3ccccc3C2=O)F 4F-935 c1ccc2c(c1)C(=O)N(C2=O)OCc3cccc(c3)F 4F-936 Cc1cccc(c1NC(=O)c2c(cn3c2nc(cc3C)C)c4ccc(cc4)Cl)C 4F-937 CCOC(=O)/C=C(/[NH3+])\Oc1ccccc1.[Cl-] 4F-938 CCOC(=O)/C=C(\N)/Nc1ccc(cc1)Cl.Cl 4F-939 CCOC(=O)/C=C(\N)/Nc1ccc(cc1)C.Cl 4F-940 CCOC(=O)c1cc([nH]c1NNC(=O)c2ccccc2)c3ccc(cc3)Cl 4F-941 COC(=O)c1ccccc1SCC#N 4F-942 Cc1cc(n2cc(c(c2n1)C(=O)Nc3ccc(cc3)Cl)c4ccc(cc4)Cl)C 4F-943 Cc1cc(n2cc(c(c2n1)C(=O)Nc3cccc(c3)Cl)c4ccc(cc4)Cl)C 4F-944 CN1CCN(CC1)c2c3c(c4ccccc4[nH]3)ncn2 4F-945 c1ccc(c(c1)/C=N/Nc2c(=O)[nH]c3ccccc3n2)Cl 4F-946 c1ccc2c(c1)[nH]c(=O)c(n2)N/N=C/c3cccc(c3)Cl 4F-947 c1ccc2c(c1)[nH]c(=O)c(n2)N/N=C/c3ccc(cc3)Cl 4F-948 c1ccc(cc1)/C=C\C=N\Nc2c(=O)[nH]c3ccccc3n2 4F-949 COc1ccc(cc1)/C=N/Nc2c(=O)[nH]c3ccccc3n2 4F-950 c1ccc(c(c1)CON)F.Cl 4F-951 c1cc(cc(c1)F)CON.Cl 4F-952 c1ccc2c(c1)c(c(s2)C#N)O 4F-953 CCOC(=O)c1cc([nH]c1Nc2ccc(cc2)Cl)c3ccc(cc3)Cl 4F-954 CCOC(=O)c1cc([nH]c1Nc2ccc(cc2)C)c3cccc(c3)[N+](=O)[O-] 4F-955 COC(=O)CSc1c2c(c3ccccc3[nH]2)ncn1 4F-957 c1cc(cc(c1)OCCON)C(F)(F)F.Cl 4F-958 CCOC(=O)c1c(c([nH]c1N2CCN(CC2)c3ccc(cc3)Cl)c4ccccc4)c5ccccc5 4F-962 CCOC(=O)/C=C(\N)/NNC(=O)c1ccncc1 4F-963 CCOC(=O)c1c(cn2c1nc(cc2C)C)c3ccccc3 4F-964 Cc1ccc(cc1)/C=N/Nc2c(=O)[nH]c3ccccc3n2 4F-965 c1ccc2c(c1)[nH]c(=O)c(n2)N/N=C/c3ccc(cc3)F 4F-966 c1ccc2c(c1)[nH]c(=O)c(n2)N/N=C/c3c(cccc3Cl)F 4F-967 c1ccc2c(c1)[nH]c(=O)c(n2)N/N=C/c3cccc(c3)C(F)(F)F 4F-968 c1ccc2c(c1)c(c(s2)C#N)OCC#N 4F-969 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Sc3cc(cnc3C#N)C(F)(F)F)Cl 4G-003 Cc1c[nH]nc1c2ccc3c(c2)ccc(c3Br)OC 4G-004 c1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 4G-005 c1c(cnc(c1Cl)c2ncc3n2cc(cc3Cl)C(F)(F)F)C(F)(F)F 4G-006 CO/N=C/C(c1ccc(cc1)Cl)S(=O)(=O)c2cc(cnc2C#N)C(F)(F)F 4G-008 c1cc(ccc1N/N=C/c2c(cc(cn2)C(F)(F)F)Cl)Cl 4G-010 Cc1cn(nc1c2ccc3c(c2)ccc(c3Br)OC)c4ccc(cc4)F 4G-011 Cc1cn(nc1c2ccc3c(c2)ccc(c3Br)OC)c4c(cc(cn4)C(F)(F)F)Cl 4G-012 Cc1cnc(nc1c2ccc3c(c2)ccc(c3Br)OC)N 4G-014 CCC(=O)Nc1ccc(cc1)Sc2cc(cnc2C#N)C(F)(F)F 4G-015 C(=N/N)(\N[NH3+])/NN.[Cl-] 4G-016 c1cc(ccc1C(=O)n2ccc(n2)/C=C/c3c(cc(cn3)C(F)(F)F)Cl)Cl 4G-017 Cc1cc(n(n1)C2=NN=C(NN2)n3c(cc(n3)C)C)C 4G-018 c1cn(nc1/C=C/c2c(cc(cn2)C(F)(F)F)Cl)c3c(cc(cn3)C(F)(F)F)Cl 4G-019 c1ccc(cc1)C(c2cc(no2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 4G-020 c1cc(ccc1C#N)N/N=C/c2c(cc(cn2)C(F)(F)F)Cl 4G-021 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)c2csc([nH+]2)COc3cccc(c3)C(F)(F)F.[Br-] 4G-022 c1cn(nc1/C=C/c2c(cc(cn2)C(F)(F)F)Cl)C(=O)CCl 4G-023 c1c(cnc(c1N2CCCC2)C#N)C(F)(F)F 4G-025 Cc1cc(n(n1)c2nnc(nn2)N3CCN(CC3)c4ccccc4)C 4G-027 COc1ccc(cc1)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 4G-028 Cc1cc(n(n1)c2nnc(nn2)NCc3ccc(cc3)Cl)C 4G-029 Cc1cc(n(n1)c2nnc(nn2)NCc3ccncc3)C 4G-031 c1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)Sc3cc(cnc3C#N)C(F)(F)F)Cl 4G-032 CN1C(=O)CCC1(c2ccccc2)O 4G-034 CC(/C=N/OC)C(=O)c1ccc2c(c1)ccc(c2Br)OC 4G-036 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)c2csc([nH+]2)c3ccc(cc3)Cl.[Br-] 4G-037 c1cc(ccc1NC(=O)/C(=N/Nc2ccc(cc2)Cl)/N=N/c3ccc(cc3)Cl)Cl 4G-038 c1cc(ccc1NC(=O)/C(=N/Nc2ccc(c(c2)Cl)Cl)/N=N/c3ccc(c(c3)Cl)Cl)Cl 4G-039 CS(=O)(=O)n1ccc(n1)/C=C/c2c(cc(cn2)C(F)(F)F)Cl 4G-040 c1cc(c(cc1Cl)Cl)N/C=C(\[N+](=O)[O-])/Br 4G-042 CC(/C=N/OCc1ccc(cc1Cl)Cl)C(=O)c2ccc3c(c2)ccc(c3Br)OC 4G-045 CC(/C=N/OCc1c(cccc1Cl)Cl)C(=O)c2ccc3c(c2)ccc(c3Br)OC 4G-046 c1c(cnc(c1N=N#N)C#N)C(F)(F)F 4G-049 c1c(cnc2c1n3c(c(nn3)C#N)nc2N)C(F)(F)F 4G-050 c1ccc(cc1)c2c3nc(c4c(n3nn2)cc(cn4)C(F)(F)F)N 4G-051 COc1ccc(cc1OC)c2c3nc(c4c(n3nn2)cc(cn4)C(F)(F)F)N 4G-053 Cn1cccc1c2c3nc(c4c(n3nn2)cc(cn4)C(F)(F)F)N 4G-054 c1cc(c(cc1Cl)Cl)c2c3nc(c4c(n3nn2)cc(cn4)C(F)(F)F)N 4G-055 c1cc(ccc1c2c3nc(c4c(n3nn2)cc(cn4)C(F)(F)F)N)Cl 4G-056 c1cc(c(c(c1)Cl)c2c3nc(c4c(n3nn2)cc(cn4)C(F)(F)F)N)F 4G-058 Cc1ccc(cc1)N/N=C(/c2c(cc(cn2)C(F)(F)F)Cl)\N=N\c3ccc(cc3)C 4G-059 c1cc(ccc1C(F)(F)F)N/N=C(/C(=O)Nc2ccc(cc2)Cl)\N=N\c3ccc(cc3)C(F)(F)F 4G-061 c1ccc(cc1)S(=O)(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 4G-062 c1cc(cc(c1)C(=O)Nc2ccc(cc2)Cl)C#N 4G-301S CCCC/N=C(\c1cccnc1)/Nc2cccc(c2)C(F)(F)F 4G-302S Cc1c(snn1)S(=O)C(C)(C)C 4G-304S c1cc(ccc1NC(=O)c2ccc(nc2)Cl)Cl 4G-307S Cc1ncn(n1)c2ccc(cn2)C(=O)Oc3ccccc3 4G-308S Cc1c(snn1)S(=O)C(C)C 4G-310S c1cc(ccc1NC(=O)c2ccc(cc2F)F)Cl 4G-311S Cc1ncn(n1)c2ccc(cn2)C(=O)OCc3ccccc3 4G-312S Cc1ncn(n1)c2ccc(cn2)C(=O)OCC(F)(F)F 4G-313S COC(=O)c1ccc(cc1)c2[nH]ccn2 4G-314S Cc1c(snn1)SCCN(C)C 4G-317S COc1cccc2c1OCC(=C2)C#N 4G-318S COc1cccc2c1OCC(=C2)C(=O)O 4G-319S c1ccc2c(c1)C=C(CO2)C#N 4G-320S COC(=O)c1ccc(cc1)c2nc(cs2)c3cccnc3 4G-321S c1cc(ccc1c2[nH]ccn2)C(=O)O 4G-322S c1ccc2c(c1)C=C(CO2)C(=O)O 4G-323S CC(C)/N=C(\c1cccnc1)/Nc2cccc(c2)C(F)(F)F 4G-324S c1cc(cc(c1)C(F)(F)F)C(=N)Nc2ccc(cc2)Cl 4G-325S Cn1c(c(c(n1)C(F)(F)F)C=O)Sc2cccc(c2)C(F)(F)F 4G-327S Cn1c(c(c(n1)C(F)(F)F)CO)Sc2ccccc2 4G-329S COc1cccc2c1OCC(=C2)C(=O)OC 4G-332S COC(=O)C1=Cc2ccccc2OC1 4G-333S Cn1c(c(c(n1)C(F)(F)F)CO)Sc2ccc(cc2)Cl 4G-334S Cn1c(c(c(n1)C(F)(F)F)CO)Sc2cccc(c2)C(F)(F)F 4G-335S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2ccc(cc2)Cl)Sc3ccccc3 4G-336S CC(=O)OCc1c(nn(c1Sc2ccccc2)C)C(F)(F)F 4G-337S CC(=O)OCc1c(nn(c1Sc2cccc(c2)C(F)(F)F)C)C(F)(F)F 4G-339S C/N=C(/c1ccc(nc1)Cl)\Nc2ccc(cc2)Cl 4G-341S Cc1c(snn1)SCCN 4G-342S CC(C)OC(=O)C1=Cc2cccc(c2OC1)OC 4G-345S c1ccc(cc1)NC(=O)c2cccnc2 4G-346S C/N=C(\c1cccnc1)/Nc2ccccc2 4G-347S CC(C)/N=C(\c1cccnc1)/Nc2ccccc2 4G-348S Cc1ncn(n1)c2ccc(cn2)C(=O)OCC=C 4G-349S CC(C)OC(=O)c1ccc(nc1)n2cncn2 4G-351S Cn1c(c(c(n1)C(F)(F)F)C=O)Sc2ccc(cc2)Br 4G-352S Cn1c(c(c(n1)C(F)(F)F)CO)Sc2ccc(cc2)Br 4G-353S COc1cccc2c1OCC(=C2)C(=O)OCc3ccccc3 4G-354S COc1ccc(cc1)COC(=O)C2=Cc3cccc(c3OC2)OC 4G-357S CCCCOC(=O)C1=Cc2cccc(c2OC1)OC 4G-360S CCOC(=O)C1=Cc2cccc(c2OC1)OC 4G-361S CCCSc1c(nns1)C 4G-362S CCCCSc1c(nns1)C 4G-363S CCC(C)Sc1c(nns1)C 4G-364S COc1cccc2c1OCC(=C2)C(=O)OCc3cccnc3 4G-366S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Sc3ccc(cc3)Cl 4G-367S c1ccc(cc1)COC(=O)C2=Cc3ccccc3OC2 4G-368S COc1ccc(cc1)COC(=O)C2=Cc3ccccc3OC2 4G-369S CC(=O)OCc1c(nn(c1Sc2ccc(cc2)Br)C)C(F)(F)F 4G-372S CC(=O)OCc1c(nn(c1Sc2ccc(cc2)Cl)C)C(F)(F)F 4G-373S c1ccc2c(c1)C=C(CO2)C(=O)OCc3cccnc3 4G-374S c1cc2c(cc1Cl)C=C(CO2)C#N 4G-375S c1ccc(cc1)NC(=O)C2=Cc3ccccc3OC2 4G-376S CCCS(=O)(=O)c1c(nns1)C 4G-377S CCCCS(=O)(=O)c1c(nns1)C 4G-378S CCC(C)S(=O)(=O)c1c(nns1)C 4G-379S CCCS(=O)c1c(nns1)C 4G-380S CCCCS(=O)c1c(nns1)C 4G-381S CCC(C)S(=O)c1c(nns1)C 4G-382S CCCC/N=C(\c1cccnc1)/Nc2ccccc2 4G-383S c1ccc2c(c1)C=C(CO2)C(=O)Nc3cccc(c3)C(F)(F)F 4G-384S Cn1c(c(c(n1)C(F)(F)F)COC(=O)C(Cl)Cl)Sc2ccc(cc2)Br 4G-385S Cn1c(c(c(n1)C(F)(F)F)COC(=O)C(Cl)Cl)Sc2ccc(cc2)Cl 4G-386S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2ccc(cc2)Cl)Sc3ccc(cc3)Br 4G-387S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Sc3ccc(cc3)Br 4G-388S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Sc3ccccc3 4G-389S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Sc3cccc(c3)C(F)(F)F 4G-390S Cn1c(c(c(n1)C(F)(F)F)C=O)Sc2ccc(cc2)F 4G-391S Cn1c(c(c(n1)C(F)(F)F)CO)Sc2ccc(cc2)F 4G-392S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Sc3ccc(cc3)F 4G-393S Cn1c(c(c(n1)C(F)(F)F)C=O)Oc2ccc(cc2)Cl 4G-395S Cn1c(c(c(n1)C(F)(F)F)/C=N/c2ccc(cc2)F)Sc3ccc(cc3)F 4G-396S Cn1c(c(c(n1)C(F)(F)F)/C=N/c2ccc(cc2F)F)Sc3ccc(cc3)F 4G-397S Cc1c(sc(n1)c2ccccc2)C(=O)NN 4G-398S c1cc2c(cc1Cl)C=C(CO2)C(=O)O 4G-399S COc1cccc2c1OCC(=C2)C(=O)NCc3cccc(c3)C(F)(F)F 4G-401S COc1ccc2c(c1)C=C(CO2)C#N 4G-403S Cn1c(c(c(n1)C(F)(F)F)CO)Oc2ccc(cc2)Cl 4G-404S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Br 4G-405S c1ccc2c(c1)C=C(CO2)C(=O)NCc3cccc(c3)C(F)(F)F 4G-406S Cc1c(snn1)Sc2ccccc2C(=O)O 4G-409S c1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(cc3F)F 4G-411S c1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(cc3)F 4G-412S c1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(cc3)Cl 4G-413S COc1cccc2c1OCC(=C2)C(=O)Nc3cccc(c3)C(F)(F)F 4G-414S Cc1c(sc(n1)c2ccccc2)c3nnc(n3CC=C)S 4G-415S CCOC(=O)c1csc(n1)c2ccccc2 4G-416S C=CCn1c(nnc1S)c2csc(n2)c3ccccc3 4G-417S COC(=O)C1=Cc2cc(ccc2OC1)Cl 4G-418S CCOC(=O)C1=Cc2cc(ccc2OC1)Cl 4G-419S C=CCOC(=O)C1=Cc2cc(ccc2OC1)Cl 4G-421S c1cc(sc1)S(=O)(=O)c2cnns2 4G-422S Cn1c(c(c(n1)C(F)(F)F)CNc2ccc(cc2)F)Sc3ccc(cc3)F 4G-423S c1cc(cc(c1)S(=O)c2cnns2)C(F)(F)F 4G-424S c1c(snn1)SC2CCCCC2 4G-425S c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)CON.Cl 4G-901 CCOC(=O)NC(=O)C(=CNNc1c(cc(cn1)C(F)(F)F)Cl)C(=O)NC(=O)OCC 4G-903 c1cc(ccc1N2C(=O)C=CC2=O)Cl 4G-904 c1cn(c(=O)nc1N)c2c(cc(cn2)C(F)(F)F)Cl 4G-905 c1cc(cc(c1)N2C(=O)C=CC2=O)C(F)(F)F 4G-906 COc1ccc(cc1)C2C3C(C(=O)N(C3=O)c4ccccc4)C(N2)(Cc5ccccc5)C(=O)OC 4G-909 COC(=O)C1(C2C(C(=O)N(C2=O)c3cccc(c3)C(F)(F)F)ON1)C(=O)OC 4G-910 COC(=O)C1(C2C(C(=O)N(C2=O)c3ccc(cc3)Cl)ON1)C(=O)OC 4G-911 c1ccc(cc1)CSc2c3nncn3c4ccccc4n2 4G-912 c1ccc2c(c1)nc(c3n2cnn3)Sc4ccccc4Cl 4G-913 COc1ccc(cc1)Sc2c3nncn3c4ccccc4n2 4G-914 c1ccc2c(c1)nc(c3n2cnn3)N4CCOCC4 4G-915 COc1ccc(cc1)C2C3C(C(=O)N(C3=O)c4ccc(cc4)Cl)C(N2)(Cc5ccccc5)C(=O)OC 4G-916 COc1ccc(cc1)C2C3C(C(=O)N(C3=O)c4cccc(c4)C(F)(F)F)C(N2)(Cc5ccccc5)C(=O)OC 4G-917 COC(=O)c1ccccc1N2C(=O)C=CC2=O 4G-920 C=CCSc1c2nncn2c3ccccc3n1 4G-922 c1cc(ccc1N2C(=O)[C@@H]3[C@H]4CCCCN4O[C@@H]3C2=O)Cl 4G-923 c1cc(cc(c1)OCCN(CCNc2c(cc(cn2)C(F)(F)F)Cl)Cc3ccc(cc3)Cl)C(F)(F)F 4G-924 COc1ccc(cc1)C2C3C(C(=O)N(C3=O)c4ccccc4C(=O)OC)C(N2)(Cc5ccccc5)C(=O)OC 4G-925 c1cn(c(=O)nc1Nc2c(cc(cn2)C(F)(F)F)Cl)c3c(cc(cn3)C(F)(F)F)Cl 4G-927 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 4G-930 c1cc(cc(c1)N2C(=O)[C@@H]3[C@H]4CCCCN4O[C@@H]3C2=O)C(F)(F)F 4G-931 Cc1ccc(cc1)S(=O)(=O)Nc2ccn(c(=O)n2)c3c(cc(cn3)C(F)(F)F)Cl 4G-932 c1ccc2c(c1)C(C(=O)N2)c3c(cc(cn3)C(F)(F)F)Cl 4G-934 c1cc(c(c(c1)Cl)C(=O)Nc2ccn(c(=O)n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 4G-935 c1ccc2c(c1)nc(c3n2c(nn3)C(F)(F)F)Sc4ccc(cc4)Cl 4G-937 c1ccc(cc1)CSc2c3nnc(n3c4ccccc4n2)C(F)(F)F 4G-938 Cc1cc(nc(n1)NC(=O)CC(=O)C)C 4G-940 CC(=O)CC(=O)Nc1ccc(cc1)F 4G-941 c1cc(cc(c1)Cl)NCc2c(snn2)Cl 4G-942 c1ccc2c(c1)nc(c3n2c(nn3)C(F)(F)F)Sc4ccccn4 4G-943 c1ccc(cc1)Sc2c3nnc(n3c4ccccc4n2)C(F)(F)F 4G-944 COc1ccc(cc1)Sc2c3nnc(n3c4ccccc4n2)C(F)(F)F 4G-945 Cc1cc(nc(c1)NC(=O)CC(=O)C)C 4G-947 C/C(=C/C(=O)Nc1ccc(cc1)Cl)/N2CCCC2 4G-948 CN(C)/C=C/C(=O)c1cccc(c1)Cl 4G-949 CCOC(=O)c1c(con1)C(=O)c2ccc(cc2)F 4G-950 CN(C)/C=C/C(=O)c1cccnc1 4G-951 CN(C)/C=C/C(=O)c1ccc(cc1)[N+](=O)[O-] 4G-952 C/C(=C/C(=O)Nc1cccc(c1)C(F)(F)F)/N2CCCC2 4G-953 Cc1cc(nc(n1)NC(=O)/C=C(\C)/N2CCCC2)C 4G-954 C/C(=C\C(=O)Nc1ccc(cc1)F)/N2CCCC2 4G-955 Cc1cc(nc(c1)NC(=O)/C=C(\C)/N2CCCC2)C 4G-956 C1COCCN1Cc2c(snn2)Cl 4G-957 CCOC(=O)c1c(con1)C(=O)c2ccc(cc2)[N+](=O)[O-] 4G-958 COC(=O)/C=C/COc1ccc2ccccc2c1C=O 4G-999 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)N 4H-004 c1ccc(cc1)S(=O)(=O)/N=C(/NNc2c(cc(cn2)C(F)(F)F)Cl)\N3CCOCC3 4H-005 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)OC3=CC(=O)CCC3 4H-006 COc1ccc(cc1)NC(=S)NC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 4H-007 c1ccc(c(c1)C(=O)Nc2ccccc2Sc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 4H-008 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NC(=S)Nc3ccc(c(c3)Cl)Oc4ccc(cn4)C(F)(F)F 4H-011 c1ccc(cc1)CN/C(=N\S(=O)(=O)c2ccccc2)/NNc3c(cc(cn3)C(F)(F)F)Cl 4H-012 CN(C)/C=N/C(=O)CCC(c1c(cc(cn1)C(F)(F)F)Cl)S(=O)(=O)c2ccccc2 4H-013 c1ccc(cc1)S(=O)(=O)/N=C(\NN)/NNc2c(cc(cn2)C(F)(F)F)Cl 4H-014 c1ccc(cc1)S(=O)(=O)C(CCc2nc[nH]n2)c3c(cc(cn3)C(F)(F)F)Cl 4H-016 c1ccc(cc1)c2csc(n2)CCC(c3c(cc(cn3)C(F)(F)F)Cl)S(=O)(=O)c4ccccc4 4H-017 CC(=O)C(=O)N(C)c1ccccc1 4H-018 c1ccc(c(c1)C#N)C(C#N)c2ccc(cc2)F 4H-019 c1ccc2c(c1)c(c(nc2Br)N)c3ccc(cc3)F 4H-020 Cn1c(cnc1S)C(=O)OC 4H-021 c1ccc(cc1)c2c3ccccc3c(nc2N)Br 4H-022 c1ccc(cc1)CO/N=C\C([N+](=O)[O-])S(=O)(=O)c2ccccc2 4H-024 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C/Nc4cccc(c4)C(F)(F)F)F 4H-025 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C/Nc4ccccc4[N+](=O)[O-])F 4H-026 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C/Nc4cccc(c4)C#N)F 4H-027 Cc1ccc(cc1)CSc2ncc(n2C)C(=O)OC 4H-028 CCOC1=NN(C(=O)C1)c2c(cc(cn2)C(F)(F)F)Cl 4H-029 c1ccc(cc1)C2CC(=O)c3c2cccc3N4CCN(CC4)c5ccccc5 4H-030 c1cc(ccc1CSc2ncc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 4H-032 c1c(cnc(c1Cl)c2cnc(nc2)[S-])C(F)(F)F.[K+] 4H-033 CCOC\1=NN(C(=O)/C1=C/N(C)C)c2c(cc(cn2)C(F)(F)F)Cl 4H-034 c1ccc(cc1)C2CC(=O)c3c2cccc3N4CCN(CC4)c5ccc(cc5)F 4H-035 COc1cccc(c1)C(C#N)N2CCOCC2 4H-036 COc1ccc(cc1)c2cnn3c2ncc(c3)c4c(cc(cn4)C(F)(F)F)Cl 4H-037 c1ccc(cc1)/C=C/c2ccnc(n2)Sc3c(cccn3)[N+](=O)[O-] 4H-039 c1ccc(c(c1)CSc2ncc(cn2)C#N)[N+](=O)[O-] 4H-040 c1ccc(cc1)C(=O)/C=C/NCC#N 4H-041 c1c(cnc(c1Cl)c2cnc(nc2)Cn3cncn3)C(F)(F)F 4H-042 c1cc(cc(c1)C(F)(F)F)/C=C/c2c(cc(cn2)C(F)(F)F)Cl 4H-043 CSc1nc2ncc(cn2n1)c3c(cc(cn3)C(F)(F)F)Cl 4H-045 CC(C(=O)C)Sc1ncc(cn1)C#N 4H-047 c1ccc2c(c1)CCNC2CC(=O)O 4H-048 c1cc(sc1)/C=C/c2c(cc(cn2)C(F)(F)F)Cl 4H-049 COc1cccc(c1)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 4H-051 c1ccc(cc1)S(=O)(=O)C(C2c3ccccc3CCN2)[N+](=O)[O-] 4H-055 c1ccc(cc1)Cc2cccc(n2)Cl 4H-100 COc1ccc(cc1)N2C(=O)CS(=O)CC2=O 4H-301S Cc1ccc(cc1)N2C(=O)CS(=O)CC2=O 4H-302S c1cc(c(cc1N2C(=O)CS(=O)CC2=O)Cl)Cl 4H-309S c1cc(cc(c1)NC(=O)CSCC(=O)O)C(F)(F)F 4H-311S c1cc(cc(c1)N2C(=O)CSCC2=O)C(F)(F)F 4H-312S c1cc(c(c(c1)Cl)S(=O)c2cnns2)Cl 4H-313S COc1ccc(cc1)S(=O)(=O)c2cnns2 4H-314S c1cc(ccc1Oc2cnns2)F 4H-315S c1cc(cc(c1)Oc2cnns2)C(F)(F)F 4H-320S c1ccc2c(c1)c(ccc2Cl)Oc3cnns3 4H-322S c1cc(cc(c1)Cl)NC(=O)CSCC(=O)O 4H-323S c1cc(cc(c1)Cl)N2C(=O)CSCC2=O 4H-325S c1cc(c(c(c1)Cl)Cl)Oc2cnns2 4H-326S c1cc(c(cc1Cl)Cl)Oc2cnns2 4H-327S c1cc(ccc1Sc2c(nns2)c3ccc(c(c3)Cl)Cl)Cl 4H-329S c1cc(cc(c1)Sc2c(nns2)c3ccc(c(c3)Cl)Cl)C(F)(F)F 4H-330S c1ccc(c(c1)Sc2c(nns2)c3ccc(c(c3)Cl)Cl)Cl 4H-331S COC(=O)CSc1c(nns1)c2ccc(c(c2)Cl)Cl 4H-332S c1ccc(cc1)Oc2cnns2 4H-335S c1cc(cc(c1)Cl)N2C(=O)CS(=O)CC2=O 4H-337S CSc1c(nns1)c2ccc(c(c2)Cl)Cl 4H-338S c1cc(ccc1C(F)(F)F)NC(=O)CSCC(=O)O 4H-339S c1ccc(c(c1)NC(=O)CSCC(=O)O)Cl 4H-342S Cc1ccccc1NC(=O)CSCC(=O)O 4H-343S c1ccc(c(c1)N2C(=O)CSCC2=O)Cl 4H-346S c1c(cc(cc1Cl)Cl)Oc2cnns2 4H-347S c1cc(c(cc1Oc2cnns2)Cl)Cl 4H-348S c1cc(cc(c1)Oc2cnns2)[N+](=O)[O-] 4H-349S COC(=O)c1ccc(cc1)Oc2cnns2 4H-350S c1c(c(cc(c1Cl)Cl)Cl)Oc2cnns2 4H-351S c1cc(ccc1C(F)(F)F)N2C(=O)CSCC2=O 4H-352S Cc1ccccc1N2C(=O)CSCC2=O 4H-353S CN(C)c1nc2cc(c(cc2c(=O)o1)OC)OC 4H-356S c1cc(ccc1CNC(=O)CSCC(=O)O)Cl 4H-357S c1cc(ccc1CN2C(=O)CSCC2=O)Cl 4H-358S COc1ccc(cc1OC)N2C(=O)CS(=O)CC2=O 4H-359S Cc1cc(nc(n1)C)OC(=O)c2ccc(cc2Cl)Cl 4H-360S Cc1cc(nc(c1C#N)OC(=O)c2c(cc(cc2Cl)Cl)Cl)C 4H-361S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3ccc(cc3Cl)Cl)C 4H-362S Cc1cc(nc(n1)OC(=O)c2ccc(cc2Cl)Cl)C 4H-363S c1cc(c(cc1Cl)C(F)(F)F)NC(=O)CSCC(=O)O 4H-364S c1cc(c(c(c1)Cl)NC(=O)CSCC(=O)O)Cl 4H-365S c1cc(ccc1CN2C(=O)CS(=O)(=O)CC2=O)Cl 4H-367S c1cc(cc(c1)NC(=O)CS(=O)(=O)CC(=O)O)C(F)(F)F 4H-368S Cc1cc(nc(n1)C)OC(=O)c2c(cc(cc2Cl)Cl)Cl 4H-369S Cc1cc(nc(n1)OC(=O)c2c(cc(cc2Cl)Cl)Cl)C 4H-370S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3c(cc(cc3Cl)Cl)Cl)C 4H-371S c1cc(c(cc1Cl)C(F)(F)F)N2C(=O)CSCC2=O 4H-372S c1cc(c(c(c1)Cl)N2C(=O)CSCC2=O)Cl 4H-373S c1ccc(cc1)NC(=O)CS(=O)(=O)CC(=O)O 4H-374S Cc1cc(nc(c1C#N)OC(=O)c2ccc(cc2Cl)S(=O)(=O)C)C 4H-375S Cc1cc(nc(n1)C)OC(=O)c2c(cccc2Cl)Cl 4H-376S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3c(cccc3Cl)Cl)C 4H-377S c1ccc(cc1)N2C(=O)CS(=O)(=O)CC2=O 4H-378S c1cc(c(cc1Cl)Cl)CNC(=O)CSCC(=O)O 4H-382S c1ccc(c(c1)N2C(=O)CS(=O)CC2=O)Cl 4H-386S Cc1cc(nc(c1C#N)OC(=O)c2cc(c(cc2Cl)F)F)C 4H-388S COc1ccc(cc1)CNC(=O)CSCC(=O)O 4H-391S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3c(cccc3F)F)C 4H-392S Cc1ccc(cc1)CNC(=O)CSCC(=O)O 4H-393S Cc1ccccc1N2C(=O)CS(=O)CC2=O 4H-394S Cn1c(nnc1SC)CNS(=O)(=O)c2ccc(cc2)Cl 4H-401S Cn1c(nnc1SCc2ccc(cc2)Cl)CNS(=O)(=O)c3ccc(cc3)Cl 4H-402S Cn1c(nnc1SCC=C)CNS(=O)(=O)c2ccc(cc2)Cl 4H-403S Cn1c(nnc1SCc2cccc(c2)C(F)(F)F)CNS(=O)(=O)c3ccc(cc3)Cl 4H-404S Cn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])CNS(=O)(=O)c3ccc(cc3)Cl 4H-405S Cn1c(nnc1SCC(=O)OC)CNS(=O)(=O)c2ccc(cc2)Cl 4H-406S c1cc(ccc1F)S(=O)(=O)NCC(=O)NN 4H-410S Cn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)Br 4H-413S Cn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)F 4H-414S c1ccc(cc1)SCC(=NOCc2ccc(cc2Cl)Cl)CSc3ccccc3 4H-418S c1ccc(cc1)SCC(=NOCc2ccc(c(c2)Cl)Cl)CSc3ccccc3 4H-419S c1ccc(cc1)SCC(=NOCc2ccc(cc2)Cl)CSc3ccccc3 4H-420S c1ccc(cc1)SCC(=NO)CSc2ccccc2 4H-421S Cn1c(nnc1SC)CNS(=O)(=O)c2ccc(cc2)Br 4H-422S Cn1c(nnc1SCC#C)CNS(=O)(=O)c2ccc(cc2)Br 4H-423S CC(=C)CSc1nnc(n1C)CNS(=O)(=O)c2ccc(cc2)Br 4H-424S Cn1c(nnc1SCc2ccc(cc2)Br)CNS(=O)(=O)c3ccc(cc3)Br 4H-425S Cn1c(nnc1SCc2ccc(c(c2)Cl)Cl)CNS(=O)(=O)c3ccc(cc3)Br 4H-426S Cn1c(nnc1SCc2cccc(c2)Cl)CNS(=O)(=O)c3ccc(cc3)Br 4H-427S Cn1c(nnc1SCc2ccc(cc2)C(F)(F)F)CNS(=O)(=O)c3ccc(cc3)Br 4H-428S c1cc(ccc1SCC(=NO)CSc2ccc(cc2)Br)Br 4H-429S Cc1ccc(cc1)SCC(=NO)CSc2ccc(cc2)C 4H-430S c1ccc(cc1)N2CCN(CC2)CC(CSc3ccc(cc3)Cl)O 4H-433S Cc1ccc(cc1)SCC(CN2CCN(CC2)c3ccccc3)O 4H-434S c1ccc(cc1)N2CCN(CC2)CC(CSc3cccc(c3)C(F)(F)F)O 4H-435S c1ccc(cc1)N2CCN(CC2)CC(CSc3cccc(c3)Cl)O 4H-436S c1ccc(cc1)N2CCN(CC2)CC(CSc3ccccc3Cl)O 4H-437S Cc1cccc(c1)SCC(CN2CCN(CC2)c3ccccc3)O 4H-438S c1ccc(cc1)N2CCN(CC2)CC(CSc3ccc(cc3)F)O 4H-439S c1ccc(cc1)N2CCN(CC2)CC(CSc3ccc(cc3)Br)O 4H-440S c1cc(ccc1N2CCN(CC2)CC(CSc3ccc(cc3)Cl)O)F 4H-443S c1cc(ccc1N2CCN(CC2)CC(CSc3ccc(cc3)F)O)F 4H-444S CCC(C)Sc1nnc(n1C)CNS(=O)(=O)c2ccc(cc2)F 4H-445S Cn1c(nnc1SCC(=O)OC)CNS(=O)(=O)c2ccc(cc2)Br 4H-446S CC(C)(C)c1ccc(cc1)CSc2nnc(n2C)CNS(=O)(=O)c3ccc(cc3)F 4H-447S Cn1c(nnc1SCc2ccc(cc2)OC)CNS(=O)(=O)c3ccc(cc3)F 4H-448S Cn1c(nnc1SCc2cccc(c2)F)CNS(=O)(=O)c3ccc(cc3)F 4H-449S CCn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)Cl 4H-452S C=CCn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)Cl 4H-453S c1cc(cc(c1)Cl)SCC(CN2CCN(CC2)c3ccc(cc3)F)O 4H-454S Cc1ccc(cc1)SCC(CN2CCN(CC2)c3ccc(cc3)F)O 4H-455S c1ccc(c(c1)N2CCN(CC2)CC(CCl)O)F 4H-456S Cc1ccc(cc1)SCC(CN2CCN(CC2)c3ccccc3F)O 4H-457S c1ccc(c(c1)N2CCN(CC2)CC(CSc3ccc(cc3)Cl)O)F 4H-458S c1ccc(c(c1)N2CCN(CC2)CC(CSc3c(cccc3Cl)Cl)O)F 4H-459S c1ccc(cc1)SCC(CN2CCN(CC2)c3ccccc3F)O 4H-460S c1ccc(c(c1)N2CCN(CC2)CC(CSc3ccc(cc3)F)O)F 4H-461S c1ccc(c(c1)N2CCN(CC2)CC(CSc3cccc(c3)Cl)O)F 4H-462S c1ccc(c(c1)N2CCN(CC2)CC(CSc3ccccc3Cl)O)F 4H-463S c1cc(ccc1SCC(=NO)CSc2ccc(cc2)Cl)Cl 4H-464S Cc1ccc(cc1)S(=O)(=O)NCc2nnc(n2C)S 4H-465S CCn1c(nnc1SC)CNS(=O)(=O)c2ccc(cc2)Cl 4H-469S CCn1c(nnc1SCc2cccc(c2)OC)CNS(=O)(=O)c3ccc(cc3)Cl 4H-470S CCn1c(nnc1SCc2ccc(cc2)F)CNS(=O)(=O)c3ccc(cc3)Cl 4H-471S CCn1c(nnc1SCc2ccc(cc2)Cl)CNS(=O)(=O)c3ccc(cc3)Cl 4H-472S CCn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])CNS(=O)(=O)c3ccc(cc3)Cl 4H-473S c1ccc(c(c1)N2CCN(CC2)CC(CSc3cccc(c3)C(F)(F)F)O)F 4H-475S c1ccc(cc1)SCC(CN2CCN(CC2)c3ccc(cc3)F)O 4H-476S c1cc(ccc1N2CCN(CC2)CC(CSc3ccc(cc3)Br)O)F 4H-477S c1cc(ccc1N2CCN(CC2)CC(CSc3ccc(c(c3)Cl)Cl)O)F 4H-478S c1cc(c(c(c1)Cl)SCC(CN2CCN(CC2)c3ccc(cc3)F)O)Cl 4H-479S c1ccc(c(c1)SCC(CN2CCN(CC2)c3ccc(cc3)F)O)Cl 4H-480S CCCCSc1nnc(n1CC)CNS(=O)(=O)c2ccc(cc2)Cl 4H-481S CCn1c(nnc1SCC=C)CNS(=O)(=O)c2ccc(cc2)Cl 4H-482S CCn1c(nnc1SCc2cccc(c2)C(F)(F)F)CNS(=O)(=O)c3ccc(cc3)Cl 4H-483S CCn1c(nnc1SCc2c(cccc2Cl)F)CNS(=O)(=O)c3ccc(cc3)Cl 4H-484S c1cc(cc(c1)Cl)N2CCN(CC2)CC(CSc3ccc(cc3)Cl)O 4H-486S Cc1ccc(cc1)SCC(CN2CCN(CC2)c3cccc(c3)Cl)O 4H-488S c1cc(cc(c1)Cl)N2CCN(CC2)CC(CSc3ccc(cc3)F)O 4H-489S c1cc(cc(c1)SCC(CN2CCN(CC2)c3cccc(c3)Cl)O)C(F)(F)F 4H-491S c1ccc(c(c1)SCC(CN2CCN(CC2)c3cccc(c3)Cl)O)Cl 4H-492S c1cc(cc(c1)Cl)N2CCN(CC2)CC(CSc3cccc(c3)Cl)O 4H-493S c1cc(cc(c1)N2CCN(CC2)CC(CCl)O)C(F)(F)F 4H-494S Cc1ccc(cc1)SCC(CN2CCN(CC2)c3cccc(c3)C(F)(F)F)O 4H-495S c1cc(cc(c1)N2CCN(CC2)CC(CSc3ccc(cc3)Cl)O)C(F)(F)F 4H-496S c1ccc(cc1)SCC(=NOC(=O)c2ccc(cc2)Cl)CSc3ccccc3 4H-497S c1cc(cc(c1)N2CCN(CC2)CC(CSc3ccc(cc3)F)O)C(F)(F)F 4H-498S c1cc(cc(c1)Cl)N2CCN(CC2)CC(CSc3ccc(cc3)Br)O 4H-499S Cc1cccc(c1)SCC(CN2CCN(CC2)c3ccccc3F)O 4H-500S CSc1nnc(n1CC=C)CNS(=O)(=O)c2ccc(cc2)Cl 4H-501S CC(C)(C)c1ccc(cc1)CSc2nnc(n2CC=C)CNS(=O)(=O)c3ccc(cc3)Cl 4H-502S C=CCn1c(nnc1SCc2c(cccc2Cl)Cl)CNS(=O)(=O)c3ccc(cc3)Cl 4H-503S C=CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)CNS(=O)(=O)c3ccc(cc3)Cl 4H-504S C=CCn1c(nnc1SCc2ccc(cc2)C(F)(F)F)CNS(=O)(=O)c3ccc(cc3)Cl 4H-505S COc1cccc(c1)CSc2nnc(n2CC=C)CNS(=O)(=O)c3ccc(cc3)Cl 4H-506S C=CCn1c(nnc1SCc2ccc(cc2)F)CNS(=O)(=O)c3ccc(cc3)Cl 4H-507S C=CCn1c(nnc1SCc2ccccc2)CNS(=O)(=O)c3ccc(cc3)Cl 4H-508S C=CCn1c(nnc1SCc2ccc(cc2)Br)CNS(=O)(=O)c3ccc(cc3)Cl 4H-509S C=CCn1c(nnc1SCC=C)CNS(=O)(=O)c2ccc(cc2)Cl 4H-510S C=CCn1c(nnc1SCC#C)CNS(=O)(=O)c2ccc(cc2)Cl 4H-511S c1cc(cc(c1)SCC(CN2CCN(CC2)c3ccc(cc3)F)O)C(F)(F)F 4H-845S c1cc(ccc1N2CCN(CC2)C(=N)CC#N)F 4H-900 CNC(=S)/C(=C(\N)/N1CCOCC1)/C#N 4H-901 c1cc(ccc1C(=O)OCC2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl 4H-902 c1ccc(cc1)SC2CC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 4H-903 COC(=O)C1CC(CN1C(=O)c2ccc(cc2)F)O 4H-904 COc1ccc(cc1)SC2CC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 4H-905 CNC(=S)/C(=C(\N)/N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)/C#N 4H-906 COC(=O)C1CC(CN1C(=O)NC2CCCCC2)O 4H-907 c1cc(ccc1C(=O)N2CC(=O)CC2C(=O)O)F 4H-908 CNC(=S)/C(=C(\N)/N1CCN(CC1)c2ccc(cc2)F)/C#N 4H-909 Cn1c(cnc1S)CO 4H-910 c1ccc(cc1)N2C(=O)C3CC(=O)CN3C2=O 4H-911 Cn1c(cnc1SCc2ccc(cc2)F)CO 4H-912 CNc1c(c(ns1)N2CCOCC2)C#N 4H-913 Cn1c(cnc1SCc2ccc(cc2)F)COC(=O)c3ccco3 4H-914 c1cc(sc1)S(=O)(=O)N2CC(=O)CC2C(=O)O 4H-915 Cn1c(cnc1SCc2c(cccc2Cl)Cl)CO 4H-916 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)CO 4H-918 c1cc(cc(c1)SC2CC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 4H-919 Cn1c(cnc1SCc2c(cccc2Cl)Cl)COC(=O)Nc3ccc(cc3)[N+](=O)[O-] 4H-920 Cn1c(nnc1S)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 4H-921 Cn1c(cnc1SCc2c(snn2)Cl)CO 4H-922 Cn1c(cnc1SCc2c(cccc2Cl)Cl)CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 4H-923 Cn1c(cnc1SCC(=O)c2ccc(cc2)Cl)CO 4H-924 C/[N+](=C\C([N+](=O)[O-])S(=O)(=O)c1ccccc1)/[O-] 4H-926 CCOC(=O)C1=NOC2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F 4H-929 COc1ccc(cc1OC)CCn2c(cnc2S)CO 4H-931 CNC(=S)/C(=C(\N)/N1CCC(CC1)C(=O)OC)/C#N 4H-932 c1ccc2c(c1)C(=O)N(C2=O)OCC3CO3 4H-933 CNc1c(c(ns1)N2CCC(CC2)C(=O)OC)C#N 4H-935 COC(=O)c1ccccc1C(=O)N2CC(CO2)O 4H-936 C1C(CON1)O.Cl 4H-937 COc1ccc(cc1OC)CCn2c(cnc2Sc3c(cc(cn3)C(F)(F)F)Cl)CO 4H-938 c1cc(ccc1C2CC(=O)C(=CN3CC(CO3)O)C(=O)C2)Cl 4H-939 CCOC1CC(N(O1)c2ccccc2)c3ccccc3 4H-940 COC(=O)C1C/C(=N/OCc2cccc(c2)C(F)(F)F)/CN1S(=O)(=O)c3cccs3 4H-943 c1cc(ccc1C(=O)/C=C\N2CC(CO2)O)[N+](=O)[O-] 4H-944 CC(=O)C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 4H-945 Cn1c(cnc1SCCOc2cccc(c2)C(F)(F)F)CO 4H-946 Cn1c(cnc1SCCOc2ccc(cc2)OC)CO 4H-947 CN1[C@H]2c3c4ccccc4ccc3OC[C@H]2[C@@H](O1)C(=O)OC 4H-948 COC(=O)C1CC(=O)CN1S(=O)(=O)c2cccs2 4H-949 Cn1c(cnc1SCC(=O)c2ccc(cc2)Br)CO 4H-951 CN(C)/C=C/C(=O)C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 4H-952 Cn1c(cnc1SCC(=O)c2ccc(cc2)F)CO 4H-953 COc1ccc(cc1)N/C=C/C(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 4H-954 C/[N+](=C/c1c2ccccc2ccc1OCc3ccccc3)/[O-] 4H-955 CC1(NC(=O)N(N1)c2ccccc2)C3=NOC(C3)CNc4c(cc(cn4)C(F)(F)F)Cl 4H-957 c1ccc(cc1)COc2ccc3ccccc3c2C=O 4H-959 COc1ccc(cc1)N2C(=O)CC(=N2)C(F)(F)F 4H-961 C/[N+](=C/c1ccccc1OCc2ccccc2)/[O-] 4H-962 COC(=O)C1CC(CN1C(=O)c2ccccc2)O 4H-964 COC(=O)C1CC(CN1C(=O)Nc2cccc(c2)C(F)(F)F)O 4H-965 COC(=O)C1CC(CN1C(=O)Nc2ccc(c(c2)Cl)Cl)O 4H-966 Cc1c(c(n(n1)C)Cl)S(=O)(=O)NNc2c(cc(cn2)C(F)(F)F)Cl 4J-001 COC(=O)c1cnc(c2c1cccc2)C(C#N)c3ccccn3 4J-002 Cn1cccc1C(C#N)c2c3ccccc3c(cn2)C(=O)OC 4J-003 CCOC(=O)CSc1c(cc(cn1)C(F)(F)F)Cl 4J-004 COC(=O)C1CCC(=O)c2n1ccc2 4J-005 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Cl 4J-006 c1c(cnc(c1Cl)N/N=C(/CCC(=O)O)\C(=O)O)C(F)(F)F 4J-007 c1ccc2c(c1)ccc3c2C4CCC(O3)O4 4J-008 CCOC(=O)NOC 4J-009 c1c(cnc(c1Cl)SCC(=O)O)C(F)(F)F 4J-010 CCOC(=O)CC(c1c(cc(cn1)C(F)(F)F)Cl)(C(=O)OCC)C(=O)OCC 4J-011 CCOC(=O)N(c1c(cc(cn1)C(F)(F)F)Cl)OC 4J-012 CCOC(=O)/C(=C\N(C)C)/Sc1c(cc(cn1)C(F)(F)F)Cl 4J-013 c1c(cnc(c1Cl)SCC(=O)NN)C(F)(F)F 4J-014 c1cc(ccc1C(=O)c2ccc(s2)CC#N)Cl 4J-016 C(=O)c1c(c([nH]c1Cl)C=O)Cl 4J-018 c1cc(nc2c1scc2C=O)Cl 4J-019 c1ccc2c(c1)ccc3c2C4CCC(N4Nc5ccc(cc5[N+](=O)[O-])[N+](=O)[O-])O3 4J-020 CCOC(=O)/C(=C\Nc1ccc(cc1)OC)/Sc2c(cc(cn2)C(F)(F)F)Cl 4J-021 c1c(cnc(c1Cl)C(CC(=O)O)C(=O)O)C(F)(F)F 4J-022 c1c(cnc(c1Cl)CCC(=O)O)C(F)(F)F 4J-023 c1cnc(nc1)NC(=O)CCCCl 4J-024 c1ccc2c(c1)OS(=O)(=O)O2 4J-025 c1cnc(nc1)N2CCCC2=O 4J-026 c1ccc(cc1)CNS(=O)(=O)Oc2ccccc2O 4J-027 c1ccc(c(c1)O)OS(=O)(=O)NCc2cccnc2 4J-028 Cc1c([n+](c2ccccc2[n+]1[O-])[O-])C(=O)C 4J-029 CN(C)/C=C\1/CCN(C1=O)c2ncccn2 4J-030 CC(=O)c1c([n+](c2ccccc2[n+]1[O-])[O-])/C=C/N(C)C 4J-031 CCOC(=O)CSC(C)(C)CNc1c(cc(cn1)C(F)(F)F)Cl 4J-032 CC1([N+](=c2ccccc2=[N+]1[O-])[O-])C 4J-034 Cc1c(c(n(n1)C)C(C#N)c2cccs2)S(=O)(=O)N(C)C 4J-036 Cc1c(c(n(n1)C)Cl)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 4J-037 CN(C)/C=N/NC(=O)CSc1c(cc(cn1)C(F)(F)F)Cl 4J-038 CC(C(=O)C)SC(C)(C)CNc1c(cc(cn1)C(F)(F)F)Cl 4J-039 CC(C)(Cn1cccc1)SCc2ccc(cc2)Cl 4J-040 Cc1n(c2ccccc2[n+]1[O-])O 4J-041 CC(C)(CNc1c(cc(cn1)C(F)(F)F)Cl)SCC#N 4J-046 c1cc(cnc1)c2nnc(o2)Sc3c(cc(cn3)C(F)(F)F)Cl 4J-050 CO/N=C/C(=C\Nc1ccc(cc1)Cl)/[N+](=O)[O-] 4J-051 CO/N=C/C(=C/Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl)/[N+](=O)[O-] 4J-052 CO/N=C/C(=C\Nc1ccc(cc1)C(F)(F)F)/[N+](=O)[O-] 4J-053 CCOC(=O)c1ccc(cc1)N/C=C(\C=N\OC)/[N+](=O)[O-] 4J-054 CN(C)S(=O)(=O)c1ccc(cc1)N/C=C(\C=N\OC)/[N+](=O)[O-] 4J-055 CCOC(=O)C(/C=N/OC)Sc1c(cc(cn1)C(F)(F)F)Cl 4J-056 c1c(cnc(c1Cl)SC2C=NNC2=O)C(F)(F)F 4J-057 Cc1ccc(cc1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)F)C)C 4J-301S CC(C)C(C(=O)O)NC(=O)c1ccccc1Cl 4J-305S CC(C)C(C(=O)O)NC(=O)c1cccc(c1)Cl 4J-306S COc1cnc(nc1Cl)SCc2ccc(cc2)Cl 4J-307S COc1cnc(nc1OC)SCc2ccc(cc2)Cl 4J-308S Cc1ccc(cc1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(ccc4Cl)Cl)C)C 4J-311S CC(C)C(c1[nH]c2ccccc2n1)NC(=O)c3cccc(c3)Cl 4J-312S Cc1ccc2c(c1)nc([nH]2)C(C(C)C)NC(=O)c3cccc(c3)Cl 4J-313S Cc1ccc(cc1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(cc(c4)Cl)Cl)C)C 4J-314S Cc1cc2c(c(c1C)[N+](=O)[O-])ncn2C(C)C 4J-316S Cc1cc2c(c(c1C)N)ncn2C(C)C 4J-317S Cc1cccc(c1)Cn2cnc3c2cc(c(c3N(=O)=O)C)C 4J-318S Cc1cccc(c1)Cn2cnc3c2cc(c(c3N)C)C 4J-319S COc1cnc(nc1Sc2ccc(cc2)Cl)SCc3ccc(cc3)Cl 4J-320S COc1cnc(nc1Sc2ccccc2)SCc3ccc(cc3)Cl 4J-321S COc1cnc(nc1Oc2cccc(c2)C(F)(F)F)SCc3ccc(cc3)Cl 4J-322S COc1cnc(nc1Oc2ccccc2)SCc3ccc(cc3)Cl 4J-323S COc1cnc(nc1Oc2ccc(cc2)Cl)SCc3ccc(cc3)Cl 4J-324S COc1cnc(nc1Oc2ccccc2Cl)SCc3ccc(cc3)Cl 4J-325S Cc1ccc(cc1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cccc(c4)C(F)(F)F)C)C 4J-327S COc1ccc(cc1)Sc2c(cnc(n2)SCc3ccc(cc3)Cl)OC 4J-328S COc1cnc(nc1Sc2cccc(c2)C(F)(F)F)SCc3ccc(cc3)Cl 4J-329S COc1cnc(nc1Sc2ccccc2Cl)SCc3ccc(cc3)Cl 4J-330S CC(C)C(c1[nH]c2ccccc2n1)NC(=O)c3ccccc3Cl 4J-331S Cc1cc2c(cc1C)nc([nH]2)C(C(C)C)NC(=O)c3ccccc3Cl 4J-332S Cc1ccc(cc1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)C)C)C 4J-333S Cc1ccc(cc1)S(=O)(=O)Nc2c(c(cc3c2ncn3C(C)C)C)C 4J-334S COc1cnc(nc1Oc2cc(cc(c2)Cl)Cl)SCc3ccc(cc3)Cl 4J-335S COc1cnc(nc1SCc2ccc(cc2)Cl)SCc3ccc(cc3)Cl 4J-336S CC(C)(C)c1ccc(cc1)Oc2c(cnc(n2)SCc3ccc(cc3)Cl)OC 4J-337S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(ccc3Cl)Cl)ncn2C(C)C 4J-340S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)ncn2C(C)C 4J-341S c1cc(ccc1c2cc(c(=O)[nH]c2)C#N)Cl 4J-342S CN(C)c1ncc(c(n1)Sc2ccc(cc2)Cl)OC 4J-344S CN(C)c1ncc(c(n1)OC)OC 4J-345S CCOC(=O)CSc1ncc(c(n1)Cl)OC 4J-346S CCOC(=O)CSc1ncc(c(n1)Sc2ccc(cc2)Cl)OC 4J-347S CCOC(=O)CSc1ncc(c(n1)Sc2ccc(cc2)OC)OC 4J-348S CC(=C)Cn1cc(cc(c1=O)C#N)c2ccc(cc2)Cl 4J-350S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)Cl)ncn2C(C)C 4J-351S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3)C(F)(F)F)ncn2C(C)C 4J-352S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)F)ncn2C(C)C 4J-353S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccccc3Cl)ncn2C(C)C 4J-354S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(cc(c3)Cl)Cl)ncn2C(C)C 4J-355S Cc1cc2c(c(c1C)NS(=O)(=O)N(C)C)ncn2C(C)C 4J-356S Cc1c(cc(c(=O)[nH]1)C#N)c2ccccc2 4J-357S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)F)C)C 4J-358S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)OC)C)C 4J-359S CCOC(=O)CSc1ncc(c(n1)Oc2cccc(c2)C(F)(F)F)OC 4J-360S CCOC(=O)CSc1ncc(c(n1)Oc2ccc(c(c2)Cl)Cl)OC 4J-361S CCOC(=O)CSc1ncc(c(n1)Oc2cc(cc(c2)Cl)Cl)OC 4J-362S CCOC(=O)CSc1ncc(c(n1)Sc2ccccc2)OC 4J-363S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(ccc4Cl)Cl)C)C 4J-364S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cccc(c4Cl)Cl)C)C 4J-365S CCCn1cnc2c1cc(c(c2[N+](=O)[O-])C)C 4J-366S CCCn1cnc2c1cc(c(c2N)C)C 4J-367S CN(C)/C=C(\C=O)/c1ccc(cc1Cl)Cl 4J-368S COc1cnc(nc1OC)SCC(=O)OC 4J-369S c1ccc(cc1)NC(=O)NNc2ccc(nn2)Cl 4J-370S CCOC(=O)CSc1ncc(c(n1)Oc2cccc(c2)[N+](=O)[O-])OC 4J-371S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(c(c4)Cl)Cl)C)C 4J-372S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4Cl)Cl)C)C 4J-373S CCOC(=O)CSc1ncc(c(n1)Oc2ccc(cc2)OC)OC 4J-374S CCOC(=O)CSc1ncc(c(n1)Sc2ccccc2Cl)OC 4J-375S CCOC(=O)CSc1ncc(c(n1)Sc2cccc(c2)C(F)(F)F)OC 4J-376S c1ccc(cc1)Nc2nnc3n2nc(cc3)Cl 4J-377S c1ccc(cc1)Cn2cc(cc(c2=O)C#N)c3ccc(cc3)Cl 4J-379S C=CCn1cc(cc(c1=O)C#N)c2ccc(cc2)Cl 4J-380S COc1ccc(cc1)Cn2cc(cc(c2=O)C#N)c3ccc(cc3)Cl 4J-381S c1ccc(c(c1)Cn2cc(cc(c2=O)C#N)c3ccc(cc3)Cl)F 4J-382S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(cc(c4)Cl)Cl)C)C 4J-383S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(c(cc4Cl)Cl)Cl)C)C 4J-384S c1cc(ccc1c2cc(c(=O)n(c2)Cc3ccc(cc3Cl)Cl)C#N)Cl 4J-385S Cn1cc(cc(c1=O)C#N)c2ccc(cc2)Cl 4J-386S c1cc(cc(c1)F)Cn2cc(cc(c2=O)C#N)c3ccc(cc3)Cl 4J-387S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(c(c4Cl)Cl)Cl)C)C 4J-388S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4c(cc(cc4Cl)Cl)Cl)C)C 4J-389S CC(C)n1cc(cc(c1=O)C#N)c2ccc(cc2)Cl 4J-390S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)Cl)C)C 4J-391S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccccc4Cl)C)C 4J-392S CCOC(=O)C(C)Sc1ncc(c(n1)OC)OC 4J-393S CCOC(=O)C(C)Sc1ncc(c(n1)Sc2ccc(cc2)Cl)OC 4J-394S CCOC(=O)C(C)Sc1ncc(c(n1)Sc2ccc(cc2)Br)OC 4J-395S COc1cnc(nc1Cl)SC 4J-396S Cc1cc2c(c(c1C)N(=O)=O)ncn2Cc3ccc(cc3)OC 4J-397S Cc1cc2c(c(c1C)N)ncn2Cc3ccc(cc3)OC 4J-398S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)C)C)C 4J-399S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cccc(c4)C(F)(F)F)C)C 4J-400S Cc1ccccc1Cn2cnc3c2cc(c(c3N(=O)=O)C)C 4J-402S Cc1ccccc1Cn2cnc3c2cc(c(c3N)C)C 4J-403S Cc1c(cc(c(n1)Cl)C#N)c2ccccc2 4J-404S Cc1cccc(c1)Cn2cnc3c2cc(c(c3NS(=O)(=O)C(F)(F)F)C)C 4J-405S CCCn1cnc2c1cc(c(c2NS(=O)(=O)c3ccc(cc3)OC)C)C 4J-406S CCCn1cnc2c1cc(c(c2NS(=O)(=O)c3ccc(cc3)Cl)C)C 4J-407S c1ccc(cc1)c2cc(c(=O)[nH]c2)C#N 4J-408S Cc1c(cc(c(n1)Sc2ccccc2)C#N)c3ccccc3 4J-409S Cc1c(cc(c(n1)Oc2ccc(cc2)OC)C#N)c3ccccc3 4J-410S CCCn1cnc2c1cc(c(c2NS(=O)(=O)c3ccc(cc3)F)C)C 4J-411S CCCn1cnc2c1cc(c(c2NS(=O)(=O)c3cccc(c3)C(F)(F)F)C)C 4J-412S CCCn1cnc2c1cc(c(c2NS(=O)(=O)c3cc(ccc3Cl)Cl)C)C 4J-413S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CSc4ccc(cc4)Br 4J-501S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CSc4cccc(c4)C(F)(F)F 4J-502S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CSc4ccc(c(c4)Cl)Cl 4J-503S Cc1ccc(cc1)SCc2c3ccccc3oc2C(=O)c4ccccc4 4J-504S c1ccc(cc1)S(=O)Cc2c3ccccc3oc2C(=O)c4ccc(cc4)Cl 4J-505S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)c4ccc(cc4Cl)Cl 4J-506S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)c4ccc(cc4)Cl 4J-507S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)(=O)c4ccc(cc4)Br 4J-508S Cc1ccc(cc1)S(=O)(=O)Cc2c3ccccc3oc2C(=O)c4ccccc4 4J-509S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)(=O)c4cccc(c4)C(F)(F)F 4J-510S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)(=O)c4ccc(c(c4)Cl)Cl 4J-511S Cc1ccc(cc1)S(=O)Cc2c3ccccc3oc2C(=O)c4ccccc4 4J-513S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)c4cccc(c4)C(F)(F)F 4J-514S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)c4ccc(c(c4)Cl)Cl 4J-515S CC1(CO1)C(=O)Nc2ccc(cc2)Cl 4J-518S CC(CS(=O)(=O)c1ccc(cc1)Br)(C(=O)Nc2ccc(cc2)Cl)O 4J-519S Cc1c2ccccc2oc1C(=O)c3ccc(c(c3)Cl)Cl 4J-520S c1cc(ccc1C(=O)NCCS(=O)(=O)c2ccc(cc2)Cl)F 4J-521S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CSCc4cccc(c4)C(F)(F)F 4J-523S CC(CS(=O)(=O)c1ccc(cc1)F)(C(=O)Nc2ccc(cc2)Cl)O 4J-526S CC(CS(=O)(=O)c1ccccc1)(C(=O)Nc2ccc(cc2)Cl)O 4J-527S CC(CS(=O)(=O)C1CCCCC1)(C(=O)Nc2ccc(cc2)Cl)O 4J-528S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CSc4ccc(cc4)Br 4J-530S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CSc4ccccc4Cl 4J-531S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CSc4c(cccc4Cl)Cl 4J-532S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CSCc4cccc(c4)C(F)(F)F 4J-536S CCCn1c2ccccc2nc1c3cccnc3Cl 4J-537S CC(CS(=O)(=O)c1ccc(c(c1)Cl)Cl)(C(=O)Nc2ccc(cc2)Cl)O 4J-538S CC(CS(=O)(=O)c1cc(cc(c1)Cl)Cl)(C(=O)Nc2ccc(cc2)Cl)O 4J-539S CC(CS(=O)c1ccc(cc1)Cl)(C(=O)Nc2ccc(cc2)Cl)O 4J-540S CC(CS(=O)(=O)c1cccc(c1)C(F)(F)F)(C(=O)Nc2ccc(cc2)Cl)O 4J-541S CC(CS(=O)(=O)Cc1ccc(cc1)Cl)(C(=O)Nc2ccc(cc2)Cl)O 4J-542S CC(CS(=O)(=O)c1cccc(c1)Cl)(C(=O)Nc2ccc(cc2)Cl)O 4J-544S Cc1ccc(cc1)S(=O)(=O)CC(C)(C(=O)Nc2ccc(cc2)Cl)O 4J-545S CC(CS(=O)(=O)c1ccc(cc1)OC)(C(=O)Nc2ccc(cc2)Cl)O 4J-546S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)(=O)c4c(cccc4Cl)Cl 4J-548S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)c4ccc(cc4)Br 4J-549S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)c4ccccc4Cl 4J-550S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)c4c(cccc4Cl)Cl 4J-551S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)(=O)Cc4cccc(c4)C(F)(F)F 4J-552S CC(=C)C(=O)Nc1cccc(c1)C(F)(F)F 4J-553S CC1(CO1)C(=O)Nc2cccc(c2)C(F)(F)F 4J-554S CC(CS(=O)(=O)c1ccccc1)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-555S CC(CS(=O)(=O)c1ccc(c(c1)Cl)Cl)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-556S CC(CSc1ccc(cc1)Br)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-557S CC(CS(=O)(=O)c1ccc(cc1)Br)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-558S Cc1ccc(cc1)S(=O)(=O)CC(C)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-559S CC(CS(=O)(=O)c1ccc(cc1)OC)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-560S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CSc4ccccc4 4J-561S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CSc4ccccc4Cl 4J-562S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CSc4ccc(cc4)Cl 4J-563S COc1ccc(cc1)SCc2c3ccccc3oc2C(=O)c4ccccc4 4J-564S Cc1ccccc1SCc2c3ccccc3oc2C(=O)c4ccccc4 4J-565S CC(CS(=O)(=O)c1ccc(cc1)Cl)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-567S CC(CS(=O)(=O)c1ccc(cc1)F)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-568S CC(CS(=O)(=O)Cc1ccc(cc1)Cl)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-569S CC(CS(=O)(=O)Cc1ccccc1Cl)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-570S CC(CS(=O)(=O)Cc1ccccc1)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-571S CC(CS(=O)(=O)Cc1cccc(c1)C(F)(F)F)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-572S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)c4ccccc4 4J-574S Cc1ccccc1S(=O)Cc2c3ccccc3oc2C(=O)c4ccccc4 4J-575S COc1ccc(cc1)S(=O)Cc2c3ccccc3oc2C(=O)c4ccccc4 4J-576S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)c4ccccc4Cl 4J-577S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)c4ccc(cc4)Cl 4J-578S Cc1ccccc1S(=O)(=O)Cc2c3ccccc3oc2C(=O)c4ccccc4 4J-580S COc1ccc(cc1)S(=O)(=O)Cc2c3ccccc3oc2C(=O)c4ccccc4 4J-581S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)(=O)c4ccccc4Cl 4J-582S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)(=O)c4ccc(cc4)Cl 4J-583S CC(CS(=O)(=O)c1cccc(c1)C(F)(F)F)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-584S CC1(CO1)C(=O)Nc2ccc(cc2Cl)Cl 4J-585S CC(CS(=O)(=O)c1ccc(cc1)Br)(C(=O)Nc2ccc(cc2Cl)Cl)O 4J-586S CC(CS(=O)(=O)c1ccccc1)(C(=O)Nc2ccc(cc2Cl)Cl)O 4J-587S CC(CS(=O)(=O)c1ccc(cc1)Cl)(C(=O)Nc2ccc(cc2Cl)Cl)O 4J-588S CC(CS(=O)(=O)Cc1ccccc1)(C(=O)Nc2ccc(cc2Cl)Cl)O 4J-589S CC(CSc1ccc(cc1)Cl)(C(=O)Nc2ccc(cc2)Cl)O 4J-590S CC(CS(=O)(=O)c1ccc(cc1)Cl)(C(=O)Nc2ccc(cc2)Cl)O 4J-591S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)Cc4cccc(c4)C(F)(F)F 4J-592S c1ccc(cc1)C(=O)c2c(c3ccccc3o2)CS(=O)(=O)Cc4cccc(c4)C(F)(F)F 4J-593S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(c(c3)Cl)Cl)CSc4cccc(c4)C(F)(F)F 4J-595S Cc1c2ccccc2oc1C(=O)c3ccc(cc3)OC 4J-596S COc1cnc(nc1Cl)SCc2ccc(cc2Cl)Cl 4J-597S c1cc(ccc1SCCNC(=O)c2ccc(c(c2)Cl)Cl)Cl 4J-599S COc1cccc(c1)C(=O)NCCSc2ccc(cc2)Cl 4J-600S c1cc(cc(c1)Cl)C(=O)NCCS(=O)(=O)c2ccc(cc2)Cl 4J-601S COc1cnc(nc1OC)SCc2ccc(cc2Cl)Cl 4J-602S COc1cnc(nc1Oc2ccc(cc2)Cl)SCc3ccc(cc3Cl)Cl 4J-604S COc1cnc(nc1Oc2cc(cc(c2)Cl)Cl)SCc3ccc(cc3Cl)Cl 4J-605S CC(C)(C)S(=O)(=O)CC(C)(C(=O)Nc1cccc(c1)C(F)(F)F)O 4J-606S CC(CS(=O)(=O)C1CCCCC1)(C(=O)Nc2cccc(c2)C(F)(F)F)O 4J-607S COc1ccc(cc1)Oc2c(cnc(n2)SCc3ccc(cc3Cl)Cl)OC 4J-609S COc1cnc(nc1Oc2ccc(c(c2)Cl)Cl)SCc3ccc(cc3Cl)Cl 4J-610S c1cc(ccc1S(=O)(=O)CCNC(=O)c2ccc(c(c2)Cl)Cl)Cl 4J-611S Cc1c(nn(c1c2ccccc2)Cc3ccc(c(c3)Cl)Cl)c4ccccc4 4J-650S C/C(=C\c1ccc(cc1)Cl)/C(=O)c2ccccc2 4J-651S COc1cnc(nc1OC)SCc2cccc(c2)C(F)(F)F 4J-653S COc1cnc(nc1Sc2ccc(cc2)Br)SCc3cccc(c3)C(F)(F)F 4J-654S COc1cnc(nc1O)SCc2ccc(c(c2)Cl)Cl 4J-655S COc1cnc(nc1Cl)SCc2ccc(c(c2)Cl)Cl 4J-656S CC(C)(C)c1ccc(cc1)CSc2ncc(c(n2)O)OC 4J-657S COc1ccc(cc1)Sc2c(cnc(n2)SCc3ccc(c(c3)Cl)Cl)OC 4J-658S COc1cnc(nc1Sc2cccc(c2)C(F)(F)F)SCc3ccc(c(c3)Cl)Cl 4J-659S COc1cnc(nc1SCc2ccc(cc2)Cl)SCc3ccc(c(c3)Cl)Cl 4J-660S COc1cnc(nc1Sc2ccc(cc2)Br)SCc3ccc(c(c3)Cl)Cl 4J-661S COc1cnc(nc1Sc2ccc(cc2)Cl)SCc3ccc(c(c3)Cl)Cl 4J-662S COc1cnc(nc1OC)SCc2ccc(c(c2)Cl)Cl 4J-663S COc1ccc(cc1)Sc2c(cnc(n2)SCc3cccc(c3)C(F)(F)F)OC 4J-665S COc1cnc(nc1SCc2ccc(cc2)Cl)SCc3cccc(c3)C(F)(F)F 4J-666S COc1cnc(nc1SC)SCc2ccc(c(c2)Cl)Cl 4J-667S COc1cnc(nc1Sc2c(c(c(c(c2F)F)F)F)F)SCc3ccc(c(c3)Cl)Cl 4J-668S COc1cnc(nc1Sc2cccc(c2)Cl)SCc3ccc(c(c3)Cl)Cl 4J-669S COc1cnc(nc1Sc2ccccc2Cl)SCc3ccc(c(c3)Cl)Cl 4J-670S COc1cnc(nc1Sc2ccccc2)SCc3ccc(c(c3)Cl)Cl 4J-671S COc1cnc(nc1Oc2ccccc2)SCc3ccc(c(c3)Cl)Cl 4J-672S COc1cnc(nc1Oc2cc(cc(c2)Cl)Cl)SCc3ccc(c(c3)Cl)Cl 4J-673S COc1cnc(nc1Oc2ccc(c(c2)Cl)Cl)SCc3ccc(c(c3)Cl)Cl 4J-674S COc1cnc(nc1Oc2ccc(cc2)F)SCc3ccc(c(c3)Cl)Cl 4J-675S COc1cnc(nc1Oc2cc(c(cc2Cl)Cl)Cl)SCc3ccc(c(c3)Cl)Cl 4J-676S COc1cnc(nc1Oc2cccc(c2)C(F)(F)F)SCc3ccc(c(c3)Cl)Cl 4J-678S COc1cnc(nc1Oc2ccc(cc2Cl)Cl)SCc3ccc(c(c3)Cl)Cl 4J-679S c1ccc2c(c1)c(c(o2)C(=O)c3ccc(cc3)Cl)CS(=O)(=O)c4ccc(cc4)Br 4J-846S COC(=O)C1CSC(N1C(=O)Nc2ccc(cc2)Cl)C(=O)OC 4J-900 COC(=O)C1CSC(N1C(=O)CON2C(=O)c3ccccc3C2=O)C(=O)OC 4J-901 COC(=O)C1N2C(CS1)C(=O)N(CC2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 4J-903 c1ccc(cc1)C(=O)Nc2cc(c3ccccn3c2=O)C#N 4J-905 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2cc(ccc2Cl)Cl 4J-906 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)C 4J-907 c1ccc2c(c1)NC(=O)CC(=O)N2 4J-909 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2cccc(c2)C(F)(F)F 4J-910 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC=C)S(=O)(=O)c2cc(ccc2Cl)Cl 4J-911 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC=C)S(=O)(=O)C 4J-912 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2ccc(cc2)OC 4J-913 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC=C)S(=O)(=O)c2cccc(c2)C(F)(F)F 4J-914 CN1C(CC(O1)CNC(=O)C2CCN(CC2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])c4ccc(cc4)OC 4J-915 CC(=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl)N(C)C 4J-916 COC(=O)C1CCN(CC1)c2ccc(nn2)Cl 4J-917 CC(=O)C1=NOC(C1)CN(N(C)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)c3cccc(c3)C(F)(F)F 4J-918 c1cc(nnc1N2CCC(CC2)C(=O)O)Cl 4J-920 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC2CC(N(O2)c3ccccc3)c4ccccc4)S(=O)(=O)C 4J-922 CC1=NN(C(=O)C1C(c2ccccc2)N(c3ccccc3)O)c4ccccc4 4J-923 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC=C)S(=O)(=O)c2ccc(cc2)OC 4J-925 C=CCNC(=O)C1CCN(CC1)c2ccc(nn2)Cl 4J-926 CN(C)CCNC=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 4J-927 COCCCNC=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl 4J-928 CC(=O)C1=NOC(C1)CN(N(C)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)C 4J-929 c1ccc(cc1)C(=O)NC(=S)NCCc2ccccn2 4J-930 CC1(OCCO1)c2ccc(c(c2)[N+](=O)[O-])Cl 4J-931 c1ccc(cc1)S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C3OCCO3 4J-932 CN1C(CC(O1)CN(N(C)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)C)c3ccc(cc3)OC 4J-934 CN1C(CC(O1)CNC(=O)C2CCN(CC2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])c4ccccc4 4J-935 CC(=O)C1=NOC2C1C(=O)N(C2=O)c3cccc(c3)C(F)(F)F 4J-936 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/C2=NOC3C2C(=O)N(C3=O)c4cccc(c4)C(F)(F)F 4J-937 c1ccc(cc1)S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C=O 4J-938 CC1(OCCO1)c2ccc(c(c2)CS(=O)(=O)c3ccccc3)[N+](=O)[O-] 4J-941 CN1C(CC(O1)CN(N(C)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)C)c3ccccc3 4J-942 CC(=O)c1ccc(c(c1)CS(=O)(=O)c2ccccc2)[N+](=O)[O-] 4J-943 CN(C)/C=C/C(=O)c1ccc(c(c1)CS(=O)(=O)c2ccccc2)[N+](=O)[O-] 4J-944 c1ccc(cc1)S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])c3cc[nH]n3 4J-945 CC1(OCCO1)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 4J-946 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)O)Cl 4J-947 c1ccc(cc1)S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])c3ccn(n3)c4c(cc(cn4)C(F)(F)F)Cl 4J-948 c1ccc2c(c1)CCN3C2CC(O3)CNC(=O)C4CCN(CC4)c5ccc(nn5)Cl 4J-949 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC2CC(N(O2)Cc3ccccc3)c4ccccc4)S(=O)(=O)C 4J-950 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)N3CCOCC3)Cl 4J-952 CSC(=C(C#N)c1ccc(cc1)[N+](=O)[O-])SC 4K-002 c1ccc(cc1)S(=O)(=O)C/C=C/C#N 4K-004 CN(C)/C=C(/C=C/C#N)\S(=O)(=O)c1ccccc1 4K-005 Cc1c(c(no1)c2c(cccc2Cl)F)C(=S)/N=C/N(C)C 4K-006 Cc1c(c(no1)c2c(cccc2Cl)F)c3ncc(s3)C(=O)c4ccc(cc4)Cl 4K-008 Cc1cc(nc(c1C#N)S)C 4K-009 CC1CC(CC2(C1)CC(=O)OC2=O)(C)C 4K-010 Cc1cc(nc(c1C#N)SC/C=C/C#N)C 4K-011 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)Cl)/C=C/C#N 4K-012 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)C(F)(F)F)/C=C/C#N 4K-013 COc1ccnc(c1C(=O)N)S(=O)(=O)c2ccc(cc2)Cl 4K-014 COc1ccc(cc1)N/C=C(\C=C\C#N)/S(=O)(=O)c2ccccc2 4K-015 c1cn(c(n1)S)c2c(cc(cn2)C(F)(F)F)Cl 4K-018 Cc1cc(nc2c1c(c(s2)/C=C/C#N)N)C 4K-019 COC(=O)/C=C/CS(=O)(=O)c1ccccc1 4K-020 CN(C)/C=C(\C=C\C(=O)OC)/S(=O)(=O)c1ccccc1 4K-021 CC1CC(CC2(C1)CC(=O)N(C2=O)c3cccc(c3)C(F)(F)F)(C)C 4K-022 COc1ccc(cc1)N/C=C(\C=C\C(=O)OC)/S(=O)(=O)c2ccccc2 4K-023 Cc1c2ccccc2ncc1c3c(cc(cn3)C(F)(F)F)Cl 4K-026 Cc1cc(nc2c1c(c(s2)/C=C/C#N)n3cccc3)C 4K-027 c1cc(ccc1C(=O)CSc2nccn2c3c(cc(cn3)C(F)(F)F)Cl)Cl 4K-029 COC(=O)c1ccccc1N/C=C/c2c(cc(cn2)C(F)(F)F)Cl 4K-031 Cc1cc(nc(c1C#N)SC/C=C/C(=O)OC)C 4K-035 COC(=O)/C=C/C(=C\Nc1ccc(cc1)F)/S(=O)(=O)c2ccccc2 4K-036 Cc1cc(nc2c1c(c(s2)/C=C/C(=O)OC)N)C 4K-037 Cc1cc(nc(c1S(=O)(=O)c2cccc(c2)C(F)(F)F)OCC(C)C)C 4K-301S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)C(C)(C)C)OCC(C)C)C 4K-302S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)COC(=O)c4ccc(cc4)Cl 4K-303S Cc1ccc(cc1)S(=O)(=O)c2c(c(nn2C)c3ccccc3)COC(=O)c4ccc(cc4)Cl 4K-304S Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)COC(=O)Nc4ccc(cc4)Cl 4K-305S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)COC(=O)Nc4ccccc4 4K-306S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)COC(=O)C 4K-307S CC(CS(=O)(=O)Cc1ccccc1)(c2ccc(c(c2)Cl)Cl)O 4K-308S CC(CS(=O)(=O)Cc1ccc(cc1)Cl)(c2ccc(c(c2)Cl)Cl)O 4K-309S CC(CS(=O)(=O)Cc1cccc(c1)C(F)(F)F)(c2ccccc2)O 4K-310S CC(CS(=O)(=O)Cc1cccc(c1)C(F)(F)F)(c2ccc(cc2)Cl)O 4K-311S CC(CS(=O)(=O)Cc1ccc(cc1)Cl)(c2ccccc2Cl)O 4K-312S CC(CS(=O)(=O)Cc1ccccc1)(c2ccccc2Cl)O 4K-313S Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)COC(=O)c4ccccc4Cl 4K-314S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)COC(=O)c4ccccc4Cl 4K-315S Cc1ccc(cc1)S(=O)(=O)c2c(c(nn2C)c3ccccc3)COC(=O)c4ccccc4Cl 4K-316S Cn1c(c(c(n1)c2ccccc2)C=O)Sc3ccc(cc3)Cl 4K-317S Cn1c(c(c(n1)c2ccccc2)C=O)Sc3ccccc3Cl 4K-318S Cn1c(c(c(n1)c2ccccc2)C=O)Sc3ccccc3 4K-319S Cn1c(c(c(n1)c2ccccc2)C=O)Sc3ccc(cc3)Br 4K-320S Cn1c(c(c(n1)c2ccccc2)CO)Sc3ccc(cc3)Cl 4K-321S Cn1c(c(c(n1)c2ccccc2)CO)Sc3ccccc3Cl 4K-322S Cn1c(c(c(n1)c2ccccc2)CO)Sc3ccccc3 4K-323S CC(CS(=O)(=O)Cc1ccc(cc1)OC)(c2ccccc2Cl)O 4K-324S CC(CS(=O)(=O)Cc1ccc(cc1Cl)Cl)(c2ccc(c(c2)Cl)Cl)O 4K-325S Cc1ccc(cc1)C(C)(CS(=O)(=O)Cc2ccc(cc2)Cl)O 4K-326S Cn1c(c(c(n1)c2ccccc2)CO)Sc3ccc(cc3)Br 4K-327S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OCCN(C)C)C)C 4K-328S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OCCN3CCOCC3)C)C 4K-329S Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)COC(=O)CCl 4K-330S Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)COC(=O)Nc4cccc(c4)Cl 4K-331S Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)COC(=O)c4ccc(cc4)F 4K-332S Cc1ccc(cc1)Oc2c(c(nn2C)c3ccccc3)COC(=O)c4ccc(cc4)Cl 4K-333S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)COC(=O)c4cccc(c4)Cl 4K-334S CC(CS(=O)(=O)Cc1ccc(cc1)OC)(c2ccc(c(c2)Cl)Cl)O 4K-335S CC(CS(=O)(=O)Cc1ccccc1Cl)(c2ccc(cc2)Cl)O 4K-337S Cc1ccc(cc1)C(C)(CS(=O)(=O)Cc2ccccc2)O 4K-338S Cc1ccc(cc1)C(C)(CS(=O)(=O)Cc2ccccc2Cl)O 4K-339S COc1ccc(cc1)NC(=O)Cc2c(nc(s2)c3ccccc3)c4ccccc4 4K-340S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)C(F)(F)F)Cl)C 4K-342S Cc1ccc(cc1S(=O)(=O)c2c(cc([nH]c2=O)C)C)F 4K-345S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)C(F)(F)F)OCC(C)C)C 4K-346S CCOC(=O)c1c(nc(nn1)c2ccccc2)O 4K-350S Cc1ccc(cc1S(=O)(=O)c2c(cc(nc2Cl)C)C)F 4K-351S Cc1ccc(cc1)S(=O)(=O)c2c(c(nn2C)c3ccccc3)COC(=O)c4cccc(c4)Cl 4K-354S Cc1cc(c(c(n1)Oc2cccc(c2)C(F)(F)F)C#N)C(F)(F)F 4K-355S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)COC(=O)c4cccc(c4)C 4K-356S Cc1ccc(cc1)S(=O)(=O)c2c(c(nn2C)c3ccccc3)COC(=O)c4cccc(c4)C 4K-357S Cn1c(c(c(n1)c2ccccc2)CCl)Sc3ccc(cc3)Cl 4K-358S Cc1cc(c(c(=O)n1c2ccc(cc2Cl)Cl)C#N)C(F)(F)F 4K-359S Cn1c(c(c(n1)c2ccccc2)COC)Sc3ccc(cc3)Cl 4K-360S Cn1c(c(c(n1)c2ccccc2)CO)Oc3ccc(cc3)F 4K-361S CN(c1cnns1)NC(=O)C(=C(Cl)Cl)Cl 4K-363S CN(c1cnns1)N(S(=O)(=O)C)S(=O)(=O)C 4K-364S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccc(cc2C)F)C 4K-366S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2C)F)Cl)C 4K-367S Cn1c(c(c(n1)c2ccccc2)CO)Oc3cccc(c3)C(F)(F)F 4K-368S Cn1c(c(c(n1)c2ccccc2)CO)Sc3cccc(c3)C(F)(F)F 4K-369S Cn1c(c(c(n1)c2ccccc2)COC(=O)Nc3cccc(c3)Cl)Sc4ccc(cc4)Cl 4K-370S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl 4K-371S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)Cl)S(=O)(=O)c4ccc(cc4)Cl 4K-372S Cn1c(c(c(n1)c2ccccc2)COc3c(cccc3Cl)Cl)Sc4ccc(cc4)Cl 4K-373S C=CCn1c(c(nc1SCc2ccc(cc2)Cl)c3ccccc3)c4ccccc4 4K-501S C#CCn1c(c(nc1SCc2ccc(cc2)Cl)c3ccccc3)c4ccccc4 4K-502S Cn1c(c(nc1SCc2ccc(c(c2)Cl)Cl)c3ccccc3)c4ccccc4 4K-503S CCCn1c(c(nc1SCc2ccc(c(c2)Cl)Cl)c3ccccc3)c4ccccc4 4K-504S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)Br)Cl 4K-506S Cn1c(c(c(n1)c2ccccc2)CSc3cc(ccc3Cl)Cl)Cl 4K-508S Cn1c(c(c(n1)c2ccccc2)CSc3ccc(cc3Cl)Cl)Cl 4K-509S Cn1c(c(c(n1)c2ccccc2)CSc3cccc(c3Cl)Cl)Cl 4K-510S Cn1c(c(c(n1)c2ccccc2)CS(=O)(=O)c3ccccc3OC)Cl 4K-511S Cn1c(c(c(n1)c2ccccc2)COC(=O)Nc3ccc(cc3)Cl)Cl 4K-512S C=CCn1c(c(nc1SCc2ccc(c(c2)Cl)Cl)c3ccccc3)c4ccccc4 4K-516S Cn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)Cl)c3ccccc3)c4ccccc4 4K-518S CCCn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)Cl)c3ccccc3)c4ccccc4 4K-519S Cn1c(c(nc1S(=O)(=O)Cc2ccc(c(c2)Cl)Cl)c3ccccc3)c4ccccc4 4K-521S CCCn1c(c(nc1S(=O)(=O)Cc2ccc(c(c2)Cl)Cl)c3ccccc3)c4ccccc4 4K-522S c1ccc(cc1)C(=O)C(CC(=O)O)Br 4K-525S COC(=O)Cc1c(nc(s1)c2ccccc2)c3ccccc3 4K-526S C=CCn1c(c(nc1S(=O)(=O)Cc2ccc(c(c2)Cl)Cl)c3ccccc3)c4ccccc4 4K-528S Cn1c(c(c(n1)c2ccccc2)COCC=C)Cl 4K-530S Cn1c(c(c(n1)c2ccccc2)COC(=O)Nc3ccccc3)Cl 4K-531S c1ccc(cc1)c2c(nc([nH]2)SCc3cccc(c3)C(F)(F)F)c4ccccc4 4K-532S CC(C)(C)c1ccc(cc1)CSc2[nH]c(c(n2)c3ccccc3)c4ccccc4 4K-533S c1ccc(cc1)c2c(nc([nH]2)SCc3c(cccc3Cl)Cl)c4ccccc4 4K-534S Cn1c(c(nc1SCc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4 4K-535S CCCn1c(c(nc1SCc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4 4K-536S C=CCn1c(c(nc1SCc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4 4K-537S C#CCn1c(c(nc1SCc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4 4K-538S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)O 4K-539S Cn1c(c(c(n1)c2ccccc2)CO)Sc3c(cccc3Cl)Cl 4K-542S Cn1c(c(c(n1)c2ccccc2)CCl)Sc3c(cccc3Cl)Cl 4K-543S Cn1c(c(c(n1)c2ccccc2)COC)Sc3c(cccc3Cl)Cl 4K-544S Cn1c(c(c(n1)c2ccccc2)COCC=C)Sc3c(cccc3Cl)Cl 4K-545S Cn1c(c(c(n1)c2ccccc2)COCc3ccc(cc3)OC)Sc4c(cccc4Cl)Cl 4K-546S CC(C)(C)c1ccc(cc1)CSc2nc(c(n2C)c3ccccc3)c4ccccc4 4K-548S CCCn1c(c(nc1SCc2ccc(cc2)C(C)(C)C)c3ccccc3)c4ccccc4 4K-549S CC(C)(C)c1ccc(cc1)CSc2nc(c(n2CC=C)c3ccccc3)c4ccccc4 4K-550S CC(C)(C)c1ccc(cc1)CSc2nc(c(n2CC#C)c3ccccc3)c4ccccc4 4K-551S Cn1c(c(nc1SCc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-552S CCCn1c(c(nc1SCc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-553S C=CCn1c(c(nc1SCc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-554S C#CCn1c(c(nc1SCc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-555S Cn1c(c(nc1S(=O)(=O)Cc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4 4K-557S CCCn1c(c(nc1S(=O)(=O)Cc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4 4K-558S C=CCn1c(c(nc1S(=O)(=O)Cc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4 4K-559S CC(C)(C)c1ccc(cc1)CS(=O)(=O)c2nc(c(n2C)c3ccccc3)c4ccccc4 4K-560S CCCn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)C(C)(C)C)c3ccccc3)c4ccccc4 4K-561S CC(C)(C)c1ccc(cc1)CS(=O)(=O)c2nc(c(n2CC=C)c3ccccc3)c4ccccc4 4K-562S CCCn1c(c(nc1S(=O)(=O)Cc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-564S C=CCn1c(c(nc1S(=O)(=O)Cc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-565S C#CCn1c(c(nc1S(=O)(=O)Cc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-566S CC(C)(C)c1ccc(cc1)CS(=O)(=O)c2nc(c(n2CC#C)c3ccccc3)c4ccccc4 4K-567S CCOC(=O)Cn1c(c(nc1SCc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-568S c1ccc(cc1)c2c(nc([nH]2)SCc3ccccc3Cl)c4ccccc4 4K-569S c1ccc(cc1)c2c(nc([nH]2)SCc3ccc(cc3)F)c4ccccc4 4K-570S COc1ccc(cc1)CSc2[nH]c(c(n2)c3ccccc3)c4ccccc4 4K-571S CCOC(=O)Cn1c(c(nc1S(=O)(=O)Cc2c(cccc2Cl)Cl)c3ccccc3)c4ccccc4 4K-572S Cn1c(c(c(n1)c2ccccc2)COCc3ccccc3)Cl 4K-573S Cn1c(c(nc1SCc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-574S CCCn1c(c(nc1SCc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-575S C=CCn1c(c(nc1SCc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-576S Cn1c(c(c(n1)c2ccccc2)COCc3ccc(cc3)OC)Cl 4K-577S Cn1c(c(c(n1)c2ccccc2)COCc3c(cccc3Cl)Cl)Cl 4K-578S Cn1c(c(c(n1)c2ccccc2)COCc3ccc(cc3Cl)Cl)Cl 4K-579S C#CCn1c(c(nc1SCc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-580S CCOC(=O)Cn1c(c(nc1SCc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-581S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)Nc4ccc(cc4)F 4K-582S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)Nc4ccc(cc4)Cl 4K-583S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)Nc4ccccc4 4K-584S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)Nc4ccc(c(c4)Cl)Cl 4K-585S Cn1c(c(nc1SCc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-586S CCCn1c(c(nc1SCc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-587S C=CCn1c(c(nc1SCc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-588S C#CCn1c(c(nc1SCc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-589S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)Nc4ccc(cc4)OC(F)(F)F 4K-590S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)Nc4cccc(c4)C(F)(F)F 4K-591S CCOC(=O)Cn1c(c(nc1SCc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-592S Cn1c(c(nc1SCc2ccc(cc2)OC)c3ccccc3)c4ccccc4 4K-593S CCCn1c(c(nc1SCc2ccc(cc2)OC)c3ccccc3)c4ccccc4 4K-594S COc1ccc(cc1)CSc2nc(c(n2CC=C)c3ccccc3)c4ccccc4 4K-595S COc1ccc(cc1)CSc2nc(c(n2CC#C)c3ccccc3)c4ccccc4 4K-596S CCOC(=O)Cn1c(c(nc1SCc2ccc(cc2)OC)c3ccccc3)c4ccccc4 4K-597S Cn1c(c(nc1S(=O)(=O)Cc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-598S CCCn1c(c(nc1S(=O)(=O)Cc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-599S C=CCn1c(c(nc1S(=O)(=O)Cc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-600S C#CCn1c(c(nc1S(=O)(=O)Cc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-601S CCOC(=O)Cn1c(c(nc1S(=O)(=O)Cc2ccccc2Cl)c3ccccc3)c4ccccc4 4K-602S Cn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-603S C=CCn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-604S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)Nc4ccc(cc4F)F 4K-605S C#CCn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-606S CCOC(=O)Cn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)F)c3ccccc3)c4ccccc4 4K-607S Cn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)OC)c3ccccc3)c4ccccc4 4K-608S CCCn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)OC)c3ccccc3)c4ccccc4 4K-609S COc1ccc(cc1)CS(=O)(=O)c2nc(c(n2CC#C)c3ccccc3)c4ccccc4 4K-611S CCOC(=O)Cn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)OC)c3ccccc3)c4ccccc4 4K-612S c1ccc(cc1)c2c(nc([nH]2)SCc3cccc(c3)F)c4ccccc4 4K-613S Cc1ccc(cc1)CSc2[nH]c(c(n2)c3ccccc3)c4ccccc4 4K-614S c1ccc(cc1)c2c(nc([nH]2)SCc3ccc(cc3)[N+](=O)[O-])c4ccccc4 4K-615S c1ccc(cc1)c2c(sc(n2)c3ccccc3)CC(=O)NC4CCCCC4 4K-618S C=CCNC(=O)Cc1c(nc(s1)c2ccccc2)c3ccccc3 4K-619S Cn1c(c(c(n1)c2ccccc2)COCc3ccc(cc3)Cl)Cl 4K-620S Cn1c(c(c(n1)c2ccccc2)COCc3cccc(c3)C(F)(F)F)Cl 4K-621S COC(=O)Cc1c(nc(s1)c2ccc(cc2)Cl)c3ccccc3 4K-622S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)O 4K-623S COc1ccc(cc1)NC(=O)Cc2c(nc(s2)c3ccc(cc3)Cl)c4ccccc4 4K-624S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)Nc4ccc(cc4)Cl 4K-625S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)Nc4ccc(c(c4)Cl)Cl 4K-626S Cn1c(c(nc1SCc2cccc(c2)F)c3ccccc3)c4ccccc4 4K-627S CCCn1c(c(nc1SCc2cccc(c2)F)c3ccccc3)c4ccccc4 4K-628S C=CCn1c(c(nc1SCc2cccc(c2)F)c3ccccc3)c4ccccc4 4K-629S C#CCn1c(c(nc1SCc2cccc(c2)F)c3ccccc3)c4ccccc4 4K-630S CCOC(=O)Cn1c(c(nc1SCc2cccc(c2)F)c3ccccc3)c4ccccc4 4K-631S Cn1c(c(c(n1)c2ccccc2)C(c3ccccc3)O)Cl 4K-632S Cc1ccc(cc1)CSc2nc(c(n2C)c3ccccc3)c4ccccc4 4K-633S CCCn1c(c(nc1SCc2ccc(cc2)C)c3ccccc3)c4ccccc4 4K-634S Cc1ccc(cc1)CSc2nc(c(n2CC=C)c3ccccc3)c4ccccc4 4K-635S Cc1ccc(cc1)CSc2nc(c(n2CC#C)c3ccccc3)c4ccccc4 4K-636S CCOC(=O)Cn1c(c(nc1SCc2ccc(cc2)C)c3ccccc3)c4ccccc4 4K-637S CCOC(=O)Cn1c(c(nc1SCc2ccc(cc2)[N+](=O)[O-])c3ccccc3)c4ccccc4 4K-641S c1ccc(cc1)N2CCN(CC2)C(=O)c3cccnc3Sc4c(cc(cn4)C(F)(F)F)Cl 4K-900 c1cncc(c1C(=O)O)N 4K-902 CN1C(C2C(O1)CCCC2=O)c3ccccc3 4K-903 CC(=O)Nc1cnccc1C(=O)O 4K-904 c1ccc(cc1)OCCN2C(=O)c3ccccc3C2=O 4K-905 c1cncc(c1C(=O)O)O 4K-906 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)c3cccc(c3C2=O)[N+](=O)[O-] 4K-907 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)c3cccc(c3C2=O)N 4K-909 CCOC(=O)C(C#N)c1cc(ccc1[N+](=O)[O-])C(F)(F)F 4K-911 CCOC(=O)c1c2cc(ccc2[nH]c1N)C(F)(F)F 4K-912 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)c3cccc(c3C2=O)n4cccc4 4K-913 c1cc2c(c(c1)[N+](=O)[O-])C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 4K-914 COC(=O)c1ccncc1O 4K-915 CCOC(=O)C(C#N)c1c(cccn1)[N+](=O)[O-] 4K-916 CC1(C2NC(=S)N(N2C(=S)N1)c3ccccc3)c4ccccc4 4K-919 c1ccc(cc1)OCCNC(=O)c2cccnc2Sc3c(cc(cn3)C(F)(F)F)Cl 4K-920 CCOC(=O)C(C#N)c1ccccc1[N+](=O)[O-] 4K-921 Cc1ccc(cc1)SCC(=O)Nc2ncc3c(n2)-c4ccccc4CC3 4K-922 Cc1ccc(cc1)/C=[N+](/C)\[O-] 4K-924 CCOC(=O)NC(=O)/C(=N/Nc1cc(cc(c1)C)C)/C(=O)C 4K-927 CCOC(=O)NC(=O)/C(=N\Nc1ccc(cc1)C(F)(F)F)/C(=O)C 4K-928 CC(=O)c1c(=O)[nH]c(=O)n(n1)c2ccc(cc2)C(F)(F)F 4K-929 Cn1c(=O)c(nn(c1=O)c2ccc(cc2)C(F)(F)F)C(=O)/C=C\N(C)C 4K-930 CC(C)(C)c1ccc(cc1)Oc2cc(cnc2C(=O)N)C(F)(F)F 4L-001 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)NN3CCOCC3 4L-002 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)OC 4L-003 CC(C)NC(=O)c1cnc(n1C)Sc2c(cc(cn2)C(F)(F)F)Cl 4L-004 c1cc(ccc1CO/N=C/c2ccnn2c3c(cc(cn3)C(F)(F)F)Cl)Cl 4L-005 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCc3cccc(c3)OC 4L-006 Cc1csc2c1c(ncn2)NCCc3ccccn3 4L-007 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCc3cccs3 4L-008 CCCNC(=O)c1cnc(n1C)Sc2c(cc(cn2)C(F)(F)F)Cl 4L-009 c1cc(cc(c1)OCCO/N=C\c2ccnn2c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 4L-010 Cn1c(cnc1Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C(=O)OC 4L-011 CCCCCCCCSc1ncc(n1C)C(=O)OC 4L-012 Cn1c(cnc1SCc2ccc(cc2)Cl)C(=O)OC 4L-013 c1cnn(c1C=C(C#N)C#N)c2c(cc(cn2)C(F)(F)F)Cl 4L-014 c1ccc(cc1)C(=O)/C(=C\c2ccnn2c3c(cc(cn3)C(F)(F)F)Cl)/C#N 4L-016 c1cc(ccc1NC(=O)NC(=O)Cn2cncn2)Cl 4L-017 C/C(=C/c1ccnn1c2c(cc(cn2)C(F)(F)F)Cl)/[N+](=O)[O-] 4L-018 COc1ccc(cc1)/C=C/c2ccnc(n2)[S-].[K+] 4L-021 c1cc(ccc1/C=C/c2ccnc(n2)[S-])Cl.[K+] 4L-022 CO/N=C/C(=C/c1cccn1c2c(cc(cn2)C(F)(F)F)Cl)/C#N 4L-023 c1ccc(cc1)S(=O)(=O)C(/C=N/OCc2c(cccc2Cl)F)[N+](=O)[O-] 4L-024 CO/N=C/C(=C/c1cccnc1)/C#N 4L-026 CN(C)c1ccc(cc1)/C=C(/C=N/OC)\C#N 4L-027 CO/N=C/C(=C/c1ccc(cc1)F)/C#N 4L-028 CO/N=C/C(=C/c1ccc[nH]1)/C#N 4L-029 COc1ccc(cc1OC)/C=C(/C=N/OC)\C#N 4L-030 CO/N=C/C(C#N)C1c2ccccc2C(=O)O1 4L-031 CO/N=C/C(=C/c1cccs1)/C#N 4L-032 CO/N=C/C(=C/c1ccccc1[N+](=O)[O-])/C#N 4L-033 c1cc(c(cc1C(=O)/C=C/c2ccnn2c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl 4L-034 CN(C)/C=C/C(=O)/C=C/c1ccc(cc1Cl)Cl 4L-035 c1cc(c(c(c1)Cl)CSc2nccc(n2)/C=C/c3ccc(cc3)Cl)Cl 4L-036 c1cc(sc1)/C=C/c2ccnc(n2)[S-].[K+] 4L-037 CC(=O)c1ccc(cc1)Oc2cc(cnc2C#N)C(F)(F)F 4L-038 c1cc(ccc1/C=C/c2ccnc(n2)SCC#N)Cl 4L-039 c1ccc(cc1)S(=O)(=O)C(/C=N/OCc2ccccc2Br)[N+](=O)[O-] 4L-040 COc1ccc(cc1)/C=C/c2ccnc(n2)SCc3c(cccc3Cl)Cl 4L-041 COc1ccc(cc1)/C=C/c2ccnc(n2)SCC#N 4L-042 c1cc(c(cc1Cl)Cl)/C=C/c2ccnc(n2)[S-].[K+] 4L-043 COc1ccc(cc1)/C=C/c2ccnc(n2)SCCC#N 4L-044 c1cc(c(c(c1)Cl)CSc2nccc(n2)/C=C/c3cccs3)Cl 4L-045 c1cc(sc1)/C=C/c2ccnc(n2)SCC#N 4L-046 c1cc(sc1)/C=C/c2ccnc(n2)Sc3c(cc(cn3)C(F)(F)F)Cl 4L-048 c1cc(c(cc1Cl)Cl)/C=C/c2ccnc(n2)SCC#N 4L-049 c1ccc(cc1)NC(=O)OCc2cccnc2Sc3ccc(cc3)Cl 4L-301S c1cc(c(nc1)Sc2ccc(cc2)Cl)COC(=O)Nc3ccc(cc3)Cl 4L-302S c1cscc1C(C(=O)O)N 4L-303S CC(=O)Nc1cc(c(cc1Cl)Cl)O 4L-304S c1ccc(cc1)/C=C/NC(=O)OCc2ccccc2Cl 4L-305S Cc1ccc(cc1)NC(=O)N/C=C/c2ccccc2 4L-306S COc1ccc(cc1)NC(=O)N/C=C/c2ccccc2 4L-307S c1ccc(cc1)/C=C/NC(=O)Nc2ccc(cc2)Cl 4L-308S c1ccc(cc1)/C=C\NC(=O)NCc2ccc(cc2)Cl 4L-309S c1ccc(cc1)/C=C\NC(=O)NCc2ccc(cc2Cl)Cl 4L-310S CC(=O)Nc1cc(c(cc1Cl)Cl)OC 4L-311S c1cc(sc1)C(C(=O)O)N 4L-313S c1cc(c(nc1)Sc2ccc(cc2)Cl)COC(=O)Nc3cc(cc(c3)Cl)Cl 4L-314S CC(C)NC(=O)OCc1cccnc1Sc2ccc(cc2)Cl 4L-315S c1cc(c(nc1)Sc2ccc(cc2)Cl)COC(=O)NC3CCCCC3 4L-316S Cc1ccccc1NC(=O)OCc2cccnc2Sc3ccc(cc3Cl)Cl 4L-317S COc1ccc(cc1)COC(=O)N/C=C/c2ccc(c(c2)Cl)Cl 4L-321S c1cc(ccc1NC(=O)N/C=C/c2ccc(c(c2)Cl)Cl)Cl 4L-323S CN(C)/C=C/1\C(=O)OC(=N1)c2ccccc2 4L-326S CC(=O)/C=N/Nc1ccccc1 4L-327S COC(=O)c1nc(on1)c2ccccc2 4L-330S c1cc(c(nc1)Sc2ccc(cc2Cl)Cl)COC(=O)Nc3ccc(cc3)Cl 4L-331S c1ccc(c(c1)Sc2c(cccn2)COC(=O)Nc3cccc(c3)C(F)(F)F)Cl 4L-332S Cc1ccc(cc1)/C=C/NC(=O)NCc2cccc(c2)Cl 4L-336S Cc1ccc(cc1)/C=C/NC(=O)OCc2ccc(cc2)OC 4L-340S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)C 4L-342S c1ccc(cc1)Sc2c(cccn2)COC(=O)Nc3cccc(c3)C(F)(F)F 4L-344S Cc1ccccc1NC(=O)OCc2cccnc2Sc3ccccc3 4L-345S COc1cc(c(cc1Cl)Cl)N 4L-348S c1cc(ccc1C(C(=O)O)N)C(F)(F)F 4L-350S CC(C)Oc1cc(c(cc1Cl)Cl)N 4L-351S Cc1ccc(cc1)Sc2cc(nc(n2)C)CSc3ccc(cc3)Cl 4L-352S Cc1nc(cc(n1)O)CSc2ccccc2 4L-353S Cc1nc(cc(n1)Cl)CS(=O)c2ccccc2 4L-355S CCOC(=O)Oc1ccc(cc1Cl)Cl 4L-356S Cc1nc(cc(n1)NC)CSc2ccc(cc2)Cl 4L-358S Cc1nc(cc(n1)N(C)C)CSc2ccc(cc2)Cl 4L-359S CCOC(=O)Oc1cc(c(cc1Cl)Cl)[N+](=O)[O-] 4L-360S Cc1nc(cc(n1)NCc2ccccc2OC)CSc3ccc(cc3)Cl 4L-361S c1c(c(cc(c1O)Cl)Cl)[N+](=O)[O-] 4L-362S Cc1ccc(cc1)COc2cc(nc(n2)C)CSc3ccccc3 4L-363S Cc1nc(cc(n1)OCc2ccc(cc2)Cl)CSc3ccccc3 4L-364S Cc1nc(cc(n1)OCc2ccc(cc2Cl)Cl)CSc3ccccc3 4L-365S COc1ccccc1CNC(=O)N/C=C/c2ccccc2Cl 4L-367S c1ccc(c(c1)/C=C/NC(=O)NCc2cccc(c2)Cl)Cl 4L-368S c1ccc(c(c1)/C=C/NC(=O)NCc2ccc(cc2)Cl)Cl 4L-369S Cc1nc(cc(n1)N2CCOCC2)CS(=O)c3ccccc3 4L-371S Cc1nc(cc(n1)NCc2ccc(cc2Cl)Cl)CS(=O)c3ccccc3 4L-372S COCCOc1cc(c(cc1Cl)Cl)N 4L-373S Cc1nc(cc(n1)Sc2ccc(cc2)Cl)CSc3ccc(cc3)Cl 4L-374S Cc1nc(cc(n1)Sc2ccc(cc2Cl)Cl)CSc3ccc(cc3)Cl 4L-375S CCOC(=O)COc1cc(c(cc1Cl)Cl)[N+](=O)[O-] 4L-376S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)[N+](=O)[O-] 4L-377S Cc1ccc(cc1)NC(=O)N/C=C/c2ccco2 4L-378S Cc1ccc(cc1C)NC(=O)N/C=C/c2ccco2 4L-379S c1cc(ncc1[N+](=O)[O-])NN 4L-380S Cc1nc(cc(n1)Sc2c(cccc2Cl)Cl)CSc3ccc(cc3)Cl 4L-382S Cc1nc(cc(n1)N2CCOCC2)CS(=O)(=O)c3ccccc3 4L-383S Cc1nc(cc(n1)N2CCCCC2)CS(=O)(=O)c3ccccc3 4L-384S Cc1nc(cc(n1)Cl)CS(=O)(=O)c2ccc(cc2)Cl 4L-386S CN(C)/C=C/1\C(=O)OC(=N1)c2ccc(cc2)F 4L-387S Cc1ccc(c(c1)C)NC(=O)N/C=C/c2ccco2 4L-390S Cc1nc(cc(n1)N2CCN(CC2)C)CS(=O)(=O)c3ccccc3 4L-392S Cc1nc(cc(n1)NCc2ccc(cc2)Cl)CSc3ccc(cc3)Cl 4L-393S Cc1nc(cc(n1)NCc2cccc(c2)OC)CSc3ccc(cc3)Cl 4L-394S Cc1nc(cc(n1)N2CCOCC2)CS(=O)c3ccc(cc3)Cl 4L-395S COCc1cc(nc(n1)c2ccccc2)O 4L-511S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3ccc(cc3)OC 4L-513S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3ccc(cc3)Br 4L-514S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3ccc(cc3)Cl 4L-515S COCc1cc(nc(n1)c2ccccc2)Cl 4L-516S COCc1cc(nc(n1)c2ccccc2)N3CCOCC3 4L-517S CNc1cc(nc(n1)c2ccccc2)COC 4L-518S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3cccc(c3Cl)Cl 4L-519S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3c(cccc3Cl)Cl 4L-520S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3cc(ccc3Cl)Cl 4L-521S Cc1ccc(cc1)SCc2c(nn(c2Cl)C)CSc3ccc(cc3)C 4L-522S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3ccc(cc3)F 4L-523S CSc1cc(n(c(=O)c1C#N)Cc2c(cccc2Cl)Cl)c3ccccc3 4L-525S CSc1cc(n(c(=O)c1C#N)Cc2ccc(cc2Cl)Cl)c3ccccc3 4L-526S COCc1cc(nc(n1)c2ccccc2)NCC=C 4L-527S COCc1cc(nc(n1)c2ccccc2)N3CCCC3 4L-528S COCc1cc(nc(n1)c2ccccc2)N3CCCCC3 4L-529S CC1CN(CC(O1)C)c2cc(nc(n2)c3ccccc3)COC 4L-530S CSc1cc(n(c(=O)c1C#N)Cc2ccc(cc2)Cl)c3ccccc3 4L-531S CSc1cc(n(c(=O)c1C#N)Cc2ccccc2)c3ccccc3 4L-532S Cc1ccc(cc1)Cn2c(cc(c(c2=O)C#N)SC)c3ccccc3 4L-533S CSc1cc(n(c(=O)c1C#N)Cc2cccc(c2)C(F)(F)F)c3ccccc3 4L-534S CC(C)(C)c1ccc(cc1)Cn2c(cc(c(c2=O)C#N)SC)c3ccccc3 4L-535S Cn1c(cc(c(c1=O)C#N)SC)c2ccccc2 4L-536S CCOC(=O)Cn1c(cc(c(c1=O)C#N)SC)c2ccccc2 4L-537S CSc1cc(n(c(=O)c1C#N)CC=C)c2ccccc2 4L-538S CCCn1c(cc(c(c1=O)C#N)SC)c2ccccc2 4L-539S Cc1ccc(cc1)SCc2c(c(n(n2)C)Cl)CSc3ccccc3Cl 4L-541S CSc1cc([nH]c(=O)c1C#N)c2ccc(cc2)Cl 4L-544S Cn1c(c(c(n1)CSc2ccccc2)CSc3c(cccc3Cl)Cl)Cl 4L-547S Cn1c(c(c(n1)CSc2ccccc2)CSc3cccc(c3Cl)Cl)Cl 4L-548S Cn1c(c(c(n1)CSc2ccccc2)CSc3ccc(cc3)OC)Cl 4L-549S CS(=O)(=O)Cc1cc(nc(n1)c2ccccc2)N3CCOCC3 4L-550S CS(=O)Cc1cc(nc(n1)c2ccncc2)NC3CCCCC3 4L-551S COCc1cc(nc(n1)c2cccnc2)O 4L-555S COCc1cc(nc(n1)c2cccnc2)Cl 4L-556S COCc1cc(nc(n1)c2ccccc2)N3CCSCC3 4L-557S COCc1cc(nc(n1)c2ccccc2)N3CCN(CC3)c4ccccc4F 4L-558S CC(C)Nc1cc(nc(n1)c2ccccc2)COC 4L-559S COCc1cc(nc(n1)c2ccccc2)N3CCN(CC3)c4cccc(c4)Cl 4L-560S COCc1cc(nc(n1)c2ccccc2)Sc3cccc(c3Cl)Cl 4L-561S COCc1cc(nc(n1)c2ccccc2)Sc3c(cccc3Cl)Cl 4L-562S COCc1cc(nc(n1)c2ccccc2)Sc3ccc(cc3Cl)Cl 4L-563S COCc1cc(nc(n1)c2ccccc2)Sc3ccc(cc3)Br 4L-564S CCCNc1cc(nc(n1)c2ccccc2)COC 4L-565S COCc1cc(nc(n1)c2ccccc2)NCc3ccccc3 4L-566S c1ccc(cc1)c2nc(cc(n2)O)CSCc3ccc(cc3)Cl 4L-568S CSc1cc(n(c(=O)c1C#N)Cc2ccc(cc2)F)c3ccc(cc3)Cl 4L-569S CSc1cc(n(c(=O)c1C#N)Cc2ccc(cc2)Cl)c3ccc(cc3)Cl 4L-570S CSc1cc(n(c(=O)c1C#N)Cc2c(cccc2Cl)Cl)c3ccc(cc3)Cl 4L-571S CSc1cc(n(c(=O)c1C#N)Cc2cccc(c2)Cl)c3ccc(cc3)Cl 4L-573S Cc1ccc(cc1)Cn2c(cc(c(c2=O)C#N)SC)c3ccc(cc3)Cl 4L-574S Cc1ccccc1Cn2c(cc(c(c2=O)C#N)SC)c3ccc(cc3)Cl 4L-575S CSc1cc(n(c(=O)c1C#N)Cc2ccccc2)c3ccc(cc3)Cl 4L-576S CCn1c(cc(c(c1=O)C#N)SC)c2ccc(cc2)Cl 4L-577S CSc1cc(n(c(=O)c1C#N)Cc2ccc(c(c2)Cl)Cl)c3ccc(cc3)Cl 4L-578S CCCn1c(cc(c(c1=O)C#N)SC)c2ccc(cc2)Cl 4L-579S CSc1cc(n(c(=O)c1C#N)CC=C)c2ccc(cc2)Cl 4L-580S CCOC(=O)Cn1c(cc(c(c1=O)C#N)SC)c2ccc(cc2)Cl 4L-581S CSc1cc(n(c(=O)c1C#N)Cc2cccc(c2)F)c3ccccc3 4L-582S CSc1cc(n(c(=O)c1C#N)Cc2ccccc2Cl)c3ccccc3 4L-583S Cc1cccc(c1)Cn2c(cc(c(c2=O)C#N)SC)c3ccccc3 4L-584S CS(=O)(=O)Cc1cc(nc(n1)c2ccccn2)NCC=C 4L-589S CS(=O)(=O)Cc1cc(nc(n1)c2ccccc2)Oc3ccc(cc3)Cl 4L-590S COc1cc(nc(n1)c2ccccc2)CS(=O)(=O)C 4L-591S CSc1cc(nc(n1)c2ccccc2)CS(=O)(=O)C 4L-592S CS(=O)(=O)Cc1cc(nc(n1)c2ccccc2)N3CCCC3 4L-594S CS(=O)(=O)Cc1cc(nc(n1)c2ccccc2)NCC=C 4L-595S Cn1c(c(c(n1)CSc2ccccc2)CSc3ccc(cc3)Br)Cl 4L-596S c1ccc(cc1)c2nc(cc(n2)Cl)CSCc3ccc(cc3)Cl 4L-603S c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])CO)Cl 4L-604S COCc1cc(nc(n1)c2ccccc2)Sc3ccc(cc3)OC 4L-606S COCc1cc(nc(n1)c2ccccc2)SCc3ccc(cc3Cl)Cl 4L-607S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)COC 4L-608S c1cc(cc(c1)Cl)NC(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl 4L-610S c1cc(cc(c1)Cl)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl 4L-612S c1ccc(cc1)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccccc3 4L-613S c1ccc(cc1)NC(=O)OCc2ccc(cc2[N+](=O)[O-])Oc3ccccc3 4L-614S COC(=O)c1ccccc1S(=O)C 4L-615S COC(=O)c1ccccc1S(=O)(=O)C 4L-617S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3)Br)CSCc4ccc(cc4)Cl 4L-619S Cc1cc(=O)n(c(n1)/N=C/N(C)C)Cc2ccc(cc2)[N+](=O)[O-] 4L-900 c1ccc2c(c1)C(=O)N(C2=O)OCc3c(cccc3Cl)Cl 4L-901 Cn1c(=O)c(cn(c1=O)CC2CC(=NO2)C(=O)NN)C#N 4L-902 c1c(cnc(c1Cl)n2c(=O)c(c(cn2)N3CCOCC3)Cl)C(F)(F)F 4L-903 Cc1ccc(cc1)N2C(=O)NC3(N2)CCN(CC3)C(=O)N 4L-904 CCOC(=O)C/C(=N/CC/N=C(/C)\CC(=O)OCC)/C.O 4L-905 Cn1c(=O)c(cn(c1=O)CC2CC(N(O2)C)c3ccccc3)C#N 4L-906 CCOC(=O)c1c(n(c2c1cc(c3c2cccc3)O)CCn4c(c(c5c4c6ccccc6c(c5)O)C(=O)OCC)C)C 4L-907 CCOC(=O)c1c(n(c2c1cc(c3c2cccc3)OC)CCn4c(c(c5c4c6ccccc6c(c5)OC)C(=O)OCC)C)C 4L-908 Cc1cc(=O)n(c(n1)N)Cc2ccc(cc2)[N+](=O)[O-] 4L-909 c1ccn(c1)c2c(c3c(s2)CN(CC3)c4cccc(n4)F)C#N 4L-910 COc1ccc(cc1)n2c(=O)c(c(cn2)N3CCc4c(sc(c4C#N)n5cccc5)C3)Cl 4L-911 CCOC(=O)CNC(=S)NCC(c1ccc2ccccc2c1)O 4L-913 Cn1c(=O)c(cn(c1=O)c2cccnc2Cl)C(=O)/C=C/N(C)C 4L-914 C/C(=N\O)/c1cnc(s1)c2ccc(cc2)Cl 4M-001 c1ccc(cc1)C(=O)/C(=N/Nc2cccc(c2)C(F)(F)F)/C=O 4M-002 CO/N=C/CC(=O)c1cnc(s1)c2ccc(cc2)Cl 4M-003 c1ccc(c(c1)CO/N=C/CC(=O)c2cnc(s2)c3ccc(cc3)Cl)Br 4M-004 c1ccc(c(c1)CO/N=C/CC(=O)c2cnc(s2)c3ccc(cc3)Cl)F 4M-005 c1cc(ccc1c2ncc(s2)C(=O)C/C=N/OCc3ccc(cc3Cl)F)Cl 4M-006 c1cc(cc(c1)OCCO/N=C/CC(=O)c2cnc(s2)c3ccc(cc3)Cl)C(F)(F)F 4M-007 Cc1ccc(cc1)c2c(cnc(n2)C)/N=N\c3cc(cc(c3)Cl)Cl 4M-008 c1ccc(cc1)N/N=C(\C=N\N)/C(=O)c2cccs2 4M-009 c1ccc(cc1)C(=O)/C(=N/Nc2ccccc2Cl)/C=O 4M-010 COc1ccc(cc1)N/N=C(\C=O)/C(=O)c2ccccc2 4M-011 c1cc(ccc1c2ncc(s2)c3ccno3)Cl 4M-012 c1cc(ccc1c2ncc(s2)c3cc[nH]n3)Cl 4M-013 c1ccc(cc1)N/N=C(\C=N\N)/C(=O)c2ccco2 4M-014 c1ccc(cc1)C(=O)/C(=N/Nc2ccccc2)/C=N/O 4M-015 c1ccc(cc1)c2ncc(s2)c3ccn(n3)C(=O)c4ccc(cc4)F 4M-016 Cc1ccc(cc1)C(=O)n2ccc(n2)c3cnc(s3)c4ccccc4 4M-017 COc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3cnc(s3)c4ccccc4 4M-018 c1ccc(cc1)c2c(cnc(n2)c3ccccc3)/N=N\c4ccccc4 4M-019 c1cc(ccc1c2ncc(s2)c3ccnc(n3)N)Cl 4M-020 c1ccc(cc1)c2ncc(s2)c3ccn(n3)S(=O)(=O)c4cccs4 4M-021 c1ccc(cc1)c2ncc(s2)c3ccn(n3)S(=O)(=O)c4ccccc4 4M-022 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)OC)/C=N/O 4M-023 COc1ccc(cc1)c2c(cnc(n2)c3ccccc3)/N=N\c4ccc(cc4)OC 4M-024 COc1ccc(cc1)N/N=C(\C=N\O)/C(=O)c2ccccc2 4M-025 COc1ccc(cc1)/N=N\c2cnc(nc2c3ccccc3)c4ccccc4 4M-026 COc1ccc(cc1)/N=N\c2cnc(nc2c3ccccc3)c4ccncc4 4M-027 COc1ccc(cc1)c2c(cnc(n2)c3ccccn3)/N=N\c4ccc(cc4)OC 4M-028 c1ccc(cc1)c2ncc(s2)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Oc5c(cc(cn5)C(F)(F)F)Cl 4M-029 Cc1cccc(c1)/N=N\c2cnc(nc2c3cccs3)c4ccncc4 4M-030 c1ccc(cc1)c2ncc(s2)c3ccn(n3)c4c(cc(cn4)C(F)(F)F)Cl 4M-031 Cc1cccc(c1)/N=N\c2cnc(nc2c3cccs3)c4ccccn4 4M-032 Cc1ncc(c(n1)c2ccccc2)/N=N\c3ccccc3Cl 4M-033 c1ccc(cc1)c2c(cnc(n2)c3ccncc3)/N=N\c4ccccc4Cl 4M-034 c1ccc(cc1)c2ncc(s2)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl 4M-035 Cc1ccc(cc1)Cn2ccc(n2)c3cnc(s3)c4ccccc4 4M-036 c1ccc(cc1)c2c(cnc(n2)N)/N=N\c3ccccc3Cl 4M-037 c1ccc(cc1)c2c(cnc(n2)c3ccccc3)/N=N\c4cccc(c4)C(F)(F)F 4M-038 c1ccc(cc1)c2c(cnc(n2)c3cccnc3)/N=N\c4cccc(c4)C(F)(F)F 4M-039 c1ccc(cc1)c2ncc(c(n2)c3ccco3)/N=N\c4ccccc4 4M-040 c1cc(ccc1C(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/C=N/O)Br 4M-041 c1ccc(cc1)c2ncc(s2)c3ccn(n3)S(=O)(=O)c4ccc(cc4)F 4M-042 c1ccc(cc1)c2ncc(s2)c3ccn(n3)c4c(cccn4)[N+](=O)[O-] 4M-043 c1cc(cnc1)c2ncc(c(n2)c3ccco3)/N=N\c4ccc(cc4)Cl 4M-044 c1cc(cnc1)c2ncc(c(n2)c3cccs3)/N=N\c4ccc(cc4)Cl 4M-045 Cc1cccc(c1)/N=N\c2cnc(nc2c3ccc(cc3)Br)c4cccnc4 4M-046 c1ccc(cc1)c2ncc(s2)c3ccn(n3)CCOc4ccc(cc4Cl)Cl 4M-047 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/C=N/O)Br 4M-048 c1ccc(cc1)c2ncc(s2)c3ccn(n3)c4cccc(n4)Cl 4M-049 c1ccc(cc1)c2c(cnc(n2)c3ccncc3)/N=N\c4cccc(c4)C(F)(F)F 4M-050 c1cc(ccc1c2c(cnc(n2)N)/N=N\c3ccc(cc3)C(F)(F)F)Br 4M-051 c1ccc(cc1)N/N=C(/C=N/O)\C(=O)c2ccc(cc2Cl)Cl 4M-052 Cc1ncc(c(n1)c2ccco2)/N=N\c3ccc(cc3)Cl 4M-053 c1ccc(cc1)c2c(cnc(n2)N)/N=N\c3cccc(c3)C(F)(F)F 4M-054 c1ccc(cc1)c2ncc(c(n2)c3ccc(cc3Cl)Cl)/N=N\c4ccccc4 4M-055 c1ccc(cc1)c2ncc(s2)c3ccn(n3)Cc4ccc(cc4)F 4M-056 c1ccc(cc1)Cn2ccc(n2)c3cnc(s3)c4ccccc4 4M-057 COc1ccc(cc1)C(=O)n2ccc(n2)c3cnc(s3)c4ccccc4 4M-058 c1ccc(cc1)c2ncc(s2)c3ccn(n3)C(=O)c4ccccc4 4M-059 Cc1ccc(cc1)c2c(cnc(n2)c3cccnc3)/N=N\c4cc(cc(c4)Cl)Cl 4M-060 c1ccc(cc1)/N=N\c2cnc(nc2c3ccc(cc3Cl)Cl)N 4M-061 c1ccc(cc1)/N=N\c2cnc(nc2c3ccc(cc3Cl)Cl)c4cccnc4 4M-062 c1ccc(cc1)/C(=N/O)/COc2ccccc2[N+](=O)[O-] 4M-301S CC(C)(C)C(=O)COc1ccccc1[N+](=O)[O-] 4M-302S Cc1ccc(cc1)Sc2cnccc2C#N 4M-303S Cc1ccc(cc1)S(=O)c2cnccc2C#N 4M-304S c1cc(ccc1Sc2cnccc2C#N)Cl 4M-307S c1cc(ccc1S(=O)c2cnccc2C#N)Cl 4M-308S CC(C)(C)/C(=N/O)/COc1ccccc1[N+](=O)[O-] 4M-311S Cc1ccc2c(c1)/C(=N\c3ccc(cc3)F)/C(=O)N2Cc4c(cccc4Cl)Cl 4M-312S Cc1ccc2c(c1)/C(=N\c3ccc(cc3)Cl)/C(=O)N2Cc4c(cccc4Cl)Cl 4M-313S Cc1ccc2c(c1)/C(=N\c3ccc(cc3)OC)/C(=O)N2Cc4c(cccc4Cl)Cl 4M-314S c1ccc(cc1)/C(=N\OCc2ccc(cc2Cl)Cl)/COc3ccccc3[N+](=O)[O-] 4M-315S CC(C)(C)/C(=N/OCc1ccc(cc1Cl)Cl)/COc2ccccc2[N+](=O)[O-] 4M-316S c1ccc(cc1)/C(=N\OC(=O)Nc2cccc(c2)Cl)/COc3ccccc3[N+](=O)[O-] 4M-317S CCOC(=O)c1cn(c2cc(ccc2c1=O)F)Cc3ccc(cc3)C 4M-321S CC1COc2ccccc2N1S(=O)(=O)c3ccc(cc3)OC 4M-323S CC1COc2ccccc2N1S(=O)(=O)c3ccc(cc3)Cl 4M-324S CC1COc2ccccc2N1S(=O)(=O)c3cc(ccc3Cl)Cl 4M-325S CC(C)(C)C1COc2ccccc2N1 4M-326S Cc1ccc(cc1)C(=O)N2c3ccccc3OCC2C 4M-327S CC1COc2ccccc2N1C(=O)c3cccnc3Cl 4M-328S CC1COc2ccccc2N1C(=O)c3ccccc3Cl 4M-329S Cn1c2c(cc(s2)c3nnc(o3)c4ccccc4)c(n1)C(F)(F)F 4M-330S Cn1c2c(cc(s2)c3nnc(n3C)S)c(n1)C(F)(F)F 4M-331S Cc1ccc(cc1)Cn2cc(c(=O)c3c2cc(cc3)F)C(=O)NN 4M-333S c1ccc(c(c1)CCC(=O)O)[N+](=O)[O-] 4M-336S CC1COc2ccccc2N1C(=O)c3ccc(cc3)Cl 4M-337S Cc1cccc(c1NC(=O)O/N=C(/COc2ccccc2[N+](=O)[O-])\C(C)(C)C)C 4M-338S Cc1cccc(c1NC(=O)O/N=C(\COc2ccccc2[N+](=O)[O-])/c3ccccc3)C 4M-339S Cc1ccc(cc1)c2nnc(o2)c3cc4c(nn(c4s3)C)C(F)(F)F 4M-340S Cn1c2c(cc(s2)c3nnc(o3)c4cccc(c4)OC)c(n1)C(F)(F)F 4M-341S CC(C)c1nnc(o1)c2cc3c(nn(c3s2)C)C(F)(F)F 4M-342S Cn1c2c(cc(s2)c3nnc(n3C)SCC=C)c(n1)C(F)(F)F 4M-347S Cn1c2c(cc(s2)c3nnc(n3C)SCC#C)c(n1)C(F)(F)F 4M-348S CCCCSc1nnc(n1C)c2cc3c(nn(c3s2)C)C(F)(F)F 4M-349S CC1COc2ccccc2N1C(=O)c3ccc(cc3)F 4M-350S CC1COc2ccccc2N1C(=O)c3ccc(cc3Cl)Cl 4M-351S CC(C)(C)C1COc2ccccc2N1S(=O)(=O)c3ccc(cc3)OC 4M-352S CC(C)(C)C1COc2ccccc2N1S(=O)(=O)c3ccc(cc3)Cl 4M-354S Cc1ccc(cc1)S(=O)(=O)N2c3ccccc3OCC2C(C)(C)C 4M-355S CC(C)(C)C1COc2ccccc2N1C(=O)c3ccccc3Cl 4M-356S Cc1ccc(cc1)C(=O)N2c3ccccc3OCC2c4ccccc4 4M-358S CCOC(=O)c1[nH]c(nn1)c2ccccc2 4M-441S c1ccc(cc1)C(=O)Nc2ccc(oc2=O)c3ccc(cc3)Cl 4M-507S c1cc(ccc1C(=O)C(F)(F)F)N 4M-508S Cc1nc(cc(n1)NCc2ccc(cc2)Cl)COC 4M-510S Cc1nc(cc(n1)N2CCOCC2)COC 4M-511S Cc1nc(cc(n1)NCC=C)COC 4M-512S Cc1nc(cc(n1)SCc2ccc(cc2)Cl)COC 4M-513S Cc1nc(cc(n1)Sc2ccc(cc2)Cl)COC 4M-514S Cc1nc(cc(n1)SC2CCCCC2)COC 4M-515S Cc1ccc(cc1)c2c(c3ccccc3[nH]c2=O)C(=O)O 4M-516S c1ccc(cc1)C(=O)Nc2ccc(oc2=O)c3ccc(cc3)Br 4M-522S c1cc(ccc1c2ccc(c(=O)o2)NC(=O)c3ccc(cc3)Cl)Br 4M-523S c1ccc(cc1)c2ccc(c(=O)o2)NC(=O)c3ccc(cc3)Cl 4M-524S c1cc(ccc1c2ccc(c(=O)o2)NC(=O)c3ccc(cc3)Cl)Cl 4M-525S c1ccc(cc1)c2ccc(c(=O)o2)NC(=O)c3ccccc3 4M-526S Cc1nc(cc(n1)Oc2ccc(cc2)Cl)COC 4M-527S Cc1nc(cc(n1)S(=O)c2ccc(cc2)Cl)COC 4M-529S Cc1nc(cc(n1)S(=O)(=O)c2ccc(cc2)Cl)COC 4M-530S Cc1nc(cc(n1)S(=O)(=O)C2CCCCC2)COC 4M-531S COCc1cc(nc(n1)S(=O)Cc2ccc(cc2)Cl)N3CCOCC3 4M-532S COCc1cc(nc(n1)SC)Sc2ccc(cc2)Cl 4M-533S COCc1cc(nc(n1)SC)Oc2cccc(c2)C(F)(F)F 4M-534S COCc1cc(nc(n1)SCc2ccc(cc2)Cl)N3CCCC3 4M-535S COCc1cc(nc(n1)SCc2ccc(cc2)Cl)Sc3ccccc3C(=O)OC 4M-536S C=CCNC(=O)c1cc(ccn1)Cl 4M-537S CNC(=O)c1cc(ccn1)Cl 4M-538S COC(=O)c1cc(ccn1)Sc2ccc(cc2)Br 4M-543S Cc1ccc(cc1)c2nnc(o2)c3c(nn(c3Cl)C)c4ccccc4 4M-545S Cn1c(c(c(n1)c2ccccc2)c3nnc(o3)c4ccccc4)Cl 4M-547S Cn1c(c(c(n1)c2ccccc2)c3nnc(o3)c4ccc(cc4)Cl)Cl 4M-549S Cn1c(c(c(n1)c2ccccc2)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl 4M-553S Cn1c(c(c(n1)c2ccccc2)C(=O)Nc3ccc(cc3)Cl)Cl 4M-554S COCc1cc(nc(n1)SC)N2CCOCC2 4M-556S COCc1cc(nc(n1)SC)N2CCCC2 4M-557S COCc1cc(nc(n1)SCc2ccc(cc2)Cl)Oc3ccc(cc3)Cl 4M-559S CSc1ccccc1C#N 4M-561S COC(=O)c1cc(ccn1)Sc2cccc(c2Cl)Cl 4M-562S COC(=O)c1cc(ccn1)Sc2c(cccc2Cl)Cl 4M-563S Cn1c(cc(n1)OC(=O)Nc2ccccc2)C(F)(F)F 4M-568S Cn1c(cc(n1)OCC(=O)N2CCOCC2)C(F)(F)F 4M-571S c1cc(ccc1n2c(=O)c(c(cn2)Br)Br)F 4M-584S CCOC(=O)C1=C(NC2=C(C1c3ccccc3)C(=O)CCC2)C 4M-701 CCO.Cc1cc2c(cc1C)NC3=C(C(N2)c4ccccc4)C(=O)CCC3 4M-702 c1ccc(cc1)c2nc3n(n2)C(=O)C(=C(C3)N)C#N 4M-703 Cc1ccc(cc1)C2C3=C(CCCC3=O)Nc4cc(c(cc4N2)C)C 4M-704 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccc(cc4)[N+](=O)[O-])C(=O)CCC3 4M-705 CN(C)c1nc(n(n1)Cc2ccc(cc2)Cl)N(C)C 4M-708 CCO.Cc1cc2c(cc1C)NC3=C(C(N2)c4cccc(c4)Br)C(=O)CCC3 4M-709 Cc1ccc(cc1)Cn2c(nc(n2)N(C)C)N(C)C 4M-710 CN(C)c1nc(n(n1)Cc2ccc(cc2)Br)N(C)C 4M-712 Cc1ccc(cc1)n2nc(c(n2)C(=O)O)C 4M-713 CC1(CN(C1=O)C(Cc2ccccc2)C(=O)N)C 4M-714 CN(C)c1nc(n(n1)Cc2c(cccc2Cl)Cl)N(C)C 4M-715 CN(C)c1nc(n(n1)Cc2ccc(cc2)F)N(C)C 4M-716 CCOC(=O)c1c(nc2c(c1c3ccccc3)C(=O)CCC2)C 4M-717 CCOC(=O)c1cnc2ccc(cc2c1NCc3ccc(cc3)Cl)C(F)(F)F 4M-723 CCOC(=O)c1cnc2ccc(cc2c1N3CCN(CC3)c4ccc(cc4)Cl)C(F)(F)F 4M-724 Cc1nnc2n1nc(cc2)N3CCOCC3 4M-726 CCO.Cc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)Nc4cc(c(cc4N2)C)C 4M-727 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccc(cc4)OCc5ccccc5)C(=O)CC(C3)(C)C 4M-728 C/C(=N\Nc1ccc(cc1)F)/C(=N/O)/C(=O)Nc2ccccc2 4M-729 C/C(=N\Nc1ccc(cc1)OC(F)(F)F)/C(=N/O)/C(=O)Nc2ccccc2 4M-730 c1cc(nn2c1nnc2C(F)(F)F)Cl 4M-731 c1cc(nn2c1nnc2C(F)(F)F)N3CCOCC3 4M-732 CCOC(=O)NNc1c(cc(cn1)C(F)(F)F)Cl 4M-733 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccc(cc4)OC)C(=O)CC(C3)(C)C 4M-734 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccc(cc4)C(C)C)C(=O)CC(C3)(C)C 4M-735 C/C(=N\Nc1ccc(cc1)OC)/C(=N/O)/C(=O)Nc2ccccc2 4M-737 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccccc4C(F)(F)F)C(=O)CC(C3)(C)C 4M-739 c1ccc(cc1)n2c(=O)cc(c(n2)C#N)Oc3ccccc3 4M-740 Cc1cc2c(cc1C)NC3=C(C(N2)c4cccc(c4)O)C(=O)CC(C3)(C)C 4M-743 c1ccc(cc1)N2CCN(CC2)c3ccc4nnc(n4n3)C(F)(F)F 4M-744 CN1C(=O)c2ccccc2/C(=N\O)/C1=O 4M-745 Cc1c(nn(n1)c2ccc(cc2)F)C(=O)O 4M-746 Cc1cc2c(cc1C)NC3=C(C(N2)c4c5ccccc5ccc4O)C(=O)CC(C3)(C)C 4M-748 Cc1ccsc1C2C3=C(CC(CC3=O)(C)C)Nc4cc(c(cc4N2)C)C 4M-749 c1cc(nn2c1nnc2C(F)(F)F)N3CCCC3 4M-750 C/C(=N\Nc1cccc(n1)F)/C(=N/O)/C(=O)Nc2ccccc2 4M-751 c1ccc(cc1)C(=O)NNc2ccc(nn2)Cl 4M-752 CC(=O)Oc1nnc2n1cc(cc2Cl)C(F)(F)F 4M-753 COc1ccc(cc1)N2CCN(CC2)c3ccc4nnc(n4n3)C(F)(F)F 4M-754 CN1CCN(CC1)c2ccc3nnc(n3n2)C(F)(F)F 4M-757 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccccc4OC)C(=O)CC(C3)(C)C 4M-758 c1c(cnc(c1Cl)NNC(=O)C(F)(F)F)C(F)(F)F 4M-761 CC1(CN(C1=O)C(Cc2ccccc2)C(=O)N/C=N/OCc3ccc(cc3Cl)F)C 4M-762 c1cc(nn2c1nnc2C(F)(F)F)N3CCNCC3 4M-764 COc1ccc(cc1)Oc2ccc3nnc(n3n2)C(F)(F)F 4M-765 c1cc(cc(c1)NC(=O)OCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 4M-900 c1cc(ccc1N2CCN(CC2)CCO)[N+](=O)[O-] 4M-901 c1ccc(cc1)NC(=O)OCCN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 4M-902 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)CCO 4M-903 c1cc(ccc1C(=O)OCCN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])F 4M-904 c1cc(cc(c1)Cl)C(=O)OCCN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 4M-905 c1cc(sc1)C(=O)OCCN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F 4M-907 c1cc(cc(c1)C(F)(F)F)C(=O)OCCN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F 4M-908 c1cc(cc(c1)NC(=O)OCCN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F 4M-909 c1cc(ccc1C(=O)OCCN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)F 4M-910 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2ccc(cc2)F 4M-912 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC#C)S(=O)(=O)c2ccc(cc2)F 4M-913 c1ccc(cc1)c2c3cc(ccc3[nH]c2c4cccs4)Cl 4M-914 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2cccs2 4M-915 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)CCOC(=O)c3ccc(cc3Cl)Cl 4M-916 CC1=C(CCC(=O)N1Cc2ccc(cc2)F)C#N 4M-917 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2ccc3ccccc3c2 4M-918 CN(c1c(cc(cn1)C(F)(F)F)Cl)N(CC#C)S(=O)(=O)c2ccc3ccccc3c2 4M-919 CC1=C(CCC(=O)N1Cc2ccc(cc2Cl)Cl)C#N 4M-920 Cc1cc(c(c(c1)C)CN2C(=C(CCC2=O)C#N)C)C 4M-921 CC1=C(CCC(=O)N1Cc2c(cccc2Cl)F)C#N 4M-922 CC1=C(CCC(=O)N1Cc2ccc(cc2)Br)C#N 4M-923 CC(=O)c1cc(on1)CN(N(C)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)c3ccc4ccccc4c3 4M-924 c1cc(ccc1C(F)(F)F)NS(=O)(=O)c2ccc(cc2)Cl 4M-926 CCOC(=O)c1c(c2ccccc2n1c3c(cc(cn3)C(F)(F)F)Cl)c4ccccc4 4M-929 COc1ccc(cc1)CN2C(=O)CCC(=C2C(=O)OC)C(=O)OC 4M-931 Cc1ccc(cc1)CN/C(=C/C(=O)Nc2cccc(c2)C(F)(F)F)/C 4M-932 CC1=C(CCC(=O)N1CCOc2ccc(cc2Cl)Cl)C#N 4M-933 CC1=C(CCC(=O)N1Cc2ccc(cc2)Cl)C(=O)OC 4M-934 C/C(=C/C(=O)Nc1ccc(cc1)Cl)/NCc2ccccc2 4M-935 Cc1ccc(cc1)CN2C(=C(CCC2=O)C(=O)Nc3cccc(c3)C(F)(F)F)C 4M-936 CN(C)c1ccc(cc1)/C=N/NC(=O)c2c(c3ccccc3[nH]2)c4ccccc4 4M-938 c1ccc(cc1)c2c3ccccc3[nH]c2C(=O)N/N=C/c4ccc(cc4)[N+](=O)[O-] 4M-939 CC1=C(CCC(=O)N1Cc2ccccc2)C(=O)Nc3ccc(cc3)Cl 4M-940 C/C(=C\C(=O)Nc1ccc(cc1)OC)/NCc2ccccc2 4M-941 CC1=C(CCC(=O)N1Cc2ccccc2)C(=O)Nc3ccc(cc3)OC 4M-942 C/C(=C\C(=O)Nc1ccc(cc1Cl)Cl)/NCCNc2c(cc(cn2)C(F)(F)F)Cl 4M-943 Cc1cc(=O)c(c(n1N(C)c2c(cc(cn2)C(F)(F)F)Cl)C)C(=O)NN(C)c3c(cc(cn3)C(F)(F)F)Cl 4M-944 CC1=C(CCC(=O)N1CCNc2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3Cl)Cl 4M-945 CCOC(=O)C1=C(N(C(=O)CC1)CCN2C(=C(CCC2=O)C(=O)OCC)C)C 4M-948 Cc1cc(nc(n1)N)C(F)(F)Cl 4M-950 COc1ccc(cc1)NC(=O)Nc2ccc(cn2)I 4M-951 c1cc(ncc1I)NC(=O)CCCCl 4M-954 c1ccn(c1)c2ccc(cn2)I 4M-955 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cn2)I 4M-956 c1cc(ccc1c2cnc3n2cc(cc3)I)Cl 4M-957 c1cc(ncc1I)NC(=S)N 4M-958 CN(C)/C=N/C(=S)Nc1ccc(cn1)I 4M-959 c1cc(ccc1c2csc(n2)Nc3ccc(cn3)I)F 4M-960 c1cc(ccc1CON/C=N/C(=S)Nc2ccc(cn2)I)Cl 4M-961 Cn1c2c(c(=O)n(c1=O)C)CCC(=O)N2 4M-962 c1cc2c(cc1C3CC3/C(=N/OCc4ccc(cc4Cl)Cl)/c5ccc(c(c5)[N+](=O)[O-])Cl)OCO2 4N-002 CC(C)(C)[C@@H](C(=O)OC)N 4N-004 Cc1ccc(cc1)C2CC2/C(=N/OCc3ccccc3F)/c4ccc(cc4)F 4N-005 Cc1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccc(cc3)C)/c4ccc(cc4)F 4N-006 Cc1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccc(cc3)OC)/c4ccc(cc4)F 4N-007 CC(C)(C)C(C(=O)OC)NC(=O)Nc1ccc(cc1)Cl 4N-008 c1ccc2c(c1)nc(c3n2ccc3)n4ccnc4 4N-009 Cc1c2ccc(nc2ccn1)Oc3ccc(cc3)NC(=O)C 4N-010 Cc1ccc(cc1)C2CC2/C(=N/OC(=O)C3CC3)/c4ccc(cc4)F 4N-011 Cc1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccc(cc3)F)/c4ccc(cc4)F 4N-012 Cc1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccco3)/c4ccc(cc4)F 4N-013 Cc1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccc(c(c3)Cl)Cl)/c4ccc(cc4)F 4N-014 c1ccc(cc1)C2CC2/C(=N/OCc3ccc(cc3)Cl)/c4ccccn4 4N-015 c1cc(ccc1C2CC2/C(=N/OCc3ccc(cc3Cl)Cl)/c4ccc(cc4)Br)Cl 4N-016 COc1ccc(cc1)C2CC2C(=O)c3ccccc3 4N-017 Cc1ccc(cc1)C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 4N-018 c1(c(c(nc(c1Cl)Cl)Cl)Cl)O 4N-019 CC(C)(C)C(C(=O)OC)NC(=O)Nc1ccccc1 4N-020 c1ccc2c(c1)nc(c3n2ccc3)n4cccn4 4N-021 COc1ccc(cc1)C(=O)/C=C/c2ccc3c(c2)OCO3 4N-022 c1ccc(cc1)C2CC2/C(=N/OCc3ccc(cc3)[N+](=O)[O-])/c4ccccn4 4N-024 c1ccc(c(c1)C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 4N-025 COc1ccc(cc1)C2CC2/C(=N/O)/c3ccccc3 4N-026 c1cc(ccc1C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)F 4N-027 CC(C)(C)C(C(=O)O)N1Cc2ccccc2C1=O 4N-029 c1ccc2c(c1)CN(C2=O)C(CC3CCCCC3)C(=O)O 4N-030 COc1ccc(cc1)C(=O)C2CC2c3ccc4c(c3)OCO4 4N-031 CC(C)(C)C(C(=O)OC)NC(=O)NC1CCCCC1 4N-032 c1ccc(cc1)C(=O)NC(=S)Nc2ccc-3c(c2)Cc4c3cccc4 4N-033 c1cc2c(cc1[N+](=O)[O-])cc(o2)C(=O)O 4N-034 c1ccc-2c(c1)Cc3c2ccc(c3)NC(=S)N 4N-035 COc1ccc(cc1)CO/N=C(\c2ccc(cc2)OC)/C3CC3c4ccc5c(c4)OCO5 4N-036 COc1ccc(cc1)/C(=N/O)/C2CC2c3ccc4c(c3)OCO4 4N-037 Cc1ccc(cc1)C(=O)O/N=C(\c2ccccc2)/C3CC3c4ccc(cc4)OC 4N-038 c1cc2c(cco2)cc1[N+](=O)[O-] 4N-039 COc1ccc(cc1)/C(=N\OC(=O)c2ccc(cc2F)F)/C3CC3c4ccc5c(c4)OCO5 4N-040 COc1ccc(cc1)/C(=N\OC(=O)c2ccco2)/C3CC3c4ccc5c(c4)OCO5 4N-041 c1ccc(cc1)C(CO)N2Cc3ccccc3C2=O 4N-042 CC(C)(C)C(C(=O)OC)NC(=S)NC(C)(C)C 4N-043 COc1ccc(cc1)/C(=N\OCCOc2cccc(c2)C(F)(F)F)/C3CC3c4ccc5c(c4)OCO5 4N-044 CC(C)(C)C(C(=O)OC)NC(=O)c1cc(cc(c1)Cl)Cl 4N-045 c1cc(ccc1C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Br 4N-046 c1cc(ccc1C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] 4N-047 COc1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccc(cc3)OC)/c4ccccc4 4N-048 c1cc(cc(c1)Cl)C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 4N-049 COC(=O)C(CC1CCCCC1)[NH3+].[Cl-] 4N-050 COc1ccc(cc1)C2CC2/C(=N/OC(=O)c3cccs3)/c4ccccc4 4N-051 COc1ccc(cc1)/C(=N\OC(=O)c2ccc(cc2Cl)Cl)/C3CC3c4ccc5c(c4)OCO5 4N-052 COc1ccc(cc1)/C(=N\OCc2ccc(cc2Cl)Cl)/C3CC3c4ccc5c(c4)OCO5 4N-053 COc1ccc(cc1)/C(=N/OC(=O)c2ccc(cc2)OC)/C3CC3c4ccc5c(c4)OCO5 4N-054 COc1ccc(cc1)/C(=N\OCc2ccccc2)/C3CC3c4ccc5c(c4)OCO5 4N-055 COc1ccc(cc1)C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 4N-056 COc1ccc(cc1)C2CC2/C(=N/O)/c3ccccn3 4N-057 COc1ccc(cc1)/C(=N\OCc2ccc(cc2)Cl)/C3CC3c4ccc5c(c4)OCO5 4N-058 CC(C)O/N=C(\c1ccc(cc1)OC)/C2CC2c3ccc4c(c3)OCO4 4N-059 c1ccc(cc1)C2CC2/C(=N\O)/c3ccc(cc3)Cl 4N-061 c1cc(ccc1/C(=N\OC(=O)c2ccc(c(c2)Cl)Cl)/C3CC3c4ccc(cc4Cl)Cl)Cl 4N-062 CC(=O)NC(C(=O)NC)C(C)(C)C 4N-063 Cc1ccc(cc1)C(=O)O/N=C(\c2ccccn2)/C3CC3c4ccc(cc4)OC 4N-066 COc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)Cl 4N-067 c1ccc(cc1)C(CO)N2CCS(=O)(=O)CC2 4N-068 COc1ccc(cc1)C2CC2/C(=N/OC(=O)c3ccc(cc3)OC)/c4ccccn4 4N-069 CC(C)(C)C(C(=O)NC)NC(=S)Nc1ccc(cc1)Cl 4N-070 COC(=O)C(CC1CCCCC1)N2CCS(=O)(=O)CC2 4N-072 c1ccc(cc1)CC(CO)N2CCS(=O)(=O)CC2 4N-073 c1cc2c(cco2)cc1N 4N-074 COc1ccc(cc1)C(=O)C2CC2c3ccc(cc3)Cl 4N-075 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)cco3 4N-076 c1ccc(cc1)C(CO)NC(=S)Nc2ccc(cc2)[N+](=O)[O-] 4N-078 c1ccc(cc1)C(CO)NC(=S)Nc2ccccc2 4N-079 c1csc2c1/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/CCS2(=O)=O 4N-301S c1csc2c1/C(=N\Nc3c(cc(cc3Cl)C(F)(F)F)Cl)/CCS2(=O)=O 4N-302S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)C(=O)C(F)(F)F 4N-304S Cc1ccc(cc1)N/N=C(/c2cc(n(c2C)c3cccc(c3)C(F)(F)F)c4ccc(cc4)S(=O)(=O)C)\C(F)(F)F 4N-305S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)/C(=N/Nc4ccc(cc4)Cl)/C(F)(F)F 4N-306S COc1ccc(cc1)Oc2c(c(cc(n2)c3ccccc3)C(F)(F)F)C#N 4N-307S c1ccc(cc1)c2cc(c(c(n2)Sc3ccc(cc3)Cl)C#N)C(F)(F)F 4N-308S c1ccc(cc1)c2cc(c(c(n2)N3CCOCC3)C#N)C(F)(F)F 4N-309S CN(C)/N=C/1\CCS(=O)(=O)c2c1ccs2 4N-311S c1csc2c1/C(=N/O)/CCS2(=O)=O 4N-312S c1cc(ccc1N/N=C/2\CCS(=O)(=O)c3c2ccs3)F 4N-313S c1ccc(cc1)c2cc(c(c(n2)Oc3ccccc3)C#N)C(F)(F)F 4N-314S c1ccc(cc1)c2cc(c(c(n2)Oc3ccc(cc3)Cl)C#N)C(F)(F)F 4N-315S c1ccc(cc1)c2cc(c(c(n2)Oc3ccc(cc3Cl)Cl)C#N)C(F)(F)F 4N-316S c1ccc(cc1)c2cc(c(c(n2)Oc3ccc4ccccc4c3)C#N)C(F)(F)F 4N-317S c1ccc(cc1)c2cc(c(c(n2)Sc3ccccc3)C#N)C(F)(F)F 4N-318S Cc1ccc(cc1)Sc2c(c(cc(n2)c3ccccc3)C(F)(F)F)C#N 4N-319S c1ccc(cc1)c2cc(c(c(n2)Sc3ccc(cc3)Br)C#N)C(F)(F)F 4N-320S c1ccc(cc1)c2cc(c(c(n2)Sc3ccc(cc3)C(F)(F)F)C#N)C(F)(F)F 4N-321S Cc1ccc(cc1)N/N=C/2\CCS(=O)(=O)c3c2ccs3 4N-322S c1cc(cc(c1)Cl)N/N=C/2\CCS(=O)(=O)c3c2ccs3 4N-323S c1cc(c(cc1Cl)N/N=C/2\CCS(=O)(=O)c3c2ccs3)Cl 4N-324S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)CO 4N-326S Cc1cccc(c1)C(=O)OCc2cc(n(c2C)c3cccc(c3)C(F)(F)F)c4ccc(cc4)S(=O)(=O)C 4N-327S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)COC(=O)c4cccc(c4)OC 4N-328S CNc1c(c(cc(n1)c2ccccc2)C(F)(F)F)C#N 4N-329S CN(C)c1c(c(cc(n1)c2ccccc2)C(F)(F)F)C#N 4N-330S c1ccc(cc1)c2cc(c(c(n2)N3CCCC3)C#N)C(F)(F)F 4N-331S CCN(CC)c1c(c(cc(n1)c2ccccc2)C(F)(F)F)C#N 4N-332S Cc1c(cc(c(n1)Oc2cccc(c2)NC(=O)C)C#N)C(=O)C 4N-335S c1cc(ccc1N/N=C/2\CCS(=O)(=O)c3c2ccs3)Cl 4N-336S c1cc(c(cc1N/N=C/2\CCS(=O)(=O)c3c2ccs3)Cl)Cl 4N-337S c1csc2c1/C(=N/N3CCOCC3)/CCS2(=O)=O 4N-338S COc1ccc(cc1)/N=C\2/CCS(=O)(=O)c3c2ccs3 4N-339S CC(C)(C)N/N=C/1\CCS(=O)(=O)c2c1ccs2 4N-340S c1cc(c(cc1Cl)Cl)N/N=C/2\CCS(=O)(=O)c3c2ccs3 4N-341S CC(=O)CCC(=O)c1ccco1 4N-342S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)COC(=O)c4ccc(cc4)OC 4N-343S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)COC(=O)c4ccc(cc4)F 4N-344S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)COC(=O)C(C)(C)CCl 4N-345S Cc1c(cc(c(n1)NCc2cc(no2)c3ccccc3)C#N)C(=O)OC 4N-348S Cc1c(cc(c(n1)NCc2cc(no2)c3ccc(cc3)OC)C#N)C(=O)OC 4N-349S Cc1c(cc(c(n1)NCc2cc(no2)c3ccc(cc3)Cl)C#N)C(=O)OC 4N-350S Cc1c(cc(c(n1)NCc2cc(no2)c3ccc(cc3)Cl)C#N)C(=O)C 4N-351S Cc1c(cc(c(n1)NCc2cc(no2)c3ccccc3)C#N)C(=O)C 4N-352S Cc1c(cc(c(n1)NCc2cc(no2)c3ccc(cc3)OC)C#N)C(=O)C 4N-353S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)COC(=O)c4ccc(cc4Cl)Cl 4N-354S c1ccc(c(c1)c2cc(c(c(n2)O)C#N)C(F)(F)F)Cl 4N-355S c1cc(cc(c1)Cl)c2cc(c(c(n2)O)C#N)C(F)(F)F 4N-356S c1cc(ccc1c2cc(c(c(n2)O)C#N)C(F)(F)F)Cl 4N-357S Cc1ccc(n1c2cc(ccc2Cl)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C 4N-359S c1cc(ccc1/N=C\2/CCS(=O)(=O)c3c2ccs3)Cl 4N-361S Cn1c2ccccc2c(c1Oc3cccc(c3)C(F)(F)F)/C=N/c4ccc(cc4)OC 4N-363S CC(=O)Nc1ccc(cc1)/C=C/c2nc3ccccc3o2 4N-367S c1cc(ccc1c2cc(on2)CNC(=O)CCl)Cl 4N-369S Cn1c2ccccc2c(c1Oc3cccc(c3)C(F)(F)F)/C=N/c4ccc(cc4)Cl 4N-372S Cc1ccc(n1c2cc(cc(c2)Cl)Cl)c3ccc(cc3)S(=O)(=O)C 4N-374S Cc1cc(cc(c1)NC(=O)c2cc(n(c2C)c3cccc(c3)C(F)(F)F)c4ccc(cc4)S(=O)(=O)C)C 4N-375S c1cc(ccc1c2cc(c(c(n2)Cl)C#N)C(F)(F)F)Cl 4N-376S c1ccc2c(c1)nc(o2)/C=C/c3ccc(cc3)NC(=O)c4ccc(cc4)F 4N-377S c1cc(ccc1c2cc(on2)CNC(=O)CN3CCOCC3)Cl 4N-379S Cc1c(cc(n1c2cc(ccc2Cl)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)C(=O)C(F)(F)F 4N-380S CCN(CC)CC(=O)NCc1cc(no1)c2ccc(cc2)Cl 4N-381S c1cc(ccc1c2cc(on2)CNC(=O)CN3CCCC3)Cl 4N-382S Cc1c(cc(n1c2cc(cc(c2)Cl)Cl)c3ccc(cc3)S(=O)(=O)C)C(=O)C(F)(F)F 4N-383S c1cc(ccc1c2cc(c(c(n2)Sc3ccc(cc3)Cl)C#N)C(F)(F)F)Cl 4N-384S c1cc(ccc1c2cc(c(c(n2)N3CCOCC3)C#N)C(F)(F)F)Cl 4N-385S c1cc(ccc1c2cc(c(c(n2)Oc3ccc(cc3F)F)C#N)C(F)(F)F)Cl 4N-386S COc1ccc(cc1)Oc2c(c(cc(n2)c3ccc(cc3)Cl)C(F)(F)F)C#N 4N-387S Cc1ccc(cc1C)/N=C/c2c3ccccc3n(c2Oc4ccc(cc4)C(F)(F)F)C 4N-389S Cn1c2ccccc2c(c1Cl)C(=O)Nc3ccc(cc3)OC 4N-390S Cc1ccc(cc1)C(=O)OCc2cc(n(c2C)c3cccc(c3)C(F)(F)F)c4ccc(cc4)S(=O)(=O)C 4N-392S Cc1c(cc(n1c2cccc(c2)C(F)(F)F)c3ccc(cc3)S(=O)(=O)C)COC(=O)C4CC4 4N-393S CN(Cc1ccccc1)CC(=O)NCc2cc(no2)c3ccc(cc3)Cl 4N-396S COc1ccc(cc1)c2cc(on2)CNC(=O)CCl 4N-397S c1cc(cc(c1)Cl)c2cc(c(c(n2)Cl)C#N)C(F)(F)F 4N-398S c1ccc(c(c1)c2cc(c(c(n2)Cl)C#N)C(F)(F)F)Cl 4N-399S Cn1c2ccccc2c(c1Cl)C(=O)Nc3ccccc3 4N-400S Cc1ccc(cc1)NC(=O)c2c3ccccc3n(c2Cl)C 4N-401S Cc1ccc(cc1)Sc2c(c3ccccc3n2C)C(=O)Nc4ccc(cc4)OC 4N-402S Cc1c(cc(n1c2cc(cc(c2)Cl)Cl)c3ccc(cc3)S(=O)(=O)C)C=O 4N-403S Cc1cc(nc2c1cccc2)Cl 4N-501S Cc1ccc(cc1)Sc2cc(c3cccc(c3n2)C)C 4N-504S Cc1ccc(cc1)Sc2cc(c3cc(ccc3n2)Cl)C 4N-505S Cc1cc(nc2c1cc(cc2)Cl)Oc3ccc(cc3)OC 4N-506S Cc1cc(nc2c1cc(cc2)Cl)N3CCOCC3 4N-507S Cc1cccc2c1nc(cc2C)N3CCCCC3 4N-508S Cc1cc(nc2c1cc(cc2)Cl)Sc3cccc(c3)C(F)(F)F 4N-509S Cc1cc(nc2c1cc(cc2)Cl)Oc3ccc(cc3F)F 4N-510S Cc1cc(nc2c1cc(cc2)Cl)N3CCCCC3 4N-511S COC(=O)c1cc(n(n1)c2cccc(c2)Cl)c3ccc(cc3)Cl 4N-515S COC(=O)c1cc(n(n1)c2ccccc2Cl)c3ccc(cc3)Cl 4N-516S COC(=O)c1cc(n(n1)c2ccc(cc2Cl)Cl)c3ccc(cc3)Cl 4N-517S COC(=O)c1cc(n(n1)c2cc(ccc2Cl)Cl)c3ccc(cc3)Cl 4N-518S COC(=O)c1cc(n(n1)c2cc(cc(c2)Cl)Cl)c3ccc(cc3)Cl 4N-519S COC(=O)c1cc(n(n1)c2ccc(c(c2)Cl)Cl)c3ccc(cc3)Cl 4N-520S Cc1ccc(cc1)n2c(cc(n2)C(=O)OC)c3ccc(cc3)Cl 4N-521S COC(=O)C(=O)CC(=O)c1ccc(c(c1)Cl)Cl 4N-522S c1ccc(c(c1)c2csc(n2)NC(=O)CN3CCOCC3)Cl 4N-523S c1ccc(c(c1)c2csc(n2)NC(=O)CN3CCSCC3)Cl 4N-524S CN(C)CC(=O)Nc1nc(cs1)c2ccccc2Cl 4N-525S Cc1cc(nc2c1cccc2)Sc3ccc(cc3)Cl 4N-531S Cc1cc(nc2c1cccc2)Sc3cccc(c3)C(F)(F)F 4N-532S Cc1ccc(cc1)Sc2cc(c3ccccc3n2)C 4N-533S Cc1cc(nc2c1cccc2)Oc3cccc(c3)C(F)(F)F 4N-534S Cc1cc(nc2c1cccc2)Oc3ccc(cc3F)F 4N-535S Cc1cc(nc2c1cccc2)Oc3ccc(cc3)OC 4N-536S Cc1cc(nc2c1cccc2)N3CCN(CC3)C 4N-537S Cc1cc(nc2c1cccc2)N3CCOCC3 4N-538S Cc1cc(nc2c1cccc2)N3CCCC3 4N-539S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)SCc5ccc(cc5Cl)Cl 4N-540S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)SCc5c(cccc5Cl)Cl 4N-541S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)SCc5ccc(cc5)F 4N-542S COC(=O)c1cc(n(n1)c2cc(ccc2Cl)Cl)c3ccc(c(c3)Cl)Cl 4N-544S COC(=O)c1cc(n(n1)c2ccc(cc2)S(=O)(=O)N)c3ccc(c(c3)Cl)Cl 4N-545S Cc1cccc(c1C)n2c(cc(n2)C(=O)OC)c3ccc(c(c3)Cl)Cl 4N-546S COC(=O)c1cc(n(n1)c2cccc(c2)Cl)c3ccc(c(c3)Cl)Cl 4N-547S c1ccc(cc1)c2c(sc(n2)c3ccccc3)Cc4nnc(o4)SCc5c(cccc5Cl)F 4N-548S c1ccc(cc1)n2c(cc(n2)C(=O)O)c3ccc(cc3)Cl 4N-549S c1cc(cc(c1)Cl)n2c(cc(n2)C(=O)O)c3ccc(cc3)Cl 4N-550S COC(=O)C(=O)CC(=O)c1ccccc1 4N-551S COC(=O)C(=O)CC(=O)c1ccccc1Cl 4N-552S c1ccc(cc1)c2csc(n2)NC(=O)CN3CCOCC3 4N-554S c1ccc(cc1)c2csc(n2)NC(=O)CN3CCCCC3 4N-555S CN(C)CC(=O)Nc1nc(cs1)c2ccccc2 4N-556S c1cc(ccc1c2cc(nn2c3cc(ccc3Cl)Cl)C(=O)O)Cl 4N-558S c1ccc(c(c1)n2c(=O)cc(c(n2)C(=O)c3ccc(cc3)Cl)C(F)(F)F)Cl 4N-559S c1cc(cc(c1)Cl)n2c(=O)cc(c(n2)C(=O)c3ccc(cc3)Cl)C(F)(F)F 4N-560S c1cc(ccc1C(=O)c2c(cc(=O)n(n2)c3ccc(cc3)Cl)C(F)(F)F)Cl 4N-561S COC(=O)c1cc(n(n1)c2ccc(cc2Cl)Cl)c3ccc(c(c3)Cl)Cl 4N-562S COc1ccc(cc1)CSc2nnc(o2)Cc3c(nc(s3)c4ccccc4)c5ccccc5 4N-565S COC(=O)c1cc(n(n1)c2ccccc2)c3ccc(c(c3)Cl)Cl 4N-569S COC(=O)c1cc(n(n1)c2ccc(cc2)F)c3ccc(c(c3)Cl)Cl 4N-570S COC(=O)c1cc(n(n1)c2cc(cc(c2)Cl)Cl)c3ccc(c(c3)Cl)Cl 4N-571S c1cc(ccc1c2cc(nn2c3ccc(cc3)Cl)C(=O)O)Cl 4N-572S c1cc(ccc1c2cc(nn2c3ccc(c(c3)Cl)Cl)C(=O)O)Cl 4N-573S c1cc(ccc1c2cc(nn2c3ccc(cc3Cl)Cl)C(=O)O)Cl 4N-574S Cc1ccc(cc1)n2c(cc(n2)C(=O)OC)c3ccc(c(c3)Cl)Cl 4N-575S Cc1ccc(cc1)n2c(cc(n2)C(=O)O)c3ccc(cc3)Cl 4N-577S c1cc(ccc1c2cc(nn2c3ccc(cc3)F)C(=O)O)Cl 4N-578S c1ccc(cc1)Sc2nc(c(s2)C=O)Cl 4N-581S c1cc(ccc1c2cc(nn2c3ccc(cc3)S(=O)(=O)N)C(=O)O)Cl 4N-582S c1ccc(c(c1)c2csc(n2)NC(=O)CN3CCN(CC3)c4ccccc4F)Cl 4N-584S c1cc(ccc1c2csc(n2)NC(=O)CN3CCOCC3)Cl 4N-585S c1cc(ccc1c2csc(n2)NC(=O)CN3CCCCC3)Cl 4N-586S CC(=O)C(C(=O)Nc1ccccc1)Cl 4N-587S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)c3cccc(c3)Cl)C(F)(F)F 4N-592S c1ccc(c(c1)c2cc(nn2c3ccc(cc3Cl)Cl)C(=O)O)Cl 4N-593S c1ccc(c(c1)c2cc(nn2c3cccc(c3)Cl)C(=O)O)Cl 4N-594S c1ccc(c(c1)c2cc(nn2c3ccc(cc3)Cl)C(=O)O)Cl 4N-595S CCN(CC)CC(=O)Nc1nc(cs1)c2ccc(cc2)Cl 4N-597S c1ccc(c(c1)c2cc(nn2c3ccc(cc3)F)C(=O)O)Cl 4N-598S c1ccc(c(c1)c2cc(nn2c3ccc(c(c3)Cl)Cl)C(=O)O)Cl 4N-599S c1ccc(cc1)n2c(cc(n2)C(=O)O)c3ccccc3Cl 4N-600S CN(Cc1ccccc1)CC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 4N-603S COC(=O)c1cc(n(n1)c2ccc(c(c2)Cl)Cl)c3ccccc3Cl 4N-604S COC(=O)c1cc(n(n1)c2ccc(cc2)Cl)c3ccccc3Cl 4N-605S c1ccc(c(c1)n2c(=O)cc(c(n2)C(=O)c3cccc(c3)Cl)C(F)(F)F)Cl 4N-607S c1cc(ccc1c2cc(nn2c3cc(ccc3Cl)Cl)C(=O)N4CCOCC4)Cl 4N-611S C=CCNC(=O)c1cc(n(n1)c2cc(ccc2Cl)Cl)c3ccc(cc3)Cl 4N-612S c1cc(ccc1c2cc(nn2c3cc(ccc3Cl)Cl)C(=O)Nc4ccc(cc4)Cl)Cl 4N-613S c1cc(ccc1c2cc(nn2c3cc(ccc3Cl)Cl)C(=O)Nc4ccc(c(c4)Cl)Cl)Cl 4N-614S COc1ccc(c(c1)NC(=O)c2cc(n(n2)c3ccc(cc3Cl)Cl)c4ccccc4Cl)OC 4N-617S Cc1ccc(cc1)n2c(cc(n2)C(=O)N3CCOCC3)c4ccc(cc4)Cl 4N-618S c1ccc(c(c1)C(=O)c2c(cc(=O)n(n2)c3cccc(c3)Cl)C(F)(F)F)Cl 4N-619S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)c3ccc(cc3)C(F)(F)F)C(F)(F)F 4N-620S c1ccc(cc1)n2c(cc(n2)C(=O)O)c3ccc(c(c3)Cl)Cl 4N-623S c1cc(cc(c1)Cl)n2c(cc(n2)C(=O)O)c3ccc(c(c3)Cl)Cl 4N-624S c1cc(c(cc1c2cc(nn2c3ccc(cc3Cl)Cl)C(=O)O)Cl)Cl 4N-625S c1cc(ccc1n2c(cc(n2)C(=O)O)c3ccc(c(c3)Cl)Cl)F 4N-626S c1cc(ccc1n2c(cc(n2)C(=O)O)c3ccc(c(c3)Cl)Cl)Cl 4N-627S CNC(=O)c1cc(n(n1)c2cc(ccc2Cl)Cl)c3ccc(cc3)Cl 4N-633S c1cc(ccc1c2cc(nn2c3cc(ccc3Cl)Cl)C(=O)NC4CC4)Cl 4N-634S c1cc(cc(c1)NC(=O)c2cc(n(n2)c3cc(ccc3Cl)Cl)c4ccc(cc4)Cl)C(F)(F)F 4N-635S c1cc(ccc1c2cc(nn2c3cc(ccc3Cl)Cl)C(=O)Nc4ccc(cc4)C(F)(F)F)Cl 4N-636S c1ccc(cc1)c2cc(nn2c3ccc(cc3)Cl)C(=O)O 4N-637S c1ccc(cc1)c2cc(nn2c3ccc(cc3Cl)Cl)C(=O)O 4N-638S Cc1ccc(cc1)n2c(cc(n2)C(=O)O)c3ccccc3 4N-640S c1ccc(cc1)c2cc(nn2c3ccc(cc3)F)C(=O)O 4N-641S Cc1cccc2c1nc(cc2C(F)(F)F)Sc3ccc(cc3)OC 4N-643S Cc1cccc2c1nc(cc2C(F)(F)F)Oc3cccc(c3)C(F)(F)F 4N-644S Cc1cccc2c1nc(cc2C(F)(F)F)Oc3ccc(cc3F)F 4N-645S Cc1cccc2c1nc(cc2C(F)(F)F)N3CCCC3 4N-646S Cc1cccc2c1nc(cc2C(F)(F)F)N3CCOCC3 4N-647S COc1ccc(c(c1)NC(=O)c2cc(n(n2)c3ccccc3)c4ccc(cc4)Cl)OC 4N-650S CNC(=O)c1cc(n(n1)c2ccccc2)c3ccc(cc3)Cl 4N-651S CO/N=C(/CN1CCOCC1)\c2ccc(cc2)Cl 4N-652S COc1ccc(cc1)c2cc(on2)CNC(=O)c3cc(no3)c4ccccc4Cl 4N-653S c1ccc(cc1)c2cc(on2)CNC(=O)c3cc(no3)c4ccccc4Cl 4N-654S COc1ccc(cc1)N(Cc2ccccc2)C(=O)c3cc(no3)c4ccccc4Cl 4N-655S Cc1ccc(cc1C)NC(=O)c2cc(n(n2)c3ccccc3)c4ccccc4Cl 4N-659S Cn1c(c(c(n1)C(F)(F)F)CO/N=C/c2ccc(cc2)Cl)Sc3ccc(cc3)Br 4N-661S Cn1c(c(c(n1)C(F)(F)F)CO/N=C/c2ccc(cc2Cl)Cl)Sc3ccc(cc3)Br 4N-662S Cc1ccc(cc1C)NC(=O)c2cc(n(n2)c3ccc(cc3Cl)Cl)c4ccc(cc4)Cl 4N-663S Cc1ccc(cc1C)NC(=O)c2cc(n(n2)c3ccc(cc3)Cl)c4ccccc4Cl 4N-665S c1ccc2c(c1)nc(o2)/C=C/c3ccc(cc3)NC(=O)c4cccc(c4)C(F)(F)F 4N-667S COc1cccc(c1)C(=O)Nc2ccc(cc2)/C=C/c3nc4ccccc4o3 4N-668S c1ccc2c(c1)nc(o2)/C=C/c3ccc(cc3)NC(=O)c4c(cccc4F)F 4N-669S CC(=O)N1CC(=O)N(/C(=C/c2ccc(cc2)OC)/C1=O)Cc3ccc(cc3)C(C)(C)C 4N-700 CC(c1ccccc1)/N=C/c2ccc(c(c2O)Cc3c(cccc3Cl)F)O 4N-701 COc1ccc(cc1)/C=C/2\C(=O)NCC(=O)N2Cc3ccc(cc3)F 4N-702 c1ccc2c(c1)CC(=O)N(C2=O)CC(=O)N 4N-704 CC(C)(C)NC(=O)C1Cc2ccccc2CN1c3c(cccn3)[N+](=O)[O-] 4N-705 c1ccc(cc1)S(=O)(=O)CCC(=C(F)F)F 4N-706 CC(=O)N1CC(=O)N(/C(=C/c2ccccc2)/C1=O)Cc3ccccc3 4N-707 c1ccc(cc1)CN\2C(=O)CNC(=O)/C2=C\c3ccccc3 4N-710 c1ccc2c(c1)nc(s2)SCCC(=C(F)F)F 4N-711 CC(=O)N1CC(=O)N(/C(=C/c2ccc(cc2)F)/C1=O)Cc3ccccc3 4N-713 CC(c1ccnc2n1ncn2)Oc3ccc(cc3)Cc4c(cc(cn4)C(F)(F)F)Cl 4N-714 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)Nc3ccc(cc3)OC 4N-715 c1ccc(cc1)CC2C(=O)NC(C(=O)N2)Cc3ccccc3 4N-716 CC(=O)N1C(C(=O)N(C(C1=O)Cc2ccccc2)C(=O)C)Cc3ccccc3 4N-717 CC(=O)N1CC(=O)N(/C(=C/c2ccc(cc2)N(C)C)/C1=O)Cc3ccccc3 4N-718 CN(C)c1ccc(cc1)/C=C/2\C(=O)NCC(=O)N2Cc3ccccc3 4N-719 COc1ccc(cc1)/C=C/2\C(=O)N(CC(=O)N2Cc3ccccc3)Cc4ccc(cc4)F 4N-720 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)c3ccc(cc3)OC 4N-721 C(CSc1[nH]nc(n1)N)C(=C(F)F)F 4N-723 CN1CC(C(C1)C(=O)c2ccc(cc2)Cl)c3ccccc3 4N-725 Cc1ccc(cc1)C2CN(CC2C(=O)c3ccc(cc3)F)C 4N-726 CN1CC(C(C1)C(=O)c2cccc(c2)OC)c3ccc(cc3)Cl 4N-728 CN1CC(C(C1)C(=O)c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3)Cl 4N-729 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)Nc3ccc(cc3)Cl 4N-730 c1ccc2c(c1)[nH]c(n2)SCCC(=C(F)F)F 4N-731 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)Cl 4N-734 COc1ccc(cc1)NC(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 4N-735 CN(C)c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Cl 4N-736 CN1CC(C(C1)C(=O)c2ccc(cc2)F)c3c(cccc3Cl)F 4N-737 COc1ccc(cc1)C(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 4N-738 c1cc(ccc1CSc2nccc(n2)c3cc(sc3Cl)Cl)Cl 4N-739 c1cc(c(cc1Cl)Cl)CSc2nccc(n2)c3cc(sc3Cl)Cl 4N-740 C(CSc1nnc(s1)N)C(=C(F)F)F 4N-741 CCOC(=O)C(CSCCC(=C(F)F)F)N 4N-742 c1cc(ccc1n2c(ccn2)c3cc(sc3Cl)Cl)F 4N-745 COc1ccc(cc1)n2c(ccn2)c3cc(sc3Cl)Cl 4N-746 CN1CC(C(C1)C(=O)c2ccc(cc2)Cl)c3ccc(cc3Cl)Cl 4N-747 c1cnc([nH]c1=O)SCCC(=C(F)F)F 4N-749 c1cc(ccc1n2c(ccn2)c3cc(sc3Cl)Cl)Cl 4N-751 CC(C)(C)NC(=O)C1Cc2ccccc2CN1c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 4N-753 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)c3cccc(c3)C(F)(F)F 4N-754 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)c3ccsc3 4N-756 c1ccc(cc1)c2ccc(cc2)c3ccnc4n3nc(n4)SCCC(=C(F)F)F 4N-758 c1cc(ccc1c2ccnc3n2nc(n3)SCCC(=C(F)F)F)F 4N-759 C1CSC(=NC#N)S1 4N-760 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)Oc3ccc(nn3)Cl 4N-761 COc1ccc(cc1)CSc2nccc(n2)c3cc(sc3Cl)Cl 4N-764 COC(=O)c1ccsc1N 4N-801 CC(=O)Nc1c(ccs1)C(=O)OC 4N-802 CC(=O)Nc1c(ccs1)C(=O)O 4N-803 CC(=O)Nc1c(cc(s1)Cl)C(=O)OC 4N-804 CC(=O)Nc1c(cc(s1)Cl)C(=O)NN 4N-806 c1csc(c1C#N)N 4N-807 CC(=O)Nc1c(ccs1)C(=O)NN 4N-808 CC(=O)Nc1c(ccs1)C(=O)Nc2ccc(cc2)Cl 4N-809 CN(C)/C=N/c1c(ccs1)C(=O)OC 4N-810 COC(=O)c1ccsc1N/C=N/OC 4N-811 COC(=O)c1ccsc1NC(=O)CCCl 4N-812 COC(=O)c1ccsc1NC(=O)c2ccco2 4N-813 COC(=O)c1ccsc1NC(=O)c2cccc(c2)Cl 4N-814 COC(=O)c1ccsc1N/C=N/OCc2ccccc2 4N-815 COc1ccc(cc1)C(=O)Nc2c(ccs2)C(=O)OC 4N-816 COC(=O)c1ccsc1NS(=O)(=O)C 4N-817 COC(=O)c1ccsc1NS(=O)(=O)c2ccccc2 4N-818 CCOC(=O)NC(=O)/C(=C/Nc1c(ccs1)C(=O)OC)/C(=O)C 4N-819 CCOC(=O)NC(=O)/C(=C\Nc1c(ccs1)C(=O)OC)/C#N 4N-820 c1csc2c1c(=O)[nH]cn2 4N-821 Cc1ccc(cc1)n2c3c(c(n2)C)C(C(=C(O3)N)C#N)c4ccc(cc4)OC 4N-822 COc1ccc(cc1)n2cnc3c(c2=O)ccs3 4N-823 COC(=O)c1ccsc1n2cc(c(=O)[nH]c2=O)C#N 4N-825 Cc1c2c(n(n1)C3=NCCCN3)NC(=O)C(C2c4ccc(cc4)OC)C#N 4N-826 c1ccc(cc1)C(COC(=O)c2cccs2)NC(=O)c3cccs3 4N-901 c1ccc(cc1)C(COC(=O)C2CC2)NC(=O)C3CC3 4N-902 c1ccc(cc1)C(CO)NC(=O)Nc2cccc(c2)Cl 4N-903 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC(CO)c2ccccc2 4N-904 c1cc(ccc1c2c(n3cc(ccc3n2)Cl)Cl)Cl 4P-001 c1cc2cn[nH]c2c(c1)NC(=S)N 4P-002 c1cc2cc[nH]c2c(c1)NC(=S)N 4P-003 COc1cccc(c1)c2c(c[nH]n2)/C=N/NC(=O)c3c(ccs3)OCc4ccc(cc4)Cl 4P-005 COc1cccc(c1)c2c(c[nH]n2)/C=N/NC(=O)Cn3cncn3 4P-008 c1cc2c(cn[nH]2)c(c1)[N+](=O)[O-] 4P-009 Cc1ccc(cc1)COc2ccsc2C(=O)N/N=C/c3c[nH]nc3c4cccc(c4)OC 4P-011 c1ccc2c(c1)nc(c(n2)F)O 4P-012 CN1CC(C(C1)C(=O)c2ccc(cc2)Cl)c3ccco3 4P-014 COc1ccc(cc1)n2cnc(c2N)C#N 4P-016 c1ccc(cc1)/N=C/c2cccs2 4P-017 CC(=O)/C=C/c1ccccc1Oc2ccccc2 4P-018 COC(=O)c1cc2ccccc2[nH]1 4P-019 c1ccc2c(c1)cc([nH]2)C(=O)NN 4P-020 c1ccc(c(c1)/C=N\O)Oc2ccc(c(c2)F)F 4P-021 c1ccc2c(c1)c(=S)ss2 4P-022 c1ccc(c(c1)/C=N\O)Oc2ccc(c(c2)F)Cl 4P-024 c1ccc(c(c1)/C=N\O)Oc2cccc(c2)C(F)(F)F 4P-025 C=CCOC(=O)C(CC(=O)O)c1ccccc1 4P-026 c1ccc(cc1)c2cc(c(c(c2)c3ccccc3)Nc4nc(cs4)c5cccs5)c6ccccc6 4P-029 c1ccc2c(c1)cc([nH]2)C(=O)N 4P-033 c1cc(sc1)C(=O)CN2CCN(CC2)c3ccc(cc3)F 4P-034 c1cc(c(cc1Cl)N)I 4P-037 C1CN2CCC1/C(=N/O)/C2 4P-039 CC(=O)/C=C/c1ccccc1Oc2cccc(c2)Cl 4P-040 CN1C(=O)/C(=C/N(C)C)/SC1=O 4P-042 c1cc(cc(c1)N2CCN(CC2)CC(=O)c3cccs3)C(F)(F)F 4P-043 c1ccc(c(c1)C2=NCCN2)S 4P-049 Cc1cccn2c1nc(c2Br)c3ccc(cc3)Cl 4P-053 Cc1cc(ccc1NC(=S)NC(=O)c2ccccc2)[N+](=O)[O-] 4P-055 Cc1c(cccc1[N+](=O)[O-])NC(=S)NC(=O)c2ccccc2 4P-056 CC(=O)/C=C/c1ccccc1Oc2cccc(c2)C(F)(F)F 4P-059 CC1CN(CC(O1)C)Cc2c(nc3n2cc(cc3)Cl)c4ccccc4 4P-062 Cc1c(cccc1[N+](=O)[O-])NC(=S)N 4P-063 CC(=O)/C=C/c1ccccc1Oc2ccc(c(c2)F)F 4P-064 c1ccc(c(c1)/C=N\O)Oc2ccc(cc2F)Br 4P-065 CC(=O)/C=C/c1ccccc1Oc2ccc(cc2F)Br 4P-067 CC(=O)/C=C/c1ccccc1Oc2ccc(c(c2)F)Cl 4P-068 CCOC(=O)C(F)(F)Sc1c(cc(cn1)C(F)(F)F)Cl 4P-070 COc1ccc(cc1)c2cn3ccccc3n2 4P-071 Cc1cc(ccc1NC(=S)N)[N+](=O)[O-] 4P-072 CC1(CC(=O)C(=Cc2c[nH]c3c2cccc3)C(=O)C1)C 4P-074 CCN(CC)c1ccc(c(c1)C)NC(=S)NC(=O)c2ccccc2 4P-075 Cc1ccc(cc1)S(=O)(=O)/C(=C\N(C)C)/c2cnc(s2)Cl 4P-077 COc1ccc(cc1)c2cn3cccnc3n2 4P-080 CCOc1c(cc(cn1)[N+](=O)[O-])C#N 4P-081 CC(=O)Nc1ccc(cc1)Oc2ccccc2C=O 4P-082 Cc1cccn2c1nc(c2)c3ccc(cc3)OC 4P-083 CC(C)OC(=O)c1cccc(n1)C(=O)Nc2ccc(cc2)F 4P-084 CCN(CC)c1ccc(c(c1)C)NC(=S)N 4P-085 c1ccc(c(c1)C=O)Oc2ccc(cc2)C#N 4P-090 c1ccc2c(c1)c(c[nH]2)C(=O)NN 4P-091 COc1ccc(cc1)c2c(n3ccccc3n2)Cl 4P-092 COc1ccc(cc1)c2c(n3cccnc3n2)Br 4P-093 c1c(cnc(n1)N)Br 4P-094 c1ccc(c(c1)C=O)Oc2ccccc2C#N 4P-096 c1cc(c2cn[nH]c2c1)N 4P-101 Cc1ccc2cccnc2c1N 4P-105 c1ccc(cc1)CNCC(C(F)(F)F)O 4P-106 c1ccc(c(c1)C=O)Oc2ccc(cc2)[N+](=O)[O-] 4P-107 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2cn[nH]3 4P-108 Cc1ccc2c(c1NC(=S)NC(=O)c3ccccc3)CCCN2 4P-109 CC(C)(C)OC(=O)/C(=N\OC)/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3.[Br-] 4P-302S CCOC(=O)/C(=N\OC)/C[P+](c1ccccc1)(c2ccccc2)c3ccccc3.[Br-] 4P-305S Cc1ccc(cc1)C(=O)Nc2c(c(no2)C)C#N 4P-308S Cc1c(c(on1)NC(=O)c2cccc(c2Cl)Cl)C#N 4P-309S Cc1c(c(on1)NC(=O)c2cccnc2Cl)C#N 4P-310S Cc1c(c(on1)NC(=O)c2cccs2)C#N 4P-311S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=O)N2 4P-314S Cc1c(n(c(c1C#N)N)Cc2ccc(cc2)OC)C 4P-315S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=S)N2 4P-319S CC(C)(C)OC(=O)N1CCC(CC1)Nc2ncccn2 4P-322S Cc1c(c(on1)N)C(=O)N 4P-323S COc1ccc(cc1)S(=O)(=O)/N=c/2\c3ccccc3[nH]c(=O)n2c4ccccc4 4P-326S Cc1ccc(cc1)S(=O)(=O)/N=c/2\c3ccccc3[nH]c(=O)n2c4ccccc4 4P-327S Cc1c(n(c(c1C#N)NC(=O)Nc2ccccc2)Cc3ccc(cc3)OC)C 4P-328S Cc1ccc(cc1)CSC\2=Nc3ccccc3/C2=N/Nc4cccc(c4)C(F)(F)F 4P-329S CCSC\1=Nc2ccccc2/C1=N/Nc3cccc(c3)C(F)(F)F 4P-330S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=N2)SCc4ccc(cc4)Cl 4P-331S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=N2)SCc4cccc(c4)C(F)(F)F 4P-332S c1ccc(cc1)CSC\2=Nc3ccccc3/C2=N/Nc4cccc(c4)C(F)(F)F 4P-338S COc1ccc(cc1)CSC\2=Nc3ccccc3/C2=N/Nc4cccc(c4)C(F)(F)F 4P-339S c1ccc(cc1)n2/c(=N/S(=O)(=O)c3ccccc3)/c4ccccc4[nH]c2=O 4P-340S c1ccc(cc1)n2/c(=N/S(=O)(=O)c3ccc(cc3)Cl)/c4ccccc4[nH]c2=O 4P-341S Cc1ccccc1C(=O)O/N=C/c2c3ccccc3n(c2N4CCOCC4)C 4P-345S Cc1cccc(c1)C(=O)O/N=C/c2c3ccccc3n(c2N4CCOCC4)C 4P-346S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=N2)SCc4ccc(cc4)F 4P-347S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=N2)SCc4cccc(c4)F 4P-348S c1ccc(c(c1)CSC\2=Nc3ccccc3/C2=N/Nc4cccc(c4)C(F)(F)F)Cl 4P-349S Cc1cccc(c1)CSC\2=Nc3ccccc3/C2=N/Nc4cccc(c4)C(F)(F)F 4P-350S Cc1ccc(cc1)C(=O)O/N=C/c2c3ccccc3n(c2N4CCOCC4)C 4P-353S Cn1c2ccccc2c(c1N3CCOCC3)/C=N/OC(=O)c4ccc(cc4)F 4P-355S Cc1ccc(cc1)Sc2c3c(noc3ncn2)C 4P-357S Cn1c2ccccc2c(c1N3CCOCC3)/C=N/OC(=O)c4cccnc4Cl 4P-358S CC(C)(C)c1ccc(cc1)CSC\2=Nc3ccccc3/C2=N/Nc4cccc(c4)C(F)(F)F 4P-359S Cc1ccccc1CSC\2=Nc3ccccc3/C2=N/Nc4cccc(c4)C(F)(F)F 4P-360S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=N2)SCc4cccc(c4)Cl 4P-361S CCN(CC)CC(=O)Nc1ccccc1SCC(=O)Nc2ccsc2C(=O)OC 4P-367S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)CNCC=C 4P-368S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)CNC3CC3 4P-369S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)CN3CCOCC3 4P-370S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=N2)SCc4c(cccc4Cl)Cl 4P-372S c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=N2)SCc4ccc(cc4Cl)Cl 4P-373S CSC\1=Nc2ccccc2/C1=N/Nc3cccc(c3)C(F)(F)F 4P-375S Cc1c2c(ncnc2Sc3ccc(cc3)Cl)on1 4P-377S Cc1c2c(ncnc2Sc3ccc(cc3)OC)on1 4P-379S Cc1c2c(ncnc2Sc3cccc(c3)C(F)(F)F)on1 4P-380S Cc1ccc(c(c1)C)Sc2c3c(noc3ncn2)C 4P-381S CC(C)NCC(=O)Nc1ccccc1SCC(=O)Nc2ccsc2C(=O)OC 4P-383S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)CNC3CCCCC3 4P-384S c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3nnc(s3)C(F)(F)F)F 4P-501S c1cc(ccc1N2CCN(CC2)CC(=O)Nc3nnc(s3)C(F)(F)F)F 4P-505S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)Nc4nnc(s4)C(F)(F)F 4P-506S c1cc(sc1)CN2C(CCC2=O)C(=O)O 4P-507S c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3nnc(s3)C(F)(F)F 4P-508S C1CCN(CC1)CC(=O)Nc2nnc(s2)C(F)(F)F 4P-509S c1cc(cc(c1)NC(=O)C2CCC(=O)N2Cc3cccs3)C(F)(F)F 4P-512S c1cc(sc1)CN2C(CCC2=O)C(=O)Nc3ccc(cc3)Cl 4P-513S c1ccc(cc1)C2C(=C(C(=O)O2)Br)Br 4P-514S c1cc(sc1)CN2C(CCC2=O)C(=O)N3CCOCC3 4P-515S CN(C)C(=O)C1CCC(=O)N1Cc2cccs2 4P-516S COc1ccc(cc1)NC(=O)C2CCC(=O)N2Cc3cccs3 4P-517S c1cc(sc1)CN2C(CCC2=O)C(=O)Nc3ccc(cc3F)F 4P-518S c1ccc(c(c1)CN2C(CCC2=O)C(=O)O)Cl 4P-519S c1ccc(c(c1)CN2C(CCC2=O)C(=O)Nc3cccc(c3)C(F)(F)F)Cl 4P-522S c1ccc(c(c1)CN2C(CCC2=O)C(=O)Nc3ccc(cc3)C(F)(F)F)Cl 4P-523S c1ccc(c(c1)CN2C(CCC2=O)C(=O)Nc3ccc(cc3)Cl)Cl 4P-524S c1ccc(c(c1)CN2C(CCC2=O)C(=O)Nc3ccccc3Br)Cl 4P-526S c1ccc(c(c1)CN2C(CCC2=O)C(=O)Nc3ccc(cc3)Br)Cl 4P-527S c1ccc(c(c1)CN2C(CCC2=O)C(=O)Nc3ccc(cc3Cl)Cl)Cl 4P-528S c1ccc(c(c1)CN2C(CCC2=O)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl 4P-529S c1ccc(c(c1)N)SCC(=O)Nc2nnc(s2)C(F)(F)F 4P-530S c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)F)SCC(=O)Nc3nnc(s3)C(F)(F)F 4P-531S c1ccc(c(c1)NS(=O)(=O)c2ccccc2F)SCC(=O)Nc3nnc(s3)C(F)(F)F 4P-532S c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)Cl)SCC(=O)Nc3nnc(s3)C(F)(F)F 4P-533S Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3nnc(s3)C(F)(F)F 4P-534S COc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3nnc(s3)C(F)(F)F 4P-535S c1cc(sc1)CN2C(CCC2=O)C(=O)Nc3ccc(cc3)C(F)(F)F 4P-536S COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)c3ccccc3 4P-540S Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)c3ccccc3 4P-541S c1ccc(cc1)C(=O)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 4P-542S c1ccc(cc1)C(=O)N2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)Cl 4P-543S CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3nnc(s3)C(F)(F)F 4P-544S c1ccc2c(c1)nc(s2)C3CCNCC3 4P-546S c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3ccccc3C(F)(F)F 4P-547S c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3cccc(c3)Cl 4P-548S c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3cccs3 4P-549S c1ccc(cc1)C(=O)N2CCN(CC2)S(=O)(=O)c3ccccc3F 4P-550S c1ccc(cc1)C(=O)N2CCN(CC2)S(=O)(=O)c3ccccc3C(F)(F)F 4P-551S c1ccc(cc1)c2cc(c(o2)NC(=O)c3cccc(c3Cl)Cl)C#N 4P-564S COc1ccccc1C(=O)N(c2c(cc(o2)c3ccccc3)C#N)C(=O)c4ccccc4OC 4P-567S c1ccc(cc1)c2cc(c(o2)N(S(=O)(=O)c3ccc(cc3)F)S(=O)(=O)c4ccc(cc4)F)C#N 4P-568S COc1ccc(cc1)S(=O)(=O)N(c2c(cc(o2)c3ccccc3)C#N)S(=O)(=O)c4ccc(cc4)OC 4P-569S c1ccc(cc1)c2cc(c(o2)NC(=O)c3cccs3)C#N 4P-570S CC(C)C(=O)Nc1c(cc(o1)c2ccccc2)C#N 4P-571S c1ccc(cc1)c2cc(c(o2)N(S(=O)(=O)c3ccc(cc3)Cl)S(=O)(=O)c4ccc(cc4)Cl)C#N 4P-572S c1ccc(cc1)c2cc(c(o2)NC(=O)c3ccccc3)C#N 4P-574S c1ccc(cc1)c2cc(c(o2)N(S(=O)(=O)c3ccccc3)S(=O)(=O)c4ccccc4)C#N 4P-575S Cc1ccc(cc1)C(=O)Nc2c(cc(o2)c3ccccc3)C#N 4P-578S Cc1ccc(cc1)S(=O)(=O)N(c2c(cc(o2)c3ccccc3)C#N)S(=O)(=O)c4ccc(cc4)C 4P-580S CCCC(=O)Nc1c(cc(o1)c2ccccc2)C#N 4P-582S Cc1c(n(c(c1C#N)NC(=O)Nc2cccc(c2)C(F)(F)F)Cc3ccc(cc3)OC)C 4P-596S Cc1c(n(c(c1C#N)NC(=O)Nc2cccc(c2)Cl)Cc3ccc(cc3)OC)C 4P-597S Cc1c(n(c(c1C#N)NC(=O)Nc2ccc(cc2)Cl)Cc3ccc(cc3)OC)C 4P-602S Cc1cccc(c1)NC(=O)Nc2c(c(c(n2Cc3ccc(cc3)OC)C)C)C#N 4P-603S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccccc5Cl 4P-643S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)C(F)(F)F 4P-644S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc(cc5)Cl 4P-645S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)Cl 4P-646S Cc1cc(nc(c1C#N)Sc2ccccc2NC(=O)c3cccs3)C 4P-647S Cc1cc(nc(c1C#N)Sc2ccccc2NC(=O)c3ccc(cc3)F)C 4P-651S Cc1cc(nc(c1C#N)Sc2ccccc2NC(=O)c3cccc(c3)OC)C 4P-652S Cc1cccc(c1)C(=O)Nc2ccccc2Sc3c(c(cc(n3)C)C)C#N 4P-653S Cn1c(c(c(n1)c2ccccc2)c3nc(no3)c4ccccc4Cl)Cl 4P-658S Cn1c(c(c(n1)c2ccccc2)c3nc(no3)c4cccc(c4)C(F)(F)F)Cl 4P-659S Cn1c(c(c(n1)c2ccccc2)c3nc(no3)c4cccc(c4)Cl)Cl 4P-660S Cn1c(c(c(n1)c2ccccc2)c3nc(no3)c4ccc(cc4)Cl)Cl 4P-661S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)C(=O)N/N=C/c4ccc(cc4)OC 4P-664S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)C(=O)N/N=C/c4ccccc4Cl 4P-665S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)C(=O)N/N=C/c4cccc(c4)C(F)(F)F 4P-666S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)C(=O)N/N=C/c4ccc(cc4Cl)Cl 4P-669S c1cc(cc(c1)Cl)c2nc(on2)C3CCCN3S(=O)(=O)c4ccc(cc4)Cl 4P-670S c1cc(ccc1c2nc(on2)C3CCCN3S(=O)(=O)c4ccc(cc4)Cl)Cl 4P-671S c1ccc(c(c1)c2nc(on2)C3CCCN3S(=O)(=O)c4ccc(cc4)Cl)Cl 4P-672S c1cc(cc(c1)C(F)(F)F)c2nc(on2)C3CCCN3S(=O)(=O)c4ccc(cc4)Cl 4P-673S Cc1c(cccc1Cl)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)C(F)(F)F 4P-674S Cc1c(cccc1Cl)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc(cc5)Cl 4P-675S Cc1c(cccc1Cl)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)Cl 4P-676S Cc1c(cccc1Cl)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccccc5Cl 4P-677S CCOC(=O)C(Cc1ccc(cc1Cl)Cl)C(=O)/C=C/N(C)C 4P-701 c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)CC3CC3)O 4P-702 CCOC(=O)CNC=C(C(=O)OCC)C(=O)OCC 4P-704 c1ccc(cc1)/C=C/Cc2c(ccn(c2=O)CCc3ccccn3)O 4P-705 c1c(cnc(c1Cl)O)C(F)(F)F 4P-706 CCOC(=O)C(=CNCC(=O)OC)C(=O)OCC 4P-707 CCOC(=O)C(Cc1c(cccc1Cl)F)(Cc2c(cccc2Cl)F)C(=O)C 4P-708 CCOC(=O)Cn1ccc(c(c1=O)Cc2ccc(cc2Cl)Cl)O 4P-711 c1ccc(cc1)CCn2ccc(c(c2=O)Cc3ccc(cc3Cl)Cl)O 4P-712 c1ccc2c(c1)c(c[nH]2)CCn3ccc(c(c3=O)Cc4ccc(cc4Cl)Cl)O 4P-713 c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)Cc3ccncc3)O 4P-714 c1cc(ccc1Cn2ccc(c(c2=O)Cc3ccc(cc3Cl)Cl)O)Cl 4P-715 Cn1cccc1C(=O)Nn2ccc(c(c2=O)Cc3ccc(cc3Cl)Cl)O 4P-717 CCOC(=O)C(C(=O)C)(C/C=C\c1ccccc1)C/C=C\c2ccccc2 4P-719 CCOC(=O)C(Cc1ccc(cc1Cl)Cl)C(=O)/C=C/NCC(F)(F)F 4P-721 c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)CC(F)(F)F)O 4P-722 c1ccn2c(c1)c(cc(c2=O)N)C#N 4P-723 Cc1cc(no1)NC(=O)CC2N(C(=O)N(O2)C)c3ccc(cc3)Cl 4P-724 c1cc(ccc1NN/C=N\c2c3ccsc3ncn2)F 4P-725 c1ccc(cc1)C(c2ccc[nH]2)c3ccc[nH]3 4P-901 c1cc([nH]c1)C(c2ccc(cc2)[N+](=O)[O-])c3ccc[nH]3 4P-902 CC1(OC(=O)C(C(=O)O1)Cc2c[nH]c3c2cccc3)C 4P-907 CC(C)(C)OC(=O)CSC1=Nc2ccccc2C3=NC(=O)CN31 4R-0001 c1ccc(cc1)CN2CCN(CC2)C(=S)NC(=O)c3ccccc3 4R-0002 c1ccc(cc1)n2ccnc2SCC(C(F)(F)F)O 4R-0003 Cc1ccc(cc1)S(=O)(=O)NNC(=O)C2CC=CCC2C(=O)O 4R-0004 Cc1ccccc1CSc2nccn2c3ccccc3 4R-0005 c1cc(cc(c1)C(F)(F)F)C(=O)Nn2cnnc2 4R-0008 COc1ccc(cc1)C(=O)Nn2cnnc2 4R-0009 Cc1cc(c2nncn2n1)OC(=O)c3ccc(cc3)F 4R-0010 Cc1cc(c2nncn2n1)OC(=O)c3cccs3 4R-0011 COC(=O)CCCSC1=Nc2ccccc2C3=NC(=O)CN31 4R-0013 c1ccc2c(c1)C3=NC(=O)CN3C(=N2)SCc4ccc(cc4)Br 4R-0014 c1cc(ccc1C(=O)Nn2cnnc2)F 4R-0015 c1cc(sc1)C(=O)Nn2cnnc2 4R-0016 c1cc(cc(c1)OCCCSc2ccc(c(c2)Cl)Cl)C(F)(F)F 4R-0020 Cc1ccc(cc1)C(=O)Oc2cc(nn3c2nnc3)C 4R-0021 Cc1ccc(cc1)C(=O)Nn2cnnc2 4R-0022 CC(C(=O)OC)Sc1nccn1c2ccccc2 4R-0023 CC1(C(=O)NC(CS1)C(=O)OC)C 4R-0024 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCCOCCSCC(C(=O)O)NC(=O)OC(C)(C)C 4R-0025 CC(C)(C)OC(=O)CSc1nccn1c2ccccc2 4R-0026 c1cc(ccc1N2CCN(CC2)C(=O)C3CC=CCC3C(=O)O)[N+](=O)[O-] 4R-0027 COC(=O)CCCSc1nccn1c2ccccc2 4R-0028 c1ccc(cc1)n2ccnc2SCc3cccc(c3)Cl 4R-0032 Cc1ccccc1CSC2=Nc3ccccc3C4=NC(=O)CN42 4R-0033 c1ccc2c(c1)C3=NC(=O)CN3C(=N2)SCc4ccc(cc4)C(F)(F)F 4R-0034 c1ccc2c(c1)C3=NC(=O)CN3C(=N2)SCc4cccc(c4)F 4R-0035 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nn2cnnc2 4R-0036 CN(C)/C=N/n1cnnc1 4R-0037 c1cc(ccc1F)S(=O)(=O)Nn2cnnc2 4R-0038 COc1ccc(cc1)S(=O)(=O)Nn2cnnc2 4R-0039 COC(=O)C1CC2C(O2)CC1C(=O)OC 4R-0040 COc1cc(cc(c1)OC)NC(=O)C2CC=CCC2C(=O)O 4R-0041 c1cc(sc1)C(=O)NNC(=O)C2CC=CCC2C(=O)O 4R-0042 c1ccc(c(c1)N)N2C(=O)C3CC=CCC3C2=O 4R-0044 c1ccc2cc(ccc2c1)S(=O)(=O)Nn3cnnc3 4R-0045 c1ccc(c(c1)C(=O)Nn2cnnc2)C(=O)O 4R-0046 c1ccc2c(c1)C3=NC(=O)CN3C(=N2)SCc4c(cccc4Cl)F 4R-0048 c1ccc2c(c1)C3=NC(=O)CN3C(=N2)SCc4ccc(cc4Cl)Cl 4R-0049 CCc1ccc(cc1)CSC2=Nc3ccccc3C4=NC(=O)CN42 4R-0051 c1ccc2c(c1)C(=O)N(C2=O)n3cnnc3 4R-0052 CCOC(=O)CNC(=S)Nn1cnnc1 4R-0053 c1ccc(cc1)n2ccnc2SCc3c(cccc3Cl)F 4R-0054 Cc1c(c(n2c(n1)cc(n2)c3c(ccs3)n4cccc4)O)Cc5ccccc5 4R-0056 CCCc1cc(n2c(n1)cc(n2)c3c(ccs3)n4cccc4)O 4R-0057 c1cnc([n+](c1)[O-])N.C1C=CC[C@@H]([C@@H]1C(=O)O)C(=O)O 4R-0058 c1ccc(c(c1)CSC2=Nc3ccccc3C4=NC(=O)CN42)F 4R-0059 c1ccc2c(c1)C3=NC(=O)CN3C(=N2)SCc4cnc(s4)Cl 4R-0060 CC(C(=O)O)Sc1nccn1c2ccccc2 4R-0061 c1ccc(cc1)n2ccnc2SCc3ccc(cc3Cl)Cl 4R-0065 Cc1ccc(cc1)CSC2=Nc3ccccc3C4=NC(=O)CN42 4R-0067 Cc1ccc(cc1)S(=O)(=O)Oc2cc(nn3c2nnc3)C 4R-0068 Cc1cc(c2nncn2n1)OS(=O)(=O)c3ccc(cc3)OC 4R-0069 CCOc1c(cc(cn1)Br)C(=O)O 4R-0072 c1ccc(cc1)n2ccnc2SCCCC(=O)O 4R-0073 c1ccc(cc1)n2ccnc2SCc3ccccc3F 4R-0076 c1ccc(cc1)n2ccnc2SCc3ccc(cc3)Br 4R-0080 C=CCSc1nccn1c2ccccc2 4R-0081 c1ccc(cc1)CCSc2nccn2c3ccccc3 4R-0082 CCc1ccc(cc1)CSc2nccn2c3ccccc3 4R-0083 COc1ccc(cc1OC)Cc2cccc(c2C#N)O 4R-0084 COc1cc2c(cc1OC)NC(=S)N3C2=NC(=O)C3 4R-0087 CN1C(=O)C(C(=O)N(C1=O)C)CCCC(=O)OC 4R-0088 c1ccc(cc1)n2ccnc2SCC(=O)O 4R-0091 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccn(n3)C(=O)c4ccc(cc4)[N+](=O)[O-] 4R-0200 COC(c1ccnc2n1ncc2C#N)OC 4R-0201 c1cc(c(cc1Cl)Cl)C(C#N)c2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 4R-0202 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccnc(n3)c4ccncc4 4R-0203 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccnc(n3)N 4R-0204 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccnc4n3ncn4 4R-0205 CN(CCOc1ccc(cc1)c2ccnc(n2)N)c3ccccn3 4R-0207 c1cc(cnc1)c2nccc(n2)NC(=O)/C=C/c3ccc(cc3)OCCCF 4R-0208 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccnc4n3ncc4C#N 4R-0209 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)C(=O)c4ccc(cc4)[N+](=O)[O-] 4R-0210 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5ccc(cc5)Cl 4R-0211 c1ccc(cc1)NC(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 4R-0212 Cc1ccc(cc1)c2nc3c(c(ccn3n2)c4ccccc4)C#N 4R-0216 C#CCNC(=O)c1ccc(cc1Cl)OCc2ccccc2 4R-0217 COC(c1ccnc(n1)c2cccnc2)OC 4R-0218 c1ccc(cc1)COc2ccc(c(c2)Cl)C(=O)NCc3ccc(cc3)Cl 4R-0219 c1ccc2c(c1)cc(cn2)/C=C/C(=O)NNc3ccc(cc3)F 4R-0220 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])C\2CCCC/C2=N/O 4R-0221 Cc1ccc(cc1)NC(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 4R-0223 Cc1cc2nccc(n2n1)C(OC)OC 4R-0224 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])C\2CCCC/C2=N\OC(=O)NC3CCCCC3 4R-0225 CCNC(=O)O/N=C/1\CCCCC1c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] 4R-0227 c1ccc(c(c1)NC(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl 4R-0229 c1ccc(cc1)C(C#N)c2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 4R-0231 c1ccc(c(c1)C(=O)Nc2ccnc(n2)c3cccnc3)Cl 4R-0232 Cc1cccc(c1)C(=O)Nc2ccnc(n2)c3cccnc3 4R-0233 c1cc(cc(c1)OCc2c(cccc2Cl)F)C(=O)/C=C/Nc3cccc(c3)[N+](=O)[O-] 4R-0234 Cc1ccc(cc1)S(=O)(=O)Nc2ccnc(n2)c3cccnc3 4R-0238 c1cc(cc(c1)Cl)Cn2ccc(n2)c3cccc(c3)OCc4c(cccc4Cl)F 4R-0240 COCCNC(=O)N 4R-0241 COC(=O)/C=C/OC(=O)c1ccc(cc1)[N+](=O)[O-] 4R-0243 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)C(=O)c4ccc(c(c4)Cl)Cl 4R-0244 COc1ccc(cc1Cl)N/C=C/C(=O)c2ccccc2OCc3ccc(cc3Cl)Cl 4R-0245 CCc1ccc(cc1)N/C=C/C(=O)c2cccc(c2)OCc3ccc(cc3Cl)Cl 4R-0246 c1cc(ccc1C#N)N2CCNCC2 4R-0247 c1ccc(cc1)COc2ccc(cc2)/C=N/O 4R-0248 c1ccc(c(c1)Cn2ccc(n2)c3cccc(c3)OCc4c(cccc4Cl)F)F 4R-0249 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)C(=O)c4ccc(cc4)I 4R-0250 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)C(=O)c4ccc(cc4)Cl 4R-0251 Cc1cc2nccc(n2n1)c3cccc(c3)OCc4ccc(cc4Cl)Cl 4R-0252 COc1ccc(cc1)C(=O)n2ccc(n2)c3cccc(c3)OCc4ccc(cc4Cl)Cl 4R-0253 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)C(=O)c4cccs4 4R-0254 c1cc(cnc1)c2nccc(n2)NC(=O)c3cccs3 4R-0255 CO/N=C/c1ccc(cc1)OCc2ccccc2 4R-0256 COc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0260 c1cc(ccc1C#N)N2CCN(CC2)C(=O)c3ccc(cc3)Cl 4R-0261 CCOC(=O)C(Cc1ccc(cc1)OCc2c(cccc2Cl)F)(C(=O)OCC)NC(=O)C 4R-0262 COc1ccc(cc1)C(=O)Nc2ccnc(n2)c3cccnc3 4R-0265 Cc1ccc(cc1)NC(=O)Nc2ccnc(n2)c3cccnc3 4R-0266 c1cc(ccc1NC(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl 4R-0267 c1cc(cc(c1)NC(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])C(F)(F)F 4R-0268 c1cc(ccc1C#N)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 4R-0272 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0273 c1ccc(cc1)COc2ccc(cc2)/C=N/OC(=O)c3ccc(cc3)Cl 4R-0274 Cc1ccc(cc1)C(=O)Nc2ccnc(n2)c3cccnc3 4R-0276 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3cccc(c3)OCc4c(cccc4Cl)F 4R-0277 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)/C=C/O 4R-0278 c1ccc(cc1)c2ccn3c(c2C#N)nc(n3)c4cccs4 4R-0280 Cc1cc(c(c(c1)C)S(=O)(=O)Nc2ccnc(n2)c3cccnc3)C 4R-0282 c1cc(cnc1)c2nccc(n2)NS(=O)(=O)c3ccc(cc3)Cl 4R-0283 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)S(=O)(=O)c4ccc(cc4)F 4R-0284 Cc1ccc(cc1)C(=O)n2ccc(n2)c3cccc(c3)OCc4ccc(cc4Cl)Cl 4R-0285 c1ccc(cc1)COc2ccc(cc2)/C=N/OC(=O)c3ccc(cc3)F 4R-0286 c1ccc(cc1)COc2ccc(cc2)/C=N/OC(=O)c3ccc(cc3)C(F)(F)F 4R-0287 c1ccc(cc1)COc2ccc(cc2)/C=N/OC(=O)c3cccs3 4R-0288 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccn(n3)S(=O)(=O)c4ccc(cc4)F 4R-0289 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)S(=O)(=O)c4cc(ccc4Cl)Cl 4R-0290 c1cc(cc(c1)OCc2c(cccc2Cl)F)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl 4R-0291 Cc1cc(c(c(c1)C)S(=O)(=O)n2ccc(n2)c3cccc(c3)OCc4ccc(cc4Cl)Cl)C 4R-0292 CCOc1ccc(cc1)Oc2c(nc3ccccc3n2)Cc4ccccc4 4R-0293 COc1ccc(cc1)Oc2c(nc3ccccc3n2)Cc4ccccc4 4R-0294 c1cc(cc(c1)Cl)NC(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 4R-0295 c1cc(ccc1C#N)N2CCN(CC2)C(=O)c3ccc(cc3)C(F)(F)F 4R-0296 c1cc(ccc1C#N)N2CCN(CC2)C(=O)c3ccc(cc3)F 4R-0297 c1cc(ccc1C#N)N2CCN(CC2)S(=O)(=O)c3ccc(cc3Cl)Cl 4R-0298 c1cc(ccc1C#N)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl 4R-0299 c1cc(sc1)C(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0300 COc1cccc(c1)C(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0301 CC(C)(C)c1ccc(cc1)C(=O)O/C=C/C(=O)OC 4R-0302 c1cc(c(c(c1)Cl)Cl)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0304 c1cc(ccc1C#N)N2CCN(CC2)S(=O)(=O)c3ccc(c(c3)Cl)Cl 4R-0305 c1cc(cc(c1)Cl)NC(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0306 COC(=O)/C=C/OC(=O)c1ccc(cc1)C(F)(F)F 4R-0307 c1cc(cc(c1)Cl)C(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0308 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)Cc4ccc(cc4)F 4R-0311 c1ccn(c1)c2ccnc(n2)c3cccnc3 4R-0312 COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0313 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)C#N 4R-0314 c1ccc(cc1)c2ccn3c(c2C#N)nc(n3)c4cccc(c4)C(F)(F)F 4R-0315 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)c3ccn(n3)Cc4ccc(c(c4)Cl)Cl 4R-0316 Cc1cccc(c1)Cn2ccc(n2)c3cccc(c3)OCc4ccc(cc4Cl)Cl 4R-0317 c1ccc(cc1)Cc2c(nc3ccccc3n2)Oc4ccc(c(c4)Cl)Br 4R-0319 Cc1ccc(c(c1)C)Oc2c(nc3ccccc3n2)Cc4ccccc4 4R-0320 c1ccc(cc1)Cc2c(nc3ccccc3n2)Oc4cccc(c4)F 4R-0321 c1cc(cc(c1)Cl)Cn2cc(cc2C#N)C(=O)Cc3ccc(cc3)Cl 4R-0323 COc1cc(cc(c1OC)OC)C(=O)O/C=C/C(=O)OC 4R-0326 COC(=O)/C=C/OC(=O)c1ccc(cc1)N 4R-0328 CC(=O)c1ccccc1OCc2ccc(cc2)Cl 4R-0329 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)C/C=N/OCc3ccc(cc3)Cl 4R-0330 Cc1ccccc1Cn2cc(cc2C#N)C(=O)Cc3ccc(cc3)Cl 4R-0331 Cc1cccc(c1)COc2ccc(c(c2)F)c3ccccc3 4R-0332 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)C/C=N/OCc3ccc(cc3Cl)Cl 4R-0333 c1cc(cc(c1)OCc2ccc(cc2Cl)Cl)C(=O)C/C=N/OCc3c(cccc3Cl)Cl 4R-0334 c1ccc2c(c1)CCc3ccccc3N2/C=C/C(=O)C(F)(F)F 4R-0600 c1ccc(cc1)N2CCN(CC2)/C=C/C(=O)C(F)(F)F 4R-0601 c1ccc(cc1)/N=N/c2ccc(cc2)N/C=C/C(=O)C(F)(F)F 4R-0602 c1ccc(cc1)Oc2ccccc2N/C=C/C(=O)C(F)(F)F 4R-0605 c1ccc(cc1)S(=O)(=O)c2ccc(cn2)[N+](=O)[O-] 4R-0606 Cc1cc(cnc1NC(=O)c2ccco2)I 4R-0607 c1ccc(cc1)S(=O)(=O)c2c(cccn2)N 4R-0608 c1ccc(cc1)C(=O)N2CCN=C(C=C2)C(F)(F)F 4R-0609 c1ccc(cc1)CN/C=C/C(=O)C(F)(F)F 4R-0611 c1ccc(cc1)CN2CCN(CC2)/C=C/C(=O)C(F)(F)F 4R-0612 Cc1cc(nc2c1c(nn2C)N)C 4R-0613 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2cc(cc(c2O)OC)Br 4R-0615 COc1cc(cc(c1O)/C=N/Cc2cccc(c2)C(F)(F)F)Br 4R-0616 c1ccnc(c1)SCC(C(F)(F)F)O 4R-0617 Cc1cc(nc2c1c(nn2C)NC(=O)Nc3cccc(c3)F)C 4R-0618 c1cnc(nc1)SC[C@H](C(F)(F)F)O 4R-0619 c1ccc2c(c1)c(c[nH]2)CCN/C=C/C(=O)C(F)(F)Cl 4R-0621 Cc1cc(nc2c1c(n[nH]2)NC(=S)NC(=O)c3ccccc3)C 4R-0622 c1cc2nc(cn2cc1Cl)C(=O)O 4R-0623 c1ccc2c(c1)c(cn2Cc3ccc(cc3)C(F)(F)F)CCN4CCS(=O)(=O)CC4 4R-0625 Cn1c2c(c(n1)C(F)(F)F)c(n[nH]2)N 4R-0626 c1c(cnc(c1Cl)SCC(C(F)(F)F)O)C(F)(F)F 4R-0628 Cc1cc(nc2c1c(nn2Cc3ccc(c(c3)Cl)Cl)n4cccc4)C 4R-0631 c1ccc(cc1)CN2CCN(CC2)/C=C/C(C(F)(F)F)O 4R-0632 c1ccc2c(c1)nc(s2)SCC(C(F)(F)F)O 4R-0635 c1cc(cc(c1)F)NC(=O)OCc2cnc(s2)Cl 4R-0638 c1ccc(c(c1)C(=O)OCc2cnc(s2)Cl)Cl 4R-0639 c1cc(c(c(c1)F)C(=O)OCc2cnc(s2)Cl)F 4R-0641 Cc1cc(nc2c1c(nn2CC#N)n3cccc3)C 4R-0642 Cc1cccc(c1)Cn2c3c(c(cc(n3)C)C)c(n2)n4cccc4 4R-0643 Cc1cc(nc2c1c(nn2Cc3cnc(s3)Cl)n4cccc4)C 4R-0644 c1ccc2c(c1)c(cn2Cc3ccc(c(c3)Cl)Cl)CCN4CCS(=O)(=O)CC4 4R-0645 Cc1cc(nc2c1c(n[nH]2)NC(=S)N)C 4R-0647 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)Nc3cccc(c3)F)C 4R-0649 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)Nc3ccccc3Cl)C 4R-0650 CCNC(=O)Nc1ccc(nc1)n2c(c(c(n2)C)C(=O)OCC)C 4R-0651 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)Nc3ccccc3)C 4R-0652 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)Nc3ccc(cc3)C)C 4R-0653 c1[nH]c2c(n1)c(ncn2)SCC(C(F)(F)F)O 4R-0654 c1cc(cc(c1)NCCC(C(F)(F)F)O)C(F)(F)F 4R-0656 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=S)NC(=O)c3ccccc3)C 4R-0657 c1cc(ccc1C(=O)NN2CCS(=O)(=O)CC2)C(F)(F)F 4R-0659 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=S)N)C 4R-0661 c1ccc2c(c1)c(c[nH]2)CCN3CC(CC3=O)C(=O)O 4R-0665 Cc1ccc(cc1)C(=O)n2c3c(c(cc(n3)C)C)c(n2)n4cccc4 4R-0666 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)/C=C\C(=O)O)C 4R-0667 c1cc(ncc1Cl)N/C=C/C(=O)C(F)(F)F 4R-0668 COC(=O)c1ccc(cc1)N2CCS(=O)(=O)CC2 4R-0669 Cc1c(c(n(n1)c2ccc(cn2)N)C)C(=O)O 4R-0670 Cc1ccc(cc1)C(=O)n2cc(c3c2cccc3)CCN4CCS(=O)(=O)CC4 4R-0673 c1cc(ccc1NCCC(C(F)(F)F)O)OC(F)(F)F 4R-0676 COc1ccc(cc1)NC(=O)OCc2cnc(s2)Cl 4R-0677 CCOC(=O)c1c(nn(c1C)c2c(cc(cn2)C(F)(F)F)Cl)C 4R-0678 c1cc(ncc1C(F)(F)F)NN 4R-0680 Cc1cc(ccc1NC(=O)Cn2cncn2)Cl 4R-0800 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccncn3 4R-0803 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)NC 4R-0804 c1ccc2c(c1)c(c[nH]2)CCNc3cccc(n3)F 4R-0805 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3ccc(cc3)Cl 4R-0806 Cc1c(sc(n1)c2ccccc2Cl)C(=O)C 4R-0807 c1cc(ccc1n2c(c(cn2)n3cncn3)O)Cl 4R-0809 Cc1ccc(cc1/N=C/c2ccc(c(c2)OC)OC)[N+](=O)[O-] 4R-0810 c1cc2c(cc1CNC(=O)Cn3cncn3)OCO2 4R-0812 c1cc(ccc1CC(=O)O)Oc2c(cc(cn2)C(F)(F)F)Cl 4R-0813 CC(C)(C)c1ccc(cc1)n2c(c(cn2)n3cncn3)O 4R-0814 CC(=O)c1ccc(cc1)n2cc(nn2)C(=O)c3ccccn3 4R-0816 Cc1c(sc(n1)c2ccccc2Cl)C(=O)/C=C/N(C)C 4R-0817 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)NC(=O)C 4R-0818 CC(=O)c1cnc(s1)c2ccccc2Cl 4R-0819 CC(=O)c1ccc(cc1)n2cc(nn2)c3ccccc3 4R-0820 COC(=O)Cn1cncn1 4R-0821 Cc1c(sc(n1)c2ccccc2Cl)c3ccnc(n3)N 4R-0823 Cc1c(sc(n1)c2ccccc2Cl)c3ccn[nH]3 4R-0824 c1cc(ccc1n2c(c(cn2)n3cncn3)Oc4c(cc(cn4)C(F)(F)F)Cl)Cl 4R-0825 Cc1ccc(c(c1)n2c(c(cn2)n3cncn3)O)C 4R-0826 c1cc(c(cc1F)F)n2c(c(cn2)n3cncn3)O 4R-0827 c1cc(nc(c1)Cl)n2c(c(cn2)n3cncn3)O 4R-0828 CN(C)/C=C/C(=O)c1cnc(s1)c2ccccc2Cl 4R-0829 Cc1c(sc(n1)c2ccc[n+](c2)C)C(=O)/C=C/c3ccc(cc3)Cl.[I-] 4R-0830 Cc1c(sc(n1)c2cccnc2)C(=O)/C=C/Nc3ccccc3 4R-0831 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/Nc3cccnc3 4R-0833 c1ccc(c(c1)c2ncc(s2)c3ccnc(n3)N)Cl 4R-0834 Cc1ccc(cc1Cl)NC(=O)Cc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 4R-0835 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3ccc(cc3)Br 4R-1001 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3ccc(cc3)Cl 4R-1002 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3ccc(cc3Cl)Cl 4R-1003 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3cccc(c3Cl)Cl 4R-1004 Cc1ccc(cc1)SCC(=O)c2c(nc(s2)c3ccccc3)C 4R-1005 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3ccccc3C(=O)OC 4R-1006 Cc1c(sc(n1)c2ccccc2)c3csc(n3)c4ccccc4 4R-1007 Cc1c(sc(n1)c2ccccc2)C(=O)COc3ccc(c4c3cccc4)Cl 4R-1009 Cc1cccc(c1C)OCC(=O)c2c(nc(s2)c3ccccc3)C 4R-1010 CCn1c(nnc1S)c2cnn(c2c3ccccc3)c4ccccc4 4R-1011 CCn1c(nnc1SC)c2cnn(c2c3ccccc3)c4ccccc4 4R-1012 c1ccc(cc1)c2c(cnn2c3ccccc3)C(=O)NNC(=O)c4cnn(c4c5ccccc5)c6ccccc6 4R-1013 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3cccc(c3)OC 4R-1014 Cc1c(sc(n1)c2ccccc2)/C(=N/OC)/CBr 4R-1015 Cc1ccn2cc(nc2c1)c3c(nc(s3)c4ccccc4)C 4R-1016 c1ccc(cc1)c2c(cnn2c3ccccc3)c4nnc(o4)c5cnn(c5c6ccccc6)c7ccccc7 4R-1017 Cc1c(sc(n1)c2ccccc2)C(=O)CS(=O)(=O)c3ccccc3 4R-1019 Cc1c(sc(n1)c2ccccc2)/C(=N\OC)/CSc3ccccc3C(=O)OC 4R-1020 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3nc4ccccc4o3 4R-1022 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3ccccc3 4R-1024 Cc1c(sc(n1)c2ccccc2)C(=O)CSc3ccc(cc3)F 4R-1025 Cc1c(cccc1Br)NC(=O)c2c(ccs2)n3cccc3 4R-1027 Cc1cccc(c1C)NC(=O)c2c(ccs2)n3cccc3 4R-1028 Cc1c(sc(n1)c2ccccc2)C(=O)/C(=C/N(C)C)/S(=O)(=O)c3ccccc3 4R-1029 Cc1c(sc(n1)c2ccccc2)c3c(cnc(n3)c4ccccc4)S(=O)(=O)c5ccccc5 4R-1030 Cc1c(sc(n1)c2ccccc2)C(=O)COc3ccc(cc3Br)Cl 4R-1032 Cc1c(sc(n1)c2ccccc2)C(=O)COc3ccsc3C(=O)OC 4R-1033 Cc1c(sc(n1)c2ccccc2)c3c(cnc(n3)c4ccncc4)S(=O)(=O)c5ccccc5 4R-1036 Cc1c(sc(n1)c2ccccc2)c3c(cnc(n3)c4cccnc4)S(=O)(=O)c5ccccc5 4R-1037 Cc1c(sc(n1)c2ccccc2)c3c(cnc(n3)c4cccs4)S(=O)(=O)c5ccccc5 4R-1038 c1cc(ccc1S(=O)(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3)Cl 4R-1039 c1cc(ccc1S(=O)(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3)Br 4R-1040 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 4R-1041 Cc1c(sc(n1)c2ccccc2)c3c(cnc(n3)N)S(=O)(=O)c4ccccc4 4R-1042 Cc1c(sc(n1)c2ccccc2)c3c(cnn3c4ccccc4)S(=O)(=O)c5ccccc5 4R-1043 c1ccc(cc1)CSc2nnc(o2)/C=C/c3ccc(cc3Cl)Cl 4R-1060 Cc1ccc(cc1)OCC2(CCN(CC2)S(=O)(=O)c3ccc(cc3)C)O 4R-1063 c1ccc(cc1)/C=C/C(=O)NNC(=O)/C=C\c2ccccc2 4R-1066 c1ccc(cc1)/C=C/c2nnc(o2)S 4R-1067 Cc1ccc(cc1)CSc2nnc(o2)/C=C/c3ccccc3 4R-1068 CCSc1nnc(o1)/C=C/c2ccccc2 4R-1069 c1ccc(cc1)/C=C/c2nnc(o2)SCc3ccc(cc3)Cl 4R-1070 c1ccc(cc1)/C=C/c2nnc(o2)SCc3ccc(cc3Cl)Cl 4R-1071 c1ccc(cc1)/C=C/c2nnc(o2)SCc3ccc(cc3)F 4R-1072 c1ccc(cc1)/C=C/c2nnc(o2)SCc3cccc(c3)Cl 4R-1073 c1ccc(cc1)/C=C/c2nnc(o2)SCc3ccc(c(c3)Cl)Cl 4R-1074 C=CCSc1nnc(o1)/C=C/c2ccccc2 4R-1075 CSc1nnc(o1)/C=C/c2ccccc2 4R-1076 Cc1c(cnc(n1)SCC(=O)O)C(=O)C 4R-1121 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3)OC 4R-1123 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)Nc3cccc(c3)C(F)(F)F 4R-1124 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3)Cl 4R-1125 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)C3C(=O)CCCC3=O 4R-1126 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)C3C(=O)CC(CC3=O)(C)C 4R-1127 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NC3CCCCC3 4R-1128 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)N3CCOCC3 4R-1129 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NC3CC3 4R-1130 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NC(C)C 4R-1131 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)NCC=C 4R-1132 c1cc(ccc1S(=O)(=O)N2CCC(CC2)C(=O)O)Cl 4R-1137 Cc1c(cnc(n1)Oc2cc(c(cc2Cl)Cl)Cl)C(=O)C 4R-1138 Cc1c(cnc(n1)N2CCCCCC2)C(=O)N3CCCCCC3 4R-1139 Cc1c(cnc(n1)Oc2cc(ccc2Cl)Cl)C(=O)C 4R-1140 Cc1c(cnc(n1)Oc2ccc3ccccc3c2)OC 4R-1141 Cc1c(cnc(n1)NC2CCCCC2)C(=O)NC3CCCCC3 4R-1143 c1cc(ccc1S(=O)(=O)N2CCC(CC2)NC(=O)N3CCOCC3)Cl 4R-1146 COC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 4R-1149 Cc1c(cnc(n1)Sc2ccc(cc2)Cl)C(=O)C 4R-1150 CC(C)NC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 4R-1153 c1cc(ccc1S(=O)(=O)N2CCC(CC2)NC(=O)N3CCCC3)Cl 4R-1154 C=CCNC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 4R-1155 Cc1c(cno1)C(=O)NC(C)C 4R-1157 COc1cc(nc(n1)SC)C(F)(F)F 4R-1158 c1cc(ccc1COC(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)Cl 4R-1160 c1cc(ccc1S(=O)(=O)N2CCC(CC2)NC(=O)OCc3ccc(cc3Cl)Cl)Cl 4R-1161 COc1ccc(cc1)COC(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 4R-1162 CC(C)OC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 4R-1163 C=CCOC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl 4R-1164 COc1cc(nc(n1)Oc2cc(ccc2Cl)Cl)C(F)(F)F 4R-1165 COc1cc(nc(n1)Oc2cc(c(cc2Cl)Cl)Cl)C(F)(F)F 4R-1166 Cc1ccn2c(c1)nc(c2/C(=N/OC)/CSc3ccc(cc3)Cl)C 4R-1182 Cc1ccn2c(c1)nc(c2/C(=N/OCc3ccc(cc3Cl)Cl)/CSc4ccc(cc4)Cl)C 4R-1183 CC1=C(N2C=CC=CC2N1)C(=O)CN3CCN(CC3)c4ccccc4 4R-1184 Cc1ccn2c(c1)nc(c2/C(=N/OCc3ccc(cc3)F)/CSc4ccc(cc4)Cl)C 4R-1185 Cc1ccn2c(c1)nc(c2/C(=N/OCc3cccc(c3)C(F)(F)F)/CSc4ccc(cc4)Cl)C 4R-1186 Cc1cccc(c1)CO/N=C(\CSc2ccc(cc2)Cl)/c3c(nc4n3ccc(c4)C)C 4R-1187 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2c(nc3n2ccc(c3)C)C 4R-1188 Cc1ccn2c(c1)nc(c2/C(=N/OC(=O)c3ccc(cc3)Cl)/C)C 4R-1200 Cc1ccn2c(c1)nc(c2/C(=N/OC(=O)c3ccccc3)/C)C 4R-1203 Cc1ccn2c(c1)nc(c2/C(=N/OCc3ccc(cc3)Cl)/CSc4ccc(cc4)Cl)C 4R-1204 Cc1ccn2c(c1)nc(c2/C(=N/OCc3cccc(c3)Cl)/CSc4ccc(cc4)Cl)C 4R-1205 Cc1ccn2c(c1)nc(c2/C(=N/OCc3ccc(cc3)C(F)(F)F)/CSc4ccc(cc4)Cl)C 4R-1206 c1ccc-2c(c1)CCc3c2nnc(c3)SCc4ccc(c(c4)Cl)Cl 4R-1242 c1ccc-2c(c1)CCc3c2nnc(c3)SCc4ccc(cc4Cl)Cl 4R-1243 c1ccc-2c(c1)CCc3c2nnc(c3)SCc4ccc(cc4)F 4R-1244 c1ccc-2c(c1)CCc3c2nnc(c3)SCc4ccccc4Cl 4R-1245 c1ccc(cc1)CSc2cc3c(nn2)-c4ccccc4CC3 4R-1246 Cc1ccccc1CSc2cc3c(nn2)-c4ccccc4CC3 4R-1247 c1ccc-2c(c1)CCc3c2nnc(c3)SCc4cccc(c4)[N+](=O)[O-] 4R-1248 c1ccc-2c(c1)CCc3c2nnc(c3)SCc4c(cccc4Cl)Cl 4R-1250 c1ccc-2c(c1)CCc3c2nnc(c3)SCc4ccc(cc4)Cl 4R-1251 c1coc2c1C(=S)NCCC2 4R-1300 COC(=O)C1CSC(N1)c2ccc(cc2)Cl 4R-1301 CCn1c(nnc1S)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC 4R-1302 Cc1ccc(cc1)C(=O)O/N=C\2/CCCc3c2cco3 4R-1304 Cc1ccc(cc1)C(=O)N2C(CSC2c3ccc(cc3)Cl)C(=O)OC 4R-1307 Cc1ccc(cc1)C(=O)N2C(CSC2c3ccc(cc3)Cl)C(=O)NN 4R-1308 CCn1c(nnc1SCC=C)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC 4R-1309 CCn1c(nnc1SCc2ccc(cc2)C)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)OC 4R-1310 Cc1cc(nc2c1c3c(s2)c(nc(n3)S)O)C 4R-1311 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)O)C)C 4R-1312 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)Cl)C)C 4R-1313 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)N5CCOCC5)C)C 4R-1314 c1ccc(cc1)C(=O)O/N=C\2/CCCc3c2cco3 4R-1315 c1cc(ccc1C(=O)O/N=C\2/CCCc3c2cco3)Cl 4R-1317 c1cc(sc1)C(=O)O/N=C\2/CCCc3c2cco3 4R-1318 c1coc2c1/C(=N\OC(=O)C3CC3)/CCC2 4R-1319 c1cc(c(c(c1)Cl)Cl)C(=O)O/N=C\2/CCCc3c2cco3 4R-1320 COc1ccc(cc1)C(=O)O/N=C\2/CCCc3c2cco3 4R-1321 c1cc(ccc1F)S(=O)(=O)O/N=C\2/CCCc3c2cco3 4R-1322 c1cc(ccc1S(=O)(=O)O/N=C\2/CCCc3c2cco3)Br 4R-1324 c1cc(ccc1S(=O)(=O)O/N=C\2/CCCc3c2cco3)Cl 4R-1325 Cc1ccc(cc1)S(=O)(=O)O/N=C\2/CCCc3c2cco3 4R-1326 c1ccc(cc1)S(=O)(=O)O/N=C\2/CCCc3c2cco3 4R-1327 CS(=O)(=O)O/N=C\1/CCCc2c1cco2 4R-1328 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)O 4R-1329 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCC(CC2)C(=O)O 4R-1331 c1cc(ccc1S(=O)(=O)N2CCC(CC2)C(=O)O)Br 4R-1332 c1cc(ccc1F)S(=O)(=O)N2CCC(CC2)C(=O)O 4R-1333 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)O 4R-1334 c1ccc2c(c1)nc(n2CC(=O)NCc3cccnc3)C(F)(F)F 4R-1501 c1ccc(c(c1)CNC(=O)Cn2c3ccccc3nc2C(F)(F)F)Cl 4R-1502 CCOC(=O)C(C(=O)Nc1ccc(cc1)OC)NC(=O)C 4R-1504 CCOC(=O)C(C(=O)Nc1ccc(cc1C)C)NC(=O)C 4R-1505 CCOC(=O)C(C(=O)Nc1ccc(cc1)F)NC(=O)C 4R-1506 CCOC(=O)C(C(=O)Nc1cccc(c1)C(F)(F)F)NC(=O)C 4R-1507 CCOC(=O)C(C(=O)Nc1c(cccc1C)C)NC(=O)C 4R-1510 COc1ccc(cc1)CNC(=O)Cn2c3ccccc3nc2C(F)(F)F 4R-1513 c1ccc(cc1)CN2CCC3(CCNC3)CC2 4R-1514 CC(C)(C)OC(=O)N1CCC2(C1)CCN(CC2)Cc3ccccc3 4R-1515 CCOC(=O)C(C(=O)Nc1ccc(cc1)C(C)(C)C)NC(=O)C 4R-1516 CCOC(=O)C(C(=O)Nc1ccc(cc1)C(C)C)NC(=O)C 4R-1517 CC(=O)NC(C(=O)Nc1ccc(cc1)OC)C(=O)O 4R-1518 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Sc3ccc(cc3)Cl 4R-1519 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Sc3ccc(cc3)F 4R-1520 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Sc3cccc(c3)C(F)(F)F 4R-1521 c1ccc(cc1)CSc2c(nnc(n2)c3ccccc3)C(F)(F)F 4R-1522 Cc1ccc(cc1)CSc2c(nnc(n2)c3ccccc3)C(F)(F)F 4R-1523 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)SCc3cccc(c3)C(F)(F)F 4R-1524 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Oc3ccccc3 4R-1525 CC(=O)NC(C(=O)Nc1ccc(cc1)OC)C(=O)Nc2ccc(cc2)F 4R-1528 CCOC(=O)CSc1c(nnc(n1)c2ccccc2)C(F)(F)F 4R-1529 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Sc3ccccc3 4R-1530 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)N3CCOCC3 4R-1531 COC(=O)c1ccccc1NC(=O)c2ccncc2 4R-1532 CNc1c(nnc(n1)c2ccccc2)C(F)(F)F 4R-1542 CN(C)c1c(nnc(n1)c2ccccc2)C(F)(F)F 4R-1543 CN(Cc1ccccc1)c2c(nnc(n2)c3ccccc3)C(F)(F)F 4R-1544 c1ccc2c(c1)nc(n2CC(=O)N3CCCCC3)C(F)(F)F 4R-1546 c1ccc2c(c1)nc(n2CC(=O)N3CCOCC3)C(F)(F)F 4R-1547 c1ccc2c(c1)nc(n2CC(=O)N3CCCC3)C(F)(F)F 4R-1548 CC1CN(CC(O1)C)C(=O)Cn2c3ccccc3nc2C(F)(F)F 4R-1549 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)NC3CCCCC3 4R-1550 c1cc(ccc1Sc2c(nc(s2)n3c(c(cn3)C(=O)O)C(F)(F)F)c4ccc(cc4Cl)Cl)Cl 4T-0004 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(c(s2)S(=O)(=O)c3ccc(cc3)Cl)c4ccc(cc4Cl)Cl 4T-0008 Cc1cc(nc(c1C#N)O)O 4T-0009 CC(C)(C)Oc1ccc(nn1)Cl 4T-0010 c1cscc1c2cn[nH]c2N 4T-0011 Cc1c(c(n(c(=O)c1C#N)C)O)CN2CCOCC2 4T-0013 Cc1cc(n(n1)c2nc(c(s2)S(=O)(=O)c3ccc(cc3)Cl)c4ccccc4)C 4T-0014 Cc1ccc(cc1)COc2ccsc2c3[nH]c(nn3)SC(=O)Cc4ccccc4 4T-0015 CC(C)(C)Oc1ccc(cc1)Br 4T-0017 Cc1ccc(n1c2ccsc2c3cc([nH]n3)/N=c/4\c5cc(ccc5occ4C=O)F)C 4T-0024 c1ccc(cc1)C(=O)COC(=O)c2cc(cc(c2N)Cl)Cl 4T-0025 c1cc2c(cc1[N+](=O)[O-])n(c(=O)o2)CC(=O)N 4T-0026 COC(=O)c1cnn2c1C(=O)N(CC2)Cc3cccs3 4T-0039 c1ccc(cc1)c2c(sc(n2)n3c(c(cn3)c4ccc(cc4)Cl)N)Sc5ccc(cc5)Cl 4T-0040 c1cc(sc1)CN2CCn3c(cc(n3)C(=O)O)C2=O 4T-0047 c1ccc(cc1)c2c(sc(n2)n3c(c(cn3)c4ccc(cc4)F)N)Sc5ccc(cc5)Cl 4T-0050 CC(C)(C)S(=O)(=O)c1cnn(c1N)c2nc(c(s2)Sc3ccc(cc3)Cl)c4ccccc4 4T-0054 c1cc(ccc1c2cnn(c2N)c3nc(c(s3)Sc4ccc(cc4)Cl)c5ccc(cc5Cl)Cl)Cl 4T-0055 c1cc(c(cc1c2ccc3c([nH]nc3n2)N)Cl)Cl 4T-0056 c1cc(ccc1c2cnn(c2N)c3nc(c(s3)Sc4ccc(cc4)Cl)c5ccc(cc5Cl)Cl)F 4T-0057 c1ccc(cc1)c2c(sc(n2)n3c(c(cn3)c4ccsc4)N)Sc5ccc(cc5)Cl 4T-0058 c1ccnc(c1)c2cn[nH]c2N 4T-0060 c1ccc(cc1)c2c(sc(n2)n3c(c(cn3)c4cccs4)N)Sc5ccc(cc5)Cl 4T-0062 Cn1c(ccn1)N 4T-0063 c1cc(ccc1c2c(n3ccsc3n2)/C=N/NC(=O)c4ccc(cc4)C(F)(F)F)Br 4T-0200 CN1CCN(CC1)c2ccc3c(c2)[nH]c(n3)c4cccc5c4cccc5 4T-0201 CN1c2cc(ccc2OCC1=O)[N+](=O)[O-] 4T-0202 CN1CCN(CC1)c2c(ccc[nH+]2)NC(=O)c3ccc(cc3)Cl.[Cl-] 4T-0205 Cc1ccc(cc1)c2c3c(c(c(n2)SCc4ccccc4)C#N)CCCC3 4T-0208 COC(=O)c1ccc(cc1)Oc2ccc(c(c2)N)[N+](=O)[O-] 4T-0210 CN(C)/C=C/C(=O)c1ccc2c(c1)OCO2 4T-0211 c1ccc(cc1)CO/N=C/c2c(nc3n2ccs3)c4ccc(cc4)Br 4T-0212 CCCc1ccc(cc1)C(=O)/C=C/c2c(nc3n2ccs3)c4ccc(cc4)Br 4T-0213 c1ccc(c(c1)C(=O)/C=C/c2c(nc3n2ccs3)c4ccc(cc4)Br)F 4T-0214 c1cc2c(cc1c3ccn[nH]3)OCO2 4T-0220 c1ccc(cc1)c2c(c(=O)c3ccccc3[nH]2)O 4T-0221 c1cc(ccc1c2c(n3ccsc3n2)/C=N/OCC(=O)N4CCOCC4)Br 4T-0222 c1cc2c(cc1c3ccnc(n3)N)OCO2 4T-0223 CCNC(=S)Nc1ccccc1N 4T-0225 c1cc2c(cc1c3ccnc4n3ncn4)OCO2 4T-0226 c1cc2c(cc1c3ccnc4n3ncc4C#N)OCO2 4T-0227 Cc1nnc(n1Cc2ccccc2OC)c3cnn(c3N)C 4T-0228 Cc1nnc(n1Cc2ccc(cc2)Cl)c3cnn(c3N)C 4T-0229 c1cc(ccc1CC(=O)Nc2ccc(cc2Cl)Cl)O 4T-0231 CSc1nc2nccc(n2n1)c3ccc4c(c3)OCO4 4T-0232 c1ccnc(c1)C(=O)/C=C/c2c(nc3n2ccs3)c4ccc(cc4)Br 4T-0233 CC(C)(C)N/N=C(\c1ccc2c(c1)NC(=O)CO2)/c3ccccc3C(=O)O 4T-0234 c1ccc(cc1)c2nccc(n2)c3ccc4c(c3)OCO4 4T-0235 Cc1nccc(n1)c2ccc3c(c2)OCO3 4T-0236 CCOC(=O)c1cnn(c1N)c2ccc(cc2Cl)Cl 4T-0237 c1ccc2c(c1)ncn2c3ccc(cc3)c4ccnc(n4)N 4T-0238 c1ccc(cc1)c2c3c(c(c(n2)SCC(=O)c4ccccc4F)C#N)CCC3 4T-0239 COC(=O)c1ccc(cc1)c2cnco2 4T-0240 c1cc(cc(c1)OCCO/N=C/c2c(nc3n2ccs3)c4ccc(cc4)Br)C(F)(F)F 4T-0241 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)O 4T-0242 CN1CCN(CC1)c2ccc3c(c2)[nH]c(n3)c4cc(c(c(c4)OC)OC)OC 4T-0244 c1cc(c(c(c1)Cl)C(c2ccc(nn2)Sc3ccc(cc3F)F)C(=O)N)Cl 4T-0246 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)NCc4cccc(c4)Cl 4T-0249 c1ccc(cc1)c2c3c(c(c(n2)SCC(=O)c4ccc(cc4)Cl)C#N)CCC3 4T-0252 CN1CCN(CC1)c2c(ccc[nH+]2)NC(=O)c3cc(c(c(c3)OC)OC)OC.[Cl-] 4T-0253 c1cnn(c1)c2ccc(cc2)c3cnco3 4T-0254 Cc1cccc(c1)c2c3c(c4c(c(sc4n2)C(=O)C)N)CCC3 4T-0255 Cc1nnc(n1Cc2ccccc2F)c3cnn(c3N)C 4T-0260 CCOC(=O)c1c([nH]c(=O)s1)C(F)(F)F 4T-0262 CC(=O)Nc1ccccc1C(=O)N 4T-0264 c1cc(ccc1CC(=O)Nc2ccc(cc2)F)O 4T-0267 c1nc-2c(nc(nc(c2n1)N)N)N 4T-0269 Cc1nnc(n1CCNc2c(cc(cn2)C(F)(F)F)Cl)c3cnn(c3N)C 4T-0270 c1ccc(cc1)CSc2c(c3c(c(n2)c4cccc(c4)C(F)(F)F)CCC3)C#N 4T-0271 Cc1ccccc1CSc2c(c3c(c(n2)c4cccc(c4)C(F)(F)F)CCC3)C#N 4T-0272 c1ccc(c(c1)CSc2c(c3c(c(n2)c4cccc(c4)C(F)(F)F)CCC3)C#N)Cl 4T-0273 c1ccc(cc1)c2ccc(s2)CO 4T-0274 Cc1nnc(n1CC2CCCO2)c3cnn(c3N)C 4T-0276 CCCCCCCc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O 4T-0280 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)Cl)C2=O 4T-0281 c1ccc(cc1)c2nccc(n2)c3ccc(cc3)n4cnc5c4cccc5 4T-0282 c1ccc(cc1)Cn2cnc(c2C#N)C#N 4T-0283 Cc1nnc(n1Cc2cccs2)c3cnn(c3N)C 4T-0284 Cc1nnc(n1CCCN2CCOCC2)c3cnn(c3N)C 4T-0285 Cc1c(c(c2c(n1)-c3ccccc3C2=O)c4cc(c(c(c4)OC)OC)OC)C#N 4T-0286 CCCCCCCc1ccc(cc1)C2C(=C(NC3=C2C(=O)c4c3cccc4)C)C#N 4T-0287 c1cc(cc(c1)F)COc2cc(c(cc2Cl)Cl)[N+](=O)[O-] 4T-0290 c1ccc2c(c1)C3=C(C2=O)C(NC(=S)N3)c4ccc(cc4)Cl 4T-0291 Cc1nccc(n1)c2ccc(cc2)n3cnc4c3cccc4 4T-0293 c1cc(cc(c1)F)COc2cc(c(cc2Cl)Cl)N 4T-0294 CCCCCCCc1ccc(cc1)c2c(c(nc-3c2C(=O)c4c3cccc4)C)C#N 4T-0296 c1ccc(cc1)CN(Cc2ccccc2)C(=O)C3CCN(CC3)C4=C(C(=O)c5ccccc5C4=O)Cl 4T-0297 c1ccc2c(c1)CCN2C(=O)C3CCN(CC3)C4=C(C(=O)c5ccccc5C4=O)Cl 4T-0298 CCCC(=O)N/C(=C(/C#N)\[NH3+])/C#N.[Cl-] 4T-0299 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)N4CCOCC4 4T-0300 c1cc(ccc1c2ccnc(n2)N)n3cncn3 4T-0301 c1cc(ccc1c2ccn[nH]2)n3cncn3 4T-0302 CN(C1CCCCC1)C(=O)C2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl 4T-0303 c1ccc2c(c1)ncn2c3ccc(cc3)c4ccnc5n4ncn5 4T-0305 Cc1cc2nccc(n2n1)c3ccc(cc3)n4cnc5c4cccc5 4T-0306 CC1CN(CC(O1)C)C(=O)C2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl 4T-0307 CC1CCCN(C1)C(=O)C2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl 4T-0308 CC(C)(C)c1ccc(cc1)Cn2cnc(c2C#N)C#N 4T-0309 CCCCCCCc1ccc(cc1)c2c(c(nc-3c2C(=O)c4c3cccc4)/C=C/N(C)C)C#N 4T-0311 COc1cc(cc(c1OC)OC)c2c(c(nc-3c2C(=O)c4c3cccc4)/C=C/c5ccc(cc5)F)C#N 4T-0312 CCCCCCCc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=S)N2 4T-0313 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)C2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl 4T-0314 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)N4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 4T-0315 CC(C(=O)C)Oc1ccc2c(c1)OCO2 4T-0317 c1ccc2c(c1)ncn2c3ccc(cc3)c4ccnc(n4)c5ccncc5 4T-0318 c1cc(c(c(c1)Cl)Cn2cnc(c2C#N)C#N)Cl 4T-0319 c1ccc(c(c1)CNC(=O)C2CCCN2C3=C(C(=O)c4ccccc4C3=O)Cl)F 4T-0320 CN(Cc1ccccc1)C(=O)C2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl 4T-0322 Cc1c(c(c2c(n1)-c3ccccc3C2=O)c4ccccc4F)C#N 4T-0323 COC(=O)c1ccc(cc1)Oc2ccc(c(c2)N)N 4T-0326 CC1=C(C(C2=C(N1)c3ccccc3C2=O)c4ccc(cc4)Cl)C#N 4T-0327 CCCCCCCc1ccc(cc1)C2C3=C(c4ccccc4C3=O)N=C5N2C(=O)CS5 4T-0328 c1cc(ccc1C(c2cc3c(cc2O)OCO3)N4CCCC4)Br 4T-0329 CC(c1ccnc(n1)N)Oc2ccc3c(c2)OCO3 4T-0330 CC(c1ccnc(n1)c2ccccc2)Oc3ccc4c(c3)OCO4 4T-0331 Cc1c(c(c2c(n1)-c3ccccc3C2=O)c4ccc5c(c4)OCO5)C#N 4T-0332 Cc1ccc(cc1)c2c(c(nc-3c2C(=O)c4c3cccc4)C)C#N 4T-0333 Cc1c(c(c2c(n1)-c3ccccc3C2=O)c4ccco4)C#N 4T-0334 CC1C(c2cc3c(cc2OC1(C)N4CCCC4)OCO3)c5ccc(cc5)Br 4T-0335 CC1C(c2cc3c(cc2OC1(C)O)OCO3)c4ccc(cc4)Br 4T-0336 COc1cccc(c1)/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccccc5F)C#N 4T-0338 CC1C(c2cc3c(cc2OC1(C)O)OCO3)c4ccccc4Oc5cccc(c5)C(F)(F)F 4T-0341 c1ccc2c(c1)ncn2c3ccc(cc3)c4ccn(n4)C(=O)C5CCCCC5 4T-0342 Cc1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)n4cnc5c4cccc5 4T-0343 Cc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)n3cnc4c3cccc4 4T-0344 c1ccc2c(c1)ncn2c3ccc(cc3)c4ccnc(n4)c5ccccn5 4T-0345 c1ccc2c(c1)ncn2c3ccc(cc3)c4ccn(n4)C(=O)c5ccc(cc5)Cl 4T-0346 CN(C)/C=C(\c1ccc(cc1)OC)/C(=O)c2ccc(cc2)OC 4T-0351 c1cc(ccc1S(=O)(=O)n2c(ccn2)c3ccc4c(c3)OCO4)Cl 4T-0352 c1cc(ccc1F)S(=O)(=O)n2c(ccn2)c3ccc4c(c3)OCO4 4T-0353 CC(=O)Nc1ccc(cc1)S(=O)(=O)n2c(ccn2)c3ccc4c(c3)OCO4 4T-0354 c1cc(n(c1)c2nccs2)C#N 4T-0600 c1ccn2cc(nc2c1)c3cccc(c3)N 4T-0601 c1cc(c(cc1Cl)Cl)C(CC(=O)O)N 4T-0602 Cc1ccccc1CO/N=C\c2cccn2c3nccs3 4T-0603 Cc1cc(c(cc1[NH+]2CCN(CC2)c3ccccc3)N)[N+](=O)[O-].[Cl-] 4T-0604 c1ccn2cc(nc2c1)c3ccc(cc3)[N+](=O)[O-] 4T-0605 Cc1ccn2cc(nc2c1)c3cccc(c3)[N+](=O)[O-] 4T-0606 c1cc(cc(c1)N)c2cn3cc(ccc3n2)I 4T-0607 c1cnc2nc(cn2c1)c3ccc(cc3)[N+](=O)[O-] 4T-0608 c1ccc2c(c1)ncc(n2)c3cccc(c3)N 4T-0610 CC1(OC(=O)C(=Cc2cccn2c3nccs3)C(=O)O1)C 4T-0612 COC(=O)CC(c1cccc2c1cccc2)NC(=O)c3ccco3 4T-0613 COC(=O)CC(c1cccc2c1cccc2)NS(=O)(=O)c3cccs3 4T-0614 c1ccn2cc(nc2c1)c3ccc(cc3)N 4T-0615 Cc1ccn2cc(nc2c1)c3cccc(c3)N 4T-0616 c1cc(cc(c1)N)c2cn3cccnc3n2 4T-0617 c1cnc2nc(cn2c1)c3ccc(cc3)N 4T-0625 Cc1ccc(o1)C=C2C(=O)OC(OC2=O)(C)C 4T-0626 c1cc(cc(c1)[N+](=O)[O-])c2cn3cc(ccc3n2)Cl 4T-0627 c1ccc2c(c1)n3cc(nc3s2)c4cccc(c4)[N+](=O)[O-] 4T-0628 Cc1ccc(o1)/C=N/O 4T-0629 CN1CCN(CC1)C(=O)CC(c2ccc(cc2)OC)NC(=O)C(F)(F)F 4T-0630 COC(=O)CC(c1cccc2c1cccc2)NC(=O)c3cccc(c3)Cl 4T-0631 Cc1ccn2c(c1)nc(c2Cl)c3cccc(c3)[N+](=O)[O-] 4T-0632 Cc1cc(c(c(c1OCC#N)Br)C(C)C)Br 4T-0633 COc1ccc(cc1)C(CC(=O)Nc2ccc(cc2F)Cl)NC(=O)C(F)(F)F 4T-0634 c1ccc2c(c1)ccc3c2cc(c(=O)o3)C(=O)O 4T-0635 COc1ccc(cc1)C(CC(=O)N2CCCCC2)NC(=O)C(F)(F)F 4T-0637 c1ccc2c(c1)n3cc(nc3s2)c4cccc(c4)N 4T-0640 COc1ccc(cc1)C(CC(=O)N)NC(=O)C(F)(F)F 4T-0641 c1ccn2c(c1)nc(c2Br)c3ccc(cc3)[N+](=O)[O-] 4T-0645 c1c(cnc(c1Br)N)Cl 4T-0646 CCOc1ccc2c(c1)sc3n2cc(n3)c4cccc(c4)[N+](=O)[O-] 4T-0647 c1ccc2c(c1)/C(=C\c3cccn3c4nccs4)/C(=O)N2 4T-0650 c1cc(n(c1)c2nccs2)/C=C\C(=O)O 4T-0653 COc1cccc2c1oc(=O)c(c2)C(=O)N 4T-0658 c1ccc2c(c1)NC(=O)CC(S2)c3ccc(cc3)Cl 4T-0660 c1ccc2c(c1)n3cc(nc3s2)c4ccc(cc4)Cl 4T-0661 CN1C(=O)C(=Cc2cccn2c3nccs3)C(=O)N(C1=O)C 4T-0662 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2cccn2c3nccs3 4T-0663 c1cc(n(c1)c2nccs2)/C=N/NC(=O)c3ccco3 4T-0664 CC(C)c1ccc(cc1)C(CC(=O)OC)NC(=O)CCl 4T-0665 COc1cccc2c1oc(c2)c3cc[nH]n3 4T-0666 CCOC(=O)c1cn2c(c(cn2)c3ccc(cc3)Cl)nc1C(F)(F)F 4T-0800 c1cc(ccc1c2cnc3c(cnn3c2N)c4ccc(cc4)F)F 4T-0801 Cc1cc(n(n1)c2nc(cs2)C(=O)NNC(=S)NC)C(F)(F)F 4T-0802 Cc1cc(n(n1)c2nc(cs2)C(=O)NNC(=S)Nc3cccc(c3)C(F)(F)F)C(F)(F)F 4T-0803 CC(C)(C)S(=O)(=O)c1cnc2c(cnn2c1N)c3ccc(cc3)Cl 4T-0808 Cc1cc(n(n1)c2nc(cs2)C(=O)N/N=C/c3ccc(cc3)OC)C(F)(F)F 4T-0809 Cc1cc(n(n1)c2nc(cs2)C(F)(F)F)C(F)(F)F 4T-0810 Cc1ccc(n1c2ccsc2c3cc4nc(c5c(n4n3)CCC5)C)C 4T-0812 CC(c1c(cc(cn1)C(F)(F)F)Cl)OC(=O)C 4T-0813 COc1ccc(cc1)c2c(sc(n2)c3cccnc3)Sc4ccc(cc4)Cl 4T-0815 Cc1cc(n(n1)c2nc(cs2)C(=O)N/N=C/c3cccc(c3)OC)C(F)(F)F 4T-0817 Cc1cc(n(n1)c2nc(cs2)C(=O)N/N=C/c3cccnc3)C(F)(F)F 4T-0818 Cc1cc2nc(c3c(n2n1)CCC3)C 4T-0819 CCOC(=O)c1cnc2c(cnn2c1C(F)(F)F)c3ccc(cc3)Cl 4T-0822 CC(c1c(cc(cn1)C(F)(F)F)Cl)O 4T-0824 CC(=O)c1c(cc(cn1)C(F)(F)F)N2CCN(CC2)C 4T-0825 CC(=O)/C=C/c1cccc(c1)Oc2ccc(cc2)C(C)(C)C 4T-0826 Cc1c2c(n3c(n1)c(cn3)c4ccc(cc4)F)CCC2 4T-0827 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)S)C(F)(F)F 4T-0828 COC(=O)Cc1c(ccn(c1=O)Cc2[nH]c3ccccc3n2)O 4T-0829 Cc1c2c(n3c(n1)c(c(n3)C)Cl)CCC2 4T-0830 COc1ccc(cc1)c2c(sc(n2)N3CCOCC3)Sc4ccc(cc4)Cl 4T-0831 Cc1cc(n(n1)c2nc(cs2)C(=O)NNC(=S)NCC=C)C(F)(F)F 4T-0832 Cc1c2c(n3c(n1)c(c(n3)C)Br)CCC2 4T-0833 c1ccc(cc1)c2c(sc(n2)n3c(c(cn3)c4ccsc4)N)CC(=O)O 4T-0834 Cc1c2c(n3c(n1)c(cn3)c4ccc(cc4)Cl)CCC2 4T-0835 CCNC(=S)NNC(=O)c1csc(n1)n2c(cc(n2)C)C(F)(F)F 4T-0837 Cc1c(sc(n1)c2ccc(cc2)F)c3c(cnc(n3)N)Br 4T-0839 Cc1c(sc(n1)Nc2ccc(cc2)C(F)(F)F)c3ccnc(n3)N 4T-0840 c1cc(sc1)c2csc(n2)N 4T-0841 c1cc(ccc1c2cn[nH]c2N/C=C/C(=O)c3ccc(o3)c4ccc(cc4Cl)Cl)Cl 4T-0842 Cc1ccc(n1c2ccsc2c3cc4nc(c5c(n4n3)CCCC5)C)C 4T-0843 Cc1c2c(n3c(n1)c(cn3)c4ccc(cc4)Cl)CCCC2 4T-0844 CCn1c(nnc1S)c2csc(n2)n3c(cc(n3)C)C(F)(F)F 4T-0845 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)S)C(F)(F)F 4T-0846 c1ccc2cc(ccc2c1)C(=O)c3cn(nn3)c4ccc(c(c4)Cl)F 4T-0853 CN(C)/C=C/C(=O)c1cnc(s1)N(c2cccc(c2)C(F)(F)F)C(=O)c3ccccc3 4T-0854 Cc1cc2nc(c3c(n2n1)CCCC3)C 4T-0855 COc1ccc(cc1)N2CCN(CC2)C(=S)N 4T-0856 COc1cc2c(cc1OC)C3Cc4c(cnc5n4ncc5c6ccsc6)C(=O)N3CC2 4T-0859 COc1cc2c(cc1OC)C3Cc4c(cnc5n4c6ccccc6n5)C(=O)N3CC2 4T-0860 COc1cc2c(cc1OC)C3Cc4c(cnc5n4ncc5c6ccc(cc6)Cl)C(=O)N3CC2 4T-0861 COc1cc2c(cc1OC)C3Cc4c(cnc5n4ncc5c6ccc(cc6)F)C(=O)N3CC2 4T-0862 COc1cc2c(cc1OC)C3Cc4c(cnc5n4ncc5C#N)C(=O)N3CC2 4T-0863 Cc1c(c(n2c(n1)ncn2)C)C/C=C/c3ccccc3 4T-0865 Cc1cc(nc2n1nnn2)c3ccccc3 4T-0866 Cc1cc(n(n1)c2nc(cs2)C(=O)N3CCN(CC3)C)C(F)(F)F 4T-0867 COc1ccc(cc1)N2CCN(CC2)c3nc(cs3)c4ccccc4 4T-0870 Cc1c(nn(c1C)C(=S)N)C 4T-0871 Cc1ccc(n1c2ccsc2c3cc4ncc5c(n4n3)CC6c7cc(c(cc7CCN6C5=O)OC)OC)C 4T-0872 COc1ccc(cc1)N2CCN(CC2)c3nc(c(s3)CC(=O)O)c4ccccc4 4T-0873 Cc1ccc(cc1)S(=O)(=O)c2cnc3cc(nn3c2N)C 4T-0874 Cc1ccc(cc1)S(=O)(=O)c2cnc3cc(nn3c2N)c4c(ccs4)n5c(ccc5C)C 4T-0875 c1cc(ccc1c2cnn3c2nccc3c4ccc(o4)c5ccc(cc5Cl)Cl)F 4T-0876 c1cc(ccc1c2cnn3c2nccc3c4ccc(o4)c5ccc(cc5Cl)Cl)Cl 4T-0877 CN(C)c1ccc(cc1)/C=C/C=N/c2c(ccs2)C#N 4T-0879 CS(=O)(=O)c1cnc2c(cnn2c1N)c3ccc(cc3)Cl 4T-0881 Cc1cc2ncc(c(n2n1)N)S(=O)(=O)C 4T-0883 CS(=O)(=O)c1cnc2c(cnn2c1N)c3ccc(cc3)F 4T-0884 CS(=O)(=O)c1cnc2nc(nn2c1N)N3CCN(CC3)C(c4ccccc4)c5ccccc5 4T-0885 Cc1c(c(n2c(n1)nc(n2)N)C)C/C=C/c3ccccc3 4T-0886 COc1cc2c(cc1OC)C3Cc4c(cnn4c5ccccc5)C(=O)N3CC2 4T-0887 COc1cc2c(cc1OC)C3Cc4c(cnn4c5cccc(c5)C(F)(F)F)C(=O)N3CC2 4T-0888 COc1cc(cc(c1OC)OC)C2CC(=O)C=C(C2n3cncn3)O 4T-0889 CC(C)(C)c1ccc(cc1)Oc2cccc(c2)C3CC(=O)C=C(C3n4cncn4)O 4T-0890 Cc1ccc(cc1)c2ccnc(n2)n3cc(nn3)C(=O)c4ccc(cc4)C 4T-0891 Cc1ccc(cc1)C(=O)c2cn(nn2)c3ccc(c(c3)Cl)F 4T-0892 c1cc(ccc1C(=O)c2cn(nn2)c3ccc(c(c3)Cl)F)F 4T-0893 COc1ccc(cc1)N2CCN(CC2)c3nc(cs3)c4ccc(cc4)F 4T-0894 c1c(nc(s1)N2CCOCC2)C(F)(F)F 4T-0895 c1ccc(cc1)S(=O)(=O)c2cnc3c(cnn3c2N)c4ccc(cc4)Cl 4T-0897 c1ccc(cc1)S(=O)(=O)c2cnc3c(cnn3c2N)c4ccc(cc4)F 4T-0898 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4nc5nc(c(cn5n4)N)S(=O)(=O)c6ccccc6 4T-0899 CS(=O)(=O)c1cnc2c(cnn2c1N)c3ccsc3 4T-0900 Cc1ccc(cc1)S(=O)(=O)c2cnc3c(cnn3c2N)c4ccc(cc4)Cl 4T-0901 Cc1cc([nH]n1)N/C=C(\C#N)/S(=O)(=O)c2ccccc2 4T-0902 Cc1ccc(cc1)CSc2nc3ncc4c(n3n2)CC5c6cc(c(cc6CCN5C4=O)OC)OC 4T-0903 CN(C)/C=C/C(=O)c1cnc(s1)Nc2ccc(cc2)C(F)(F)F 4T-0904 COc1ccc(cc1)c2csc(n2)N 4T-0907 CCOC(=O)/C=C(\C)/Nc1ccc(cc1)Cl 4T-0908 CC(C)(CCl)C(=O)Nc1c(c2c(s1)CCCC2)C#N 4T-0910 COc1ccc(cc1)c2c(sc(n2)n3c(c(cn3)c4ccsc4)N)Sc5ccc(cc5)Cl 4T-0915 COc1cc2c(cc1OC)C3Cc4c(cnc5n4nc(n5)N)C(=O)N3CC2 4T-0919 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)S(=O)(=O)C)C 4T-0920 c1cc(c2cc(sc2c1)C(=O)NC3CC3)F 4T-1121 COc1ccc(cc1)CNC(=O)c2cc3c(cccc3s2)F 4T-1122 c1ccc(cc1)CNC(=O)c2cc3c(cccc3s2)F 4T-1123 c1cc(c2cc(sc2c1)C(=O)N3CCCC3)F 4T-1124 c1cc(cc(c1)NC(=O)c2cc3c(cccc3s2)F)C(F)(F)F 4T-1125 Cc1c(cn(n1)c2ccc(cc2)[N+](=O)[O-])c3ccccc3OC 4T-1240 Cc1c(cn(n1)c2ccc(cc2)Cl)c3ccccc3OC 4T-1242 Cc1c(cn(n1)c2ccc(c(c2)Cl)Cl)c3ccccc3OC 4T-1243 COC(=O)c1cc2c(cccc2s1)F 4T-1304 c1cc(c2cc(sc2c1)C(=O)O)F 4T-1305 CC(=O)OCn1c(=O)c(c(cn1)N2CCOCC2)Br 4T-1482 c1c(c(c(=O)n(n1)COC(=O)CCl)Br)Br 4T-1484 c1c(c(c(=O)n(n1)COC(=O)CCl)Cl)Cl 4T-1486 c1ccc(cc1)n2c(=O)c(c(cn2)Br)Br 4T-1488 Cc1ccc(cc1)Oc2cnn(c(=O)c2Br)c3ccccc3 4T-1491 COC(=O)c1cc2cc(ccc2s1)C(F)(F)F 4T-1505 c1cc2c(cc1C(F)(F)F)cc(s2)C(=O)O 4T-1506 CCN(CC)CCNC(=O)c1cc2cc(ccc2s1)C(F)(F)F 4T-1510 c1cc2c(cc1C(F)(F)F)cc(s2)C(=O)N3CCOCC3 4T-1512 c1ccc(cc1)NC(=O)c2cc3cc(ccc3s2)C(F)(F)F 4T-1513 c1cc(ccc1CNC(=O)c2cc3cc(ccc3s2)C(F)(F)F)Cl 4T-1514 C=CCNC(=O)c1cc2cc(ccc2s1)C(F)(F)F 4T-1517 c1cc2c(cc1C(F)(F)F)NC(=O)C2 4W-0019 Cc1cccc(c1N2CCN(CC2)c3cc(nc(n3)N)Cl)C 4W-0036 c1cc2c(c(c(oc2=O)O)C=O)nc1 4W-0039 Cc1ccc(cc1)c2cc(c(c(n2)C)C(=O)N)c3cc(c(c(c3)OC)OC)OC 4W-0043 c1cc(ccc1SCc2cnc(s2)Cl)Cl 4W-0045 Cc1cc(ccc1OCc2c(nc(s2)c3ccc(cc3)Cl)C)Cl 4W-0201 Cc1c(sc(n1)c2ccc(cc2)Cl)COc3ccccc3NC(=O)C 4W-0202 c1ccc2c(c1)c(c(o2)C(=O)NCc3cccc(c3)C(F)(F)F)n4cccc4 4W-0204 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)/C=C(\C#N)/c5ccc(cc5Cl)Cl 4W-0205 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)C 4W-0206 Cc1c(c(=O)n(n1C(=O)c2ccc(cc2)F)C)CCO 4W-0207 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)/C=C(\C#N)/c5cccs5 4W-0208 c1ccc2c(c1)c(c[nH]2)/C=N/NC(=O)c3ccc4c(c3)cccn4 4W-0209 Cc1ccc(cc1)CNC(=O)c2c(c3ccccc3o2)n4cccc4 4W-0210 c1cc(ccc1C(=O)OCCC2C(=O)Nc3cc(ccc3O2)Cl)F 4W-0211 Cc1c(c(=O)[nH]n1C(=O)c2ccc(cc2)F)CCO 4W-0213 Cc1c(c(=O)n(n1C(=O)c2cccc(c2)[N+](=O)[O-])C)CCO 4W-0215 Cc1c(c(=O)n([nH]1)c2ccc(cc2)F)CCOC(=O)c3ccc(cc3)F 4W-0216 CSC1=NC(=O)/C(=C/c2cn(nc2c3ccc(cc3)C4CCCCC4)c5ccccc5)/S1 4W-0217 Cc1c(c(=O)n(n1C(=O)c2ccc(cc2)OC)C)CCO 4W-0220 Cc1c(c(=O)[nH]n1C(=O)c2c(cccc2F)F)CCO 4W-0221 Cc1c(c(=O)[nH]n1C(=O)c2ccc(cc2)OC)CCO 4W-0224 Cc1c(c(=O)n([nH]1)C(=N)N)CCO 4W-0227 COc1ccc(cc1OC)/C(=C/c2cn(nc2c3ccc(cc3)C4CCCCC4)c5ccccc5)/C#N 4W-0231 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)C4CCCCC4)/C=C(\C#N)/c5cccc(c5)F 4W-0232 c1cc(ccc1C(=O)O)n2c(=O)c3c([nH]2)CCCC3 4W-0233 c1ccc2c(c1)C(CCC2O)c3ccc(c(c3)Cl)Cl 4W-0234 c1ccc(cc1)/C=C/c2c3c(c4cc(ccc4n2)Oc5ccccc5)SCC3 4W-0236 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5c(cccc5Cl)Cl)CCS4 4W-0237 c1ccc(cc1)Oc2ccc3c(c2)c4c(c(n3)/C=C/c5cccc6c5cccc6)CCS4 4W-0238 Cc1ncc2c(n1)-c3ccccc3C(C2)c4ccc(c(c4)Cl)Cl 4W-0242 CCOC(=O)c1cnn(c1N)c2ccc(cc2)C 4W-0243 CCOC(=O)c1cnn(c1N)c2ccc(cc2)F 4W-0244 CCOC(=O)c1cnn(c1I)c2ccc(cc2)F 4W-0248 CC(C)CN1CCCc2c1cccc2 4W-0249 Cc1c(sc(n1)c2ccc(cc2)Cl)CNS(=O)(=O)c3ccccc3Cl 4W-0250 CN(C)/C=N/c1nc(cs1)c2ccc3c(c2)OCO3 4W-0251 CN(C)/C=C/C(=O)c1cc(ccc1[N+](=O)[O-])N2CCOCC2 4W-0252 c1ccc\2c(c1)C(CC/C2=N\O)c3ccc(c(c3)Cl)Cl 4W-0253 CCOC(=O)CC1C(=O)Nc2ccccc2S1 4W-0254 CCCCCC(=O)NCc1c(nc(s1)c2ccc(cc2)Cl)C 4W-0256 CC(C)CN1CCCc2c1ccc(c2)C=O 4W-0257 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CN 4W-0258 c1cc(cc(c1)C(F)(F)F)c2c3c(nn2c4ccc(cc4)C(=O)O)CCC3 4W-0261 Cc1c(sc(n1)c2ccc(cc2)Cl)CNS(=O)(=O)c3ccc(cc3)C(C)(C)C 4W-0262 Cc1c(sc(n1)c2ccc(cc2)Cl)CNC(=O)c3ccco3 4W-0263 Cc1c(sc(n1)c2ccc(cc2)Cl)CNC(=O)c3ccc(cc3)C(F)(F)F 4W-0264 c1cc(c(cc1N2CCOCC2)c3ccn4c(n3)c(cn4)C#N)[N+](=O)[O-] 4W-0266 Cc1cc2nc(ccn2n1)c3cc(ccc3[N+](=O)[O-])N4CCOCC4 4W-0267 CSc1nc2nc(ccn2n1)c3cc(ccc3[N+](=O)[O-])N4CCOCC4 4W-0268 c1ccc(cc1)NNC(=O)NO 4W-0270 c1cc(c(cc1Cl)Cl)n2cc(cn2)O 4W-0271 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)CNC(=O)c3ccc(cc3)Cl 4W-0273 c1ccc2c(c1)NC(=O)C(S2)CC(=O)O 4W-0274 CCOc1ccc(cc1)/C=C/c2c3c(c4cc(ccc4n2)Oc5ccccc5)SCC3 4W-0276 c1cc2c(cc1/C=C/3\C(=O)N=C(S3)NO)OCO2 4W-0278 Cc1ccc(cc1)C(=O)NCc2c(nc(s2)c3ccc(cc3)Cl)C 4W-0279 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CNC(=O)C(C)(C)CCl 4W-0280 CCOC(=O)c1cnn(c1Br)c2ccc(cc2)C 4W-0283 c1cc2c(nc1)NC(=O)C(O2)CCOC(=O)c3ccc(cc3)Cl 4W-0284 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc3c(c2)CCCN3CC(C)C)/C#N 4W-0286 c1cc2cc(ccc2nc1)c3nnc(o3)c4ccc(cc4)Cl 4W-0287 C1CCc2c(c(=O)n([nH]2)C(=N)N)C1 4W-0288 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CNC(=O)c3ccco3 4W-0289 CCOC(=O)c1cnn(c1N)c2cccc(c2)Cl 4W-0290 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CNC(=O)c3ccc(cc3)C(C)(C)C 4W-0291 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CNC(=O)c3ccc(cc3)Cl 4W-0293 c1ccc(cc1)CC(C(=O)O)NC2=NC(=O)/C(=C\c3ccc4c(c3)OCO4)/S2 4W-0294 CC(C)C(C(=O)O)NC1=NC(=O)/C(=C\c2ccc3c(c2)OCO3)/S1 4W-0295 c1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3O 4W-0298 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CNS(=O)(=O)c3ccccc3Cl 4W-0299 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CN3CC(C3=O)(C)C 4W-0300 CC(C(=O)O)NC1=NC(=O)/C(=C/c2ccccc2n3cccn3)/S1 4W-0301 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CNC(=O)c3ccc(cc3)OC 4W-0302 CCOC(=O)c1cnn(c1Br)c2cccc(c2)Cl 4W-0304 CCOC(=O)C1CCN(CC1)c2ccc(c(c2)C(=O)C)[N+](=O)[O-] 4W-0306 c1cc(cc(c1)C(F)(F)F)c2c3c(nn2c4ccc(cc4)C(=O)NCc5ccc(cc5)Cl)CCC3 4W-0307 COc1ccc(cc1OC)c2cn(nc2C(=O)O)c3ccccc3 4W-0308 c1cc(cc(c1)C(F)(F)F)c2c3c(nn2c4ccc(cc4)C(=O)NCc5ccco5)CCC3 4W-0312 c1cc(cc(c1)C(F)(F)F)c2c3c(nn2c4ccc(cc4)C(=O)NCCC5=CCCCC5)CCC3 4W-0314 c1ccc(cc1)CCNC(=O)c2ccc(cc2)n3c(c4c(n3)CCC4)c5cccc(c5)C(F)(F)F 4W-0315 Cc1ccc(cc1)c2nc(no2)c3ccc(cc3)N4CCN(CC4)C(=O)OC(C)(C)C 4W-0318 c1ccc2c(c1)C(CCC2=C(C#N)C#N)c3ccc(c(c3)Cl)Cl 4W-0319 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NO 4W-0320 c1cc(cc(c1)Cl)n2c(c(cn2)C(=O)O)Br 4W-0321 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])C)CCO 4W-0324 c1cc(cc(c1)[N+](=O)[O-])C(=O)OCCC2C(=O)Nc3ccc(cc3O2)[N+](=O)[O-] 4W-0325 C/C(=N/O)/c1cc2c(cc1N3Cc4ccccc4C3)OCO2 4W-0326 c1ccc(cc1)n2c(nnc2S)c3ccc4c(c3)cccn4 4W-0327 c1cc(ccc1c2nc(nc(n2)N)c3ccc(cc3)Br)Br 4W-0328 c1cc(ccc1c2nc(nc(n2)N)c3ccc(cc3)Cl)Cl 4W-0329 c1cc(c(nc1)n2c(c(cn2)C#N)N)[N+](=O)[O-] 4W-0330 c1cc2c(cc1[N+](=O)[O-])OC(C(=O)N2)CCCl 4W-0331 c1cc(cc(c1)C(F)(F)F)c2nc(on2)CCC(=O)O 4W-0335 c1ccc(c(c1)C(=O)c2cnn(c2)c3ccc(cc3)C(=O)O)O 4W-0337 c1cc2c(nc1)NC(=O)C(O2)CCOC(=O)c3ccc(cc3)F 4W-0338 Cc1ccc(cc1)c2cc(n(n2)c3ccc(cc3)F)N 4W-0340 Cc1ccc(cc1)c2cc(n(n2)c3ccc(cc3)Cl)N 4W-0341 COC(=O)C(c1ccccc1)NC(=O)Cc2nc(no2)c3cccc(c3)C(F)(F)F 4W-0342 c1ccc2c(c1)c(c(cn2)C=O)Cl 4W-0344 CCOc1cc(ccc1Oc2ccc(cn2)[N+](=O)[O-])C=O 4W-0345 Cc1c2c(n[nH]1)NC3=C(C2c4ccc(cc4)NC(=O)C)C(=O)CC(C3)(C)C 4W-0401 Cc1ccc(cc1)/C=N\NC(=O)c2ccc3c(c2)cccn3 4W-0402 Cc1nc2ccc(cc2o1)C(=O)O 4W-0404 c1cc2cc(ccc2nc1)C(=O)N/N=C/c3cccs3 4W-0406 Cc1ccc(cc1)C(=O)NNC(=O)c2ccc3c(c2)cccn3 4W-0412 c1cc2cc(ccc2nc1)C(=O)NNC(=O)c3ccc(cc3)Cl 4W-0416 Cc1c2c(n[nH]1)NC3=C(C2c4ccccc4OC)C(=O)CC(C3)(C)C 4W-0418 Cc1c2c(n[nH]1)NC3=C(C2c4cccnc4)C(=O)CC(C3)(C)C 4W-0419 CC(C)(C)NC(=S)NNC(=O)c1ccc2c(c1)cccn2 4W-0420 c1cc(ccc1c2cc(n(n2)c3ccc(cc3)F)N)Br 4W-0423 CCOc1cc(ccc1O)C2c3c([nH]nc3NC4=C2C(=O)CC(C4)(C)C)C 4W-0424 Cc1ccc(cc1)c2nnc(o2)c3ccc4c(c3)cccn4 4W-0427 c1ccc(c(c1)C(=O)/C=C/c2cccs2)N 4W-0430 c1cc(ccc1c2cc(n(n2)c3ccc(cc3Cl)Cl)N)Br 4W-0432 Cc1ccc(n1c2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3)I)C 4W-0433 c1ccc(cc1)NC(=S)NNC(=O)c2ccc3c(c2)cccn3 4W-0440 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4ccc(cc4Cl)Cl)[nH]c2=O 4W-0604 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4ccccc4Cl)[nH]c2=O 4W-0605 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)CC(=O)OC 4W-0612 c1cn[nH]c1c2c(ccs2)Br 4W-0801 c1ccc2c(c1)c(n[nH]2)n3cccc3 4W-0802 Cc1cccc(c1)C(CC(=O)O)n2cccc2 4W-0804 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccnc2n3c(cc(n3)C(F)(F)F)C(F)(F)F 4W-0805 CCCCCC(=O)Nc1cccnc1n2c(cc(n2)C(F)(F)F)C(F)(F)F 4W-0806 c1cc(c(nc1)n2c(cc(n2)C(F)(F)F)C(F)(F)F)NC(=O)c3ccco3 4W-0807 c1csc\2c1C(C/C2=N\O)NC(=O)C(F)(F)F 4W-0809 c1csc2c1C3C(C2=O)N3C(=O)C(F)(F)F 4W-0810 Cc1c(c(nc(c1Br)C)OC)C#N 4W-0811 Cc1c(c(nc(c1Br)C)N2CCN(CC2)C)C#N 4W-0812 Cc1c(c(nc(c1Br)C)N2CCOCC2)C#N 4W-0813 c1ccc(c(c1)C(CC(=O)O)n2cccc2)F 4W-0815 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccc(cc3)OC)C(F)(F)F 4W-0816 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccc(cc3)NC(=O)C)C(F)(F)F 4W-0817 CCOc1c(cccn1)C(=O)Nc2ccc(cc2)Cl 4W-0818 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccccc3)C(F)(F)F 4W-0819 CCOc1c(cccn1)C(=O)/N=C\2/N(CCS2)C(=O)c3cccnc3OCC 4W-0820 CCOc1c(cccn1)C(=O)Nc2cccc(c2)C(F)(F)F 4W-0821 CCOc1c(cccn1)C(=O)NC2CCCCCC2 4W-0822 CCOc1c(cccn1)C(=O)Nc2ccc(cc2)F 4W-0823 c1cc(ccc1c2cnn3c2nccc3c4c(cc(cn4)C(F)(F)F)Cl)Cl 4W-0824 CCc1ccc(cc1)C(CC(=O)N)NC(=O)C(F)(F)F 4W-0826 COc1ccc(cc1)C(=O)COc2ccccc2C(=O)N 4W-0827 CN1CCN(CC1)CC#Cc2ccccc2 4W-0828 CCC(c1cc(cc(n1)Cl)C(F)(F)F)(C(=O)OCC)C(=O)OCC 4W-0830 CCCc1cc(cc(n1)Cl)C(F)(F)F 4W-0831 CCOc1c(cccn1)C(=O)NCc2ccc(cc2)OC 4W-0832 C/C(=N/OC(=O)c1cccc(c1)C(F)(F)F)/c2cnccn2 4W-0833 Cc1c2c(n[nH]c2nc(c1Br)C)N 4W-0834 CN1C(=O)C(SC1=O)Cc2ccc(cc2)C#N 4W-0835 COc1cc2c(cc1OC)C(=O)CC2NC(=O)CCl 4W-0836 Cc1ccc(cc1)S(=O)(=O)c2cc3ccccc3nc2N 4W-0838 Cc1ccc(cc1)S(=O)(=O)c2cc3cc(cc(c3nc2N)Br)Br 4W-0839 c1ccc(cc1)S(=O)(=O)c2cc3ccccc3nc2N 4W-0840 c1ccc(cc1)S(=O)(=O)c2cc3cc(cc(c3nc2N)Br)Br 4W-0841 CS(=O)(=O)c1cc2ccccc2nc1N 4W-0842 CS(=O)(=O)c1cc2cc(cc(c2nc1N)Br)Br 4W-0843 COc1ccc(cc1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N 4W-0844 Cc1c(c(nc(c1Br)C)Sc2ncccn2)C#N 4W-0846 CCc1ccc(cc1)C(CC(=O)N2CCN(CC2)Cc3ccccc3)NC(=O)C(F)(F)F 4W-0847 c1cc(sc1c2ccnc(n2)S)Br 4W-0848 c1cc(sc1c2ccnc(n2)S)Cl 4W-0849 c1ccc(c(c1)C(CC(=O)O)n2cccc2C(=O)C(F)(F)F)F 4W-0851 CS(=O)(=O)N(c1cccnc1n2c(cc(n2)C(F)(F)F)C(F)(F)F)S(=O)(=O)C 4W-0852 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cccnc2n3c(cc(n3)C(F)(F)F)C(F)(F)F 4W-0854 CCc1ccc(cc1)C(CC(=O)N2CCN(CC2)c3ccccc3F)NC(=O)C(F)(F)F 4W-0856 CCc1ccc(cc1)C(CC(=O)N2CCC(CC2)C(=O)OCC)NC(=O)C(F)(F)F 4W-0857 Cc1ccc(n1C(CC(=O)O)c2ccsc2)C 4W-0858 c1ccn(c1)C(CC(=O)O)c2ccc(cc2)Br 4W-0859 c1cc(c(nc1)n2c(cc(n2)C(F)(F)F)C(F)(F)F)NS(=O)(=O)c3cccs3 4W-0860 c1cc(oc1)C(=O)O/N=C/2\CC(c3c2scc3)NC(=O)C(F)(F)F 4W-0862 COc1cccc(c1)C(=O)O/N=C/2\CC(c3c2scc3)NC(=O)C(F)(F)F 4W-0863 COc1ccc(cc1)C2=COc3ccccc3C(=O)N2 4W-0865 c1ccn(c1)C(CC(=O)O)c2ccsc2 4W-0866 Cc1cc(n(n1)c2nc(cs2)C(=O)Nc3cccc(c3)C(=O)C)C(F)(F)F 4W-0867 Cc1cc(n(n1)c2nc(cs2)C(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F 4W-0868 Cc1cc(n(n1)c2nc(cs2)C(=O)NCc3cccnc3)C(F)(F)F 4W-0869 c1cc(cc(c1)NC(=O)NCCCl)C(F)(F)F 4W-0871 c1ccn(c1)C(CC(=O)O)C2CCCCC2 4W-0872 c1ccc(cc1)C(=O)c2ccccc2n3cccc3 4W-0876 c1cnc2ncnn2c1c3c(cc(cn3)C(F)(F)F)Cl 4W-0879 CSc1nc2nccc(n2n1)c3c(cc(cn3)C(F)(F)F)Cl 4W-0880 c1cc(sc1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N 4W-0881 c1ccn(c1)C(CC(=O)O)c2ccc(cc2)[N+](=O)[O-] 4W-0882 c1ccc(c(c1)C(=O)N)OCC(=O)c2ccc(cc2)Cl 4W-0883 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccccc3[N+](=O)[O-])C(F)(F)F 4W-0884 Cc1cc(n(n1)c2nc(cs2)C(=O)NNS(=O)(=O)C)C(F)(F)F 4W-0885 c1cc(cc(c1)N2CCNC2=O)C(F)(F)F 4W-0886 c1cc(ccc1F)S(=O)(=O)N(c2c(ccs2)C#N)S(=O)(=O)c3ccc(cc3)F 4W-0888 CCc1ccc(cc1)C(CC(=O)N/N=C/Cc2ccc3c(c2)OCO3)NC(=O)C(F)(F)F 4W-0889 Cc1ccc(n1C(CC(=O)O)c2ccc3c(c2)OCO3)C 4W-0890 c1ccc2c(c1)C(=O)NC(=CO2)c3ccc(cc3)Cl 4W-0891 CCOC(=O)C(=O)CC(=O)c1cccc(c1)[N+](=O)[O-] 4W-0892 c1ccc(c(c1)C(=O)N)OCC(=O)c2cccc(c2)[N+](=O)[O-] 4W-0893 C#CCOc1cccc2c1cccc2 4W-0894 C#CCOc1ccc2c(c1)OCO2 4W-0896 Cc1ccc(cc1)NC(=O)Nc2cccnc2n3c(cc(n3)C(F)(F)F)C(F)(F)F 4W-0899 c1ccn(c1)C(CC(=O)O)c2cccc(c2)Cl 4W-0900 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)Cl 4X-0200 COc1ccc(cc1OC)/C(=C/c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)/C#N 4X-0201 CSc1nc2nc(ccn2n1)c3cccc(c3)C(F)(F)F 4X-0202 c1ccc(cc1)CC2CCN(CC2)Cc3c(c(=O)cc(o3)CO)O 4X-0204 c1ccc(cc1)CN2CCN(CC2)Cc3c(c(=O)cc(o3)CO)O 4X-0205 COc1ccc(cc1)N2CCN(CC2)Cc3c(c(=O)cc(o3)CO)O 4X-0206 CN(Cc1c(c(=O)cc(o1)CO)O)CC2OCCO2 4X-0207 CN(Cc1ccccc1)Cc2c(c(=O)cc(o2)CO)O 4X-0208 CC1CCN(CC1)Cc2c(c(=O)cc(o2)CO)O 4X-0209 c1cc(cc(c1)C(F)(F)F)c2ccn3c(n2)c(cn3)c4ccc(cc4)F 4X-0214 c1cc(cc(c1)C(F)(F)F)c2ccn3c(n2)c(cn3)C#N 4X-0215 c1cc(cc(c1)N2CCN(CC2)Cc3c(c(=O)cc(o3)CO)O)C(F)(F)F 4X-0219 CC(C)CC(=O)N1CCC(CC1)(CS(=O)(=O)c2ccccc2Cl)O 4X-0220 Cc1ccccc1CS(=O)(=O)CC2(CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F)O 4X-0224 c1ccc(c(c1)CS(=O)(=O)CC2(CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F)O)Cl 4X-0225 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCC(CC2)(CS(=O)(=O)Cc3ccc(cc3)Cl)O 4X-0226 c1ccc(cc1)CS(=O)(=O)CC2(CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F)O 4X-0227 CC(C)(C)c1ccc(cc1)CS(=O)(=O)CC2(CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F)O 4X-0228 COc1ccc(cc1)CS(=O)(=O)CC2(CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F)O 4X-0229 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCC(CC2)(CS(=O)(=O)c3ccc(c(c3)Cl)Cl)O 4X-0230 Cc1cccc(c1C)N2CCN(CC2)Cc3c(c(=O)cc(o3)CO)O 4X-0231 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=C(\C#N)/c3ccc4c(c3)OCO4)Cl 4X-0234 c1cc(sc1)/C(=C/c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)/C#N 4X-0235 COc1ccc(cc1OC)NC(=O)NNC(=O)c2ccc(cc2Cl)Cl 4X-0240 CN1C(=O)C(=Cc2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)C(=O)N(C1=O)C 4X-0242 c1ccc(cc1)c2cc(=O)n([nH]2)c3[nH]c(=O)cc(n3)c4ccccc4 4X-0245 Cc1cc(=O)[nH]c(n1)n2c(=O)cc([nH]2)c3ccccc3 4X-0246 c1cc(cnc1)CN(Cc2cccnc2)Cc3c(c(=O)cc(o3)CO)O 4X-0247 c1cnc(nc1)N2CCN(CC2)Cc3c(c(=O)cc(o3)CO)O 4X-0251 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=C\3/C(=O)C4CCN3CC4)F 4X-0257 c1cc(c(cc1CC(=O)O)NC(=O)/C=C/C(=O)O)O 4X-0258 c1ccc(cc1)c2c(c3nc(c(cn3n2)CCN4CCOCC4)c5ccc(cc5)F)Br 4X-0264 CSc1c(c2nc(c(cn2n1)CCN3CCOCC3)c4ccc(cc4)F)C#N 4X-0265 c1cc(c(cc1C=C2C(=O)NC(=O)NC2=O)[N+](=O)[O-])N3CCOCC3 4X-0268 c1cc(ccc1CO/N=C/c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)C(F)(F)F 4X-0269 c1cc(cc(c1)C(F)(F)F)c2ccn3c(n2)ncn3 4X-0271 Cc1cc2nc(ccn2n1)c3cccc(c3)C(F)(F)F 4X-0278 Cc1c(c(=O)[nH]c(n1)n2c(=O)cc([nH]2)c3ccccc3)Cc4ccccc4 4X-0280 Cc1ccc(cc1)/C(=C\c2ccccc2Oc3ccc(cc3Cl)Cl)/C#N 4X-0281 CSc1c(c2nc(ccn2n1)c3cccc(c3)C(F)(F)F)C#N 4X-0283 c1ccn(c1)c2ccc(cc2)CC#N 4X-0288 C1COC(=O)C1SC(=N)N.Br 4X-0289 c1cc2c(cc1C(F)(F)F)NC(=O)C3N2CCCC3 4X-0290 c1cc(cc(c1)C(F)(F)F)c2ccnc(n2)N 4X-0293 CC(C)(C)c1ccc(cc1)/C=C(\C#N)/c2ccc(cc2)n3cccc3 4X-0294 CSc1ccc(cc1)/C=C(/C#N)\c2nc(cs2)CCN3C(=O)c4ccccc4C3=O 4X-0296 c1ccc2c(c1)n(c(=O)n2CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)CCCCl 4X-0297 Cc1ccc(cc1)/C=C(/C#N)\c2nc(cs2)CCN3C(=O)c4ccccc4C3=O 4X-0298 c1ccc(cc1)COc2ccc(cc2)/C=C(/C#N)\c3nc(cs3)CCN4C(=O)c5ccccc5C4=O 4X-0301 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)/C(=C\c4cccc(c4)C(F)(F)F)/C#N 4X-0302 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)/C(=C\c4ccc(cc4)F)/C#N 4X-0303 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)/C(=C\c4ccoc4)/C#N 4X-0305 COc1cccc(c1)/C(=C/c2ccccc2Oc3ccc(cc3Cl)Cl)/C#N 4X-0308 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(nc2)n3cccn3)Cl 4X-0309 CC(C)CN1CCCc2c1ccc(c2)/C=C(\C#N)/c3nc(cs3)CCN4C(=O)c5ccccc5C4=O 4X-0311 c1ccc(c(c1)/C=C(\C#N)/c2nc(cs2)CCN3C(=O)c4ccccc4C3=O)Oc5ccc(cc5Cl)Cl 4X-0312 c1ccc(c(c1)/C=C(\C#N)/c2cccs2)Oc3ccc(cc3Cl)Cl 4X-0313 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)/C(=C/c4ccncc4)/C#N 4X-0314 CN1CCN(CC1)c2c3ccccc3nc(n2)SC 4X-0316 COc1cccc(c1)/C(=C/c2ccc(nc2)N3CCCCC3)/C#N 4X-0317 Cn1cccc1C(=O)N/N=C\c2ccccc2Oc3ccc(cc3Cl)Cl 4X-0318 c1ccc(c(c1)/C=C(\C#N)/C(=S)N)Oc2ccc(cc2Cl)Cl 4X-0322 c1ccc(c(c1)/C=C(\C#N)/c2ccc(cc2)n3cccc3)C(F)(F)F 4X-0325 c1ccn(c1)c2ccc(cc2)/C(=C/c3ccc4c(c3)OCO4)/C#N 4X-0326 COc1ccccc1/C=C(\C#N)/c2ccc(cc2)n3cccc3 4X-0327 COc1ccc(c(c1)/C=C(\C#N)/c2ccc(cc2)n3cccc3)OC 4X-0328 c1cc(ccc1c2nc3c4ccsc4ncn3n2)Cl 4X-0329 CN(C)/C=C(/C#N)\c1ccc(cc1)n2cccc2 4X-0331 c1ccc2c(c1)ccc3c2occ(c3=O)/C=N/O 4X-0334 CCOC(=O)C1CCN(CC1)c2ccc(cn2)/C=N/NC(=O)c3cccn3C 4X-0335 c1ccc2c(c1)cccc2/C=C(\C#N)/c3ccc(cc3)n4cccc4 4X-0340 COc1ccc(cc1OC)/C=C(\C#N)/c2ccc(cc2)n3cccc3 4X-0341 CCOC(=O)C1CCN(CC1)c2ccc(cn2)C=C3C(=O)N(C(=O)N(C3=O)C)C 4X-0347 c1cc(ncc1C=C2C(=O)NC(=O)NC2=O)N3CCSCC3 4X-0348 c1cc2c(cc1Br)sc(n2)N 4X-0349 c1c(cnc(c1C=O)Cl)Cl 4X-0701 c1c(cnc(c1C(=O)O)O)S(=O)(=O)O 4X-0702 COC(=O)c1cc(ccn1)Cl 4X-0703 c1cc(c(nc1)N2CCCCC2)C#N 4X-0709 c1cc(ncc1C=O)N2CCCCC2 4X-0710 c1cc(ncc1C=O)N2CCSCC2 4X-0715 CC1CN(CC(O1)C)c2ccc(cn2)C=O 4X-0716 CCOC(=O)C1CCN(CC1)c2ccc(cn2)C=O 4X-0717 c1cc(ncc1C=O)N2CCOCC2 4X-0718 c1ccc(cc1)CN2CCN(CC2)c3ccc(cn3)C=O 4X-0719 c1ccc(c(c1)C=O)OCc2c(cccc2Cl)F 4X-0720 c1cc(cc(c1)OCc2c(cccc2Cl)F)C=O 4X-0721 CC(C)(C)Sc1ccc(cc1)Br 4X-0722 COc1ccc(cc1)C(=O)CO 4X-0724 COC(=O)c1ccc(nc1)n2cccc2 4X-0727 c1cc(ccc1C(=O)CO)Br 4X-0729 c1cc(ccc1C(=O)CO)Cl 4X-0730 CC(C)(C)Sc1ccc(cc1)C=O 4X-0731 CCOC(=O)C(C1CCCCC1)C(=O)OCC 4X-0732 CC(C)(C=O)N1CCOCC1 4X-0733 COC(=O)c1cccc(c1CN2CCCCC2)N 4X-0800 CCCCCC(=O)Nc1ccc(cc1)Oc2ccccc2C(=O)OC 4X-0804 COC(=O)c1ccccc1Oc2ccc(cc2)NS(=O)(=O)C 4X-0805 Cn\1ccc(n/c1=N/C#N)c2cccs2 4X-0806 CN(C#N)c1nccc(n1)c2cccs2 4X-0807 COC(=O)c1ccccc1Oc2ccc(cc2)NC(=O)c3ccco3 4X-0809 COC(=O)c1ccccc1Oc2ccc(cc2)NC(=O)CCCl 4X-0810 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3ccccc3C(=O)OC 4X-0812 COC(=O)c1ccccc1Oc2ccc(cc2)NC(=O)c3ccc(cc3F)F 4X-0813 CCCC(=O)CC(=O)C(F)(F)F 4X-0815 C#CCN1CCN(CC1)c2cccc(c2)C(F)(F)F 4X-0816 c1cc(ccc1/C(=N\O)/N)OCc2ccc(nc2)Cl 4X-0818 Cc1nn(c(=O)n1c2ccc(cc2)C(C)(C)C)C/C(=N/O)/N 4X-0820 Cn1c(cc(=O)n(c1=O)C)N/N=C/c2ccc3c(c2)OCO3 4X-0823 c1ccc(cc1)/N=C/c2ccc3c(c2)OCO3 4X-0824 COC(=O)c1ccccc1Oc2ccc(cc2)NS(=O)(=O)c3ccccc3 4X-0825 COC(=O)c1ccccc1Oc2ccc(cc2)NS(=O)(=O)c3cccc(c3)Br 4X-0826 CCC(C)(C)c1ccc2c(c1)NC(=O)c3cccc(c3CO2)[N+](=O)[O-] 4X-0827 Cc1ccc2c(c1)NC(=O)c3cccc(c3CO2)[N+](=O)[O-] 4X-0828 C1COCCN1N2CCS(=O)(=O)CC2 4X-0829 CC(=O)OCc1ccc(nc1)Cl 4X-0830 COC(=O)c1cc2c(ncnc2s1)N3CCC(CC3)Cc4ccccc4 4X-0832 COC(=O)c1cc2c(nc(nc2s1)N)N3CCCCC3 4X-0833 c1ccc(c(c1)NC(=S)NCCN2CCN(CC2)C(=S)Nc3ccccc3F)F 4X-0834 COc1ccccc1C(=O)NOCc2ccc(nc2)Cl 4X-0835 Cc1nc2cc(ccc2o1)CC(=O)O 4X-0836 COc1ccc(cc1OC)CC/N=C/c2ccc(c(c2)Cl)OC 4X-0837 c1cc(c(cc1CN2CCS(=O)(=O)CC2)C(F)(F)F)Cl 4X-0838 CC(=O)N1CCN(CC1)Cc2cnc(s2)Oc3ccc(cc3)I 4X-0839 c1ccc(cc1)CC2CCN(CC2)c3c4cc(sc4ncn3)C(=O)O 4X-0840 c1ccc(cc1)c2nc3cc(ccc3o2)CC(=O)O 4X-0842 c1cc(sc1)CN2CCS(=O)(=O)CC2 4X-0843 C1CCN(CC1)N2CCS(=O)(=O)CC2 4X-0844 CC1(c2c(c3cc(ccc3[nH]2)OC)CCN1)CCc4ccc(nc4)Cl 4X-0845 CC1(c2c(c3cc(ccc3[nH]2)OC)CC[NH2+]1)Cc4ccc(c(c4)OC)OC.[Cl-] 4X-0846 CCCc1cc(c(c(n1)O)C#N)C(F)(F)F 4X-0847 c1ccc(cc1)CC2CCN(CC2)c3c4cc(sc4ncn3)C(=O)NN 4X-0850 c1ccc(cc1)CN2CCC(CC2)N3CCS(=O)(=O)CC3 4X-0852 c1c(c[nH]c1C=C(C#N)C#N)C(=O)CCl 4X-0854 CC(C)(C)NNC(=O)OC(C)(C)C 4X-0858 CC(C)(C)n1c(c(cn1)C(=O)NCc2ccco2)C(F)(F)F 4X-0859 c1ccc2c(c1)C(=O)C(=Cc3cc(c[nH]3)C(=O)CCl)C2=O 4X-0860 CC(C)(C)OC(=O)NCCN1CCS(=O)(=O)CC1 4X-0861 c1ccc2c(c1)/C(=C/c3cc(c[nH]3)C(=O)CCl)/C(=O)N2 4X-0866 C1CN(CCN1CCNC(=S)NC23CC4CC(C2)CC(C4)C3)C(=S)NC56CC7CC(C5)CC(C7)C6 4X-0867 Cc1cc(n2c(n1)c(c(n2)SC)C#N)C 4X-0868 Cc1nn(c(=O)n1c2ccc(cc2)C(C)(C)C)C/C(=N/OC(=O)c3ccc(cc3)F)/N 4X-0869 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(C(C)(C)C)NC(=O)OC(C)(C)C 4X-0870 Cc1cc(ccc1NC(=S)NCCN2CCN(CC2)C(=S)Nc3ccc(cc3C)Cl)Cl 4X-0871 CCc1nc2cc(ccc2o1)CC(=O)O 4X-0873 CCCNC(=O)Nc1ccc(cc1)Oc2ccccc2C(=O)OC 4X-0874 c1ccc(cc1)C(=O)/C(=C/c2cc(c[nH]2)C(=O)CCl)/C#N 4X-0875 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3ccc(cc3)I 4X-0876 c1c(cc(cc1Cl)Cl)NC(=S)NCCN2CCN(CC2)C(=S)Nc3cc(cc(c3)Cl)Cl 4X-0877 CC(C)(C)c1ccc(cc1)NC(=S)NCCN2CCN(CC2)C(=S)Nc3ccc(cc3)C(C)(C)C 4X-0878 c1ccnc(c1)c2nc3cc(ccc3o2)CC(=O)O 4X-0880 COC(=O)c1cnc(cc1O)O 4X-0881 Cc1ccc(n1c2ccc(cc2)Oc3ccccc3C(=O)OC)c4ccco4 4X-0882 c1cc(c(nc1)NCCC(=O)O)[N+](=O)[O-] 4X-0883 c1ccc2c(c1)/C(=C/c3cnc[nH]3)/C(=O)N2 4X-0884 c1ccc2c(c1)/C(=C/c3ccc(c(c3)[N+](=O)[O-])O)/C(=O)N2 4X-0886 c1ccc2c(c1)/C(=C\c3ccc(c(c3)[N+](=O)[O-])Cl)/C(=O)N2 4X-0887 c1ccc2c(c1)/C(=C\c3cccc(c3)C(=O)O)/C(=O)N2 4X-0888 c1ccc2c(c1)/C(=C/c3ccc(cc3)F)/C(=O)N2 4X-0889 c1cc2c(cc1CC(=O)O)nc(o2)c3ccncc3 4X-0890 c1ccc2c(c1)nc3c(n2)OCC4N3CCCC4 4X-0891 CN1C(=O)C(=Cc2c[nH]c3c2cc(cc3)OC)C(=O)N(C1=O)C 4X-0892 CC(C(=O)OC)/N=C/c1ccccc1 4X-0893 c1cc(cnc1)c2nc3cc(ccc3o2)CC(=O)O 4X-0895 Cc1c(c(=O)n(n1C)c2ccccc2)/N=C\3/c4ccccc4NC3=O 4X-0897 Cc1c(c(=O)n(n1C)c2ccccc2)/N=C\3/c4cc(ccc4NC3=O)Br 4X-0898 Cc1ccc(n1C(CC(=O)O)C2CCCCC2)C 4X-0899 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl 4X-0900 COC(=O)Cc1ccc2c(c1)NC(=O)CO2 4X-0904 COc1ccc2c(c1)c(c[nH]2)CCNc3ncccn3 4X-0910 c1ccc(cc1)COc2ccc(cn2)[N+](=O)[O-] 4X-5009 COc1ccc(cc1OC)CCNCc2ccc(c(c2)Cl)OC 4X-5091 CC(C)(C)OC(=O)NC1CCN(CC1)C(c2ccccc2)C(=O)OC 4X-5096 CS(=O)(=O)c1ccc(cc1)c2csc(n2)c3cccnc3 4Y-0010 CS(=O)(=O)c1ccc(cc1)c2csc(n2)c3ccc(cc3)Cl 4Y-0016 c1cc(ccc1OCCCl)OCCCl 4Y-0018 c1ccc2c(c1)c(cn2Cc3cccc(c3)C(F)(F)F)C4=CCC5(CC4)OCCO5 4Y-0032 c1ccc(cc1)Cn2cc(c3c2cccc3)C4=CCC5(CC4)OCCO5 4Y-0033 c1cc2c(cc1Br)c(c[nH]2)C3=CCC4(CC3)OCCO4 4Y-0048 c1cc(sc1S(=O)(=O)Oc2c(c(c(c(c2F)F)F)F)F)Br 4Y-0246 c1cc(ccc1C(=O)N2CCN(CC2)C3CCCCC3)[N+](=O)[O-] 4Y-0248 c1cnc(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)[N+](=O)[O-] 4Y-0252 CCNCc1cc(ccc1Br)O 4Y-0300 C=CS(=O)(=O)Oc1c(c(c(c(c1F)F)F)F)F 4Y-0324 CCOC(=O)Cn1cccn1 4Y-0601 c1ccc(cc1)Cn2cc(cc(c2=O)Br)C(=O)O 4Y-0700 c1cc(ccc1c2ccc(cn2)[N+](=O)[O-])C(=O)O 4Y-0702 c1cc(ccc1C=O)c2ccc(cn2)[N+](=O)[O-] 4Y-0703 c1cc(ccc1c2ccc(cn2)[N+](=O)[O-])F 4Y-0704 COc1ccc(cc1)c2ccc(cn2)N 4Y-0705 c1cc(c(nc1)c2ccc(cc2)C=O)[N+](=O)[O-] 4Y-0706 c1ccc(cc1)c2ccc(cn2)N 4Y-0708 c1cc(c(nc1)c2ccc(cc2)F)[N+](=O)[O-] 4Y-0709 COc1ccc(cc1)c2c(cccn2)[N+](=O)[O-] 4Y-0710 c1ccc(cc1)CN2CCN(CC2)c3ccc(c(c3)N)[N+](=O)[O-] 4Y-0714 c1cc(c(cc1C=O)[N+](=O)[O-])N2CCCCC2 4Y-0715 COC(=O)c1ccnc(c1)Cl 4Y-0718 c1c(cncc1Br)C(=O)NN 4Y-0719 c1cnc(cc1CO)Cl 4Y-0721 CCOC(=O)c1c(nn(c1C)c2cccc(c2)Br)C 4Y-0801 Cc1c(nn(c1C(=O)O)c2cccc(c2)F)C 4Y-0802 c1cc(cnc1)c2cc[nH]n2 4Y-0803 c1cc(cnc1)c2ccnc(n2)N 4Y-0804 CCOc1c(ccc(n1)c2cccnc2)C(=O)N 4Y-0805 CC(=O)Nc1ccc(cc1OC(F)(F)F)Cl 4Y-0806 CCOC(=O)c1c(nn(c1C)c2ccccc2Br)C 4Y-0809 c1cc(c(cc1Cl)OC(F)(F)F)N 4Y-0810 Cc1c(c(n(n1)c2cccc(c2)Br)C)C(=O)O 4Y-0811 c1ccc(cc1)c2c(nc(s2)c3cccnc3)O 4Y-0813 Cc1c(c(n(n1)c2ccccc2Br)C)C(=O)O 4Y-0814 Cc1c(c(n(n1)c2ccccc2F)C)C(=O)O 4Y-0815 COC(=O)C(c1ccccc1)Oc2ccc(cc2)C=O 4Y-0816 CC1(C(=O)N(C(=O)N1c2ccc(cn2)[N+](=O)[O-])Cc3ccc(cc3)Cl)C 4Y-0819 COc1ccc(cc1)c2c3cnc4cc5c(cc4c3ccn2)OCO5 4Y-0820 CC1(C(=O)N(C(=O)N1CCCCOc2ccccc2)Cc3ccc(cc3)F)C 4Y-0821 Cc1ccc(c(c1)I)N 4Y-0823 c1ccc2c(c1)c(cn2Cc3ccc(nc3)Cl)C=O 4Y-0824 CC(=O)c1cn(c2c1cccc2)Cc3ccc(nc3)Cl 4Y-0825 Cc1cc(nc(n1)n2cc(nn2)c3cccc(c3)N4CC(C4=O)(C)C)C 4Y-0826 c1ccc(cc1)C2CC(=O)CC(=O)C2n3cncn3 4Y-0828 Cc1c(c(n2c(n1)nc(n2)N)C)Cc3ccc(cc3)Cl 4Y-0830 c1cc(ccc1C(=O)CC#N)Br 4Y-0832 c1cc(c(cc1/C=C/2\CSc3ccc(cc3C2=O)Cl)[N+](=O)[O-])Cl 4Y-0923 c1cc(ccc1/C=C/2\CSc3ccc(cc3C2=O)Cl)F 4Y-0929 c1cc(ccc1/C=C\2/CSc3ccc(cc3C2=O)Cl)C#N 4Y-0930 c1cc(ccc1c2cc(c3cc(ccc3n2)Cl)C(=O)O)Cl 4Y-0933 CCn1c2ccccc2c(c(c1=O)/C(=N/Cc3ccco3)/CC(=O)NCc4ccco4)O 4Y-0941 CC(=O)Oc1ccccc1I 4Y-0965 CC(=O)Oc1ccccc1Cl 4Y-0976 c1ccc(cc1)CNC(=O)c2cc(ccc2O)[N+](=O)[O-] 4Y-5000 c1ccc(cc1)Cn2c(=O)c3cc(ccc3oc2=O)[N+](=O)[O-] 4Y-5011 c1cc2c(c(c1)[N+](=O)[O-])CN(C2=O)CCN3CCOCC3 4Y-5014 COC(=O)c1c(ccs1)Oc2ccc(cc2)NC(=O)c3ccccc3F 4Y-5021 COC(=O)c1c(ccs1)Oc2ccc(cc2)NC(=O)CCc3ccccc3 4Y-5022 CC(C)CC(=O)Nc1ccc(cc1)Oc2ccsc2C(=O)OC 4Y-5023 CC(C)(C)C(=O)Nc1ccc(cc1)Oc2ccsc2C(=O)OC 4Y-5024 COC(=O)c1c(ccs1)Oc2ccc(cc2)NC(=O)c3cccs3 4Y-5025 COCC(=O)Nc1ccc(cc1)Oc2ccsc2C(=O)OC 4Y-5026 COC(=O)c1c(ccs1)Oc2ccc(cc2)NC(=O)C3CC3 4Y-5027 COC(=O)c1c(ccs1)Oc2ccc(cc2)NC(=O)c3ccccc3 4Y-5028 COC(=O)c1c(ccs1)Oc2ccc(cc2)NC(=O)COCc3ccccc3 4Y-5029 COC(=O)c1c(ccs1)Oc2ccc(cc2)NS(=O)(=O)c3ccccc3 4Y-5030 COC(=O)c1c(ccs1)Oc2ccc(cc2)NS(=O)(=O)C 4Y-5031 COc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)OC 4Y-5034 COC(=O)c1c(ccs1)Oc2ccc(cc2)NS(=O)(=O)Cc3ccccc3 4Y-5035 COC(=O)c1c(ccs1)Oc2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl 4Y-5036 COC(=O)c1c(ccs1)Oc2ccc(cc2)NS(=O)(=O)c3cccc(c3)F 4Y-5037 COC(=O)c1c(ccs1)Oc2ccc(cc2)NS(=O)(=O)c3cccs3 4Y-5038 COC(=O)c1c(ccs1)Oc2ccc(cc2)NS(=O)(=O)CC(F)(F)F 4Y-5039 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O)F 4Y-5040 c1ccc(cc1)CCC(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5041 CC(C)CC(=O)Nc1ccc(cc1)Oc2ccsc2C(=O)O 4Y-5042 CC(C)(C)C(=O)Nc1ccc(cc1)Oc2ccsc2C(=O)O 4Y-5043 c1cc(sc1)C(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5044 COCC(=O)Nc1ccc(cc1)Oc2ccsc2C(=O)O 4Y-5045 c1cc(ccc1NC(=O)C2CC2)Oc3ccsc3C(=O)O 4Y-5046 c1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5047 c1ccc(cc1)COCC(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5048 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5049 CS(=O)(=O)Nc1ccc(cc1)Oc2ccsc2C(=O)O 4Y-5050 COc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5053 c1ccc(cc1)CS(=O)(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5054 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Cl)Oc3ccsc3C(=O)O 4Y-5055 c1cc(cc(c1)S(=O)(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O)F 4Y-5056 c1cc(sc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccsc3C(=O)O 4Y-5057 COC(=O)c1cccc(c1COc2ccc(cc2)C=O)[N+](=O)[O-] 4Y-5060 CCOC(=O)C(=CNc1ccc2c(c1)c(=O)n(c(=O)o2)CCc3ccc(c(c3)OC)OC)C(=O)OCC 4Y-5062 CC(Cc1ccc2c(c1)OCC2)N.Cl 4Z-0005 CSc1nccc(n1)c2c(=O)ccn(n2)c3ccc(cc3)Cl 4Z-0201 c1cc(nc(c1)F)N2CCc3c(sc4c3c(ncn4)Nc5ccc(cc5)F)C2 4Z-0211 CN(C)/C=N/c1c(c2c(s1)CN(CC2)Cc3ccccc3)C#N 4Z-0227 C1[C@H]2[C@@H]1C3C(=O)NC(=O)N3C2 4Z-0246 c1cc(c(cc1N2CCCC2)N)[N+](=O)[O-] 4Z-0700 c1cc(c(cc1N2CCCCC2)N)[N+](=O)[O-] 4Z-0701 c1cc(c(cc1c2ccsc2)F)C#N 4Z-0702 c1cc(c(cc1c2ccsc2)C#N)F 4Z-0703 c1cc(oc1C=O)c2ccsc2 4Z-0704 c1ccc(cc1)n2cc(nn2)CN 4Z-0706 COC(=O)c1ccc(cc1)c2c(cccn2)[N+](=O)[O-] 4Z-0708 c1cc(ccc1C(=O)CN)F.Cl 4Z-0709 c1cc(ccc1c2nc(cs2)CC(=O)O)C(F)(F)F 4Z-0711 CCOC(=O)c1csc(n1)c2ccc(cc2)C(F)(F)F 4Z-0712 c1cc(ccc1c2nc(cs2)C(=O)O)C(F)(F)F 4Z-0713 CCOC(=O)c1ccc(s1)c2ccc(cc2)F 4Z-0714 c1cc(sc1c2ccsc2)C(=O)O 4Z-0715 CCOC(=O)c1ccc(s1)c2cccc(c2)[N+](=O)[O-] 4Z-0716 CCOC(=O)c1ccc(s1)c2ccccc2 4Z-0717 c1cc(cc(c1)[N+](=O)[O-])c2ccc(s2)C(=O)O 4Z-0718 c1ccc(cc1)c2ccc(s2)C(=O)O 4Z-0719 c1cc(ccc1C(CN)O)F 4Z-0721 c1cc(ccc1n2cc(nn2)CN)Cl 4Z-0722 Cc1ccc(cc1Oc2ccccc2C=O)C(C)C 4Z-0801 CCCCc1nnc(s1)N 4Z-0810 CC(C)(C)c1ccc2c(c1)NC(=O)CO2 4Z-0811 c1cc(sc1)/C(=N/O)/N 4Z-0812 CCCc1nnc(s1)N 4Z-0813 CCOC(=O)c1c(nn(c1C)c2c(cccc2Cl)Cl)C 4Z-0814 c1cnc(cn1)/C(=N/O)/N 4Z-0815 COC(=O)c1nc(no1)c2ccccc2 4Z-0816 CCOC(=O)c1csc2n1cc(n2)c3ccc(cc3)Br 4Z-0817 CCCc1[nH]c2cc(c(cc2n1)Cl)Cl 4Z-0820 CN(C)/C=C(\C#N)/C(=O)c1ccccc1Br 4Z-0827 c1cc(c(cc1Br)C(CC(=O)O)N)F 4Z-0828 Cc1ccc(cc1F)C(CC(=O)O)N 4Z-0829 Cc1cc(cc(c1N)N)Br 4Z-0830 c1cc(c(cc1Br)F)C(CC(=O)O)N 4Z-0832 c1c[nH]c2c1c(ccn2)Cl 4Z-5015 COc1cc(cc(c1O)/C=N\c2ccccc2)Br 5B-001 COc1cc(cc(c1O)/C=N\c2ccccc2Cl)Br 5B-002 COc1cc(cc(c1O)/C=N\c2cccc(c2)Cl)Br 5B-003 Cc1ccc(cc1)/N=C\c2cc(cc(c2O)OC)Br 5B-004 COc1ccc(cc1)/N=C\c2cc(cc(c2O)OC)Br 5B-005 COc1cc(cc(c1O)/C=N\c2cccc(c2)C(F)(F)F)Br 5B-006 c1cc(ccc1C(=O)O/N=C(\C#N)/C(=O)N)Cl 5B-007 c1ccc2c(c1)NCCS2 5B-009 c1ccc(c(c1)NC(=O)N2CCSc3c2cccc3)Cl 5B-011 c1ccc2c(c1)N(CCS2)C(=O)Nc3cccc(c3)Cl 5B-012 c1ccc2c(c1)N(CCS2)C(=O)Nc3ccc(cc3)Cl 5B-013 Cc1ccc(cc1)NC(=O)N2CCSc3c2cccc3 5B-014 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N\c2ccccc2 5B-015 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N\c2ccc(cc2)C 5B-016 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N\c2cccc(c2)C(F)(F)F 5B-018 Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2)S(=O)(=O)N 5B-019 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N\c2cccc(c2)Cl 5B-020 CCOC(=O)COc1c(cc(cc1OC)Br)/C=N\c2ccc(cc2)OC 5B-021 c1ccc(cc1)S(=O)(=O)O/N=C(/C#N)\C(=O)N 5B-022 c1ccc2c(c1)N(CCS2)C(=O)Nc3cccc(c3)C(F)(F)F 5B-023 c1ccc(cc1)NC(=O)N2CCSc3c2cccc3 5B-024 Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2)S(=O)(=O)/N=C/N(C)C 5B-026 c1cc(ccc1CSc2nc3cc(ccc3o2)Cl)Cl 5B-028 CC(C)(C)c1ccc(c(n1)O)C(=O)/C=C/N(C)C 5B-029 c1cc(cnc1)CSc2nc3cc(ccc3o2)Cl 5B-030 CC1(OC(=O)C(=Cc2ccccc2)C(=O)O1)C 5B-032 c1cc(ccc1C(=O)Sc2nc3cc(ccc3o2)Cl)Cl 5B-034 c1cc(cc(c1)Cl)C(=O)Sc2nc3cc(ccc3o2)Cl 5B-035 c1ccc(c(c1)C(=O)Sc2nc3cc(ccc3o2)Cl)Cl 5B-036 CC1(CC2=C(C(CC(=O)O2)c3ccccc3)C(=O)C1)C 5B-054 CN(C)c1nnc(o1)CC#N 5B-056 CC1(CC2=C(C(CC(=O)O2)c3ccc(cc3)Cl)C(=O)C1)C 5B-057 CC1(OC(=O)C(=Cc2ccc(cc2)OC)C(=O)O1)C 5B-058 CC1(CC2=C(C(CC(=O)O2)c3ccc(cc3)OC)C(=O)C1)C 5B-061 CC1(OC(=O)C(=Cc2cccs2)C(=O)O1)C 5B-062 CC1(OC(=O)C(=C/C=C/c2ccccc2)C(=O)O1)C 5B-063 Cn1c(c(c(n1)Cl)Cl)N(C)/N=C/c2ccccc2 5B-066 c1cc(ccc1C2CC(=O)CC(=O)C2)Cl 5B-067 Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2)S(=O)(=O)NC3CCCCC3 5B-070 c1cc(ccc1C2CC3=C(C(CC(=O)O3)c4ccc(cc4)Cl)C(=O)C2)Cl 5B-072 Cn1c(c(c(n1)Cl)Cl)N(C)NC(=O)Nc2ccc(cc2)Cl 5B-076 Cn1c(c(c(n1)Cl)Cl)N(C)NC(=O)Nc2cccc(c2)C(F)(F)F 5B-077 Cc1ccc(cc1)NC(=O)NN(C)c2c(c(nn2C)Cl)Cl 5B-078 CCCCCCCCCCCCCNS(=O)(=O)c1ccc(cc1)Oc2c(c(nn2C)Cl)Cl 5B-079 c1ccc(cc1)/C=C/CSc2cccc[n+]2[O-] 5B-082 c1ccc(cc1)C(=O)NNC2=NCCCCC2 5B-083 c1cc(ccc1C(=O)NNC2=NCCCCC2)Cl 5B-084 c1ccc(cc1)c2nnc3n2CCCCC3 5B-085 c1cc(ccc1c2nnc3n2CCCCC3)Cl 5B-086 CN(C)C=C1C=NNC1=O 5B-088 c1cc(ccc1NC=C2C=NNC2=O)Cl 5B-089 CCOC(=O)c1cc2c(cc[nH]c2=O)nc1C 5B-090 COC(c1ccc(c(=O)n1Cc2ccc(cc2)Cl)C#N)OC 5B-093 c1ccc(cc1)Nn2cnc3ccsc3c2=O 5B-095 c1cc(cc(c1)Cl)c2nnc3n2CCCCC3 5B-096 COC(c1ccc(c(=O)n1Cc2ccccc2)C#N)OC 5B-097 c1ccc(cc1)c2nnc3n2CCCC3 5B-098 c1cc(c(cc1c2nnc3n2CCCCC3)Cl)Cl 5B-101 CN(C)n1cnc2ccsc2c1=O 5B-104 CCOC(=O)Cn1nc(nn1)N(Cc2ccccc2Cl)Cc3ccccc3Cl 5B-105 c1cc(c(cc1c2nnc3n2CCCC3)Cl)Cl 5B-106 c1cc(nc(c1)Cl)Nn2cnc3ccsc3c2=O 5B-107 CS(=O)(=O)c1ccccc1O 5B-108 C(C(=C(C#N)C#N)N)Cl 5C-001 c1cnccc1C(=C(C#N)C#N)N 5C-002 c1cc(cnc1)C(=C(C#N)C#N)N 5C-005 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)N 5C-009 Cn1c(c(cn1)C#N)N 5C-010 c1ccc(cc1)n2c(nc3ccccc3c2=O)/C=C/c4ccc(cc4Cl)Cl 5C-012 Cc1c(c(n(n1)c2ccccc2)C)Cc3ccc(cc3)O 5C-014 c1cc(ccc1SCC(=C(C#N)C#N)N)Cl 5C-015 Cc1c(c(n(n1)C)C)Cc2ccc(cc2)OC(=O)Nc3ccccc3 5C-020 Cc1c(c(n(n1)C)C)Cc2ccc(cc2)OC(=O)Nc3cccc(c3)C(F)(F)F 5C-032 Cc1c(c(n(n1)C)C)Cc2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl 5C-035 COc1ccc(cc1)/C=N/c2ccccc2 5C-039 COc1ccc(cc1)/C=C/c2nc3ccccc3c(=O)n2c4ccccc4 5C-043 CCOC\1=NN(C(=O)/C1=C\N(C)C)c2ccccc2 5C-044 Cc1c(c(n(n1)C)C)Cc2ccc(cc2)OC(=O)c3ccccc3 5C-045 COc1cccc(c1)/C=C/c2nc3ccccc3c(=O)n2c4ccccc4 5C-047 Cc1ccc(cc1)/C=C/c2nc3ccccc3c(=O)n2c4ccccc4 5C-052 Cn1/c(=C\[N+](=O)[O-])/s/c(=C/c2ccccc2O)/c1=O 5C-053 c1ccc(cc1)n2c(nc3ccccc3c2=O)/C=C/c4ccc(cc4)C#N 5C-057 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)Cl)c3ccccc3 5C-060 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)C(=O)OC)c3ccccc3 5C-061 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2F)F)c3ccccc3 5C-062 CCOC\1=NN(C(=O)/C1=C\Nc2cc(cc(c2)Cl)Cl)c3ccccc3 5C-063 CCOC\1=NN(C(=O)/C1=C\Nc2ccccc2)c3ccccc3 5C-064 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)C)c3ccccc3 5C-065 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)OC)c3ccccc3 5C-066 CCOC\1=NN(C(=O)/C1=C\N(C)C)c2ccc(cc2)Cl 5C-067 CCOC\1=NN(C(=O)/C1=C\NCc2cccnc2)c3ccccc3 5C-069 CN(C)/C=C/C(=O)c1ccccn1 5C-070 CCOC\1=NN(C(=O)/C1=C\NCc2ccc(cc2Cl)Cl)c3ccccc3 5C-071 CCOC\1=NN(C(=O)/C1=C\NCc2cccs2)c3ccccc3 5C-072 CCOC\1=NN(C(=O)/C1=C\NCc2ccncc2)c3ccccc3 5C-074 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(c(c2)C)C)c3ccc(cc3)Cl 5C-075 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)Cl)c3ccc(cc3)Cl 5C-076 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)C)c3ccc(cc3)Cl 5C-079 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)OC)c3ccc(cc3)Cl 5C-080 CCOC\1=NN(C(=O)/C1=C\NN2CCOCC2)c3ccc(cc3)Cl 5C-081 Cc1ccc2c(c1)c(=O)c(co2)C=O 5C-082 CCOC\1=NN(C(=O)/C1=C\NCC(=O)OC)c2ccccc2 5C-083 Cc1ccc(cc1)N/C=C/c2c(c(ns2)SC)C#N 5C-084 CSc1c(c(sn1)/C=C/Nc2ccc(cc2)C(=O)O)C#N 5C-085 CSc1c(c(sn1)/C=C/Nc2ccc(cc2)Cl)C#N 5C-086 CSc1c(c(sn1)/C=C/Nc2ccc(cc2)F)C#N 5C-087 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2OC)OC)c3ccc(cc3)Cl 5C-088 CCOC\1=NN(C(=O)/C1=C\NN2CCCCC2)c3ccc(cc3)Cl 5C-089 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2F)F)c3ccc(cc3)Cl 5C-090 CCOC\1=NN(C(=O)/C1=C\Nc2cccc(c2)C(F)(F)F)c3ccc(cc3)Cl 5C-091 CCOC\1=NN(C(=O)/C1=C\NCc2cccnc2)c3ccc(cc3)Cl 5C-092 Cc1ccc2c(c1)c(=O)c(co2)/C=N/O 5C-093 CCOC\1=NN(C(=O)/C1=C\NCC(=O)OC)c2ccc(cc2)Cl 5C-094 CCOC\1=NN(C(=O)/C1=C\NCc2cccs2)c3ccc(cc3)Cl 5C-095 CCOC\1=NN(C(=O)/C1=C\NCc2ccc(cc2)Cl)c3ccc(cc3)Cl 5C-096 CCOC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)O)c3ccc(cc3)Cl 5C-097 CSc1c(c(sn1)/C=C/Nc2cccc(c2)Cl)C#N 5C-099 CSc1c(c(sn1)/C=C/Nc2cccc(c2)C(F)(F)F)C#N 5C-100 Cc1ccc2c(c1)c(=O)c(c(o2)N)C=O 5C-101 Cc1ccc(cc1C)N/C=C/c2c(c(ns2)SC)C#N 5C-103 CSc1c(c(sn1)/C=C/Nc2cc(cc(c2)Cl)Cl)C#N 5C-104 CSc1c(c(sn1)/C=C/Nc2ccccc2c3ccccc3)C#N 5C-105 CCc1c(cc2c(=O)c3cc(ccc3oc2n1)C)C(=O)OC 5C-106 Cc1cc(ccc1N/C=C/c2c(c(ns2)SC)C#N)O 5C-107 CN(C)c1nnnn1c2c(cc(cn2)C(F)(F)F)Cl 5C-110 Cc1c(c(n(n1)C)C)Cc2ccc(cc2)OC(=O)Nc3ccc(cc3)OC(F)(F)F 5C-111 CCOC(=O)c1cc2c(=O)c3cc(ccc3oc2nc1C)C 5C-112 Cc1ccc2c(c1)c(=O)c3cc(c(nc3o2)COC)C(=O)OC 5C-113 Cc1ccc2c(c1)c(=O)c3cc(c(nc3o2)C)C(=O)O 5C-114 Cc1ccc2c(c1)c(=O)c3cc(c(nc3o2)C)C(=O)OC 5C-115 Cc1ccc2c(c1)c(=O)c3cc(c(nc3o2)C)C(=O)Nc4ccc(cc4)Cl 5C-116 Cc1ccc2c(c1)c(=O)c3cc(c(nc3o2)C)C(=O)Nc4cccc(c4)C(F)(F)F 5C-117 Cc1ccc2c(c1)c(=O)c3cc(c(nc3o2)C)C(=O)NCc4ccccc4 5C-118 Cc1ccc2c(c1)c(=O)c3cc(c(nc3o2)C)C(=O)NCc4ccc(cc4)Cl 5C-119 Cc1ccc2c(c1)c(=O)c3cc(cnc3o2)C(=O)NC(C)(C)C 5C-120 CSc1c(c(sn1)/C=C/Nc2ccc(cc2F)F)C#N 5C-121 c1ccc(cc1)n2c(nc3ccccc3c2=O)/C=C/c4cccc(c4)C(F)(F)F 5C-123 c1ccc(cc1)/C=C\c2ccnc3n2nc(n3)SCc4c(cccc4Cl)F 5D-001 COc1ccc(cc1)c2ccnc3n2nc(n3)SCc4c(cccc4Cl)F 5D-002 c1ccnc(c1)c2ccnc3n2nc(n3)SCc4c(cccc4Cl)F 5D-006 C(C#N)Sc1nc([nH]n1)N 5D-007 CC(c1ccnc2n1nc(n2)SCc3c(cccc3Cl)F)Oc4ccc(cc4Cl)Cl 5D-008 c1ccc(cc1)N2CCN(CC2)/C=C\3/c4ccccc4C(=O)O3 5D-010 c1cc(ccc1COc2ccsc2C(=O)NN)F 5D-011 COc1cc(c(s1)C(=O)OC)O 5D-012 CCOC(=O)c1cc(nnc1Cl)c2ccccc2 5D-013 c1ccc(cc1)/C=C/CSc2nc3nccc(n3n2)c4ccccc4 5D-014 c1ccc(cc1)N2CCN(CC2)Cc3c4ccccc4c(=O)[nH]n3 5D-015 c1ccc2c(c1)/C(=C/Nc3[nH]ncn3)/OC2=O 5D-016 c1ccc2c(c1)/C(=C/Nc3ccc(cc3F)F)/OC2=O 5D-017 c1ccc2c(c1)/C(=C/NN/C(=N/c3ccc(cc3)Cl)/C[N+](=O)[O-])/OC2=O 5D-018 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3F)F 5D-019 CC(=O)[O-].c1ccc2c(c1)/C(=C/NNc3c(cc(c[nH+]3)C(F)(F)F)Cl)/OC2=O 5D-020 c1ccc(cc1)/C=C/CSc2nc3nccc(n3n2)/C=C\c4ccccc4 5D-021 c1ccc(cc1)/C=C/CSc2nc3nccc(n3n2)c4ccc(cc4)F 5D-022 c1ccc2c(c1)/C(=C/NNC(=O)CC#N)/OC2=O 5D-023 CN(C)c1c(cc(nn1)c2ccccc2)C#N 5D-025 c1ccc(cc1)n2c(=O)c3c(ccs3)[nH]c2=S 5D-026 c1ccc(cc1)CNc2c(cc(nn2)c3ccccc3)C#N 5D-027 c1ccc(cc1)c2cc(c(nn2)Oc3ccc(cc3)Cl)C#N 5D-028 COc1ccc(cc1)Oc2c(cc(nn2)c3ccccc3)C#N 5D-029 COc1ccc(cc1)c2cnc3nc(nn3c2N)SC/C=C/c4ccccc4 5D-030 c1ccc(cc1)/C=C/CSc2nc3ncc(c(n3n2)N)c4ccc(cc4)Cl 5D-031 COc1ccc(cc1)c2ccnc3n2nc(n3)SC/C=C/c4ccccc4 5D-032 c1ccc(cc1)Oc2ccc(cc2)N/C=C\3/c4ccccc4C(=O)O3 5D-034 c1ccc(cc1)Oc2ccc(cc2)NCc3c4ccccc4c(=O)[nH]n3 5D-035 Cc1ccc(cc1)N/N=C(/C(=O)CC(=O)OC)\C(=O)OC 5D-036 COC(=O)CC(=O)/C(=N/Nc1cccc(c1)C(F)(F)F)/C(=O)OC 5D-039 c1cc(c(cc1Cl)N2CSCC2=O)Cl 5D-042 COc1ccc(cc1)N2CSCC2=O 5D-043 c1cc(ccc1N2CS(=O)CC2=O)Cl 5D-044 c1cc(c(cc1Cl)N2CS(=O)(=O)CC2=O)Cl 5D-045 Cc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)O)O 5D-046 c1cc(c(cc1Cl)Cl)n2c(=O)cc(c(n2)C(=O)O)O 5D-047 c1cc(cc(c1)n2c(=O)cc(c(n2)C(=O)O)O)C(F)(F)F 5D-048 c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)O)O 5D-049 Cc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)OC)O 5D-052 COC(=O)c1c(cc(=O)n(n1)c2ccccc2)O 5D-056 COC(=O)c1c(cc(=O)n(n1)c2cccc(c2)C(F)(F)F)O 5D-057 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2Cl)Cl)O 5D-058 COc1ccc(cc1)N2CS(=O)CC2=O 5D-059 COc1ccc(cc1)N2CS(=O)(=O)CC2=O 5D-060 CC(C)(C)S(=O)(=O)/C(=C/N(C)C)/C#N 5D-065 c1ccc(cc1)c2cc(c(nn2)Oc3ccccc3)C#N 5D-069 c1ccc(cc1)c2cc(c(nn2)Oc3ccc(cc3)F)C#N 5D-070 c1cc(ccc1N/C=C/2\C(=O)N(CS2(=O)=O)c3ccc(cc3)Cl)Cl 5D-072 Cc1ccc(c(c1)C(=O)C)O 5D-073 c1ccc(cc1)c2cc(c(nn2)Oc3ccccc3Cl)C#N 5D-074 c1ccc(cc1)c2cc(c(nn2)Oc3cccc(c3)C(F)(F)F)C#N 5D-076 Cc1ccc(cc1)Oc2c(cc(nn2)c3ccccc3)C#N 5D-077 c1ccc(cc1)c2cc(c(nn2)NCc3ccc(cc3)Cl)C#N 5D-078 CN(C)/C=C/1\C(=O)N(CS1(=O)=O)c2ccc(cc2)OC 5D-079 CN(C)/C=C/1\C(=O)N(CS1=O)c2ccc(cc2)Cl 5D-080 CCSC(NC(=O)Nc1ccc(cc1)OC(F)(F)F)SCC 5D-086 CCSC(NC(=O)Nc1cccc(c1)C(F)(F)F)SCC 5D-088 CCSC(NC(=O)Nc1ccc(cc1Cl)Cl)SCC 5D-089 CCSC(NC(=O)Nc1ccc(cc1)C)SCC 5D-090 CCSC(NC(=O)Nc1ccc(cc1)OC)SCC 5D-091 Cn1cccc1C(=O)C(Cl)(Cl)Cl 5D-093 c1cc(c(c(c1)Cl)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)Cl 5D-095 COc1ccc(cc1)N/C=C/2\C(=O)N(C[S+]2[O-])c3ccc(cc3)Cl 5D-096 c1cc(ccc1N/C=C/2\C(=O)N(C[S+]2[O-])c3ccc(cc3)Cl)Cl 5D-097 c1cc(cc(c1)N/C=C/2\C(=O)N(C[S+]2[O-])c3ccc(cc3)Cl)C(F)(F)F 5D-098 c1cc(ccc1N2CSCC2=O)F 5D-099 COc1ccc(cc1)C(C#N)c2ccc(nn2)Cl 5D-109 c1cc(ccc1N2CS(=O)CC2=O)F 5D-110 CN(C)/C=C/1\C(=O)N(C[S+]1[O-])c2ccc(cc2)OC 5D-111 COc1ccc(cc1)N/C=C/2\C(=O)N(CS2(=O)=O)c3ccc(cc3)Cl 5D-112 COc1ccc(cc1)C(C#N)c2ccc(nn2)O 5D-114 c1cc(ccc1C(F)(F)F)N2CSCC2=O 5D-116 CCOC(=O)c1cc(nnc1Sc2ccccc2)c3ccccc3 5D-117 CCOC(=O)c1cc(nnc1Sc2ccc(cc2)Cl)c3ccccc3 5D-118 CN(C)/C=C/1\C(=O)N(CS1=O)c2ccc(cc2)F 5D-119 CCOC(=O)c1cc(nnc1Oc2ccccc2)c3ccccc3 5D-120 Cn1c(c(cn1)C#N)N/C=C\2/c3ccccc3C(=O)O2 5D-123 COc1ccc(cc1)Cc2ccc(nn2)O 5D-124 Cn1c(c(cn1)C#N)NCc2c3ccccc3c(=O)[nH]n2 5D-125 c1ccc(cc1)C(C#N)c2ccc(nn2)Cl 5D-128 Cn1cc(cc1C(=O)C(Cl)(Cl)Cl)C(=O)c2cccc(c2Cl)Cl 5D-129 c1cc(c(c(c1)Cl)Cl)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 5D-130 COc1ccc(cc1)C(c2ccc(nn2)O)C(=O)O 5D-132 c1ccc(cc1)C(C#N)c2ccc(nn2)O 5D-133 Cn1cc(cc1C(=O)OC)C(=O)c2cccc(c2Cl)Cl 5D-135 COC(=O)c1cc(c[nH]1)C(=O)c2cccc(c2Cl)Cl 5D-136 c1cc(ccc1N/C=C/2\C(=O)N(C[S+]2[O-])c3ccc(cc3)F)F 5D-138 Cc1ccc(cc1)N2CSCC2=O 5D-139 CCOC(=O)c1cc(nnc1Sc2ccc(cc2)F)c3ccccc3 5D-140 COC(=O)c1cc(c[nH]1)C(=O)c2c(cccc2Cl)Cl 5D-141 CNC(=O)c1cc(c[nH]1)C(=O)c2c(cccc2Cl)Cl 5D-143 Cc1ccc(cc1)N2CS(=O)(=O)CC2=O 5D-144 Cc1ccc(cc1)N2CS(=O)CC2=O 5D-145 Cc1ccc(cc1)N2CS(=O)/C(=C/N(C)C)/C2=O 5D-146 Cc1ccc(cc1)N2CS(=O)(=O)/C(=C/N(C)C)/C2=O 5D-147 CC(=O)c1cc(n(c1)C)C(=O)C(Cl)(Cl)Cl 5D-148 c1ccc(cc1)Cc2ccc(nn2)O 5D-149 CC(=O)c1cc(n(c1)C)C(=O)N 5D-151 c1cc(ccc1N2CSCC2=O)Br 5D-153 c1csc2n1cc(n2)Cl 5D-154 c1cc(ccc1N2CS(=O)CC2=O)Br 5D-156 c1cc(ccc1N2CS(=O)(=O)CC2=O)Br 5D-159 Cc1ccc(cc1)N/C=C/2\C(=O)N(C[S+]2[O-])c3ccc(cc3)C 5D-160 Cc1ccc(cc1)N2C[S+](/C(=C/Nc3ccc(cc3)Cl)/C2=O)[O-] 5D-161 Cc1ccc(cc1)N/C=C/2\C(=O)N(CS2(=O)=O)c3ccc(cc3)C 5D-162 CC(=O)c1cc(n(c1)C)C(=O)OC 5D-163 CN(C)/C=C/1\C(=O)N(C[S+]1[O-])c2ccc(cc2)Br 5D-165 c1cc(ccc1C(F)(F)F)N2CS(=O)(=O)CC2=O 5D-167 CN(C)/C=C/1\C(=O)N(CS1(=O)=O)c2ccc(cc2)Br 5D-168 CNC(=O)c1cc(cn1C)C(=O)c2cccc(c2Cl)Cl 5D-171 Cn1cc(cc1C(=O)N)C(=O)c2cccc(c2Cl)Cl 5D-172 c1ccc(cc1)Cc2ccc(nn2)Cl 5D-173 Cn1cc(cc1C#N)C(=O)c2cccc(c2Cl)Cl 5D-174 c1cc(c(c(c1)Cl)Cl)C(=O)c2cc([nH]c2)C(=O)N 5D-175 CN(C)/C=C(\C#N)/C(=O)NC(=O)c1ccccc1 5E-004 c1cc(c(cc1CO/N=C(/c2ccncc2)\N)Cl)Cl 5E-005 c1cc(ccc1CO/N=C(/c2ccncc2)\N)[N+](=O)[O-] 5E-007 c1cc(cnc1)/C(=N/OCc2ccc(cc2Cl)Cl)/N 5E-009 c1cc(c(c(c1)Cl)CO/N=C(/c2cccnc2)\N)Cl 5E-010 CC(=O)NC(=O)/C(=C/N(C)C)/C#N 5E-011 c1cc(cnc1)/C(=N/OCc2ccc(cc2)[N+](=O)[O-])/N 5E-012 c1ccnc(c1)/C(=N/OCc2ccc(cc2Cl)Cl)/N 5E-013 c1ccnc(c1)/C(=N/OCc2c(cccc2Cl)Cl)/N 5E-014 c1cc(cnc1)/C(=N/OCc2ccc(c(c2)Cl)Cl)/N 5E-015 COC(=O)c1cc(c[nH]1)C(=O)c2ccccc2 5E-016 c1cc(c(cc1Cl)Cl)C(=O)NC(=O)CC(=O)NC(=O)c2ccc(cc2Cl)Cl 5E-018 c1ccnc(c1)/C(=N/OCc2ccc(cc2)[N+](=O)[O-])/N 5E-020 c1ccc(cc1)c2ccn(n2)c3cccc(n3)F 5E-021 CC(C)(C#N)N1CCN(CC1)C(c2ccccc2)c3ccccc3 5E-022 CN(C)/C=C(\C1c2ccccc2C(=O)O1)/[N+](=O)[O-] 5E-023 c1c(cnc(n1)N2CCOCC2)C#N 5E-024 c1ccc(cc1)NC(=O)NNc2cccc(n2)F 5E-026 c1ccc(cc1)C(=O)NNc2cccc(n2)F 5E-027 c1ccc(cc1)S(=O)(=O)NNc2cccc(n2)F 5E-028 c1c(cnc(n1)NN)C#N 5E-029 c1ccc(cc1)Sc2ncc(cn2)C#N 5E-030 CC(C)(C#N)N1CCN(CC1)c2ccc(c(c2)Cl)Cl 5E-031 CC(C)(C#N)N1CCN(CC1)Cc2ccc3c(c2)OCO3 5E-032 c1cc(nc(c1)F)NNC(=O)N 5E-033 c1ccc(cc1)Nc2ncc(cn2)C#N 5E-035 c1ccc(cc1)c2cn(nc2N)c3cccc(n3)F 5E-036 c1cc(nc(c1)F)n2cc(c(n2)N)c3ccc(cc3)Cl 5E-037 c1cc(nc(c1)F)n2cnc(n2)O 5E-038 CO/C(=C(\C#N)/N=C/c1ccccc1Cl)/N 5E-039 CC(C)(C(=O)N)N1CCN(CC1)c2ccc(c(c2)Cl)Cl 5E-040 c1cc(c(cc1Cl)Cl)CON.Cl 5E-041 c1cc(c(cc1CON)Cl)Cl.Cl 5E-042 c1cc(c(c(c1)Cl)CO[NH3+])Cl.[Cl-] 5E-043 c1cc(ccc1CON)Cl.Cl 5E-044 c1cc(cc(c1)Cl)N2CCN(CC2)c3ncc(cn3)C#N 5E-046 c1ccc(cc1)N/C=C(\C2c3ccccc3C(=O)O2)/[N+](=O)[O-] 5E-047 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3ccc(cc3)Cl)/[N+](=O)[O-] 5E-048 c1ccc(cc1)/C=C/C=C\2/c3ccccc3C(=O)O2 5E-050 c1c(ccc(c1)Cl)/C=C(\C(=O)O)/C(=C/c2ccc(cc2)Cl)/C(=O)O 5E-051 CC(C)(C#N)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 5E-080 CC(C)(C(=O)N)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 5E-081 CC(C)(C#N)N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 5E-082 CC(C)(C(=O)N)N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 5E-083 CC(C)(C#N)N1CCN(CC1)c2ccc(cc2)OC 5E-084 CC(C)(C(=O)N)N1CCN(CC1)c2ccc(cc2)OC 5E-085 CC(C)(C#N)N1CCN(CC1)c2cccc(c2)C(F)(F)F 5E-086 CC(C)(C(=O)N)N1CCN(CC1)c2cccc(c2)C(F)(F)F 5E-087 CC(C)(C#N)N1CCN(CC1)c2ccc(cc2)F 5E-088 CC(C)(C(=O)N)N1CCN(CC1)c2ccc(cc2)F 5E-089 COC(=O)c1ccc[nH]c1=O 5E-302S COC(=O)c1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 5E-303S CCOC(=O)C(C)Sc1cc(nc(n1)c2ccccn2)C(F)(F)F 5E-304S CN(C)S(=O)(=O)NCCN1CCOCC1 5E-305S c1ccnc(c1)c2nc(cc(n2)Oc3ccc(cc3)C#N)C(F)(F)F 5E-306S COC(=O)c1ccccc1Oc2cc(nc(n2)c3ccccn3)C(F)(F)F 5E-307S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)O 5E-308S COC(=O)c1cccn(c1=O)Cc2c(cccc2Cl)Cl 5E-309S Cc1c(snn1)Cl 5E-310S c1ccc(c(c1)Oc2cc(nc(n2)c3ccccn3)C(F)(F)F)Cl 5E-311S c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)O)Cl 5E-312S CNC(=O)c1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 5E-314S c1ccnc(c1)c2nc(cc(n2)NCc3ccc(cc3)Cl)C(F)(F)F 5E-315S c1ccnc(c1)c2nc(cc(n2)NCc3cccs3)C(F)(F)F 5E-316S c1ccc(cc1)Nc2cc(nc(n2)c3ccccn3)C(F)(F)F 5E-317S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 5E-318S c1ccc(cc1)CNC(=O)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 5E-319S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)Nc3ccc(cc3)Cl 5E-320S CN(C)C(=O)c1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 5E-321S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)NCc3ccc(cc3)Cl 5E-322S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 5E-323S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)N3CCOCC3 5E-324S c1ccc(c(c1)CNc2cc(nc(n2)c3ccccn3)C(F)(F)F)C(F)(F)F 5E-326S c1ccc(c(c1)CNc2cc(nc(n2)c3ccccn3)C(F)(F)F)Cl 5E-327S Cn1c(cc(n1)C(F)(F)F)O 5E-328S Cn1c(c(c(n1)C(F)(F)F)C=O)Cl 5E-329S CNC(=O)c1cccn(c1=O)Cc2c(cccc2Cl)Cl 5E-330S CN(C)C(=O)c1cccn(c1=O)Cc2c(cccc2Cl)Cl 5E-331S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3c(cccc3Cl)Cl 5E-332S c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3)Cl)Cl 5E-333S c1cc(cc(c1)NC(=O)c2cccn(c2=O)Cc3c(cccc3Cl)Cl)C(F)(F)F 5E-334S c1ccc(cc1)CNC(=O)c2cccn(c2=O)Cc3c(cccc3Cl)Cl 5E-335S COC(=O)c1cccn(c1=O)Cc2cccc(c2)C(F)(F)F 5E-336S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2c(cccc2Cl)Cl)Cl 5E-337S COC(=O)c1cccn(c1=O)Cc2cccc(c2)Cl 5E-338S c1cc(cc(c1)C(F)(F)F)Cn2cccc(c2=O)C(=O)O 5E-339S c1cc(cc(c1)Cl)Cn2cccc(c2=O)C(=O)O 5E-340S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 5E-343S c1cc(cc(c1)C(F)(F)F)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3)Cl 5E-344S c1cc(cc(c1)C(F)(F)F)Cn2cccc(c2=O)C(=O)Nc3cccc(c3)C(F)(F)F 5E-345S c1cc(cc(c1)C(F)(F)F)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3F)F 5E-346S CNC(=O)c1cccn(c1=O)Cc2cccc(c2)C(F)(F)F 5E-347S CN(C)C(=O)c1cccn(c1=O)Cc2cccc(c2)C(F)(F)F 5E-348S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3cccc(c3)Cl 5E-349S c1cc(cc(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3)Cl 5E-350S c1cc(cc(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3cccc(c3)C(F)(F)F 5E-351S c1cc(cc(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3F)F 5E-352S CNC(=O)c1cccn(c1=O)Cc2cccc(c2)Cl 5E-353S CN(C)CCNC(=O)c1cccn(c1=O)Cc2cccc(c2)C(F)(F)F 5E-355S c1cc(cc(c1)Cl)Cn2cccc(c2=O)C(=O)N3CCOCC3 5E-357S CN1CCN(CC1)C(=O)c2cccn(c2=O)Cc3cccc(c3)Cl 5E-358S c1ccc(cc1)Cn2cccc(c2=O)C(=O)O 5E-360S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(cc2Cl)Cl)Cl 5E-361S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(c(c2)Cl)Cl)Cl 5E-362S Cn1c(c(c(n1)C(F)(F)F)/C=N/OCc2ccc(cc2)[N+](=O)[O-])Cl 5E-363S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC)Cl 5E-364S Cn1c(c(c(n1)C(F)(F)F)/C=N/O)Cl 5E-365S Cn1c(cc(n1)O)C(F)(F)F 5E-366S COC(=O)c1ccc(=O)[nH]c1 5E-367S CN(C)CCNC(=O)c1cccn(c1=O)Cc2c(cccc2Cl)Cl 5E-368S CN1CCN(CC1)C(=O)c2cccn(c2=O)Cc3c(cccc3Cl)Cl 5E-369S c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3F)F)Cl 5E-370S c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl 5E-371S c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3c(cccc3Cl)Cl)Cl 5E-372S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccccc2)Cl 5E-373S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2ccc(cc2)Cl)Cl 5E-374S Cn1c(c(c(n1)C(F)(F)F)/C=N/OC(=O)c2cccc(c2)C(F)(F)F)Cl 5E-375S CC1CN(CC(O1)C)C(=O)c2cccn(c2=O)Cc3c(cccc3Cl)Cl 5E-376S c1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccccc3 5E-378S c1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3)Cl 5E-379S c1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3F)F 5E-380S c1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3cccc(c3)C(F)(F)F 5E-381S c1ccc(cc1)Cn2cccc(c2=O)C(=O)Nc3ccc(cc3)OC(F)(F)F 5E-382S COC(=O)c1ccc(=O)n(c1)Cc2ccc(c(c2)Cl)Cl 5E-383S CN(c1ccccc1)C(=O)c2cccn(c2=O)Cc3ccccc3 5E-385S c1ccc(cc1)CNC(=O)c2cccn(c2=O)Cc3ccccc3 5E-386S c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)NCCN3CCOCC3)Cl.Cl 5E-387S COC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2)Cl 5E-388S c1cc(c(cc1Cn2cc(ccc2=O)C(=O)O)Cl)Cl 5E-389S c1cc(c(=O)n(c1)Cc2ccc3c(c2)OC(O3)(F)F)C(=O)O 5E-501 c1cc(ncc1C(F)(F)F)O 5E-502 c1ccc(c(c1)C(F)(F)F)NC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-504 c1cc(cc(c1)NC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F)C(F)(F)F 5E-505 c1cc(c(=O)n(c1)Cc2ccc3c(c2)OC(O3)(F)F)C(=O)Nc4ccc(cc4)C(F)(F)F 5E-506 c1cc(c(=O)n(c1)Cc2ccc3c(c2)OC(O3)(F)F)C(=O)Nc4ccc(cc4F)F 5E-508 Cc1cccc(c1NC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F)C 5E-509 CNC(=O)c1cccn(c1=O)Cc2ccc3c(c2)OC(O3)(F)F 5E-511 CN(C)C(=O)c1cccn(c1=O)Cc2ccc3c(c2)OC(O3)(F)F 5E-512 c1cc(c(=O)n(c1)Cc2ccc3c(c2)OC(O3)(F)F)C(=O)NCc4ccc(cc4)Cl 5E-514 COc1ccccc1CNC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-515 CC(C)Oc1cccc(c1)NC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-516 CC(C)N(c1ccc(cc1)Cl)C(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-517 CC(C)N(Cc1ccccc1Cl)C(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-518 CC(C)C(C)(C(=O)N)NC(=O)c1cccn(c1=O)Cc2ccc3c(c2)OC(O3)(F)F 5E-520 Cc1ccc(nc1)NC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-521 CC(C)(C(=O)OC)NC(=O)c1cccn(c1=O)Cc2ccc3c(c2)OC(O3)(F)F 5E-522 CC(c1ccccc1)NC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-524 c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 5E-525 c1cc(ccc1Cn2cc(cc(c2=O)[N+](=O)[O-])C(F)(F)F)Cl 5E-542 COc1cc(cn(c1=O)Cc2ccc(cc2)Cl)C(F)(F)F 5E-544 c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)C(=O)N=N#N 5E-551 c1cc(c(cc1Cn2cc(cc(c2=O)[N+](=O)[O-])C(F)(F)F)Cl)Cl 5E-552 c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)NC(=O)Nc3ccc(cc3F)F 5E-553 Cc1cccc(c1NC(=O)Nc2cccn(c2=O)Cc3ccc(cc3)Cl)C 5E-554 c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)NC(=O)Nc3cc(cc(c3)Cl)Cl 5E-555 Cc1ccc(nc1)NC(=O)Nc2cccn(c2=O)Cc3ccc(cc3)Cl 5E-556 c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)N=N#N 5E-557 CNC(=O)Nc1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 5E-558 CN(C)C(=O)Nc1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 5E-559 CN1CCN(CC1)C(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 5E-560 c1cc(cc(c1)NC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl)C(F)(F)F 5E-561 COC(=O)c1ccccc1NC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 5E-562 CC(C)Oc1cccc(c1)NC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 5E-563 c1ccc(cc1)SC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 5E-564 CCOC(=O)CSC(=O)Nc1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 5E-565 C#CCOC(=O)Nc1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 5E-566 c1ccc(cc1)n2ccc(n2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F 5E-717 COC(=O)C(/C=N/OCc1c(cccc1Cl)Cl)NC(=O)c2ccccc2 5E-903 COC(=O)C(/C=N/OCc1ccc(c(c1)Cl)Cl)NC(=O)c2ccccc2 5E-904 COC(=O)C(/C=N/OCc1ccc(cc1)[N+](=O)[O-])NC(=O)c2ccccc2 5E-905 c1ccc(cc1)SCCC(=O)O 5E-906 CC1(C2CC3CC(C2)CC1C3)CC(=O)Nc4cccc(c4)C(F)(F)F 5E-907 CC1(C2CC3CC(C2)CC1C3)CC(=O)Nc4ccc(cc4Cl)Cl 5E-908 COC(=O)C(/C=N/O)NC(=O)c1ccccc1 5E-909 c1ccc2c(c1)C(=O)C(CO2)(CO)CO 5E-911 c1ccc2c(c1)C(=O)C(CS2)(CO)CO 5E-912 c1ccc(cc1)C2OCC3(COc4ccccc4C3=O)CO2 5E-913 c1ccc2c(c1)C(=O)C3(CO2)COC(OC3)c4ccc(cc4)Cl 5E-914 c1ccc2c(c1)C(=O)C3(COC(OC3)c4ccc(cc4)Cl)CS2 5E-915 c1ccc2c(c1)C(=O)C(CS2)(COC(=O)c3cccc(c3)C(F)(F)F)COC(=O)c4cccc(c4)C(F)(F)F 5E-916 c1ccc(cc1)C(=O)OCC2(CSc3ccccc3C2=O)COC(=O)c4ccccc4 5E-917 c1ccc(cc1)C(=O)OCC2(COc3ccccc3C2=O)COC(=O)c4ccccc4 5E-918 c1ccc2c(c1)C(=O)C(CO2)(COC(=O)c3cccc(c3)C(F)(F)F)COC(=O)c4cccc(c4)C(F)(F)F 5E-919 c1ccc(cc1)C2OCC3(CO2)CSc4ccccc4C3=O 5E-920 COC(=O)C(/C=N/OC)NC(=O)c1ccccc1 5E-923 c1ccc2c(c1)C(=O)C3(CC3C#N)CO2 5E-924 c1cc(c(cc1Cl)Cl)C(=O)NCC(=O)O 5E-925 c1ccc2c(c1)C(=O)C3(CC3C#N)CS2 5E-926 Cc1ccc(cc1)N2C(=O)CC(=N2)C(F)(F)F 5E-929 Cc1ccc(cc1)N2C(=O)CC(=N2)C 5E-930 c1ccc(cc1)C2=NN(C(=O)C2)c3ccccc3 5E-933 COC(=O)C(/C=N/OCc1ccc(cc1)Cl)NC(=O)c2ccccc2 5E-934 CCOC(=O)c1c(=O)c2cc(ccc2oc1c3ccccc3)C 5E-936 COc1ccc2cc(c(=O)oc2c1)NC(=O)c3ccccc3 5E-937 CCOC(=O)c1cc(c(=O)oc1C(F)(F)F)NC(=O)c2ccc(cc2Cl)Cl 5E-940 Cn1c(=O)c2cc(c(=O)oc2n(c1=O)C)NC(=O)c3ccc(cc3Cl)Cl 5E-942 c1cc(cc2c1cc(c(=O)o2)NC(=O)c3ccc(cc3Cl)Cl)O 5E-943 COc1ccc(cc1)C(=O)Nc2cc3ccc(cc3oc2=O)O 5E-944 Cc1ccc2c(c1)c(=O)c(c(o2)c3ccccc3)C(=O)O 5E-950 COc1ccc2cc(c(=O)oc2c1)NC(=O)c3ccc(cc3Cl)Cl 5E-951 c1cc(cc(c1)n2c(=O)cc3c(n2)c(n[nH]3)O)C(F)(F)F 5F-002 c1ccnc(c1)SCc2ncn(n2)c3cccc(n3)F 5F-004 COC(=O)c1c(ccs1)Oc2c(cc(cn2)C(F)(F)F)Cl 5F-005 CCOC(=O)Cc1[nH]nc(n1)COc2ncn(n2)c3ccccc3 5F-006 Cc1ccc(cc1)/N=C(/C[N+](=O)[O-])\NN/C=C\2/c3ccccc3C(=O)O2 5F-009 COC(=O)c1ccccc1OC/C(=N/NC(=O)c2ccccc2)/N 5F-010 COC(=O)c1ccccc1OC/C(=N/Nc2cccc(n2)Cl)/N 5F-011 c1ccc(cc1)NC(=O)Nc2c(ccs2)OCc3ccc(cc3)F 5F-014 COC(=O)c1c(cc(=O)n(n1)c2ccccc2)Oc3ccc(cc3)Cl 5F-015 CN(C)/C=C(\C(=O)OC)/N=C/c1ccc(cc1)Cl 5F-017 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)Sc3ncccn3 5F-019 COC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)Sc3cccc[n+]3[O-] 5F-020 c1ccc(c(c1)C(=O)NN)OCc2ncn(n2)c3cccc(n3)Cl 5F-022 c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)Oc3ccc(cc3)Cl 5F-023 c1ccc2c(c1)-c3c(cccn3)C2O 5F-024 c1ccc(c(c1)C(=O)NNC(=N)COc2ccc(cc2Cl)Cl)OCc3ncn(n3)c4cccc(n4)Cl 5F-025 COC(=O)c1c(ccs1)Oc2cccc(n2)Cl 5F-027 COC(=O)c1c(ccs1)Oc2ccc(nn2)Cl 5F-029 CC(=O)c1ccc(o1)c2ccc(cc2Cl)Cl 5F-031 CCOC(=O)C[n+]1ccccc1.[Br-] 5F-032 Cc1c(nc(s1)c2ccc(cc2)Cl)O 5F-033 c1cc[n+](cc1)C2C(C(=C(NC2=O)[O-])C#N)c3ccc(cc3)Cl 5F-034 c1cc(ccc1Oc2ccc(c(c2)Cl)c3csc(n3)N)Cl 5F-035 Cc1nc(cs1)c2ccc(cc2Cl)Oc3ccc(cc3)Cl 5F-036 c1cc([nH]c1)C=C(C#N)C#N 5F-037 c1cc(ccc1/C=C\c2ccnc(n2)Cn3cncn3)Cl 5F-038 c1cc(c(cc1Cl)Cl)c2ccc(o2)C(=O)C(Br)Br 5F-039 Cc1c(nc(s1)c2c(cccc2F)F)O 5F-040 Cc1ccc(cc1)CONC(=O)N 5F-041 Cc1ccc(cc1)CONC(=O)/N=C/N(C)C 5F-042 c1ccc(cc1)C(=O)NC(=O)Nc2ccccc2 5F-043 c1cc(c(cc1Cl)Cl)c2ccc(o2)C=O 5F-045 Cc1ccc(cc1)CONC(=O)N/C=N/OC 5F-046 Cc1c(c(on1)/C=C/c2ccc(o2)c3ccc(cc3Cl)Cl)[N+](=O)[O-] 5F-047 CC(c1ccnc(n1)Cn2cncn2)Oc3ccc(cc3)Cl 5F-048 c1ccc(c(c1)C(=O)NNC(=N)COc2ccc(cc2)F)OCc3ncn(n3)c4cccc(n4)Cl 5F-049 c1ccc(c(c1)c2nnc(o2)COc3ccc(cc3)F)OCc4ncn(n4)c5cccc(n5)Cl 5F-050 c1ccc2c(c1)/C(=C/c3ccc(o3)c4ccc(cc4Cl)Cl)/OC2=O 5F-051 C1C(=O)CNC(=O)NC1=O 5F-053 c1cc(c(cc1Cl)Cl)c2ccc(o2)C(=O)CBr 5F-054 c1ccc2c(c1)c(n[nH]c2=O)Cc3ccc(o3)c4ccc(cc4Cl)Cl 5F-055 COC(c1ccccc1)P(=O)(OC)OC 5F-057 c1cc(c(cc1C(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl)Cl)Cl 5F-301S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl 5F-303S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)F)c4ccc(cc4)Cl 5F-304S Cc1ccc(cc1)C(=O)OCc2cn(nn2)c3ccc(c(c3)Cl)Cl 5F-308S c1ccc(cc1)n2cc(nn2)COC(=O)CCl 5F-309S c1ccc(cc1)NC(=O)OCc2cn(nn2)c3ccccc3 5F-311S c1cc(cc(c1)[N+](=O)[O-])NC(=O)c2cc(cc(c2)Cl)Cl 5F-313S c1cc2c(c(sc2nc1)C(=O)Nc3ccc(cc3)Cl)OCc4ccc(c(c4)Cl)Cl 5F-314S c1ccc(cc1)COCc2cn(nn2)c3ccccc3 5F-317S Cc1cc(cc(c1)C(=O)NCc2cccc(c2)C(F)(F)F)C 5F-319S Cc1cc(cc(c1)C(=O)NCc2ccc(cc2)C(F)(F)F)C 5F-320S c1cc(cc(c1)NC(=O)c2c(c3cccnc3s2)OCc4ccc(c(c4)Cl)Cl)C(F)(F)F 5F-321S c1cc2c(c(sc2nc1)C(=O)Nc3ccc(cc3)OC(F)(F)F)OCc4ccc(c(c4)Cl)Cl 5F-322S CN(c1ccc(cc1)C(F)(F)F)C(=O)c2cc(cc(c2)Cl)Cl 5F-323S CN(c1cccc(c1)[N+](=O)[O-])C(=O)c2cc(cc(c2)Cl)Cl 5F-324S COc1ccc(cc1)COc2c3cccnc3sc2C(=O)OC 5F-325S c1ccc(cc1)n2cc(nn2)C=O 5F-326S CCOC(=O)COc1c2cccnc2sc1C(=O)OC 5F-327S CCOC(=O)C(C)Oc1c2cccnc2sc1C(=O)OC 5F-328S c1ccc(cc1)NC(=O)c2c(c3cccnc3s2)OCc4ccc(c(c4)Cl)Cl 5F-329S c1cc(cc(c1)Cl)NC(=O)c2c(c3cccnc3s2)OCc4ccc(c(c4)Cl)Cl 5F-331S CCNC(=O)OCc1cn(nn1)c2ccccc2 5F-332S Cc1ccc(cc1)C(=O)OCc2cn(nn2)c3ccccc3 5F-333S Cc1cc(cc(c1)C(=O)Nc2cccc(c2)C(F)(F)F)C 5F-334S Cc1cc(cc(c1)C(=O)Nc2ccc(cc2)C(F)(F)F)C 5F-335S Cc1cc(cc(c1)C(=O)N(C)c2ccc(cc2)C(F)(F)F)C 5F-337S Cc1cc(cc(c1)C(=O)N(C)c2cccc(c2)C(F)(F)F)C 5F-338S c1ccc(cc1)n2cc(nn2)COC(=O)Nc3cccc(c3)Cl 5F-339S c1ccc(cc1)n2cc(nn2)COC(=O)Nc3ccc(cc3)Cl 5F-340S Cn1c(c(c(n1)C(F)(F)F)C#N)Sc2ccccc2 5F-341S Cn1c(c(c(n1)C(F)(F)F)C#N)SCc2ccc(cc2)Cl 5F-342S c1ccc(cc1)COc2c3cccnc3sc2C(=O)O 5F-344S c1ccc2c(c1)cnn(c2=O)c3c(cc(cc3Cl)Cl)Cl 5F-345S Cc1ccc(cc1)S(=O)(=O)NC(=O)OCc2cn(nn2)c3ccccc3 5F-347S CC(C)(C)C(=O)OCc1cn(nn1)c2ccccc2 5F-349S c1ccc(cc1)n2cc(nn2)COC(=O)C3CC3 5F-350S Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2ccc(cc2)Cl 5F-351S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)c2ccccc2C(=O)OC 5F-352S CC(C)CC(=O)OCc1cn(nn1)c2ccccc2 5F-353S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)c2ccccc2 5F-354S Cc1cc(cc(c1)C(=O)N(C)Cc2ccc(cc2)C(F)(F)F)C 5F-355S Cc1cc(cc(c1)C(=O)N(C)Cc2cccc(c2)C(F)(F)F)C 5F-356S c1c(c[nH]c(=O)c1C(=O)O)Br 5F-357S c1ccc(cc1)n2cc(nn2)COC(=O)c3cccc(c3)C(F)(F)F 5F-359S Cc1ccc(cc1)S(=O)(=O)c2c(c(nn2C)C(F)(F)F)C#N 5F-360S Cc1cc(cc(c1)C(=O)Nc2cccc(c2)[N+](=O)[O-])C 5F-363S COC(=O)c1cc(cn(c1=O)Cc2cccc(c2)C(F)(F)F)Br 5F-365S c1ccc2c(c1)cnn(c2=O)c3ccc(cc3)Cl 5F-366S Cc1ccccc1CS(=O)(=O)c2c(c(nn2C)C(F)(F)F)C#N 5F-367S c1ccc(cc1)n2cc(nn2)/C=N/OCc3ccc(cc3Cl)Cl 5F-368S CC(C)(C)c1ccc(cc1)COc2c(c(nn2C)C(F)(F)F)C#N 5F-369S Cc1cc(cc(c1)C(=O)N(C)c2ccc(cc2)[N+](=O)[O-])C 5F-370S Cc1cc(cc(c1)C(=O)N(C)c2cccc(c2)[N+](=O)[O-])C 5F-371S Cn1c(c(c(n1)C(F)(F)F)C#N)OCC#C 5F-374S Cn1c(c(c(n1)C(F)(F)F)C#N)OCc2ccc(cc2)OC 5F-376S Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2ccc(cc2)C(=O)OC 5F-377S Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2ccc(cc2Cl)Cl 5F-378S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Br)c4ccc(cc4)Cl 5F-379S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3)Cl 5F-380S c1cc(ccc1CS(=O)(=O)CC(CN2CCCC2=O)O)Cl 5F-381S c1cc(ccc1S(=O)(=O)CC(CN2CCCC2=O)O)Cl 5F-382S c1ccc(cc1)n2cc(nn2)/C=N/OCc3ccc(cc3)Cl 5F-383S Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2cccc(c2)[N+](=O)[O-] 5F-384S c1ccc(cc1)n2cc(nn2)/C=N/O 5F-385S c1cc(ccc1C[NH2+]CC(CN2CCCC2=O)O)Cl.[Cl-] 5F-386S c1ccc(c(c1)CS(=O)(=O)CC(CN2CCCC2=O)O)Cl 5F-387S c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)CC(CN2CCCC2=O)O 5F-388S c1ccc(cc1)CS(=O)(=O)CC(CN2CCCC2=O)O 5F-389S Cc1ccccc1CS(=O)(=O)CC(CN2CCCC2=O)O 5F-390S Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2cccc(c2)C(F)(F)F 5F-391S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)Cc2cccc(c2)C(F)(F)F 5F-392S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)C(=O)O)Br 5F-393S CC(C)(C)c1ccc(cc1)CS(=O)(=O)CC(CN2CCCC2=O)O 5F-394S c1ccc(cc1)S(=O)(=O)CC(CN2CCCC2=O)O 5F-395S Cc1ccc(cc1)S(=O)(=O)CC(CN2CCCC2=O)O 5F-396S CC(C)(C)c1ccc(cc1)CS(=O)(=O)c2c(c(nn2C)C(F)(F)F)C#N 5F-398S c1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3cccc(c3)C(F)(F)F)Br 5F-401S c1ccc(cc1)c2nc3ccccc3n2O 5F-403S c1ccc2c(c1)cnn(c2=O)c3ccc(cc3Cl)Cl 5F-404S c1ccc2c(c1)cnn(c2=O)c3ccc(cc3)F 5F-405S COc1ccc(cc1)S(=O)(=O)CC(CN2CCCC2=O)O 5F-406S c1cc(cc(c1)S(=O)(=O)CC(CN2CCCC2=O)O)C(F)(F)F 5F-407S c1ccc2c(c1)cnn(c2=O)c3ccc(cc3)Br 5F-408S c1ccnc(c1)c2nc(c(c(n2)O)Br)C(F)(F)F 5F-411S c1ccc(c(c1)CNCC(CN2CCCC2=O)O)Cl.Cl 5F-412S c1cc(cc(c1)Cl)C[NH2+]CC(CN2CCCC2=O)O.[Cl-] 5F-413S Cc1ccccc1C[NH2+]CC(CN2CCCC2=O)O.[Cl-] 5F-414S Cc1ccc(cc1)CNCC(CN2CCCC2=O)O.Cl 5F-416S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3)F 5F-417S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3Cl)Cl 5F-418S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3)Br 5F-419S c1ccc2c(c1)cnn(c2=O)c3ccc(cc3F)F 5F-420S c1ccc(c(c1)CNc2ccccc2[N+](=O)[O-])Cl 5F-422S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)OC(F)(F)F)c4ccc(cc4)Cl 5F-423S c1ccc2c(c1)cnn(c2=O)c3ccc(cc3)OC(F)(F)F 5F-424S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3)OC(F)(F)F 5F-425S c1ccc2c(c1)cnn(c2=O)c3ccc(cc3)C(F)(F)F 5F-432S CCOC(=O)/C=C(\[NH3+])/Nc1cccc(c1)C(F)(F)F.[Cl-] 5F-900 CCOC(=O)/C=C(\N)/Nc1ccc(cc1)OC.Cl 5F-901 Cc1cc(n(n1)c2c3c(c4ccccc4[nH]3)ncn2)C 5F-902 Cc1ccc(cc1)c2[nH]c(=O)c(c(n2)C)CC#C 5F-904 CC(=O)c1ccc(cc1)NC(=O)CC2(C3CC4CC(C3)CC2C4)c5ccccc5 5F-905 Cc1c(c(=O)[nH]c(=S)[nH]1)CC#C 5F-906 Cc1nnc2n1cnc3c2[nH]c4c3cccc4 5F-908 c1ccc2c(c1)c3c([nH]2)c(ncn3)n4cc(c(n4)N)c5ccc(cc5)Cl 5F-909 CN(C)/C=C/C(=O)c1ccc(cc1)NC(=O)CC2(C3CC4CC(C3)CC2C4)c5ccccc5 5F-911 c1coc2c1C(=O)CCC2 5F-912 C/C(=N/OCc1ccc(cc1Cl)Cl)/c2ccc(cc2)NC(=O)CC3(C4CC5CC(C4)CC3C5)c6ccccc6 5F-914 Cc1ccc(cc1)c2nc(c(c(n2)Cl)CC#C)C 5F-915 c1coc2c1-c3c(cnc(n3)N)CC2 5F-916 c1ccc2c(c1)CC3=C2C(=O)CCS3 5F-917 c1ccc2c(c1)CC3=C2/C(=N/OCc4ccc(cc4Cl)Cl)/CCS3 5F-919 c1ccc2c(c1)c3c([nH]2)c(ncn3)N/N=C/c4ccc(cc4Cl)Cl 5F-921 c1ccc(cc1)C(=O)CC2C(=O)CCCC2=O 5F-922 Cc1ccc(cc1)n2c(cc3c2CCCC3=O)c4ccccc4 5F-923 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)NCC(CO)O 5F-924 c1ccc(cc1)N2C(=O)CC(=N2)c3cccnc3 5F-926 c1ccc2c(c1)CC3=C2SCC(=C3Cl)/C=N/OCc4ccc(cc4Cl)Cl 5F-927 Cc1c(c(=O)[nH]c(n1)N)CC#C 5F-930 c1cc(cnc1)C2=NN(C(=O)C2)c3ccc(cc3Cl)Cl 5F-931 COc1cc(ccc1O)/C=N/Nc2c(=O)[nH]c3ccccc3n2 5F-933 c1ccc(c(c1)/C=N/Nc2c(=O)[nH]c3ccccc3n2)O 5F-934 Cc1ccc(cc1)c2nc(c(c(n2)N3CCN(CC3)c4ccc(cc4)OC)CC#C)C 5F-935 CC1=NN(C(=O)C1CC#C)c2c(cc(cc2Cl)Cl)Cl 5F-937 Cc1ccc(cc1)n2c(cc\3c2CCC/C3=N/OCc4ccc(cc4)Cl)c5ccccc5 5F-939 c1cc(sc1)C(=O)Nc2ncc3c(n2)-c4ccoc4CC3 5F-940 c1ccc(cc1)N2C(=O)/C(=C\Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)/C(=N2)c4cccnc4 5F-941 COc1ccc(cc1)N/C=C/2\c3ccccc3C4=C2C(=O)CCS4 5F-942 CN1C(CC(O1)COC(=O)c2ccc(cc2)OC)c3ccccc3 5F-943 c1cc(ccc1N2CCC(=O)CC2)[N+](=O)[O-] 5F-944 c1cc(ccc1CON=C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])Cl 5F-945 c1c(cc(c(c1[N+](=O)[O-])N2CCC(=O)CC2)[N+](=O)[O-])C(F)(F)F 5F-946 CN1C(CC(O1)COC(=O)c2ccc(cc2Cl)Cl)c3ccccc3 5F-947 CN1C(CC(O1)COC(=O)c2ccc(cc2)F)c3ccccc3 5F-948 CN1C(CC(O1)COC(=O)c2ccccc2)c3ccccc3 5F-949 CN1C(CC(O1)COC(=O)c2cccc(c2)C(F)(F)F)c3ccccc3 5F-950 CN(C)/C=C\1/CN(CCC1=O)c2ccc(cc2)[N+](=O)[O-] 5F-951 c1cc(ccc1N2CCC(CC2)O)[N+](=O)[O-] 5F-952 c1ccc2c(c1)/C(=N/OCc3ccc(cc3Cl)Cl)/CC24C5CC6CC(C5)CC4C6 5F-953 Cc1ccc(cc1)c2ncc3c(n2)CCN(C3)c4ccc(cc4)[N+](=O)[O-] 5F-954 c1cc(ccc1N2CCc3c(c[nH]n3)C2)[N+](=O)[O-] 5F-955 c1ccc(cc1)n2cc3c(n2)CN(CC3)c4ccc(cc4)[N+](=O)[O-] 5F-956 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3ccccc3)C(=O)c4ccccc4 5F-957 c1ccc(cc1)C(=O)c2cc(c([nH]2)N3CCN(CC3)c4ccccc4)C#N 5F-958 c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccccc3 5F-959 Cc1c2c(nc(n1)c3ccccc3O)Oc4ccccc4C2 5F-960 Cc1ccc(cc1)c2[nH]c(=O)cc(n2)c3cccnc3 5F-965 c1ccc2c(c1)/C(=N/N)/CC23C4CC5CC(C4)CC3C5 5F-966 CCOC(=O)/C(=C(/C(=C/c1ccccc1)/NC(=O)c2ccccc2)\O)/C#N 5F-967 c1ccc(c(c1)/C=N/Nc2c(=O)[nH]c3ccccc3n2)F 5F-969 CCOC(=O)Cn1nc(nn1)c2ccccc2 5F-970 c1ccc2c(c1)/C(=N/NC(=O)Nc3ccc(cc3)Cl)/CC24C5CC6CC(C5)CC4C6 5F-971 c1ccc2c(c1)/C(=N/NC(=O)c3ccc(cc3Cl)Cl)/CC24C5CC6CC(C5)CC4C6 5F-972 CC(C)(C(=O)/C(=C/c1ccc(cc1)OC)/C#N)n2cncn2 5G-001 CC(C)(C(=O)/C(=C/c1ccc(cc1Cl)Cl)/C#N)n2cncn2 5G-002 c1cc(sc1)CN/C(=N\Cc2cccs2)/c3c(cc(cn3)C(F)(F)F)Cl 5G-003 c1cc(cnc1)Oc2cc(cnc2C#N)C(F)(F)F 5G-004 Cn1c(c(c(c1Cl)C=O)C=O)c2ccccc2 5G-005 c1cc(cc(c1)Oc2cc(cnc2C(=O)N)C(F)(F)F)C(F)(F)F 5G-006 c1cc(cc(c1)Oc2cc(cnc2C#N)C(F)(F)F)C(F)(F)F 5G-007 c1cc(cc(c1)F)Oc2cc(cnc2C#N)C(F)(F)F 5G-008 c1cc(ccc1NC(=O)/C(=N/Nc2ccc(c(c2)Cl)Cl)/N=N/c3ccc(c(c3)Cl)Cl)OC(F)(F)F 5G-009 COc1ccc(cc1)Oc2cc(cnc2C#N)C(F)(F)F 5G-011 c1cc(ccc1C(F)(F)F)N/N=C(/C(=O)Nc2ccc(cc2)OC(F)(F)F)\N=N\c3ccc(cc3)C(F)(F)F 5G-012 CN(C)/C=C(/c1c(cc(cn1)C(F)(F)F)Cl)\S(=O)(=O)c2ccccc2 5G-013 CO/N=C/C(c1c(cc(cn1)C(F)(F)F)Cl)S(=O)(=O)c2ccccc2 5G-014 c1ccc(cc1)S(=O)(=O)C(/C=N/OCc2c(cccc2Cl)Cl)c3c(cc(cn3)C(F)(F)F)Cl 5G-015 COc1ccc(cc1)N/N=C(/C=N\OC)\C(=O)c2ccccc2 5G-016 c1cc(ccc1Oc2cc(cnc2C#N)C(F)(F)F)F 5G-017 c1c(cnc(c1Cl)C(=O)N)C(F)(F)F 5G-018 c1c(cnc2c1n3c(c(nn3)C(=O)N)nc2N)C(F)(F)F 5G-019 Cc1c(nnn1c2cc(cnc2C#N)C(F)(F)F)C(=O)C 5G-020 c1cc(cc(c1)F)Oc2cc(cnc2C(=O)N)C(F)(F)F 5G-021 c1cc(ccc1Oc2cc(cnc2C(=O)N)C(F)(F)F)F 5G-022 CO/N=C/C(=N\Nc1ccc(cc1)[N+](=O)[O-])/C(=O)c2ccccc2 5G-023 CO/N=C/C(=N\Nc1ccc(cc1)Cl)/C(=O)c2ccccc2 5G-024 Cc1c(nnn1c2cc(cnc2C#N)C(F)(F)F)/C(=N/O)/C 5G-025 CO/N=C/C(=N\Nc1ccccc1)/C(=O)c2ccccc2 5G-026 c1cnn(c1)c2c(cc(cn2)C(F)(F)F)Cl 5G-027 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/C(=N\Nc2c(cc(cn2)C(F)(F)F)Cl)/C 5G-028 c1cc(ccc1Sc2cc(cnc2c3nc[nH]n3)C(F)(F)F)Cl 5G-029 CC(C)(C(=O)/C(=C/c1cccs1)/C#N)n2cncn2 5G-031 CC(C)(C(=O)/C(=C/c1ccco1)/C#N)n2cncn2 5G-032 c1cc(ccc1NC(=O)NC(=O)c2c(cc(cn2)C(F)(F)F)Sc3ccc(cc3)Cl)Cl 5G-033 CC(C)(C(=O)c1cnoc1N)n2cncn2 5G-035 c1cc(ccc1C(F)(F)F)Oc2cc(cnc2C#N)C(F)(F)F 5G-036 COc1ccc(cc1)Oc2cc(cnc2C(=O)N)C(F)(F)F 5G-038 CC(C)(c1c(cnn1S(=O)(=O)c2ccc(cc2Cl)Cl)C#N)n3cncn3 5G-039 c1ccc(cc1)NC(=O)/C(=N/Nc2ccc(cc2)Cl)/N=N/c3ccc(cc3)Cl 5G-040 CN(C)/C=N/C(=O)c1c(cc(cn1)C(F)(F)F)Cl 5G-041 c1cc(cnc1)Oc2cc(cnc2C(=O)N)C(F)(F)F 5G-042 c1ccc(cc1)NC(=O)/C(=N/Nc2ccc(c(c2)Cl)Cl)/N=N/c3ccc(c(c3)Cl)Cl 5G-043 c1cc(ccc1Nc2cc(cnc2C#N)C(F)(F)F)F 5G-044 c1ccc(cc1)NC(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/N=N/c3ccc(cc3)C(F)(F)F 5G-045 CC1(CC(=CC(=O)C1)/C=C/Nc2cccc(c2)C(F)(F)F)C 5G-046 CC1(CC(=CC(=O)C1)/C=C/Nc2ccc(cc2)C(F)(F)F)C 5G-047 CC1(CC(=CC(=O)C1)/C=C/Nc2cc(cc(c2)Cl)Cl)C 5G-048 CC1(CC(=CC(=O)C1)/C=C/Nc2ccc(cc2)[N+](=O)[O-])C 5G-049 c1cc(ccc1N2CCN(CC2)c3cc(cnc3C#N)C(F)(F)F)F 5G-050 CC(C)(C(=O)/C(=C/c1cccc(c1)C(F)(F)F)/C#N)n2cncn2 5G-051 c1cc(ccc1C(F)(F)F)Oc2cc(cnc2C(=O)N)C(F)(F)F 5G-052 CC(C)(c1c(cnn1S(=O)(=O)C)C#N)n2cncn2 5G-054 c1ccc(cc1)OP(=O)(C(c2ccncc2)O)Oc3ccccc3 5G-055 c1ccc(cc1)OP(=O)(C(c2ccc(cc2Cl)Cl)O)Oc3ccccc3 5G-056 CCCCOC(=O)C1=Cc2cc(ccc2OC1)Cl 5G-301S COc1ccc2c(c1)C=C(CO2)C(=O)O 5G-302S CCn1c(nnc1S)c2csc(n2)c3ccccc3 5G-303S c1cc(cc(c1)Cl)NC(=O)C2=Cc3cc(ccc3OC2)Cl 5G-304S c1cc(ccc1CNC(=O)C2=Cc3cc(ccc3OC2)Cl)Cl 5G-305S Cn1c(c(c(n1)C(F)(F)F)C=O)Oc2ccccc2 5G-307S Cn1c(c(c(n1)C(F)(F)F)CO)Oc2ccccc2 5G-308S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Oc3ccc(cc3)Cl 5G-309S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2ccc(cc2)Cl)Oc3ccc(cc3)Cl 5G-310S Cn1c(c(c(n1)C(F)(F)F)CO)S(=O)(=O)c2ccc(cc2)F 5G-311S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3cccc(c3)C(F)(F)F 5G-312S Cn1c(c(c(n1)C(F)(F)F)COC(=O)CCl)Sc2ccc(cc2)F 5G-314S CCC(=O)OCc1c(nn(c1Sc2ccc(cc2)F)C)C(F)(F)F 5G-315S CC(=O)OCc1c(nn(c1S(=O)(=O)c2ccc(cc2)Cl)C)C(F)(F)F 5G-316S CC(=O)OCc1c(nn(c1Oc2ccccc2)C)C(F)(F)F 5G-317S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Oc3ccccc3 5G-318S CC(=O)OCc1c(nn(c1Oc2ccc(cc2)Cl)C)C(F)(F)F 5G-319S CCn1c(nnc1S)c2c(nc(s2)c3ccccc3)C 5G-320S CCn1c(nnc1SCc2cccc(c2)C(F)(F)F)c3csc(n3)c4ccccc4 5G-321S CCn1c(nnc1SCc2ccc(cc2)Cl)c3csc(n3)c4ccccc4 5G-322S CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3csc(n3)c4ccccc4 5G-323S c1cc(cc(c1)NC(=O)C2=Cc3cc(ccc3OC2)Cl)C(F)(F)F 5G-324S COc1ccc2c(c1)C=C(CO2)C(=O)OC 5G-325S Cc1ccc(cc1)NC(=O)C2=Cc3cccc(c3OC2)OC 5G-326S COc1ccc(cc1)NC(=O)C2=Cc3cccc(c3OC2)OC 5G-327S CCn1c(nnc1SC)c2c(nc(s2)c3ccccc3)C 5G-328S c1c(snn1)S(=O)C2CCCCC2 5G-329S c1c(snn1)S(=O)(=O)C2CCCCC2 5G-330S COc1cccc2c1OCC(=C2)C(=O)Nc3ccc(cc3Cl)Cl 5G-331S COc1cccc2c1OCC(=C2)C(=O)Nc3ccc(cc3)OC(F)(F)F 5G-332S COc1cccc2c1OCC(=C2)C(=O)Nc3nccs3 5G-333S CCOC(=O)C(C)Sc1cnns1 5G-334S Cn1c(c(c(n1)C(F)(F)F)CNc2ccc(cc2F)F)Sc3ccc(cc3)F 5G-336S CC(C)S(=O)c1cnns1 5G-337S c1cc(ccc1NC(=O)c2ccncc2)Cl 5G-339S COc1cccc2c1OCC(=C2)C(=O)n3cccn3 5G-340S Cc1c(sc(n1)c2ccccc2)c3nnc(n3C)S 5G-341S COc1cccc2c1OCC(=C2)C(=O)Nc3c(cc(cc3Cl)OC(F)(F)F)Cl 5G-342S Cc1c(sc(n1)c2ccccc2)c3nnc(n3C)SCC#C 5G-345S Cc1c(sc(n1)c2ccccc2)c3nnc(n3C)SC 5G-346S CCC(=O)OCc1c(nn(c1Sc2ccc(cc2)Cl)C)C(F)(F)F 5G-349S Cn1c(c(c(n1)C(F)(F)F)CO)S(=O)(=O)c2ccc(cc2)Cl 5G-351S Cn1c(c(c(n1)C(F)(F)F)CO)S(=O)(=O)c2ccc(cc2)Br 5G-352S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 5G-353S Cn1c(c(c(n1)C(F)(F)F)CO)Oc2cccc(c2)C(F)(F)F 5G-355S Cn1c(c(c(n1)C(F)(F)F)COC(=O)CCl)S(=O)(=O)c2ccc(cc2)F 5G-357S COc1cccc2c1OCC(=C2)C(=O)NCc3ccc(cc3Cl)Cl 5G-359S c1c(cc(c2c1C=C(CO2)C(=O)O)Cl)Cl 5G-360S Cc1c(cccc1Cl)NC(=O)C2=Cc3cccc(c3OC2)OC 5G-361S COc1cccc(c1)CNC(=O)C2=Cc3cccc(c3OC2)OC 5G-362S COc1cccc2c1OCC(=C2)C(=O)Nc3cc(ccc3Cl)Cl 5G-363S CC(C)/N=C(\c1ccncc1)/Nc2ccc(cc2)Cl 5G-364S Cn1c(nnc1S)c2csc(n2)c3ccccc3 5G-365S Cc1c(sc(n1)c2ccccc2)c3nnc(n3C)SCC=C 5G-366S Cc1c(sc(n1)c2ccccc2)c3nnc(n3C)SCc4ccc(cc4)Cl 5G-367S CC(=O)OCc1c(nn(c1Oc2cccc(c2)C(F)(F)F)C)C(F)(F)F 5G-368S CCC(=O)OCc1c(nn(c1Oc2cccc(c2)C(F)(F)F)C)C(F)(F)F 5G-370S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)Oc3cccc(c3)C(F)(F)F 5G-371S COc1cccc2c1OCC(=C2)C(=O)Nc3ccc(c(c3)Cl)Cl 5G-372S CC(C)NC(=O)C1=Cc2cccc(c2OC1)OC 5G-373S c1cc(ccc1NC(=O)C2=Cc3cc(ccc3OC2)Cl)Cl 5G-374S c1cc(c(cc1F)F)NC(=O)C2=Cc3cc(ccc3OC2)Cl 5G-375S Cn1c(c(c(n1)C(F)(F)F)CO)SCc2ccc(cc2)Cl 5G-377S Cn1c(nnc1SCc2ccccc2)c3csc(n3)c4ccccc4 5G-378S COc1ccc2c(c1)C=C(CO2)C(=O)Nc3ccccc3 5G-379S COc1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(cc3)F 5G-380S c1cc(cc(c1)NC(=O)c2ccncc2)C(F)(F)F 5G-381S C/N=C(\c1ccncc1)/Nc2cccc(c2)C(F)(F)F 5G-382S COc1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(cc3F)F 5G-383S CC(=O)OCc1c(nn(c1SCc2ccc(cc2)Cl)C)C(F)(F)F 5G-384S Cn1c(c(c(n1)C(F)(F)F)COC(=O)c2ccc(cc2)Cl)SCc3ccc(cc3)Cl 5G-386S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)SCc3ccc(cc3)Cl 5G-387S c1ccc(cc1)c2nc(cs2)c3nnc(o3)S 5G-388S COc1ccc2c(c1)C=C(CO2)C(=O)NCc3cccc(c3)C(F)(F)F 5G-389S COc1ccc2c(c1)C=C(CO2)C(=O)Nc3cccc(c3)C(F)(F)F 5G-390S COc1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(cc3)Cl 5G-391S c1cc(ccc1c2nc(cs2)C(=O)NN)Cl 5G-393S c1ccc(cc1)c2nc(cs2)c3nnc(o3)SCc4ccc(cc4)Cl 5G-394S c1ccc(cc1)c2nc(cs2)c3nnc(o3)SCc4cccc(c4)C(F)(F)F 5G-395S CCOC(=O)c1c(snn1)Sc2ccc(cc2)Cl 5G-398S CC(C)/N=C(\c1ccncc1)/Nc2cccc(c2)C(F)(F)F 5G-399S Cc1ccc(cc1)NC(=O)C2=Cc3cc(ccc3OC2)OC 5G-400S COc1ccc2c(c1)C=C(CO2)C(=O)Nc3cccc(c3)Cl 5G-401S Cn1c(nnc1S)c2csc(n2)c3ccc(cc3)Cl 5G-402S CCn1c(nnc1S)c2csc(n2)c3ccc(cc3)Cl 5G-403S Cn1c(c(c(n1)C(F)(F)F)COC(=O)C2CC2)Sc3ccc(cc3)F 5G-404S COc1ccc2c(c1)C=C(CO2)C(=O)NCc3ccc(cc3)Cl 5G-405S c1ccc(cc1)c2nc(cs2)c3nnc(o3)c4cccc(c4)C(F)(F)F 5G-406S c1cc(ccc1Sc2c(nns2)C(=O)O)Cl 5G-408S c1ccc(cc1)/C=N/n2cc(nc2N)c3ccc(cc3)Cl 5G-409S Cn1c(c(c(n1)C(F)(F)F)COC(=O)C2CC2)S(=O)(=O)c3ccc(cc3)F 5G-410S CC(=O)OCc1c(nn(c1S(=O)(=O)Cc2ccc(cc2)Cl)C)C(F)(F)F 5G-411S CCC(=O)OCc1c(nn(c1S(=O)(=O)Cc2ccc(cc2)Cl)C)C(F)(F)F 5G-412S COc1ccc2c(c1)C=C(CO2)C(=O)OCCc3ccccc3 5G-413S COc1ccc2c(c1)C=C(CO2)C(=O)OCc3cccnc3 5G-414S COc1ccc(cc1)COC(=O)C2=Cc3cc(ccc3OC2)OC 5G-415S COc1ccccc1NC(=O)c2ccc(nc2)n3cncn3 5G-417S C=CCn1c(nnc1S)c2csc(n2)c3ccc(cc3)Cl 5G-418S Cn1c(nnc1SCc2cccc(c2)C(F)(F)F)c3csc(n3)c4ccc(cc4)Cl 5G-419S Cn1c(nnc1SCc2cccc(c2)Cl)c3csc(n3)c4ccc(cc4)Cl 5G-420S CCC(=O)OCc1c(nn(c1S(=O)(=O)Cc2ccccc2Cl)C)C(F)(F)F 5G-428S Cn1c(c(c(n1)C(F)(F)F)COC(=O)C2CC2)S(=O)(=O)Cc3ccccc3Cl 5G-429S Cn1c(c(c(n1)C(F)(F)F)COC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)Cc3ccc(cc3)Cl 5G-430S c1ccc2c(c1)C=C(CO2)C(=O)NCc3ccc(cc3)Cl 5G-431S c1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(cc3Cl)Cl 5G-432S CCn1c(nnc1SCC#C)c2csc(n2)c3ccc(cc3)Cl 5G-434S c1ccc2cc(ccc2c1)Sc3cnns3 5G-435S c1ccc2cc(ccc2c1)S(=O)c3cnns3 5G-436S c1ccc2c(c1)C=C(CO2)C(=O)NCc3ccc(cc3Cl)Cl 5G-437S COc1ccc(cc1OC)c2nc(cs2)C(=O)NN 5G-440S c1cc(ccc1c2cn(c(n2)N)N)Cl 5G-441S c1ccc2cc(ccc2c1)S(=O)(=O)c3cnns3 5G-442S C/N=C(\c1ccncc1)/Nc2ccc(cc2)Cl 5G-444S c1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc(c(c3)Cl)Cl 5G-445S Cc1c(cccc1Cl)NC(=O)C2=Cc3ccccc3OC2 5G-446S Cn1c(nnc1S)c2csc(n2)c3cccc(c3)C(F)(F)F 5G-448S COc1ccc(cc1OC)c2nc(cs2)c3nnc(n3CC=C)S 5G-449S c1cc(ccc1F)S(=O)(=O)c2cnns2 5G-454S COc1ccc(cc1)NC(=O)C2=Cc3ccccc3OC2 5G-457S c1cc(cc(c1)C(F)(F)F)c2nc(cs2)c3nnc(o3)c4ccc(cc4Cl)Cl 5G-458S COc1ccc(cc1OC)c2nc(cs2)c3nnc(o3)c4ccc(cc4)Cl 5G-459S c1cc(c(cc1Cl)Cl)NC(=O)C2=Cc3cc(ccc3OC2)Cl 5G-462S Cn1c(nnc1SC)c2csc(n2)c3cccc(c3)C(F)(F)F 5G-463S COc1ccc(cc1OC)c2nc(cs2)c3nnc(n3CC=C)SCc4c(cccc4Cl)Cl 5G-464S Cc1ccccc1NC(=O)c2ccc(nc2)n3cncn3 5G-465S CCOC(=O)/C(=N/Nc1ccccc1)/C(=O)C(F)(F)F 5G-466S c1cc(c(cc1[N+](=O)[O-])CBr)Cl 5G-471S c1cc(ccc1C(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)[N+](=O)[O-] 5G-900 c1cc(sc1)C(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5G-901 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5G-902 c1cc(c(cc1Cl)Cl)NC(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5G-903 c1c(cnc(c1Cl)N2CCC3(CC2)N(CCO3)C(=O)NC4CCCCC4)C(F)(F)F 5G-904 c1cc(ccc1NC(=S)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)[N+](=O)[O-] 5G-905 C=CCNC(=S)N1CCOC12CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 5G-906 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCOC34CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 5G-907 c1cc(c(cc1Cl)Cl)/C=N/NC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 5G-909 c1ccnc(c1)SCc2c(snn2)Cl 5G-910 c1cc(ccc1C(F)(F)F)NC(=O)N2CCOC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5G-911 CCOC(=O)c1c(c(on1)C)C(=O)Nc2ccc(cc2)F 5G-912 CCOC(=O)c1c(c(on1)C)C(=O)Nc2ccc(cc2)Cl 5G-913 c1ccc(cc1)C2=CSC3=NCCN23 5G-914 Cc1c(c(no1)C(=O)N)C(=O)Nc2ccc(cc2)Cl 5G-915 c1cnc(nc1)N2CCC(=O)CC2 5G-917 CCOC(=O)c1c(c(on1)C)C(=O)Nc2cccc(c2)C(F)(F)F 5G-918 Cc1c(c(no1)C(=O)N)C(=O)Nc2cccc(c2)C(F)(F)F 5G-919 COc1ccc(cc1)/C=N/NC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 5G-920 c1ccc(cc1)/C=N/NC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 5G-921 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 5G-922 Cc1ccc(cc1)NC(=O)N2CCOC23CCN(CC3)c4ncccn4 5G-924 c1ccc2c(c1)C(=O)N(C2=O)OCc3c(snn3)Cl 5G-925 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNC(=O)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5G-926 C=CCNc1c(cc(cn1)C(F)(F)F)Cl 5G-927 c1cc(cc(c1)SCc2c(snn2)Cl)C(F)(F)F 5G-928 Cc1c(c(no1)c2ccccc2)C(=O)NNC(=O)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5G-929 CCOC(=O)c1c(c(on1)C)C(=O)Nc2nc(cc(n2)C)C 5G-932 Cc1c(c(no1)/C=N\O)C(=O)Nc2ccc(cc2)F 5G-934 CC1(CNC2(N1)CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C 5G-935 CC1(CN(C2(N1)CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)Nc4ccccc4)C 5G-936 CCOC(=O)c1c(c(on1)C)C(=O)Nc2cc(cc(n2)C)C 5G-938 Cc1cc(nc(c1)NC(=O)c2c(onc2C(=O)N)C)C 5G-939 c1ccc(cc1)NC(=O)NNC(=O)C=C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 5G-940 CN(C)/C=C/C(=O)c1ccccc1F 5G-941 CCOC(=O)c1c(con1)C(=O)c2cccc(c2)C(F)(F)F 5G-942 CCOC(=O)c1c(con1)C(=O)c2cccc(c2)Cl 5G-943 Cc1c(c(no1)C#N)C(=O)Nc2ccc(cc2)Cl 5G-944 CCOC(=O)c1c(con1)C(=O)c2ccccn2 5G-945 CN(C)c1ccc(cc1)/C=N/c2c(c3c(s2)CN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C#N 5G-946 CCOC(=O)c1c(con1)C(=O)c2ccco2 5G-948 CCOC(=O)c1c(con1)C(=O)c2cccnc2 5G-949 CCOC(=O)c1c(con1)C(=O)c2ccccc2F 5G-950 c1cc(ccc1F)SCc2c(snn2)Cl 5G-951 c1cc(ccc1CON=C2CCN(CC2)C(=O)N)[N+](=O)[O-] 5G-952 CN(C)/C=N/c1ccn(c(=O)n1)c2c(cc(cn2)C(F)(F)F)Cl 5G-954 CCOC(=O)C1C(C2COCCN2O1)(C(F)(F)F)O 5G-957 c1c(cnc(c1Cl)N2CCC(=C(C#N)C#N)CC2)C(F)(F)F 5G-961 c1ccc2c(c1)C(=O)N(C2=O)CCN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5G-963 CC1=CSC2=NCCN12 5G-964 CCOC(=O)C[N+]1=C2N(CC1)C(=CS2)C.[Br-] 5G-965 CC1=CSC2=[N+](CCN12)CC(=O)c3ccc(cc3)Cl.[Br-] 5G-966 c1ccc2c(c1)CCN(C2CC#N)C(=O)Nc3cccc(c3)Cl 5H-001 CCOC(=O)c1c(sc(=S)s1)S 5H-004 c1ccc(cc1)c2c3cccc(c3c(nc2N)Br)F 5H-005 c1cc2c(c(c1)F)c(nc(c2c3ccc(cc3)F)N)Br 5H-007 c1cc2c(c(c1)F)c(nc(c2c3ccc(cc3)Cl)N)Br 5H-009 CSC(=S)NNc1c(cc(cn1)C(F)(F)F)Cl 5H-010 CCOC(=O)c1c(sc(=S)s1)SCc2ccc(cc2)Cl 5H-011 CCOC(=O)c1c(sc(=S)s1)SCC(=O)c2ccc(cc2)Cl 5H-012 CCOC(=O)C1=C(NC(=O)C1)C 5H-013 CCOC(=O)/C=C(\C)/c1ccc(cc1)Cl 5H-014 CCOC(=O)C\1=C(NC(=O)/C1=C\N(C)C)C 5H-015 c1ccc(cc1)NC(=O)CC2c3ccccc3CCN2 5H-016 c1ccc(cc1)C(C#N)c2cccc(c2C#N)Cl 5H-017 c1cc(sc1)C(C#N)N2CCOCC2 5H-018 c1cc(c(c(c1)Cl)C#N)C(C#N)c2ccc(cc2)F 5H-020 CCOC(=O)C\1=C(NC(=O)/C1=C\Nc2ccccc2)C 5H-022 c1ccc2c(c1)CCN3C2CC(=O)CC3=O 5H-023 c1cc(ccc1/C=C/c2c(cc(cn2)C(F)(F)F)Cl)C#N 5H-024 CN(C)/C=C/1\C(=O)CC2c3ccccc3CCN2C1=O 5H-025 c1cc(sc1)C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3 5H-026 CO/N=C/C1C(=O)CC2c3ccccc3CCN2C1=O 5H-027 c1cc(cnc1)/C=C/c2c(cc(cn2)C(F)(F)F)Cl 5H-028 c1cc2c(c(c1)Cl)c(nc(c2c3ccc(cc3)F)N)Br 5H-029 c1cc(sc1)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 5H-030 c1ccc2c(c1)CCN3C2CC(=O)/C(=C\Nc4ccc(cc4)Cl)/C3=O 5H-031 c1cc(c(c(c1)Cl)C#N)C(C#N)c2ccc(cc2)Cl 5H-033 c1cc(ccc1c2cnn3c2ncc(c3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 5H-034 Cc1cc(c([nH]1)/C(=N\O)/c2ccccc2)C(F)(F)F 5H-037 Cc1cc2ncc(cn2n1)c3c(cc(cn3)C(F)(F)F)Cl 5H-038 c1ccc2c(c1)CCN3C2Cc4c(cno4)C3=O 5H-040 c1ccc(cc1)c2cn[nH]c2N 5H-041 Cc1c(c(ns1)S/C=C/C(=O)c2ccccc2)C#N 5H-042 c1cc(ccc1C(=O)/C=C\SCc2c(cc(cn2)C(F)(F)F)Cl)Cl 5H-044 c1cc(ccc1C(=O)/C=C\Sc2c(cc(cn2)C(F)(F)F)Cl)Cl 5H-045 c1ccc(cc1)c2cc3ncc(cn3n2)c4c(cc(cn4)C(F)(F)F)Cl 5H-047 c1cc(ccc1C(=O)/C=C/n2cc(cc(c2=S)Cl)C(F)(F)F)Cl 5H-049 Cc1c(c2ncc(cn2n1)c3c(cc(cn3)C(F)(F)F)Cl)Br 5H-050 c1cc(ccc1C(=O)/C=C/Sc2nc[nH]n2)Cl 5H-051 c1c(cnc(c1Cl)Sc2nc[nH]n2)C(F)(F)F 5H-052 c1ccc(cc1)/C(=N\OC(=O)Nc2ccc(cc2Cl)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 5H-053 c1cc(sc1)c2cn[nH]c2N 5H-054 c1ccc(cc1)c2c(c3ncc(cn3n2)c4c(cc(cn4)C(F)(F)F)Cl)Br 5H-055 c1cc(ccc1c2ccnc3n2nc(n3)N)F 5H-056 COC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3cccs3 5H-057 c1ccn(c1)c2nc3nccc(n3n2)c4ccc(cc4)F 5H-058 c1cc(ccc1C(C#N)N2CCOCC2)Cl 5H-059 c1cc(sc1)c2cnn3c2ncc(c3)c4c(cc(cn4)C(F)(F)F)Cl 5H-060 CN(C)/C=N/c1nc2nccc(n2n1)c3ccc(cc3)F 5H-061 Cc1cc2ncc(cn2n1)C(=O)N 5H-063 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)no2 5H-064 COc1ccc(cc1)C(C#N)N2CCOCC2 5H-065 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)on2 5H-066 CO/N=C/Nc1nc2nccc(n2n1)c3ccc(cc3)F 5H-067 c1cc(ccc1C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3)Cl 5H-068 c1cc(cnc1)C(C#N)N2CCOCC2 5H-069 Cc1cc2ncc(cn2n1)C(=O)/N=C/N(C)C 5H-070 c1cc(ccc1C(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl 5H-072 COc1ccc(cc1)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 5H-074 c1cc(cnc1)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 5H-076 c1ccc(cc1)c2cnn3c2ncc(c3)c4c(cc(cn4)C(F)(F)F)Cl 5H-077 c1ccc2c(c1)CCN(C2CC#N)C(=O)Nc3ccc(cc3)Cl 5H-078 c1ccc(cc1)N2C(=O)CS(=O)CC2=O 5H-301S c1cc(c(cc1Cl)Cl)CN2C(=O)CSCC2=O 5H-302S CCc1cccc(c1N2C(=O)CSCC2=O)CC 5H-303S c1cc(c(cc1Cl)Cl)CN2C(=O)CS(=O)CC2=O 5H-304S Cc1cc(nc(c1C(=O)c2ccccc2)OC(=O)c3c(cc(cc3Cl)Cl)Cl)C 5H-305S Cc1ccc(cc1)CN2C(=O)CSCC2=O 5H-306S CCc1cccc(c1N2C(=O)CS(=O)CC2=O)CC 5H-307S Cc1cc(nc(n1)C)OC(=O)c2cc(c(cc2Cl)F)F 5H-308S Cc1cc(nc(n1)C)OC(=O)c2c(cccc2Cl)F 5H-310S COc1ccc(cc1)CN2C(=O)CSCC2=O 5H-311S c1cc(c(cc1Cl)Cl)CN2C(=O)CS(=O)(=O)CC2=O 5H-312S Cc1cc(nc(c1C#N)OC(=O)c2c(cc(cc2F)F)F)C 5H-313S Cc1cc(nc(n1)C)OC(=O)c2c(cc(cc2F)F)F 5H-314S Cc1ccc(cc1)CN2C(=O)CS(=O)(=O)CC2=O 5H-315S Cc1ccc(cc1)CN2C(=O)CS(=O)CC2=O 5H-316S c1cc(c(c(c1)Cl)N2C(=O)CS(=O)CC2=O)Cl 5H-317S c1cc(c(cc1CNC(=O)CSCC(=O)O)Cl)Cl 5H-318S COc1ccc(cc1)CN2C(=O)CS(=O)CC2=O 5H-320S c1cc(cc(c1)C(F)(F)F)CNC(=O)CSCC(=O)O 5H-321S c1cc(cc(c1)C(F)(F)F)CN2C(=O)CSCC2=O 5H-322S COc1ccc(cc1)CN2C(=O)CS(=O)(=O)CC2=O 5H-323S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3c(cc(cc3F)F)F)C 5H-324S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3cc(c(cc3Cl)F)F)C 5H-325S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3c(cccc3Cl)F)C 5H-326S c1cc(c(cc1CN2C(=O)CSCC2=O)Cl)Cl 5H-327S c1cc(cc(c1)C(F)(F)F)CNC(=O)CS(=O)CC(=O)O 5H-328S Cc1cc(c2c(c1)c(=O)oc(n2)N(C)C)C 5H-329S c1ccc(c(c1)CNC(=O)CSCC(=O)O)Cl 5H-334S c1cc(c(cc1CNC(=O)CS(=O)CC(=O)O)Cl)Cl 5H-335S Cc1cc(nc(c1C(=O)c2ccccc2)OC(=O)c3c(cc(cc3F)F)F)C 5H-336S Cc1cc(nc(c1C(=O)c2ccccc2)OC(=O)c3cc(c(cc3Cl)F)F)C 5H-337S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC(=O)c3c(ccc(c3F)F)F)C 5H-338S c1cc(c(cc1CN2C(=O)CS(=O)CC2=O)Cl)Cl 5H-342S c1cc(c(cc1CN2C(=O)CS(=O)(=O)CC2=O)Cl)Cl 5H-343S CCCCOc1cnns1 5H-345S CCOCCOc1cnns1 5H-346S c1c(snn1)OCCCCl 5H-347S Cc1ccc(cc1)NC(=O)CS(=O)CC(=O)O 5H-351S Cc1ccc(cc1)NC(=O)CS(=O)(=O)CC(=O)O 5H-352S c1cc(cc(c1)NC(=O)CS(=O)CC(=O)O)C(F)(F)F 5H-354S c1ccc(c(c1)CN2C(=O)CSCC2=O)Cl 5H-355S Cc1cc(c(cc1Cl)C)S(=O)c2cnns2 5H-356S c1cc(cc(c1)C(F)(F)F)CNC(=O)CS(=O)(=O)CC(=O)O 5H-357S Cc1ccc(cc1)N2C(=O)CS(=O)(=O)CC2=O 5H-358S COc1ccc(cc1)NC(=O)CS(=O)CC(=O)O 5H-360S COc1ccc(cc1)NC(=O)CS(=O)(=O)CC(=O)O 5H-361S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl 5H-363S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(cc2Cl)Cl 5H-364S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(c(c2)Cl)Cl 5H-365S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(cc2)NC(=O)C 5H-366S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2cccc(c2)C(F)(F)F 5H-367S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(cc2)OC 5H-368S CCOC(=O)CC1C(=O)NCCN1C(=O)c2cccc(c2)C(F)(F)F 5H-369S CC(C)(C)C(=O)Nc1ccsc1C(=O)OC 5H-370S CC(C)(C)C(=O)Nc1ccsc1C(=O)O 5H-372S CCOc1cnns1 5H-373S c1ccc(cc1)N2CCN(CC2)CC(CSc3ccc(c(c3)Cl)Cl)O 5H-401S CCOC(=O)CC1C(=O)NCCN1 5H-402S CCOC(=O)CC1C(=O)NCCN1C(=O)c2ccc(c(c2)Cl)Cl 5H-403S CCOC(=O)CC1C(=O)NCCN1C(=O)c2c(cccc2Cl)Cl 5H-404S CCOC(=O)CC1C(=O)NCCN1C(=O)c2ccc(cc2Cl)Cl 5H-405S Cc1ccc(cc1)S(=O)(=O)NCc2nnc(n2C)SCc3ccc(cc3)C(F)(F)F 5H-406S Cc1ccc(cc1)S(=O)(=O)NCc2nnc(n2C)SCc3cccc(c3)C(F)(F)F 5H-407S Cc1ccc(cc1)S(=O)(=O)NCc2nnc(n2C)SCc3ccc(cc3)C(C)(C)C 5H-408S CCn1c(nnc1S)C(C)NS(=O)(=O)c2ccc(cc2)Cl 5H-411S CCOC(=O)CC1C(=O)NCCN1C(=O)c2ccc(cc2)Cl 5H-412S CCOC(=O)CC1C(=O)NCCN1C(=O)c2ccccc2 5H-413S CCOC(=O)CC1C(=O)NCCN1C(=O)c2ccc(cc2)C 5H-414S CCn1c(nnc1S)C(Cc2ccccc2)NS(=O)(=O)c3ccc(cc3)F 5H-417S CCCSc1nnc(n1C)CNS(=O)(=O)c2ccc(cc2)C 5H-421S Cc1ccc(cc1)S(=O)(=O)NCc2nnc(n2C)SCC=C 5H-422S Cc1cc(nc(c1)N2C(C(N(C2=O)C)O)O)C 5H-423S CCOC(=O)CC1C(=O)NCCN1C(=O)c2ccc(cc2F)F 5H-424S CCOC(=O)CC1C(=O)NCCN1C(=O)c2c(cccc2F)F 5H-425S Cc1cc(nc(c1)NC(=O)NC)C 5H-426S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(cc2)C 5H-427S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(cc2)Br 5H-428S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(cc2)Cl 5H-429S CCn1c(nnc1SCc2cccc(c2)F)C(C)NS(=O)(=O)c3ccc(cc3)Cl 5H-430S CCn1c(nnc1SCc2ccccc2Cl)C(C)NS(=O)(=O)c3ccc(cc3)Cl 5H-431S CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)C(C)NS(=O)(=O)c3ccc(cc3)Cl 5H-432S CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)C(C)NS(=O)(=O)c3ccc(cc3)Cl 5H-433S CCn1c(nnc1SCc2ccc(cc2)OC)C(C)NS(=O)(=O)c3ccc(cc3)Cl 5H-434S CCn1c(nnc1SCC=C)C(C)NS(=O)(=O)c2ccc(cc2)Cl 5H-435S CCn1c(nnc1SC)C(C)NS(=O)(=O)c2ccc(cc2)Cl 5H-436S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccccc2 5H-437S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccccc2Cl 5H-438S CCOC(=O)CC1C(=O)NCCN1S(=O)(=O)c2ccc(cc2)F 5H-439S Cn1c(nnc1S)C(Cc2ccccc2)NS(=O)(=O)c3ccc(cc3)Cl 5H-440S C=CCn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)Br 5H-441S CCn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)Br 5H-443S CCn1c(nnc1SC)C(Cc2ccccc2)NS(=O)(=O)c3ccc(cc3)F 5H-444S CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)C(Cc3ccccc3)NS(=O)(=O)c4ccc(cc4)F 5H-445S CCn1c(nnc1SCC=C)C(Cc2ccccc2)NS(=O)(=O)c3ccc(cc3)F 5H-446S CCn1c(nnc1SCc2cccc(c2)F)C(Cc3ccccc3)NS(=O)(=O)c4ccc(cc4)F 5H-447S CCn1c(nnc1SCc2cccc(c2)OC)C(Cc3ccccc3)NS(=O)(=O)c4ccc(cc4)F 5H-448S C/C(=N\O)/C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 5H-900 Cc1c(c(n(n1)c2ccccc2)OCC=C)C=C3C(=O)N(C(=O)N(C3=O)C)C 5H-903 c1ccc(cc1)n2c(c(c(n2)C(F)(F)F)C=O)Cl 5H-904 CCOC(=O)C1=NOC(C1)COc2ccccc2C=O 5H-906 C=CCOc1ccc(cc1C=O)Cl 5H-907 CN1C(=O)C(=Cc2cc(ccc2OCC=C)Cl)C(=O)N(C1=O)C 5H-909 c1ccc(cc1)COc2c(cc(cc2Cl)Cl)C=O 5H-911 Cn1c(=O)c2c(n(c1=O)C)OCC3C2c4cc(ccc4OC3)Cl 5H-912 C/[N+](=C/c1cc(cc(c1OCc2ccccc2)Cl)Cl)/[O-] 5H-913 CCOC(=O)c1cc(c(nc1NNS(=O)(=O)c2cccs2)O)C(=O)OCC 5H-917 CCOC(=O)C1=NOC(C1)COc2ccc(cc2C=O)Cl 5H-919 CCOC(=O)C1=NOC(C1)COc2ccccc2/C=N/OC 5H-920 c1cc(ccc1C=O)OCc2c(snn2)Cl 5H-921 Cc1c(c(no1)C(=O)C)C(=O)Nc2ccc(cc2)F 5H-922 c1cc(ccc1/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)OCc3c(snn3)Cl 5H-923 C/[N+](=C\c1ccc(cc1)OCc2c(snn2)Cl)/[O-] 5H-924 c1ccc(c(c1)C=O)OCc2c(snn2)Cl 5H-925 CC(=O)c1c(con1)C(=O)c2ccc(cc2)OC 5H-926 C(c1c(snn1)Cl)O[NH3+].[Cl-] 5H-927 CO/N=C\c1ccccc1OCc2c(snn2)Cl 5H-929 CCOC(=O)C1=NOC(C1)COc2ccc(cc2/C=N\O)Cl 5H-930 CN(C)/C=C/C(=O)c1c(con1)C(=O)c2ccc(cc2)OC 5H-931 CC(=O)c1ccc(s1)CC#N 5J-002 c1cnc(nc1)N2CC/C(=C/Nc3ccc(cc3)Cl)/C2=O 5J-003 CO/N=C\C1CCN(C1=O)c2ncccn2 5J-004 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)N/C=C\3/CCN(C3=O)c4ncccn4 5J-005 c1ccc(cc1)N/C=C\2/CCN(C2=O)c3ncccn3 5J-006 c1cnc(nc1)N2CC/C(=C/Nc3ccc(cc3)OC(F)(F)F)/C2=O 5J-007 CC(=O)c1ccc(s1)/C(=C/N(C)C)/C#N 5J-008 CC(C)(CNc1c(cc(cn1)C(F)(F)F)Cl)SC 5J-009 C/C(=N/O)/c1ccc(s1)CC#N 5J-010 C/C(=N/OC)/c1ccc(s1)CC#N 5J-011 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)OC(F)(F)F)/SC2=O 5J-014 c1ccc2c(c1)/C(=C/Nc3cccc(c3)C(F)(F)F)/SC2=O 5J-015 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)/SC2=O 5J-016 c1ccc(cc1)Oc2ccc(cc2)N/C=C\3/c4ccccc4C(=O)S3 5J-017 C/C(=N/OC)/c1ccc(s1)/C(=C/N(C)C)/C#N 5J-018 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)Cl)/SC2=O 5J-019 c1ccc2c(c1)C(SC2=O)/C=N/OCc3ccc(cc3)Cl 5J-020 C/C(=N\OCc1ccc(cc1Cl)Cl)/c2ccc(s2)CC#N 5J-021 COC(=O)CC1=NN(C(=O)C1)C2CCS(=O)(=O)C2 5J-022 c1ccc(cc1)CNS(=O)(=O)Oc2ccccc2OC(=O)Nc3ccc(cc3)Cl 5J-023 CCOC(=O)C(=CNc1ccc(cc1)Cl)C(=O)OCC 5J-024 CCOC(=O)C(=CNc1ccccc1Cl)C(=O)OCC 5J-025 CCOC(=O)c1cnc2ccc(cc2c1O)Cl 5J-026 CCOC(=O)C(=CNc1ccc(cc1)F)C(=O)OCC 5J-027 CCOC(=O)C(=CNc1cc(cc(c1)C)C)C(=O)OCC 5J-028 CCOC(=O)C(=CNc1ccc(cc1F)F)C(=O)OCC 5J-029 CCOC(=O)c1cnc2c(c1O)cccc2Cl 5J-030 CCOC(=O)c1cnc2ccc(cc2c1O)F 5J-031 CCOC(=O)C(=CNc1ccc(cc1)C)C(=O)OCC 5J-032 CCOC(=O)c1cnc2cc(cc(c2c1O)C)C 5J-033 c1cc(ccc1C(C#N)c2c(cc(cn2)C(F)(F)F)Cl)OS(=O)(=O)c3ccc(cc3)Cl 5J-034 CCOC(=O)c1cnc2ccc(cc2c1Cl)Cl 5J-036 CCOC(=O)c1cnc2c(c1O)cc(cc2F)F 5J-037 CCOC(=O)c1cnc2ccc(cc2c1Cl)F 5J-038 CCOC(=O)c1cnc2c(c1Cl)cccc2Cl 5J-039 CCOC(=O)C(=CNc1ccc(cc1)C(F)(F)F)C(=O)OCC 5J-040 CCOC(=O)c1cnc2ccc(cc2c1O)C 5J-041 CCOC(=O)c1cnc2c(c1Cl)cc(cc2F)F 5J-042 CCOC(=O)c1cnc2cc(cc(c2c1Cl)C)C 5J-043 CCOC(=O)C(=CNc1cc(ccc1C)C)C(=O)OCC 5J-045 CCOC(=O)c1cnc2c(ccc(c2c1O)C)C 5J-046 CCOC(=O)c1cnc2ccc(cc2c1Cl)C 5J-047 CCOC(=O)C(=CNc1ccc(cc1)Br)C(=O)OCC 5J-048 CCOC(=O)C(=CNc1ccc(cc1C)Cl)C(=O)OCC 5J-049 CCOC(=O)c1cnc2c(cc(cc2c1O)Cl)C 5J-050 CCOC(=O)c1cnc2c(cc(cc2c1Cl)Cl)C 5J-051 CCOC(=O)c1cnc2c(ccc(c2c1Cl)C)C 5J-052 CCOC(=O)c1cnc2ccc(cc2c1O)Br 5J-053 CCOC(=O)C(=CNc1ccccc1F)C(=O)OCC 5J-054 CCOC(=O)c1cnc2c(c1O)cccc2F 5J-055 CCOC(=O)c1cnc2c(c1Cl)cccc2F 5J-056 CCOC(=O)C(=CNc1cccc(c1Cl)Cl)C(=O)OCC 5J-057 CCOC(=O)c1cnc2c(c1O)ccc(c2Cl)Cl 5J-058 CCOC(=O)c1cnc2c(c1Cl)ccc(c2Cl)Cl 5J-059 CNc1c(cnc(n1)SCc2ccc(c(c2)Cl)Cl)OC 5J-301S CC(C)Nc1c(cnc(n1)SCc2ccc(c(c2)Cl)Cl)OC 5J-303S CCCn1cnc2c1cc(c(c2NS(=O)(=O)C(F)(F)F)C)C 5J-304S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)OC)C)C 5J-305S c1ccc(cc1)Cn2cc(cc(c2=O)C#N)c3ccccc3 5J-306S c1ccc(cc1)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)C#N 5J-307S c1ccc(cc1)c2cc(c(=O)n(c2)Cc3cccc(c3)C(F)(F)F)C#N 5J-308S c1ccc(cc1)c2cc(c(=O)n(c2)Cc3ccc(cc3)F)C#N 5J-309S COc1cnc(nc1OC)SC 5J-310S COc1cnc(nc1Sc2ccc(cc2)Cl)SC 5J-311S c1cc(ccc1c2cc(c(nc2)Cl)C#N)Cl 5J-312S Cn1cc(cc(c1=O)C#N)c2ccccc2 5J-313S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)F)C)C 5J-314S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)Cl)C)C 5J-315S Cc1cc2c(c(c1C)N(=O)=O)ncn2Cc3cccc(c3)OC 5J-316S Cc1cc2c(c(c1C)N)ncn2Cc3cccc(c3)OC 5J-317S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(c(cc4Cl)Cl)Cl)C)C 5J-318S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cccc(c4)C(F)(F)F)C)C 5J-319S c1ccc(cc1)Oc2c(cc(cn2)c3ccc(cc3)Cl)C#N 5J-320S c1cc(ccc1c2cc(c(nc2)Oc3ccc(cc3)F)C#N)Cl 5J-322S c1cc(ccc1c2cc(c(nc2)Oc3ccc(cc3F)F)C#N)Cl 5J-323S CN(C)/C=C(\C=O)/c1cccc(c1)Cl 5J-324S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)C)C)C 5J-325S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(cc(c4)Cl)Cl)C)C 5J-326S COc1ccc(cc1)Oc2c(cc(cn2)c3ccc(cc3)Cl)C#N 5J-327S Cc1cc2c(cc1C)nc([nH]2)C 5J-328S Cc1cc2c(c(c1C)[N+](=O)[O-])nc([nH]2)C 5J-329S Cc1cccc(c1)Cn2c(nc3c2cc(c(c3N(=O)=O)C)C)C 5J-330S Cc1cccc(c1)Cn2c(nc3c2cc(c(c3N)C)C)C 5J-331S c1cc(cc(c1)Cl)c2cc(c(=O)[nH]c2)C#N 5J-332S c1cc(ccc1Cn2cc(cc(c2=O)C#N)c3ccc(cc3)Cl)F 5J-333S c1cc(ccc1c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)C#N)Cl 5J-334S c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)C#N)c3ccc(cc3)Cl)Cl 5J-335S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)C#N)c3ccc(cc3)Cl 5J-336S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4cc(ccc4Cl)Cl)C)C 5J-337S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4c(cc(cc4Cl)Cl)Cl)C)C 5J-338S CN(C)c1ncc(c(n1)Sc2ccc(cc2)Br)OC 5J-342S CN(C)c1ncc(c(n1)Sc2cccc(c2)C(F)(F)F)OC 5J-343S CN(C)c1ncc(c(n1)Sc2ccc(cc2)OC)OC 5J-344S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(c(c4)Cl)Cl)C)C 5J-345S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4Cl)Cl)C)C 5J-346S Cc1ccc(cc1)Sc2c(cnc(n2)N(C)C)OC 5J-347S CN(C)c1ncc(c(n1)Sc2cccc(c2)Cl)OC 5J-348S CN(C)c1ncc(c(n1)SCc2cccc(c2)C(F)(F)F)OC 5J-349S CCOC(=O)CSc1c(cnc(n1)N(C)C)OC 5J-350S Cc1ccccc1Cn2cnc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)C(C)(C)C)C)C 5J-351S c1ccc(cc1)Cn2cc(cc(c2=O)C#N)c3cccc(c3)Cl 5J-353S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)C#N)c3cccc(c3)Cl 5J-354S c1cc(cc(c1)Cl)c2cc(c(=O)n(c2)Cc3ccc(cc3Cl)Cl)C#N 5J-355S C=CCn1cc(cc(c1=O)C#N)c2cccc(c2)Cl 5J-356S CN(C)/C=C(\C=O)/c1c(cccc1Cl)Cl 5J-357S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)F)ncn2Cc4ccc(cc4)OC 5J-358S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)OC)ncn2Cc4ccc(cc4)OC 5J-359S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)Cl)ncn2Cc4ccc(cc4)OC 5J-361S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccccc3Cl)ncn2Cc4ccc(cc4)OC 5J-362S COc1ccc(cc1)Sc2c(cc(cn2)c3ccc(cc3)Cl)C#N 5J-363S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3)C(F)(F)F)ncn2Cc4ccc(cc4)OC 5J-364S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)ncn2Cc4ccc(cc4)OC 5J-365S CCCCCCCCn1cnc2c1cc(c(c2N(=O)=O)C)C 5J-366S CCCCCCCCn1cnc2c1cc(c(c2N)C)C 5J-367S CCOC(=O)CSc1ncc(c(n1)OC(=O)N(C)C)OC 5J-368S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(c(c3Cl)Cl)Cl)ncn2Cc4ccc(cc4)OC 5J-369S Cc1cc2c(c(c1C)NS(=O)(=O)c3c(cc(cc3Cl)Cl)Cl)ncn2Cc4ccc(cc4)OC 5J-370S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(cc(c3)Cl)Cl)ncn2Cc4ccc(cc4)OC 5J-371S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(ccc3Cl)Cl)ncn2Cc4ccc(cc4)OC 5J-372S CCOC(=O)Cn1c2ccccc2nc1C(C)NC(=O)c3ccc(cc3Cl)Cl 5J-373S c1ccc(cc1)Sc2c(cc(cn2)c3ccc(cc3)Cl)C#N 5J-374S c1ccc(c(c1)Sc2c(cc(cn2)c3ccc(cc3)Cl)C#N)Cl 5J-375S Cc1cc2c(c(c1C)NS(=O)(=O)C)ncn2Cc3ccc(cc3)OC 5J-379S Cc1cc2c(c(c1C)N(=O)=O)nc(n2Cc3ccc(cc3)OC)C 5J-380S Cc1cc2c(c(c1C)N)nc(n2Cc3ccc(cc3)OC)C 5J-381S c1cc(cc(c1)Cl)Sc2c(cc(cn2)c3ccc(cc3)Cl)C#N 5J-382S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)OC)ncn2Cc4cccc(c4)OC 5J-384S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)F)ncn2Cc4cccc(c4)OC 5J-385S c1cc(ccc1c2cc(c(nc2)Sc3ccc(cc3)F)C#N)Cl 5J-386S c1cc(c(c(c1)Cl)Sc2c(cc(cn2)c3ccc(cc3)Cl)C#N)Cl 5J-387S CC(C)Nc1ncc(c(n1)OC)OC 5J-389S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3)C(F)(F)F)ncn2Cc4cccc(c4)OC 5J-390S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3Cl)Cl)ncn2Cc4cccc(c4)OC 5J-391S c1cc(cc(c1)Oc2c(cc(cn2)c3ccc(cc3)Cl)C#N)C(F)(F)F 5J-392S COc1ccccc1Oc2c(cc(cn2)c3ccc(cc3)Cl)C#N 5J-393S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3Cl)Cl)ncn2Cc4cccc(c4)OC 5J-394S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(c(c3)Cl)Cl)ncn2Cc4cccc(c4)OC 5J-395S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(ccc3Cl)Cl)ncn2Cc4cccc(c4)OC 5J-396S CCCCCCCCn1cnc2c1cc(c(c2NS(=O)(=O)c3ccc(cc3)F)C)C 5J-397S c1ccc(cc1)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)C#N 5J-398S COc1cccc(c1)Cn2cc(cc(c2=O)C#N)c3ccccc3 5J-399S COc1cnc(nc1O)SCC(=O)O 5J-400S CCOC(=O)/C(=C/c1ccccc1[N+](=O)[O-])/C#N 5J-401S CCCCCCCCn1cnc2c1cc(c(c2NS(=O)(=O)c3ccc(cc3)OC)C)C 5J-402S CCCCCCCCn1cnc2c1cc(c(c2NS(=O)(=O)c3ccc(c(c3)Cl)Cl)C)C 5J-403S c1ccc(cc1)c2cc(c(=O)n(c2)Cc3ccccc3Cl)C#N 5J-404S c1ccc(cc1)c2cc(c(=O)n(c2)Cc3cccc(c3)Cl)C#N 5J-405S CN(C)c1ncc(c(n1)Oc2cc(cc(c2)Cl)Cl)OC 5J-406S CN(C)c1ncc(c(n1)Oc2cccc(c2)[N+](=O)[O-])OC 5J-407S CN(C)c1ncc(c(n1)Oc2ccc(cc2)C#N)OC 5J-408S c1ccc(cc1)c2cc(c(nc2)Cl)C#N 5J-410S c1cc(cc(c1)Cl)c2cc(c(=O)n(c2)Cc3ccc(cc3)F)C#N 5J-411S c1cc(cc(c1)Cl)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)C#N 5J-412S COc1cnc(nc1Sc2ccc(cc2)Cl)SCc3ccc(cc3Cl)Cl 5J-501S COc1ccc(cc1)Sc2c(cnc(n2)SCc3ccc(cc3Cl)Cl)OC 5J-502S COc1cnc(nc1Sc2ccccc2)SCc3ccc(cc3Cl)Cl 5J-504S CN(C)c1c(cnc(n1)SCc2ccc(cc2Cl)Cl)OC 5J-506S COc1cnc(nc1Sc2ccccc2)SC 5J-510S COc1cnc(nc1Sc2cccc(c2)C(F)(F)F)SC 5J-511S COc1ccc(cc1)Sc2c(cnc(n2)SC)OC 5J-512S COc1cnc(nc1Sc2ccc(c(c2)Cl)Cl)SC 5J-513S COc1cnc(nc1Oc2cc(cc(c2)Cl)Cl)SC 5J-516S c1ccc(cc1)C(=O)NCCSc2ccc(cc2)Br 5J-519S c1cc(ccc1SCCNC(=O)c2ccc(cc2Cl)Cl)Br 5J-520S c1cc(ccc1C(=O)NCCSc2ccc(cc2)Br)F 5J-521S c1cc(ccc1C(=O)NCCS(=O)(=O)c2ccc(cc2)Br)F 5J-522S c1cc(ccc1S(=O)(=O)CCNC(=O)c2ccc(cc2Cl)Cl)Br 5J-523S c1ccc(cc1)C(=O)NCCS(=O)(=O)c2ccc(cc2)Br 5J-524S c1cc(cc(c1)Cl)C(=O)NCCS(=O)c2ccc(cc2)Cl 5J-525S COc1cnc(nc1O)SCc2c(cccc2Cl)Cl 5J-527S Cc1c(nn(c1c2ccccc2)OCc3ccc(c(c3)Cl)Cl)c4ccccc4 5J-529S Cc1c(nn(c1c2ccccc2)OCc3c(cccc3Cl)Cl)c4ccccc4 5J-530S COc1cnc(nc1Cl)SCc2c(cccc2Cl)Cl 5J-531S COc1cnc(nc1OC)SCc2c(cccc2Cl)Cl 5J-533S COc1cnc(nc1Oc2ccc(cc2)Cl)SCc3c(cccc3Cl)Cl 5J-535S COc1cnc(nc1Oc2cc(cc(c2)Cl)Cl)SCc3c(cccc3Cl)Cl 5J-536S COc1cnc(nc1Sc2ccc(cc2)Cl)SCc3c(cccc3Cl)Cl 5J-537S COc1ccc(cc1)Sc2c(cnc(n2)SCc3c(cccc3Cl)Cl)OC 5J-538S COc1cnc(nc1Sc2cccc(c2)C(F)(F)F)SCc3c(cccc3Cl)Cl 5J-539S COc1cnc(nc1Sc2ccccc2)SCc3c(cccc3Cl)Cl 5J-540S COc1cnc(nc1Oc2ccc(c(c2)Cl)Cl)SCc3c(cccc3Cl)Cl 5J-541S COc1ccc(cc1)Oc2c(cnc(n2)SCc3c(cccc3Cl)Cl)OC 5J-542S COc1ccc(cc1)Oc2c(cnc(n2)SC)OC 5J-543S COc1cnc(nc1Oc2ccc(c(c2)Cl)Cl)SC 5J-544S COc1cnc(nc1Oc2ccc(cc2Cl)Cl)SC 5J-545S c1ccc(c(c1)C(=O)NCCSc2ccc(cc2)Br)Cl 5J-547S c1ccc(c(c1)C(=O)NCCS(=O)(=O)c2ccc(cc2)Br)Cl 5J-548S c1cc(cc(c1)C(F)(F)F)C(=O)NCCSc2ccc(cc2)Br 5J-549S c1cc(ccc1C(=O)NCCS(=O)(=O)c2ccc(cc2)Br)Cl 5J-550S c1cc(ccc1SCCNS(=O)(=O)c2ccc(c(c2Cl)Cl)Cl)Br 5J-551S c1cc(cc(c1)Cl)c2cnn(c2)c3cccc(c3)Cl 5J-554S Cc1c(nn(c1c2ccccc2)OS(=O)(=O)N(C)C)c3ccccc3 5J-555S Cc1c(nn(c1c2ccccc2)OCc3cccc(c3)C(F)(F)F)c4ccccc4 5J-557S Cc1c(nn(c1c2ccccc2)OCc3ccc(cc3)C(=O)OC)c4ccccc4 5J-558S c1cc(cc(c1)Cl)c2cnn(c2)c3cccc(c3)[N+](=O)[O-] 5J-559S c1cc(cc(c1)Cl)c2cnn(c2)c3cccc(c3)C(F)(F)F 5J-560S c1cc(cc(c1)Cl)c2cnn(c2)c3ccc(c(c3Cl)Cl)Cl 5J-561S c1ccc(c(c1)c2cnn(c2)c3c(cc(cc3Cl)C(F)(F)F)Cl)Cl 5J-562S Cc1cccc(c1)n2cc(cn2)c3cccc(c3)Cl 5J-563S c1cc(cc(c1)Cl)c2cnn(c2)c3cccc(c3)F 5J-565S CC1(CO1)C(=O)Nc2ccc(cc2)C(F)(F)F 5J-567S COc1cnc(nc1Oc2cc(cc(c2)Cl)Cl)SCc3cccc(c3)C(F)(F)F 5J-570S Cc1ccc(cc1)Sc2c(cccn2)c3nc4cc(ccc4o3)Cl 5J-576S c1cc(cc(c1)C(F)(F)F)C(=O)NCCS(=O)(=O)c2ccc(cc2)Br 5J-577S c1cc(c(c(c1)F)C(=O)NCCS(=O)(=O)c2ccc(cc2)Br)F 5J-578S CN(C)/C=C(\C=O)/c1cccc(c1)C(F)(F)F 5J-579S c1ccc(cc1)/C(=C\c2ccc(cc2)F)/C(=O)c3ccccc3 5J-582S c1cc(cc(c1)C(F)(F)F)c2cnn(c2)c3c(cc(cc3Cl)C(F)(F)F)Cl 5J-586S CC(CS(=O)(=O)c1ccccc1)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-590S CC(CS(=O)(=O)c1ccc(cc1)Br)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-591S CC(CS(=O)(=O)c1cccc(c1)C(F)(F)F)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-592S CC(CS(=O)(=O)c1c(cccc1Cl)Cl)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-593S CC(CS(=O)(=O)Cc1ccccc1)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-594S CC(CS(=O)(=O)c1ccc(cc1)F)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-595S CC(CS(=O)(=O)C1CCCCC1)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-596S CC(CS(=O)(=O)c1ccc(cc1)Cl)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-597S CC(CSc1ccc(cc1)OC)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-598S CC(CS(=O)(=O)c1ccc(cc1)OC)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-599S CC(CS(=O)(=O)c1cc(cc(c1)Cl)Cl)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-600S CC(CS(=O)(=O)Cc1ccccc1Cl)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-601S CC(CS(=O)(=O)Cc1cccc(c1)C(F)(F)F)(C(=O)Nc2ccc(cc2)C(F)(F)F)O 5J-602S c1ccc(cc1)Sc2c(cccn2)c3nc4cc(ccc4o3)Cl 5J-603S c1cc(c(nc1)Sc2ccc(cc2)Br)c3nc4cc(ccc4o3)Cl 5J-605S c1cc(cc(c1)Sc2c(cccn2)c3nc4cc(ccc4o3)Cl)C(F)(F)F 5J-606S c1cc(cc(c1)C(F)(F)F)c2cnn(c2)c3cccc(c3)Cl 5J-608S c1cc(cc(c1)C(F)(F)F)c2cnn(c2)c3cccc(c3)[N+](=O)[O-] 5J-610S Cc1cccc(c1)n2cc(cn2)c3cccc(c3)C(F)(F)F 5J-611S c1cc(cc(c1)C(F)(F)F)c2cnn(c2)c3cccc(c3)Br 5J-612S c1cc(cc(c1)Cl)c2cnn(c2)c3cccc(c3)Br 5J-613S COC(CNC(=S)Nc1ccc(cc1)Cl)OC 5J-900 c1cc(ccc1n2ccnc2S)Cl 5J-901 CC(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 5J-902 c1cc(ccc1n2ccnc2SCc3c(snn3)Cl)Cl 5J-903 c1cc(ccc1N2C(=O)NC3(N2)CCC4(CC3)OCCO4)Cl 5J-904 c1cc(ccc1N2C(=O)NC3(N2)CCC(=O)CC3)Cl 5J-905 c1ccc(cc1)N2C(=O)NC3(N2)CCC4(CC3)NC(=O)N(N4)c5ccc(cc5)Cl 5J-906 c1cc(ccc1N2C(=O)NC3(N2)CCC4(CC3)NC(=O)N(N4)c5ccc(cc5)Cl)Cl 5J-907 CN1C(CC(O1)CN(N(C)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)c3ccc(cc3)OC)c4ccc(cc4)OC 5J-908 Cc1ccc(cc1)n2c(cc(nc2=O)N3CCN(CC3)c4ccc(cc4)OC)N 5J-909 COc1ccc(cc1)N2CCN(CC2)c3cc(n(c(=O)n3)C4CCCCC4)O 5J-910 c1c(cnc(c1Cl)C(C#N)C#N)C(F)(F)F 5K-001 COc1ccnc(c1C#N)Oc2cccc(c2)C(F)(F)F 5K-002 Cc1cc(nc2c1c(c(s2)/C=C/C(=O)OC)n3cccc3)C 5K-006 Cc1cc(nc2c1c(c(s2)/C=C/C#N)/N=C/N(C)C)C 5K-007 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 5K-008 COc1cc(cc(c1)OC)N/N=C(\C=N\OC)/C(=O)c2ccccc2 5K-009 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)N 5K-010 COc1ccc(cc1)NC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 5K-011 CC(C)c1ccc(cc1)NC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 5K-012 Cc1cc(cc(c1)NC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl)C 5K-013 c1cc(cc(c1)NC(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 5K-014 Cc1cc(nc2c1c(c(s2)/C=C/C(=O)OC)/N=C/N(C)C)C 5K-015 COc1ccnc(c1C(=O)N)Oc2cccc(c2)C(F)(F)F 5K-016 C#CCSc1nccn1c2c(cc(cn2)C(F)(F)F)Cl 5K-017 COC(=O)/C=C/Cn1cncn1 5K-018 CSc1nccn1c2c(cc(cn2)C(F)(F)F)Cl 5K-019 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Br 5K-020 c1cc(ccc1CSc2nccn2c3c(cc(cn3)C(F)(F)F)Cl)Cl 5K-021 Cc1c2ccccc2oc1/C=C/C(=O)OC 5K-022 CO/N=C/C(C#N)c1ccc(cc1)Cl 5K-023 COC(=O)/C=C/c1cc2ccccc2o1 5K-024 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)F 5K-025 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3F)F 5K-026 c1ccc2c(c1)CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl 5K-027 CN(C)/C=C/C(=O)c1cccc(c1)[N+](=O)[O-] 5K-030 c1ccc(cc1)S(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl 5K-032 c1ccc(cc1)S(=O)(=O)c2c(cc(cn2)C(F)(F)F)O 5K-033 CON/C=C/C(=O)c1ccc(cc1)[N+](=O)[O-] 5K-034 COc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)F 5K-035 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)NN 5K-036 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)OC)/C=N/OC 5K-037 c1ccc(cc1)NC(=S)NNC(=O)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 5K-038 CNC(=S)NNC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3ccccc3 5K-039 COc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)c2ccc(c(c2)Cl)Cl 5K-040 Cn1c(nnc1S)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4ccccc4 5K-041 c1ccc(cc1)n2c(nnc2S)c3c(c4c(s3)cc(cn4)C(F)(F)F)c5cccs5 5K-042 c1ccc2c(c1)CCN(C2=O)c3c(cc(cn3)C(F)(F)F)Cl 5K-043 c1cc(ccc1Sc2c(cc(cn2)C(F)(F)F)Cl)Cl 5K-044 COc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)Cl 5K-046 COc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)Br 5K-047 Cn1c(nnc1SC)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4ccccc4 5K-048 CSc1nnc(n1c2ccccc2)c3c(c4c(s3)cc(cn4)C(F)(F)F)c5cccs5 5K-049 CCSc1nnc(n1C)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 5K-050 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)c3ccc(cc3)Cl 5K-053 Cc1c(c(=O)cco1)OCc2ccc(cc2)F 5K-054 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)NS(=O)(=O)c3ccc(cc3)Cl 5K-055 Cc1ccc(cc1)Cn2ccc(=O)c(c2C)OCc3c(cccc3Cl)Cl 5K-056 Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cccc(c3)C(F)(F)F)Sc4ccc(cc4)Cl 5K-301S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cccc(c3)C(F)(F)F)S(=O)(=O)c4ccc(cc4)Cl 5K-302S Cc1ccc(cc1S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C)F 5K-304S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3Cl)Cl)Sc4ccc(cc4)Cl 5K-305S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3Cl)Cl)S(=O)(=O)c4ccc(cc4)Cl 5K-306S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Sc4ccc(cc4)Cl 5K-307S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)S(=O)(=O)c4ccc(cc4)Cl 5K-308S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)C#N)Sc4ccc(cc4)Br 5K-309S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)C#N)S(=O)(=O)c4ccc(cc4)Br 5K-310S Cc1ccccc1S(=O)(=O)c2c(cc(nc2Nc3ccccc3)C)C 5K-311S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cccc(c3)Cl)Sc4ccc(cc4)Br 5K-312S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cccc(c3)Cl)S(=O)(=O)c4ccc(cc4)Br 5K-313S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3Cl)Cl)Oc4ccc(cc4)F 5K-315S Cc1ccccc1C(=O)OCc2c(nn(c2Sc3ccc(cc3)Br)C)c4ccccc4 5K-316S Cc1ccccc1C(=O)OCc2c(nn(c2S(=O)(=O)c3ccc(cc3)Br)C)c4ccccc4 5K-317S Cc1cc([nH]c(=O)c1S(=O)(=O)c2cccc(c2C)Br)C 5K-318S Cc1cc([nH]c(=O)c1S(=O)(=O)Cc2ccccc2)C 5K-319S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)Br)Oc4ccc(cc4)F 5K-320S Cc1cc([nH]c(=O)c1S(=O)(=O)CCC(C)C)C 5K-321S Cc1cc([nH]c(=O)c1S(=O)(=O)C(C)C)C 5K-322S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3c(cccc3Cl)F)Oc4ccc(cc4)F 5K-323S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccccc3Cl)Oc4ccc(cc4)F 5K-324S Cn1c(c(c(n1)c2ccccc2)COC(=O)Nc3cccc(c3)Cl)Sc4ccc(cc4)Br 5K-325S Cc1cc(nc(c1S(=O)(=O)Cc2ccccc2)Cl)C 5K-326S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cccc(c3)C(F)(F)F)Oc4ccc(cc4)F 5K-328S Cc1cc(nc(c1S(=O)(=O)c2cccc(c2C)Br)Cl)C 5K-329S COc1c(nnc(n1)c2ccccc2)C(=O)OC 5K-333S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)F)S(=O)(=O)c4ccccc4 5K-336S Cc1cc(nc(c1S(=O)(=O)C(C)C)Cl)C 5K-337S Cc1cc(nc(c1S(=O)(=O)Cc2ccccc2)OC(C)C)C 5K-338S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cccc(c3)Cl)Sc4ccccc4 5K-339S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cccc(c3)Cl)S(=O)(=O)c4ccccc4 5K-340S Cc1cc(nc(c1S(=O)(=O)c2cccc(c2C)Br)OCC(C)C)C 5K-341S Cc1cc(nc(c1S(=O)(=O)C(C)C)OC(C)C)C 5K-342S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccc(cc3)Cl 5K-345S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3cccc(c3)C(F)(F)F 5K-346S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccc(cc3)OC 5K-347S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(c(c3)Cl)Cl)Sc4ccccc4 5K-348S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(c(c3)Cl)Cl)S(=O)(=O)c4ccccc4 5K-349S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)C#N)Oc4cccc(c4)C(F)(F)F 5K-350S CC(C)Oc1c(nnc(n1)c2ccccc2)C(=O)OC(C)C 5K-351S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(c(c3)Cl)Cl)Oc4cccc(c4)C(F)(F)F 5K-352S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)F)Oc4cccc(c4)C(F)(F)F 5K-354S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3c(cccc3F)F)Oc4cccc(c4)C(F)(F)F 5K-355S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Oc4cccc(c4)C(F)(F)F 5K-357S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3Cl)Cl)Oc4cccc(c4)C(F)(F)F 5K-358S Cn1c(c(c(n1)c2ccccc2)COC(=O)Nc3cccc(c3)Cl)Sc4ccccc4 5K-359S c1ccc(cc1)c2c(nsn2)Cl 5K-360S CC(=O)OCc1c(nn(c1Sc2ccccc2Cl)C)c3ccccc3 5K-361S Cn1c(c(c(n1)c2ccccc2)CCl)Sc3ccccc3Cl 5K-362S Cn1c(c(c(n1)c2ccccc2)COC)Sc3ccccc3Cl 5K-363S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Sc4ccccc4Cl 5K-364S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(c(c3)Cl)Cl)Sc4ccccc4Cl 5K-365S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccccc3 5K-366S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccc(cc3Cl)Cl 5K-367S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)F)Sc4cccc(c4)C(F)(F)F 5K-370S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3)C#N)Sc4cccc(c4)C(F)(F)F 5K-371S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Sc4cccc(c4)C(F)(F)F 5K-374S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)S(=O)(=O)c4cccc(c4)C(F)(F)F 5K-375S Cn1c(c(nc1S(=O)(=O)Cc2cccc(c2)F)c3ccccc3)c4ccccc4 5K-501S CCCn1c(c(nc1S(=O)(=O)Cc2cccc(c2)F)c3ccccc3)c4ccccc4 5K-502S C=CCn1c(c(nc1S(=O)(=O)Cc2cccc(c2)F)c3ccccc3)c4ccccc4 5K-503S C#CCn1c(c(nc1S(=O)(=O)Cc2cccc(c2)F)c3ccccc3)c4ccccc4 5K-504S CC(c1c(nn(c1Cl)C)c2ccccc2)O 5K-505S CCC(c1c(nn(c1Cl)C)c2ccccc2)O 5K-506S Cn1c(c(c(n1)c2ccccc2)C(C#Cc3ccccc3)O)Cl 5K-507S Cn1c(c(c(n1)c2ccccc2)C(c3cccs3)O)Cl 5K-508S Cn1c(c(c(n1)c2ccccc2)C(CC=C)O)Cl 5K-509S CCOC(=O)Cn1c(c(nc1S(=O)(=O)Cc2cccc(c2)F)c3ccccc3)c4ccccc4 5K-510S Cc1ccc(cc1)CS(=O)(=O)c2nc(c(n2C)c3ccccc3)c4ccccc4 5K-511S CCCn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)C)c3ccccc3)c4ccccc4 5K-512S Cc1ccc(cc1)CS(=O)(=O)c2nc(c(n2CC#C)c3ccccc3)c4ccccc4 5K-515S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3ccc(cc3)Br 5K-523S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3cccc(c3)C(F)(F)F 5K-524S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3c(cccc3Cl)Cl 5K-525S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)Nc4ccccc4 5K-526S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)Nc4ccc(cc4)OC(F)(F)F 5K-527S C#CCn1c(c(nc1SCc2cccc(c2)Cl)c3ccccc3)c4ccccc4 5K-529S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3ccc(cc3)OC 5K-531S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3ccccc3C 5K-532S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3cc(ccc3C)C 5K-533S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)Nc4ccc(cc4)F 5K-534S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)Nc4ccc(cc4F)F 5K-535S c1ccc(cc1)c2c(sc(n2)c3ccc(cc3)Cl)CC(=O)Nc4cccc(c4)C(F)(F)F 5K-536S COC(=O)Cc1c(nc(s1)c2ccccc2Cl)c3ccccc3 5K-537S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)O 5K-538S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)Nc4ccc(cc4)Cl 5K-541S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)Nc4ccc(c(c4)Cl)Cl 5K-542S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)Nc4ccccc4 5K-543S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)Nc4ccc(cc4)OC(F)(F)F 5K-544S COc1ccc(cc1)NC(=O)Cc2c(nc(s2)c3ccccc3Cl)c4ccccc4 5K-545S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)Nc4cccc(c4)C(F)(F)F 5K-546S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)Nc4ccc(cc4)F 5K-547S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)Nc4ccc(cc4F)F 5K-548S Cn1c(c(c(n1)c2ccccc2)C(=O)OC)Cl 5K-549S CCOC(=O)Cn1c(c(nc1S(=O)(=O)Cc2ccc(cc2)Cl)c3ccccc3)c4ccccc4 5K-553S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)O 5K-554S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3ccccc3Cl 5K-555S Cc1c(c(n(n1)C)Cl)/C=C/c2ccccc2 5K-557S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3ccc(cc3)C 5K-558S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3ccc(cc3)F 5K-559S CCOC(=O)c1c(nc(nn1)c2ccccc2)Sc3ccccc3C(=O)OC 5K-560S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3ccc(cc3)Cl 5K-561S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccc(cc3)Br 5K-562S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3ccc(cc3)C 5K-563S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3cccc(c3)C(F)(F)F 5K-564S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3ccc(cc3)F 5K-565S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3c(cccc3Cl)Cl 5K-566S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3c(cccc3C)C 5K-567S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3ccccc3Cl 5K-568S CCOC(=O)c1c(nc(nn1)c2ccccc2)Oc3ccc(cc3)OC 5K-569S Cc1cccc(c1NC(=O)c2cc(cc(c2N)Cl)Cl)C 5K-576S Cc1cccc(c1n2c(nc3c(c2=O)cc(cc3Cl)Cl)CCl)C 5K-583S CSCc1nc2ccccc2c(=O)n1c3ccc(c(c3)Cl)Cl 5K-584S c1ccc(cc1)c2c(sc(n2)c3ccccc3Cl)CC(=O)NC4CCCCC4 5K-586S C=CCNC(=O)Cc1c(nc(s1)c2ccccc2Cl)c3ccccc3 5K-587S Cc1cccc(c1n2c(nc3c(c2=O)cc(cc3Cl)Cl)CSCc4ccccc4)C 5K-588S Cc1cccc(c1n2c(nc3c(c2=O)cc(cc3Cl)Cl)CSc4cccc(c4)C(F)(F)F)C 5K-589S Cc1cccc(c1n2c(nc3c(c2=O)cc(cc3Cl)Cl)CSc4ccc(cc4)Br)C 5K-590S c1cc(ccc1c2csc(n2)N)Cl 5K-591S c1cc(ccc1c2csc(n2)NC(=O)CCl)Cl 5K-592S c1ccc(c(c1)c2csc(n2)N)Cl 5K-594S c1ccc(c(c1)c2csc(n2)NC(=O)CCl)Cl 5K-595S c1cc(ccc1c2csc(n2)N)F 5K-596S c1cc(ccc1c2csc(n2)NC(=O)CCl)F 5K-597S c1ccc(cc1)c2csc(n2)N 5K-598S c1ccc(cc1)c2csc(n2)NC(=O)CCl 5K-599S Cn1c(c(c(n1)c2ccccc2)C(c3ccccc3)OC)Cl 5K-600S c1cc(ccc1c2csc(n2)NC(=O)CSc3ccc(cc3)Cl)Cl 5K-602S Cc1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-603S c1cc(cc(c1)Cl)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-604S c1ccc(c(c1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl)Cl 5K-605S Cc1cccc(c1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-606S CCCCSCc1nc2c(cc(cc2Cl)Cl)c(=O)n1c3c(cccc3C)C 5K-607S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccccc3Cl 5K-610S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3cccc(c3)Cl 5K-611S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccccc3C(=O)OC 5K-612S Cc1cccc(c1n2c(nc3c(c2=O)cc(cc3Cl)Cl)CS(=O)(=O)c4cccc(c4)C(F)(F)F)C 5K-613S Cc1ccccc1NC(=O)c2cc(ccc2N)Cl 5K-616S Cc1cccc(c1n2c(nc3c(c2=O)cc(cc3Cl)Cl)CSc4ccc(cc4)F)C 5K-617S Cc1cccc(c1n2c(nc3c(c2=O)cc(cc3Cl)Cl)CSc4ccc(cc4)OC)C 5K-618S c1cc(c(c(c1)Cl)Cl)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-622S c1cc(cc(c1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl)C(F)(F)F 5K-623S Cc1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccccc3Cl 5K-624S c1ccc(c(c1)c2csc(n2)NC(=O)CSc3ccc(cc3)Cl)Cl 5K-625S c1ccc(c(c1)c2csc(n2)NC(=O)CSc3c(cccc3Cl)Cl)Cl 5K-626S c1ccc(c(c1)c2csc(n2)NC(=O)CSc3ccc(cc3)Br)Cl 5K-627S c1cc(ccc1c2csc(n2)NC(=O)CSc3ccc(cc3)Br)F 5K-628S c1cc(ccc1c2csc(n2)NC(=O)CSc3ccc(cc3)Cl)F 5K-629S Cc1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)F 5K-630S c1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)F 5K-631S c1ccc(cc1)c2csc(n2)NC(=O)CSc3ccc(cc3)Cl 5K-632S Cc1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccccc3 5K-633S c1ccc2c(c1)c(=O)n(c(n2)CCl)c3cccc(c3)C(F)(F)F 5K-634S c1ccc(cc1)n2c(nc3ccccc3c2=O)CCl 5K-635S Cc1cc(ccc1n2c(nc3ccccc3c2=O)CCl)Cl 5K-636S Cc1ccc(c(c1)SCc2nc3ccccc3c(=O)n2c4ccccc4)C 5K-638S c1ccc(cc1)n2c(nc3ccccc3c2=O)CSc4cccc(c4)Cl 5K-639S c1ccc(cc1)n2c(nc3ccccc3c2=O)CSc4cccc(c4Cl)Cl 5K-640S Cc1cc(cc(c1)SCc2nc3ccccc3c(=O)n2c4cccc(c4)C(F)(F)F)C 5K-641S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Oc3ccccc3 5K-642S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Oc3ccc(cc3)Cl 5K-643S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Oc3cccc(c3)C(F)(F)F 5K-644S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Oc3ccccc3C(=O)OC 5K-645S c1ccc(cc1)c2csc(n2)NC(=O)CSc3ccccc3 5K-646S c1ccc(cc1)c2csc(n2)NC(=O)CSc3ccc(cc3)F 5K-647S Cc1ccccc1SCC(=O)Nc2nc(cs2)c3ccccc3 5K-648S Cc1cccc(c1)SCC(=O)Nc2nc(cs2)c3ccccc3 5K-649S c1ccc(cc1)c2csc(n2)NC(=O)CSc3cccc(c3)Cl 5K-650S c1cc(c(cc1Cl)Cl)c2csc(n2)N 5K-651S c1cc(c(cc1Cl)Cl)c2csc(n2)NC(=O)CCl 5K-652S c1ccc2c(c1)c(=O)n(c(n2)CSc3cc(ccc3Cl)Cl)c4cccc(c4)C(F)(F)F 5K-653S c1ccc2c(c1)c(=O)n(c(n2)CSc3ccccc3Cl)c4cccc(c4)C(F)(F)F 5K-655S Cc1cccc(c1)SCc2nc3ccccc3c(=O)n2c4cccc(c4)C(F)(F)F 5K-656S c1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl 5K-657S c1cc(cc(c1)Cl)SCC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl 5K-658S Cc1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl 5K-659S c1cc(ccc1SCC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl)Cl 5K-660S Cc1ccc(c(c1)SCC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl)C 5K-661S Cc1ccccc1SCC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl 5K-662S c1cc(c(cc1Cl)Cl)c2csc(n2)NC(=O)CSc3cc(c(cc3Cl)Cl)Cl 5K-663S c1cc(cc(c1)SCC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl)C(F)(F)F 5K-664S c1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-665S Cc1ccccc1SCc2nc3ccccc3c(=O)n2c4cccc(c4)C(F)(F)F 5K-668S Cc1cc(ccc1n2c(nc3ccccc3c2=O)CSc4c(cccc4Cl)Cl)Cl 5K-670S c1cc(ccc1c2csc(n2)NC(=O)CSc3cc(ccc3Cl)Cl)Cl 5K-671S COC(=O)c1ccccc1SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-672S Cc1ccccc1SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-673S c1ccc(c(c1)S(=O)CC(=O)Nc2nc(cs2)c3ccc(cc3)Cl)Cl 5K-674S Cc1cccc(c1)S(=O)(=O)CC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 5K-675S CCOC(=O)c1c(nc(nn1)c2cccc(c2)C(F)(F)F)Oc3ccc(cc3)OC 5K-676S CC1(C2NC(=S)N(N2C(=S)N1)c3ccc(cc3)OC)c4ccccc4 5K-902 Cc1cc(cc(c1)n2c(=O)[nH]c(=O)c(n2)C(=O)C)C 5K-904 CCOC(=O)NC(=O)/C(=N\Nc1cccc(c1)OC)/C#N 5K-905 COc1cccc(c1)n2c(=O)[nH]c(=O)c(n2)C#N 5K-906 CC1(C2NC(=S)N(N2C(=S)N1)c3ccccc3)c4ccc(cc4)[N+](=O)[O-] 5K-911 CCOC(=O)NC(=O)/C(=N/Nc1cccc(c1)C(F)(F)F)/C#N 5K-914 c1cc(cc(c1)n2c(=O)[nH]c(=O)c(n2)C#N)C(F)(F)F 5K-915 CCOC(=O)NC(=O)/C(=N\Nc1cccc(c1)Cl)/C#N 5K-916 c1cc(cc(c1)Cl)n2c(=O)[nH]c(=O)c(n2)C#N 5K-917 CCOC(=O)NC(=O)/C(=N/Nc1ccc(cc1)F)/C#N 5K-919 c1cc(ccc1n2c(=O)[nH]c(=O)c(n2)C#N)F 5K-921 c1cc(ccc1Cn2c(=O)c(nn(c2=O)c3ccc(cc3)F)C#N)[N+](=O)[O-] 5K-922 Cn1c(=O)c(nn(c1=O)c2ccc(cc2)F)C#N 5K-923 c1ccc(cc1)NC(=S)/C(=C(\N)/N2CCN(CC2)c3ccccc3)/C#N 5K-925 c1ccc(cc1)NC(=S)/C(=C(\N)/N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)/C#N 5K-926 COc1cc2c(cc1OC)nc(sc2=N)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 5K-927 CC1(C2NC(=S)N(N2C(=S)N1)c3ccccc3)c4ccc(cc4)Cl 5K-932 CC1(C2NC(=S)N(N2C(=S)N1)c3ccc(cc3)Cl)c4ccc(cc4)Cl 5K-933 CC1(C2NC(=S)N(N2C(=S)N1)c3ccccc3)c4ccc(c(c4)Cl)Cl 5K-935 CCCSCC(=O)Nc1ncc2c(n1)-c3ccccc3CC2 5K-937 CC(C)SCC(=O)Nc1ncc2c(n1)-c3ccccc3CC2 5K-938 COc1cc(c(cc1OC)NC(=S)/C(=C(\N)/N2CCN(CC2)c3cccc(n3)Cl)/C#N)C#N 5K-939 c1ccc(cc1)C(=O)c2c(c(c(s2)Nc3ccccc3)C#N)N 5K-940 c1ccc(cc1)Nc2c(c(c(s2)C(=O)c3ccc(c(c3)Cl)Cl)N)C#N 5K-941 COc1cc(c(cc1OC)Nc2c(c(c(s2)C(=O)c3ccc(cc3)Cl)N)C#N)C#N 5K-942 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)CSc4ccc(cc4)Cl 5K-943 CCOC(=O)/C(=N/Nc1c(cccc1F)F)/C#N 5K-945 CN(C)/C=C/C(=O)c1ccc(cc1)Oc2cc(cnc2C#N)C(F)(F)F 5L-001 CO/N=C/C(=N\Nc1ccc(cc1)F)/C#N 5L-002 c1cc(ccc1C(=O)c2c(cc(cn2)C(F)(F)F)N3CCCC3)Cl 5L-003 C1CC(=O)NC1SCC(=O)O 5L-004 Cc1ccc(cc1)CO/N=C/C([N+](=O)[O-])S(=O)(=O)c2ccccc2 5L-006 C#CCSc1nccc(n1)/C=C/c2ccc(cc2)Cl 5L-007 CO/N=C\C(=N/Nc1ccc(cc1)Oc2ccccc2)\C#N 5L-008 COc1ccc(cc1)N/N=C(\C=N\OC)/C#N 5L-009 c1ccc(cc1)n2c(c(cn2)C#N)C(F)(F)F 5L-010 c1cc(ccc1C(=O)c2c(cc(cn2)C(F)(F)F)Oc3ccc(cc3)O)Cl 5L-011 c1cc(c(cc1Cl)Cl)/C=C/c2ccnc(n2)Sc3c(cc(cn3)C(F)(F)F)Cl 5L-012 COc1ccc(cc1)n2c(c(cn2)C#N)C(F)(F)F 5L-013 c1c(cc(cc1Cl)Cl)N/C=C/C#N 5L-014 C1CC(=O)N2C1SCC2=O 5L-015 c1cc(ccc1C(=O)c2c(cc(cn2)C(F)(F)F)N3CCCCCC3)Cl 5L-017 c1cc(ccc1C#N)N/C=C/C#N 5L-018 c1cc(cc(c1)Cl)n2c(c(cn2)C#N)C(F)(F)F 5L-019 c1cc(ccc1C(=O)c2c(cc(cn2)C(F)(F)F)N3CCOCC3)Cl 5L-020 Cc1ccc(cc1)S(=O)(=O)c2cc(cnc2C(=O)c3ccc(cc3)Cl)C(F)(F)F 5L-023 c1cc(c(cc1Cl)Cl)CO/N=C/CC#N 5L-024 CC(=O)c1ccc(cc1)Oc2cc(cnc2C(=O)N)C(F)(F)F 5L-025 CCOC(=O)C(=O)/C(=C/Nc1ccc(cc1)C#N)/C#N 5L-026 CCOC(=O)C1=C(NC(=O)CC1c2c(cccc2Cl)F)C 5L-027 CCOC(=O)c1c(cnn1c2ccc(cc2)C)C#N 5L-028 c1cc(oc1)/C=C(\C#N)/c2nnc(s2)N 5L-030 c1ccc(c(c1)/C=C(\C#N)/c2nnc(s2)N)F 5L-031 CCOC(=O)c1c(cnn1c2ccc(cc2)F)C#N 5L-032 CCOC(=O)C1=C(NC(=O)CC1c2cccc(c2)Br)C 5L-038 CN(C)/C=C/C(=O)/C=C/c1cccc(c1)C(F)(F)F 5L-039 COc1ccc(cc1)N2CCN(CC2)Cc3ccc(nc3)Cl 5L-040 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2)Cl)C 5L-041 c1cc(ccc1N2CCN(CC2)Cc3ccc(nc3)Cl)F 5L-042 c1cnc(nc1)N2CCN(CC2)Cc3ccc(nc3)Cl 5L-043 C[NH2+]C.c1c(c([nH]n1)C(=O)[O-])C#N 5L-044 c1c(cc(cc1Cl)Cl)Oc2cc(cnc2C#N)C(F)(F)F 5L-045 Cc1cc(ccc1Oc2cc(cnc2C#N)C(F)(F)F)Cl 5L-046 c1cc(ccc1CO/N=C/CC#N)F 5L-047 c1cc(ncc1CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 5L-048 c1ccnc(c1)SCc2ccc(nc2)Cl 5L-049 c1cc(ccc1/C(=N\O)/c2c(cc(cn2)C(F)(F)F)Cl)Cl 5L-050 CCOC(=O)c1c(cn[nH]1)C#N 5L-051 c1cc(sc1)C(=N)N.Cl 5L-0512 c1ccc(cc1)S(=O)(=O)c2cc(cnc2C(=O)c3ccc(cc3)Cl)C(F)(F)F 5L-052 CCOC(=O)c1c(cnn1c2ccc(cc2)Cl)C#N 5L-054 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2Cl)Cl)C 5L-055 CCOC(=O)C1=C(NC(=O)CC1c2ccccc2F)C 5L-056 c1cc(ccc1C(F)(F)F)N/C=C/2\C(=O)N3C(S2)CCC3=O 5L-059 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2)[N+](=O)[O-])C 5L-060 c1ccc(cc1)S(=O)(=O)Cc2ccc(nc2)Cl 5L-061 CC(C)(C)C1=C(C(CC(=O)N1)c2c(cccc2Cl)F)C#N 5L-062 CCOC(=O)C(=O)/C(=C/Nc1cc(cc(c1)C)C)/C#N 5L-063 CN(C)/C=C(/c1ccc(nc1)Cl)\S(=O)(=O)c2ccccc2 5L-064 CCOC(=O)C1=C(NC(=O)CC1c2cccc(c2)Br)C(F)(F)F 5L-065 C/C(=C/N(C)C)/[N+](=O)[O-] 5L-066 COc1ccc(cc1)N/C=C(\c2ccc(nc2)Cl)/S(=O)(=O)c3ccccc3 5L-067 CO/N=C/C(c1ccc(nc1)Cl)S(=O)(=O)c2ccccc2 5L-068 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2)Cl)C(F)(F)F 5L-069 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2Cl)Cl)C(F)(F)F 5L-070 CCOC(=O)C1=C(NC(=O)CC1c2ccccc2F)C(F)(F)F 5L-071 c1cc(ncc1CSc2c(cc(cn2)C(F)(F)F)Cl)Cl 5L-072 c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Cl)/c3ccc(nc3)Cl 5L-074 Cc1ccc(cc1C)N/C=C(/c2ccc(nc2)Cl)\S(=O)(=O)c3ccccc3 5L-075 c1ccc(cc1)S(=O)(=O)C(/C=N/OCc2ccc(cc2Cl)F)c3ccc(nc3)Cl 5L-076 c1ccc(cc1)S(=O)(=O)C(/C=N/OCc2cccc(c2Cl)Cl)c3ccc(nc3)Cl 5L-077 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2)[N+](=O)[O-])C(F)(F)F 5L-078 CO/N=C/C(=C\Nc1ccc(cc1)OC(F)(F)F)/[N+](=O)[O-] 5L-079 CCOC(=O)C(=O)/C(=C/Nc1ccc(cc1)F)/C#N 5L-080 CO/N=C/C(=C\Nc1ccc(cc1)C#N)/[N+](=O)[O-] 5L-081 c1ccc(cc1)Oc2ccc(cc2)N/C=C/3\C(=O)N4C(S3)CCC4=O 5L-082 CCOC(=O)C(=O)/C(=C/Nc1ccccc1C(=O)O)/C#N 5L-083 CC(C)(C)C1=C(C(CC(=O)N1)c2ccc(cc2)Cl)C#N 5L-084 c1cc(c(c(c1)Cl)C2CC(=O)NC3=C2C(=O)OC3)F 5L-085 c1cc(cc(c1)Br)C2CC(=O)NC3=C2C(=O)OC3 5L-086 CN(C)/C=C(/c1c(c(no1)c2ccccc2)C(=O)OC)\C(=O)C(F)(F)F 5L-087 c1ccc(cc1)COc2cc(c(cc2Cl)Cl)N 5L-301S Cc1nc(cc(n1)Sc2ccc(cc2)Cl)CS(=O)c3ccc(cc3)Cl 5L-302S CCOC(=O)COc1cc(c(cc1Cl)Cl)N 5L-303S Cc1nc(cc(n1)Oc2ccc(cc2)OC)CS(=O)c3ccc(cc3)Cl 5L-304S COc1ccc(cc1)NC(=O)c2nc(on2)c3ccccc3 5L-305S Cc1nc(cc(n1)N2CC(OC(C2)C)C)CSc3ccc(cc3)Cl 5L-306S Cc1nc(cc(n1)NCc2ccccc2)CSc3ccc(cc3)Cl 5L-307S Cc1nc(cc(n1)NCc2ccccc2Cl)CSc3ccc(cc3)Cl 5L-308S Cc1nc(cc(n1)NCc2ccc(cc2Cl)Cl)CS(=O)c3ccc(cc3)Cl 5L-309S c1c(c(cc(c1O)Cl)Cl)N 5L-310S Cc1nc(cc(n1)NC)CS(=O)c2ccc(cc2)Cl 5L-311S Cc1nc(cc(n1)SCc2ccc(cc2)Cl)CS(=O)c3ccc(cc3)Cl 5L-312S Cc1nc(cc(n1)Oc2ccc(cc2Cl)Cl)CS(=O)c3ccc(cc3)Cl 5L-313S Cc1nc(cc(n1)Sc2ccc(cc2)C(C)(C)C)CS(=O)c3ccc(cc3)Cl 5L-314S Cc1nc(cc(n1)OCc2ccc(c(c2)Cl)Cl)CSc3ccc(cc3)Cl 5L-315S Cc1nc(cc(n1)OCc2ccc(cc2Cl)Cl)CSc3ccc(cc3)Cl 5L-316S Cc1nc(cc(n1)OCc2ccc(cc2)Cl)CSc3ccc(cc3)Cl 5L-317S Cc1nc(cc(n1)OCc2cccc(c2)Cl)CSc3ccc(cc3)Cl 5L-318S COC(=O)c1nc(on1)c2ccc(cc2)F 5L-319S Cc1nc(cc(n1)OCc2ccc(cc2)F)CS(=O)(=O)c3ccc(cc3)Cl 5L-322S Cc1nc(cc(n1)OCc2ccccc2Cl)CS(=O)(=O)c3ccc(cc3)Cl 5L-323S Cc1nc(cc(n1)Sc2ccc(cc2)Cl)CS(=O)(=O)c3ccc(cc3)Cl 5L-324S Cc1nc(cc(n1)Sc2ccc(cc2)Cl)CS(=O)(=O)c3ccccc3 5L-325S CNC(=O)c1nc(on1)c2ccccc2 5L-327S Cc1ccc(cc1)Sc2cc(nc(n2)C)CS(=O)(=O)c3ccccc3 5L-328S Cc1nc(cc(n1)Sc2ccc(cc2)Br)CS(=O)(=O)c3ccccc3 5L-329S Cc1nc(cc(n1)N2CCN(CC2)c3ccccc3F)CS(=O)(=O)c4ccccc4 5L-330S c1cc(ccc1c2nc(no2)C(=O)O)F 5L-331S Cc1nc(cc(n1)Sc2ccccc2Cl)CS(=O)(=O)c3ccccc3 5L-332S Cc1nc(cc(n1)Sc2ccc(cc2Cl)Cl)CS(=O)(=O)c3ccccc3 5L-333S Cc1nc(cc(n1)Sc2ccc(cc2)OC)CS(=O)(=O)c3ccccc3 5L-334S Cc1nc(cc(n1)OC)CS(=O)(=O)c2ccc(cc2)Cl 5L-335S Cc1ccc(cc1)NC(=O)c2nc(on2)c3ccccc3 5L-336S c1ccc(cc1)c2nc(no2)C(=O)Nc3ccc(cc3)Oc4ccccc4 5L-338S Cc1nc(cc(n1)Sc2ccccc2Cl)CS(=O)(=O)c3ccc(cc3)Cl 5L-339S Cc1nc(cc(n1)Sc2cccc(c2)Cl)CS(=O)(=O)c3ccc(cc3)Cl 5L-343S Cc1nc(cc(n1)NCC=C)CS(=O)(=O)c2ccc(cc2)Cl 5L-344S Cc1nc(cc(n1)Oc2ccc(cc2Cl)Cl)CS(=O)(=O)c3ccc(cc3)Cl 5L-345S Cc1nc(cc(n1)Sc2ccc(cc2)C(C)(C)C)CS(=O)(=O)c3ccc(cc3)Cl 5L-346S Cc1nc(cc(n1)N2CCOCC2)CS(=O)(=O)c3ccc(cc3)Cl 5L-347S c1cc(ncc1CO)Cl 5L-348S c1cc(ncc1C=O)Cl 5L-349S Cc1ccc(cc1)Sc2ccc(cn2)C=O 5L-350S Cc1ccc(cc1)Sc2ccc(cn2)/C=N/O 5L-351S Cc1ccc(cc1)CO/N=C/c2ccc(nc2)Sc3ccc(cc3)C 5L-352S Cc1ccc(cc1)Sc2ccc(cn2)/C=N/OCc3ccc(cc3Cl)Cl 5L-353S Cc1ccc(cc1)Sc2ccc(cn2)/C=N/OC(=O)c3cccc(c3)OC 5L-354S Cc1ccc(cc1)Oc2ccc(cn2)C=O 5L-355S c1cc(ccc1Sc2ccc(cn2)C=O)Cl 5L-356S Cc1ccc(cc1)Oc2ccc(cn2)/C=N/OC 5L-357S c1cc(c(cc1C=O)[N+](=O)[O-])Oc2ccc(cc2F)F 5L-501S c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)c3ccc(c(c3)Cl)Cl 5L-502S c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3cc(cc(c3)Cl)Cl 5L-503S Cc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)c3ccc(c(c3)Cl)Cl 5L-504S Cc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3cc(cc(c3)Cl)Cl 5L-505S COCc1cc(nc(n1)c2ccccc2)Sc3ccc(cc3)Cl 5L-507S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)CSCc4ccc(cc4)Cl 5L-508S c1ccc(cc1)c2nc(cc(n2)Sc3c(cccc3Cl)Cl)CSCc4ccc(cc4)Cl 5L-509S c1ccc(cc1)c2nc(cc(n2)Sc3cccc(c3)Cl)CSCc4ccc(cc4)Cl 5L-510S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3Cl)Cl)CSCc4ccc(cc4)Cl 5L-511S Cc1cc([nH]c(=O)c1)C 5L-514S COc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)CSCc4ccc(cc4)Cl 5L-516S COCc1cc(nc(n1)c2ccccc2)SCc3cccc(c3)C(F)(F)F 5L-517S c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)c3ccc(cc3)[N+](=O)[O-] 5L-518S c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3ccc(cc3)Cl 5L-519S c1cc(ccc1C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl)[N+](=O)[O-] 5L-520S c1cc(cc(c1)NC(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl)C(F)(F)F 5L-521S Cc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)c3ccc(cc3)Cl 5L-522S c1cc(c(cc1CO)[N+](=O)[O-])Oc2ccc(cc2F)F 5L-523S Cc1c(snn1)NC(=O)OCc2ccc(cc2)C(C)(C)C 5L-526S Cc1c(snn1)NC(=O)OCc2ccc(cc2)C(F)(F)F 5L-527S Cc1c(snn1)NC(=O)OCC(C)(C)C 5L-528S Cc1c(snn1)NC(=O)OC 5L-529S c1ccnc(c1)c2nc(cc(n2)Sc3ccc(cc3Cl)Cl)CSCc4ccc(cc4)Cl 5L-531S c1ccnc(c1)c2nc(cc(n2)Sc3ccc(cc3)Br)CSCc4ccc(cc4)Cl 5L-532S c1ccnc(c1)c2nc(cc(n2)Sc3ccc(cc3)Cl)CSCc4ccc(cc4)Cl 5L-533S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccn3)CSCc4ccc(cc4)Cl 5L-534S c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)c3ccc(cc3)Cl 5L-535S c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3cccc(c3)Cl 5L-536S c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])COC(=O)Nc3cccc(c3)C(F)(F)F 5L-537S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3)Cl)CSCc4ccc(cc4)Cl 5L-538S c1cc(cc(c1)Cl)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3F)F 5L-539S c1cc(c(cc1COC(=O)c2ccc(c(c2)Cl)Cl)[N+](=O)[O-])Oc3ccc(cc3F)F 5L-540S c1cc(ccc1NC(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3F)F)Cl 5L-541S c1cc(cc(c1)NC(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3F)F)C(F)(F)F 5L-542S Cc1ccc(cc1)Sc2nc(cc(n2)OC)OC 5L-544S COc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(cc2)Cl 5L-545S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3)F)CSCc4ccc(cc4)Cl 5L-546S COc1ccc(cc1)Sc2cc(nc(n2)c3ccccn3)CSCc4ccc(cc4)Cl 5L-547S c1ccnc(c1)c2nc(cc(n2)Sc3ccc(cc3)F)CSCc4ccc(cc4)Cl 5L-548S c1ccnc(c1)c2nc(cc(n2)Sc3cccc(c3)Cl)CSCc4ccc(cc4)Cl 5L-549S c1ccnc(c1)c2nc(cc(n2)Sc3c(cccc3Cl)Cl)CSCc4ccc(cc4)Cl 5L-550S COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccc(cc3)Cl 5L-551S CS(=O)c1ccccc1C(=O)O 5L-554S Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2Cl)Cl)OC 5L-556S COc1cc(c(cc1Cl)Cl)NS(=O)(=O)c2ccc(cc2)Cl 5L-557S COc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2Cl)Cl)OCc3ccccc3 5L-558S COc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(cc2)[N+](=O)[O-] 5L-559S COc1cc(c(cc1Cl)Cl)NC(=O)c2cccc(c2)C(F)(F)F 5L-560S COc1cc(c(cc1Cl)Cl)NC(=O)c2c(cccc2F)F 5L-561S COc1ccc(cc1)C(=O)Nc2cc(c(cc2Cl)Cl)OC 5L-562S CCOC(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)c2ccc(cc2)C 5L-564S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2ccccc2 5L-565S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(c(c2)Cl)Cl 5L-566S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2ccccc2Cl 5L-568S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2cccc(c2)OC 5L-569S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2cc(c(cc2Cl)Cl)OC 5L-571S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3ccc(cc3)Cl 5L-573S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3cccc(c3)C(F)(F)F 5L-574S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3ccc(cc3)[N+](=O)[O-] 5L-575S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3c(cccc3F)F 5L-576S COc1ccc(cc1)C(=O)Nc2cc(c(cc2Cl)Cl)OCc3ccccc3 5L-577S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccccc2)c3cc(c(cc3Cl)Cl)OC 5L-578S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(cc2)Cl)c3cc(c(cc3Cl)Cl)OC 5L-579S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(c(c2)Cl)Cl)c3cc(c(cc3Cl)Cl)OC 5L-580S c1ccnc(c1)c2nc(cc(n2)SCc3ccc(cc3Cl)Cl)CSCc4ccc(cc4)Cl 5L-581S COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccc(cc3)[N+](=O)[O-] 5L-582S COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3cccc(c3)C(F)(F)F 5L-583S COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3c(cccc3F)F 5L-584S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2ccccc2 5L-585S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(c(c2)Cl)Cl 5L-586S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2ccccc2Cl 5L-588S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2cccc(c2)OC 5L-589S CCOC(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)c2ccc(cc2)Cl 5L-592S Cn1c(c(c(n1)C(F)(F)F)NC(=O)OCC=C)Oc2cccc(c2)C(F)(F)F 5L-594S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(cc2)Cl 5L-595S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(cc2)[N+](=O)[O-] 5L-596S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)c2cccc(c2)C(F)(F)F 5L-597S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(cc2)OC 5L-599S COc1ccc(cc1)c2nnnn2c3cc(c(cc3Cl)Cl)OC 5L-600S COc1cc(c(cc1Cl)Cl)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)Cl 5L-601S CS(=O)(=O)c1ccccc1C(=O)O 5L-603S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 5L-604S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl 5L-605S CC(C)SCc1cc(nc(n1)c2ccccc2)N3CCCC3 5L-607S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccccc3 5L-610S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccc(c(c3)Cl)Cl 5L-611S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccccc3Cl 5L-612S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)c3cccc(c3)OC 5L-613S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3c(nnn3)c4ccc(cc4)Cl 5L-614S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3c(nnn3)c4cccc(c4)C(F)(F)F 5L-615S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3c(nnn3)c4ccc(cc4)[N+](=O)[O-] 5L-616S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3c(nnn3)c4c(cccc4F)F 5L-617S COc1ccc(cc1)c2nnnn2c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-618S CC(C)SCc1cc(nc(n1)c2ccccc2)N3CCN(CC3)c4cccc(c4)Cl 5L-620S Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2Cl)Cl)OCc3ccccc3 5L-621S COc1cc(c(cc1Cl)Cl)NS(=O)(=O)c2ccc(cc2)F 5L-622S CCOC(=O)CN(c1cc(c(cc1Cl)Cl)OCc2ccccc2)S(=O)(=O)c3ccc(cc3)C 5L-623S CCOC(=O)CN(c1cc(c(cc1Cl)Cl)OCc2ccccc2)S(=O)(=O)c3ccc(cc3)OC 5L-624S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cccc(c2Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl 5L-625S CCOC(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)c2ccc(cc2)F 5L-626S CNC(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)c2ccc(cc2)Cl 5L-627S CN(C)C(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)c2ccc(cc2)Cl 5L-628S COCCOc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccccc3 5L-629S COCCOc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccc(c(c3)Cl)Cl 5L-630S COCCOc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccccc3Cl 5L-632S COCCOc1cc(c(cc1Cl)Cl)n2c(nnn2)c3cccc(c3)OC 5L-633S CCOC(=O)COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccc(cc3)Cl 5L-634S CCOC(=O)COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccc(cc3)[N+](=O)[O-] 5L-635S CCOC(=O)COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3cccc(c3)C(F)(F)F 5L-636S CCOC(=O)COc1cc(c(cc1Cl)Cl)n2c(nnn2)c3ccc(cc3)OC 5L-637S COc1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2cc(c(cc2Cl)Cl)OCc3ccccc3 5L-638S CC(C)Oc1cc(c(cc1Cl)Cl)NS(=O)(=O)c2ccc(cc2)Cl 5L-639S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)CSCc4ccc(cc4)Cl 5L-640S CC1CN(CC(O1)C)c2cc(nc(n2)c3ccccc3)CSCc4ccc(cc4)Cl 5L-641S c1ccc(cc1)c2nc(cc(n2)N3CCCC3)CSCc4ccc(cc4)Cl 5L-642S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2cc(c(cc2Cl)Cl)OCc3ccccc3 5L-643S CN(C)c1cc(nc(n1)c2ccccc2)CSCc3ccc(cc3)Cl 5L-647S c1ccc(cc1)c2nc(cc(n2)N3CCCCC3)CSCc4ccc(cc4)Cl 5L-648S COc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(cc2)Cl)c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-649S COc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(cc2)F)c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-650S COc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-651S CCOC(=O)CN(c1cc(c(cc1Cl)Cl)OC(C)C)S(=O)(=O)c2ccc(cc2)Cl 5L-653S CN(C)C(=O)CN(c1cc(c(cc1Cl)Cl)OCc2ccccc2)S(=O)(=O)c3ccc(cc3)OC 5L-654S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2F)F)S(=O)(=O)c3ccc(cc3)Cl 5L-655S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(cc2)Cl)c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-656S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(cc2)Br)c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-657S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(c(c2)Cl)Cl)c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-658S COc1cc(c(cc1Cl)Cl)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)F 5L-659S CNc1cc(nc(n1)c2ccccc2)CSCc3ccc(cc3)Cl 5L-664S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2cccc(c2)C(F)(F)F)c3cc(c(cc3Cl)Cl)OCc4ccccc4 5L-665S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)NC)c2cc(c(cc2Cl)Cl)OCc3ccccc3 5L-666S c1cc(ccc1F)S(=O)(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl 5L-900 C=CCN(CCNc1c(cc(cn1)C(F)(F)F)Cl)S(=O)(=O)c2ccc(cc2)F 5L-901 c1cc(ccc1N/N=C\2/CCCNC2=O)F 5L-902 c1cc2c(cc1F)c3c([nH]2)C(=O)NCC3 5L-904 CN(C)/C=C/c1ccc2c(c1)C(=O)c3ccccc3C2=O 5L-907 CO/N=C/Cc1ccc2c(c1)C(=O)c3ccccc3C2=O 5L-908 c1cc(ccc1F)S(=O)(=O)N(CCNc2c(cc(cn2)C(F)(F)F)Cl)CC3CC(=NO3)C(=O)NN 5L-911 c1ccc2c(c1)C(=O)c3ccc(cc3C2=O)C/C=N/OCc4ccc(cc4Cl)F 5L-912 c1ccc(c(c1)CO/N=C/Cc2ccc3c(c2)C(=O)c4ccccc4C3=O)Br 5L-913 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C/Cc2ccc3c(c2)C(=O)c4ccccc4C3=O 5L-914 c1cc(ccc1/C=N/NC(=O)C2=NOC(C2)CN(CCNc3c(cc(cn3)C(F)(F)F)Cl)S(=O)(=O)c4ccc(cc4)F)F 5L-915 c1cc(ccc1/C=N\NC(=O)C2=NOC(C2)CN(CCNc3c(cc(cn3)C(F)(F)F)Cl)S(=O)(=O)c4ccc(cc4)F)C(F)(F)F 5L-916 c1ccc2c(c1)C(=O)c3ccc(cc3C2=O)C/C=N/O 5L-917 Cc1ccc(cc1)NC(=O)C/C=N/OC 5L-918 c1ccc(cc1)NC(=O)NNC(=O)C2=NOC(C2)CN(CCNc3c(cc(cn3)C(F)(F)F)Cl)S(=O)(=O)c4ccc(cc4)F 5L-920 c1cc(cc(c1)[N+](=O)[O-])C(=O)C[N+]23CN4CN(C2)CN(C4)C3.[Br-] 5L-921 COc1ccc(cc1)c2c(cnc(n2)c3ccncc3)/N=N\c4ccc(cc4)F 5M-001 COc1ccc(cc1)c2c(cnc(n2)c3cccnc3)/N=N\c4ccc(cc4)F 5M-002 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)F)/C=N/O 5M-003 Cc1ncc(c(n1)c2ccccc2)/N=N\c3ccc(cc3)OC 5M-004 Cc1ncc(c(n1)c2ccc(cc2)Cl)/N=N\c3ccc(cc3)F 5M-005 Cc1ccc(cc1)c2c(cnc(n2)N)/N=N\c3cc(cc(c3)Cl)Cl 5M-006 Cc1ccc(cc1)c2c(cnc(n2)c3ccccc3)/N=N\c4cc(cc(c4)Cl)Cl 5M-007 c1ccc(cc1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 5M-008 c1cc(ccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])S(=O)(=O)Cl 5M-009 c1cc(c(cc1NC(=O)C2CC2)Cl)Oc3ccc(cn3)C(F)(F)F 5M-010 c1ccc(cc1)c2ncc(s2)c3ccn(n3)C(=O)C4CC4 5M-011 c1cc(ccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])S(=O)(=O)N3CCOCC3 5M-012 c1ccc(cc1)c2ncc(c(n2)c3ccc(cc3)Br)/N=N\c4ccc(cc4)C(F)(F)F 5M-013 c1cc(ccc1c2c(cnc(n2)c3ccncc3)/N=N\c4cc(cc(c4)Cl)Cl)Br 5M-014 Cc1ccc(cc1)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-016 c1ccc(cc1)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-017 c1cc(oc1)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-018 c1cc(c(cc1F)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)F 5M-019 c1cc(sc1)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-020 COc1ccc(cc1)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-021 c1cc(cc(c1)C(F)(F)F)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-022 c1ccc(cc1)/C=C/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-023 CN1CCN(CC1)S(=O)(=O)c2ccc(cc2)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 5M-024 c1cc2c(cnc(n2)N)c(c1)Cl 5M-025 c1ccnc(c1)CNS(=O)(=O)c2ccc(cc2)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 5M-026 c1cc(cc(c1)C(F)(F)F)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 5M-027 c1cc(cc(c1)Cl)/C=N/Nc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 5M-028 c1ccc(cc1)/C=C/c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 5M-029 c1cc(sc1)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 5M-030 c1ccc2c(c1)nc(c(n2)N/N=C/c3ccc(cc3)C(F)(F)F)C(F)(F)F 5M-031 c1cc(cc(c1)Cl)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 5M-032 c1ccc(c(c1)/C=N/Nc2c(nc3ccccc3n2)C(F)(F)F)F 5M-033 c1cc(c(cc1F)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F)F 5M-034 c1ccc2c(c1)nc(c(n2)N/N=C/c3c(cccc3Cl)F)C(F)(F)F 5M-035 Cc1ccsc1/C=N/Nc2c(nc3ccccc3n2)C(F)(F)F 5M-036 CC(=O)Nc1ncc2c(n1)cccc2Cl 5M-037 c1ccc(cc1)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 5M-038 c1ccc(c(c1)c2nnc3n2c4ccccc4nc3C(F)(F)F)F 5M-039 c1ccc2c(c1)nc(c(n2)N/N=C/c3ccc(cc3)Br)C(F)(F)F 5M-040 Cc1ccc(cc1)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 5M-041 c1ccc2c(c1)nc(c(n2)N/N=C/c3c(cccc3Cl)Cl)C(F)(F)F 5M-042 c1ccc(cc1)/C=C/C=N/Nc2c(nc3ccccc3n2)C(F)(F)F 5M-043 c1ccc2c(c1)nc(c3n2c(nn3)c4ccc(cc4)C(F)(F)F)C(F)(F)F 5M-044 c1ccc(cc1)C2COc3ccccc3N2C(=O)CCl 5M-301S CC(C)(C)c1nnc(o1)c2cc3c(nn(c3s2)C)C(F)(F)F 5M-304S CCOC(=O)Cn1c2ccccc2oc1=O 5M-307S CC(C)CC(=O)N1c2ccccc2OCC1c3ccccc3 5M-309S c1ccc(cc1)C2COc3ccccc3N2S(=O)(=O)c4ccc(cc4)Cl 5M-310S c1cc(ccc1c2cc(on2)CCl)Cl 5M-311S Cc1ccc(cc1)S(=O)(=O)N2c3ccccc3OCC2c4ccccc4 5M-315S COc1ccc(cc1)S(=O)(=O)N2c3ccccc3OCC2c4ccccc4 5M-316S CCOC(=O)c1cn(c2cc(ccc2c1=O)F)CC=C 5M-317S c1ccc(cc1)C2COc3ccccc3N2S(=O)(=O)c4ccc(cc4)F 5M-318S c1ccc(cc1)C2COc3ccccc3N2C(=O)C(Cl)Cl 5M-319S c1ccc(cc1)C2COc3ccccc3N2C(=O)CCCl 5M-320S CCCNC(=O)Cn1c2ccccc2oc1=O 5M-321S c1ccc(cc1)c2cc(on2)CCl 5M-323S c1ccc(cc1)C2COc3ccccc3N2C(=O)c4cccnc4Cl 5M-324S CC(C)(C)C1COc2ccccc2N1C(=O)c3cccc(c3)Cl 5M-325S c1ccc(cc1)c2cc(on2)CSc3ccc(cc3)Cl 5M-329S c1ccc(cc1)CSCc2cc(no2)c3ccccc3 5M-330S CC(C)(C)C1COc2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F 5M-331S CC(C)(C)C1COc2ccccc2N1C(=O)c3ccc(cc3)F 5M-332S Cc1ccccc1C(=O)N2c3ccccc3OCC2C(C)(C)C 5M-333S c1ccc(cc1)c2cc(on2)CN3C(=O)c4ccccc4C3=O 5M-334S c1ccc(cc1)c2cc(on2)CSc3ccccc3 5M-335S Cc1ccc(c(c1)[N+](=O)[O-])OCC(=O)C(C)(C)C 5M-337S Cc1ccc(c(c1)[N+](=O)[O-])OC/C(=N\O)/C(C)(C)C 5M-338S Cc1ccc2c(c1)NC(CO2)C(C)(C)C 5M-339S CCS(=O)(=O)Cc1cc(no1)c2ccccc2 5M-340S CC(=O)N(/C=C\1/C(=O)OC(=N1)c2ccccc2)C3=NCCS3 5M-341S c1ccc2c(c1)C(=O)N(C2=O)Cc3cc(no3)c4ccc(cc4)Cl 5M-344S c1ccc(cc1)SCc2cc(no2)c3ccc(cc3)Cl 5M-345S Cc1ccc(cc1)SCc2cc(no2)c3ccc(cc3)Cl 5M-346S Cc1ccc2c(c1)N(C(CO2)C(C)(C)C)S(=O)(=O)c3ccc(cc3)Cl 5M-347S Cc1ccc2c(c1)N(C(CO2)C(C)(C)C)S(=O)(=O)c3ccc(cc3)OC 5M-348S Cc1ccc(cc1)S(=O)(=O)N2c3cc(ccc3OCC2C(C)(C)C)C 5M-349S Cc1ccc2c(c1)N(C(CO2)C(C)(C)C)S(=O)(=O)c3ccc(cc3)F 5M-350S c1ccc(cc1)c2cc(on2)CS(=O)(=O)c3ccccc3 5M-351S c1ccc(cc1)S(=O)(=O)Cc2cc(no2)c3ccc(cc3)Cl 5M-352S Cc1ccc(cc1)S(=O)(=O)Cc2cc(no2)c3ccc(cc3)Cl 5M-353S CC(C)(C)/C(=N\OC(=O)NC1CCCCC1)/COc2ccccc2[N+](=O)[O-] 5M-354S CC(C)(C)/C(=N\OC(=O)Nc1cccc(c1)Cl)/COc2ccccc2[N+](=O)[O-] 5M-355S CCCNC(=O)O/N=C(/COc1ccccc1[N+](=O)[O-])\C(C)(C)C 5M-356S COc1ccc(cc1)c2cc(on2)CCl 5M-357S Cc1ccc(c(c1)[N+](=O)[O-])OC/C(=N/OC(=O)NC2CCCCC2)/C(C)(C)C 5M-358S Cc1ccc(c(c1)[N+](=O)[O-])OC/C(=N/OC(=O)Nc2cccc(c2)Cl)/C(C)(C)C 5M-359S c1cc(sc1)C(=O)Nc2ccc(oc2=O)c3ccc(cc3)Cl 5M-502S c1cc(sc1)C(=O)Nc2ccc(oc2=O)c3ccc(cc3)Br 5M-503S Cc1ccc(cc1)n2c(=O)c(c(cn2)N3CCOCC3)Cl 5M-512S Cn1c(cc(n1)OCC(CS(=O)(=O)c2ccc(cc2)Cl)O)C(F)(F)F 5M-516S Cc1ccc(cc1)n2c(=O)c(c(cn2)NC)Cl 5M-517S Cc1ccc(cc1)n2c(=O)c(c(cn2)N(C)C)Cl 5M-518S Cc1ccc(cc1)n2c(=O)c(c(cn2)NCC=C)Cl 5M-519S CC(C)Nc1cnn(c(=O)c1Br)c2ccc(cc2)F 5M-524S CN1CCN(CC1)c2cnn(c(=O)c2Br)c3ccc(cc3)F 5M-525S CN(Cc1ccccc1)c2cnn(c(=O)c2Br)c3ccc(cc3)F 5M-528S c1ccc(cc1)CNc2cnn(c(=O)c2Br)c3ccc(cc3)F 5M-529S Cc1c(cno1)C(=O)C 5M-531S CSc1nnc(n1c2ccccc2)CNC(=O)c3ccc(cc3)F 5M-532S CCOC(=O)CSc1nnc(n1c2ccccc2)CNC(=O)c3ccc(cc3)F 5M-533S C=CCSc1nnc(n1c2ccccc2)CNC(=O)c3ccc(cc3)F 5M-534S c1cc(ccc1n2c(=O)c(c(cn2)N3CCCC3)Cl)F 5M-536S c1cc(ccc1n2c(=O)c(c(cn2)N3CCCCC3)Cl)F 5M-537S CCCNc1cnn(c(=O)c1Cl)c2ccc(cc2)F 5M-538S C=CCNc1cnn(c(=O)c1Cl)c2ccc(cc2)F 5M-539S CCOC(=O)C(C)S(=O)(=O)c1ccc(cn1)C(F)(F)F 5M-544S CCOC(=O)C(C)S(=O)c1ccc(cn1)C(F)(F)F 5M-545S Cc1c(cno1)c2csc(n2)C 5M-547S Cc1c(cno1)c2csc(n2)c3ccccc3Cl 5M-548S Cc1c(cno1)c2csc(n2)c3ccccc3 5M-549S Cc1ccc2nc(cn2c1)c3cnoc3C 5M-550S Cc1ccc(cc1)CSc2nnc(n2c3ccccc3)CNC(=O)c4ccc(cc4)F 5M-552S CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)CNC(=O)c3ccc(cc3)Cl 5M-553S CCn1c(nnc1SCC=C)CNC(=O)c2ccc(cc2)Cl 5M-555S CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)CNC(=O)c3ccc(cc3)Cl 5M-556S CCOC(=O)CS(=O)(=O)c1ccc(cn1)C(F)(F)F 5M-558S CCOC(=O)CS(=O)c1ccc(cn1)C(F)(F)F 5M-559S c1cc(ncc1C(F)(F)F)S(=O)(=O)CC(=O)O 5M-560S Cc1c(cno1)/C(=N/OCc2ccc(cc2)F)/C 5M-563S CC(C(=O)O)S(=O)(=O)c1ccc(cn1)C(F)(F)F 5M-564S Cc1ccc(cc1)Sc2cnn(c(=O)c2Cl)c3ccc(c(c3)Cl)Cl 5M-570S c1ccc(cc1)Cn2c(cnc2S(=O)Cc3ccc(cc3)Cl)CO 5M-571S c1ccc(cc1)Cn2c(cnc2S(=O)(=O)Cc3ccc(cc3)Cl)CO 5M-572S CS(=O)(=O)c1ncc(n1Cc2ccccc2)CO 5M-573S Cn1c(cnc1S(=O)Cc2ccc(cc2)Cl)CO 5M-574S Cn1c(cnc1S(=O)(=O)Cc2ccc(cc2)Cl)CO 5M-575S Cc1cccc(c1)CS(=O)(=O)c2ncc(n2C)CO 5M-576S Cn1c(cnc1S(=O)(=O)Cc2ccc(cc2)[N+](=O)[O-])CO 5M-577S CCOC(=O)CS(=O)(=O)c1c(cc(cn1)Cl)Cl 5M-582S c1cc(ccc1C(=O)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)F 5M-586S Cc1ccc(cc1)n2c(=O)c(c(cn2)Cl)Oc3ccc(cc3)OC 5M-588S COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccc(c(c3)Cl)Cl)Cl 5M-590S Cc1ccc(cc1)n2c(=O)c(c(cn2)N3CCOCC3)Oc4ccc(cc4)OC 5M-591S COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccc(cc3)F)Cl 5M-593S COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccccc3)Cl 5M-594S Cc1cccc(c1C)n2c(=O)c(c(cn2)Cl)Oc3ccc(cc3)OC 5M-595S c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)CNC(=O)c2ccc(cc2Cl)Cl 5M-597S c1c(cnc(c1Cl)S(=O)(=O)CC(=O)O)Cl 5M-600S c1ccc(cc1)n2c(=O)c(c(cn2)Cl)Cl 5M-603S CNC(=O)c1c(cnn1c2ccccc2)Cl 5M-604S Cc1ccc(cc1)n2c(c(cn2)Cl)C(=O)NC 5M-605S CC1(Cc2c(c(c3ccccc3n2)N)C(=O)C1)C 5M-700 c1ccc(cc1)CNc2ccc3nnc(n3n2)C(F)(F)F 5M-701 Cc1cccc(c1N2CCN(CC2)c3ccc4nnc(n4n3)C(F)(F)F)C 5M-702 Cc1cc2c(cc1C)NC3=C(C(N2)c4ccc(cc4)N(C)C)C(=O)CC(C3)(C)C 5M-703 Cc1cc(c(c(c1)C)CSC(C)(C)CNC(=O)c2cccc(c2)[N+](=O)[O-])C 5M-706 Cc1cc(c(c(c1)C)CSC(C)(C)CNC(=O)CCCl)C 5M-707 Cc1cc(c(c(c1)C)CSC(C)(C)CNc2c(cccn2)[N+](=O)[O-])C 5M-709 Cc1cc(c(c(c1)C)CSC(C)(C)CNC(=O)c2cc(ccc2Cl)Cl)C 5M-710 Cc1cc(c(c(c1)C)CSC(C)(C)CNC(=O)c2ccc(cc2)OC)C 5M-711 CC1(CN(C1=O)C(Cc2ccccc2)C(=O)N/C=N/OCc3ccc(cc3)OC)C 5M-714 Cc1cc(nc(n1)O)/C=N/O 5M-715 CCOC(=O)CC(=O)c1cc2cc(ccc2oc1=O)Cl 5M-716 CC(C)(CN)SCc1cccc(c1)C(F)(F)F 5M-717 CC(=O)C(Cc1c(cccc1Cl)Cl)C(=O)C 5M-721 Cc1c(c(on1)C)Cc2c(cccc2Cl)Cl 5M-723 c1cc(nc(c1)F)NNC(=O)C(F)(F)F 5M-726 c1cc(c(c(c1)C#N)N2CCC(CC2)C(=O)N)C#N 5M-727 Cc1c(c(=O)ccn1c2nc[nH]n2)Cc3c(cccc3Cl)Cl 5M-728 Cc1cc(c(c(c1)C)CSC(C)(C)CN2C(=O)Cc3ccccc3C2=O)C 5M-730 c1cc(c(c(c1)C#N)N2CCC(CC2)C#N)C#N 5M-731 c1ccc\2c(c1)CCC/C2=N\O 5M-732 Cc1c(cno1)/C(=N/OCc2ccc(cc2Cl)Cl)/C 5M-860S c1cc(cc(c1)F)CON/C=N/C(=S)Nc2ccc(cn2)I 5M-900 c1cc(cc(c1)OCCON/C=N/C(=S)Nc2ccc(cn2)I)C(F)(F)F 5M-901 Cn1c2c(c(=O)n(c1=O)C)CCC(=O)N2Cc3ccc(cc3)Br 5M-902 c1ccc2c(c1)c(c[nH]2)C3CC(=O)N(C3=O)c4cccc(c4)C(F)(F)F 5M-903 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)Nc3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl 5M-906 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)Nc3ccc(cc3)F 5M-907 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)Nc3ccc(cc3)OC(F)(F)F 5M-909 COc1ccc2c(c1)c(c[nH]2)C3CC(=O)N(C3=O)c4cccc(c4)C(F)(F)F 5M-910 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)CC(C2=O)c3c[nH]c4c3cccc4 5M-912 CC(=C1C=C(c2c1cccc2)C(C)(C)C3=CC(=C(C)C)c4c3cccc4)C 5M-913 c1ccc2c(c1)c(c[nH]2)C3CC(=O)N(C3=O)c4ccc(cc4Cl)Cl 5M-915 c1ccc(cc1)n2ccc(=O)c(n2)c3cc[nH]n3 5M-917 CC(=O)C(=NNc1ccc(cc1)Cl)C(=O)C 5M-918 c1ccc(cc1)n2ccc(=O)c(n2)c3ccn(n3)c4ccc(cc4)Cl 5M-919 Cc1ccc(cc1)n2ccc(n2)c3c(=O)ccn(n3)c4ccccc4 5M-920 c1ccc(cc1)n2ccc(=O)c(n2)c3ccn(n3)C4CCS(=O)(=O)C4 5M-921 CC(=O)C(=NNc1cccc(c1)C(F)(F)F)C(=O)C 5M-922 Cc1ccc(cc1)C(=O)n2ccc(n2)c3c(=O)ccn(n3)c4ccccc4 5M-923 c1ccc(cc1)n2ccc(=O)c(n2)c3ccn(n3)C(=O)c4ccc(cc4)F 5M-924 COc1cccc(c1)C(=O)n2ccc(n2)c3c(=O)ccn(n3)c4ccccc4 5M-925 c1cc(ccc1n2ccc(=O)c(n2)c3cc[nH]n3)Cl 5M-927 c1cc(cc(c1)n2ccc(=O)c(n2)c3ccn(n3)c4cccc(c4)[N+](=O)[O-])C(F)(F)F 5M-929 c1ccc(cc1)n2ccc(n2)c3c(=O)ccn(n3)c4cccc(c4)C(F)(F)F 5M-930 COc1ccc(cc1)n2ccc(n2)c3c(=O)ccn(n3)c4cccc(c4)C(F)(F)F 5M-931 c1cc(cc(c1)n2ccc(=O)c(n2)c3ccn(n3)c4cccc(c4)Cl)C(F)(F)F 5M-932 c1cc(cc(c1)[N+](=O)[O-])C(=O)n2ccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl 5M-933 c1cc(sc1)C(=O)n2ccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl 5M-934 c1ccc(cc1)NC(=O)n2ccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl 5M-935 c1ccc(c(c1)n2ccc(n2)c3c(=O)ccn(n3)c4cccc(c4)C(F)(F)F)F 5M-936 c1ccc(c(c1)C(=O)/C=C/c2ccco2)Cl 5M-937 c1cc(oc1)/C=C/C(=O)c2ccc(cc2)Cl 5M-938 c1cc(oc1)/C=C/C(=O)c2ccc(cc2Cl)Cl 5M-939 c1cc(oc1)/C=C/C(=O)c2ccc(c(c2)Cl)Cl 5M-940 c1ccnc(c1)C(=O)/C=C/c2ccco2 5M-941 c1cc(oc1)/C=C/C(=O)c2ccco2 5M-942 c1ccc2cc(ccc2c1)C(=O)/C=C/c3ccco3 5M-943 c1ccc(cc1)c2ccc(cc2)C(=O)/C=C/c3ccco3 5M-944 c1cc(ccc1n2ccc(=O)c(n2)c3ccn(n3)C(=O)c4ccc(c(c4)Cl)Cl)Cl 5M-945 c1ccc(c(c1)C(=O)n2ccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl)Cl 5M-946 c1ccc(cc1)C(=O)/C=C/c2cccs2 5M-948 c1cc(ccc1n2ccc(=O)c(n2)c3ccn(n3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 5M-949 c1ccc(cc1)/C=C/C(=O)n2ccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl 5M-950 c1c(c(cc2c1OCO2)Br)C=O 5M-952 c1cc(cnc1)C(=O)/C=C/c2ccco2 5M-953 c1ccc(cc1)C(=O)/C=C/c2ccoc2 5M-954 c1cc(ncc1I)NC(=O)N 5M-956 c1cc2c(cco2)cc1NC(=S)N 5N-001 Cc1c2ccc(nc2ccn1)Oc3ccc(cc3Cl)Cl 5N-002 COc1ccc(cc1)/C(=N\O)/C2CC2c3ccc(cc3)Cl 5N-005 CC(C)(C)C(C(=O)NC)NC(=O)c1cccc(c1)OC 5N-006 COc1ccc(cc1)/C(=N\OCc2ccc(cc2Cl)Cl)/C3CC3c4ccc(cc4)Cl 5N-007 COc1ccc(cc1)/C(=N\OCc2ccc(cc2)[N+](=O)[O-])/C3CC3c4ccc(cc4)Cl 5N-008 CN(C)c1ccc(cc1)C2CC2C(=O)c3ccc(cc3)Cl 5N-009 Cc1ccc(cc1)CO/N=C(\c2ccc(cc2)OC)/C3CC3c4ccc(cc4)Cl 5N-010 COc1ccc(cc1)/C(=N\OCc2ccc(cc2)Cl)/C3CC3c4ccc(cc4)Cl 5N-011 c1ccc(cc1)C(COC(=O)c2ccc(c(c2)Cl)Cl)N3CCS(=O)(=O)CC3 5N-012 Cc1ccc(cc1)C(=O)O/N=C(\c2ccc(cc2)OC)/C3CC3c4ccc(cc4)Cl 5N-013 COc1ccc(cc1)/C(=N\OC(=O)c2ccc(c(c2)Cl)Cl)/C3CC3c4ccc(cc4)Cl 5N-014 CC(C)(C)C(C(=O)OC)NC(=O)Nc1ccccc1Cl 5N-015 CC(C)(C)C(C(=O)OC)NC(=O)Nc1cccc(c1)C(F)(F)F 5N-016 C1CCC(CC1)CC(C(=O)O)N2CCS(=O)(=O)CC2 5N-017 c1ccc(cc1)CC(CO)NC(=O)Nc2ccc(cc2)Cl 5N-018 c1ccc(cc1)C(CO)NC(=O)Nc2ccc(cc2)Cl 5N-019 CC(C)(C)C(C(=O)NC)NC(=O)c1ccc(cc1F)F 5N-020 COc1ccc(cc1)/C(=N\OC(=O)c2ccc(cc2F)F)/C3CC3c4ccc(cc4)Cl 5N-021 c1ccc(cc1)CC(CO)NC(=O)NC2CCCCC2 5N-022 c1ccc(cc1)C(CO)NC(=O)NC2CCCCC2 5N-023 CC(C)(C)C(C(=O)NC)NC(=O)c1ccc(cc1)Cl 5N-024 CC(C)(C)C(C(=O)NC)NC(=S)NC(=O)c1ccc(cc1)F 5N-025 CC(C)(C)C(C(=O)NC)NS(=O)(=O)c1ccc(cc1)Br 5N-026 COc1ccc(cc1)NC(=O)NC(COC(=O)Nc2ccc(cc2)OC)c3ccccc3 5N-028 CC(C)(C)C(C(=O)NC)NC(=O)c1cccc(c1)C(F)(F)F 5N-029 Cc1c2ccc(nc2ccn1)Oc3ccc(cc3)C#N 5N-030 CCOC(=O)NC(=O)/C(=C/NC(Cc1ccccc1)CO)/C#N 5N-031 c1ccc(cc1)CC(CO)NC(=S)NC(=O)c2ccc(cc2)F 5N-032 c1ccc(cc1)C(COC(=O)Nc2ccccc2)NC(=O)Nc3ccccc3 5N-033 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(C(=O)NC)C(C)(C)C 5N-034 c1cc(ccc1c2c(c[nH]n2)C=O)F 5N-036 CCOC(=O)NC(=O)/C(=C/NC(CO)c1ccccc1)/C#N 5N-037 CC(C)(C)C(C(=O)O)N1CCS(=O)(=O)CC1 5N-038 c1cc(ccc1C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)OC(F)(F)F 5N-039 c1ccc(cc1)CC(COC(=O)Nc2ccc(c(c2)Cl)Cl)NC(=O)Nc3ccc(c(c3)Cl)Cl 5N-040 c1ccc(cc1)C(CO)NC(=S)NC(=O)c2ccc(cc2)F 5N-041 CC(C)(C)C(C(=O)NC)NC(=O)c1c(cccc1F)F 5N-043 C1c2c(c(c(nc2OC1CO)N)C#N)N 5N-044 c1ccc(cc1)CC2COC3(N2C(=O)Nc4ccc(cc4)Cl)CCN(CC3)c5c(cc(cn5)C(F)(F)F)Cl 5N-045 CCOC(=O)NC(=O)/C(=C\NC(C(=O)NC)C(C)(C)C)/C#N 5N-046 Cc1c2ccc(nc2ccn1)N3CCOCC3 5N-047 Cc1ccc(cc1)NC(=S)NC(Cc2ccccc2)CO 5N-048 Cc1ccc(cc1)NC(=O)N2C(COC23CCN(CC3)c4ccc(cc4)[N+](=O)[O-])c5ccccc5 5N-049 COc1ccc(c(c1)NC(=O)C(CC2CCCCC2)N3CCS(=O)(=O)CC3)OC 5N-050 Cc1ccc(cc1)NC(=O)N2C(COC23CCN(CC3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])c5ccccc5 5N-051 CC(C)(C)C(C(=O)OC)n1cccc1 5N-052 CC(C)(C)C(C(=O)O)n1cccc1 5N-053 c1cc(ccc1C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)C(F)(F)F 5N-054 COc1ccc(cc1)C(=O)N2C(COC23CCN(CC3)c4ccc(cc4)[N+](=O)[O-])c5ccccc5 5N-055 c1ccc(cc1)C2COc3c2c(c(c(n3)N)C#N)N 5N-056 COC(=O)C(CC1CCCCC1)n2cccc2 5N-057 c1ccc(cc1)C(CO)NC(=O)c2ccc(cc2)Cl 5N-058 c1ccc(cc1)CC(CO)NC(=O)c2ccc(c(c2)Cl)Cl 5N-059 c1ccc(cc1)C(CO)NC(=O)c2ccco2 5N-060 c1ccc(cc1)C2COC3(N2C(=O)c4ccc(cc4)F)CCN(CC3)c5c(cc(cc5[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 5N-061 C1c2c(c(c(nc2OC1CCl)N)C#N)N 5N-062 CCOc1ccc2c(c1)sc(n2)NC(=O)c3cccs3 5N-063 c1ccc(cc1)C(CO)NC(=O)C2CC2 5N-064 c1ccc(cc1)C(CCl)NC(=O)c2ccc(cc2)Cl 5N-065 CCOC(=O)c1ccc(cc1)N2CCCC2=O 5N-066 c1ccc2c(c1)CN(C2=O)C(CC3CCCCC3)C(=O)Nc4ccc(cc4)Oc5c(cc(cn5)C(F)(F)F)Cl 5N-067 Cc1ccc(cc1)NC(=O)NC(C(=O)NC)C(C)(C)C 5N-068 c1cc(ccc1n2cn[nH]c2=O)Br 5N-069 c1ccc(cc1)C(COC(=O)c2ccc(c(c2)Cl)Cl)NC(=O)CNC(=O)c3ccc(cc3)Cl 5N-070 c1ccc(cc1)n2cn[nH]c2=O 5N-071 Cc1cccc(c1)C(=O)OCC(Cc2ccccc2)NC(=O)Nc3ccc(cc3)Cl 5N-072 CC(C)c1ccc(cc1)n2cn[nH]c2=O 5N-076 c1ccn(c1)C(CC2CCCCC2)C(=O)N/N=C/c3ccc(cc3)[N+](=O)[O-] 5N-077 c1cc(cc(c1)n2cn[nH]c2=O)C(F)(F)F 5N-078 CC(C)(C)C(C(=O)NC)Nc1c(cccn1)[N+](=O)[O-] 5N-079 c1ccc(cc1)c2cc(n(n2)c3ccccc3)N 5N-080 COc1ccc(cc1)C2CC(=O)Nc3c2c(nn3c4ccccc4)c5ccccc5 5N-081 CC(C)(C)C(C(=O)NC)Nc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 5N-082 CCOC(=O)CNC(=S)NC(C(=O)NC)C(C)(C)C 5N-083 Cc1cc(nc2c1c(nn2c3ccccc3)c4ccccc4)C 5N-085 COc1cc(cc(c1OC)OC)NC(=O)C(CC2CCCCC2)N3Cc4ccccc4C3=O 5N-086 c1ccc2c(c1)CN(C2=O)C(CC3CCCCC3)C(=O)NNC(=O)c4ccc(cc4)Cl 5N-087 CC(C)(C)C(C(=O)OC)Nc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 5N-088 c1ccc(cc1)CC(COC(=O)c2cccc(c2)Cl)NC(=O)c3ccc(c(c3)Cl)Cl 5N-089 Cc1ccc(n1c2cccc(c2)C(F)(F)F)c3ccco3 5N-301S Cc1ccc(n1c2cc(cc(c2)Cl)Cl)c3ccco3 5N-302S c1cc(cc(c1)Cl)c2cc(c(c(n2)Sc3ccc(cc3)Br)C#N)C(F)(F)F 5N-303S c1ccc2cc(ccc2c1)Oc3c(c(cc(n3)c4cccc(c4)Cl)C(F)(F)F)C#N 5N-304S CCN(CC)c1c(c(cc(n1)c2ccc(cc2)Cl)C(F)(F)F)C#N 5N-305S C1CCc2c(c(nc(n2)S)O)C1 5N-306S Cc1ccc(cc1)CSc2nc3c(c(n2)O)CCCC3 5N-307S Cc1ccc(cc1)CSc2nc3c(c(n2)Cl)CCCC3 5N-308S COc1ccc(cc1)c2cc(on2)CNC(=O)CN3CCCC3 5N-309S CCN(CC)CC(=O)NCc1cc(no1)c2ccc(cc2)OC 5N-310S CN(Cc1ccccc1)CC(=O)NCc2cc(no2)c3ccc(cc3)OC 5N-311S COc1ccc(cc1)c2cc(on2)CNC(=O)CN3CCOCC3 5N-312S COc1ccc(cc1)c2cc(on2)CNC(=O)CN3CCCCC3 5N-313S CN1CCN(CC1)CC(=O)NCc2cc(no2)c3ccc(cc3)OC 5N-314S c1ccc(cc1)Sc2c(c(cc(n2)c3ccc(cc3)Cl)C(F)(F)F)C#N 5N-315S Cc1ccc(cc1)Sc2c(c(cc(n2)c3ccc(cc3)Cl)C(F)(F)F)C#N 5N-316S c1ccc2cc(ccc2c1)Oc3c(c(cc(n3)c4ccc(cc4)Cl)C(F)(F)F)C#N 5N-317S c1cc(cc(c1)Sc2c(c(cc(n2)c3ccc(cc3)Cl)C(F)(F)F)C#N)C(F)(F)F 5N-318S c1cc(ccc1c2cc(c(c(n2)Oc3ccc(cc3Cl)Cl)C#N)C(F)(F)F)Cl 5N-319S Cc1ccc(cc1)Sc2c(c(cc(n2)c3ccccc3Cl)C(F)(F)F)C#N 5N-320S c1ccc(c(c1)c2cc(c(c(n2)N3CCOCC3)C#N)C(F)(F)F)Cl 5N-321S c1ccc2cc(ccc2c1)Oc3c(c(cc(n3)c4ccccc4Cl)C(F)(F)F)C#N 5N-322S COc1ccc(cc1)Oc2c(c(cc(n2)c3ccccc3Cl)C(F)(F)F)C#N 5N-323S c1ccc(c(c1)CSc2nc3c(c(n2)O)CCCC3)Cl 5N-327S c1ccc(cc1)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-328S Cc1cccc(c1)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-329S Cn1c2ccccc2c(c1Cl)C(=O)Nc3ccc(cc3)Cl 5N-330S Cc1ccc(cc1)Sc2c(c3ccccc3n2C)C(=O)Nc4ccc(cc4)Cl 5N-331S Cn1c2ccccc2c(c1Sc3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)Cl 5N-332S c1c(c(c(nc1C2CC2)Cl)C#N)C(F)(F)F 5N-333S c1ccc(c(c1)CSc2nc3c(c(n2)Cl)CCCC3)Cl 5N-334S Cc1ccc(cc1)CSc2nc3c(c(n2)N4CCOCC4)CCCC3 5N-335S Cn1c2ccccc2c(c1Sc3ccc(cc3Cl)Cl)C(=O)Nc4ccc(cc4)Cl 5N-336S Cn1c2ccccc2c(c1Sc3cccc(c3)OC)C(=O)Nc4ccc(cc4)Cl 5N-337S Cc1cccc(c1)Sc2c(c3ccccc3n2C)C(=O)Nc4ccc(cc4)Cl 5N-338S Cn1c2ccccc2c(c1SCc3ccccc3)C(=O)Nc4ccc(cc4)Cl 5N-339S Cc1ccc(cc1)CSc2nc3c(c(n2)N4CCCCC4)CCCC3 5N-340S Cc1ccc(cc1)CSc2nc3c(c(n2)NCC=C)CCCC3 5N-341S c1csc2c1C(CCS2(=O)=O)O 5N-343S c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-344S c1cc(ccc1C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3)Cl 5N-345S c1cc(ccc1C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3)F 5N-346S c1cc(sc1)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-347S c1cc(c(cc1C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3)Cl)Cl 5N-348S Cc1ccccc1C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-349S COc1cccc(c1)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-350S COc1ccc(cc1)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-351S Cc1ccc(cc1)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-352S c1cc(cc(c1)Cl)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-353S c1cc(c(cc1Cl)Cl)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3 5N-354S c1cc(c(c(c1)F)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3)F 5N-355S Cc1ccc(cc1)CSc2nc3c(c(n2)NC4CC4)CCCC3 5N-356S Cc1ccc(cc1)CSc2nc3c(c(n2)NC(C)C)CCCC3 5N-357S Cc1ccc(cc1)CSc2nc3c(c(n2)N4CCN(CC4)C)CCCC3 5N-358S Cc1ccc(cc1)CSc2nc3c(c(n2)NC)CCCC3 5N-359S Cc1ccc(cc1)CSc2nc3c(c(n2)N(C)C)CCCC3 5N-360S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)S(=O)(=O)Cc4ccc(cc4)Cl)CCCC3 5N-361S Cn1c2ccccc2c(c1Sc3ccc(cc3)Br)C(=O)Nc4ccc(cc4)Cl 5N-362S Cn1c2ccccc2c(c1Sc3ccc(cc3)F)C(=O)Nc4ccc(cc4)Cl 5N-363S Cn1c2ccccc2c(c1Sc3cccc(c3)Cl)C(=O)Nc4ccc(cc4)Cl 5N-364S Cn1c2ccccc2c(c1Sc3cccc(c3)C(F)(F)F)C(=O)Nc4ccc(cc4)Cl 5N-365S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)S(=O)(=O)C4CCCCC4)CCCC3 5N-366S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccc(cc4)C)CCCC3 5N-367S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccc(cc4)Cl)CCCC3 5N-368S c1c(c(c(nc1C2CC2)N3CCCC3)C#N)C(F)(F)F 5N-369S c1c(c(c(nc1C2CC2)N3CCOCC3)C#N)C(F)(F)F 5N-370S CCN(CC)c1c(c(cc(n1)C2CC2)C(F)(F)F)C#N 5N-371S CC(C)(C)c1cc(c(c(n1)O)C#N)C(F)(F)F 5N-373S c1ccc(cc1)CN(c2ccccc2)C(=O)CCl 5N-374S c1ccc(cc1)C(=O)OC2CCS(=O)(=O)c3c2ccs3 5N-375S CSc1nc2c(c(n1)O)CCCC2 5N-376S c1cc(ccc1CSc2nc3c(c(n2)O)CCCC3)Cl 5N-377S c1cc(ccc1CSc2nc3c(c(n2)Cl)CCCC3)Cl 5N-378S c1ccc(c(c1)C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3)C(F)(F)F 5N-379S c1csc2c1/C(=N/OC(=O)C3CC3)/CCS2(=O)=O 5N-380S CC(C)(C)C(=O)O/N=C/1\CCS(=O)(=O)c2c1ccs2 5N-381S CC(C)C(=O)O/N=C/1\CCS(=O)(=O)c2c1ccs2 5N-382S CC(C)(C)c1cc(c(c(n1)NC)C#N)C(F)(F)F 5N-384S Cc1cc(c(c(n1)Sc2ccccc2C(=O)OC)C#N)C(F)(F)F 5N-388S CCN(CC)c1c(c(cc(n1)C)C(F)(F)F)C#N 5N-389S Cc1cc(c(c(n1)Oc2ccccc2)C#N)C(F)(F)F 5N-390S Cc1cc(c(c(n1)Sc2ccc(cc2)Cl)C#N)C(F)(F)F 5N-391S Cc1cc(c(c(n1)Sc2ccccc2)C#N)C(F)(F)F 5N-392S Cc1cc(c(c(n1)N2CCCC2)C#N)C(F)(F)F 5N-393S Cc1ccc(cc1)Sc2c(c(cc(n2)C)C(F)(F)F)C#N 5N-394S Cc1cc(c(c(n1)NC)C#N)C(F)(F)F 5N-395S Cc1cc(c(c(n1)N2CCOCC2)C#N)C(F)(F)F 5N-396S Cc1cc(c(c(n1)Oc2ccc3ccccc3c2)C#N)C(F)(F)F 5N-397S Cc1cc(c(c(n1)Oc2ccc(cc2F)F)C#N)C(F)(F)F 5N-398S COc1ccc2c(c1)c(cc(n2)O)C(F)(F)F 5N-504S Cc1cc(cc(c1)NC(=O)c2cc(n(n2)c3ccc(cc3Cl)Cl)c4ccc(c(c4)Cl)Cl)C 5N-506S CO/N=C(/CN1CCCC1)\c2ccc(cc2)Cl 5N-511S COc1ccc(cc1)C2C(C(=O)N2c3ccccc3)CN4CCCCC4 5N-512S COc1ccc(cc1)C2C(C(=O)N2c3ccccc3)CN4CCOCC4 5N-514S COc1ccc(cc1)C2C(C(=O)N2c3ccccc3)CN4CCN(CC4)c5ccccc5F 5N-516S CC(=O)Nc1ccc(cc1)/C=N/OCc2c(nn(c2Sc3ccc(cc3)Br)C)C(F)(F)F 5N-518S Cn1c(c(c(n1)C(F)(F)F)CO/N=C/c2c(cccc2Cl)Cl)Sc3ccc(cc3)Br 5N-519S CO/N=C(/CN1CCCCC1)\c2ccc(cc2)Cl 5N-524S CN1C(=O)/C(=N\OC(=O)c2ccc(cc2Cl)Cl)/C(=N1)C(F)(F)F 5N-525S COc1ccc(cc1)N2C(C(C2=O)CN3CCCCC3)c4ccccc4 5N-526S CCN(CC)CC1C(N(C1=O)c2ccc(cc2)OC)c3ccccc3 5N-527S CN1CCN(CC1)CC2C(N(C2=O)c3ccc(cc3)OC)c4ccccc4 5N-529S COc1ccc(cc1)C2C(C(=O)N2c3ccccc3)CN4CCCC4 5N-530S CN1CCN(CC1)C/C(=N/OC)/c2ccc(cc2)Cl 5N-531S CO/N=C(/CN1CCN(CC1)c2ccccc2F)\c3ccc(cc3)Cl 5N-532S CO/N=C(/CN1CCN(CC1)C(c2ccccc2)c3ccccc3)\c4ccc(cc4)Cl 5N-533S c1cc(c(nc1)SCC(=O)O)C(F)(F)F 5N-537S COc1ccc(cc1)N2C(C(C2=O)CSc3ccc(cc3)Br)c4ccccc4 5N-538S CC(C)(C)c1ccc(cc1)SCC2C(N(C2=O)c3ccc(cc3)OC)c4ccccc4 5N-539S CSc1nc2ccccc2c(n1)N3CCOCC3 5N-542S CSc1nc2ccccc2c(n1)N3CCCCC3 5N-543S CNc1c2ccccc2nc(n1)SC 5N-544S CN(C)c1c2ccccc2nc(n1)SC 5N-545S CSc1nc2ccccc2c(n1)NCC=C 5N-546S Cc1ccc(cc1)n2c(cc(n2)C(=O)Nc3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl 5N-581S Cc1ccc(cc1)n2c(cc(n2)C(=O)Nc3ccc(cc3Cl)Cl)c4ccc(cc4)Cl 5N-582S Cc1ccc(cc1)n2c(cc(n2)C(=O)Nc3ccc(cc3C)Cl)c4ccc(cc4)Cl 5N-583S Cc1ccc(cc1)n2c(cc(n2)C(=O)Nc3cc(ccc3C)Cl)c4ccc(cc4)Cl 5N-584S Cc1ccc(cc1)n2c(cc(n2)C(=O)O)c3ccccc3Cl 5N-585S c1cc(ccc1c2cc(nn2c3ccc(cc3)Cl)C(=O)N4CCOCC4)Cl 5N-588S CNC(=O)c1cc(n(n1)c2ccc(cc2)Cl)c3ccc(cc3)Cl 5N-589S Cc1cc(ccc1NC(=O)c2cc(n(n2)c3cccc(c3)Cl)c4ccc(c(c4)Cl)Cl)Cl 5N-592S CNC(=O)c1cc(n(n1)c2cccc(c2)Cl)c3ccc(cc3)Cl 5N-593S CN(C)C(=O)c1cc(n(n1)c2ccc(cc2Cl)Cl)c3ccc(cc3)Cl 5N-595S c1cc(ccc1c2cc(nn2c3ccc(cc3Cl)Cl)C(=O)N4CCOCC4)Cl 5N-596S c1cc(ccc1c2cc(nn2c3ccc(c(c3)Cl)Cl)C(=O)N4CCOCC4)Cl 5N-597S c1cc(c(cc1c2cc(no2)CO)Cl)Cl 5N-600S c1cc(ccc1c2cc(no2)CO)Cl 5N-601S c1cc(ccc1c2cc(no2)COC(=O)C3CC3)Cl 5N-602S c1cc(c(cc1c2cc(no2)CCl)Cl)Cl 5N-603S Cc1ccc(cc1)NC(=O)OCc2cc(on2)c3ccc(cc3)Cl 5N-604S Cc1ccc(cc1)C(=O)OCc2cc(on2)c3ccc(cc3)Cl 5N-605S c1cc(cc(c1)C(F)(F)F)C(=O)OCc2cc(on2)c3ccc(c(c3)Cl)Cl 5N-606S COc1ccc(cc1)C(=O)OCc2cc(on2)c3ccc(c(c3)Cl)Cl 5N-607S c1cc(ccc1c2cc(no2)COC(=O)c3ccc(cc3Cl)Cl)Cl 5N-608S c1cc(cc(c1)C(F)(F)F)C(=O)OCc2cc(on2)c3ccc(cc3)Cl 5N-609S c1cc(ccc1c2cc(no2)COC(=O)c3ccc(cc3)F)Cl 5N-610S c1cc(c(c(c1)F)C(=O)OCc2cc(on2)c3ccc(c(c3)Cl)Cl)F 5N-611S c1cc(sc1)C(=O)OCc2cc(on2)c3ccc(c(c3)Cl)Cl 5N-612S c1cc(ccc1c2cc(no2)COC(=O)c3ccc(cc3)Cl)Cl 5N-613S CC(=O)Nc1ccc(cc1)/C=C/c2nc3ccccc3s2 5N-641S COc1cccc(c1)C(=O)Nc2ccc(cc2)/C=C/c3nc4ccccc4s3 5N-647S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3)NC(=O)c4cccc(c4)C(F)(F)F 5N-648S Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)/C=C/c3nc4ccccc4s3 5N-649S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3)NS(=O)(=O)c4cccc(c4)C(F)(F)F 5N-651S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3)NS(=O)(=O)c4ccc(cc4)Cl 5N-652S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3)NS(=O)(=O)c4ccc(cc4)F 5N-653S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3)NC(=O)c4ccc(cc4)Cl 5N-654S c1ccc2c(c1)nc(s2)/C=C/c3ccc(cc3)NC(=O)c4ccc(cc4Cl)Cl 5N-659S CCOC(=O)/C(=N\Nc1ccccc1)/Cl 5N-666S c1ccc(cc1)n2c(=O)cc(c(n2)S(=O)(=O)c3ccccc3)C(F)(F)F 5N-671S Cc1ccc(cc1)OC(=O)CN(c2ccccc2)S(=O)(=O)c3ccccc3 5N-672S c1ccc(cc1)N(CC(=O)Oc2ccc(cc2)F)S(=O)(=O)c3ccccc3 5N-673S CN1CC(C(C1)C(=O)c2ccc(cc2)Cl)c3ccc(cc3)N(C)C 5N-700 c1cc(oc1)c2ccnc3n2nc(n3)SCCC(=C(F)F)F 5N-701 c1cc(cc(c1)O)/C=C/C(=O)c2ccc(cc2)Cl 5N-702 c1ccc(cc1)/C=C/C(=O)c2ccc(cc2Cl)Oc3ccc(cc3)Cl 5N-704 c1ccc(cc1)CSc2nccc(n2)c3cc(sc3Cl)Cl 5N-705 CN1CC(C(C1)C(=O)c2ccc(cc2)F)c3ccc(cc3)F 5N-706 CCNC(=O)OCc1ccoc1 5N-708 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCc3ccc(cc3)C(=O)NN 5N-709 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)Nc3cccc(c3)C(F)(F)F 5N-710 Cc1ccc(cc1)NC(=O)N2Cc3ccccc3CC2C(=O)NC(C)(C)C 5N-711 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)Nc3cccc(c3)Cl 5N-712 CCNC(=O)N1Cc2ccccc2CC1C(=O)NC(C)(C)C 5N-713 COC(=O)c1ccccc1SCCC(=C(F)F)F 5N-715 c1ccc(c(c1)/C=C/C(=O)c2ccc(cc2)Cl)F 5N-717 CN1CC(C(C1)C(=O)c2ccc(cc2Cl)Oc3ccc(cc3)Cl)c4ccccc4 5N-718 c1c2c(nc3n1nc(n3)SCCC(=C(F)F)F)CCCC2=O 5N-720 CN1CC(C(C1)C(=O)c2ccc(cc2)OC)c3ccc(cc3)Cl 5N-721 CN1CC(C(C1)C(=O)c2ccc(cc2)Cl)c3ccccc3F 5N-723 c1cc(ccc1C(=O)/C=C/c2ccc(o2)c3ccc(cc3Cl)Cl)Cl 5N-725 CCOC(=O)CSCCC(=C(F)F)F 5N-727 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)Nc3ccccc3Cl 5N-728 CN1CC(C(C1)C(=O)c2ccc(cc2)Cl)c3ccc(o3)c4ccc(cc4Cl)Cl 5N-729 c1cc(c(c(c1)F)C#N)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 5N-732 c1ccc(cc1)C2CC(=NN2c3ccc(cc3)F)c4ccc(cc4)Cl 5N-733 CCOC(=O)CN1C(=O)C2Cc3ccccc3CN2C1=S 5N-734 c1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccc(cc4)Cl 5N-737 CN(C)/C=C\1/C(=O)SC(=N1)SC 5N-741 CC(=O)Nc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Cl 5N-742 c1ccc(cc1)c2cnc3nc(nn3c2N)SCCC(=C(F)F)F 5N-743 COc1ccc(cc1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccccc4 5N-744 c1ccc(cc1)N2C(=O)C3Cc4ccccc4CN3C2=S 5N-745 COc1cccc(c1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccccc4 5N-746 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)Cl)c4ccc(cc4Cl)Cl 5N-747 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=S)NC(C)(C)C 5N-748 COc1ccc(cc1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccc(cc4)F 5N-749 CC(=O)Nc1ccc(cc1)C2CN(CC2C(=O)c3ccc(cc3)Cl)C 5N-750 CC(C)(C)NC(=O)C1Cc2ccccc2CN1C(=O)c3cc(cc(c3)Cl)Cl 5N-751 c1ccc(cc1)C2CC(=NN2c3ccc(cc3F)F)c4ccc(cc4)Cl 5N-752 CC(=O)Nc1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccc(cc4)Cl 5N-753 c1ccc(cc1)N/N=C(\C=C\c2ccc(cc2)Cl)/c3ccc(cc3)[N+](=O)[O-] 5N-754 c1ccc(cc1)C2CC(=NN2c3ccc(cc3)Cl)c4ccc(cc4)Cl 5N-755 CC(C)(C)NC(=O)C1Cc2ccccc2CN1S(=O)(=O)c3ccc(cc3)OC 5N-756 c1ccc2c(c1)CC3C(=O)N(C(=S)N3C2)c4ccc(cc4)Cl 5N-757 COc1cccc(c1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccc(cc4)F 5N-758 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)Cl)c4ccco4 5N-759 CN1C(=O)C2Cc3ccccc3CN2C1=S 5N-760 CCN1C(=O)C2Cc3ccccc3CN2C1=S 5N-762 Cc1cccc(c1)C(=O)N2Cc3ccccc3CC2C(=O)NC(C)(C)C 5N-763 Cc1ccccc1CSc2nccc(n2)c3cc(sc3Cl)Cl 5N-764 Cc1ccc(cc1)CSc2nccc(n2)c3cc(sc3Cl)Cl 5N-765 c1cc(ccc1Cn2cnc3c(c2=O)ccs3)Cl 5N-803 COc1ccc(cc1)Cn2cnc3c(c2=O)ccs3 5N-804 c1ccc(c(c1)Cn2cnc3c(c2=O)ccs3)F 5N-805 c1cc(cc(c1)C(F)(F)F)Cn2cnc3c(c2=O)ccs3 5N-806 Cc1cccc(c1)Cn2cnc3c(c2=O)ccs3 5N-807 CC(=O)Nc1c(ccs1)C(=O)Nc2ccc(cc2)OC 5N-808 COC(=O)c1ccsc1NC(=S)Nc2ccccc2 5N-809 COC(=O)c1ccsc1NC(=O)Nc2cccc(c2)Cl 5N-810 CC(=O)Nc1c(cc(s1)Cl)C(=O)O 5N-811 COC(=O)c1ccsc1/N=C/Nc2nncs2 5N-812 Cn1c(=O)c(cn(c1=O)c2c(ccs2)C(=O)OC)C#N 5N-813 COC(=O)c1ccsc1NC(=S)Nc2ccc(cc2)[N+](=O)[O-] 5N-814 c1cc(ccc1C(=O)Nc2c(ccs2)C#N)Cl 5N-815 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2c(ccs2)C#N 5N-816 c1csc(c1C#N)NC(=O)CCl 5N-817 C1CCN(CC1)C(=O)CC#N 5N-819 C1COCCN1C(=O)CC#N 5N-820 c1cc(cc(c1)Cl)SCC(=O)Nc2c(ccs2)C#N 5N-821 C1CCN(C1)C(=O)CC#N 5N-822 CCOC(=O)NC(=O)/C(=C/Nc1c(ccs1)C#N)/C#N 5N-823 CN(C)/C=N/c1c(ccs1)C#N 5N-824 c1cc(ccc1NC(=O)Nc2c(ccs2)C#N)Cl 5N-825 c1cc(ccc1NC(=S)Nc2c(ccs2)C#N)Cl 5N-826 c1ccc(cc1)/C=N/c2c(ccs2)C#N 5N-827 c1cc(cc(c1)C(F)(F)F)CC(=O)OCC(=O)Nc2c(ccs2)C#N 5N-828 Cc1ccc(n1c2c(ccs2)C#N)C 5N-830 c1cc(ccc1N/C=N/c2c(ccs2)C#N)Cl 5N-831 c1cc(cc(c1)N/C=N/c2c(ccs2)C#N)C(F)(F)F 5N-832 c1cc(cc(c1)SCC(=O)Nc2c(ccs2)C#N)C(F)(F)F 5N-833 c1csc(c1C#N)n2cc(c(=O)[nH]c2=O)C#N 5N-834 c1cc(ccc1F)S(=O)(=O)Nc2c(ccs2)C#N 5N-835 c1csc(c1C#N)NC(=O)CSc2c(cc(cn2)C(F)(F)F)Cl 5N-836 c1csc(c1C#N)NC(=O)CSC2CCCCC2 5N-837 c1ccc(c(c1)/C=N/c2c(ccs2)C#N)Cl 5N-838 Cc1ccc(cc1)/C=N/c2c(ccs2)C#N 5N-839 c1ccc(c(c1)/C=N/c2c(ccs2)C#N)C(F)(F)F 5N-840 c1csc2c1c(ncn2)N 5N-841 CC(=O)Nc1ccccc1OCC(=O)Nc2c(ccs2)C#N 5N-843 c1ccc2c(c1)c(ccc2Cl)OCC(=O)Nc3c(ccs3)C#N 5N-844 COc1ccc(cc1)NC(=O)N2C(COC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cc5ccccc5 5N-900 c1ccc(cc1)C(CO)NC(=O)CNC(=O)c2ccc(cc2)Cl 5N-901 c1ccc(cc1)CC(COC(=O)c2ccc(cc2F)F)NC(=O)c3ccc(cc3F)F 5N-902 CC(C)(C)C(C(=O)NC)NC(=O)CNC(=O)c1ccc(cc1)Cl 5N-903 c1ccc(cc1)C(CO)N2C(=O)CNC2=S 5N-905 Cc1ccc(cc1)NC(=O)N2C3(CCN(CC3)c4ccc(cc4)[N+](=O)[O-])CC(=O)N2 5N-910 COC(=O)c1c2c(sc1N(S(=O)(=O)C)S(=O)(=O)C)CN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 5N-911 C=C(c1cn(c2c1cccc2)Cc3ccc(cc3Cl)Cl)c4cn(c5c4cccc5)Cc6ccc(cc6Cl)Cl 5N-915 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(COC(=O)c3c(onc3c4c(cccc4Cl)F)C)c5ccccc5 5N-916 CCOC(=O)NC(=O)/C(=N\Nc1ccc(cc1)Cl)/C#N 5N-918 c1cc(ccc1n2c(=O)[nH]c(=O)c(n2)C#N)Cl 5N-919 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3c(cccc3C)C)c4cccs4 5P-001 c1cc2c(cn[nH]2)c(c1)NC(=S)N 5P-002 Cc1ccc2c(c1NC(=S)N)CCCN2 5P-003 COc1ccc(c(c1)N/C=N/C(=C(/C#N)\N)/C#N)OC 5P-006 C1CCC(CC1)NCC(C(F)(F)F)O 5P-007 C1CCC(=CC(=O)O)CC1 5P-014 CCCCCCCCCc1ccc(cc1)Oc2ccccc2C=O 5P-015 Cc1ccc2cccnc2c1NC(=S)NC(=O)c3ccccc3 5P-016 CCOC(=O)c1cc([nH]c1N2CCN(CC2)c3cccc(c3)Cl)c4cccs4 5P-019 CC(c1ccccc1)NCC(C(F)(F)F)O 5P-023 C1CCN(CC1)CC(C(F)(F)F)O 5P-024 c1ccc(cc1)/C(=N/O)/Nc2ccccc2Cl 5P-025 COc1ccc(c(c1)n2cnc(c2N)C#N)OC 5P-028 c1cc(cc(c1)Cl)/C=N/O 5P-032 c1ccc2c(c1)cc([nH]2)C(=S)N 5P-033 COc1ccc(c2c1[nH]c(n2)C(F)(F)F)OC 5P-035 c1ccc(cc1)/C(=N/O)/Nc2ccc(cc2)Cl 5P-038 Cc1ccc2ccccc2c1N 5P-039 c1ccc(cc1)CN2CCN(CC2)CC(C(F)(F)F)O 5P-043 COc1ccc(c(c1N)NC(=O)C(F)(F)Cl)OC 5P-045 COc1ccc(c2c1[nH]c(n2)C(C(C(F)(F)F)(F)F)(F)F)OC 5P-046 Cc1ccc2ccccc2c1NC(=S)NC(=O)c3ccccc3 5P-048 c1ccc2c(c1)cc([nH]2)C#N 5P-050 c1ccc(cc1)/C(=N\O)/Nc2ccccc2 5P-051 c1ccc2c(c1)c(c[nH]2)C(=O)N 5P-052 Cc1ccc2ccccc2c1NC(=S)N 5P-054 c1cc(ccc1/C(=N/O)/Nc2ccc(cc2)Cl)Cl 5P-058 c1cc(cnc1)/C=N/O 5P-059 c1ccc2c(c1)CCN(C2)CC(C(F)(F)F)O 5P-062 c1ccc(cc1)/C(=N/O)/Nc2cccc(c2)Cl 5P-065 Cn1c2ccccc2c(=O)c3c1cccc3O 5P-071 c1cc(cc(c1)Oc2ccc(cc2)C#N)C(F)(F)F 5P-072 C1CCCC(CC1)NCC(C(F)(F)F)O 5P-073 CCOn1ccnc1 5P-074 Cc1ccc(cc1)COn2ccnc2C=O 5P-075 C1=CC(=O)c2c([nH]c(n2)C(F)(F)F)C1=O 5P-076 c1ccc(cc1)N/C(=N\O)/c2ccc(cc2)Cl 5P-077 c1ccc(cc1)CCOn2ccnc2C=O 5P-078 CCOC(=O)c1c(nc2ccccn2c1=O)O 5P-079 Cc1ccc2cccnc2c1NC(=S)N 5P-081 Cc1cc(ccc1N/C=N\C(=C(\C#N)/N)\C#N)OC 5P-082 CC(=O)N1CCC(CC1)C(=O)O 5P-083 CCOC(=O)c1c(nc2n(c1=O)c3ccccc3s2)O 5P-086 Cc1ccc2c(c1N)cccn2 5P-087 CCOC(=O)C(C(C(=O)OCC)NCc1ccco1)C(=O)OCC 5P-088 CCOC(=O)C(C(C(=O)OCC)N1CCOCC1)C(=O)OCC 5P-089 C/C(=C/C(=O)C(F)(F)F)/Nc1ccsc1C(=O)OC 5P-090 Cc1ccc2c(c1NC(=S)NC(=O)c3ccccc3)cccn2 5P-092 CN(C)/C=C/C(=C/C(=O)C(F)(F)F)/Nc1ccsc1C(=O)OC 5P-094 c1ccn(c1)c2ccsc2C(=O)NN 5P-306S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)COc3ccccc3 5P-309S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)COc3ccc(cc3Cl)F 5P-310S COC(=O)c1c(ccs1)NC(=O)CSc2ccccc2NC(=O)COc3ccc4ccccc4c3 5P-311S CSc1c(ccc(n1)C(F)(F)F)C#N 5P-314S c1cc(ccc1CSc2c(ccc(n2)C(F)(F)F)C#N)Cl 5P-316S c1cc(cc(c1)C(F)(F)F)CSc2c(ccc(n2)C(F)(F)F)C#N 5P-317S CC(C)Sc1c(ccc(n1)C(F)(F)F)C#N 5P-318S CC(C)(C)C(=O)Nc1ccccn1 5P-319S CC(C)C(=O)NNC(=O)c1c(ccs1)n2cccc2 5P-320S Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-321S Cc1ccccc1Sc2c3c(noc3ncn2)C 5P-324S Cc1c2c(ncnc2Sc3ccc(cc3)Br)on1 5P-325S Cc1c2c(ncnc2Sc3c(cccc3Cl)Cl)on1 5P-326S Cc1c2c(ncnc2Sc3ccccc3Cl)on1 5P-327S Cc1c2c(ncnc2Sc3ccccc3C(=O)OC)on1 5P-328S Cc1c2c(ncnc2Oc3ccccc3)on1 5P-330S Cc1cccc(c1C)Oc2c3c(noc3ncn2)C 5P-331S Cc1c2c(ncnc2Oc3ccc(cc3)F)on1 5P-333S Cc1c2c(ncnc2Oc3cccc(c3)C(F)(F)F)on1 5P-334S Cc1cccc(c1)Oc2c3c(noc3ncn2)C 5P-335S Cc1cc(ccc1Oc2c3c(noc3ncn2)C)Cl 5P-336S c1ccc(cc1)C(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-337S c1ccn(c1)c2ccsc2C(=O)NNC(=O)c3cccc(c3)Cl 5P-338S c1ccn(c1)c2ccsc2C(=O)NNS(=O)(=O)c3ccc(cc3)Cl 5P-339S c1ccn(c1)c2ccsc2C(=O)NNS(=O)(=O)c3ccc(cc3)F 5P-340S Cc1c(sc2n1c3ccccc3n2)C(=O)C 5P-343S CS(=O)(=O)c1nc2ccccc2s1 5P-344S CC(C)(C)C(=O)Nc1c(cccn1)C(c2ccccc2)O 5P-345S CC(C)(C)C(=O)Nc1c(cccn1)C(c2cccc(c2)C(F)(F)F)O 5P-346S COC(=O)c1c(c2ccc(nc2s1)C(F)(F)F)N 5P-349S CCOC(=O)c1ccc(n(c1=O)Cc2ccc(cc2)Cl)C(F)(F)F 5P-350S c1cc(ccc1Cn2c(ccc(c2=O)C(=O)O)C(F)(F)F)Cl 5P-351S COc1cccc(c1)C(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-355S Cc1ccc(cc1)C(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-356S c1ccn(c1)c2ccsc2C(=O)NNS(=O)(=O)c3cc(cc(c3)Cl)Cl 5P-357S COc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-358S c1ccc(cc1)NC(=O)N2CC2C#N 5P-359S c1ccc2c(c1)nc(s2)N3CCNCC3 5P-361S Cc1ccc(c(c1)[N+](=O)[O-])Oc2c3c(noc3ncn2)C 5P-362S Cc1c2c(ncnc2Oc3ccccc3Cl)on1 5P-363S Cc1c2c(ncnc2Oc3ccc(cc3Cl)Cl)on1 5P-364S Cc1c2c(ncnc2Oc3ccc(cc3)C(C)(C)C)on1 5P-365S Cc1c2c(ncnc2Oc3ccc(cc3Br)Cl)on1 5P-366S Cc1ccc(c(c1)Oc2c3c(noc3ncn2)C)C(C)C 5P-367S Cc1c2c(ncnc2Oc3cc(ccc3Cl)Cl)on1 5P-369S Cc1c2c(ncnc2Oc3ccc4ccccc4c3)on1 5P-370S c1ccn(c1)c2ccsc2C(=O)NNC(=O)c3ccc(cc3)Cl 5P-371S c1ccc(c(c1)C(=O)NNC(=O)c2c(ccs2)n3cccc3)Cl 5P-372S c1ccn(c1)c2ccsc2C(=O)NNC(=O)c3ccc(cc3)F 5P-373S c1ccc(cc1)NC(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-374S Cc1c2c(ncnc2on1)N3CCCC3 5P-376S CCN(CC)c1c2c(noc2ncn1)C 5P-377S c1ccc(cc1)S(=O)(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-378S c1ccn(c1)c2ccsc2C(=O)NNS(=O)(=O)c3ccc(cc3)Br 5P-379S c1ccc(c(c1)F)S(=O)(=O)NNC(=O)c2c(ccs2)n3cccc3 5P-380S COc1cccc(c1)C(=O)N2CCN(CC2)C(=O)c3ccccc3 5P-501S c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3cccc(c3Cl)Cl 5P-502S c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3ccc(cc3Cl)Cl 5P-503S c1ccc2c(c1)C(=O)N(C2=O)COc3cccc(c3)Cl 5P-504S c1ccc2c(c1)nc(s2)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 5P-505S c1ccc2c(c1)nc(s2)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)F 5P-506S Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3nc4ccccc4s3 5P-507S c1ccc2c(c1)nc(s2)C3CCN(CC3)S(=O)(=O)C(F)(F)F 5P-508S CNC(=O)c1c(=O)ccn(n1)c2ccc(cc2)Cl 5P-511S COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3nc4ccccc4s3 5P-512S c1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3nc4ccccc4s3 5P-513S c1ccc(cc1)CS(=O)(=O)N2CCC(CC2)c3nc4ccccc4s3 5P-514S c1ccc(cc1)S(=O)(=O)N2CCCC2c3nc4ccccc4s3 5P-516S c1ccc2c(c1)nc(s2)C3CCCN3S(=O)(=O)c4ccc(cc4)Cl 5P-517S Cc1ccc(cc1)S(=O)(=O)N2CCCC2c3nc4ccccc4s3 5P-518S COc1ccc(cc1)S(=O)(=O)N2CCCC2c3nc4ccccc4s3 5P-519S c1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3nnc(s3)C(F)(F)F 5P-520S c1cc(ccc1n2ccc(=O)c(n2)C(=O)O)Cl 5P-522S c1ccc2c(c1)nc(s2)C3CCCN3S(=O)(=O)c4cc(cc(c4)Cl)Cl 5P-523S c1ccc(cc1)CS(=O)(=O)N2CCCC2c3nc4ccccc4s3 5P-524S c1ccc2c(c1)nc(s2)C3CCCN3S(=O)(=O)c4cc(ccc4Cl)Cl 5P-525S c1ccc2c(c1)nc(s2)C3CCCN3S(=O)(=O)c4ccc(cc4)Br 5P-526S c1ccc(cc1)c2ccc(=O)[nH]n2 5P-527S c1cc(ccc1n2ccc(=O)c(n2)C(=O)NN)Cl 5P-528S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)S 5P-531S Cc1c(n(c(c1C#N)NC(=O)Nc2ccc(c(c2)Cl)Cl)Cc3ccc(cc3)OC)C 5P-561S Cc1c(n(c(c1C#N)NC(=O)Nc2ccc(cc2)F)Cc3ccc(cc3)OC)C 5P-563S COc1ccc(cc1)Sc2c3cc(oc3ncn2)c4ccccc4 5P-565S c1ccc(cc1)c2cc3c(o2)ncnc3Sc4ccc(cc4)Br 5P-568S c1ccc(cc1)c2cc3c(o2)ncnc3Sc4ccc(cc4)Cl 5P-570S c1ccc(cc1)c2cc3c(o2)ncnc3Sc4ccccc4 5P-572S Cc1ccc(c(c1)C)Sc2c3cc(oc3ncn2)c4ccccc4 5P-573S Cc1ccccc1Sc2c3cc(oc3ncn2)c4ccccc4 5P-575S c1ccc(cc1)c2cc3c(o2)ncnc3Sc4ccccc4Cl 5P-576S Cc1ccccc1Oc2c3cc(oc3ncn2)c4ccccc4 5P-577S COc1cccc(c1)C(=O)Nc2c(c3c(o2)cccn3)C#N 5P-578S Cc1cccc(c1C)Oc2c3cc(oc3ncn2)c4ccccc4 5P-580S c1ccc(cc1)c2cc3c(o2)ncnc3Oc4ccc(cc4)Cl 5P-581S c1ccc(cc1)c2cc3c(o2)ncnc3Oc4ccccc4 5P-584S Cc1ccc(c(c1)Oc2c3cc(oc3ncn2)c4ccccc4)C(C)C 5P-585S c1cc2c(c(c(o2)NC(=O)c3cccs3)C#N)nc1 5P-588S c1ccc(cc1)C(=O)Nc2c(c3c(o2)cccn3)C#N 5P-589S c1cc2c(c(c(o2)NC(=O)c3ccc(cc3)Cl)C#N)nc1 5P-590S Cc1cc(ccc1Oc2c3cc(oc3ncn2)c4ccccc4)Cl 5P-593S CCOC(=O)c1nc(no1)CS(=O)(=O)c2ccccc2 5P-644S Cc1ccc(cc1)C(=O)NNC(=O)c2c3ccccc3c(=O)n(n2)c4cccc(c4C)Cl 5P-647S Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)C(=O)NNS(=O)(=O)c4cc(ccc4Cl)Cl 5P-648S Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(c(c4)C)C 5P-649S c1ccc(cc1)S(=O)(=O)C/C(=N/OC(=O)C2CC2)/N 5P-651S c1ccc(cc1)S(=O)(=O)C/C(=N/OC(=O)c2cccs2)/N 5P-652S c1ccc(cc1)S(=O)(=O)C/C(=N/OC(=O)c2ccc(cc2)F)/N 5P-653S Cc1cccc(c1)C(=O)O/N=C(/CS(=O)(=O)c2ccccc2)\N 5P-655S COc1cccc(c1)C(=O)O/N=C(/CS(=O)(=O)c2ccccc2)\N 5P-657S c1ccc(cc1)S(=O)(=O)C/C(=N/OC(=O)c2ccccc2C(F)(F)F)/N 5P-658S c1ccc(c(c1)S(=O)(=O)N2CCCC2c3nc(no3)c4cccc(c4)C(F)(F)F)Cl 5P-660S c1ccc(c(c1)S(=O)(=O)N2CCCC2c3nc(no3)c4ccc(cc4)Cl)Cl 5P-661S c1ccc(c(c1)S(=O)(=O)N2CCCC2c3nc(no3)c4cccc(c4)Cl)Cl 5P-662S c1ccc(c(c1)c2nc(on2)C3CCCN3S(=O)(=O)c4ccccc4Cl)Cl 5P-663S c1ccc(cc1)S(=O)(=O)Cc2nc(on2)C3CCCN3S(=O)(=O)c4ccccc4Cl 5P-664S COc1cccc(c1)c2nc(no2)CS(=O)(=O)c3ccccc3 5P-665S CCOC(=O)c1c2ccccc2c(=O)n(n1)c3cccc(c3C)Cl 5P-667S Cc1c(cccc1Cl)n2c(=O)c3ccccc3c(n2)C(=O)NN 5P-668S Cc1c(cccc1Cl)n2c(=O)c3ccccc3c(n2)C(=O)N/N=C/c4ccc(c(c4)F)F 5P-670S Cc1c(cccc1Cl)n2c(=O)c3ccccc3c(n2)C(=O)N/N=C/c4cccc(c4)OC 5P-672S c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)NC(=O)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)O 5P-701 Cc1cccc(n1)n2cc(nc2)C(=O)OC 5P-703 CN1C(=O)N(C(O1)CC(=O)NC2CCCCCC2)c3ccc(cc3)Cl 5P-705 CSc1cccc(c1)n2ccc(c(c2=O)Cc3ccc(cc3Cl)Cl)O 5P-709 CC(C)(Cn1ccc(c(c1=O)Cc2ccc(cc2Cl)Cl)O)SCc3cccc(c3)C(F)(F)F 5P-712 c1cc(ccc1COc2ccsc2C(=O)Nn3ccc(c(c3=O)Cc4ccc(cc4Cl)Cl)O)F 5P-713 Cc1ccc(cc1)/C=C(/c2c(cc(cn2)C(F)(F)F)Cl)\C(=O)OC 5P-714 CCOC(=O)C(Cc1ccc(cc1Cl)Cl)c2ccno2 5P-715 CCC(=O)C(c1ccc(cc1Cl)Cl)c2ccnc3n2nc(n3)N 5P-716 c1c(cnc(c1Cl)CC(=O)NN)C(F)(F)F 5P-720 C(C(CBr)Br)N(C=O)NC=O 5P-721 c1cc(ccc1CC(C(=O)O)NS(=O)(=O)c2ccc(cc2F)F)C#N 5P-725 Cc1ccc(cc1)C(=O)CSc2nccc(n2)CCc3ccc(cc3Cl)Cl 5P-726 C/C(=N\NC(=O)Cc1c(cc(cn1)C(F)(F)F)Cl)/C(=O)C 5P-728 Cc1c(nnc(c1c2c(cc(cn2)C(F)(F)F)Cl)O)C 5P-729 CC1(CC(=C(C(=O)C1)Br)O)C 5P-730 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4ccc(c(c4)Cl)Cl 5R-0001 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4ccc(cc4)C(F)(F)F 5R-0002 Cc1ccc(cc1)CSC2=Nc3cc(c(cc3C4=NC(=O)CN42)OC)OC 5R-0003 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4ccc(cc4)F 5R-0004 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4cccc(c4)F 5R-0005 Cc1cccc(c1)CSC2=Nc3cc(c(cc3C4=NC(=O)CN42)OC)OC 5R-0006 C1CCC(CC1)NC(=O)[C@H]2CCCC[C@H]2C(=O)O 5R-0008 Cn1c(ccc1C(C#N)c2ccccc2C#N)C=O 5R-0010 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4cccc(c4)Cl 5R-0011 CC(C)(C)OC(=O)CSC1=Nc2cc(c(cc2C3=NC(=O)CN31)OC)OC 5R-0012 Cc1ccccc1CSC2=Nc3cc(c(cc3C4=NC(=O)CN42)OC)OC 5R-0014 c1nncn1N2C(=O)C3CC=CCC3C2=O 5R-0015 C=CCNC(=S)Nn1cnnc1 5R-0017 c1ccc(c(c1)C(F)(F)F)NC(=O)[C@H]2CCCC[C@H]2C(=O)O 5R-0018 CCc1ccc(cc1)CSC2=Nc3cc(c(cc3C4=NC(=O)CN42)OC)OC 5R-0022 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4ccccc4F 5R-0024 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCC#N 5R-0025 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCCC(=C(F)F)F 5R-0027 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4cc(cc(c4)C(F)(F)F)C(F)(F)F 5R-0028 c1ccc(cc1)C2C(CCC(=O)N2C3CCCCC3)C(=O)n4ccnc4 5R-0029 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4c(cccc4Cl)F 5R-0031 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4ccccc4 5R-0032 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4ccc(cc4Cl)Cl 5R-0033 Cc1cc(n2c(n1)cc(n2)c3c(ccs3)n4cccc4)C(F)(F)F 5R-0041 c1ccn(c1)c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)C(F)(F)F 5R-0042 c1ccc(cc1)n2ccnc2SCC(C(F)(F)F)OC(=O)c3cccc(c3)C(F)(F)F 5R-0044 c1ccn(c1)c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5cccc(c5)Cl 5R-0045 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C)C)C 5R-0048 CC(=O)Nc1cccc(c1)c2[nH]nnn2 5R-0049 c1cc(ccc1c2[nH]nnn2)OCCOCCO 5R-0050 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCC=C 5R-0051 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCc4c(cccc4Cl)Cl 5R-0052 Cc1ccc(n1c2ccsc2c3cc([nH]n3)N)C 5R-0053 Cc1nnc(o1)c2cccc(c2)NC(=O)C 5R-0060 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3)SCCCC(=O)OC 5R-0062 CCOC(=O)C(=CNn1cnnc1)C(=O)OCC 5R-0063 c1ccc(cc1)n2ccnc2SCC(C(F)(F)F)OC(=O)c3ccco3 5R-0066 c1ccc(cc1)n2ccnc2SCC(C(F)(F)F)OC(=O)c3cccc(c3)Cl 5R-0067 Cc1cc(nn2c1nnc2)C 5R-0072 Cc1ccc(n1n2cnnc2)C 5R-0073 CCOC(=O)NC(c1ccccc1F)C2CCCCC2=O 5R-0075 CCOC(=O)NC(c1ccccc1)C2CCCCC2=O 5R-0076 CC(=O)NC(c1ccccc1F)C2CCCCC2=O 5R-0077 Cc1ccc(n1c2ccsc2c3c(c4nc(cc(n4n3)C)C)C)C 5R-0078 c1ccn(c1)c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5cccs5 5R-0079 Cc1cc(c(n1n2cnnc2)C)C=O 5R-0080 c1ccc(cc1)C2C(CCCN2C3CCCCC3)CO 5R-0083 CC1=C/C(=C/N(C)C)/C(=O)O1 5R-0084 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)c5ccc(cc5Cl)Cl)C)C 5R-0085 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5ccccc5)C 5R-0088 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5ccco5)C 5R-0089 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)Cl)C)C 5R-0090 Cc1ccc(cc1)C(=O)O/N=C/c2ccc(cc2)OCc3ccccc3 5R-0200 COc1ccc(cc1)C(=O)O/N=C/c2ccc(cc2)OCc3ccccc3 5R-0201 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCN(CC2)c3ccc(cc3)C#N 5R-0202 COCCN1C(=O)CC(=O)NC1=O 5R-0203 c1cc(c(c(c1)Cl)Cn2cc(cc2C#N)C(=O)Cc3ccc(cc3)Cl)F 5R-0204 c1ccc(cc1)Cc2c(nc3ccccc3n2)Oc4ccc(cc4)Cl 5R-0205 c1ccc(cc1)Cc2c(nc3ccccc3n2)Oc4cc(cc(c4)Cl)Cl 5R-0206 c1ccc(cc1)CC(=O)NCCCl 5R-0207 Cc1ccc(cc1)C(=O)O/C=C/C(=O)OC 5R-0209 c1cc(c(c(c1)Cl)Cl)C(=O)Nc2ccnc(n2)c3cccnc3 5R-0210 c1cc(nc(c1)F)N/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 5R-0213 c1cc(nc(c1)Cl)N/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 5R-0214 c1cc(cnc1)c2nccc(n2)NC(=O)c3ccco3 5R-0216 Cc1ccc(cc1)N/C=C/C(=O)c2ccccc2OCc3ccc(cc3)Cl 5R-0218 c1ccc(c(c1)C(=O)/C=C/Nc2ccc(cc2)OC(F)(F)F)OCc3ccc(cc3)Cl 5R-0219 c1ccc(cc1)N/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 5R-0220 Cc1cc2nccc(n2n1)c3ccccc3OCc4ccc(cc4)Cl 5R-0223 c1ccc(c(c1)c2cc[nH]n2)OCc3ccc(cc3)Cl 5R-0224 CC(=O)c1ccccc1OCc2ccc(cc2)F 5R-0225 CN1C(=O)C(=Cc2ccc(cc2)OCCN(C)c3ccccn3)C(=O)N(C1=O)C 5R-0226 CN(CCOc1ccc(cc1)/C=C/2\C(=O)NC(=O)N(C2=O)CCOC)c3ccccn3 5R-0227 CN(CCOc1ccc(cc1)C=C2C(=O)NC(=O)NC2=O)c3ccccn3 5R-0228 c1ccc(cc1)Cc2cc(=O)[nH]c(=S)[nH]2 5R-0229 c1ccc(c(c1)C(=O)/C=C/Nc2ccc(cc2F)Cl)OCc3ccc(cc3)Cl 5R-0230 c1ccc(c(c1)C(=O)C/C=N/OCc2ccc(cc2Cl)Cl)OCc3ccc(cc3)Cl 5R-0231 c1ccc(c(c1)c2ccnc3n2ncn3)OCc4ccc(cc4)Cl 5R-0232 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5ccccc5F 5R-0233 c1ccc(cc1)CC2=NCCO2 5R-0235 Cc1ccc(cc1)C(=O)n2ccc(n2)c3ccccc3OCc4ccc(cc4)Cl 5R-0236 c1ccc(c(c1)c2ccn(n2)C(=O)c3ccc(cc3)Cl)OCc4ccc(cc4)Cl 5R-0237 c1ccc(c(c1)c2ccn(n2)C(=O)c3cccs3)OCc4ccc(cc4)Cl 5R-0238 c1ccc(c(c1)c2ccnc(n2)N)OCc3ccc(cc3)Cl 5R-0239 c1ccc(c(c1)c2ccnc3n2ncc3C#N)OCc4ccc(cc4)Cl 5R-0241 Cc1ccc(cc1)/C=N\NC(=O)C2Cc3c4ccccc4ccc3O2 5R-0243 c1ccc(c(c1)c2ccn(n2)S(=O)(=O)c3ccc(cc3)F)OCc4ccc(cc4)Cl 5R-0244 COc1ccc(cc1)C(=O)n2ccc(n2)c3ccccc3OCc4ccc(cc4)Cl 5R-0245 c1ccc(c(c1)c2ccn(n2)C(=O)c3cccc(c3)Cl)OCc4ccc(cc4)Cl 5R-0246 c1ccc2c(c1)cccc2S(=O)(=O)n3ccc(n3)c4ccccc4OCc5ccc(cc5)Cl 5R-0248 c1ccc(c(c1)c2ccn(n2)S(=O)(=O)c3cc(ccc3Cl)Cl)OCc4ccc(cc4)Cl 5R-0249 Cc1cc(=O)[nH]c(n1)SCc2c(cccc2Cl)F 5R-0250 Cc1cc(=O)[nH]c(n1)SCc2cccc(c2)Cl 5R-0251 CCc1cc(=O)[nH]c(=S)[nH]1 5R-0252 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccccc3OCc4ccc(cc4)Cl 5R-0253 COc1cc2c(cc1OC)NC(=S)N3C2=NC(=O)C3Cc4ccccc4 5R-0254 Cc1ccc(cc1)Cn2ccc(n2)c3ccccc3OCc4ccc(cc4)Cl 5R-0255 CC(C)(C)c1cc(=O)[nH]c(=S)[nH]1 5R-0257 Cc1cc(=O)[nH]c(n1)SCc2ccc(cc2)C(F)(F)F 5R-0258 c1ccc(c(c1)c2ccn(n2)Cc3ccc(cc3)F)OCc4ccc(cc4)Cl 5R-0259 Cc1cc(=O)[nH]c(n1)SCc2cccc(c2)F 5R-0260 Cc1ccc(cc1)CSc2[nH]c(=O)cc(n2)C 5R-0261 Cc1cc(n(n1)c2c(nc3ccccc3n2)Cc4ccccc4)C 5R-0262 COCCN1C(=O)/C(=C/c2ccc(cc2)F)/C(=O)NC1=O 5R-0264 COc1ccccc1/C=C(\c2ccccc2)/C(=O)O 5R-0266 CCc1cc(=O)[nH]c(n1)SCc2c(cccc2Cl)F 5R-0267 CCc1cc(=O)[nH]c(n1)SCc2cccc(c2)Cl 5R-0268 c1ccc(c(c1)c2ccn(n2)Cc3ccc(c(c3)Cl)Cl)OCc4ccc(cc4)Cl 5R-0269 COCCN1C(=O)/C(=C/c2ccc(c(c2)OC)O)/C(=O)NC1=O 5R-0270 c1ccc(c(c1)c2ccnc(n2)c3ccncc3)OCc4ccc(cc4)Cl 5R-0271 c1ccc(c(c1)c2ccnc(n2)c3ccccn3)OCc4ccc(cc4)Cl 5R-0272 c1ccc2c(c1)[nH]c(=O)c(n2)N/N=C\3/CCCCC3c4ccc(cc4[N+](=O)[O-])[N+](=O)[O-] 5R-0273 Cc1cc2nccc(n2n1)c3ccccc3OCc4ccc(cc4)F 5R-0274 c1ccc(c(c1)c2ccnc3n2ncn3)OCc4ccc(cc4)F 5R-0275 Cc1c(c(no1)c2ccccc2)C(=O)c3cc([nH]c3)C(=O)NCc4ccncc4 5R-0276 Cc1c(c(no1)c2ccccc2)C(=O)c3cc([nH]c3)C(=O)NCc4ccccn4 5R-0277 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)NC3CCCCC3)Br 5R-0279 COCCCNC(=O)c1cc(c[nH]1)C(=O)c2ccccc2Br 5R-0280 Cc1c(c(no1)c2ccccc2)C(=O)c3cc([nH]c3)C(=O)NCCCN4CCOCC4 5R-0281 Cc1ccc(cc1)/C=N/NC(=O)C2CCN(CC2)Cc3ccccc3 5R-0283 c1ccc(c(c1)C(=O)C/C=N/OCc2ccc(cc2Cl)Cl)OCc3ccc(cc3)F 5R-0284 Cc1ccc(cc1)C(=O)NNC(=O)C2CCN(CC2)Cc3ccccc3 5R-0285 Cc1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)Cc3ccccc3 5R-0286 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3)C(F)(F)F 5R-0287 c1ccc(cc1)CN2CCC(CC2)C(=O)NNC(=O)c3cccc(c3)Cl 5R-0290 CCc1cc(=O)[nH]c(n1)SCc2ccc(cc2)F 5R-0292 CCCCCCCCCCCCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 5R-0294 c1ccc(cc1)CCNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3Cl)Cl 5R-0295 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)NCC3CCCO3 5R-0296 COc1ccccc1/C=C(/c2ccccc2)\C(=O)NCc3ccc(cc3)F 5R-0297 Cc1ccc(cc1)C(=O)n2ccc(n2)c3ccccc3OCc4ccc(cc4)F 5R-0298 c1ccc(c(c1)c2ccn(n2)C(=O)c3ccco3)OCc4ccc(cc4)F 5R-0299 c1ccc(c(c1)c2ccn(n2)C(=O)c3cccc(c3)Cl)OCc4ccc(cc4)F 5R-0300 Cc1ccc(cc1)CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)Cc5ccccc5)OC)OC 5R-0303 c1ccc(c(c1)c2ccn(n2)C(=O)c3ccc(cc3)F)OCc4ccc(cc4)F 5R-0305 COc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccccc3OCc4ccc(cc4)F 5R-0306 c1ccc(c(c1)c2ccn(n2)Cc3ccc(cc3)Cl)OCc4ccc(cc4)F 5R-0307 Cc1cc(c(c(c1)C)S(=O)(=O)n2ccc(n2)c3ccccc3OCc4ccc(cc4)F)C 5R-0308 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5ccc(cc5)C(F)(F)F 5R-0309 CCCCOc1ccc2cc(ccc2c1)/C=C/C(=O)OC 5R-0311 CN(C)/C=N/NC(=O)C1CCN(CC1)Cc2ccccc2 5R-0313 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5ccccc5 5R-0314 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5ccccc5Cl 5R-0315 c1cc(cnc1)C2=NOC(C2)C(=O)NN 5R-0316 c1ccc(cc1)CN2CCC(CC2)C(=O)NNS(=O)(=O)c3cc(ccc3Cl)Cl 5R-0317 CN1CCN(CC1)c2ccc(cn2)[N+](=O)[O-] 5R-0318 c1cc(c(nc1)SCCC(=O)O)C(=O)O 5R-0323 Cc1nnc2n1c3ccccc3nc2Cc4ccccc4 5R-0324 CCOC(=O)c1nnc2n1c3ccccc3nc2Cc4ccccc4 5R-0325 c1ccc(cc1)Cc2c(nc3ccccc3n2)N/N=C(/Cc4ccccc4)\C(=O)[O-].[Na+] 5R-0326 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5c(cccc5Cl)F 5R-0327 Cc1ccccc1CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)Cc5ccccc5)OC)OC 5R-0328 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCCc5ccccc5 5R-0329 COC(=O)c1c(ccs1)N/C=C/C(=O)C(F)(F)F 5R-0600 c1ccc(cc1)N/C=C/C(=O)C(F)(F)F 5R-0603 c1cc(ccc1C(=O)N2CCN=C(C=C2)C(F)(F)F)F 5R-0604 c1cc2c(cc1N)nccn2 5R-0605 CN(Cc1ccccc1)/C=C/C(=O)C(F)(F)F 5R-0606 c1ccc(cc1)S(=O)(=O)c2ccc(cn2)N 5R-0607 Cc1ccc(cc1)NC(=O)OCc2cnc(s2)Cl 5R-0608 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NS(=O)(=O)c3ccc(cc3F)F)C 5R-0610 c1cc(cc(c1)Cl)C(=O)N2CCN=C(C=C2)C(F)(F)F 5R-0612 C1CCN(CC1)C(=O)C(F)(F)Br 5R-0614 CCOC(=O)c1c(nn(c1C)c2ccc(cn2)NC(=O)CSCC(=O)O)C 5R-0616 c1cc2c(cc1NC(=O)/C=C/C(=O)O)nccn2 5R-0619 COc1ccc(cc1)NC(=O)Nc2ccc3c(c2)nccn3 5R-0620 c1ccc2c(c1)CCCN2C(=O)C(F)(F)Br 5R-0621 c1ccc2c(c1)CCN(C2)C(=O)C(F)(F)Br 5R-0622 CN(CCC(C(F)(F)F)O)Cc1ccccc1 5R-0624 c1ccc(cc1)NCCC(C(F)(F)F)O 5R-0626 Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)nccn3 5R-0627 c1cc(sc1)CNC(=O)c2ccc(cc2)N3CCS(=O)(=O)CC3 5R-0629 c1cc(ccc1C(=O)NN)N2CCS(=O)(=O)CC2 5R-0630 Cc1ccc(cc1)C(=O)Nc2c(cccn2)S(=O)(=O)c3ccccc3 5R-0631 c1ccc(cc1)NC(=O)Nc2ccc3c(c2)nccn3 5R-0633 c1ccc(c(c1)NC(=O)Nc2ccc3c(c2)nccn3)Cl 5R-0634 c1cc(cc(c1)Cl)NC(=O)Nc2ccc3c(c2)nccn3 5R-0635 c1cc(ccc1N2CCN(CC2)C(=O)CSCC(=O)O)F 5R-0637 c1cc(cc(c1)N2CCN(CC2)/C=C/C(=O)C(F)(F)F)C(F)(F)F 5R-0641 c1cc(ccc1C(=O)OCc2cnc(s2)Cl)Cl 5R-0643 Cc1c(nc2cc(ccc2n1)N)C 5R-0644 Cc1ccccc1C(=O)OCc2cnc(s2)Cl 5R-0645 Cc1cc(cnc1NCc2cc(cc(c2O)Br)Br)I 5R-0650 Cc1c(nc2cc(ccc2n1)NC(=O)c3ccc(cc3)I)C 5R-0652 Cc1c(nc2cc(ccc2n1)NC(=O)c3ccc(cc3)OC)C 5R-0653 Cc1c(nc2cc(ccc2n1)NC(=O)c3cccc(c3)C(F)(F)F)C 5R-0654 Cc1c(nc2cc(ccc2n1)NC(=O)/C=C/C(=O)O)C 5R-0655 c1cc(ccc1C(=O)OCc2cnc(s2)Cl)[N+](=O)[O-] 5R-0656 c1cc2c(c(c1)[N+](=O)[O-])nn[nH]2 5R-0658 Cc1c(nc2cc(ccc2n1)/N=C/c3cc(cc(c3O)OC)Br)C 5R-0659 Cc1cc(nc2c1c(nn2C)n3cccc3)C 5R-0661 c1cc(oc1)C(=O)OCc2cnc(s2)Cl 5R-0662 c1cc(cc(c1)NC(=O)OCc2cnc(s2)Cl)C(F)(F)F 5R-0663 c1cc(ccc1OCc2cnc(s2)Cl)Cl 5R-0666 Cc1ccc(cc1OCc2cnc(s2)Cl)C(C)C 5R-0667 c1cc(ccc1NC(=O)OCc2cnc(s2)Cl)[N+](=O)[O-] 5R-0668 c1ccc(cc1)/C=C/C(=O)OCc2cnc(s2)Cl 5R-0669 Cc1c(nc2cc(ccc2n1)NC(=O)Nc3ccccc3Cl)C 5R-0670 Cc1c(nc2cc(ccc2n1)NC(=O)Nc3ccc(cc3)OC)C 5R-0672 Cc1cc2c(cc1C)nc(cn2)NC(=O)Nc3cccc(c3)F 5R-0673 Cc1cc(n(n1)Cc2cnc(s2)Cl)C 5R-0674 c1cc(cc(c1)Cl)C(=O)OCc2cnc(s2)Cl 5R-0676 c1ccc2c(c1)ccc(c2C=O)OCc3cnc(s3)Cl 5R-0677 CCc1ccc(cc1)OCc2cnc(s2)Cl 5R-0678 CC(=O)Nc1cccc(c1)OCc2cnc(s2)Cl 5R-0679 c1cc2c(ccc(c2nc1)OCc3cnc(s3)Cl)Cl 5R-0680 c1cc(ccc1CC#N)OCc2cnc(s2)Cl 5R-0681 Cc1ccc2c(c1[N+](=O)[O-])nn[nH]2 5R-0683 CC(C)(C)c1cc(ccc1OCc2cnc(s2)Cl)OC 5R-0684 COc1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)CCN4CCS(=O)(=O)CC4 5R-0685 c1ccc(cc1)CC(=O)OCc2cnc(s2)Cl 5R-0686 Cc1c(nc2cc(ccc2n1)NC(=O)c3ccco3)C 5R-0688 Cc1c(nc2cc(ccc2n1)NS(=O)(=O)c3cccc(c3)C(F)(F)F)C 5R-0689 Cc1c(nc2cc(ccc2n1)NS(=O)(=O)c3cccs3)C 5R-0690 Cc1c(nc2cc(ccc2n1)NS(=O)(=O)c3ccc(cc3)OC)C 5R-0691 c1cc(ccc1NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)F 5R-0800 c1cc(cc(c1)C(F)(F)F)CNC(=O)Cn2cncn2 5R-0801 c1cc(c(cc1NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cl)Oc3ccc(cn3)C(F)(F)F 5R-0802 COc1ccc(cc1)C2CC(=O)CC(=O)C2n3cncn3 5R-0803 c1cc(ccc1CNC(=O)Cn2cnnc2)Cl 5R-0804 Cc1ccc(n1NC(=O)c2ccc(cc2)Cl)C 5R-0806 c1ncn(n1)CC(=O)NCCCN2CCOCC2 5R-0807 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3ccc[n+](c3)C.[I-] 5R-0808 CC(=O)c1ccc(cc1)n2cc(nn2)c3c(c(no3)c4c(cccc4Cl)Cl)C(=O)OC 5R-0809 c1ccc(cc1)CCNC(=O)Cn2cncn2 5R-0811 CNc1nccc(n1)c2cnc(s2)c3ccc(cc3)Cl 5R-0812 Cc1c(sc(n1)c2cccc(c2)Cl)C(=O)C 5R-0813 CC(=O)c1cnc(s1)c2cccc(c2)Cl 5R-0814 Cc1c(sc(n1)c2cccc(c2)Cl)C(=O)/C=C/N(C)C 5R-0815 c1cc(ccc1c2ncc(s2)c3ccncn3)Cl 5R-0816 CN(C)/C=C/C(=O)c1cnc(s1)c2cccc(c2)Cl 5R-0817 Cc1c(sc(n1)c2cccc(c2)Cl)c3ccnc(n3)N 5R-0818 Cc1c(sc(n1)c2cccc(c2)Cl)c3ccn[nH]3 5R-0819 Cc1c(sc(n1)c2ccc[n+](c2)C)C(=O)/C=C/Nc3ccccc3.[I-] 5R-0820 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/Nc3ccc[n+](c3)C.[I-] 5R-0821 COc1ccc(cc1)C2CC(=O)CC(=O)C2c3c(cc(cn3)C(F)(F)F)Cl 5R-0822 c1cc(cc(c1)Cl)c2ncc(s2)c3ccnc(n3)N 5R-0823 CC(=O)Nc1nccc(n1)c2cnc(s2)c3ccc(cc3)Cl 5R-0824 CC(=O)c1ccc(cc1)n2c(c(nn2)CO)CO 5R-0825 Cc1c(c(n2c(c(nc2n1)C#N)C#N)C)Cc3c(cccc3Cl)Cl 5R-0826 c1cc(cc(c1)Cl)C2CC(=O)CC(=O)C2n3cncn3 5R-0827 c1cc(ccc1c2ncc(s2)C(=O)/C=C/Nc3cc(c(cc3N)Cl)Cl)Cl 5R-0828 c1c2c(cc(c1Cl)Cl)nc[nH]2 5R-0829 c1c(cnc(c1Cl)n2c(c(nn2)CO)CO)C(F)(F)F 5R-0830 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)CBr 5R-1001 c1cc(ncc1C(F)(F)F)N2CCC(CC2)(C(=O)N)N3CCCCC3 5R-1002 c1c(cnc(c1Cl)N2CCC(CC2)(C(=O)N)N3CCCCC3)C(F)(F)F 5R-1003 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)CS(=O)(=O)c3ccccc3 5R-1004 c1ccn(c1)c2ccsc2C(=O)OCC#N 5R-1005 Cc1ccc(cc1)SCC(=O)c2c(n3c4ccccc4nc3s2)C 5R-1009 c1ccn(c1)c2ccsc2C(=O)N3CCOCC3 5R-1010 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N\O)/CS(=O)(=O)c3ccccc3 5R-1011 CCNC(=O)c1c(ccs1)n2cccc2 5R-1012 CNC(=O)c1c(ccs1)n2cccc2 5R-1013 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N\OC)/CS(=O)(=O)c3ccccc3 5R-1014 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N\OCc3ccc(cc3)Cl)/CS(=O)(=O)c4ccccc4 5R-1015 c1ccn(c1)c2ccsc2C(=O)NC3CC3 5R-1017 Cc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 5R-1019 c1cc(c(c(c1)Cl)/C=C/C(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl 5R-1020 c1cc(ccc1C(=O)/C=C/c2ccc(cc2Cl)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 5R-1021 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N\OCc3cccc(c3)C(F)(F)F)/CS(=O)(=O)c4ccccc4 5R-1023 Cc1c(sc(n1)c2ccc(cc2)Cl)/C(=N\OCc3ccc(cc3)F)/CS(=O)(=O)c4ccccc4 5R-1024 Cn1ccnc1SC[C@H](C(F)(F)F)O 5R-1061 c1csc(n1)N/C=C/C(=O)C(F)(F)Cl 5R-1062 C1CCC2NCCCN2CC1 5R-1063 c1ccc2c(c1)c(c[nH]2)C(=O)C(F)(F)F 5R-1064 COc1cc(nc(n1)Oc2ccc3ccccc3c2)C(F)(F)F 5R-1121 Cc1c(cno1)C(=O)NC2CCCCC2 5R-1123 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)OC 5R-1125 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)OC(C)C 5R-1126 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)NC(C)C 5R-1127 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)N3CCCC3 5R-1128 Cc1c(cnc(n1)N2CCCC2)C(=O)N3CCCC3 5R-1129 COc1cc(nc(n1)Sc2cccc(c2Cl)Cl)C(F)(F)F 5R-1134 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)Oc3cc(c(cc3Cl)Cl)Cl 5R-1137 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)N3CCOCC3 5R-1139 CC(C)NC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(cc2)OC 5R-1140 COc1ccc(cc1)COC(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC 5R-1141 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)OCc3c(cccc3Cl)Cl 5R-1142 c1cc(ccc1NC(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)Br)Cl 5R-1146 CCOC(=O)c1cnc(nc1Oc2cc(ccc2Cl)Cl)SC 5R-1148 CSc1c(cc2ccccc2n1)C=O 5R-1152 COc1cc(nc(n1)Oc2ccc(c3c2nccc3)Cl)C(F)(F)F 5R-1153 COC(=O)NC1CCN(CC1)S(=O)(=O)c2ccccc2 5R-1156 c1cc(ccc1F)S(=O)(=O)N2CCC(CC2)NC(=O)Nc3ccc(cc3F)F 5R-1157 c1cc(cc(c1)NC(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)F)C(F)(F)F 5R-1158 c1cc(ccc1F)S(=O)(=O)N2CCC(CC2)NC(=O)Nc3ccc(cc3Cl)Cl 5R-1159 CSc1c(cc2ccccc2n1)/C=N/O 5R-1160 Cc1cc(ccc1NC(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)F)Cl 5R-1162 CCOC(=O)c1cnc(nc1Oc2ccc3ccccc3c2)SC 5R-1164 CCOC(=O)c1cnc(nc1Oc2cc(c(cc2Cl)Cl)Cl)SC 5R-1165 CCOC(=O)c1cnc(nc1Oc2ccc(cc2)F)SC 5R-1166 CCOC(=O)c1cnc(nc1Oc2cccc(c2)C(F)(F)F)SC 5R-1167 CCOC(=O)c1cnc(nc1Oc2cccc3c2nccc3)SC 5R-1168 CCOC(=O)c1cnc(nc1Oc2ccc(cc2Cl)Cl)SC 5R-1169 CCOC(=O)c1cnc(nc1Oc2cccc(c2)N)SC 5R-1170 CCOC(=O)c1cnc(nc1Oc2ccc(cc2)NC(=O)C)SC 5R-1171 CSc1c(cc2ccccc2n1)/C=N/OC(=O)c3ccc(c(c3)Cl)Cl 5R-1172 CSc1nc(cc(n1)Oc2ccc(cc2Cl)Cl)C(F)(F)F 5R-1176 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)C=O 5R-1177 Cc1cc(nc2c1c(c(s2)NC(=O)OC)n3cccc3)C 5R-1183 CCOC(=O)Nc1c(c2c(cc(nc2s1)C)C)n3cccc3 5R-1185 Cc1cc(nc2c1c(c(s2)NC(=O)OC(C)C)n3cccc3)C 5R-1186 CCCCOC(=O)Nc1c(c2c(cc(nc2s1)C)C)n3cccc3 5R-1187 Cc1cc(nc2c1c(c(s2)NC(=O)OCc3ccc(cc3)Cl)n4cccc4)C 5R-1188 Cc1cc(nc2c1c(c(s2)NC(=O)OCc3ccc(cc3)Br)n4cccc4)C 5R-1189 Cc1cc(nc2c1c(c(s2)NC(=O)Nc3ccc(cc3)Cl)n4cccc4)C 5R-1191 Cc1cc(nc2c1c(c(s2)NC(=O)Nc3ccccc3)n4cccc4)C 5R-1192 c1ccc(cc1)c2c(cnn2c3c(cc(cc3Cl)Cl)Cl)NC(=O)OCc4ccc(cc4)Cl 5R-1194 c1ccc(cc1)c2c(cnn2c3c(cc(cc3Cl)Cl)Cl)NC(=O)OCc4ccc(cc4)Br 5R-1195 Cc1cc(nc2c1c(c(s2)NC(=O)OCc3ccccc3)n4cccc4)C 5R-1197 Cc1cc(nc2c1c(c(s2)NC(=O)OCc3ccc(cc3)C(C)(C)C)n4cccc4)C 5R-1198 Cc1cc(nc2c1c(c(s2)NC(=O)OCc3ccc(cc3)OC)n4cccc4)C 5R-1201 Cc1cc(nc2c1c(c(s2)NC(=O)Nc3ccc(cc3)Br)n4cccc4)C 5R-1205 Cc1cc(cc(c1)NC(=O)Nc2c(c3c(cc(nc3s2)C)C)n4cccc4)C 5R-1208 Cc1cc(nc2c1c(c(s2)NC(=O)Nc3cccc(c3)C(F)(F)F)n4cccc4)C 5R-1210 Cc1ccccc1NC(=O)Nc2c(c3c(cc(nc3s2)C)C)n4cccc4 5R-1212 Cc1cc(nc2c1c(c(s2)NC(=O)Nc3ccc(cc3)F)n4cccc4)C 5R-1213 Cc1ccc(cc1)c2nnc(o2)/C=C/c3ccccc3 5R-1240 c1ccc(cc1)/C=C/c2nnc(o2)c3ccccc3 5R-1241 Cc1ccc(cc1)CSc2nnc(n2c3ccc(cc3)Cl)/C=C/c4ccccc4 5R-1243 c1ccc(cc1)/C=C/c2nnc(n2c3ccc(cc3)Cl)SCc4ccc(cc4)Cl 5R-1244 c1ccc(cc1)/C=C/c2nnc(o2)SCc3ccccc3Cl 5R-1245 c1ccc(cc1)/C=C/c2nnc(o2)SCc3cccc(c3)[N+](=O)[O-] 5R-1247 c1ccc(cc1)/C=C/c2nnc(o2)SCc3c(cccc3Cl)Cl 5R-1248 c1ccc(cc1)CSc2nnc(o2)/C=C/c3ccccc3 5R-1249 Cc1cccc(c1)CSc2nnc(o2)/C=C/c3ccccc3 5R-1250 COC(=O)c1ccc(cc1)CSc2nnc(o2)/C=C/c3ccccc3 5R-1251 c1ccc(cc1)/C=C/c2nnc(o2)SCC(=O)c3ccc(cc3)F 5R-1252 Cc1cccc(c1)c2nnc(o2)/C=C/c3ccccc3 5R-1254 c1ccc(cc1)/C=C/c2nnc(n2c3ccc(cc3)Cl)SCc4ccccc4Cl 5R-1256 CCn1c(nnc1SC)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC 5R-1300 CCn1c(nnc1SC(C)C)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC 5R-1301 CCn1c(nnc1SCc2ccc(cc2)F)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)OC 5R-1302 CCn1c(nnc1SCc2ccccc2)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)OC 5R-1303 COC(=O)C1CSC(N1C(=O)c2ccccc2)c3ccc(cc3)Cl 5R-1305 COc1ccc(cc1)C(=O)N2C(CSC2c3ccc(cc3)Cl)C(=O)OC 5R-1306 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCC=C)O)C 5R-1307 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCC=C)Cl)C 5R-1308 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)N5CCCC5)C)C 5R-1310 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCC=C)N4CCOCC4)C 5R-1311 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCC=C)NC4CC4)C 5R-1312 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)NCC=C)C)C 5R-1313 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)Sc5ccc(cc5)C)C)C 5R-1314 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)Sc5ccccc5)C)C 5R-1315 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)SCc5ccc(cc5)Cl)C)C 5R-1316 CC(=O)N1C(CC(=O)CC1(C)C)(C)C 5R-1317 CC(=O)N1C(CC(=NO)CC1(C)C)(C)C 5R-1318 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCC=C)Sc4ccc(cc4)Cl)C 5R-1320 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCC=C)Sc4cccc(c4)OC)C 5R-1321 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)Sc5ccccc5C(=O)OC)C)C 5R-1322 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccccc4)O)C 5R-1325 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccc(cc4)Cl)O)C 5R-1326 CCSc1nc2c3c(cc(nc3sc2c(n1)O)C)C 5R-1327 CC(=O)NC(C(=O)NCc1ccccc1)C(=O)Nc2ccc(cc2)OC 5R-1501 CC(=O)NC(C(=O)Nc1ccc(cc1)OC)C(=O)OCC(=O)c2ccc(cc2)Cl 5R-1502 c1ccc2c(c1)nc(n2CC(=O)N3CCN(CC3)c4ccc(cc4)F)C(F)(F)F 5R-1504 c1ccc(cc1)N2CCN(CC2)C(=O)Cn3c4ccccc4nc3C(F)(F)F 5R-1505 CN1CCN(CC1)C(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1506 Cc1ccc(cc1)Oc2c(nnc(n2)c3ccccc3)C(F)(F)F 5R-1507 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Oc3cccc(c3)C(F)(F)F 5R-1509 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)N3CCCC3 5R-1510 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)N3CCCCC3 5R-1511 C=CCNC(=O)Cn1c2ccccc2nc1C(F)(F)F 5R-1512 CC(C)(C)NC(=O)Cn1c2ccccc2nc1C(F)(F)F 5R-1513 CNC(=O)Cn1c2ccccc2nc1C(F)(F)F 5R-1514 CN(c1c(nnc(n1)c2ccccc2)C(F)(F)F)N 5R-1515 COc1c(nnc(n1)c2ccccc2)C(F)(F)F 5R-1516 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Oc3ccc(cc3Cl)Cl 5R-1517 c1ccc(cc1)c2nc(c(nn2)C(F)(F)F)Oc3ccc(cc3)F 5R-1518 CC(C)NC(=O)Cn1c2ccccc2nc1C(F)(F)F 5R-1520 COC(=O)c1ccccc1NC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1521 c1ccc(c(c1)C(=O)O)NC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1525 CCN(CC)CCNc1c(nnc(n1)c2ccccc2)C(F)(F)F 5R-1526 CN(C)CCNc1c(nnc(n1)c2ccccc2)C(F)(F)F 5R-1528 CCN1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 5R-1529 CCN1CCN(CC1)c2ccc(cc2)N 5R-1532 Cc1cccc(c1)OC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1533 Cc1ccccc1OC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1534 Cc1ccc(cc1)OC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1535 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2cccnc2Cl 5R-1536 CN(c1c(nnc(n1)c2ccccc2)C(F)(F)F)NC(=O)c3ccc(cc3)OC 5R-1538 CN(c1c(nnc(n1)c2ccccc2)C(F)(F)F)NC(=O)c3ccc(cc3)Cl 5R-1539 Cc1ccc(cc1)C(=O)NN(C)c2c(nnc(n2)c3ccccc3)C(F)(F)F 5R-1540 COC(=O)c1ccccc1OC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1542 c1ccc2c(c1)nc(n2CC(=O)Oc3ccc(cc3)C#N)C(F)(F)F 5R-1543 CC(C)c1ccc(cc1)NC(=O)C(C(=O)O)NC(=O)C 5R-1544 CC(=O)NC(C(=O)NCc1ccc(cc1)OC)C(=O)Nc2ccc(cc2)OC 5R-1545 CC(=O)NC(C(=O)NCc1ccccc1Cl)C(=O)Nc2ccc(cc2)OC 5R-1546 CC(=O)NC(C(=O)NCc1ccccc1OC)C(=O)Nc2ccc(cc2)OC 5R-1547 CC(=O)NC(C(=O)NCc1ccc(cc1)F)C(=O)Nc2ccc(cc2)OC 5R-1548 CC(=O)NC(C(=O)Nc1ccc(cc1)OC)C(=O)N2CCOCC2 5R-1549 CC(C)c1ccc(cc1)NC(=O)C(C(=O)NCc2ccccc2)NC(=O)C 5R-1550 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 5R-1552 CC(=O)Nc1ccc(cc1)OC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1553 CC(C)(C)c1ccc(cc1)OC(=O)Cn2c3ccccc3nc2C(F)(F)F 5R-1554 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cccn2)C(=O)Nc3ccc(cc3)OC 5R-1555 CC(C)(C)OC(=O)N1CCN(CC1)c2c(c(nc(n2)c3ccncc3)c4ccc(cc4)Cl)C#N 5R-1556 CN(c1c(nnc(n1)c2ccccc2)C(F)(F)F)NC(=O)c3cccc(c3)Cl 5R-1557 Cc1cccc(c1)C(=O)NN(C)c2c(nnc(n2)c3ccccc3)C(F)(F)F 5R-1558 CC(C)c1ccc(cc1)NC(=O)C(C(=O)NCc2ccc(cc2)OC)NC(=O)C 5R-1560 CC(C)c1ccc(cc1)NC(=O)C(C(=O)NCc2ccc(cc2)Cl)NC(=O)C 5R-1561 Cc1c(nc(nn1)c2ccc(cc2)Cl)NCCN(C)C 5R-1565 CN(c1c(nnc(n1)c2ccccc2)C(F)(F)F)NC(=O)CCl 5R-1568 CC(C)CC(=O)NN(C)c1c(nnc(n1)c2ccccc2)C(F)(F)F 5R-1569 CC(C)(C)C(=O)NN(C)c1c(nnc(n1)c2ccccc2)C(F)(F)F 5R-1570 c1ccc2c(c1)nc(n2CC(=O)Oc3ccc(cc3Cl)Cl)C(F)(F)F 5R-1571 c1ccc2c(c1)nc(n2CC(=O)Oc3cc(ccc3Cl)Cl)C(F)(F)F 5R-1572 CCCCC(=O)NN(C)c1c(nnc(n1)c2ccccc2)C(F)(F)F 5R-1573 Cc1ccc(c(c1)OC(=O)Cn2c3ccccc3nc2C(F)(F)F)C(C)C 5R-1574 Cc1c(nc(nn1)c2ccc(cc2)Cl)OC 5R-1578 COc1ccc(cc1)Cn2c3c(c(c2N)C#N)CCCC3 5T-0002 CCOC(=O)C(=CNc1ccnn1C)C(=O)OCC 5T-0006 CCOC(=O)c1cnc2c(c1Cl)cnn2C 5T-0007 c1cc(ccc1c2csc(n2)n3c(ccn3)c4ccc(cc4Cl)Cl)Cl 5T-0008 c1cc(sc1)c2csc(n2)n3c(ccn3)c4ccc(cc4Cl)Cl 5T-0009 COc1ccc(cc1)c2csc(n2)n3c(ccn3)c4ccc(cc4Cl)Cl 5T-0010 c1cc(ccc1c2csc(n2)n3c(ccn3)c4ccc(cc4Cl)Cl)F 5T-0011 COc1ccc(cc1)c2csc(n2)n3c(ccn3)c4ccccc4 5T-0012 c1ccc(cc1)c2ccnn2c3nc(cs3)c4ccc(cc4)F 5T-0013 c1ccc(cc1)c2ccnn2c3nc(cs3)c4cccs4 5T-0014 c1ccc(cc1)c2ccnn2c3nc(cs3)c4ccccc4 5T-0015 CCCCc1c(onc1O)C 5T-0019 CCOC(=O)c1cnn(c1NC(=S)NC(C)(C)C)C 5T-0021 CCOC(=O)/C(=C/Nc1ccnn1C)/C#N 5T-0022 c1cc(ccc1c2cnn(c2)c3nc(c(s3)Sc4ccc(cc4)Cl)c5ccc(cc5Cl)Cl)Cl 5T-0027 Cc1cc(n2c(n1)c3ccc(nc3n2)c4ccc(c(c4)Cl)Cl)C(F)(F)F 5T-0032 CN1C(=O)C(=Cc2ccc3c(c2)OCCO3)C(=O)N(C1=O)C 5T-0034 CCOC(=O)c1cnc2cc(nn2c1CCl)C 5T-0035 COC(=O)CSc1nccc(n1)c2cccs2 5T-0041 c1cc(oc1)c2ccnc(n2)N 5T-0042 c1ccn2cc(nc2c1)C(=O)NN 5T-0043 CN1C(=O)C(=Cc2ccc(cc2)SC)C(=O)N(C1=O)C 5T-0044 c1ccc2c(c1)/C(=C/c3cc(cs3)Br)/C(=O)N2 5T-0045 c1cnc2nc(c(n2c1)Cl)c3ccc(cc3)Cl 5T-0046 CN1c2ccccc2C(C1CCc3ccccc3)(C(F)(F)F)O 5T-0047 CN1C(=O)C(C(=O)N(C1=O)C)Cc2ccc(cc2)SC 5T-0049 c1ccc2c(c1)c(cn2Cc3cnc(s3)Cl)C=O 5T-0050 COC(=O)c1ccc(cc1)Oc2ccc3c(c2)nc(c(n3)c4ccccc4)c5ccccc5 5T-0200 c1ccc2c(c1)ncn2c3ccc(cc3)c4ccnc5n4ncc5C#N 5T-0201 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)NC4CCCC4 5T-0202 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)NCc4cccs4 5T-0204 CC(C1(OCCO1)C)Oc2ccc(cc2)[N+](=O)[O-] 5T-0207 CCc1c(nc2cc(ccc2n1)Oc3ccc(cc3)C(=O)OC)CC 5T-0208 COc1ccc(cc1)c2cnc3ncnn3c2c4ccc(cc4)OC 5T-0209 Cc1cc2ncc(c(n2n1)c3ccc(cc3)OC)c4ccc(cc4)OC 5T-0210 CCCCCCCc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=C2C(=O)OC)C 5T-0211 COc1ccc2c(c(=O)ncn2n1)c3c(cccc3Cl)Cl 5T-0212 COc1ccc(cc1)c2cnc(nc2c3ccc(cc3)OC)N 5T-0214 c1ccc2c(c1)ncn2c3ccc(cc3)C(=O)/C=C/Nc4ccc(cc4)C(F)(F)F 5T-0216 Cc1ccc(cc1)c2cn(c(n2)SCc3ccc(cc3)C(F)(F)F)CC(=O)c4ccc(cc4)C 5T-0218 c1cc(cc(c1)F)COc2cc(c(cc2Cl)Cl)NC(=O)C3CC3 5T-0219 COc1ccc(cc1)/C(=C\Nc2ccc(cc2)C(F)(F)F)/C(=O)c3ccc(cc3)OC 5T-0220 CCOC(=O)COc1ccccc1C=O 5T-0221 COc1ccc(cc1)c2c[nH]nc2c3ccc(cc3)OC 5T-0224 c1ccc2c(c1)C(=O)C(=Cc3ccc4c(c3)c(on4)c5ccc(cc5)F)C2=O 5T-0225 CCCN1c2ccccc2OCC1=O 5T-0226 c1ccc(cc1)OC(=O)Nc2ccc(cc2)CSc3ccccc3 5T-0228 c1cc(ccc1C(=O)n2c(ccn2)c3ccc4c(c3)OCO4)F 5T-0229 CC(C)(C)c1ccc(cc1)C(=O)n2c(ccn2)c3ccc4c(c3)OCO4 5T-0230 c1cc(cc(c1)C(F)(F)F)C(=O)n2c(ccn2)c3ccc4c(c3)OCO4 5T-0231 CCOC(=O)/C(=C\c1ccc2c(c1)c(on2)c3ccc(cc3)F)/C#N 5T-0232 Cc1cccc(c1)C(=O)Nc2cc(c(cc2Cl)Cl)OCc3cccc(c3)F 5T-0236 COc1ccc(cc1)c2cnc(nc2c3ccc(cc3)OC)c4ccccn4 5T-0237 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)C(=O)c4ccc(cc4)Br 5T-0238 c1ccc2c(c1)cccc2C=C3C(=O)c4ccccc4C3=O 5T-0240 CCCCCCCc1ccc(cc1)c2c(c(nc-3c2C(=O)c4c3cccc4)/C=C(\C)/N(C)C)C#N 5T-0241 CCCCCCCc1ccc(cc1)c2c(c(nc-3c2C(=O)c4c3cccc4)/C=C/c5cccc(c5)Cl)C#N 5T-0242 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)C(=O)OCc4cncs4 5T-0243 c1ccc(cc1)SCc2ccc(cc2)NC(=O)N3CCc4c3cccc4 5T-0244 CCCCCCCc1ccc(cc1)c2c(c(nc-3c2C(=O)c4c3cccc4)/C=C(\C)/Nc5ccccc5F)C#N 5T-0245 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)S(=O)(=O)c4ccc(cc4)I 5T-0246 Cc1c(cnc2n1ncc2C#N)C(=O)OCc3ccccc3 5T-0249 CN1CCN(CC1)c2ccc(cc2)NC(=O)Oc3ccccc3 5T-0251 Cc1ccccc1C(=O)n2cc(c(n2)c3ccc(cc3)OC)c4ccc(cc4)OC 5T-0252 CC(C)(C)c1ccc(cc1)C(=O)n2cc(c(n2)c3ccc(cc3)OC)c4ccc(cc4)OC 5T-0253 CCOC(=O)C1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 5T-0254 c1ccc(cc1)SCc2ccc(cc2)NC(=O)N3CCCC3C(=O)O 5T-0258 Cc1c(cnc2n1ncc2C#N)C(=O)O 5T-0259 COc1cccc(c1)/C=C/2\CCCc3ccccc3C2=O 5T-0260 CC1C(c2cc3c(cc2OC1(C)N4CCCC4)OCO3)c5cccc6c5cccc6 5T-0262 CC1C(c2cc3c(cc2OC1(C)O)OCO3)c4cccc5c4cccc5 5T-0263 C/C(=N\c1c(cn[nH]1)C#N)/C2CCOC2=O 5T-0264 c1cc(c(cc1C(c2cc3c(cc2O)OCO3)N4CCCC4)Cl)Cl 5T-0267 CCC(C(=O)OCC)Oc1ccccc1C=O 5T-0268 CN1CCN(CC1)c2ccc(cc2)NC(=O)N3CCc4c3cccc4 5T-0269 CCOc1ccccc1C(c2cc3c(cc2O)OCO3)N4CCCC4 5T-0270 CCOc1ccccc1C2c3cc4c(cc3OC(C2C)(C)N5CCCC5)OCO4 5T-0271 CC1C(c2cc3c(cc2OC1(C)N4CCCC4)OCO3)c5ccc(c(c5)Cl)Cl 5T-0272 CCCCCCCc1ccc(cc1)c2c(c(nc-3c2C(=O)c4c3cccc4)/C=C/Nc5c(cccc5C)C)C#N 5T-0274 COc1cccc(c1)C2C3=C(c4ccccc4CCC3)NC(=S)N2 5T-0275 Cc1cc(=O)n(c(=O)[nH]1)c2ccc(cc2)Cl 5T-0276 c1cc(ccc1n2c(=O)cc([nH]c2=O)C(F)(F)F)Cl 5T-0277 Cc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)n3cncn3 5T-0279 CC1C(c2cc3c(cc2OC1(C)O)OCO3)c4ccc(c(c4)Cl)Cl 5T-0281 CCOc1ccccc1C2c3cc4c(cc3OC(C2C)(C)O)OCO4 5T-0282 Cc1ccsc1/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccccc5F)C#N 5T-0283 Cc1c(c(=O)n2c([nH]1)c(cn2)C#N)CCO 5T-0284 CCOC(=O)C1CCN(CC1)c2ccc(c(c2)N)[N+](=O)[O-] 5T-0285 c1cc(ccc1c2ccn(n2)CCO)n3cncn3 5T-0287 c1cc(ccc1c2ccnc3n2ncn3)n4cncn4 5T-0288 Cc1cc2nccc(n2n1)c3ccc(cc3)n4cncn4 5T-0290 c1ccc(c(c1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)NC(=O)CO4)Cl 5T-0291 Cc1c(cnc2n1c3ccccc3n2)C(=O)O 5T-0293 Cc1c(c(n2c(n1)c(cn2)C#N)Cl)CCCl 5T-0294 c1ccnc(c1)c2nccc(n2)c3ccc(cc3)n4cncn4 5T-0295 Cc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)N3CCN(CC3)C 5T-0296 Cc1nccc(n1)c2ccc(cc2)n3cncn3 5T-0297 c1ccc2c(c1)nc3n2c(ccn3)c4ccc(cc4)n5cncn5 5T-0298 CCOC(=O)C1CCN(CC1)C(=O)c2ccc(cc2)Cl 5T-0299 CCOC(=O)C1CCN(CC1)C(=O)c2ccc(cc2)OC 5T-0300 c1ccc(cc1)n2c(=O)cc([nH]c2=S)C(F)(F)F 5T-0301 CN(C)c1ccc(cc1)/C=C/2\CCCc3ccccc3C2=O 5T-0302 CN1CCN(CC1)c2ccc(cc2)c3cc[nH]n3 5T-0303 Cc1c(sc(c1c2ccccc2)C(=O)N)C#N 5T-0305 C/C(=N\c1[nH]c2ccccc2n1)/C3CCOC3=O 5T-0306 CC1C(c2cc3c(cc2OC1(C)OC)OCO3)c4cccc5c4cccc5 5T-0307 c1ccnc(c1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)NC(=O)CO4 5T-0308 CCOC(=O)C1CCN(CC1)c2ccc(c(c2)C(=O)N)[N+](=O)[O-] 5T-0309 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)C(=O)c4ccc(cc4)F 5T-0310 CCCN1c2cc(ccc2OCC1=O)C(=O)c3ccccc3C(=O)O 5T-0312 CC(C)Sc1nc(cc(=O)n1c2ccccc2)C(F)(F)F 5T-0313 COc1ccc(c(c1)C(c2cc3c(cc2O)OCO3)N4CCCC4)OC 5T-0315 Cc1ccc(cc1)Cn2cc(c(n2)c3ccc(cc3)OC)c4ccc(cc4)OC 5T-0316 CCCN1c2cc(ccc2OCC1=O)c3c4ccccc4c(=O)[nH]n3 5T-0318 c1ccc2c(c1)N(C(=O)CO2)Cc3c(cccc3Cl)F 5T-0319 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)CCO 5T-0320 CC1C(c2cc3c(cc2OC1(C)O)OCO3)c4cc(ccc4OC)OC 5T-0323 CC1C(c2cc3c(cc2OC1(C)OC)OCO3)c4cc(ccc4OC)OC 5T-0324 CC(C)(C)c1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)N4CCN(CC4)C 5T-0326 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)C(=O)c4cccc(c4)C(F)(F)F 5T-0327 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)C(=O)c4cccs4 5T-0328 CCn1c(=O)cc([nH]c1=S)C(F)(F)F 5T-0329 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)Cc4ccc(c(c4)Cl)Cl 5T-0330 COc1ccc(cc1)c2cnc3c(cnn3c2c4ccc(cc4)OC)C#N 5T-0332 COc1ccc(cc1)c2cn(nc2c3ccc(cc3)OC)CCOc4ccc(cn4)C(F)(F)F 5T-0333 COc1ccc(cc1)C(=O)Nc2cccc(c2)c3cn4c5ccccc5sc4n3 5T-0600 Cc1ccn2cc(nc2c1)c3cccc(c3)NS(=O)(=O)c4ccc(cc4)F 5T-0601 c1cc(cc(c1)NC(=O)c2ccco2)c3cn4cc(ccc4n3)I 5T-0602 COc1cccc2c1oc(c2)c3ccnc(n3)N 5T-0603 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(cc3)Cl 5T-0604 c1ccn2cc(nc2c1)c3cccc(c3)NC(=O)CC(c4ccc(cc4)Cl)NC(=O)C(F)(F)F 5T-0606 CC(=O)c1cc2c3ccccc3ccc2o1 5T-0607 c1cc(n(c1)c2nccs2)C=C(C#N)C#N 5T-0609 c1ccc(c(c1)N/N=C/c2cccn2c3nccs3)F 5T-0610 Cc1ccn2cc(nc2c1)c3cccc(c3)NC(=O)C4CCCCC4 5T-0611 c1ccn2c(c1)nc(c2C=O)c3ccc(cc3)[N+](=O)[O-] 5T-0612 c1ccc2c(c1)nc(s2)NC(=O)CC(c3ccc(cc3)Cl)NC(=O)C(F)(F)F 5T-0614 CC(c1ccc(cc1)n2cccc2)O 5T-0617 C=CCSc1nccc(n1)c2cccs2 5T-0618 c1cc(sc1)c2ccnc(n2)SCc3cnc(s3)Cl 5T-0619 CCCCCC(=O)Nc1ccc(cc1)c2cn3cccnc3n2 5T-0620 c1cc(cc(c1)NS(=O)(=O)c2cccs2)c3cn4cc(ccc4n3)I 5T-0621 c1cc(ccc1C#N)OC(=O)CC(c2ccc(cc2)Cl)NC(=O)C(F)(F)F 5T-0622 CCOC(=O)c1cn2c3ccccc3sc2n1 5T-0623 c1cc(sc1)c2ccnc(n2)SCc3ccc(cc3)Cl 5T-0625 CCOc1ccc2c(c1)sc3n2cc(n3)C(=O)OCC 5T-0627 CCOC(=O)c1cn2ccccc2n1 5T-0628 COc1ccc(cc1)SCc2cnc(s2)Cl 5T-0631 Cc1cc(c(cc1N2CCN(CC2)c3ccccc3)N)[N+](=O)[O-] 5T-0633 Cc1ccc(n1c2ccc(cc2)C(=O)C)C 5T-0635 c1cc(n(c1)c2nccs2)/C=C\3/C(=O)NC(=O)S3 5T-0636 c1cc2c(cc1[N+](=O)[O-])c(=O)[nH]cn2 5T-0638 c1cc(n(c1)c2nccs2)/C(=N/O)/N 5T-0639 c1cc(cc(c1)N)c2cn3cc(ccc3n2)Cl 5T-0640 c1ccc(c(c1)C#N)n2cccc2 5T-0643 c1ccc2c(c1)N=CC=C(S2)c3cccnc3 5T-0645 c1cc(ccc1c2ncc(s2)c3ccnc(n3)N)F 5T-0653 c1cc(cc(c1)F)c2ncc(s2)c3ccnc(n3)N 5T-0654 CCOC(=O)/C(=C\c1ccc(cc1)Cl)/C#N 5T-0658 CCOC(=O)C1=C(N(C(=C(C1c2ccc(cc2)Cl)C(=O)OCC)N)c3ccc(cc3)Cl)C 5T-0659 COC(=O)Cc1c(nc(s1)N2CCOCC2)c3ccccc3 5T-0801 CS(=O)(=O)c1cnc2c(cnn2c1N)S(=O)(=O)c3ccccc3 5T-0802 CC(C)(C)S(=O)(=O)c1cnc2c(cnn2c1N)S(=O)(=O)c3ccccc3 5T-0803 Cc1cc(n2c(n1)c(cn2)S(=O)(=O)c3ccccc3)C(F)(F)F 5T-0804 c1ccc(cc1)c2ccc(cc2)c3csc(n3)n4c(c(cn4)c5ccsc5)N 5T-0806 c1ccc(cc1)c2ccc(cc2)c3csc(n3)n4c(c(cn4)c5cccs5)N 5T-0807 Cc1cc(n(n1)c2nc(cs2)c3cccs3)C 5T-0808 COc1cc2c(cc1OC)C3Cc4c(cnn4S(=O)(=O)c5ccc(cc5)Cl)C(=O)N3CC2 5T-0811 COC(=O)c1cc(n2c(n1)ncn2)c3cccc(c3)OCc4ccccc4 5T-0813 Cc1cc(nc(n1)n2cc(nn2)C(=O)c3ccc(cc3Cl)Cl)c4ccccc4 5T-0814 c1ccc(cc1)c2cc(n3c(n2)c(cn3)S(=O)(=O)c4ccccc4)C(F)(F)F 5T-0816 COc1ccc(cc1)c2cc(n3c(n2)c(cn3)S(=O)(=O)c4ccccc4)C(F)(F)F 5T-0817 COc1ccccc1c2cc(n3c(n2)c(cn3)S(=O)(=O)c4ccccc4)C(F)(F)F 5T-0818 CC(=O)c1cnc(s1)c2ccc(cc2)F 5T-0821 CC(=O)c1cnc(s1)c2cccc(c2)F 5T-0822 c1cnn(c1)C(=S)N 5T-0826 COc1ccc(cc1)c2c(sc(n2)N3CCN(CC3)c4ccc(cc4)OC)Sc5ccc(cc5)Cl 5T-0827 COc1ccc(cc1)N2CCN(CC2)c3[nH+]c(cs3)C(F)(F)F.[Br-] 5T-0828 c1cc(ccc1CSc2nnc(s2)N)F 5T-0829 CC(C)(C)NC(=S)N1CCN(CC1)C 5T-0830 Cc1cc2nc(c(c(n2n1)C)C/C=C/c3ccccc3)C 5T-0832 CC(=O)c1ccc(s1)N2CCN(CC2)C 5T-0834 CC(C)(C)c1ccc(cc1)Oc2cccc(c2)/C=C/C(=O)/C=C/N(C)C 5T-0835 Cc1c(c(n2c3ccccc3nc2n1)C)C/C=C/c4ccccc4 5T-0836 CCOC(=O)c1cnn2c1nc(c(c2C)C/C=C/c3ccccc3)C 5T-0837 c1cc(ccc1NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3 5T-0838 Cc1c(nn(c1C)c2nc(cs2)c3ccccc3)C 5T-0840 Cc1c(nn(c1C)c2nc(cs2)c3ccc(cc3)OC)C 5T-0841 Cc1c(nn(c1C)c2nc(cs2)c3cccs3)C 5T-0842 COc1cc2c(cc1OC)C3Cc4c(cnn4c5cc(ccc5Cl)Cl)C(=O)N3CC2 5T-0843 Cc1ccc(cc1)CSc2[nH]c(nn2)N 5T-0844 c1ccc(cc1)S(=O)(=O)c2cnn3c2nccc3c4ccc(o4)c5ccc(cc5Cl)Cl 5T-0846 Cc1cc2ncc(c(n2n1)N)S(=O)(=O)c3ccccc3 5T-0847 c1ccc(cc1)S(=O)(=O)c2cnc3c(cnn3c2N)c4ccsc4 5T-0848 COc1ccc(cc1)c2c(sc(n2)N)Sc3ccc(cc3)Cl 5T-0849 COc1ccc(cc1)N2CCN(CC2)c3nc(cs3)c4ccc(cc4)c5ccccc5 5T-0850 CC(C)(C)S(=O)(=O)c1cnc2c(cnn2c1N)c3ccsc3 5T-0851 COc1cccc(c1)CSc2nnc(s2)N 5T-0852 COC(=O)C1C2c3ccccc3CCN2C(=O)C=C1O 5T-0855 COc1ccc(cc1)n2c3c(cn2)C(=O)N4CCc5cc(c(cc5C4C3)OC)OC 5T-0856 c1cc(cc(c1)F)CSc2nnc(s2)N 5T-0857 CC(=O)Nc1nnc(s1)C(F)(F)F 5T-0858 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)N)c5ccccn5)C 5T-0859 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)N 5T-0860 c1c(sc(n1)Cl)CSc2nnc(s2)N 5T-0861 CC(C)(C)S(=O)(=O)c1cnc2nc(nn2c1N)N3CCN(CC3)C(c4ccccc4)c5ccccc5 5T-0862 CC(C)(C)S(=O)(=O)c1cnc2cc(nn2c1N)c3cnn(c3C(F)(F)F)C 5T-0863 Cn1c(c(cn1)c2cc3ncc4c(n3n2)CC5c6cc(c(cc6CCN5C4=O)OC)OC)C(F)(F)F 5T-0864 Cc1c(nc2c(cnn2c1C)S(=O)(=O)c3ccccc3)C 5T-0867 CC(C)(C)S(=O)(=O)c1cnc2c(cnn2c1N)c3ccccn3 5T-0868 c1ccnc(c1)c2cnn(c2N)c3nc(cs3)c4ccc(cc4)Cl 5T-0870 CCOC(=O)c1cnc2c(c(nn2c1C(F)(F)F)C)Br 5T-0871 CCOC(=O)c1cnc2c(c(nn2c1C(F)(F)F)C)Cl 5T-0873 Cc1cc2ncc(c(n2n1)N)c3ccccn3 5T-0874 CN(C)c1ccc(cc1)C2CC(=O)C=C(C2n3cncn3)O 5T-0881 c1cc(ccc1C2CC(=O)C=C(C2n3cncn3)O)F 5T-0882 CC(C)(C)c1ccc(cc1)Oc2cccc(c2)/C=C/c3ccnc4n3ncn4 5T-0885 CC(C)Oc1cccc(c1)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 5T-0886 Cc1c(c(n2c(n1)nnn2)C)C/C=C/c3ccccc3 5T-0887 COCc1cc(n2c(n1)c(cn2)S(=O)(=O)c3ccccc3)O 5T-0888 COc1cccc(c1)c2cc(n3c(n2)c(cn3)S(=O)(=O)c4ccccc4)C(F)(F)F 5T-0889 c1ccc(cc1)c2cc(on2)CNC=O 5T-0890 Cn1c(c(cn1)c2cc3ncc(c(n3n2)N)S(=O)(=O)C)C(F)(F)F 5T-0891 COc1cc2c(cc1OC)C3Cc4c(cnn4c5ccc(cc5)C#N)C(=O)N3CC2 5T-0892 COc1cc2c(cc1OC)C3Cc4c(cnn4c5ccc(cc5)C(F)(F)F)C(=O)N3CC2 5T-0893 c1cc(ccc1C#N)n2c(ccn2)c3cnc4n(c3=O)CCS4 5T-0895 c1cc(ccc1n2c(ccn2)c3cnc4n(c3=O)CCS4)F 5T-0896 c1cc(cc(c1)Cl)n2c(ccn2)c3cnc4n(c3=O)CCS4 5T-0897 c1ccc(c(c1)n2c(ccn2)c3cnc4n(c3=O)CCS4)F 5T-0898 Cc1cc(n(n1)c2nc(cs2)C(=O)N/N=C/c3ccc(cc3)F)C(F)(F)F 5T-0900 c1cc(ccc1c2csc(n2)N=C(N)N)Cl 5T-0906 C/C(=N\Nc1nc(cs1)c2ccc(cc2)Cl)/c3ccc(cc3)OC 5T-0907 C/C(=N/Nc1nc(cs1)c2ccc(cc2)Cl)/c3ccc4ccccc4c3 5T-0909 C/C(=N/Nc1nc(cs1)c2ccc(cc2)Cl)/c3cccs3 5T-0910 C/C(=N/Nc1nc(cs1)c2ccc(cc2)Cl)/c3ccncc3 5T-0911 Cc1cc(n2c(n1)cc(n2)c3cnn(c3C(F)(F)F)C)C(F)(F)F 5T-0913 Cn1c(c(cn1)c2cc3nc(cc(n3n2)C(F)(F)F)C(F)(F)F)C(F)(F)F 5T-0914 Cc1cc([nH]n1)NC(=O)C2C3c4ccccc4CCN3C(=O)C=C2O 5T-0916 Cc1cc(n2c(n1)cc(n2)c3cnn(c3C(F)(F)F)C)C(F)(F)Cl 5T-0917 c1ccc(cc1)c2csc(n2)N=C(N)N 5T-0918 Cc1cc(n2c(n1)c(c(n2)c3cnn(c3C(F)(F)F)C)Cl)C(F)(F)Cl 5T-0922 c1cc(sc1)c2ccnc3n2ncc3c4ccsc4 5T-0923 Cc1c(c2ncc(c(n2n1)C(F)(F)F)C(=O)O)Cl 5T-0926 c1c(c(c(=O)[nH]n1)Br)N2CCCC2 5T-1482 c1cc(c(cc1Cl)n2c(=O)c(c(cn2)Br)Br)Cl 5T-1484 CC(=O)OCn1c(=O)c(c(cn1)Cl)Cl 5T-1486 COc1ccc(cc1)Oc2cnn(c(=O)c2Br)c3ccccc3 5T-1487 CC(=O)OCn1c(=O)c(c(cn1)N2CCN(CC2)c3ccccc3)Br 5T-1494 COc1ccc(cc1)Oc2cnn(c(=O)c2Br)c3cc(ccc3Cl)Cl 5T-1495 c1cc(ccc1c2ncc(s2)c3c(cnc(n3)N)Br)F 5T-9001 c1cc(cc(c1)F)c2ncc(s2)c3c(cnc(n3)N)Br 5T-9003 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)c3c(cnc(n3)N)Br 5T-9004 Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)c3c(cnc(n3)N)Br 5T-9005 Cc1c(sc(n1)c2ccc(cc2)F)c3c(cnc(n3)N)Cl 5T-9006 c1cc(ccc1c2ncc(s2)c3c(cnc(n3)N)Cl)F 5T-9007 c1cc(cc(c1)F)c2ncc(s2)c3c(cnc(n3)N)Cl 5T-9009 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)c3c(cnc(n3)N)Cl 5T-9010 Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)c3c(cnc(n3)N)Cl 5T-9011 c1ccc(cc1)c2nc(c(s2)c3ccnc(n3)N)Cl 5T-9032 CSCc1cnc(s1)Cl 5W-0006 c1ccc(cc1)SCc2cnc(s2)Cl 5W-0007 c1ccc2cc(ccc2c1)SCc3cnc(s3)Cl 5W-0013 c1ccc(cc1)CSCc2cnc(s2)Cl 5W-0015 c1c(c(cnc1Cl)Cl)CO 5W-0016 c1cc(ccc1C(=O)O)SCc2cnc(s2)Cl 5W-0025 COC(=O)C(c1ccc(cc1[N+](=O)[O-])Br)C(=O)OC 5W-0035 c1cc(c(cc1c2csc(n2)c3nc(cs3)c4ccc(c(c4)Cl)Cl)Cl)Cl 5W-0040 COC(=O)c1cc(cc(c1)OCc2cn(nn2)c3ccc(cc3)C(F)(F)F)OCc4cn(nn4)c5ccc(cc5)C(F)(F)F 5W-0041 c1ccc(cc1)COc2cc(cc(c2)OCc3ccccc3)C(=O)O 5W-0042 COc1ccc(cc1OCc2cn(nn2)c3ccc(cc3)C(F)(F)F)C=O 5W-0043 COc1cc(ccc1OCc2ccc(cc2)CN)CC=C 5W-0044 c1ccc(cc1)CS(=O)(=O)Cc2cnc(s2)Cl 5W-0046 c1cc(ccc1C(=O)O)S(=O)(=O)Cc2cnc(s2)Cl 5W-0066 COC(=O)c1ccc(cc1)SCc2cnc(s2)Cl 5W-0067 CS(=O)(=O)Cc1cnc(s1)Cl 5W-0070 c1ccc(cc1)CSc2ccc(cc2[N+](=O)[O-])Cl 5W-0073 COC(=O)C(c1c(cccc1Cl)[N+](=O)[O-])C(=O)OC 5W-0074 COC(=O)C(c1ccc(cc1[N+](=O)[O-])Cl)C(=O)OC 5W-0075 c1cc2c(cc1Br)C(=O)CCC2 5W-0079 c1cc2c(cc1Cl)NC(=O)C2 5W-0082 Cc1ccc(cc1)C(CCc2ccc(cc2)N)O 5W-0083 c1cc2c(c(c1)Cl)CC(=O)N2 5W-0090 COC(=O)C(c1cc(ccc1[N+](=O)[O-])C(F)(F)F)C(=O)OC 5W-0092 c1cc2c(nc1)NC(=O)C(O2)CCOC(=O)c3ccc(cc3)[N+](=O)[O-] 5W-0201 c1cc2c(nc1)NC(=O)C(O2)CCOC(=O)c3ccco3 5W-0202 CC(=O)c1cc(ccc1N)N2CCOCC2 5W-0204 CCNC(=S)NNC(=O)c1ccc2c(c1)cccn2 5W-0205 Cc1ccc(cc1)c2cc(n(n2)c3ccc(cc3Cl)Cl)N 5W-0206 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)I)C)CCO 5W-0207 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])c3ccccc3)CCO 5W-0208 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)Cl)C)CCO 5W-0209 Cc1ccc(cc1)S(=O)(=O)n2c(c(c(=O)n2C)CCO)C 5W-0210 CC(=O)c1cc(ccc1[N+](=O)[O-])N2CCC(CC2)C(=O)O 5W-0211 Cc1cc2ncc(cn2n1)C(=O)c3ccccc3O 5W-0212 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])CCO 5W-0217 c1ccc(cc1)COc2ccc(cc2)CCCO 5W-0218 Cc1c(c(=O)n(n1S(=O)(=O)c2cc(ccc2Cl)Cl)C)CCO 5W-0219 COC(=O)C(c1ccccc1)NC(=O)CCc2nc(no2)c3cccc(c3)C(F)(F)F 5W-0220 Cc1c2cc(ccc2nc(c1C(=O)OC)C(=O)OC)N3CCOCC3 5W-0222 c1cc2c(cc1[N+](=O)[O-])OC(C(=O)N2)CCN3CCCC3 5W-0223 CCn1c(nnc1S)c2ccc3c(c2)cccn3 5W-0226 c1ccc2c(c1)c(c(s2)C(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5)Cl 5W-0227 c1ccc2c(c1)c(c(s2)C(=O)N3CCN(CC3)c4ccc(cc4)F)Cl 5W-0228 c1ccc2c(c1)c(c(s2)C(=O)NCc3ccc(cc3)F)Cl 5W-0229 Cc1c(c(=O)n(n1C(=O)c2ccc(cc2)Cl)C)CCO 5W-0231 Cc1cc(c(c(c1)C)S(=O)(=O)n2c(c(c(=O)n2C)CCO)C)C 5W-0232 c1cc2c(cc1CN3CCN(CC3)CCC4C(=O)Nc5ccc(cc5O4)[N+](=O)[O-])OCO2 5W-0234 Cc1cccc(c1N2CCN(CC2)CCC3C(=O)Nc4ccc(cc4O3)[N+](=O)[O-])C 5W-0235 Cc1c(c(=O)n(n1S(=O)(=O)C)C)CCO 5W-0237 c1ccc2c(c1)c(c(s2)C(=O)NCCCN3CCOCC3)Cl 5W-0238 c1ccc(cc1)C(C(=O)O)NC(=O)CCc2nc(no2)c3cccc(c3)C(F)(F)F 5W-0239 CN(C)/C=N/c1c2ccccc2oc1C(=O)OC 5W-0241 CC(C)CN1CCCc2c1ccc(c2)/C=C(\C#N)/c3ccc4c(c3)OCO4 5W-0242 COc1cc(c(cc1OC)NC(=S)N2CCOCC2)C#N 5W-0243 CCCCCC1CCC(CC1)C(=O)NNC(=S)Nc2ccccc2 5W-0244 CCCCCC1CCC(CC1)C(=O)NNC(=O)c2ccc(cc2)F 5W-0245 CCCCCC1CCC(CC1)C(=O)NNC(=O)c2cccc(c2)C 5W-0246 CCCCCC1CCC(CC1)C(=O)NNC(=S)NC 5W-0247 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)F)c3ccccc3)CCO 5W-0250 Cc1c(c(=O)n(n1S(=O)(=O)c2ccccc2[N+](=O)[O-])c3ccccc3)CCO 5W-0251 Cc1c(c(=O)n(n1S(=O)(=O)c2c(cc(cc2Cl)Cl)Cl)c3ccccc3)CCO 5W-0252 CC(C)CN1CCCc2c1ccc(c2)/C=C/3\C(=O)SC(=S)N3 5W-0253 CC(C)(C)n1c(nnc1S)c2ccc3c(c2)cccn3 5W-0254 CCCCCC1CCC(CC1)c2nnc(n2c3ccccc3)S 5W-0255 CCCCCC1CCC(CC1)c2nnc(n2C)S 5W-0256 COC(=O)c1c(c2ccccc2o1)NC(=O)/C=C/C(=O)O 5W-0257 CCCCCC1CCC(CC1)c2nnc(o2)c3ccc(cc3)F 5W-0258 Cc1c2cc(ccc2nc(c1C(=O)O)C(=O)O)N3CCOCC3 5W-0259 Cc1c(c(=O)n(n1S(=O)(=O)c2ccccc2[N+](=O)[O-])C)CCO 5W-0260 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)F)C)CCO 5W-0261 COc1cc(c(cc1OC)/N=C(\N2CCOCC2)/SCC#N)C#N 5W-0262 COC(=O)c1c(c2ccccc2o1)N3C(=O)C=CC3=O 5W-0263 COc1ccc(cc1)Cn2cnc3c4ccccc4oc3c2=O 5W-0264 c1cc(ccc1C(=O)O)n2cc(c(n2)C(F)(F)F)CCCO 5W-0267 c1ccc(cc1)CNC(=O)CCc2nc(no2)c3cccc(c3)C(F)(F)F 5W-0269 c1cc2c(cc1OCCCF)sc(c2Cl)C(=O)N 5W-0274 c1ccc(c(c1)C(=O)/C=C/c2cccs2)O 5W-0275 CCN1C(=C(C(NC1=O)c2cccc(c2)[N+](=O)[O-])C(=O)O)C 5W-0276 CCOC(=O)c1cnc2c(c1NCCC3=CCCCC3)cnn2C 5W-0280 CCCCCC1CCC(CC1)C(=O)NNC(=S)NCC 5W-0281 CCCCCC1CCC(CC1)C(=O)NNC(=S)Nc2ccc(cc2)Cl 5W-0282 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NN 5W-0283 c1ccc(cc1)C(=O)N/N=C/c2coc3ccccc3c2=O 5W-0284 c1cc(cc(c1)C(F)(F)F)c2nc(on2)CCC(=O)NCc3ccco3 5W-0286 Cc1cccc(c1C)NC(=O)CCc2nc(no2)c3cccc(c3)C(F)(F)F 5W-0287 COc1cc(c(cc1OC)NC(=S)N2CCCC2)C#N 5W-0288 CCOC(=O)c1c(nc(s1)Br)C 5W-0289 CCCCCC1CCC(CC1)c2nnc(n2c3ccc(cc3)Cl)S 5W-0294 CCCCCC1CCC(CC1)c2nnc(n2CC)S 5W-0295 CCOC(=O)c1cnc2c(c1NCCCn3ccnc3)cnn2C 5W-0296 c1c(c(nc2n1ncn2)C(F)(F)F)CCCO 5W-0298 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCCC3=CCCCC3 5W-0299 c1cc2c(nc1)NC(=O)C(O2)CCCl 5W-0300 CC(C)(C)n1cc(cn1)C(=O)c2ccccc2O 5W-0301 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)CNC(=O)c3ccc(cc3)OC 5W-0302 Cc1ccc(cc1)C(=O)NCc2ccc(cc2)N3CCN(CC3)C(=O)OC(C)(C)C 5W-0303 c1ccc2c(c1)c(c(cn2)/C=N/N)Cl 5W-0304 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCCCn3ccnc3 5W-0305 Cc1ccc(cc1)n2c(cc(n2)C)N 5W-0307 C1CCc2c(c(=O)n([nH]2)CCO)C1 5W-0309 c1ccc2c(c1)c3c(o2)c(=O)n(cn3)CCCn4ccnc4 5W-0314 c1ccc2c(c1)c3c(o2)c(=O)n(cn3)Cc4cccc(c4)C(F)(F)F 5W-0316 COc1cc(c(cc1OC)/N=C(\N2CCCC2)/SCC#N)C#N 5W-0317 c1ccc2c(c1)c(c(o2)C(=O)NN)n3cccc3 5W-0319 CCOC(=O)C(=CNc1cc(nn1c2ccc(cc2)C)C)C(=O)OCC 5W-0324 CC(C)(C)OC(=O)N1CCC2(CC1)C=Cc3c2cccc3 5W-0327 c1cc(c(c(c1[N+](=O)[O-])Cl)C#N)Cl 5W-0330 c1ccc2c(c1)c3c(o2)c(=O)n(cn3)Cc4ccc(cc4)Cl 5W-0331 COc1ccccc1CNC(=O)CCc2nc(no2)c3cccc(c3)C(F)(F)F 5W-0332 COC(=O)c1c(sc(n1)N)c2ccccc2 5W-0333 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)CCl 5W-0334 CC(=O)c1ccc2c(c1)CCC2 5W-0337 c1ccc2c(c1)c(c(o2)C(=O)NNC(=O)c3ccc(cc3)Cl)n4cccc4 5W-0340 c1ccc2c(c1)c(c(o2)C(=O)NNC(=O)c3ccco3)n4cccc4 5W-0341 CCOC(=O)c1cnc2c(c1Cl)c(nn2c3ccc(cc3)C)C 5W-0344 CC(C)c1c(nc(s1)Cl)C(=O)O 5W-0350 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)Cl)c3ccccc3)CCO 5W-0351 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)I)c3ccccc3)CCO 5W-0352 Cc1c(c(=O)n(n1S(=O)(=O)c2cc(ccc2Cl)Cl)c3ccccc3)CCO 5W-0353 Cc1cc(n(n1)c2ccc(cc2)Cl)N 5W-0357 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)CN5C(=O)c6ccccc6C5=O 5W-0369 Cc1c(c(=O)n(n1S(=O)(=O)c2ccc(cc2)OC)C(C)(C)C)CCO 5W-0373 Cc1c(c(=O)n(n1S(=O)(=O)C)C(C)(C)C)CCO 5W-0374 CCOC(=O)c1cnc2c(c1NCCCn3ccnc3)c(nn2c4ccc(cc4)C)C 5W-0375 CCCCCC1CCC(CC1)Cc2nnc(n2c3ccc(cc3)C)S 5W-0376 c1ccc(cc1)CNC(=O)C(c2ccccc2)NC(=O)CCc3nc(no3)c4cccc(c4)C(F)(F)F 5W-0377 c1ccc2c(c1)ccc3c2occ(c3=O)C=O 5W-0378 CC(C)c1ccc(cc1)NC(=O)c2c(c3c4ccccc4ccc3s2)Cl 5W-0380 c1ccc2c(c1)ccc3c2c(c(s3)C(=O)O)Cl 5W-0383 CC(C)(C)n1cc(cn1)C(=O)c2ccc3ccccc3c2O 5W-0388 c1cc2c(cc1C(=O)CCC(=O)O)CCC2 5W-0389 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccc(cc2)OC)CCO 5W-0391 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccc(cc2)F)CCO 5W-0392 Cc1ccc(cc1)n2c3c(c(n2)C)c(c(cn3)C(=O)O)NCCCn4ccnc4 5W-0394 COc1ccc(cc1)N2CCN(CC2)C(=O)c3c(c4c5ccccc5ccc4s3)Cl 5W-0395 c1cc(ccc1C(=O)NCCN2CCCCC2)[N+](=O)[O-] 5W-0607 c1cc(ccc1[N+](=O)[O-])OCCN2CCOCC2 5W-0610 c1cc(ccc1C(=O)NCCN2CCCCC2)N 5W-0617 c1cc(cc(c1)OCCO)N 5W-0636 COC(=O)c1ccc(nc1)CO 5W-0644 c1ccc(cc1)N2CCN(CC2)c3ncc(s3)/C=C/4\c5ccccc5NC4=O 5W-0800 CN1C(=O)C(=Cc2cnc(s2)N3CCN(CC3)c4ccccc4)C(=O)N(C1=O)C 5W-0801 CN1C(=O)/C(=C/C=C/c2ccccc2)/SC1=O 5W-0803 CCCCCC/C=C\1/C(=O)N(C(=O)S1)C 5W-0804 Cc1ccc(cc1)Oc2ccccc2/C=C\3/C(=O)N(C(=O)S3)C 5W-0805 c1ccc2c(c1)c(=O)[nH]c3n2ncc3C#N 5W-0806 CCOC(=O)c1cn(nn1)c2nc(cc(n2)c3ccccc3)C 5W-0809 Cc1c(c(n2c(n1)c(cn2)c3ccsc3)C)Cc4ccc(nc4)Cl 5W-0810 Cc1ccc(n1C(CC(=O)Nc2ccc(cc2)F)c3ccc4c(c3)OCO4)C 5W-0811 CCOC(=O)c1cc([nH]n1)c2cccc(c2)[N+](=O)[O-] 5W-0812 c1cc(ccc1NC(=O)NCCCl)F 5W-0813 c1ccc(cc1)OCCN2CCN(C2=O)c3cccc(c3)C(F)(F)F 5W-0815 Cc1ccc(cc1)c2cc3ccccc3nc2N 5W-0816 Cc1cccn2c1nc(c2)c3cccc(c3)[N+](=O)[O-] 5W-0817 CNc1nc(cs1)c2cccc(c2)[N+](=O)[O-] 5W-0818 Cc1cc(c(n1C(CC(=O)O)c2ccc3c(c2)OCO3)C)C(=O)C(F)(F)F 5W-0819 CCCCCc1c(nnn1c2nc(cc(n2)c3ccccc3)C)C(=O)OC 5W-0820 CCCCCc1c(nnn1c2nc(c(c(n2)C)Cc3ccc(cc3)Cl)C)C(=O)OC 5W-0822 CN1CCN(CC1)CC#CCOc2ccc3c(c2)OCO3 5W-0823 Cc1cc2c(c(c(=O)[nH]c2cc1N)C)C 5W-0826 c1cc(c(c(c1)Cl)COc2coc(cc2=O)CO)F 5W-0828 COc1ccc(cc1OC)c2cc3ccccc3nc2N 5W-0830 c1ccc2c(c1)cc(c(n2)N)c3cccs3 5W-0831 c1cc2c(cc1CN3CCN(CC3)c4ncc(s4)C=O)OCO2 5W-0832 CCOc1cc2c(cc1OC)C(/C(=C/N(C)C)/C2=O)NC(=O)C(F)(F)F 5W-0833 c1ccn(c1)C(CC(=O)NC2CCCCC2)c3ccc(cc3)Br 5W-0834 Cc1ccc(n1C(CC(=O)OC)c2ccsc2)C 5W-0836 Cc1c(c(n2c(n1)c(cn2)c3ccccn3)C)Cc4ccc(nc4)Cl 5W-0837 CNc1nc(cs1)c2cccc(c2)N 5W-0838 c1cc(ccc1N2CCNC2=O)F 5W-0840 c1ccn(c1)C(CC(=O)O)c2ccc(cc2)N 5W-0841 CCOC(=O)C(Cc1ccc(cc1)Cl)(Cc2ccc(cc2)Cl)C(=O)C 5W-0843 Cc1c(sc(n1)n2cccc2)C(=O)C 5W-0845 CCOC(=O)CC(c1cccc(c1)Cl)n2cccc2 5W-0846 Cc1c(sc2n1cc(n2)c3ccc(cc3)Cl)C(=O)C 5W-0848 c1ccc(c(c1)Cn2cccc2C=O)[N+](=O)[O-] 5W-0849 COc1ccc(cc1)N2CCN(CC2)CC#CCOc3ccc4c(c3)OCO4 5W-0852 Cc1ccc(n1C(CC(=O)O)c2ccc(cc2)[N+](=O)[O-])C 5W-0855 Cn1cc2cccc(c2n1)NC(=O)c3ccc(cc3)F 5W-0856 c1ccc(cc1)c2c(nnc(n2)SCc3ccc(cc3)Cl)c4ccccc4 5W-0857 CCOC(=O)CC(c1cccc(c1)Cl)n2cccc2C=O 5W-0859 c1ccc2c(c1)ccc(n2)c3ccc(cc3)C4CCCCC4 5W-0861 c1cc(ccc1c2ccc3cc(cc(c3n2)Br)Br)C4CCCCC4 5W-0862 C/C(=N\OCc1ccc(cc1)Cl)/C(Cc2ccc(nc2)Cl)Cc3ccc(nc3)Cl 5W-0864 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)C)Cc5ccc(nc5)Cl)C)C 5W-0865 Cc1c(c(n2c(n1)ncn2)C)Cc3ccc(cc3)Cl 5W-0866 C/C(=N\OC)/C(Cc1ccc(nc1)Cl)Cc2ccc(nc2)Cl 5W-0867 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)SCc4ccc(cc4)F)C(F)(F)F 5W-0868 CCOC(=O)c1cc(on1)c2cccc(c2)[N+](=O)[O-] 5W-0869 c1c2c(cc3c1OCO3)C(=CC2NC(=O)C(F)(F)F)Cl 5W-0870 CCCCCC(=O)Nc1cc2c(cc1C)c(cc(=O)[nH]2)COC 5W-0871 Cc1cc2c(cc(=O)[nH]c2cc1NC(=O)C(C)(C)CCl)COC 5W-0872 CCOC(=O)CC(c1ccc(cc1)[N+](=O)[O-])n2c(ccc2C)C 5W-0873 c1ccc(c(c1)Cn2cccc2/C=N/O)[N+](=O)[O-] 5W-0874 CCOc1cc2c(cc1OC)C(/C(=C/Nc3ccc(c(c3)C)C)/C2=O)NC(=O)C(F)(F)F 5W-0875 CCOC(=O)CC(c1ccc(cc1)N)n2c(ccc2C)C 5W-0876 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)SCCCCOc4ccccc4)C(F)(F)F 5W-0877 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)Sc4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 5W-0878 COc1ccc-2c(c1)CCc3c2nc4c(c3)cc(cc4Br)Br 5W-0879 Cc1c(sc(n1)n2cccc2)C(=O)/C=C/N(C)C 5W-0881 Cc1ccc(n1C(CC(=O)O)c2ccc(cc2)C#N)C 5W-0883 Cc1ccc(n1C(CC(=O)O)c2ccc(cc2)F)C 5W-0884 Cc1ccc(n1C(CC(=O)O)c2ccco2)C 5W-0885 c1ccc(cc1)COc2ccc(cc2)C(CC(=O)O)N 5W-0887 c1ccc2c(c1)cccc2C(CC(=O)O)n3cccc3 5W-0888 CCCCCC(=O)Nc1cccc(c1)c2csc(n2)NC 5W-0889 Cc1cc2c(cc(=O)[nH]c2cc1NC(=O)C3CC3)COC 5W-0891 Cc1ccc(n1C(CC(=O)OC)c2ccc(cc2)C#N)C 5W-0893 Cn1cc2cc(ccc2n1)NS(=O)(=O)c3ccc(cc3)OC 5W-0894 c1cc(n(c1)c2nccs2)/C=N/NC(=S)N 5W-0896 c1cc(n(c1)c2nccs2)/C=C\C(=O)c3ccc4c(c3)OCO4 5W-0897 CC1(CC(=O)C(=CNc2cccc(c2)OC)C(=O)C1)C 5W-0900 COc1cc(ccc1OCc2cccc(c2)C(F)(F)F)C=O 5W-0901 C1CS(=O)(=O)CCN1CCC(=O)O 5W-0902 C[NH+]1CC[NH+](CC1)CC#CCOc2ccc3c(c2)OCO3.[Cl-].[Cl-] 5W-0911 CCCc1cc(cc(n1)O)C(F)(F)F 5W-0931 CCOC(=O)c1cnc(nc1C(F)(F)F)c2ccccc2 5W-1085 c1ccc(cc1)c2ncc(c(n2)C(F)(F)F)C(=O)O 5W-1087 c1ccc(cc1)c2cc(c(=O)[nH]n2)C(=O)O 5X-0023 CCOC(=O)c1cc(nnc1O)c2ccccc2 5X-0069 c1c(c(cc(c1N2CCOCC2)Cl)[N+](=O)[O-])N 5X-0200 c1ccc(c(c1)CN2c3cc(ccc3N4CCCCC4C2=O)C(F)(F)F)Cl 5X-0201 c1ccc(c(c1)C=C(C#N)C#N)Oc2ccc(cc2Cl)Cl 5X-0204 CCOC(=O)C1CCN(CC1)c2ccc(cn2)C=C(C#N)C#N 5X-0205 c1ccn(c1)c2ccc(cc2)c3cn[nH]c3N 5X-0206 CCOC(=O)c1ccc(nc1C)c2cccc(c2)C(F)(F)F 5X-0207 CCOC(=O)C\1CCC/C1=N\Nc2ccc(cc2)C(=O)O 5X-0208 c1ccc(cc1)/C=C/C=C\2/C(=O)N=C(S2)NC(=N)N 5X-0211 c1ccc(c(c1)/C=C\2/C(=O)N=C(S2)NCCCC(=O)O)C(F)(F)F 5X-0213 c1ccc(c(c1)/C=C\2/C(=O)N=C(S2)NO)C(F)(F)F 5X-0214 CSc1ccc(cc1)/C=C/2\C(=O)NC(=S)S2 5X-0220 c1ccc2c(c1)cccc2/C=C/3\C(=O)NC(=S)S3 5X-0221 Cc1ccc(cc1)C2C(C(=C(C(C2(C#N)C#N)c3ccc(cc3)SC)C(=O)OC)O)C(=O)OC 5X-0224 Cc1cccc(c1N2CCN(CC2)CN(C3=NC(=O)/C(=C/c4ccccc4C(F)(F)F)/S3)O)C 5X-0225 CCOC(=O)c1c2c(sc1N)CN(CC2)C 5X-0229 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2ccc(cc2)SC)(C#N)C#N)c3ccc(cc3)C(F)(F)F 5X-0230 CSC1=NC(=O)/C(=C\c2cccc3c2cccc3)/S1 5X-0232 CSc1ccc(cc1)/C=C\2/C(=O)N=C(S2)SC 5X-0235 Cc1ccc(cc1)/C(=N/O)/N 5X-0240 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2ccc(cc2)SC)(C#N)C#N)c3ccc(cc3)F 5X-0241 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2ccc(cc2)SC)(C#N)C#N)c3ccncc3 5X-0242 COC(=O)C1C(C(C(C(=C1O)C(=O)OC)c2ccc(cc2)SC)(C#N)C#N)c3ccc(cc3)[N+](=O)[O-] 5X-0243 c1cc(c(c(c1)Cl)CN2c3cc(ccc3N4CCCCC4C2=O)C(F)(F)F)F 5X-0245 c1cc(cc(c1)C(F)(F)F)CN2c3cc(ccc3N4CCCCC4C2=O)C(F)(F)F 5X-0246 c1cc2c(cc1C(F)(F)F)NCC3N2CCCC3 5X-0247 Cc1ccc(cc1)c2nc(on2)c3cccnc3 5X-0253 c1cc(cnc1)c2nc(no2)c3ccc(cc3)CBr 5X-0260 c1c(c(cc(c1N2CCCC2)Cl)[N+](=O)[O-])N 5X-0261 c1cc(cnc1)c2nc(no2)c3ccc(cc3)CN4CCOCC4 5X-0263 CC1CN(CC(O1)C)c2ccc(cn2)/C=N/OCc3c(cccc3Cl)Cl 5X-0265 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)N.Br 5X-0266 c1ccc2c(c1)cccc2/C=C/3\C(=O)N=C(S3)NC(=N)N 5X-0267 Cc1ccc(cc1)c2nc(on2)c3ccncc3 5X-0268 c1cc2c(cc1F)c3c([nH]2)CCNC3 5X-0270 CCOC(=O)c1cnc([nH]c1=O)NC2=NC(=O)/C(=C\c3cccc4c3cccc4)/S2 5X-0275 c1ccn(c1)c2c(ccs2)C#N 5X-0277 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)NC(=O)c4cccs4 5X-0283 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)NC(=O)C4CCCCC4 5X-0286 c1ccn(c1)c2c(ccs2)/C(=N/O)/N 5X-0289 CC(Nc1nccs1)n2cncn2 5X-0291 CCOC(=O)C1CNc2ccccc2O1 5X-0292 Cc1ccc(cc1C)Cc2nnn(n2)C 5X-0293 c1c(c(cc(c1N2CCCCC2)Cl)[N+](=O)[O-])N 5X-0294 COc1ccc(cc1S(=O)(=O)N2CC3CCCCN3c4c2cc(cc4)C(F)(F)F)Cl 5X-0295 CCOC(=O)C1CN(c2ccccc2O1)S(=O)(=O)c3ccc(cc3)OC 5X-0299 COc1ccc(cc1)S(=O)(=O)N2CC(Oc3c2cccc3)C(=O)O 5X-0308 CCOC(=O)C1CNc2cc(ccc2O1)S(=O)(=O)CC 5X-0309 COc1ccc(cc1OC)C(=O)Nc2nc(cs2)CCN3C(=O)c4ccccc4C3=O 5X-0314 CC(C)(C)C(=O)Nc1cccc(c1)OC 5X-0602 Cc1ccc(n1c2ccc(cc2)CO)C 5X-0700 c1ccc(cc1)CN2CCCCC2CO 5X-0703 CC(C)(C)OC(=O)N1CCC(CC1)CO 5X-0704 CCCCCC#Cc1c(cccn1)C#N 5X-0706 Cc1nc2cc(ccc2o1)N 5X-0708 COC(=O)c1cnc(cc1Cl)Cl 5X-0801 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)CCCCl 5X-0802 Cc1cc(nc(n1)N)N2CCOCC2 5X-0803 c1ccnc(c1)c2nc3cc(ccc3o2)CC(=O)NCc4ccc(cc4)F 5X-0804 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(C(C)(C)C)N 5X-0805 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=C\4/c5ccccc5NC4=O 5X-0806 COc1ccc2c(c1)sc(n2)N 5X-0808 Cc1ccc2c(c1)sc(n2)N 5X-0809 CC(C)c1ccc2c(c1)sc(n2)N 5X-0810 CC(=O)C(=C(SC)SC)C(=O)C 5X-0811 COc1ccc(cc1)c2cc(cnc2c3ccc(cc3)OC)C(F)(F)F 5X-0813 COc1ccc(cc1S(=O)(=O)Cl)c2ccc(cc2Cl)C(F)(F)F 5X-0814 CN(C)/C=C/C(=O)c1cccc(c1)C#N 5X-0815 COC(=O)Cc1ccc2c(c1)nc(o2)c3cccnc3 5X-0816 c1cnc(nc1)SCC#N 5X-0817 CN1C(=O)C(C(=O)N(C1=O)C)Cc2c[nH]c3c2cc(cc3)OC 5X-0818 c1ccc2c(c1)nc3c(n2)Oc4cccnc4N3 5X-0821 c1ccc2c(c1)c(c([nH]2)C(=O)NN)Cl 5X-0824 COc1ccc(cc1S(=O)(=O)N)c2c(cc(cn2)C(F)(F)F)Cl 5X-0827 Cc1ccc(cc1)c2c(nnc(n2)S)c3ccc(cc3)C 5X-0829 CN1CCC(CC1)NS(=O)(=O)c2ccc(cc2)I 5X-0830 CCC(CC)N1CCS(=O)(=O)CC1 5X-0831 CC(C)(C)c1ccc(cc1)/C=N/O 5X-0832 COC(=O)c1cccn2c1nc(c2)c3ccc(cc3)F 5X-0833 c1cc(ccc1NC(=O)/C=C/C(=O)O)I 5X-0834 c1cc(ccc1CCN2CCS(=O)(=O)CC2)S(=O)(=O)N 5X-0835 c1cc(ccc1CNS(=O)(=O)CCCCl)F 5X-0836 CC/C(=N\OCc1ccccc1Cl)/c2cc(ccn2)C(F)(F)F 5X-0839 CC(C(=O)C)Oc1cc(ccc1OC)[N+](=O)[O-] 5X-0842 c1cc(cc(c1)N2CCN(CC2)C(=O)Cc3ccc4c(c3)nc(o4)c5cccnc5)C(F)(F)F 5X-0843 c1cc(cc(c1)C(F)(F)F)C(CCO)N2CCS(=O)(=O)CC2 5X-0844 COc1ccc(cc1OC)CCN(CN2C(=O)CCC2=O)CN3C(=O)CCC3=O 5X-0849 c1cc(ccc1C2c3ccsc3CCN2)Cl 5X-0852 COc1cc(cc(c1OC)OC)CNCc2cc(c(c(c2)OC)OC)OC 5X-0853 CCOC(=O)c1cc2c(c(sc2nc1C(F)(F)F)C(=O)OCC)N 5X-0854 c1c(occ(c1=O)O)CCl 5X-0856 Cc1c(nc2c(c(nn2c1C)SC)C#N)C 5X-0858 c1ccc2c(c1)-c3c(c[nH]n3)CO2 5X-0922 c1ccc2c(c1)-c3c(cnc(n3)N)CO2 5X-0923 Cn1cc(c(=O)c2c1cccc2)c3ccccc3C(=O)O 5X-0924 Cn1cc(c(=O)c2c1cccc2)c3ccccc3C(=O)N 5X-0925 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4ccccc4Cl)CO2 5X-0926 c1cc(ccc1C#N)OCCBr 5X-0927 CNC(=O)c1ccccc1c2cn(c3ccccc3c2=O)C 5X-0928 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4cccc(c4)Cl)CO2 5X-0929 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4ccc(cc4)Cl)CO2 5X-0930 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4cccc(c4)[N+](=O)[O-])CO2 5X-0934 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4ccc(cc4)[N+](=O)[O-])CO2 5X-0936 Cc1ccc(cc1)C(=O)Nc2ncc3c(n2)-c4ccccc4OC3 5X-0937 Cn1c2ccc(cc2sc1=N)Br 5X-0941 Cc1ccc2c(c1)sc(=N)n2C 5X-0942 Cn1c2ccc(cc2sc1=N)OC 5X-0943 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4ccc(cc4)F)CO2 5X-0944 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4ccc(cc4Cl)Cl)CO2 5X-0946 c1ccc2c(c1)-c3c(cnc(n3)NC(=O)c4ccccc4F)CO2 5X-0947 CCOC(=O)c1c(c(c(s1)SC)C(=O)C)C 5X-0949 CCOC(=O)c1c(c(sc1SC)C(=O)C)C 5X-0952 CCOC(=O)c1c(c(sc1SC)C(=O)OCC)C 5X-0953 C[NH+](C)CCC(=O)c1ccccc1.[Cl-] 5X-0955 c1cc(cc(c1)Cl)CN(Cc2cccc(c2)Cl)C#N 5X-0956 c1ccn2c(c1)cnc2Br 5X-5034 c1cc(cc(c1)F)c2ncnc(n2)Nc3cccc(c3)C(F)(F)F 5X-9000 CC(=O)N1C(CSC12CCC3(CC2)OCCO3)C(=O)O 5Y-0009 CC(=O)N1C(CSC12CCN(CC2)Cc3ccccc3)C(=O)O.Cl 5Y-0010 COc1ccc2c(c1)c(c[nH]2)C3=CCC4(CC3)OCCO4 5Y-0011 c1ccc(c(c1)C(=O)c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)C(=O)O 5Y-0037 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCOCC4 5Y-0039 c1cc(c(cc1[N+](=O)[O-])C(F)(F)F)N2CCOCC2 5Y-0055 c1ccc2c(c1)ccc(c2C(C(=O)O)O)O 5Y-0200 c1ccc2c(c1)C(C(=O)N2)CCCC(=O)O 5Y-0202 c1cc2c(nc1)nc(o2)S 5Y-0203 c1c(c(sc1C(=O)O)C=O)Br 5Y-0208 COC(c1c2ccccc2ccc1O)C(=O)OC 5Y-0212 CSc1nc2c(o1)cccn2 5Y-0215 c1ccnc(c1)N2CCN(CC2)C(=O)c3ccc(cc3)N 5Y-0217 c1cc(ccc1C(=O)N2CCN(CC2)C3CCCCC3)N 5Y-0218 c1ccc(c(c1)N2CCN(CC2)C(=O)c3ccc(cc3)N)F 5Y-0219 c1cnc(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)N 5Y-0222 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)c3ccc(cc3)N 5Y-0223 c1cc(ccc1C#N)N2CCN(CC2)C(=O)c3ccc(cc3)N 5Y-0225 CN1CCc2c(sc(c2C#N)N)C1 5Y-0232 CC(C)N1CCc2c(sc(c2C(=O)OC)N)C1.O 5Y-0238 CCOC(=O)c1c(nc(s1)Cl)C(F)(F)F 5Y-0700 COc1ccc(cc1)c2c(cccn2)N 5Y-0701 COC(=O)c1ccc(cc1)c2ccc(cn2)N 5Y-0702 COC(=O)c1cc(c(nc1)N)Br 5Y-0703 c1ccn(c1)c2ccc(cn2)C(=O)O 5Y-0705 CC(C)(C1OCc2ccccc2CO1)Br 5Y-0706 COC(=O)c1cc(c(c(c1)F)F)F 5Y-0800 CC(=O)c1ccc(cc1)OC(c2ccccc2)C(=O)OC 5Y-0801 c1cc2c(cc1CC(=O)O)NC(=O)CO2 5Y-0802 c1cc(c(cc1[N+](=O)[O-])Cl)SCC(=O)O 5Y-0803 COc1ccc(c(c1)Br)O 5Y-0804 c1ccc(cc1)C(C(=O)O)Oc2ccc(cc2)C=O 5Y-0807 C#CCOc1ccc(cc1Cl)Cl 5Y-0809 C#Cc1cccc(c1)NC(=O)c2ccc(cc2)Cl 5Y-0814 CCOC(=O)C1=C(N(C(=O)C1)CCc2cccs2)C 5Y-0816 COc1ccc(cc1OC(c2ccccc2)C(=O)OC)C=O 5Y-0817 COC(=O)CSc1ccc(cc1Cl)[N+](=O)[O-] 5Y-0818 c1cnc2nc(nn2c1C3CC3)N 5Y-0821 c1cc(ccc1c2cc([nH]n2)N)Br 5Y-0822 c1cc(ccc1[N+](=O)[O-])SCC(=O)O 5Y-0823 COC(=O)CSc1ccc(cc1)[N+](=O)[O-] 5Y-0824 Cc1ccc(cc1)COc2ccc(c(c2)O)C(=O)C 5Y-0922 c1cc(ccc1C(CNCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O)(c4ccc(cc4)Cl)O)Cl 5Y-0923 c1cc(ccc1C(=O)N2CCN(CC2)c3ccc(cc3)C(F)(F)F)N 5Y-0937 CC(=O)c1ccc(c(c1)Cl)O 5Y-0939 Cc1cccc(c1)COc2ccc(cc2F)C(=O)C 5Y-0940 Cc1ccc(cc1)C(=O)c2ccccc2C(=O)O 5Y-1180 COc1ccc(cc1)C(=O)c2ccccc2C(=O)O 5Y-1181 Cc1ccc(cc1)c2c3ccccc3c(=O)[nH]n2 5Y-1182 c1cc2cc(ccc2cc1C=O)O 5Y-5022 c1c(c(nc(n1)Cl)N)C#N 5Y-5028 CCOC(=O)C(=O)CC(=O)c1ccccn1 5Z-0610 CCOC(=O)c1cc(n[nH]1)c2ccccn2 5Z-0611 COC(=O)c1cc(ccc1c2ccc(cc2)Br)[N+](=O)[O-] 5Z-0700 c1cc2c(cc1C(F)(F)F)[nH]nc2N 5Z-0702 C/C(=C\C(=O)c1cnccn1)/N(C)C 5Z-0802 CC(C)(C)OC(=O)N1CCc2c(ccs2)C1c3ccc(cc3)[N+](=O)[O-] 5Z-0803 c1c[nH]nc1c2cnccn2 5Z-0806 Cc1cc(n[nH]1)c2cnccn2 5Z-0807 CN(C)/C=C/C(=O)c1nccs1 5Z-0809 C/C(=C\C(=O)c1nccs1)/N(C)C 5Z-0810 c1c[nH]nc1c2nccs2 5Z-0812 Cc1cc(n[nH]1)c2nccs2 5Z-0813 c1cnc(nc1c2cnccn2)N 5Z-0814 c1c(cc(cc1C(F)(F)F)F)/C=C/C(=O)O 5Z-0815 Cc1cc(ccc1Br)Oc2ccccc2C=O 5Z-0818 Cc1ccc(n1c2ccccc2C(=O)NN)C 5Z-0819 c1ccc(cc1)Oc2cc(ccc2C=O)Br 5Z-0821 c1ccc2c(c1)CN(C2=O)CCC(=O)O 5Z-0825 Cc1cccc2c1[nH]c3c2c(ccc3C)C 5Z-0826 Cc1ccc(n1CCC(=O)O)C 5Z-0827 c1cc(ccc1CN(Cc2ccc(cc2)Cl)C#N)Cl 6B-001 c1ccc(cc1)CN(Cc2ccccc2)c3[nH]nnn3 6B-002 c1ccc(cc1)/C=C/CSc2ccccn2 6B-003 c1ccc(cc1)/C=C/CSc2ccc(cn2)C(F)(F)F 6B-004 c1ccc(cc1)/C=C/CSc2ccc(cc2)Cl 6B-005 c1ccc(cc1)/C=C/CSc2ccccc2N 6B-007 c1ccc(cc1)/C=C/CS(=O)(=O)c2ccc(cc2)Cl 6B-008 c1cc(ccc1CN(Cc2ccc(cc2)Cl)c3[nH]nnn3)Cl 6B-009 CN(C)/C=C(/C=C/c1ccccc1)\S(=O)(=O)c2ccc(cc2)Cl 6B-010 c1ccc(c(c1)C(F)(F)F)NC=C2C=NNC2=O 6B-012 c1cc(cc(c1)NC=C2C=NNC2=O)C(F)(F)F 6B-013 COc1ccc(cc1)NC=C2C=NNC2=O 6B-014 CNc1c(cn(n1)C(=O)Nc2cccc(c2)C(F)(F)F)[N+](=O)[O-] 6B-015 c1ccc(c(c1)NC=C2C=NNC2=O)Cl 6B-017 c1cc(cc(c1)Cl)NC=C2C=NNC2=O 6B-018 CNc1c(cn(n1)C(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 6B-020 CNc1c(cn(n1)C(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] 6B-021 CC(=O)n1cc(c(n1)NC)[N+](=O)[O-] 6B-022 c1ccc(cc1)/C=C/C(/C=N\O)S(=O)(=O)c2ccc(cc2)Cl 6B-023 c1ccc2c(c1)N(CCS2)S(=O)(=O)c3ccc(cc3)Cl 6B-024 COc1ccc(cc1)S(=O)(=O)N2CCSc3c2cccc3 6B-025 Cc1ccc(cc1)S(=O)(=O)N2CCSc3c2cccc3 6B-026 c1ccc2c(c1)N(CCS2)C(=O)c3ccc(cc3)Cl 6B-027 CC1(OC(=O)C(=C(SC)SC)C(=O)O1)C 6B-036 CNC1=C(CC(=C(N1C)SC)[N+](=O)[O-])[N+](=O)[O-] 6B-037 c1cc(c(nc1/C=N\O)O)C#N 6B-038 CO/N=C\C(/C=C/c1ccccc1)S(=O)(=O)c2ccc(cc2)Cl 6B-043 CNc1c(cn(n1)C(=O)c2cccc(c2)C(F)(F)F)[N+](=O)[O-] 6B-045 c1cc(ccc1Nc2c(cnc(n2)N)[N+](=O)[O-])Cl 6B-047 c1ccc2c(c1)c(=O)c(co2)/C=N/O 6B-048 CNC1=C(CC(=C(N1C)N2CCOCC2)[N+](=O)[O-])[N+](=O)[O-] 6B-049 CNc1c(cn(n1)S(=O)(=O)c2cccc(c2)C(F)(F)F)[N+](=O)[O-] 6B-051 c1cc(cc(c1)Nc2c(cnc(n2)N)[N+](=O)[O-])C(F)(F)F 6B-053 CCOC(=O)c1cc2c(=O)c3ccccc3oc2nc1C 6B-055 c1ccc(cc1)/C=C/C(/C=N/OC(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 6B-059 c1cc[n+](c(c1)SCC(=O)CSc2cccc[n+]2[O-])[O-] 6B-063 CCOC(=O)Cn1nc(nn1)N(Cc2ccc(cc2)Cl)Cc3ccc(cc3)Cl 6B-064 c1ccc(cc1)SCC(=O)CSc2ccccc2 6B-065 CCOC(=O)c1cc2c(=O)c3ccccc3oc2nc1C(F)(F)F 6B-066 CN(/C=C(\Sc1ccccc1)/C(=O)/C(=C/N(C)C)/Sc2ccccc2)C 6B-067 c1cc(ccc1CN(Cc2ccc(cc2)Cl)c3nnn(n3)CC(=O)N)Cl 6B-068 CNC1=C(CC(=C(N1C)N2CCNCC2)[N+](=O)[O-])[N+](=O)[O-] 6B-073 c1cc(ccc1NC(=O)N2CCSc3c2ccc(c3)Cl)Cl 6B-074 Cc1ccc(cc1)NC(=O)N2CCSc3c2ccc(c3)Cl 6B-075 c1cc(cc(c1)NC(=O)N2CCSc3c2ccc(c3)Cl)C(F)(F)F 6B-076 CNC1=C(CC(=C(N1C)N2CCN(CC2)C(=O)Nc3ccccc3)[N+](=O)[O-])[N+](=O)[O-] 6B-077 c1cc(ccc1S(=O)(=O)N2CCSc3c2ccc(c3)Cl)Cl 6B-078 COc1ccc(cc1)S(=O)(=O)N2CCSc3c2ccc(c3)Cl 6B-079 CNC1=C(CC(=C(N1C)NCc2ccc(cc2)Cl)[N+](=O)[O-])[N+](=O)[O-] 6B-080 CNC1=C(CC(=C(N1C)NCc2ccccn2)[N+](=O)[O-])[N+](=O)[O-] 6B-081 c1ccc(c(c1)NC(=O)N2CCSc3c2ccc(c3)Cl)Cl 6B-082 c1cc(cc(c1)Cl)NC(=O)N2CCSc3c2ccc(c3)Cl 6B-083 c1ccc(cc1)NC(=O)N2CCSc3c2ccc(c3)Cl 6B-084 CN/C(=N\C)/C[N+](=O)[O-] 6B-085 Cc1ccc(cc1)S(=O)(=O)N2CCSc3c2ccc(c3)Cl 6B-086 c1ccc(cc1)S(=O)(=O)N2CCSc3c2ccc(c3)Cl 6B-087 Cc1ccc(cc1)C=C2C(=O)OC(OC2=O)(C)C 6B-092 CC1(CC2=C(C(CC(=O)O2)c3ccc(cc3)N(C)C)C(=O)C1)C 6B-094 CC1(CC2=C(C(CC(=O)O2)c3ccc(cc3Cl)Cl)C(=O)C1)C 6B-097 Cc1ccc(cc1)C2CC(=O)OC3=C2C(=O)CC(C3)(C)C 6B-100 c1cc(nc(c1)Cl)N2CCNCC2 6B-103 c1ccc(cc1)NC(=O)N2CCN(CC2)c3cccc(n3)Cl 6B-107 c1cc(ccc1C(=O)N2CCSc3c2ccc(c3)Cl)Cl 6B-108 Cc1ccc(cc1)C(=O)N2CCSc3c2ccc(c3)Cl 6B-109 Cc1c(c(ns1)SCc2c(cccc2Cl)Cl)C#N 6C-001 Cc1c(c(ns1)SCc2ccccc2C(=O)OC)C#N 6C-002 Cc1c(c(ns1)SCC#N)C#N 6C-006 Cc1c(c(ns1)SCc2ccc(cc2)Cl)C#N 6C-008 CC(=O)c1cc(ccc1O)F 6C-009 c1cc2c(cc1F)c(=O)c(co2)C=O 6C-010 c1cc2c(cc1F)c(=O)c(co2)/C=N\O 6C-011 c1ccc(cc1)C(Nc2ccccn2)Nc3ccccn3 6C-012 c1cc2c(cc1F)c(=O)c(c(o2)N)C=O 6C-013 c1ccc(cc1)n2c(nc3ccccc3c2=O)/C=C/c4cccnc4 6C-015 CCc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)OC 6C-016 COCc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)OC 6C-017 CCOC(=O)c1cc2c(=O)c3cc(ccc3oc2nc1C)F 6C-020 Cc1ccc(cc1)CSc2c(c(sn2)C)C#N 6C-022 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)O 6C-023 CS/C(=N\C#N)/N1CCOCC1 6C-024 Cc1c(c(ns1)SCc2cccc(c2)Cl)C#N 6C-025 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)Nc4ccc(cc4)Cl 6C-027 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)Nc4cccc(c4)C(F)(F)F 6C-028 C1COCCN1c2[nH]c(nn2)N 6C-029 CCOC(=O)c1cnc2nc(nn2c1N)N3CCOCC3 6C-030 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)NCc4ccccc4 6C-031 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)NCc4ccc(cc4)Cl 6C-032 CC(=O)c1cc(ccc1O)Cl 6C-033 c1c(c(n2c(n1)nc(n2)N3CCOCC3)N)C(=O)O 6C-034 CS/C(=C\[N+](=O)[O-])/Nc1ccc(cc1)OC(F)(F)F 6C-035 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)OC 6C-036 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)NC(C)(C)C 6C-037 CCN(CC)C(=O)c1cc2c(=O)c3cc(ccc3oc2nc1C)F 6C-038 c1cc(ccc1C(=O)n2cnc(c2C#N)C#N)Cl 6C-039 c1cc(ccc1N\2C(=O)CS/C2=C\[N+](=O)[O-])OC(F)(F)F 6C-040 COC(=O)c1c(nc(s1)N2CCOCC2)N 6C-041 c1cc2c(cc1Cl)c(=O)c(co2)C=O 6C-042 c1cc2c(cc1Cl)c(=O)c(co2)/C=N/O 6C-043 c1cc2c(cc1Cl)c(=O)c(c(o2)N)C=O 6C-044 CCc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)OC 6C-046 COCc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)OC 6C-047 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)OC 6C-048 CCOC(=O)c1cc2c(=O)c3cc(ccc3oc2nc1C)Cl 6C-053 CN(C)/C=C/c1c(c(ns1)SCc2ccccc2C(=O)OC)C#N 6C-054 COC(=O)c1ccccc1CSc2c(c(sn2)/C=C/Nc3ccccc3)C#N 6C-055 COC(=O)c1ccccc1CSc2c(c(sn2)/C=C/Nc3ccc(cc3)Cl)C#N 6C-056 c1cnc2nc(nn2c1N)N3CCOCC3 6C-058 CN(C)/C=C/c1c(c(ns1)SCc2c(cccc2Cl)Cl)C#N 6C-059 c1ccc(cc1)N/C=C/c2c(c(ns2)SCc3c(cccc3Cl)Cl)C#N 6C-060 c1cc(c(c(c1)Cl)CSc2c(c(sn2)/C=C/Nc3ccc(cc3)Cl)C#N)Cl 6C-061 CN(C)/C=C/c1c(c(ns1)SCc2ccc(cc2)Cl)C#N 6C-063 Cc1ccc(cc1)CSc2c(c(sn2)/C=C/N(C)C)C#N 6C-064 Cc1c(c(ns1)SCc2c(cccc2Cl)F)C#N 6C-065 Cc1c(c(ns1)SCc2ccc(cc2Cl)Cl)C#N 6C-066 CN(C)/C=C/c1c(c(ns1)SCc2ccc(cc2Cl)Cl)C#N 6C-067 CN(C)/C=C/c1c(c(ns1)SCc2c(cccc2Cl)F)C#N 6C-068 Cc1c(c(ns1)SCc2csc(n2)C)C#N 6C-069 c1ccc(cc1)N/C=C/c2c(c(ns2)SCc3ccc(cc3Cl)Cl)C#N 6C-070 c1cc(ccc1N/C=C/c2c(c(ns2)SCc3ccc(cc3Cl)Cl)C#N)Cl 6C-071 c1ccc(cc1)N/C=C/c2c(c(ns2)SCc3c(cccc3Cl)F)C#N 6C-072 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)O 6C-073 c1cc(c(c(c1)Cl)CSc2c(c(sn2)/C=C/Nc3ccc(cc3)Cl)C#N)F 6C-074 Cc1c(c(ns1)S(=O)(=O)C)C#N 6C-076 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)Nc4ccc(cc4)Cl 6C-078 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)Nc4cccc(c4)C(F)(F)F 6C-079 Cc1nc(cs1)CSc2c(c(sn2)/C=C/N(C)C)C#N 6C-080 Cc1c(c(ns1)SC)C(=O)O 6C-081 Cc1nc(cs1)CSc2c(c(sn2)/C=C/Nc3ccc(cc3)Cl)C#N 6C-082 Cc1nc(cs1)CSc2c(c(sn2)/C=C/Nc3ccccc3)C#N 6C-083 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)NCc4ccccc4 6C-084 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)NCc4ccc(cc4)Cl 6C-085 c1cc[n+](c(c1)SCC#N)[O-] 6C-087 c1cc[n+](c(c1)SCC(=C(C#N)C#N)N)[O-] 6C-088 c1cc(c(cc1Cl)Cl)C(C#N)c2ccc(nn2)Cl 6D-001 c1cc(c(cc1Cl)Cl)Cc2ccc(nn2)O 6D-002 c1cc(c(cc1Cl)Cl)C(C#N)c2ccc(nn2)O 6D-003 c1cc(c(cc1Cl)Cl)Cc2ccc(nn2)Cl 6D-004 c1ccc(cc1)Oc2ccc(cc2)N3CSCC3=O 6D-005 c1ccc(cc1)Oc2ccc(cc2)N3CS(=O)CC3=O 6D-006 c1ccc(cc1)Oc2ccc(cc2)N3CS(=O)(=O)CC3=O 6D-007 CN(C)/C=C/1\C(=O)N(CS1=O)c2ccc(cc2)Oc3ccccc3 6D-009 c1ccc(cc1)/C=N/NC(=O)CC#N 6D-011 c1ccc(cc1)C(=O)NN/C=N\O 6D-013 CN(C)/C=C(\C#N)/C(=O)N/N=C/c1ccccc1 6D-014 CN(C)/C=N/NS(=O)(=O)c1ccccc1 6D-016 c1ccc(cc1)S(=O)(=O)NN/C=N\O 6D-017 c1cc(c(cc1N2CSCC2=O)Cl)Cl 6D-019 Cn1c(=O)c2c(ccs2)nc1SCc3ccccc3 6D-020 Cn1c(=O)c2c(ccs2)nc1SCC=C 6D-021 Cn1c(=O)c2c(ccs2)nc1SCC#C 6D-022 c1cc(c(cc1N2CS(=O)CC2=O)Cl)Cl 6D-023 c1cc(c(cc1N2CS(=O)(=O)CC2=O)Cl)Cl 6D-024 CSc1nc2ccsc2c(=O)n1c3ccccc3 6D-026 C=CCSc1nc2ccsc2c(=O)n1c3ccccc3 6D-027 C#CCSc1nc2ccsc2c(=O)n1c3ccccc3 6D-028 CN(C)/C=C/1\C(=O)N(CS1(=O)=O)c2ccc(c(c2)Cl)Cl 6D-029 c1csc2n1c(c(n2)Cl)[N+](=O)[O-] 6D-030 c1ccnc(c1)C(C#N)c2ccc(nn2)Cl 6D-031 c1cc(c(c(c1)Cl)/C=[N+]/2\CCC(=O)[N-]2)F 6D-033 CN(C)/C=N/C(=S)c1ccccc1 6D-035 c1ccc(cc1)c2ncc(s2)C(=O)c3ccccc3 6D-036 c1ccc(cc1)c2ncc(s2)C(=O)c3ccc(cc3)Cl 6D-037 CC(=O)c1cnc(s1)c2ccccc2 6D-038 c1ccc(cc1)C(=S)N/C=N/O 6D-040 c1cnccc1/C=[N+]/2\CCC(=O)[N-]2 6D-043 c1ccc(cc1)Sc2c(n3ccsc3n2)[N+](=O)[O-] 6D-045 c1cscc1/C=[N+]/2\CCC(=O)[N-]2 6D-047 c1cc(cnc1)N=C=S 6D-048 c1cc(cnc1)n2c(=O)c3c(ccs3)[nH]c2=S 6D-049 c1ccnc(c1)Cc2ccc(nn2)O 6D-050 c1cc(cnc1)/C=[N+]/2\CCC(=O)[N-]2 6D-051 CN(C)/C=N/C(=S)c1ccc(cc1)Cl 6D-052 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)[N+](=O)[O-])N3N=N3 6D-053 CSc1nc2ccsc2c(=O)n1c3cccnc3 6D-055 C=CCSc1nc2ccsc2c(=O)n1c3cccnc3 6D-056 CN(C)/C=C/1\C(=O)N(CS1(=O)=O)c2ccc(cc2)Oc3ccccc3 6D-057 Cc1c(c(nc(n1)c2ccccn2)O)Cl 6D-058 c1ccc(cc1)c2ncc(s2)C(=O)c3ccc(cc3)F 6D-059 c1cc(ccc1c2ncc(s2)C(=O)c3ccc(cc3)Cl)Cl 6D-060 Cc1c(c(nc(n1)c2ccccc2)O)Cl 6D-061 COc1ccc(cc1)N/C=C/2\C(=O)N(CS2(=O)=O)c3ccc(cc3)Oc4ccccc4 6D-062 Cc1c(c(nc(n1)c2ccccn2)Cl)Cl 6D-063 Cc1c(c(nc(n1)c2ccccc2)Cl)Cl 6D-064 c1ccc(cc1)C(=O)c2cnc(s2)c3ccc(cc3)Cl 6D-065 c1ccc2c(c1)c(on2)/C=C/c3ccc(cc3)[N+](=O)[O-] 6D-066 c1ccc(c(c1)/C=[N+]/2\CCC(=O)[N-]2)Cl 6D-068 c1ccc2c(c1)c(on2)/C=C/c3ccc(cc3)F 6D-070 c1ccnc(c1)Cc2ccc(nn2)Cl 6D-071 Cc1c(c(nc(n1)c2ccccn2)SCC(=O)OC)Cl 6D-072 Cc1c(c(nc(n1)c2ccccc2)SCC(=O)OC)Cl 6D-073 Cc1c(c(nc(n1)N)Cl)Cl 6D-075 COc1ccc(cc1)/C=C/c2c3ccccc3no2 6D-076 c1cc(c(cc1/C=[N+]/2\CCC(=O)[N-]2)Cl)Cl 6D-078 CC(=O)c1cnc(s1)c2ccc(cc2)Cl 6D-079 c1ccc(c(c1)C(=O)/C=C/c2c(cccc2Cl)F)N3N=N3 6D-080 Cc1c(c(nc(n1)c2ccccn2)SCC(=O)N(C)C)Cl 6D-081 Cc1c(c(nc(n1)c2ccccc2)SCC(=O)N(C)C)Cl 6D-082 c1ccc2c(c1)c(on2)/C=C/c3c(cccc3Cl)F 6D-084 Cn1c(c(c(n1)Cl)Cl)Oc2ccc(cc2)S(=O)(=O)Oc3ccccc3 6D-085 COC(=O)c1c(ccs1)OCc2ccccc2 6D-093 Cc1c(c(nc(n1)N)SCC(=O)OC)Cl 6D-094 COC(=O)c1c(ccs1)NC(=S)Nc2ccccn2 6D-095 CSc1nc2ccsc2c(=O)n1c3ccccn3 6D-096 C=CCSc1nc2ccsc2c(=O)n1c3ccccn3 6D-097 CCOC(=O)C(=Cc1c(ccs1)CBr)C(=O)OCC 6E-002 COc1ccc(cc1)n2cc3ccsc3c2 6E-004 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)N3CCC(CC3)C(=O)N 6E-005 c1ccc(cc1)Oc2ccc(cc2)n3cc4ccsc4c3 6E-007 c1cnc(nc1)N2CCC(CC2)C(=O)N 6E-008 CN(C)/C=N\C(=O)C1CCN(CC1)c2ncccn2 6E-009 c1cc(c(c(c1)Cl)CO/N=C/NC(=O)C2CCN(CC2)c3ncccn3)Cl 6E-012 c1cnc(nc1)N2CCC(CC2)C(=O)N/C=N/OCc3ccc(cc3)Cl 6E-013 c1cnc(nc1)N2CCC(CC2)C(=O)N/C=N/OCc3ccc(c(c3)Cl)Cl 6E-014 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)N)C(F)(F)F 6E-015 CN(C)/C=N/C(=O)C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 6E-016 c1cc(c(cc1Cl)Cl)CO/N=C/NC(=O)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 6E-018 c1cc(ccc1n2cc3ccsc3c2)OC(F)(F)F 6E-021 c1cc(nc(c1)F)NNC(=O)c2cccs2 6E-023 COc1ccc(cc1)C(=O)NNc2cccc(n2)F 6E-024 c1cc(nc(c1)F)NNC(=O)c2ccc(cc2Cl)Cl 6E-025 COc1ccc(cc1)c2ccn(n2)c3cccc(n3)F 6E-026 CSc1nc(n(n1)c2cccc(n2)F)N 6E-027 c1cc(ccc1CO/N=C(/c2ccncc2)\[NH3+])Cl.[Cl-] 6E-028 c1cc(cnc1)/C(=N/OCc2ccc(cc2)Cl)/[NH3+].[Cl-] 6E-029 CN(C)c1ccc(cc1)/C=[N+]/2\CCC(=O)[N-]2 6E-031 c1ccc(cc1)/C=C/C=[N+]/2\CCC(=O)[N-]2 6E-032 COc1ccc(cc1)/C=[N+]/2\CCC(=O)[N-]2 6E-034 c1cc(cc(c1)C(F)(F)F)/C=[N+]/2\CCC(=O)[N-]2 6E-035 c1cc(ccc1N)Oc2c(cc(cn2)C(F)(F)F)Cl 6E-036 c1cc(ccc1/C=[N+]/2\CCC(=O)[N-]2)F 6E-037 c1cc(ccc1n2cc3ccsc3c2)Oc4c(cc(cn4)C(F)(F)F)Cl 6E-038 c1cc(ccc1CONC(=O)N)Cl 6E-039 CN(C)/C=N/C(=O)NOCc1ccc(cc1)Cl 6E-041 Cc1cc(n(n1)c2cccc(n2)F)C 6E-042 CC(=NNc1ccc(nn1)Cc2ccc(cc2Cl)Cl)C 6E-044 c1cc(cc(c1)C(F)(F)F)CNc2ncc(cn2)C#N 6E-047 COc1ccc(cc1)CNc2ncc(cn2)C#N 6E-048 c1cc(oc1)CNc2ncc(cn2)C#N 6E-049 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ncc(cn4)C#N 6E-051 c1cc(c(cc1Cl)Cl)CNc2ncc(cn2)C#N 6E-053 CNC(=O)c1ccc(=O)n(c1)Cc2ccc(c(c2)Cl)Cl 6E-301S c1cc(c(cc1Cn2cc(ccc2=O)C(=O)N3CCOCC3)Cl)Cl 6E-302S CCN(CC)C(=O)c1ccc(=O)n(c1)Cc2ccc(c(c2)Cl)Cl 6E-303S CN1CCN(CC1)C(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 6E-304S c1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 6E-305S COC(=O)c1cccn(c1=O)Cc2ccc(cc2)C(F)(F)F 6E-306S COC(=O)c1cccn(c1=O)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F 6E-307S c1ccc(cc1)Cn2cccc(c2=O)C(=O)NCc3cccc(c3)C(F)(F)F 6E-308S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)O 6E-309S c1ccc(cc1)CNC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 6E-310S c1cc(c(=O)n(c1)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)O 6E-311S CN(C)C(=O)c1cccn(c1=O)Cc2ccc(cc2)C(F)(F)F 6E-314S CN(c1ccccc1)C(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 6E-315S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 6E-316S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F 6E-317S c1cc(cc(c1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F)C(F)(F)F 6E-318S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)Nc3ccc(cc3)C(F)(F)F 6E-319S CNC(=O)c1cccn(c1=O)Cc2ccc(cc2)C(F)(F)F 6E-320S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F 6E-321S c1cc(c(=O)n(c1)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)Nc3ccc(cc3F)F 6E-322S c1cc(cc(c1)NC(=O)c2cccn(c2=O)Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F 6E-323S c1cc(c(=O)n(c1)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)Nc3ccc(cc3)C(F)(F)F 6E-324S CNC(=O)c1cccn(c1=O)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F 6E-325S CN(C)CCNC(=O)c1cccn(c1=O)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F 6E-326S CN(C)CCNC(=O)c1cccn(c1=O)Cc2ccc(cc2)C(F)(F)F 6E-328S CN1CCN(CC1)C(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 6E-329S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)Nc3cc(cc(c3)Cl)Cl 6E-330S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)Nc3ccc(cc3Cl)Cl 6E-331S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)N3CCOCC3 6E-332S c1ccc(c(c1)C(F)(F)F)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 6E-333S c1ccc(cc1)CNC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 6E-335S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)NCc3ccc(cc3)Cl 6E-336S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)Nc3nccs3 6E-337S c1cc(cnc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 6E-338S COC(=O)c1c(ccs1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 6E-339S c1cc(cc(c1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)C(F)(F)F 6E-341S c1cc(ccc1C(F)(F)F)NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 6E-342S c1cc(ccc1NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl 6E-343S c1cc(c(cc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3F)F)Cl)Cl 6E-344S c1cc(ccc1NC(=O)c2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)F 6E-345S c1cc(cc(c1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3)Cl)C(F)(F)F 6E-346S c1cc(ccc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)C(F)(F)F)Cl 6E-347S c1cc(ccc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)Cl)Cl 6E-348S c1cc(ccc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3F)F)Cl 6E-349S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 6E-350S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)Nc3nccs3 6E-351S c1cc(cnc1)NC(=O)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 6E-352S COC(=O)c1c(ccs1)NC(=O)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 6E-353S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)NC3=NCCS3 6E-354S COC(=O)c1ccc(=O)n(c1)Cc2cccc(c2)C(F)(F)F 6E-355S COC(=O)c1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 6E-356S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)Nc3nncs3 6E-357S c1ccnc(c1)NC(=O)c2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 6E-358S c1cc(cc(c1)C(F)(F)F)Cn2cc(ccc2=O)C(=O)O 6E-359S c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)O)Cl 6E-360S c1cc(ccc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)OC(F)(F)F)Cl 6E-361S c1ccc(cc1)CNC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3)Cl 6E-362S c1cc(ccc1Cn2cc(ccc2=O)C(=O)NCCN3CCOCC3)Cl 6E-363S CN(c1ccccc1)C(=O)c2ccc(=O)n(c2)Cc3ccc(cc3)Cl 6E-364S CN(C)CCNC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2)Cl 6E-365S CN1CCN(CC1)C(=O)c2ccc(=O)n(c2)Cc3ccc(cc3)Cl 6E-366S CN(C)CCNC(=O)c1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 6E-367S COC(=O)c1ccc(=O)n(c1)Cc2ccc(cc2)C(F)(F)F 6E-368S COC(=O)c1ccc(=O)n(c1)Cc2cccc(c2)Cl 6E-369S c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)C(=O)NC3CC3 6E-370S CNC(=O)c1ccc(=O)n(c1)Cc2cccc(c2)C(F)(F)F 6E-374S c1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3cccc(c3)C(F)(F)F 6E-375S c1cc(cc(c1)C(F)(F)F)Cn2cc(ccc2=O)C(=O)Nc3cccc(c3)C(F)(F)F 6E-376S c1cc(cc(c1)C(F)(F)F)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3F)F 6E-377S c1cc(ccc1Cn2cc(ccc2=O)C(=O)O)C(F)(F)F 6E-378S c1ccc(c(c1)CSC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl)Cl 6E-500 c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)NC(=O)OCC(F)(F)F 6E-501 c1cc(cc(c1)SC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl)C(F)(F)F 6E-502 c1ccc(c(c1)SC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl)Cl 6E-503 c1cc(cnc1)OC(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 6E-504 c1ccc(cc1)SC(=O)c2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 6E-507 c1cc(c(=O)n(c1)Cc2ccc3c(c2)OC(O3)(F)F)C(=O)N=[N+]=[N-] 6E-510 C#CCOC(=O)Nc1cccn(c1=O)Cc2ccc3c(c2)OC(O3)(F)F 6E-511 c1cc(cnc1)OC(=O)Nc2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 6E-514 CC(C)N(Cc1ccccc1Cl)C(=O)Nc2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 6E-517 CC(C)N(c1ccc(cc1)Cl)C(=O)Nc2cccn(c2=O)Cc3ccc4c(c3)OC(O4)(F)F 6E-518 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)N=[N+]=[N-])Cl 6E-520 c1ccc(cc1)NC(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl 6E-521 c1cc(cc(c1)NC(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl)C(F)(F)F 6E-522 Cc1cccc(c1NC(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl)C 6E-523 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)Nc3ccc(cc3F)F)Cl 6E-524 c1ccnc(c1)CNC(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl 6E-525 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)NCc3ccncc3)Cl 6E-526 COC(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-527 C#CCOC(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-528 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)OCC(F)(F)F)Cl 6E-529 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)OCc3cccnc3)Cl 6E-530 CC(C)(C#C)OC(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-531 c1cc(cc(c1)OC(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl)C(F)(F)F 6E-532 CCOC(=O)CSC(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-533 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)N)Cl 6E-536 c1ccc(cc1)C(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl 6E-539 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)c3ccc(cc3Cl)Cl)Cl 6E-541 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)c3ccc(c(c3)Cl)Cl)Cl 6E-542 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)c3c(cccc3Cl)Cl)Cl 6E-544 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl 6E-545 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)C(Cl)(Cl)Cl)Cl 6E-546 CC(C)(C)C(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-547 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)C(F)(F)F)Cl 6E-548 CC(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-549 c1ccc(c(c1)C(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl)C(F)(F)F 6E-550 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)c3ccc(cc3)Cl)Cl 6E-551 c1ccc(c(c1)C(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl)Cl 6E-552 Cc1ccc(cc1)C(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl 6E-554 COc1ccc(cc1)C(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl 6E-555 c1ccc(c(c1)C(=O)Nc2cccn(c2=O)Cc3c(cccc3Cl)Cl)[N+](=O)[O-] 6E-556 c1ccc(cc1)NC(=O)Nc2ccc(=O)n(c2)Cc3c(cccc3Cl)Cl 6E-559 C#CCOC(=O)Nc1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 6E-560 c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)NC(=O)Nc3ccc(c(c3)F)F)Cl 6E-561 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)C3CC3)Cl 6E-562 CCCCC(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-563 CC(C)CC(=O)Nc1cccn(c1=O)Cc2c(cccc2Cl)Cl 6E-564 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)Cc3ccc(cc3)Cl)Cl 6E-565 c1cc(c(c(c1)Cl)Cn2cccc(c2=O)NC(=O)CCCCl)Cl 6E-566 CCOC(=O)Nc1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 6E-567 CC(C)(C)NC(=O)Nc1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 6E-568 c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)NC(=O)NCc3cccnc3)Cl 6E-569 CCn1cc(ccc1=O)[N+](=O)[O-] 6E-571 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc3ccc(cc3oc2=O)O 6E-902 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc3c(=O)[nH]c(=O)[nH]c3oc2=O 6E-903 COC(=O)/C(=C\Nc1cccc(c1)C(F)(F)F)/NC(=O)c2ccccc2 6E-907 CCOC(=O)c1cc(c(=O)oc1C(F)(F)F)NC(=O)c2cccc(c2)C(F)(F)F 6E-909 COc1ccc(cc1)c2c(c(=O)c3cc(ccc3o2)OC)C(=O)Nc4ccccc4 6E-910 COc1ccc2cc(c(=O)oc2c1)NC(=O)c3cccc(c3)C(F)(F)F 6E-912 COc1ccc(cc1)N/C=C(\C(=O)OC)/NC(=O)c2ccccc2 6E-913 COc1ccc(cc1)C(=O)Nc2cc3ccc(cc3oc2=O)OC 6E-914 COC(=O)/C(=C/N/C=C(\NC(=O)c1ccccc1)/C(=O)OC)/NC(=O)c2ccccc2 6E-917 c1ccc2c(c1)c3nnc(n3c(n2)Cl)c4ccc(cc4)Cl 6E-923 COC(=O)/C(=C\Nc1cccnc1)/NC(=O)c2ccccc2 6E-924 c1cc(cc(c1)Cl)C(=O)NCC(=O)O 6E-925 CN1CCN(CC1)c2nc3ccccc3c4n2c(nn4)c5ccc(cc5)Cl 6E-926 COC(=O)/C(=C/NC(=S)N/C=C(\NC(=O)c1ccccc1)/C(=O)OC)/NC(=O)c2ccccc2 6E-927 COC(=O)/C(=C\Nc1ccc(cc1)Oc2ccccc2)/NC(=O)c3ccccc3 6E-928 c1ccc2c(c1)c(nc(n2)Cl)N/N=C/c3ccc(cc3)Cl 6E-931 COC(=O)C(/C=N/OC)NC(=O)c1ccc(cc1Cl)Cl 6E-933 COC(=O)C(/C=N/OCc1ccc(cc1Cl)Cl)NC(=O)c2ccc(cc2Cl)Cl 6E-934 COC(=O)C(/C=N/OCc1ccc(cc1)[N+](=O)[O-])NC(=O)c2ccc(cc2Cl)Cl 6E-935 COC(=O)C(/C=N/OCc1c(cccc1Cl)Cl)NC(=O)c2ccc(cc2Cl)Cl 6E-936 CN(C)/C=C(\C(=O)OC)/NC(=O)c1cccc(c1)Cl 6E-937 COC(=O)C(/C=N/OCc1ccc(cc1Cl)Cl)NC(=O)c2cccc(c2)Cl 6E-939 COC(=O)C(/C=N/OCc1ccc(cc1)[N+](=O)[O-])NC(=O)c2cccc(c2)Cl 6E-940 CCOC(=O)c1c(=O)c2cc(ccc2oc1c3ccc(cc3)OC)OC 6E-941 COC(=O)C(/C=N/OCc1ccc(cc1)[N+](=O)[O-])NC(=O)c2ccc(cc2)C(F)(F)F 6E-942 c1ccc(cc1)NC(=O)CC(=O)Nc2ccccc2 6E-943 Cc1ccc(cc1)NC(=O)CC(=O)Nc2ccc(cc2)C 6E-944 COC(=O)C(/C=N/OC)NC(=O)c1ccc(cc1)C(F)(F)F 6E-948 CCOC(=O)CC(=O)Nc1ccc(cc1)C 6E-950 COC(=O)C(/C=N/OCc1c(cccc1Cl)Cl)NC(=O)c2cccc(c2)Cl 6E-951 c1ccc(cc1)NC(=O)/C=C/c2ccc(o2)c3ccc(cc3Cl)Cl 6F-002 c1cc(nc(c1)Cl)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 6F-004 CCOC(c1ccc(cc1)/C=C(\C#N)/C(=O)N)OCC 6F-005 c1ccc2c(c1)cc(o2)C(=O)c3ccc(o3)c4ccc(cc4Cl)Cl 6F-006 Cc1c(c(on1)/C=C/c2ccc(o2)c3ccc(cc3)Cl)[N+](=O)[O-] 6F-007 Cc1c(c(on1)/C=C/c2ccc(o2)c3cccc(c3)Cl)[N+](=O)[O-] 6F-008 Cc1c(c(on1)/C=C/c2ccc(o2)c3ccccc3Cl)[N+](=O)[O-] 6F-009 c1ccc2c(c1)c(n[nH]c2=O)Cc3ccc(o3)c4ccc(cc4)Cl 6F-011 c1ccc2c(c1)c(n[nH]c2=O)Cc3ccc(o3)c4cccc(c4)Cl 6F-012 c1ccc2c(c1)c(n[nH]c2=O)Cc3ccc(o3)c4ccccc4Cl 6F-014 c1ccn(c1)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 6F-015 CCOC(c1ccc(cc1)/C=C(/C#N)\C(=O)/N=C/N(C)C)OCC 6F-016 c1cc(ccc1c2ccc(o2)C=O)Cl 6F-017 c1cc[n+](c(c1)SCC(=O)c2ccc(cc2Cl)Oc3ccc(cc3)Cl)[O-] 6F-018 Cn1cccc1/C=C(/c2ccccc2)\OC 6F-019 CS/C(=N\C#N)/NOCc1c(cccc1Cl)Cl 6F-020 Cn1cc(cc1/C=C/C(=O)Nc2ccc(cc2Cl)Cl)C(=O)c3ccc(cc3Cl)Cl 6F-021 c1ccn(c1)c2c(cc(cn2)C(F)(F)F)Cl 6F-022 c1cc(cc(c1)Cl)c2ccc(o2)C=O 6F-024 c1ccc(c(c1)c2ccc(o2)C=O)Cl 6F-027 c1cc(c(cc1Cl)Cl)c2ccc(o2)c3csc(n3)N 6F-028 Cn1c(ccc1C(=O)C(Cl)(Cl)Cl)CC#N 6F-029 c1ccc2c(c1)/C(=C/c3ccc(o3)c4ccc(cc4)Cl)/OC2=O 6F-030 Cc1nc(cs1)c2ccc(o2)c3ccc(cc3Cl)Cl 6F-031 c1ccn(c1)c2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl 6F-032 c1ccc2c(c1)/C(=C/c3ccc(o3)c4cccc(c4)Cl)/OC2=O 6F-033 c1ccc(c(c1)c2ccc(o2)/C=C\3/c4ccccc4C(=O)O3)Cl 6F-035 CC(C)(C(=O)NN)n1cncn1 6F-037 C/C(=N/O)/c1ccccc1 6F-040 c1cc(c(cc1Cl)Cl)c2ccc(o2)c3csc(n3)CC#N 6F-041 CN(C)/C=C(\C#N)/c1nc(cs1)c2ccc(o2)c3ccc(cc3Cl)Cl 6F-043 c1cc[n+](cc1)C2C(C(=C(NC2=O)[S-])C#N)c3ccc(cc3)Cl 6F-044 c1cc(ccc1/C=C(\C#N)/c2nc(cs2)c3ccc(o3)c4ccc(cc4Cl)Cl)Cl 6F-045 C/C(=N\Oc1cccc(n1)F)/c2ccc(cc2)F 6F-046 C/C(=N\Oc1cccc(n1)F)/c2ccccc2 6F-047 c1ccnc(c1)C(=N)NNC(=O)C(=O)N 6F-048 CO/C(=C\c1ccc(o1)c2ccc(cc2)Cl)/c3ccccc3 6F-049 c1c(nc2c(c(nn2c1C(F)(F)F)CC#N)C#N)C(F)(F)F 6F-051 C/C(=N\Oc1cccc(n1)F)/c2ccc(cc2Cl)Cl 6F-052 c1ccc(cc1)/C=C(\C#N)/c2c(c3nc(cc(n3n2)C(F)(F)F)C(F)(F)F)C#N 6F-053 CN(C)/C=C(\C#N)/c1c(c2nc(cc(n2n1)C(F)(F)F)C(F)(F)F)C#N 6F-054 C/C(=N\Oc1cccc(n1)F)/c2ccc(cc2)Oc3ccccc3 6F-055 CSc1nc(n(n1)c2cccc(n2)Cl)N 6F-057 Cc1c(nc(s1)c2c(cccc2F)F)OCc3ccc(cc3)Cl 6F-059 Cn1cc(cc1/C=C(\C#N)/c2ccc(cc2)Cl)C(=O)c3ccc(cc3Cl)Cl 6F-061 c1ccc(cc1)N/C=C/c2nc(cs2)c3ccc(o3)c4ccc(cc4Cl)Cl 6F-065 CC(C)(c1nnc(n1C)S)n2cncn2 6F-066 c1cc(ccc1C(=O)O/N=C(\Cn2cncn2)/N)Cl 6F-068 c1ccc(cc1)c2nc3ccccc3n2OCc4ccc(cc4)Cl 6F-301S c1ccc(cc1)COn2c3ccccc3nc2c4ccccc4 6F-302S c1ccc(c(c1)c2nc3ccccc3n2O)Cl 6F-304S Cn1c(c(c(n1)C(F)(F)F)C#N)NCc2ccccc2 6F-305S Cn1c(c(c(n1)C(F)(F)F)C#N)Sc2cccc(c2)C(F)(F)F 6F-306S c1ccc(c(c1)NCc2ccc(cc2)Cl)[N+](=O)[O-] 6F-307S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)Cc2ccccc2 6F-308S Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2ccc(cc2)C#N 6F-309S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)C(c3ccccc3)c4ccccc4 6F-311S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCOCC2 6F-312S c1ccc(cc1)c2nc3ccccc3n2OCc4c(cccc4Cl)Cl 6F-313S c1ccc(cc1)c2nc3ccccc3n2OCc4ccc(c(c4)Cl)Cl 6F-314S c1ccc(cc1)c2nc3ccccc3n2OCc4ccc(cc4Cl)Cl 6F-315S c1ccc(cc1)c2nc3ccccc3n2OCc4c(cccc4Cl)F 6F-316S Cn1c(c(c(n1)C(F)(F)F)C#N)NCc2cccc(c2)OC 6F-317S Cn1c(c(c(n1)C(F)(F)F)C#N)NCc2cccnc2 6F-318S c1ccc(c(c1)Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F)Cl 6F-320S COc1ccc(cc1)Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F 6F-321S c1ccc2c(c1)nc(n2O)c3ccc(cc3)Cl 6F-322S c1ccc(cc1)c2nc3ccccc3n2OCc4cccc(c4)Cl 6F-323S c1ccc(cc1)c2nc3ccccc3n2OCc4cccc(c4)C(F)(F)F 6F-324S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3)C(F)(F)F 6F-325S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3F)F 6F-326S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)c2cccc(c2)C(F)(F)F 6F-327S Cn1c(c(c(n1)C(F)(F)F)C#N)S(=O)(=O)c2ccc(cc2)OC 6F-328S Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2cccc(c2)Cl 6F-329S Cc1ccc(cc1)Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F 6F-331S c1ccc(c(c1)c2nc3ccccc3n2OCc4cccc(c4)C(F)(F)F)Cl 6F-332S c1ccc(c(c1)c2nc3ccccc3n2OCc4ccc(cc4)Cl)Cl 6F-333S c1ccc(cc1)COn2c3ccccc3nc2c4ccccc4Cl 6F-334S CC(C)(C)c1ccc(cc1)Oc2c(c(nn2C)C(F)(F)F)C#N 6F-335S c1ccc2c(c1)nc(n2OCc3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl 6F-336S c1ccc2c(c1)nc(n2OCc3cccc(c3)Cl)c4ccc(cc4)Cl 6F-337S c1ccc(cc1)COn2c3ccccc3nc2c4ccc(cc4)Cl 6F-338S Cn1c(c(c(n1)C(F)(F)F)C#N)NCc2ccc(cc2)OC 6F-339S c1cc(ccc1NC(=O)c2cc(cc(c2)Cl)Cl)Cl 6F-341S Cc1cc(cc(c1)C(=O)Nc2ccc(c(c2)Cl)Cl)C 6F-344S c1ccc2c(c1)nc(n2OCc3ccc(cc3Cl)Cl)c4ccc(cc4)Cl 6F-347S c1ccc(c(c1)COn2c3ccccc3nc2c4ccc(cc4)Cl)Cl 6F-348S c1cc(c(cc1Cl)Cl)CS(=O)(=O)CC(CN2CCCC2=O)O 6F-351S c1ccc2c(c1)nc(n2OCc3ccc(cc3)Cl)c4ccc(cc4)Cl 6F-353S c1ccc2c(c1)nc(n2OCc3c(cccc3Cl)Cl)c4ccc(cc4)Cl 6F-354S c1cc(c(nc1)NCc2ccc(cc2)Cl)[N+](=O)[O-] 6F-355S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)Cl)Cl)Cl)Cl 6F-356S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)F)Cl)Cl)Cl 6F-357S Cc1ccc(cc1)c2nc3ccccc3n2O 6F-358S c1ccc2c(c1)nc(n2OCc3ccc(c(c3)Cl)Cl)c4ccc(cc4)Cl 6F-359S c1ccc2c(c1)nc(n2OCc3c(cccc3Cl)F)c4ccc(cc4)Cl 6F-360S c1ccc2c(c1)cnn(c2=O)c3c(cc(cc3Cl)C(F)(F)F)Cl 6F-361S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)c4ccc(cc4)F 6F-364S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)F)c4ccc(cc4)F 6F-365S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)OC(F)(F)F)Cl)Cl)Cl 6F-366S Cc1ccc(cc1)COn2c3ccccc3nc2c4ccc(cc4)Cl 6F-367S Cc1cc(cc(c1)COn2c3ccccc3nc2c4ccc(cc4)Cl)C 6F-368S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)OC(F)(F)F)c4ccc(cc4)F 6F-369S c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)C(F)(F)F)c4ccc(cc4)F 6F-371S Cc1c2ccccc2c(=O)n(n1)c3c(cc(cc3Cl)Cl)Cl 6F-372S Cc1c2ccccc2c(=O)n(n1)c3ccc(c(c3Cl)Cl)Cl 6F-373S Cc1c2ccccc2c(=O)n(n1)c3ccc(cc3Cl)C(F)(F)F 6F-374S Cc1c2ccccc2c(=O)n(n1)c3c(cc(cc3Cl)C(F)(F)F)Cl 6F-375S Cc1ccc(cc1)c2nc3ccccc3n2OCc4cccc(c4)C(F)(F)F 6F-378S Cc1ccc(cc1)c2nc3ccccc3n2OCc4ccccc4 6F-379S Cc1ccc(cc1)COn2c3ccccc3nc2c4ccccc4 6F-380S Cc1cc(cc(c1)COn2c3ccccc3nc2c4ccccc4)C 6F-381S COc1ccc(cc1)CNc2ccccc2[N+](=O)[O-] 6F-382S c1cc(ccc1c2n[nH]nn2)Cl 6F-900 c1ccc(cc1)c2nnn(n2)CC(=O)NN 6F-903 CN(C)/C=N/NC(=O)Cn1nc(nn1)c2ccccc2 6F-904 CN(C)/C=N/NC(=O)c1ccccc1 6F-905 c1ccc(cc1)C(=O)N/N=C/NOCc2ccc(cc2)Cl 6F-906 c1ccc(cc1)c2nnn(n2)CC(=O)N/N=C/NOCc3c(cccc3Cl)F 6F-907 c1cc(ccc1C2=N/C(=C/c3ccc(cc3Cl)Cl)/C(=O)O2)Cl 6F-909 CN(C)/C=N/NC(=O)c1ccncc1 6F-910 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Cl 6F-911 CN(C)/C=N/NC(=O)c1ccc(cc1)Cl 6F-913 c1cc(ccc1CON/C=N/NC(=O)c2ccc(cc2)Cl)Cl 6F-914 COc1ccc(cc1)N/C=N/NC(=O)c2ccc(cc2)Cl 6F-915 c1ccc(cc1)C(=O)/C=C\c2ccco2 6F-917 CCOC(=O)c1cc(c(nc1N)NNC(=O)c2ccncc2)C(=O)OCC 6F-918 c1cc(c(cc1Cl)Cl)CON/C=N/NC(=O)c2ccncc2 6F-919 c1cc(ccc1C(=O)N/N=C/NO)Cl 6F-921 CCOC(=O)c1cc(cc(n1)C(=O)OCC)N2CCN(CC2)c3ccc(cc3)OC 6F-922 C/C(=C\C(=O)c1ccccc1)/NCC#N 6F-923 c1ccnc(c1)c2ncc3c(n2)CCN(C3)c4ccc(cc4)[N+](=O)[O-] 6F-924 c1cc(ccc1N2CCc3c(cnc(n3)N)C2)[N+](=O)[O-] 6F-925 CCOC(=O)CC(=N)NNC(=O)c1ccc(cc1)Cl 6F-926 CCOC(=O)c1cc(c2nnc(n2c1N)c3ccncc3)C(=O)OCC 6F-927 CCOC(=O)c1cc(c2nnc(n2c1N)c3ccccc3)C(=O)OCC 6F-928 CCOC(=O)c1cc(c2nnc(n2c1N)c3ccc(cc3)Cl)C(=O)OCC 6F-929 CCOC(=O)/C=C(\N)/NNC=O 6F-931 CN(/C=C/1\C(=O)/C(=C\N(C)C)/CN(C1)c2ccc(cc2)[N+](=O)[O-])C 6F-932 CCOC(=O)C(=CNc1c[nH]c(c1C(=O)c2ccccc2)C)C(=O)OCC 6F-933 COc1ccc(cc1)N2CCN(CC2)C(=O)CC3(C4CC5CC(C4)CC3C5)c6ccc(cc6)Cl 6F-935 c1ccc(cc1)N2CCN(CC2)C(=O)CC3(C4CC5CC(C4)CC3C5)c6ccc(cc6)Cl 6F-936 c1cc(ccc1C2(C3CC4CC(C3)CC2C4)CC(=O)N5CCCCC5)Cl 6F-937 c1cc(ccc1C2(C3CC4CC(C3)CC2C4)CC(=O)N5CCCC5)Cl 6F-938 c1cc(ccc1C2(C3CC4CC(C3)CC2C4)CC(=O)N5CCOCC5)Cl 6F-939 c1ccc(cc1)CN2CCN(CC2)C(=O)CC3(C4CC5CC(C4)CC3C5)c6ccc(cc6)Cl 6F-940 C[NH+]1CCN(CC1)C(=O)CC2(C3CC4CC(C3)CC2C4)c5ccc(cc5)Cl.[Cl-] 6F-941 c1cc(ccc1C2(C3CC4CC(C3)CC2C4)CC(=O)NCCO)Cl 6F-942 CCOC(=O)c1cc(c2nncn2c1N)C(=O)OCC 6F-943 c1ccc2c(c1)c(c([nH]2)C(=O)NN)N 6F-945 c1ccc(cc1)NC(=O)OCCNC(=O)CC2(C3CC4CC(C3)CC2C4)c5ccc(cc5)Cl 6F-946 c1cc(ccc1C2(C3CC4CC(C3)CC2C4)CC(=O)NCCOC(=O)Nc5ccc(cc5)Cl)Cl 6F-947 c1cc(nc(c1)Cl)n2cc3c(n2)CCN(C3)c4ccc(cc4)[N+](=O)[O-] 6F-949 CCOC(=O)C(=CNc1cn(c(c1C(=O)c2ccccc2)C)C)C(=O)OCC 6F-950 c1cc(ccc1CO/N=C/C2CN(CC(C2=O)/C=N\OCc3ccc(cc3)Cl)c4ccc(cc4)[N+](=O)[O-])Cl 6F-951 CCOC(=O)CC(=N)NNC(=O)OC 6F-952 c1cc(ccc1n2cc3c(n2)CCN(C3)c4ccc(cc4)[N+](=O)[O-])F 6F-953 CCOC(=O)c1ccccc1C(=O)C 6F-954 CCOC(=O)c1ccccc1C(=O)CBr 6F-955 CCOC(=O)c1ccccc1C(=O)CN2CCN(CC2)c3ccc(cc3)OC 6F-956 CCOC(=O)c1cc([nH]c1NNC(=O)OC)c2ccc(c(c2)Cl)Cl 6F-958 COC(=O)N1C(=O)C2C(=N1)NCC2(c3ccccc3)O 6F-959 CCOC(=O)C(=CNc1cn(c(c1C(=O)c2ccccc2)C)Cc3ccc(cc3)F)C(=O)OCC 6F-960 COc1ccc(cc1)NC(=O)NCC2(C3CC4CC(C3)CC2C4)c5ccccc5 6F-961 Cc1ccc(cc1)CO/N=C/C2CN(CC(C2=O)/C=N\OCc3ccc(cc3)C)c4ccc(cc4)[N+](=O)[O-] 6F-963 c1c(cnc(n1)N)C#N 6G-001 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(\c2c(cc(cn2)C(F)(F)F)Cl)/N 6G-003 c1ccc(cc1)C(=O)O/N=C(\c2c(cc(cn2)C(F)(F)F)Cl)/N 6G-004 c1ccc(cc1)NC(=O)O/N=C(\c2c(cc(cn2)C(F)(F)F)Cl)/N 6G-005 c1cc(cc(c1)C(F)(F)F)c2nc(no2)c3c(cc(cn3)C(F)(F)F)Cl 6G-006 c1ccc(cc1)c2nc(no2)c3c(cc(cn3)C(F)(F)F)Cl 6G-007 c1cc(cc(c1)N2CCN(CC2)c3cc(cnc3C#N)C(F)(F)F)C(F)(F)F 6G-011 c1cc(cnc1)COc2cc(cnc2C#N)C(F)(F)F 6G-012 CC1C(=N/C(=C\C(=S)N)/S1)O 6G-014 c1ccc(cc1)C(C#N)c2ccccc2C#N 6G-015 CO/N=C/Nc1ncc(cn1)C#N 6G-017 c1ccc(cc1)N2C(=O)C3C(C2=O)ON=C3c4c(cc(cn4)C(F)(F)F)Cl 6G-018 c1ccc(cc1)c2c(nnn2c3cc(cnc3C#N)C(F)(F)F)C(=O)c4ccccc4 6G-019 Cc1cc(n(n1)C2CCS(=O)(=O)C2)C 6G-021 c1ccc(cc1)C(C#N)c2cccc(c2C#N)F 6G-023 c1ccc(cc1)c2cnn(c2N)C3CCS(=O)(=O)C3 6G-024 c1ccc(cc1)c2ccnn2C3CCS(=O)(=O)C3 6G-025 Cn1cccc1C(C#N)c2ccccc2C#N 6G-027 c1c(cnc(c1Cl)N2CCCC2=O)C(F)(F)F 6G-028 c1c(cnc(c1N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C#N)C(F)(F)F 6G-029 c1cc(ccc1O)Oc2cc(cnc2C#N)C(F)(F)F 6G-031 c1ccc(c(c1)C#N)C(C#N)c2ccc(cc2)Cl 6G-033 c1cc2c(ccc(c2nc1)Oc3cc(cnc3C#N)C(F)(F)F)Cl 6G-034 c1cc(ccc1NC(=O)O/N=C(\c2c(cc(cn2)C(F)(F)F)Cl)/N)Cl 6G-035 c1cc2cccnc2c(c1)Oc3cc(cnc3C#N)C(F)(F)F 6G-036 CN(/C=c\1/n(c(=O)/c(=C\N(C)C)/n(c1=O)c2ncc(cc2Cl)C(F)(F)F)c3ncc(cc3Cl)C(F)(F)F)C 6G-038 c1cc(c(cc1NC(=O)O/N=C(/c2c(cc(cn2)C(F)(F)F)Cl)\N)Cl)Cl 6G-039 c1ccc(cc1)C(C#N)c2ccccc2C(=O)c3ccccc3 6G-040 c1ccc(cc1)C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 6G-041 c1ccc(c(c1)C#N)C(C#N)c2c(cccc2Cl)F 6G-042 c1ccc(cc1)C(C#N)c2ccc(cc2)C(=O)c3ccccc3 6G-043 c1cc2nnnn2c3c1c(cc(n3)C(F)(F)F)C(F)(F)F 6G-044 CN(C)/C=C/1\CCN(C1=O)c2c(cc(cn2)C(F)(F)F)Cl 6G-045 Cc1cc(n(n1)c2nnc(nn2)NCc3ccccc3)C 6G-047 CC[NH+](CC)CC.c1c(cnc(c1Cl)NNC(=S)[S-])C(F)(F)F 6G-048 c1ccc(c(c1)COc2cc(cnc2C#N)C(F)(F)F)Cl 6G-049 c1ccc(cc1)C(C#N)c2ccc(cc2)C(=O)c3ccc(cc3)F 6G-050 c1cc(ccc1C(=O)CSC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl 6G-051 c1ccc(cc1)C(c2ccc(cc2)C(=O)c3ccccc3)C(=O)N 6G-052 COc1cc(cnc1C#N)C(F)(F)F 6G-053 COC(c1ccnn1c2c(cc(cn2)C(F)(F)F)Cl)OC 6G-055 c1cc(c(c(c1)Cl)CO/N=C/c2ccnn2c3c(cc(cn3)C(F)(F)F)Cl)Cl 6G-056 c1ccc(cc1)C(C#N)c2ccc(cc2)C(c3ccccc3)O 6G-060 C/C(=C\C(=O)C(F)(F)F)/OC 6G-061 c1ccc(cc1)C(C#N)c2cccc(n2)Cl 6G-065 Cc1cc(n(n1)c2nnc(nn2)N3CCN(CC3)c4ccc(cc4)F)C 6G-071 CO/N=C/c1ccnn1c2c(cc(cn2)C(F)(F)F)Cl 6G-072 C1COCCN1C(=O)CC(=O)N2CCOCC2 6G-075 c1ccc(cc1)OC(C(=O)Nc2ccc(cc2)Cl)(F)F 6G-301S c1ccc(cc1)OC(C(=O)Nc2ccc(cc2Cl)Cl)(F)F 6G-302S CCOc1ccccc1NC(=O)c2ccc(nc2)n3cncn3 6G-303S Cc1cccc(c1NC(=O)c2ccc(nc2)n3cncn3)C 6G-304S c1ccc(cc1)OC(C(=O)Nc2ccc(c(c2)Cl)Cl)(F)F 6G-307S c1ccc(cc1)OC(C(=O)Nc2ccc(cc2)OC(F)(F)F)(F)F 6G-308S c1cc(ccc1NC(=O)c2c(snn2)Sc3ccc(cc3)Cl)F 6G-313S c1cc(ccc1Sc2c(nns2)C(=O)Nc3ccc(cc3F)F)Cl 6G-314S CCc1cccc(c1NC(=O)c2ccc(nc2)n3cncn3)CC 6G-317S c1cc(ccc1NC(=O)c2c(snn2)S(=O)(=O)c3ccc(cc3)Cl)F 6G-318S c1cc(ccc1S(=O)(=O)c2c(nns2)C(=O)Nc3ccc(cc3F)F)Cl 6G-319S c1cc(c(c(c1)F)NC(=O)c2ccc(nc2)n3cncn3)F 6G-320S c1ccc(cc1)OC(C(=O)N2CCCC2)(F)F 6G-321S c1ccc(c(c1)NC(=O)c2ccc(nc2)n3cncn3)F 6G-322S c1ccc(cc1)OC(C(=O)N2CCOCC2)(F)F 6G-323S CCOC(=O)C(Oc1cccc(c1)C(F)(F)F)(F)F 6G-324S CN1CCN(CC1)C(=O)C(Oc2ccccc2)(F)F 6G-327S c1ccc(cc1)/C=N/n2cc(nc2N)c3ccc(cc3)Br 6G-330S c1ccc(cc1)OC(C(=O)Nc2ccc(cc2F)F)(F)F 6G-331S c1ccc(cc1)NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F 6G-332S c1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)F)(F)F)C(F)(F)F 6G-333S c1cc(cc(c1)OC(C(=O)Nc2ccc(cc2F)F)(F)F)C(F)(F)F 6G-334S c1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)Cl)(F)F)C(F)(F)F 6G-335S CC(C)(CCC(=O)c1cccs1)[N+](=O)[O-] 6G-336S c1cc(cc(c1)NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F)C(F)(F)F 6G-337S c1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)OC(F)(F)F)(F)F)C(F)(F)F 6G-338S c1cc(cc(c1)OC(C(=O)Nc2ccc(c(c2)Cl)Cl)(F)F)C(F)(F)F 6G-343S c1cc(cc(c1)OC(C(=O)Nc2ccc(cc2Cl)Cl)(F)F)C(F)(F)F 6G-344S COc1ccc(cc1)NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F 6G-345S c1ccc(cc1)OC(C(=O)Nc2ccc(cc2)F)(F)F 6G-349S c1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)Br)(F)F)C(F)(F)F 6G-350S Cc1ccc(cc1)NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F 6G-351S c1cc(cc(c1)OC(C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)(F)F)C(F)(F)F 6G-352S CC(C)(CCC(=O)c1ccc(cc1)Cl)[N+](=O)[O-] 6G-353S CC(C)(CCC(=O)c1ccc(c(c1)OC)OC)[N+](=O)[O-] 6G-355S c1ccc(c(c1)C(F)(F)F)NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F 6G-365S c1cc(cc(c1)OC(C(=O)N)(F)F)C(F)(F)F 6G-370S CN1CCN(CC1)C(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F 6G-371S c1cc(cc(c1)OC(C(=O)Nc2[nH]cnn2)(F)F)C(F)(F)F 6G-373S c1ccc(cc1)C(=O)CCC(C(=O)N)S(=O)(=O)c2ccccc2 6G-374S CC1(CCC(=[N+]1[O-])c2cccs2)C 6G-375S CC1(CCC(=[N+]1[O-])c2ccc(cc2)Br)C 6G-376S CCc1cccc(c1NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F)CC 6G-378S c1c(nc(nc1O)S)C(F)(F)F 6G-379S CN(C)c1nc(cc(n1)O)C(F)(F)F 6G-380S CSc1nc(cc(n1)O)C(F)(F)F 6G-381S c1cc(cc(c1)OC(C(=O)Nc2c(cccc2Cl)Cl)(F)F)C(F)(F)F 6G-383S Cc1ccc(c(c1)C)NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F 6G-384S c1ccc(c(c1)NC(=O)C(Oc2cccc(c2)C(F)(F)F)(F)F)F 6G-385S CC(C)(CCC(=O)c1ccc(c(c1)Cl)Cl)[N+](=O)[O-] 6G-386S CC(C)(CCC(=O)c1ccc(cc1)OC)[N+](=O)[O-] 6G-387S c1cc(cc(c1)OC(C(=O)Nc2ccc(cc2)C(F)(F)F)(F)F)C(F)(F)F 6G-388S CC(C)(CCC(=O)c1ccc(cc1)Br)[N+](=O)[O-] 6G-391S CN(C)c1nc(cc(n1)Sc2ccc(cc2)Cl)C(F)(F)F 6G-393S CN(C)c1nc(cc(n1)Sc2ccc(c(c2)Cl)Cl)C(F)(F)F 6G-395S c1ccc(cc1)OCCSc2ccc(cc2)Cl 6G-396S c1ccc(cc1)OCCSc2cccc(c2)C(F)(F)F 6G-397S c1ccc(cc1)OCCCCSc2ccccc2 6G-398S CN(C)c1nc(cc(n1)Sc2ccc(cc2Cl)Cl)C(F)(F)F 6G-400S CN(C)c1nc(cc(n1)Sc2ccc(cc2)Br)C(F)(F)F 6G-401S CN(C)c1nc(cc(n1)Oc2ccc(cc2)Cl)C(F)(F)F 6G-402S CC1(CCC(=[N+]1[O-])c2ccc(c(c2)Cl)Cl)C 6G-403S CC1(CCC(=[N+]1[O-])c2ccc(cc2)OC)C 6G-404S c1cc(ccc1NC(=O)C(Oc2ccc(cc2)F)(F)F)Cl 6G-405S CN(C)c1nc(cc(n1)Sc2ccc3ccccc3c2)C(F)(F)F 6G-406S Cc1ccc(cc1)Oc2cc(nc(n2)N(C)C)C(F)(F)F 6G-407S c1ccc(cc1)OCCCCS(=O)(=O)c2cccc(c2)Cl 6G-408S c1ccc(cc1)OCCS(=O)(=O)c2ccc(cc2)Cl 6G-409S c1ccc(cc1)OCCS(=O)c2ccc(cc2)Cl 6G-410S c1cc(cc(c1)NC(=O)C(Oc2ccc(cc2)F)(F)F)C(F)(F)F 6G-411S Cc1ccc(cc1)NC(=O)C(Oc2ccc(cc2)F)(F)F 6G-412S c1ccc(cc1)OCCSc2ccc(cc2)Br 6G-414S c1ccc(cc1)OCCCCSc2ccc(cc2)Br 6G-415S COC(=O)C(Oc1ccc(cc1)F)(F)F 6G-416S c1ccc(cc1)SCCCCSc2ccccc2 6G-417S c1cc(ccc1SCCCCSc2ccc(cc2)Cl)Cl 6G-418S CN(C)c1nc(cc(n1)Oc2ccc(cc2)OC)C(F)(F)F 6G-419S CN(C)c1nc(cc(n1)Oc2ccc(cc2)[N+](=O)[O-])C(F)(F)F 6G-420S c1cc(ccc1OC(C(=O)Nc2ccc(c(c2)Cl)Cl)(F)F)F 6G-421S c1cc(ccc1OC(C(=O)Nc2ccc(cc2F)F)(F)F)F 6G-422S COc1ccc(cc1)NC(=O)C(Oc2ccc(cc2)F)(F)F 6G-424S c1cc(ccc1NC(=O)C(Oc2ccc(cc2)F)(F)F)OC(F)(F)F 6G-425S Cc1ccc(cc1)SCCOc2ccccc2 6G-426S c1cc(cc(c1)OCCCSc2ccc(cc2)Cl)C(F)(F)F 6G-427S c1cc(ccc1OC(C(=O)N2CCOCC2)(F)F)F 6G-428S CN(C)c1nc(cc(n1)Oc2ccc(cc2)C#N)C(F)(F)F 6G-429S Cc1ccc(cc1)Sc2cc(nc(n2)N(C)C)C(F)(F)F 6G-430S CN(C)c1nc(cc(n1)Oc2cccc(c2)C(F)(F)F)C(F)(F)F 6G-431S CN(C)c1nc(cc(n1)Oc2cc(cc(c2)Cl)Cl)C(F)(F)F 6G-432S C=CCNC(=O)C(Oc1ccc(cc1)F)(F)F 6G-433S c1ccc(cc1)S(=O)(=O)CCCCS(=O)(=O)c2ccccc2 6G-434S c1cc(ccc1S(=O)CCCCS(=O)c2ccc(cc2)Cl)Cl 6G-435S c1cc(ccc1S(=O)(=O)CCCCS(=O)(=O)c2ccc(cc2)Cl)Cl 6G-436S CCCNC(=O)C(Oc1ccc(cc1)F)(F)F 6G-437S c1cc(ccc1OC(C(=O)N2CCCC2)(F)F)F 6G-438S Cc1ccc(cc1)S(=O)CCOc2ccccc2 6G-439S Cc1ccc(cc1)S(=O)(=O)CCOc2ccccc2 6G-440S CN(C)c1nc(cc(n1)Oc2cccc(c2Cl)Cl)C(F)(F)F 6G-441S CN(C)c1nc(cc(n1)Oc2c(cccc2Cl)Cl)C(F)(F)F 6G-442S CCCCNC(=O)C(Oc1ccc(cc1)F)(F)F 6G-443S c1cc(cc(c1)OCCCS(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F 6G-445S CCNc1nc(cc(n1)O)C(F)(F)F 6G-446S c1cc(cc(c1)OC(C(=O)NCc2ccc(cc2)Cl)(F)F)C(F)(F)F 6G-447S CN1CCN(CC1)C(=O)C(Oc2ccc(cc2)F)(F)F 6G-448S c1cc(cc(c1)OCCCS(=O)(=O)c2ccc(c(c2)Cl)Cl)C(F)(F)F 6G-451S c1cc(cc(c1)OCCCS(=O)(=O)c2ccc(cc2)Br)C(F)(F)F 6G-452S c1ccc(cc1)C(C(=O)NO)N 6G-453S Cc1ccc(cc1)SCCCSc2ccc(cc2)C 6G-457S CC(C)OC(=O)c1cccnc1N2CCN(CC2)C(c3ccccc3)c4ccccc4 6G-458S CC(C)OC(=O)c1cccnc1N2CCN(CC2)c3ccc(cc3)F 6G-459S CC(C)OC(=O)c1cccnc1N2CCN(CC2)c3ccccc3 6G-461S CC(C)OC(=O)c1cccnc1N2CCN(CC2)Cc3ccccc3 6G-462S CC(C)OC(=O)c1cccnc1N2CCN(CC2)c3ccccc3F 6G-466S c1ccc(cc1)SCCOc2ccc(cc2Cl)Cl 6G-467S c1cc(ccc1SCCOc2ccc(cc2Cl)Cl)Cl 6G-468S COC(=O)c1cccnc1N2CCN(CC2)c3ccccc3F 6G-469S COC(=O)c1cccnc1N2CCN(CC2)c3ccc(cc3)F 6G-470S COC(=O)c1cccnc1N2CCN(CC2)C(c3ccccc3)c4ccccc4 6G-471S CC(C)OC(=O)c1cccnc1N2CCN(CC2)c3cccc(c3)Cl 6G-472S c1c(cnc(c1Cl)N2CCN(CC2)CCN)C(F)(F)F 6G-900 c1cc(ccc1C(=O)NCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 6G-901 Cc1ccc(cc1)C=C(C#N)C#N 6G-903 c1c(cnc(c1Cl)N2CCC3(CC2)C4=C(CCN(C4)c5c(cc(cn5)C(F)(F)F)Cl)C(=C(C3(C#N)C#N)N)C#N)C(F)(F)F 6G-905 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)N)Cl 6G-906 c1cc(ccc1S(=O)(=O)NCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 6G-907 c1cc(ccc1NC(=O)NCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 6G-908 CCOC(=O)C1C(C2c3ccccc3CCN2O1)(C(F)(F)F)O 6G-909 CC(=O)CC(=O)Nc1cccc(c1)F 6G-910 CCOC(=O)NCCN1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 6G-911 C/C(=C/C(=O)Nc1cccc(c1)F)/N2CCCC2 6G-912 CC1(CN(C2(N1)CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)c4ccc(cc4Cl)Cl)C 6G-914 CN1[C@@H]([C@@H]2[C@H](O1)C(=O)N(C2=O)c3ccccc3)c4ccccc4 6G-915 CN1[C@@H]([C@@H]2[C@H](O1)C(=O)N(C2=O)c3cccc(c3)C(F)(F)F)c4ccccc4 6G-916 CC1=CSC2=[N+](CCN12)CC(=O)C.[Cl-] 6G-917 CCOC(=O)c1c(c(on1)C)C(=O)Nc2cccc(c2)F 6G-918 Cc1c(c(no1)C(=O)N)C(=O)Nc2cccc(c2)F 6G-919 c1ccc(cc1)CNC(=O)/C=C\C(=O)O 6G-920 c1cc(c(cc1Cl)Cl)NC(=O)/C=C\C(=O)O 6G-921 C1COCCN1C(=O)CC(=O)C(F)(F)F 6G-922 C1CCN(C1)/C(=C/C(=O)N2CCOCC2)/C(F)(F)F 6G-923 c1ccc(cc1)CN2C(=O)C=CC2=O 6G-925 Cc1c(c(no1)C#N)C(=O)Nc2cccc(c2)C(F)(F)F 6G-926 CCOC(=O)CC1(CCCC1=O)C(=O)OCC 6G-927 c1c(cnc(c1Cl)NCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 6G-928 c1c(cnc(c1Cl)N2CCN(CC2)CCNC(=O)N)C(F)(F)F 6G-929 CN(C)/C=N/C(=O)NCCN1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 6G-930 CN1[C@H]2c3c4ccccc4ccc3OC[C@H]2CO1 6G-932 CC1(CC(=O)N(C(=O)C1)CCCCN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C 6G-933 CCOC(=O)C1=NOC2C1C(=O)N(C2=O)c3ccc(cc3)Cl 6G-935 CC(=O)CC(=O)N1CCOCC1 6G-939 CC(=O)N(C)[C@@H]1c2c3ccccc3ccc2OC[C@@H]1COC(=O)C 6G-940 CC(=O)N[C@@H]1c2c3ccccc3ccc2OC[C@@H]1COC(=O)C 6G-941 c1ccc2c(c1)ccc3c2[C@H]([C@H](CO3)CO)NC(=O)Nc4ccc(cc4)Cl 6G-942 c1ccc2c(c1)ccc3c2[C@H]([C@H](CO3)CO)NC(=S)Nc4ccc(cc4)[N+](=O)[O-] 6G-943 C/C(=C\C(=O)N1CCOCC1)/N2CCCC2 6G-944 COc1cccc(c1OCC=C)C=O 6G-945 CN1[C@H]2c3cccc(c3OC[C@H]2CO1)OC 6G-947 c1ccc2c(c1)ccc3c2[C@@H]4[C@H](CO3)COC(N4)c5ccc(cc5)Cl 6G-948 CN1[C@@H]([C@@H]2[C@H](O1)C(=O)N(C2=O)c3cccc(c3)C(F)(F)F)c4ccc(cc4)OC 6G-949 CN1C(CC(O1)CNc2c(cc(cn2)C(F)(F)F)Cl)c3ccccc3 6G-951 c1ccc(cc1)N2CCN(CC2)c3nc4ccccc4c5n3c(nn5)c6ccc(cc6)Cl 6G-956 COC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3cccnc3 6H-002 COc1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)OC 6H-005 c1ccnc(c1)C(C#N)N2CCOCC2 6H-006 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)OC 6H-007 c1ccc2c(c1)CCN(C2CC#N)C(=O)N 6H-008 c1ccc2c(c1)CCNC2C3=C(CCCC3=O)O 6H-012 CC1(CC(=C(C(=O)C1)C2c3ccccc3CCN2)O)C 6H-013 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)O 6H-014 c1ccc2c(c1)CCN3C2C/C(=N\O)/CC3=O 6H-015 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c3ccccc3c2=O)C(=O)OC 6H-017 c1ccc2c(c1)CCNC2Cc3c(cc(cn3)C(F)(F)F)Cl 6H-018 c1ccc(cc1)NC(=O)N2CCc3ccccc3C2Cc4c(cc(cn4)C(F)(F)F)Cl 6H-019 COC(=O)C1CC(=O)N(C1)Cc2ccccc2 6H-020 Cc1nc(c(s1)C(=O)NCc2ccc(cc2)OC)C(F)(F)F 6H-021 CC(=O)/C=C/c1c(cccc1Cl)F 6H-022 CN(C)/C=C(/c1c(cc(cn1)C(F)(F)F)Cl)\C(=O)C(F)(F)F 6H-023 c1cc(ccc1C2CC(=O)CC(=O)C2)F 6H-024 CC1=C(CC(=O)N1Cc2ccccc2)C(=O)OC 6H-025 c1cc(c(c(c1)Cl)C2CC(=CC(=O)C2)O)F 6H-026 c1ccc2c(c1)CCNC2C3=C(CC(CC3=O)c4ccc(cc4)F)O 6H-027 c1ccc2c(c1)CCNC2C3=C(CC(CC3=O)c4c(cccc4Cl)F)O 6H-028 CC(c1ccc(cc1)Cl)N 6H-029 COc1ccc(cc1)N2CC(=CC2=O)c3ccc(cc3)F 6H-032 Cn1c(cnc1SCC(=O)c2cccc(c2)C(F)(F)F)C(=O)OC 6H-033 c1cc(oc1)c2ccnc3n2nc(n3)N 6H-034 c1cc(sc1)c2ccnc3n2nc(n3)N 6H-035 Cn1c(cnc1SCC(=O)c2ccccc2)C(=O)OC 6H-036 CC(=O)/C=C/c1c(nc2n1ccs2)c3ccc(cc3)Cl 6H-037 c1cc(cnc1)c2ccnc3n2nc(n3)N 6H-038 c1ccc(cc1)CN2CC(CC2=O)C(=O)N 6H-040 c1ccc(cc1)CN2CC(CC2=O)C(=O)NN 6H-041 Cc1nc(c(s1)C(=O)NCc2ccccc2Cl)C(F)(F)F 6H-042 Cc1nc(c(s1)C(=O)NC(C)c2ccc(cc2)Cl)C(F)(F)F 6H-043 c1cc(ccc1/C=C/c2ccnc3n2nc(n3)N)F 6H-044 c1cc(ccc1c2cnc3nc(nn3c2N)N)F 6H-045 Cc1nc(c(s1)C(=O)NCc2cccc(c2)C(F)(F)F)C(F)(F)F 6H-046 c1ccn(c1)c2nc3nccc(n3n2)/C=C/c4ccc(cc4)F 6H-047 CN(C)/C=C(/c1c(c(no1)c2ccccc2Cl)C(=O)OC)\C(=O)C(F)(F)F 6H-048 CCOC(=O)c1c(sc(=S)s1)SCc2ccc(cc2)F 6H-049 CCOC(=O)c1c(sc(=S)s1)SCc2cccc(c2)C(F)(F)F 6H-050 CCOC(=O)c1c(sc(=S)s1)SCc2cccc(c2)C#N 6H-051 COc1ccc(cc1)N2C(=O)CC(=C2/C=N/OC)c3ccc(cc3)F 6H-052 COc1ccc(cc1)N2C(C(=CC2=O)c3ccc(cc3)F)/C=N/O 6H-053 COc1ccc(cc1)N\2C(=O)C=C(/C2=C/Nc3ccc(cc3)Cl)c4ccc(cc4)F 6H-054 CN(C)/C=N\c1nc2nccc(n2n1)/C=C/c3ccc(cc3)F 6H-055 CO/N=C/Nc1nc2nccc(n2n1)/C=C/c3ccc(cc3)F 6H-056 c1c(cnc(c1Cl)c2cnc3c(cnn3c2)C#N)C(F)(F)F 6H-057 Cn1c(cnc1Sc2ccc(nn2)Cl)C(=O)OC 6H-059 c1ccc2c(c1)CCNC2CC(=O)Nc3ccc(cc3)Cl 6H-060 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CC3c4ccccc4CCN3 6H-061 CN(C)/C=C/1\C(=C(N(C1=O)c2ccc(cc2)OC)/C=N/OC)c3ccc(cc3)F 6H-062 c1ccn(c1)c2nc3nccc(n3n2)c4cccs4 6H-063 CCOC(=O)c1c(sc(=S)s1)SCc2c(cc(cn2)C(F)(F)F)Cl 6H-064 c1ccc(c(c1)c2ncnn2c3c(cc(cn3)C(F)(F)F)Cl)n4ccnc4 6H-067 c1ccc(c(c1)c2nc[nH]n2)n3ccnc3 6H-068 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)N(C)C 6H-070 c1cc(ccc1NC(=O)CC(=O)O)F 6H-071 CN(C)/C=C/C(=O)Nc1ccc(cc1)F 6H-073 CO/N=C\CC(=O)Nc1ccc(cc1)F 6H-074 c1cc(sc1)/C=C/c2ccnc3n2nc(n3)N 6H-075 c1cc(sc1)c2cnc3nc(nn3c2N)N 6H-077 c1ccc(c(c1)CN2C(=O)CS(=O)CC2=O)Cl 6H-301S c1ccc(c(c1)CN2C(=O)CS(=O)(=O)CC2=O)Cl 6H-302S c1cc(c(cc1F)F)NC(=O)CSCC(=O)O 6H-303S c1ccc(cc1)C(=O)Nc2ccsc2C(=O)O 6H-304S c1cc(c(cc1NC(=O)CS(=O)(=O)CC(=O)O)Cl)Cl 6H-305S CC(=O)Nc1ccsc1C(=O)OC 6H-306S c1ccc(c(c1)CNC(=O)CS(=O)CC(=O)O)Cl 6H-307S c1ccc(c(c1)CNC(=O)CS(=O)(=O)CC(=O)O)Cl 6H-308S COc1ccc(cc1)N2C(=O)CS(=O)(=O)CC2=O 6H-309S c1cc(c(cc1CNC(=O)CS(=O)(=O)CC(=O)O)Cl)Cl 6H-310S CC(C)(C)c1cc(c(c(n1)N)C#N)c2ccccc2 6H-311S c1cc(c(cc1Cl)Cl)NC(=O)CS(=O)(=O)CC(=O)O 6H-312S c1cc(c(cc1Cl)Cl)NC(=O)CS(=O)CC(=O)O 6H-313S Cc1c(c(c(nc1c2ccccc2)N)C#N)c3ccc(cc3)OC 6H-314S CC(C)(C)c1cc(c(c(n1)N)C#N)c2ccc(cc2)Cl 6H-315S c1cc(c(cc1N2C(=O)CS(=O)(=O)CC2=O)Cl)Cl 6H-316S c1cc(c(cc1Cl)Cl)CNC(=O)CS(=O)(=O)CC(=O)O 6H-317S c1cc(c(cc1F)F)N2C(=O)CSCC2=O 6H-321S c1ccc(cc1)CNC(=O)CSCC(=O)O 6H-322S COC(=O)c1ccc(s1)c2ccc(cc2)F 6H-324S Cc1c(nc(c(c1c2ccccc2)C#N)N)C 6H-326S CC(C)(C)c1cc(c(c(n1)N)C#N)c2c(cccc2Cl)Cl 6H-327S COc1ccc(cc1)c2cc(c(c(n2)N)C#N)c3ccc(cc3Cl)Cl 6H-328S c1cc(c(cc1F)F)NC(=O)CS(=O)CC(=O)O 6H-330S c1cc(c(cc1F)F)NC(=O)CS(=O)(=O)CC(=O)O 6H-331S COC(=O)c1ccc(s1)c2ccc(c(c2)Cl)Cl 6H-332S c1cc(ccc1c2ccc(s2)C(=O)O)F 6H-333S c1cc(c(cc1c2ccc(s2)C(=O)O)Cl)Cl 6H-335S CNC(=O)c1ccc(s1)c2ccc(cc2)F 6H-337S c1cc(c(cc1F)F)N2C(=O)CS(=O)CC2=O 6H-338S c1ccc(cc1)NC(=O)c2ccc(s2)c3ccc(cc3)F 6H-339S Cc1nc2cc(ccc2c(=O)n1c3nncs3)Cl 6H-341S c1cc(c(c(c1)Cl)c2cc(nc(c2C#N)N)c3ccc(cc3)Cl)Cl 6H-342S COc1ccc(cc1)c2cc(c(c(n2)N)C#N)c3cccc(c3)Cl 6H-343S COC(=O)c1ccc(s1)c2ccccc2 6H-344S CNC(=O)c1ccc(s1)c2ccc(c(c2)Cl)Cl 6H-345S c1ccc(cc1)NC(=O)c2ccc(s2)c3ccc(c(c3)Cl)Cl 6H-346S c1cc(c(cc1F)F)N2C(=O)CS(=O)(=O)CC2=O 6H-347S COc1ccc(cc1OC)CN2C(=O)CSCC2=O 6H-348S COc1ccc(cc1OC)CNC(=O)CS(=O)CC(=O)O 6H-350S COc1ccc(cc1OC)CNC(=O)CS(=O)(=O)CC(=O)O 6H-351S CC(C)Cc1cc(c(c(n1)N)C#N)c2ccc(cc2)Cl 6H-352S c1ccc(cc1)CNC(=O)CS(=O)(=O)CC(=O)O 6H-353S CC(C(=O)O)SCC(=O)O 6H-354S CC1C(=O)OC(=O)CS1 6H-355S CC(=O)Nc1cc(ccc1C(=O)Nc2[nH]c3ccccc3n2)Cl 6H-356S CC(C)Cc1cc(c(c(n1)N)C#N)c2ccccc2Cl 6H-357S c1cc(sc1)c2cc(c(c(n2)N)C#N)c3ccc(cc3)Cl 6H-358S CC1C(=O)N(C(=O)CS1)c2ccc(cc2)Cl 6H-359S CN(C)S(=O)(=O)Oc1ccsc1C(=O)OC 6H-363S CNC(=O)c1ccc(s1)c2ccccc2 6H-365S c1ccc(cc1)c2ccc(s2)C(=O)Nc3ccccc3 6H-366S Cc1c(nc(c(c1c2ccc(cc2)Cl)C#N)N)C 6H-367S Cc1nc2cc(ccc2c(=O)n1c3nc[nH]n3)Cl 6H-368S c1cc(ccc1c2cc(nc(c2C#N)N)c3ccc(c(c3)Cl)Cl)Cl 6H-369S CCc1c(c(c(c(n1)N)C#N)c2ccc(cc2)Cl)C 6H-370S Cc1c(c(c(nc1c2ccccc2)N)C#N)c3ccc(cc3)Cl 6H-371S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2)Cl 6H-374S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(c(c2)Cl)Cl 6H-375S CN(c1ccccc1)C(=O)c2ccc(s2)c3ccc(cc3)F 6H-376S Cc1nc2cc(ccc2c(=O)n1c3nccs3)Cl 6H-377S c1ccc(c(c1)c2cc(c(c(n2)N)C#N)c3ccc(cc3)Cl)Cl 6H-378S c1cc(ccc1c2cc(nc(c2C#N)N)c3ccc(cc3Cl)Cl)Cl 6H-379S c1ccc(cc1)c2cc(c(c(n2)N)C#N)c3ccc(cc3)Cl 6H-380S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2F)F 6H-382S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2)F 6H-383S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2cccc(c2)C(F)(F)F 6H-384S Cc1ccc(nc1)n2c(nc3cc(ccc3c2=O)Cl)C 6H-386S Cc1cc(nc(c1)n2c(nc3cc(ccc3c2=O)Cl)C)C 6H-387S CC(C)Cc1cc(c(c(n1)N)C#N)c2cccc(c2)Cl 6H-389S CCc1c(c(c(c(n1)N)C#N)c2cccc(c2)Cl)C 6H-390S COc1ccc(cc1OC)CN2C(=O)CS(=O)CC2=O 6H-391S COc1ccc(cc1OC)CN2C(=O)CS(=O)(=O)CC2=O 6H-392S c1ccc(cc1)c2cc(nc(c2C#N)N)c3ccc(cc3)Cl 6H-393S COc1ccc(cc1OC)c2cc(c(c(n2)N)C#N)c3ccccc3 6H-394S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccccc2C(F)(F)F 6H-395S c1cc(ccc1CNC(=O)CSCC(=O)O)F 6H-397S COc1ccc(cc1)c2cc(nc(c2C#N)N)c3ccc(c(c3)OC)OC 6H-399S CCc1c(c(c(c(n1)N)C#N)c2ccc(cc2)OC)C 6H-400S CCn1c(nnc1SCc2ccc(cc2)C)C(Cc3ccccc3)NS(=O)(=O)c4ccc(cc4)F 6H-401S CCOC(=O)CC1C(=O)NCCN1C(=O)c2cccc(c2)OC 6H-402S Cn1c(nnc1SCc2ccc(cc2)Br)C(Cc3ccccc3)NS(=O)(=O)c4ccc(cc4)Cl 6H-406S Cn1c(nnc1SCc2ccc(c(c2)Cl)Cl)C(Cc3ccccc3)NS(=O)(=O)c4ccc(cc4)Cl 6H-407S Cn1c(nnc1SCc2ccc(cc2)C(F)(F)F)C(Cc3ccccc3)NS(=O)(=O)c4ccc(cc4)Cl 6H-408S c1cc(cc(c1)NC(=O)c2ccc(cc2)c3cccs3)C(F)(F)F 6H-410S Cc1ccc(cc1)NC(=O)c2ccc(cc2)c3cccs3 6H-411S Cn1c(nnc1SCC(=O)OC)C(Cc2ccccc2)NS(=O)(=O)c3ccc(cc3)Cl 6H-414S Cn1c(nnc1SCC=C)C(Cc2ccccc2)NS(=O)(=O)c3ccc(cc3)Cl 6H-415S CC(=C)CSc1nnc(n1C)C(Cc2ccccc2)NS(=O)(=O)c3ccc(cc3)Cl 6H-416S c1ccc(cc1)/C(=N/O)/CSc2ccc(cc2)Cl 6H-417S COC(=O)c1ccc(cc1)c2cccs2 6H-419S Cc1nc2c(cc(cc2Cl)Cl)c(=O)n1c3nncs3 6H-422S c1ccc(cc1)NC(=O)c2ccc(cc2)c3cccs3 6H-423S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2)C(F)(F)F 6H-426S COc1ccc(cc1)c2ccc(s2)C(=O)OC 6H-428S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2)Br 6H-429S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2)[N+](=O)[O-] 6H-430S Cn1c(c(c(n1)C(F)(F)F)/N=N/c2ccc(cc2)Cl)O 6H-431S C=CCn1c(nnc1SCc2ccc(cc2)Cl)CNS(=O)(=O)c3ccc(cc3)Br 6H-432S CC(C)(C)c1ccc(cc1)CSc2nnc(n2CC=C)CNS(=O)(=O)c3ccc(cc3)Br 6H-433S C=CCn1c(nnc1SCc2ccc(cc2)C(F)(F)F)CNS(=O)(=O)c3ccc(cc3)Br 6H-434S CSc1nnc(n1CC=C)CNS(=O)(=O)c2ccc(cc2)Br 6H-435S C=CCn1c(nnc1SCCOc2ccccc2)CNS(=O)(=O)c3ccc(cc3)Br 6H-436S COc1cccc(c1)CSc2nnc(n2CC=C)CNS(=O)(=O)c3ccc(cc3)Br 6H-437S CCOC(=O)c1ccc(cc1)CSc2nnc(n2CC=C)CNS(=O)(=O)c3ccc(cc3)Br 6H-438S c1ccc(cc1)/C(=N/OCc2ccc(cc2)Cl)/CSc3ccc(cc3)Cl 6H-439S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2)OC(F)(F)F 6H-444S c1ccc(cc1)/C(=N/OCc2c(cccc2Cl)Cl)/CSc3ccc(cc3)Cl 6H-450S CCn1c(nnc1SCc2c(cccc2Cl)Cl)CNS(=O)(=O)c3ccc(cc3)Br 6H-453S CCn1c(nnc1SCc2ccc(cc2)C(F)(F)F)CNS(=O)(=O)c3ccc(cc3)Br 6H-454S CCn1c(nnc1SC)CNS(=O)(=O)c2ccc(cc2)Br 6H-455S CCn1c(nnc1SCCOc2ccccc2)CNS(=O)(=O)c3ccc(cc3)Br 6H-456S CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)CNS(=O)(=O)c3ccc(cc3)Br 6H-457S CCn1c(nnc1SCC(=C)C)CNS(=O)(=O)c2ccc(cc2)Br 6H-458S CCn1c(nnc1SCc2cccc(c2)OC)CNS(=O)(=O)c3ccc(cc3)Br 6H-459S CCn1c(nnc1SC(C)C(=O)OCC)CNS(=O)(=O)c2ccc(cc2)Br 6H-460S c1cc(sc1)c2ccc(cc2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 6H-461S CCn1c(nnc1SCc2cccc(c2)F)CNS(=O)(=O)c3ccc(cc3)Br 6H-463S COc1ccc(cc1)c2ccc(s2)C(=O)O 6H-465S c1ccc(cc1)/C(=N/OCc2ccc(cc2)Cl)/CS(=O)(=O)c3ccc(cc3)Cl 6H-467S c1ccc(cc1)/C(=N/OCc2c(cccc2Cl)Cl)/CS(=O)(=O)c3ccc(cc3)Cl 6H-468S c1cc(ccc1CNC(=O)CS(=O)CC(=O)O)F 6H-501S Cc1ccc2c(c1)c(=O)n(c(n2)C)c3ccc(cc3)F 6H-502S Cc1c(c(c(nc1c2ccc(cc2)Cl)N)C#N)c3ccc(cc3)OC 6H-503S Cc1ccc(cc1)c2cc(c(c(n2)N)C#N)c3ccc(cc3)Cl 6H-504S c1cc(ccc1CN2C(=O)CSCC2=O)F 6H-506S Cc1ccc(cc1)c2cc(c(c(n2)N)C#N)c3cccc(c3)Cl 6H-508S CC(C)Cc1cc(c(c(n1)N)C#N)c2cccc(c2Cl)Cl 6H-509S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(c(c2)F)F 6H-510S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccc(cc2)OC 6H-511S c1cc(ccc1c2cc(nc(c2C#N)N)c3ccc(cc3)F)F 6H-513S CCc1c(c(c(c(n1)N)C#N)c2ccc(cc2)F)C 6H-514S c1cc(ccc1C2CC(=O)C(=CNOCc3c(snn3)Cl)C(=O)C2)Cl 6H-900 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NOCc3c(snn3)Cl 6H-901 Cc1c(c(no1)C(=O)C)C(=O)Nc2nccs2 6H-902 Cc1c(c(no1)C(=O)/C=C/N(C)C)C(=O)Nc2nccs2 6H-904 Cc1ccc(cc1)n2c(ccn2)c3c(c(on3)C)C(=O)Nc4nccs4 6H-905 Cc1c(c(no1)C(=O)/C=C/Nc2ccc(cc2)OC)C(=O)Nc3nccs3 6H-906 Cc1c(c(no1)C(=O)/C=C/Nc2ccc(cc2)OC(F)(F)F)C(=O)Nc3nccs3 6H-909 C1CC(=O)C(C(=O)C1)/C=N/OCc2c(snn2)Cl 6H-911 c1cc(cc(c1)OCCn2c(cnc2S)CO)C(F)(F)F 6H-912 c1c(cnc(c1Cl)NCCn2c(cnc2S)CO)C(F)(F)F 6H-913 Cc1c(c(no1)/C(=N/O)/C)C(=O)Nc2nccs2 6H-914 CCOC(=O)/C=C(\N)/NNC(=O)c1cccnc1 6H-915 CC1CN(C(ON1C)c2ccccc2)C(=O)Nc3ccc(cc3)Cl 6H-917 CCOC(=O)c1cc(c(=O)n(c1N)NC(=O)c2cccnc2)C(=O)OCC 6H-918 CN1C(=O)C(=Cc2cccc(c2OCC=C)OC)C(=O)N(C1=O)C 6H-920 COc1cccc(c1OCc2ccccc2)C=O 6H-921 CN1C(=O)C(C(=O)N(C1=O)C)C(c2cccc(c2OCC=C)OC)C3C(=O)N(C(=O)N(C3=O)C)C 6H-922 CCOC(=O)CC(=N)NN(C)c1c(cc(cn1)C(F)(F)F)Cl 6H-923 C/[N+](=C/c1cccc(c1OCc2ccccc2)OC)/[O-] 6H-925 Cn1c(=O)c2c(n(c1=O)C)OCC3C2c4cccc(c4OC3)OC 6H-926 CCOC(=O)CC(=N)NNC(=O)c1ccc(cc1Cl)Cl 6H-930 CCOC(=O)c1cc(c(=O)n(c1N)NC(=O)c2ccc(cc2Cl)Cl)C(=O)OCC 6H-932 CCOC(=O)/C=C(\NC(=O)Nc1ccccc1)/NN(C)c2c(cc(cn2)C(F)(F)F)Cl 6H-933 c1cc(ccc1N2CCN(CC2)C(=N)CC#N)Cl 6H-934 c1cc(cc(c1)Cl)N2CCN(CC2)C(=N)CC#N 6H-935 c1cc(nc(c1)Cl)N2CCN(CC2)C(=N)CC#N 6H-936 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=S)NC(=O)c2ccccc2 6H-937 c1cc(cc(c1)Cl)N2CCN(CC2)/C(=C(\C=C(C#N)C#N)/C#N)/N 6H-938 c1cc(ccc1N2CCN(CC2)/C(=C(\C=C(C#N)C#N)/C#N)/N)Cl 6H-939 CN(C)/C=N/c1c(cc(c(n1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C#N)C#N 6H-940 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=S)N 6H-941 c1cc(nc(c1)Cl)N2CCN(CC2)/C(=C(\C=C(C#N)C#N)/C#N)/N 6H-942 c1cc(ccc1CON/C=N/c2c(cc(c(n2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C#N)C#N)Cl 6H-943 CCOC(=O)c1cc(c(=O)n(c1N)N(C)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)OCC 6H-944 Cn1c(cnc1SCc2ccc(cc2)F)CS(=O)(=O)c3ccccc3 6H-945 CC(=O)C1=NOC2C1C(=O)N(C2=O)c3ccccc3 6H-948 CN1CCN(CC1)/C(=C/C#N)/N 6H-949 c1ccn(c1)c2c(cc(c(n2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C#N)C#N 6H-950 CN1CCN(CC1)/C(=C(\C=C(C#N)C#N)/C#N)/N 6H-951 CN1CCN(CC1)c2c(cc(c(n2)N)C#N)C#N 6H-952 CCOC(=O)c1cc(c(nc1n2c(cc(n2)C)C)OCc3ccc(cc3)C)C(=O)OCC 6H-953 c1ccc(cc1)S(=O)(=O)Cc2c(snn2)Cl 6H-954 c1cc(cc(c1)N2C(=O)C3CC(CN3C2=O)Cl)C(F)(F)F 6H-955 c1cc(c(cc1N2CCN(CC2)/C(=C\C#N)/N)Cl)Cl 6H-956 CC1(OCCO1)c2ccc(cc2)[N+](=O)[O-] 6H-958 CC1(OCCO1)c2ccc3c(c2)c(on3)c4ccccc4 6H-959 c1cc(c(cc1N2CCN(CC2)/C(=C(/C=C(C#N)C#N)\C#N)/N)Cl)Cl 6H-960 CN(C)/C=C/C(=O)/C=C/c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 6H-961 CC(=O)c1ccc2c(c1)c(on2)c3ccccc3 6H-962 CCOC(=O)c1cnc2ccc(cc2c1Cl)Br 6J-001 CCOC(=O)C(=CNc1ccccc1C(F)(F)F)C(=O)OCC 6J-002 CCOC(=O)c1cnc2ccc(cc2c1O)C(F)(F)F 6J-003 CCOC(=O)c1cnc2ccc(cc2c1Cl)C(F)(F)F 6J-004 CCOC(=O)C(=CNc1ccc(cc1Cl)Cl)C(=O)OCC 6J-005 CCOC(=O)c1cnc2c(c1O)cc(cc2Cl)Cl 6J-006 CCOC(=O)c1cnc2c(c1Cl)cc(cc2Cl)Cl 6J-007 CCOC(=O)C(=CNc1ccccc1Br)C(=O)OCC 6J-008 CCOC(=O)C(=CNc1cc(ccc1Cl)Cl)C(=O)OCC 6J-009 CCOC(=O)C(=CNc1cccc(c1C)Cl)C(=O)OCC 6J-010 CCOC(=O)c1cnc2c(c(ccc2c1O)Cl)C 6J-011 CCOC(=O)c1cnc2c(c(ccc2c1Cl)Cl)C 6J-012 c1cc(ccc1/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)Cl 6J-013 CC(=O)c1ccc(s1)/C(=C/c2ccc(cc2)Cl)/C#N 6J-014 CCOC(=O)c1cnc2c(ccc(c2c1O)Cl)Cl 6J-015 CCOC(=O)c1cnc2c(c1O)cccc2Br 6J-016 CCOC(=O)C(=CNc1ccccc1OC)C(=O)OCC 6J-017 CCOC(=O)c1cnc2c(c1O)cccc2OC 6J-018 CCOC(=O)C(=CNc1cc(ccc1F)F)C(=O)OCC 6J-019 CCOC(=O)c1c[nH]c2c(ccc(c2c1=O)F)F 6J-020 CCOC(=O)C(=CNc1ccccc1C)C(=O)OCC 6J-022 CCOC(=O)C(=CNc1ccc(cc1C)C)C(=O)OCC 6J-023 CCOC(=O)c1cnc2c(c1Cl)cccc2Br 6J-024 CCOC(=O)c1cnc2c(ccc(c2c1Cl)Cl)Cl 6J-025 CCOC(=O)c1cnc2c(c1O)cccc2C(F)(F)F 6J-026 CCOC(=O)c1cnc2c(c1Cl)cccc2C(F)(F)F 6J-027 CCOC(=O)c1cnc2c(cc(cc2c1O)C)C 6J-028 CCOC(=O)c1cnc2c(cccc2c1O)C 6J-029 CCOC(=O)C(=CNc1ccc(cc1Cl)C)C(=O)OCC 6J-030 CCOC(=O)c1cnc2c(c1O)cc(cc2Cl)C 6J-031 CCOC(=O)c1cnc2c(c1Cl)cc(cc2Cl)C 6J-032 CCOC(=O)c1cnc2c(cc(cc2c1Cl)C)C 6J-033 CCOC(=O)c1cnc2c(c1Cl)cccc2OC 6J-034 CN(C)/C=C/C(=O)c1ccc(s1)/C(=C/c2ccc(cc2)Cl)/C#N 6J-035 CCOC(=O)C(=CNc1ccc(cc1F)Cl)C(=O)OCC 6J-036 CCOC(=O)c1cnc2c(c1O)cc(cc2F)Cl 6J-037 CCOC(=O)c1cnc2c(c1Cl)cc(cc2F)Cl 6J-038 CCOC(=O)c1cnc2c(cccc2c1Cl)C 6J-039 c1cc(ccc1/C(=N/Nc2c(cc(cn2)C(F)(F)F)Cl)/Cl)Cl 6J-040 c1cc(ccc1c2nnc3n2cc(cc3Cl)C(F)(F)F)Cl 6J-041 CCOC(=O)C(=CNc1ccc2c(c1)OCO2)C(=O)OCC 6J-043 CCOC(=O)c1cnc2cc3c(cc2c1O)OCO3 6J-044 CCOC(=O)C(=CNc1ccc(cc1Cl)F)C(=O)OCC 6J-045 CCOC(=O)c1cnc2c(c1O)cc(cc2Cl)F 6J-046 CCOC(=O)c1cnc2c(c1Cl)cc(cc2Cl)F 6J-047 CCOC(=O)C(=CNc1ccccc1)C(=O)OCC 6J-048 CCOC(=O)c1cnc2cc3c(cc2c1Cl)OCO3 6J-049 CCOC(=O)c1c[nH]c2ccccc2c1=O 6J-050 CCOC(=O)c1cnc2ccccc2c1Cl 6J-051 CCOC(=O)C(=CNc1ccccc1C#N)C(=O)OCC 6J-052 CCOC(=O)c1cnc2cc(cc(c2c1O)Cl)Cl 6J-053 CCOC(=O)c1cnc2cc(cc(c2c1Cl)Cl)Cl 6J-054 CCOC(=O)c1cnc2c(cccc2c1O)C#N 6J-055 CCOC(=O)C(=CNc1cc(cc(c1)Cl)Cl)C(=O)OCC 6J-056 CCOC(=O)C(=CNc1cc(cc(c1)F)F)C(=O)OCC 6J-057 COC(=O)c1cc(cc(c1)N)N 6J-060 c1cc(sc1)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 6J-062 CCOC(=O)c1cnc2c(cccc2c1Cl)C#N 6J-063 c1c(cnc(c1Cl)N/N=C/C(=O)O)C(F)(F)F 6J-064 c1cc(ccc1/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 6J-065 c1cc(ccc1c2nnc3n2cc(cc3Cl)C(F)(F)F)[N+](=O)[O-] 6J-066 c1cc(c(cc1Cl)Cl)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 6J-067 CCOC(=O)c1cnc2cc(cc(c2c1O)F)F 6J-068 CCOC(=O)c1cnc2cc(cc(c2c1Cl)F)F 6J-069 CCOC(=O)c1cnc2ccc(cc2c1O)OC 6J-070 CCOC(=O)c1cnc2ccc(cc2c1Cl)OC 6J-071 CC(=O)c1ccc(s1)/C(=C/c2ccc(cc2Cl)Cl)/C#N 6J-072 CC(=O)c1ccc(s1)/C(=C/c2cccs2)/C#N 6J-073 c1cc(c(cc1Cl)Cl)c2nnc3n2cc(cc3Cl)C(F)(F)F 6J-074 c1cnccc1/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 6J-075 CCOc1ccccc1N/C(=C\[N+](=O)[O-])/SC 6J-076 c1ccc(c(c1)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)C(=O)O 6J-077 c1cnccc1c2nnc3n2cc(cc3Cl)C(F)(F)F 6J-078 c1ccc(c(c1)c2nnc3n2cc(cc3Cl)C(F)(F)F)C(=O)O 6J-079 c1ccc(cc1)/C=C/c2nnc3n2cc(cc3Cl)C(F)(F)F 6J-081 c1ccc(cc1)/C=C/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 6J-082 Cn1cc(cc1/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)C(=O)c3ccc(cc3Cl)Cl 6J-083 C=CCn1cc(cc(c1=O)C#N)c2ccccc2 6J-301S c1ccc(cc1)c2cc(c(nc2)Sc3ccccc3)C#N 6J-302S COc1ccc(cc1)Sc2c(cc(cn2)c3ccccc3)C#N 6J-303S Cc1cc(ccc1Oc2c(cc(cn2)c3ccccc3)C#N)Cl 6J-304S c1ccc(cc1)c2cc(c(nc2)Oc3ccc(cc3)F)C#N 6J-305S Cn1cc(cc(c1=O)C#N)c2cccc(c2)Cl 6J-306S c1ccc(cc1)c2cc(c(nc2)Oc3ccc(c(c3)Cl)Cl)C#N 6J-307S c1cc(cc(c1)Cl)c2cc(c(nc2)Cl)C#N 6J-308S CCCCCCCCn1cnc2c1cc(c(c2NS(=O)(=O)c3ccc(cc3)C(C)(C)C)C)C 6J-310S Cc1cccc(c1)Cn2c(nc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)OC)C)C)C 6J-311S COc1ccccc1Oc2c(cc(cn2)c3cccc(c3)Cl)C#N 6J-312S c1cc(cc(c1)Cl)c2cc(c(nc2)Oc3cccc(c3)C(F)(F)F)C#N 6J-313S Cc1cccc(c1)Cn2c(nc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)Cl)C)C)C 6J-314S Cc1cccc(c1)Cn2c(nc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)F)C)C)C 6J-315S CN(C)c1ncc(c(n1)Oc2ccc(c(c2)Cl)Cl)OC 6J-319S CN(C)c1ncc(c(n1)Oc2ccc(cc2)[N+](=O)[O-])OC 6J-320S Cc1cccc(c1)Cn2c(nc3c2cc(c(c3NS(=O)(=O)c4ccc(cc4)C(C)(C)C)C)C)C 6J-323S Cc1cccc(c1)Cn2c(nc3c2cc(c(c3NS(=O)(=O)C)C)C)C 6J-324S CN(C)c1ncc(c(n1)Oc2ccc(cc2)C(=O)OC)OC 6J-325S COc1ccc(cc1OC)c2cc(c(=O)[nH]c2)S(=O)(=O)c3ccccc3 6J-326S CN(C)c1ncc(c(n1)Oc2ccc(c3c2cccc3)Cl)OC 6J-327S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)F)nc(n2Cc4ccc(cc4)OC)C 6J-328S Cc1cc2c(c(c1C)NS(=O)(=O)c3cccc(c3)C(F)(F)F)nc(n2Cc4ccc(cc4)OC)C 6J-330S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)nc(n2Cc4ccc(cc4)OC)C 6J-331S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)Cl)ncn2Cc4cccc(c4)OC 6J-334S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccccc3Cl)ncn2Cc4cccc(c4)OC 6J-335S Cc1ccc(cc1)S(=O)(=O)c2c(cc([nH]c2=O)C)C 6J-336S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccccc2Cl)C 6J-337S Cc1cc([nH]c(=O)c1S(=O)(=O)c2cccc(c2)Cl)C 6J-338S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)ncn2Cc4cccc(c4)OC 6J-346S Cc1cc2c(c(c1C)NS(=O)(=O)C)ncn2Cc3cccc(c3)OC 6J-347S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(c(c3Cl)Cl)Cl)ncn2Cc4cccc(c4)OC 6J-348S Cc1cc2c(c(c1C)NS(=O)(=O)c3cc(cc(c3)Cl)Cl)ncn2Cc4cccc(c4)OC 6J-349S Cc1cc2c(c(c1C)NS(=O)(=O)c3ccc(cc3)C(C)(C)C)ncn2Cc4cccc(c4)OC 6J-350S Cc1ccccc1S(=O)(=O)c2c(cc([nH]c2=O)c3ccccc3)C 6J-355S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccccc2OC)C 6J-356S Cc1ccc(cc1)S(=O)(=O)Nc2c(c(cc3c2ncn3Cc4cccc(c4)OC)C)C 6J-357S CCCCCCCCn1cnc2c1cc(c(c2NS(=O)(=O)c3cc(cc(c3)Cl)Cl)C)C 6J-358S c1cc(cc(c1)C(F)(F)F)c2cc(c(=O)[nH]c2)C#N 6J-508S c1cc(cc(c1)C(F)(F)F)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)C#N 6J-512S COc1ccc(cc1)Cn2cc(cc(c2=O)C#N)c3cccc(c3)C(F)(F)F 6J-513S c1cc(cc(c1)C(F)(F)F)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)C#N 6J-514S c1cc(cc(c1)C(F)(F)F)c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)C#N 6J-515S Cn1cc(cc(c1=O)C#N)c2cccc(c2)C(F)(F)F 6J-516S C=CCn1cc(cc(c1=O)C#N)c2cccc(c2)C(F)(F)F 6J-518S Cc1ccc(cc1)Cn2cc(cc(c2=O)C#N)c3cccc(c3)C(F)(F)F 6J-519S c1cc(cc(c1)C(F)(F)F)c2cc(c(=O)n(c2)Cc3ccc(cc3)F)C#N 6J-520S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)C#N)c3cccc(c3)C(F)(F)F 6J-521S c1cc(c(nc1)Sc2ccc(cc2)Cl)c3nc4cc(ccc4o3)Cl 6J-530S c1ccc(c(c1)CSc2c(cccn2)c3nc4cc(ccc4o3)Cl)Cl 6J-532S COC(=O)c1ccc(cc1)Cn2c(cccc2=O)c3ccc(cc3)Cl 6J-535S c1ccc(cc1)Cn2c3ccccc3nc2NS(=O)(=O)c4cccc(c4Cl)Cl 6J-538S c1ccc(cc1)Cn2c3ccccc3nc2NS(=O)(=O)c4cc(ccc4Cl)Cl 6J-540S c1ccc(cc1)Cn2c3ccccc3nc2NS(=O)(=O)c4ccccc4[N+](=O)[O-] 6J-542S c1ccc(cc1)c2cc(c(nc2)Oc3ccc(cc3)Cl)C#N 6J-545S c1ccc(cc1)c2cc(c(nc2)Sc3ccc(cc3)Cl)C#N 6J-547S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Cl)C#N 6J-549S c1ccc(cc1)Cn2cc(cc(c2=O)C#N)c3cccc(c3)C(F)(F)F 6J-550S CC(C)Cn1cc(cc(c1=O)C#N)c2cccc(c2)C(F)(F)F 6J-551S c1ccc(cc1)Oc2c(cc(cn2)c3cccc(c3)C(F)(F)F)C#N 6J-552S c1ccc(c(c1)Oc2c(cc(cn2)c3cccc(c3)C(F)(F)F)C#N)Cl 6J-553S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Oc3ccc(cc3)Cl)C#N 6J-555S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Oc3ccc(cc3)F)C#N 6J-556S COc1ccc(cc1)Oc2c(cc(cn2)c3cccc(c3)C(F)(F)F)C#N 6J-557S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Oc3c(cccc3Cl)Cl)C#N 6J-558S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Oc3ccc(cc3F)F)C#N 6J-559S c1cc(c(nc1)Oc2ccc(c(c2)Cl)Cl)c3nc4cc(ccc4o3)Cl 6J-561S c1cc(c(nc1)Oc2cc(cc(c2)Cl)Cl)c3nc4cc(ccc4o3)Cl 6J-562S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Oc3cccc(c3)C(F)(F)F)C#N 6J-566S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Oc3ccc(c(c3)Cl)Cl)C#N 6J-567S c1ccc(cc1)Sc2c(cc(cn2)c3cccc(c3)C(F)(F)F)C#N 6J-568S c1ccc(c(c1)Sc2c(cc(cn2)c3cccc(c3)C(F)(F)F)C#N)Cl 6J-569S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Sc3cccc(c3)Cl)C#N 6J-570S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Sc3ccc(cc3)Cl)C#N 6J-571S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Sc3ccc(cc3)F)C#N 6J-572S COc1ccccc1Sc2c(cc(cn2)c3cccc(c3)C(F)(F)F)C#N 6J-573S c1ccc(cc1)C(CC(=O)c2ccc(cc2)Br)C#N 6J-574S c1ccc(cc1)C(=O)CC(C#N)c2cccc(c2Cl)Cl 6J-575S c1ccc(cc1)C(=O)CC(c2cccc(c2Cl)Cl)C(=O)O 6J-577S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Sc3c(cccc3Cl)Cl)C#N 6J-578S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Sc3ccc(c(c3)Cl)Cl)C#N 6J-579S c1cc(cc(c1)C(F)(F)F)c2cc(c(nc2)Sc3cccc(c3)C(F)(F)F)C#N 6J-581S Cc1ccc(cc1)c2cc(c(=O)n(c2)Cc3ccccc3)C#N 6J-583S Cc1ccc(cc1)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)C#N 6J-584S Cc1ccc(cc1)c2cc(c(=O)n(c2)Cc3ccc(cc3)F)C#N 6J-585S COC(=O)C(CC(=O)c1ccc(cc1)Br)c2ccccc2 6J-586S Cc1ccc(cc1)c2cc(c(=O)n(c2)Cc3cccc(c3)OC)C#N 6J-587S Cc1ccc(cc1)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)C#N 6J-588S Cc1ccc(cc1)c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)C#N 6J-589S Cc1ccc(cc1)c2cc(c(=O)n(c2)Cc3cccc(c3)C(F)(F)F)C#N 6J-590S c1cc(ccc1c2cc(c(nc2)OC(=O)c3ccc(cc3)Cl)C#N)Cl 6J-591S c1cc(c(nc1)Oc2ccc(cc2Cl)Cl)c3nc4cc(ccc4o3)Cl 6J-653S Cc1c(c(nc(n1)N)SCc2cccc(c2)C(F)(F)F)C#N 6J-855S CC(=O)O/C(=C(\C=N\OC)/C(=O)Nc1ccc(cc1Cl)Cl)/Nc2ccc(cc2Cl)Cl 6J-900 CN(c1c(cc(cn1)C(F)(F)F)Cl)Nc2cc(n(c(=O)n2)c3ccc(cc3Cl)Cl)O 6J-901 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)C=C 6J-903 CCOC(=O)C1=C(N(C(=O)CC1)N(C)c2c(cc(cn2)C(F)(F)F)Cl)C 6J-904 CN(c1c(cc(cn1)C(F)(F)F)Cl)Nc2cc(n(c(=O)n2)c3cccc(c3)C(F)(F)F)N 6J-906 CC(=O)C1=NOC(C1)C(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl 6J-907 c1cc(nnc1N2CCC(CC2)C(=O)NCC3CC4CCCCN4O3)Cl 6J-909 CC(C)(CO)NC(=O)c1ccccc1OC 6J-910 CC1(COC(=N1)c2ccccc2OC)C 6J-911 c1cc(cnc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)NN 6K-001 CNC(=S)NNC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3cccnc3 6K-002 COc1ccc(cc1)C=C(C#N)C#N 6K-003 COc1ccc(cc1)CC(C#N)C#N 6K-004 COc1ccc(cc1)Cc2c(nc(nc2N)N)N 6K-005 COc1ccc(cc1)Cc2c(nc(nc2N)c3ccccc3)N 6K-006 Cc1nc(c(c(n1)N)Cc2ccc(cc2)OC)N 6K-007 COc1ccc(cc1)Cc2c(nc(nc2N)c3ccccn3)N 6K-008 c1cc(c(cc1Cl)Cl)C=C(C#N)C#N 6K-009 c1cc(c(cc1Cl)Cl)CC(C#N)C#N 6K-010 c1ccnc(c1)c2nc(c(c(n2)N)Cc3ccc(cc3Cl)Cl)N 6K-011 c1cc(c(cc1Cl)Cl)Cc2c(nc(nc2N)N)N 6K-012 c1cc(c(cc1Cl)Cl)Cc2c(nc(nc2N)Cn3cncn3)N 6K-013 Cc1nc(c(c(n1)N)Cc2ccc(cc2Cl)Cl)N 6K-014 c1ccc(cc1)c2nc(c(c(n2)N)Cc3ccc(cc3Cl)Cl)N 6K-015 c1cc(c(c(c1)Cl)C=C(C#N)C#N)F 6K-016 c1ccnc(c1)c2nc(c(c(n2)N)Cc3c(cccc3Cl)F)N 6K-017 c1cc(c(c(c1)Cl)CC(C#N)C#N)F 6K-018 c1ccc(c(c1)C=C(C#N)C#N)F 6K-019 c1ccc(c(c1)CC(C#N)C#N)F 6K-020 c1ccc(c(c1)Cc2c(nc(nc2N)N)N)F 6K-021 Cn1c(nnc1S)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccnc4 6K-022 Cc1c(c(=O)ccn1Cc2ccccc2)OCc3c(cccc3Cl)Cl 6K-023 Cn1c(nnc1SC)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccnc4 6K-024 c1cc(oc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)NN 6K-027 c1ccc(cc1)c2nc(c(c(n2)N)Cc3ccccc3F)N 6K-028 c1ccc(c(c1)Cc2c(nc(nc2N)c3ccccn3)N)F 6K-029 Cc1nc(c(c(n1)N)Cc2ccccc2F)N 6K-030 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=S)N 6K-031 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=S)/N=C/N(C)C 6K-032 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3ncc(s3)C(=O)c4ccc(cc4)Cl 6K-033 c1ccc(cc1)C(=O)c2ccc(cc2)C(C#N)c3ccc(cc3)Cl 6K-034 CNC(=S)NNC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3ccco3 6K-035 Cn1c(nnc1S)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4ccco4 6K-036 Cc1nnc(n1N)n2c(ccn2)/C=C/c3ccc(cc3)Cl 6K-039 CCOC(=O)CNC(=O)c1c(onc1c2ccccc2Cl)C 6K-040 c1ccc(c(c1)Cc2c(nc(nc2N)Cn3cncn3)N)F 6K-042 COc1ccc(cc1)Cc2c(nc(nc2N)Cn3cncn3)N 6K-043 c1ccc(cc1)C(=O)c2ccc(cc2)C(c3ccc(cc3)Cl)C(=O)N 6K-044 c1ccc(cc1)C(c2ccc(cc2)C(C#N)c3ccc(cc3)Cl)O 6K-045 Cc1ccc(cc1C)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)c3ccccc3 6K-046 COc1ccc(c(c1)OC)N/N=C(/C=N/OC)\C(=O)c2ccc(cc2)c3ccccc3 6K-047 COc1ccc(c(c1)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)c3ccccc3)OC 6K-048 CCOc1cnc(o1)c2c(onc2c3ccccc3Cl)C 6K-049 c1cc(ccc1C=C(C#N)C#N)[N+](=O)[O-] 6K-051 c1cc(c(cc1Cl)Cl)CC(C#N)(C#N)c2c(cc(cn2)C(F)(F)F)Cl 6K-052 Cc1nnc(n1N)n2c(ccn2)c3cccc(c3)Oc4c(cc(cn4)C(F)(F)F)Cl 6K-056 COc1ccc(cc1)N/N=C(/C=N/OC)\C(=O)c2ccc(cc2)c3ccccc3 6K-057 Cc1c(c(=O)ccn1Cc2c(cccc2Cl)F)OCc3c(cccc3Cl)Cl 6K-058 c1ccnc(c1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)NN 6K-059 Cc1c(c(=O)cc[nH]1)OCc2ccccc2 6K-060 c1ccn(c1)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 6K-061 Cc1ccc(cc1)N/N=C(/C=N/OC)\C(=O)c2ccc(cc2)c3ccccc3 6K-062 CNC(=S)NNC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3ccccn3 6K-063 c1(nnc(n1N)NN)C(F)(F)F.Cl 6K-064 Cn1c(nnc1S)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4ccccn4 6K-065 c1cc(ccc1CC(C#N)C#N)[N+](=O)[O-] 6K-067 Cn1c(nnc1SC)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4ccccn4 6K-069 CN(C)/C=N/C(=O)C(c1ccc(cc1)C(=O)c2ccccc2)c3ccc(cc3)Cl 6K-072 CO/N=C/C(=N\Nc1ccc(cc1)[N+](=O)[O-])/C(=O)c2ccc(cc2)c3ccccc3 6K-073 Cc1c(c(=O)ccn1Cc2ccc(cc2)F)OCc3c(cccc3Cl)Cl 6K-074 Cc1c(c(=O)ccn1c2c(cc(cn2)C(F)(F)F)Cl)OCc3c(cccc3Cl)Cl 6K-075 c1cc(ccc1CC(C#N)(C#N)c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 6K-076 Cc1c(c(=O)ccn1Cc2ccc(cc2)Cl)OCc3c(cccc3Cl)Cl 6K-077 COC(=O)CNC(=O)c1cc(ccc1Cl)Cl 6K-078 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)NNC(=S)N 6K-079 c1cc(c(c(c1)F)C#N)C(C#N)c2ccc(cc2Cl)Cl 6K-080 Cc1c(c(=O)ccn1Cc2ccc(c(c2)Cl)Cl)OCc3c(cccc3Cl)Cl 6K-081 c1cc(ccc1CCc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 6K-082 Cc1c(c(=O)ccn1Cc2c(cccc2Cl)F)OCc3ccccc3 6K-083 c1ccc(cc1)C(=O)c2ccc(cc2)C(c3ccc(cc3)Cl)C(=O)N/C=N/O 6K-084 Cc1c(c(=O)ccn1c2c(cc(cn2)C(F)(F)F)Cl)OCc3ccccc3 6K-085 Cc1c(c(=O)cc[nH]1)OCc2ccc(cc2)F 6K-086 Cc1ccc(cc1)Cn2ccc(=O)c(c2C)OCc3ccccc3 6K-087 Cc1c(c(=O)ccn1Cc2ccc(cc2)OC)OCc3c(cccc3Cl)Cl 6K-088 c1ccc(cc1)C(=O)c2ccc(cc2)C(C#N)c3ccc(cc3Cl)Cl 6K-089 Cc1c(c(=O)ccn1Cc2ccc(cc2)Cl)OCc3ccccc3 6K-090 Cc1c(c(=O)ccn1Cc2ccc(cc2)F)OCc3ccccc3 6K-091 Cc1c(c(=O)cc[nH]1)O 6K-092 c1ccc(cc1)C(=O)c2ccc(cc2)C(c3ccc(cc3Cl)Cl)C(=O)N 6K-093 Cc1c(c(=O)ccn1c2c(cc(cn2)C(F)(F)F)Cl)OCc3ccc(cc3)F 6K-094 Cc1c(c(=O)ccn1Cc2ccccc2)OCc3ccccc3 6K-096 Cc1c(c(=O)ccn1Cc2ccc(c(c2)Cl)Cl)OCc3ccccc3 6K-099 c1cc(c(cc1Cl)Cl)CCc2c(cc(cn2)C(F)(F)F)Cl 6K-100 Cc1c(c(=O)ccn1Cc2ccc(c(c2)Cl)Cl)OCc3ccc(cc3)F 6K-102 CN(C)/C=N/C(=O)C(c1ccc(cc1)C(=O)c2ccccc2)c3ccc(cc3Cl)Cl 6K-103 c1ccc(cc1)C2N(C(=O)CS2)c3nc(cs3)c4ccc(cc4Cl)Cl 6K-303S Cc1ccc(cc1Sc2c(c(nn2C)c3ccccc3)COC(=O)c4ccc(c(c4)Cl)Cl)F 6K-306S Cc1ccc(cc1S(=O)(=O)c2c(c(nn2C)c3ccccc3)COC(=O)c4ccc(c(c4)Cl)Cl)F 6K-307S Cc1ccc(cc1Sc2c(c(nn2C)c3ccccc3)COC(=O)c4ccc(cc4Cl)Cl)F 6K-308S c1cc(oc1)/C=N/c2nc(cs2)c3ccc(cc3Cl)Cl 6K-309S Cn1c(c(c(n1)C(F)(F)F)C=O)Oc2ccc(cc2Cl)Cl 6K-310S Cn1c(c(c(n1)C(F)(F)F)CO)Oc2ccc(cc2Cl)Cl 6K-311S Cn1c(c(c(n1)C(F)(F)F)CCl)Oc2ccc(cc2Cl)Cl 6K-312S Cn1c(c(c(n1)C(F)(F)F)CS(=O)(=O)c2ccc(cc2)Cl)Oc3cccc(c3)C(F)(F)F 6K-318S Cn1c(c(c(n1)C(F)(F)F)CSc2c(cccc2Cl)Cl)Oc3cccc(c3)C(F)(F)F 6K-319S Cn1c(c(c(n1)C(F)(F)F)COc2cc(c(cc2Cl)Cl)Cl)Oc3cccc(c3)C(F)(F)F 6K-320S Cn1c(c(c(n1)C(F)(F)F)CSc2ccc(cc2)Br)Oc3ccc(cc3Cl)Cl 6K-321S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3Cl)Cl)Sc4ccccc4Cl 6K-324S Cn1c(c(c(n1)c2ccccc2)COC(=O)c3ccc(cc3Cl)Cl)S(=O)(=O)c4ccccc4Cl 6K-325S Cn1c(c(c(n1)c2ccccc2)CO)SCc3ccc(cc3)Cl 6K-326S CC1C(=O)N(C(S1)c2ccc(cc2Cl)Cl)c3nc(cs3)c4ccc(cc4Cl)Cl 6K-329S Cn1c(c(c(n1)c2ccccc2)CCl)SCc3ccc(cc3)Cl 6K-330S Cn1c(c(c(n1)c2ccccc2)CCl)Sc3ccc(cc3)Br 6K-331S Cn1c(c(c(n1)C(F)(F)F)CS(=O)(=O)Cc2ccccc2Cl)Oc3ccc(cc3Cl)Cl 6K-332S Cn1c(c(c(n1)C(F)(F)F)COc2c(cc(cc2Cl)Cl)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl 6K-333S Cn1c(c(c(n1)C(F)(F)F)COc2ccc(cc2)C#N)Oc3cccc(c3)C(F)(F)F 6K-334S Cn1c(c(c(n1)C(F)(F)F)COc2cc(c(cc2Cl)Cl)Cl)Oc3ccc(cc3Cl)Cl 6K-335S Cn1c(c(c(n1)C(F)(F)F)CS(=O)(=O)c2cccc(c2)C(F)(F)F)Oc3ccc(cc3Cl)Cl 6K-336S COc1ccc(cn1)NC(=O)C(=C(Cl)Cl)Cl 6K-342S COc1ccc(cn1)NC(=O)/C(=C(\SCc2ccccc2)/Cl)/Cl 6K-344S Cn1c(c(c(n1)C(F)(F)F)CSCc2ccccc2Cl)Oc3ccc(cc3Cl)Cl 6K-346S Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccccc2C(C)C)C 6K-347S Cn1c(c(c(n1)c2ccccc2)CS(=O)(=O)c3ccc(cc3)Br)S(=O)(=O)c4ccc(cc4)Br 6K-350S Cc1cc(nc(c1S(=O)(=O)c2ccccc2C(C)C)OCC(C)C)C 6K-354S Cn1c(c(c(n1)c2ccccc2)CSc3ccc(cc3Cl)Cl)SCc4ccc(cc4)Cl 6K-355S Cn1c(c(c(n1)c2ccccc2)CSc3cccc(c3)C(F)(F)F)Sc4ccc(cc4)Br 6K-356S Cn1c(c(c(n1)c2ccccc2)CSc3ccc(cc3)Cl)Sc4ccc(cc4)Br 6K-357S Cc1cc(ccc1n2c(nc3ccccc3c2=O)CSc4ccccc4OC)Cl 6K-502S Cc1cc(ccc1n2c(nc3ccccc3c2=O)CSCc4ccccc4Cl)Cl 6K-503S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CCl 6K-505S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4ccc(cc4)Cl 6K-508S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4c(cccc4Cl)Cl 6K-510S CC(C)c1ccccc1n2c(nc3cc(ccc3c2=O)Cl)CS(=O)(=O)c4ccc(cc4)Cl 6K-512S c1ccc(cc1)n2c(nc3ccccc3c2=O)CS(=O)(=O)c4ccc(cc4Cl)Cl 6K-513S COC(=O)c1ccccc1SCC(=O)Nc2nc(cs2)c3ccccc3Cl 6K-517S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4ccc(cc4)Br 6K-518S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4cc(ccc4Cl)Cl 6K-519S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4cccc(c4)Cl 6K-520S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4cc(cc(c4)C)C 6K-521S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4cccc(c4)C(F)(F)F 6K-522S Cc1ccccc1n2c(nc3ccc(cc3c2=O)Cl)CSc4ccc(cc4)OC 6K-523S Cn1c(c(c(n1)c2ccccc2)C(c3ccccc3C(F)(F)F)O)Cl 6K-526S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3ccccc3 6K-527S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3ccccc3Cl 6K-528S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3cccc(c3)Cl 6K-529S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3ccc(cc3)Cl 6K-530S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3cccc(c3)C(F)(F)F 6K-531S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3ccc(cc3)OC 6K-532S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3ccccc3C(=O)OC 6K-535S Cc1c(n(c(n1)SCc2ccc(cc2)Cl)C)C 6K-537S c1ccc(c(c1)c2csc(n2)NC(=O)CS(=O)c3ccc(cc3)Br)Cl 6K-541S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Sc3ccc(cc3)Br 6K-542S Cc1ccc(cc1)S(=O)(=O)CC(=O)Nc2nc(cs2)c3ccccc3 6K-543S c1cc(c(c(c1)Cl)Cl)S(=O)(=O)CC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 6K-544S c1ccc(cc1)c2csc(n2)NC(=O)CS(=O)(=O)c3ccc(cc3)Cl 6K-545S Cn1c(=O)c2ccccc2nn1 6K-546S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Oc3ccccc3 6K-548S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Oc3ccccc3Cl 6K-549S CCOC(=O)c1c(nc(nn1)c2cccs2)Sc3ccccc3 6K-551S CCOC(=O)c1c(nc(nn1)c2cccs2)Sc3cccc(c3)C(F)(F)F 6K-554S Cc1ccc(c(c1)S(=O)CC(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl)C 6K-557S Cc1cccc(c1)S(=O)(=O)CC(=O)Nc2nc(cs2)c3ccccc3 6K-558S CCCn1c(c(nc1SCc2ccc(c(c2)Cl)Cl)C)C 6K-563S Cc1c(n(c(n1)SCc2ccc(c(c2)Cl)Cl)CC#C)C 6K-564S CCCc1c(n(c(n1)SCc2ccc(cc2)OC)C)CCC 6K-568S CCCc1c(n(c(n1)SCc2ccc(cc2)OC)CC(=O)OCC)CCC 6K-570S Cc1cc(cc(c1)n2c(nc3ccccc3c2=O)CCl)C 6K-571S c1ccc(cc1)S(=O)(=O)CC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 6K-572S c1cc(ccc1c2csc(n2)NC(=O)CSc3ccc(cc3)Br)Cl 6K-573S COc1ccc(cc1)SCC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 6K-574S COC(=O)c1ccccc1S(=O)CC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 6K-575S Cc1ccccc1S(=O)CC(=O)Nc2nc(cs2)c3ccc(cc3)Cl 6K-576S Cn1c(c(c(n1)c2ccccc2)C(C#Cc3ccccc3)O)Sc4ccccc4 6K-577S Cn1c(c(c(n1)c2ccccc2)C(C#Cc3ccccc3)O)Sc4ccc(cc4)Cl 6K-578S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)C(C#Cc4ccccc4)O 6K-579S CCCCC#CC(c1c(nn(c1Sc2ccc(cc2)C)C)c3ccccc3)O 6K-580S CCCCC#CC(c1c(nn(c1Sc2ccccc2)C)c3ccccc3)O 6K-581S CCCCC#CC(c1c(nn(c1Sc2ccc(cc2)Cl)C)c3ccccc3)O 6K-582S Cn1c(c(c(n1)c2ccccc2)C(c3cccs3)O)Sc4ccc(cc4)Cl 6K-583S Cc1ccc(cc1)Sc2c(c(nn2C)c3ccccc3)C(c4cccs4)O 6K-584S c1cc(ccc1c2csc(n2)NC(=O)CS(=O)(=O)c3ccc(cc3)Br)Cl 6K-585S Cn1c(c(c(n1)c2ccccc2)C(c3ccc(cc3)Cl)O)Cl 6K-586S Cc1ccc(cc1)CSCc2nc3cc(ccc3c(=O)n2c4cc(cc(c4)C)C)Cl 6K-587S Cc1cc(cc(c1)n2c(nc3cc(ccc3c2=O)Cl)CSc4ccccc4Cl)C 6K-588S Cc1cc(cc(c1)n2c(nc3cc(ccc3c2=O)Cl)CSc4ccc(cc4)F)C 6K-592S Cc1cc(cc(c1)n2c(nc3cc(ccc3c2=O)Cl)CSc4cccc(c4)Cl)C 6K-593S Cc1cc(cc(c1)n2c(nc3cc(ccc3c2=O)Cl)CSCc4ccccc4)C 6K-594S CCCCCCSCc1nc2cc(ccc2c(=O)n1c3cc(cc(c3)C)C)Cl 6K-595S CCCc1c(n(c(n1)SCc2c(cccc2Cl)Cl)C)CCC 6K-602S CCCc1c(n(c(n1)SCc2c(cccc2Cl)Cl)CC#C)CCC 6K-604S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Oc3cccc(c3)C(F)(F)F 6K-612S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Oc3ccc(cc3)OC 6K-613S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Oc3ccc(cc3Cl)Cl 6K-614S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)Oc3ccccc3C(=O)OC 6K-615S Cc1ccc(cc1)c2nc(c(nn2)C(=O)OC)OC 6K-616S CC(C)Cc1c(n(c(n1)S(=O)(=O)Cc2ccc(cc2)F)C)CC(C)C 6K-621S CCCn1c(c(nc1SCc2ccc(cc2)F)CC(C)C)CC(C)C 6K-622S CC(C)Cc1c(n(c(n1)SCc2ccc(cc2)F)CC#C)CC(C)C 6K-623S CCCn1c(c(nc1SCc2c(cccc2Cl)F)CC(C)C)CC(C)C 6K-626S CCOC(=O)Cn1c(c(nc1SCc2c(cccc2Cl)F)CC(C)C)CC(C)C 6K-629S COC(=O)c1ccccc1SC 6K-630S CSc1ccccc1C(=O)NN 6K-632S c1(nnc(s1)N)C(F)(F)F 6K-633S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccccc2 6K-638S CCOC(=O)n1c2ccccc2n(c1=O)C(=O)OCC 6K-644S Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)C(=O)C 6K-650S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)OC 6K-651S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccccc2Cl 6K-652S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] 6K-653S Cc1cccc(c1S(=O)(=O)Nc2cccc(c2)C(=O)C)Cl 6K-654S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)C(C)(C)C 6K-655S CC(=O)c1cccc(c1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F 6K-656S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)C(F)(F)F 6K-657S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)NC(=O)C 6K-658S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)Br 6K-659S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)F 6K-660S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(c(c2)Cl)Cl 6K-661S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2F)F 6K-662S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2Cl)Cl 6K-663S CC(=O)c1cccc(c1)NS(=O)(=O)c2cccc(c2)C(F)(F)F 6K-664S CC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)Cl 6K-665S CC(=O)c1cccc(c1)NS(=O)(=O)C 6K-666S CC(=O)c1cccc(c1)NS(=O)(=O)N(C)C 6K-667S CC(=O)c1cccc(c1)NS(=O)(=O)Cc2ccccc2 6K-668S Cn1c(=O)c2cc(cc(c2nn1)Cl)Cl 6K-669S C(C(=O)Nc1nnc(s1)C(F)(F)F)Cl 6K-672S Cc1ccc(cc1)SCC(=O)Nc2nnc(s2)C(F)(F)F 6K-673S CN1C(=O)C(CC(=N1)c2ccc(cc2)Cl)c3ccc(cc3)Cl 6K-675S CCOC(=O)c1c(nc(nn1)c2cccs2)Oc3ccccc3 6K-676S CCOC(=O)c1c(nc(nn1)c2cccs2)Oc3cccc(c3)C(F)(F)F 6K-677S CCOC(=O)c1c(nc(nn1)c2cccs2)Oc3ccccc3C(=O)OC 6K-678S CCOC(=O)c1c(nc(nn1)c2ccccc2)N3CCOCC3 6K-679S CCOC(=O)/C(=N/Nc1ccc(cc1)Cl)/C#N 6K-902 CCOC(=O)C(=O)Nc1ccc(cc1C(=O)c2ccccc2)Cl 6K-904 c1ccc2c(c1)c3c([nH]2)ncnc3N4CCOCC4 6K-905 CCOC(=O)c1c(c2cc(ccc2[nH]1)Cl)c3ccccc3 6K-906 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3ccccc3)Cl 6K-907 c1ccc(cc1)Cn2c3ccc(cc3c(c2C(F)(F)F)c4ccccc4)Cl 6K-908 c1ccc(cc1)c2c3cc(ccc3n(c2C(F)(F)F)CCOc4ccccc4)Cl 6K-909 c1ccc(cc1)c2c3cc(ccc3[nH]c2C(=O)O)Cl 6K-910 c1ccc(cc1)c2c3cc(ccc3[nH]c2c4ccccc4)Cl 6K-911 CC1=C(C(C(=C(N1)C)C#N)c2ccccc2OC)C#N 6K-913 c1cc(ccc1Cn2c(=O)c(nn(c2=O)c3ccc(cc3)F)C#N)Cl 6K-914 Cc1c(c(c(c(n1)C)C#N)c2ccccc2OC)C#N 6K-915 CC1=C(C(C(=C(N1)C)C#N)c2ccccc2O)C#N 6K-916 CCOC(=O)NC(=O)/C(=N/Nc1c(cccc1F)F)/C#N 6K-917 c1cc(c(c(c1)F)n2c(=O)[nH]c(=O)c(n2)C#N)F 6K-918 COc1ccc(cc1)N2CCN(CC2)/C(=C(\C#N)/C(=S)Nc3ccc(cc3)Cl)/N 6K-919 c1cc(c(c(c1)F)n2c(=O)n(c(=O)c(n2)C#N)Cc3ccc(cc3)Cl)F 6K-920 c1ccc(cc1)NC(=S)/C(=C(\N)/N2CCOCC2)/C#N 6K-921 c1cc(ccc1Nc2c(c(c(s2)C(=O)c3ccc(cc3Cl)Cl)N)C#N)Cl 6K-922 c1ccc(cc1)C(=O)c2c(c(c(s2)Nc3ccccc3)C#N)n4cccc4 6K-923 c1ccc(cc1)c2c3cc(ccc3[nH]c2C(=O)N)Cl 6K-925 CCOC(=O)CNC(=S)/C(=C(\N)/N1CCN(CC1)c2cccc(c2)Cl)/C#N 6K-926 c1ccc(cc1)C2=CSC(=C(C(=N2)N3CCOCC3)C#N)Nc4ccccc4 6K-927 c1ccc(cc1)NC2=C(C(=NC(=CS2)c3ccc(c(c3)Cl)Cl)N4CCOCC4)C#N 6K-928 CCOC(=O)CNc1c(c(ns1)N2CCN(CC2)c3cccc(c3)Cl)C#N 6K-929 c1c(cnc(c1Cl)NCC(CC#N)O)C(F)(F)F 6K-930 c1ccc(cc1)c2c3cc(ccc3[nH]c2C#N)Cl 6K-931 c1cc(ccc1n2c(=O)n(c(=O)c(n2)C#N)Cc3c(cc(cn3)C(F)(F)F)Cl)F 6K-932 c1cc(ccc1Nc2c(c(c(s2)C(=O)c3c(ccs3)Cl)N)C#N)Cl 6K-933 c1cc(c(cc1Cl)Cl)C2CC(=O)NC3=C2C(=O)OC3 6L-001 CN(C)/C=C(/c1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC)\C(=O)C(F)(F)F 6L-002 c1ccc(c(c1)C2CC(=O)NC3=C2C(=O)OC3)F 6L-003 Cc1ccc(cc1)n2cc(c(n2)C(F)(F)F)c3c(c(no3)c4ccccc4Cl)C(=O)OC 6L-005 CN(C)/C=C(/c1c(c(no1)c2c(cccc2Cl)F)C(=O)OC)\C(=O)C(F)(F)F 6L-006 c1cc(ccc1C2CC(=O)NC3=C2C(=O)OC3)Cl 6L-007 CN(C)/C=C(\C=C/C#N)/C#N 6L-008 c1ccc(cc1)c2cc(=O)c3cccc(c3[nH]2)S 6L-009 CCOC(=O)C1=C(N(C(=O)CC1c2ccc(cc2)Cl)Cc3ccc(cc3)Cl)C 6L-011 CCOC(=O)CN1C(=C(C(CC1=O)c2ccc(cc2)Cl)C(=O)OCC)C 6L-012 COc1ccc(cc1)C(=O)c2ccc(s2)CC#N 6L-013 c1cc(ccc1C(=O)c2ccc(s2)CC#N)F 6L-014 COC(=O)c1c(noc1c2cnc(nc2C(F)(F)F)N)c3ccccc3Cl 6L-015 CN(C)/C=C(/C#N)\c1ccc(s1)C(=O)c2ccc(cc2)F 6L-016 CCOC(=O)C1=C(N(C(=O)CC1c2ccc(cc2)Cl)C)C 6L-017 CCOC(=O)/C(=C/Nc1ccc(cc1)Cl)/Sc2c(cc(cn2)C(F)(F)F)Cl 6L-018 COc1ccc(cc1)/C=C(\C#N)/c2ccc(s2)C(=O)c3ccc(cc3)F 6L-019 COC(=O)c1c(noc1c2cnc(nc2C(F)(F)F)N)c3ccccc3 6L-020 CCOC(=O)/C(=C/Nc1ccc(cc1)OC(F)(F)F)/Sc2c(cc(cn2)C(F)(F)F)Cl 6L-021 COc1ccc(cc1)/C=C(\C#N)/c2ccc(s2)C(=O)c3ccc(cc3)OC 6L-022 CN(C)c1ccc(cc1)/C=C(\C#N)/c2ccc(s2)C(=O)c3ccccc3F 6L-023 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)C=O)Cl)C 6L-024 Cc1ccsc1/C=C(\C#N)/c2ccc(s2)C(=O)c3ccc(cc3)Cl 6L-025 COc1ccc(cc1)C(=O)c2ccc(s2)/C(=C/c3cccc(c3)Br)/C#N 6L-026 Cc1ccc(cc1)N/C=C(\C=C/C#N)/C#N 6L-027 CCOC(=O)/C(=C/Nc1ccccc1C(F)(F)F)/Sc2c(cc(cn2)C(F)(F)F)Cl 6L-028 CCOC(=O)C(=O)/C(=C\N(C)C)/c1c(c(no1)c2ccccc2)C(=O)OC 6L-029 CCOC(=O)/C(=C\Nc1ccc(cc1)C(=O)OC)/Sc2c(cc(cn2)C(F)(F)F)Cl 6L-030 COC(=O)c1c(noc1c2cnc(nc2C(F)(F)F)N)c3c(cccc3Cl)Cl 6L-031 COC(=O)c1c(noc1c2cnc(nc2C(F)(F)F)N)c3c(cccc3Cl)F 6L-032 COc1ccc(cc1)C(=O)c2ccc(s2)/C(=C\c3cccn3c4c(cc(cn4)C(F)(F)F)Cl)/C#N 6L-033 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)/C=C(/C#N)\c3ccc(s3)C(=O)c4ccc(cc4)F 6L-034 COc1ccc(cc1)C(=O)c2ccc(s2)/C(=C/c3ccccc3)/C#N 6L-035 Cc1ccc(cc1)n2cc(c(n2)C(F)(F)F)c3c(c(no3)c4ccccc4)C(=O)OC 6L-036 c1cc(c(cc1Cl)Cl)C(=O)c2cc(cs2)CC#N 6L-037 c1cc(ccc1/C=C(\C#N)/c2ccc(s2)C(=O)c3ccc(cc3)F)Cl 6L-038 c1ccc(c(c1)C(=O)c2ccc(s2)/C(=C/c3ccc(cc3)Cl)/C#N)F 6L-039 CCOC(=O)/C(=C\Nc1ccc(cc1)I)/Sc2c(cc(cn2)C(F)(F)F)Cl 6L-040 COC(=O)c1c(noc1c2cn(nc2C(F)(F)F)c3ccccc3F)c4c(cccc4Cl)F 6L-041 COC(=O)c1c(noc1c2cn(nc2C(F)(F)F)c3ccc(cc3)F)c4c(cccc4Cl)F 6L-042 CCOC(=O)C(=O)/C(=C\N(C)C)/c1c(c(no1)c2c(cccc2Cl)F)C(=O)OC 6L-044 COC(=O)c1c(noc1c2cn(nc2C(F)(F)F)c3ccc(cc3Cl)Cl)c4c(cccc4Cl)Cl 6L-045 COC(=O)c1c(noc1c2cn(nc2C(F)(F)F)c3cccc(c3)Cl)c4c(cccc4Cl)Cl 6L-046 CCOC(=O)C(=O)/C(=C\N(C)C)/c1c(c(no1)c2ccccc2Cl)C(=O)OC 6L-047 Cc1ccc2ccccc2c1[N+](=O)[O-] 6L-048 c1cc(ccc1N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N)I 6L-049 COc1ccc(c(c1)N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N)OC 6L-050 c1cc(ccc1C(F)(F)F)N/C=C/c2c3cnc4c(cnn4c3ccn2)C#N 6L-051 c1cc(c(cc1Cl)Cl)CO/N=C/Cc2c3cnc4c(cnn4c3ccn2)C#N 6L-052 Cc1c(oc(n1)c2ccccc2)C(=O)OC 6L-301S CN(C)/C=C/1\C(=O)OC(=N1)c2ccc(cc2)OC 6L-302S COc1ccc(cc1)C(C(=O)O)N 6L-303S Cc1ccc(cc1)Oc2ccc(cn2)/C=N/OCc3ccc(cc3Cl)Cl 6L-306S Cc1ccc(cc1)Oc2ccc(cn2)/C=N/O 6L-307S Cc1ccc(cc1)Oc2ccc(cn2)/C=N/OC(=O)c3ccc(cc3)Cl 6L-308S c1cc(ccc1C#N)Oc2ccc(cn2)C=O 6L-309S CO/N=C/c1ccc(nc1)Sc2ccc(cc2)Cl 6L-312S c1cc(ccc1Sc2ccc(cn2)/C=N/OCc3ccc(cc3Cl)Cl)Cl 6L-313S COc1cc(c(cc1Cl)Cl)n2cccc2 6L-314S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3cccc3 6L-315S COCCOc1cc(c(cc1Cl)Cl)n2cccc2 6L-316S CC(C)Oc1cc(c(cc1Cl)Cl)n2cccc2 6L-317S COc1cc(c(cc1Cl)Cl)n2ccnc2S 6L-320S COc1ccc(cc1)c2nc(no2)C(=O)OC 6L-323S c1ccc(cc1)N2c3ccccc3C(=O)C2=O 6L-325S c1cc(ccc1S(=O)c2ccc(cn2)/C=N/OCc3ccc(cc3Cl)Cl)Cl 6L-326S c1cc(ccc1S(=O)(=O)c2ccc(cn2)/C=N/OCc3ccc(cc3Cl)Cl)Cl 6L-327S c1cc(ccc1Sc2ccc(cn2)/C=N/O)Cl 6L-328S c1cc(ccc1CO/N=C/c2ccc(nc2)Sc3ccc(cc3)Cl)F 6L-329S Cc1ccc(cc1)C(C(=O)O)N 6L-332S c1cc(cc(c1)F)CO/N=C/c2ccc(nc2)Sc3ccc(cc3)Cl 6L-333S COc1cc(c(cc1Cl)Cl)n2ccnc2SC 6L-334S COc1ccc(cc1)c2nc(no2)C(=O)O 6L-338S COCCOc1cc(c(cc1Cl)Cl)n2c(c(cn2)c3ccccc3)N 6L-339S c1ccc(c(c1)C(C(=O)O)N)F 6L-340S c1cc(cc(c1)F)C(C(=O)O)N 6L-341S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3ccnc3S 6L-344S CCOC(=O)COc1cc(c(cc1Cl)Cl)n2cccc2 6L-345S Cc1c(c(n(n1)c2cc(c(cc2Cl)Cl)OCCOC)N)c3ccc(cc3)Cl 6L-346S Cc1c(c(n(n1)c2cc(c(cc2Cl)Cl)OC)N)c3ccc(cc3)Cl 6L-347S c1cc(cc(c1)Br)C(C(=O)O)N 6L-348S c1cc(ccc1C(C(=O)O)N)Br 6L-349S COc1cc(c(cc1Cl)Cl)n2ccnc2SCc3ccccc3 6L-352S COc1ccc(cc1)C(=O)O/N=C/c2ccc(nc2)Sc3ccc(cc3)Cl 6L-353S COc1ccc(cc1)C(=O)O/N=C/c2ccc(nc2)S(=O)c3ccc(cc3)Cl 6L-354S COc1ccc(cc1)C(=O)O/N=C/c2ccc(nc2)S(=O)(=O)c3ccc(cc3)Cl 6L-355S CC(C)Oc1cc(c(cc1Cl)Cl)n2ccnc2S 6L-356S CSc1nccn1c2cc(c(cc2Cl)Cl)OCc3ccccc3 6L-357S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3ccnc3SCc4ccccc4 6L-358S c1cc(cc(c1)Oc2ccc(cn2)C=O)C(F)(F)F 6L-359S CC(C)Oc1cc(c(cc1Cl)Cl)n2ccnc2SC 6L-360S COCCOc1cc(c(cc1Cl)Cl)n2ccnc2S 6L-361S COCCOc1cc(c(cc1Cl)Cl)n2ccnc2SC 6L-362S COCCOc1cc(c(cc1Cl)Cl)n2ccnc2SCc3ccccc3 6L-363S CC(C)Oc1cc(c(cc1Cl)Cl)n2ccnc2SCc3ccccc3 6L-364S c1ccc(c(c1)Sc2ccc(cn2)C=O)Cl 6L-365S c1cc(cc(c1)Oc2ccc(cn2)/C=N/O)C(F)(F)F 6L-366S c1cc(cc(c1)Oc2ccc(cn2)/C=N/OCc3ccc(cc3Cl)Cl)C(F)(F)F 6L-367S Cc1ccc(cc1)Sc2ccc(cn2)/C=N/OC(=O)c3ccccc3Cl 6L-368S CC(C)CC(=O)O/N=C/c1ccc(nc1)Sc2ccc(cc2)Cl 6L-369S c1ccc(c(c1)C(C(=O)O)N)C(F)(F)F 6L-370S CC(C)c1ccc(cc1)C(C(=O)O)N 6L-371S CCOc1ccc(cc1)C(C(=O)O)N 6L-372S c1cc(c(cc1Cl)Cl)C(C(=O)O)N 6L-373S CC(C)CC(=O)O/N=C/c1ccc(nc1)S(=O)(=O)c2ccc(cc2)Cl 6L-375S c1cc(ccc1C#N)Oc2ccc(cn2)/C=N/O 6L-376S c1ccc(cc1)c2nc(cc(n2)N3CCN(CC3)c4cccc(c4)Cl)CSCc5ccc(cc5)Cl 6L-501S c1ccc(cc1)c2nc(cc(n2)N3CCN(CC3)C(c4ccccc4)c5ccccc5)CSCc6ccc(cc6)Cl 6L-502S c1ccc(cc1)CNc2cc(nc(n2)c3ccccc3)CSCc4ccc(cc4)Cl 6L-503S Cc1ccc(cc1)S(=O)(=O)N(CC(=O)N(C)C)c2cc(c(cc2Cl)Cl)OCc3ccccc3 6L-505S CNC(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)c2ccc(cc2)F 6L-506S CN(C)C(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)c2ccc(cc2)F 6L-507S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)F 6L-508S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)F 6L-509S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)F 6L-510S CS(=O)(=O)Cc1cc(nc(n1)c2cccnc2)Cl 6L-511S CC(C)Oc1cc(c(cc1Cl)Cl)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)Cl 6L-517S CC(C)Oc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)Br)S(=O)(=O)c3ccc(cc3)Cl 6L-519S CC(C)Oc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)Cl 6L-520S CC(C)Oc1cc(c(cc1Cl)Cl)N(CC(=O)N(C)C)S(=O)(=O)c2ccc(cc2)Cl 6L-521S CC(C)Oc1cc(c(cc1Cl)Cl)N(CC(=O)NC)S(=O)(=O)c2ccc(cc2)Cl 6L-522S COCCOc1cc(c(cc1Cl)Cl)NS(=O)(=O)c2ccccc2 6L-523S CSc1ccccc1C(=O)Nc2ccc(cc2)C(F)(F)F 6L-528S CSc1ccccc1C(=O)Nc2ccc(cc2)Br 6L-529S CC(=O)Nc1cccn2c1nnc2C(F)(F)F 6L-530S CSc1ccccc1C(=O)Nc2ccc(cc2)Cl 6L-531S Cc1cc(cc(c1)NC(=O)c2ccccc2SC)C 6L-534S CCOC(=O)CN(c1cc(c(cc1Cl)Cl)OCCOC)S(=O)(=O)c2ccc(cc2)Cl 6L-537S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)O)S(=O)(=O)c2ccccc2 6L-538S CSCc1cc(nc(n1)c2ccccc2)N3CCCC3 6L-541S CS(=O)(=O)Cc1cc(nc(n1)c2cccnc2)NCc3ccccc3 6L-542S CS(=O)(=O)Cc1cc(nc(n1)c2cccnc2)NC3CCCCC3 6L-543S CS(=O)(=O)Cc1cc(nc(n1)c2cccnc2)N3CCCC3 6L-544S CS(=O)(=O)Cc1cc(nc(n1)c2cccnc2)N3CCOCC3 6L-545S CS(=O)(=O)Cc1cc(nc(n1)c2ccncc2)N3CCOCC3 6L-546S CS(=O)(=O)Cc1cc(nc(n1)c2ccncc2)N3CCCC3 6L-547S CS(=O)(=O)Cc1cc(nc(n1)c2ccncc2)Sc3ccccc3 6L-548S CC(C)Oc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl 6L-551S CC(C)Oc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 6L-553S Cc1nc(cc(n1)Sc2ccc(cc2)Cl)CS(=O)(=O)C 6L-555S CS(=O)(=O)Cc1cc(nc(n1)c2ccccc2)Sc3ccc(cc3)Br 6L-556S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)Cl 6L-557S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl 6L-558S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)Br)S(=O)(=O)c3ccc(cc3)Cl 6L-559S CNC(=O)CN(c1cc(c(cc1Cl)Cl)OCCOC)S(=O)(=O)c2ccc(cc2)Cl 6L-560S CN(C)C(=O)CN(c1cc(c(cc1Cl)Cl)OCCOC)S(=O)(=O)c2ccc(cc2)Cl 6L-561S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl 6L-562S CS(=O)Cc1cc(nc(n1)c2ccccc2)N3CCOCC3 6L-566S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 6L-567S CSCc1cc(nc(n1)c2cccnc2)Sc3ccc(cc3)Cl 6L-568S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)F)S(=O)(=O)c3ccccc3 6L-570S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)S(=O)(=O)c3ccccc3 6L-571S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)Br)S(=O)(=O)c3ccccc3 6L-572S COc1cc(c(cc1Cl)Cl)NS(=O)(=O)c2cccc(c2)C(F)(F)F 6L-573S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NS(=O)(=O)c3ccccc3 6L-574S CCn1c(nnc1S)c2ccccc2SC 6L-578S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)OC 6L-581S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)OC 6L-582S CNC(=O)CN(c1cc(c(cc1Cl)Cl)OCCOC)S(=O)(=O)c2ccc(cc2)OC 6L-583S COc1cc(c(cc1Cl)Cl)n2c(nnn2)S 6L-584S COCCOc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccccc3 6L-586S COc1cc(c(cc1Cl)Cl)n2c(=O)c3ccccc3nc2SC 6L-587S COc1cc(c(cc1Cl)Cl)n2c(nnn2)SC 6L-588S COc1cc(c(cc1Cl)Cl)n2c(nnn2)SCc3ccccc3 6L-589S COc1cc(c(cc1Cl)Cl)n2c(=O)c3ccccc3nc2SCc4ccccc4 6L-590S CNC(=O)CN(c1cc(c(cc1Cl)Cl)OCCOC)S(=O)(=O)c2ccccc2 6L-591S CN(C)C(=O)CN(c1cc(c(cc1Cl)Cl)OCCOC)S(=O)(=O)c2ccccc2 6L-592S CN(C)C(=O)CN(c1cc(c(cc1Cl)Cl)OCCOC)S(=O)(=O)c2ccc(cc2)OC 6L-593S CS(=O)c1ccccc1COC(=O)Nc2ccc(cc2)Cl 6L-595S Cc1nc(cc(n1)N2CCCC2)CSC 6L-596S CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3ccccc3SC 6L-597S CCn1c(nnc1SC)c2ccccc2SC 6L-598S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)S 6L-599S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)SC 6L-600S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)SCc3ccccc3 6L-601S CSc1ccccc1COC(=O)Nc2ccccc2 6L-603S CSc1ccccc1COC(=O)Nc2cc(cc(c2)Cl)Cl 6L-604S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(nnn2)SCc3ccc(c(c3)Cl)Cl 6L-605S CCOC(=O)CSc1nnnn1c2cc(c(cc2Cl)Cl)OC(C)C 6L-606S CSc1ccccc1c2nnc(o2)S 6L-608S Cc1cccc(c1NC(=O)OCc2ccccc2SC)C 6L-609S CS(=O)c1ccccc1COC(=O)Nc2ccccc2 6L-610S CSc1ccccc1c2nnc(o2)SCc3ccc(cc3Cl)Cl 6L-611S CSc1ccccc1c2nnc(o2)SC 6L-612S CSc1ccccc1c2nnc(o2)SCC=C 6L-613S CCOC(=O)CSc1nnc(o1)c2ccccc2SC 6L-614S COCCOc1cc(c(cc1Cl)Cl)n2c(nnn2)SCc3ccccc3 6L-617S COCCOc1cc(c(cc1Cl)Cl)n2c(nnn2)SCC(=O)OC 6L-618S CSc1ccccc1COC(=O)Nc2cccc(c2)Cl 6L-621S Cc1ccc(cc1)NC(=O)OCc2ccccc2SC 6L-622S CS(=O)c1ccccc1COC(=O)Nc2cc(cc(c2)Cl)Cl 6L-623S CS(=O)(=O)c1ccccc1COC(=O)Nc2cc(cc(c2)Cl)Cl 6L-624S Cc1ccccc1NC(=O)OCc2ccccc2SC 6L-625S CS(=O)(=O)c1ccccc1COC(=O)Nc2ccc(cc2)Cl 6L-627S CSc1ccccc1COC(=O)Nc2ccc(cc2)Cl 6L-655S CC(C)(CCl)C(=O)Nc1ccc(cc1)OC 6L-700 CC1(CN(C1=O)c2ccc(cc2)OC)C 6L-701 c1c(cc(cc1Cl)Cl)Oc2cc(cnc2C(=O)N)C(F)(F)F 6L-702 Cc1cc(ccc1Oc2cc(cnc2C(=O)N)C(F)(F)F)Cl 6L-703 c1cc(c(cc1Cl)Cl)/C=C/c2ccnc(n2)Sc3cc(cnc3C#N)C(F)(F)F 6L-704 COc1ccc(cc1)N2CCN(CC2)c3cc(cnc3C#N)C(F)(F)F 6L-705 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4cc(cnc4C#N)C(F)(F)F 6L-706 c1c(cnc(c1Sc2[nH]nc(n2)N)C#N)C(F)(F)F 6L-708 c1cc(c(cc1Cl)Cl)/C=C/c2ccnc(n2)Sc3cc(cnc3C(=O)N)C(F)(F)F 6L-709 c1cc(c(cc1C(=O)C[N+]23CN4CN(C2)CN(C4)C3)Cl)Cl.[Br-] 6L-900 CCOC(=O)c1c(c[nH]c1N)c2cccc(c2)[N+](=O)[O-] 6L-902 c1cc(cc(c1)[N+](=O)[O-])c2c[nH]c(c2C#N)N 6L-903 COc1ccc(cc1OC2CCCC=C2)C=O 6L-905 CCOC(=O)c1c(c2ccccc2[nH]1)NC(=O)c3cccc(c3)C(F)(F)F 6L-907 c1cc(ccc1N/C=C/C(=O)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-])OC(F)(F)F 6L-908 CCOC(=O)c1c(c2ccccc2n1Cc3ccc(cc3Cl)Cl)N(Cc4ccc(cc4Cl)Cl)C(=O)c5cccc(c5)C(F)(F)F 6L-909 c1cc(ccc1CNC(=O)CO/N=C/CC(=O)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-])Cl 6L-910 COc1ccc(cc1)N/C=C/C(=O)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 6L-911 c1ccc2c(c1)C(=O)c3ccc(cc3C2=O)CC#N 6L-912 c1ccc2c(c1)C(=O)c3ccc(cc3C2=O)CC(=O)O 6L-914 c1cc(ccc1C(=O)OC(CC#N)CNc2c(cc(cn2)C(F)(F)F)Cl)Cl 6L-916 c1ccc2c(c1)C(=O)c3ccc(cc3C2=O)CC(=O)N4CCOCC4 6L-917 C/C(=C(/C#N)\C(=O)Nc1cccc(c1)C(F)(F)F)/O 6L-918 COc1ccc2c(c1O)C3CCC=CC3=C2 6L-920 Cc1c(c(sc1C(=O)N/C=N/OCc2ccc(cc2)Cl)C#N)c3ccccc3 6M-001 Cc1c(c(sc1C(=O)N/C=N/OCc2c(cccc2Cl)F)C#N)c3ccccc3 6M-002 Cc1ccc(cc1)C(=O)NNc2c(nc3ccccc3n2)C(F)(F)F 6M-003 Cc1ccc(cc1)/C=N/Nc2c(nc3ccccc3n2)C(F)(F)F 6M-004 c1ccc2c(c1)nc(c(n2)NNS(=O)(=O)c3ccc(cc3)Br)C(F)(F)F 6M-005 c1ccc2c(c1)nc(c3n2c(nn3)c4ccc(cc4)Br)C(F)(F)F 6M-006 c1cc(c(c(c1)Cl)c2nnc3n2c4c(cccn4)cc3C(F)(F)F)F 6M-007 c1ccc(cc1)/C=C/c2nnc3n2c4ccccc4nc3C(F)(F)F 6M-008 c1ccc2c(c1)nc(c3n2c(nn3)c4c(cccc4Cl)Cl)C(F)(F)F 6M-009 COc1ccc(cc1)C(=O)NNc2c(nc3ccccc3n2)C(F)(F)F 6M-010 COc1ccc(cc1)c2nnc3n2c4c(cc3)c(cc(n4)C(F)(F)F)C(F)(F)F 6M-011 c1ccc2c(c1)nc(c(n2)N/N=C/c3ccc(c(c3)[N+](=O)[O-])Cl)C(F)(F)F 6M-012 c1ccc2c(c1)nc(c3n2c(nn3)c4ccc(c(c4)[N+](=O)[O-])Cl)C(F)(F)F 6M-013 c1ccc(cc1)C(=O)NNc2c(nc3ccccc3n2)C(F)(F)F 6M-014 c1ccc2c(c1)nc(c(n2)NNC(=O)c3ccco3)C(F)(F)F 6M-015 Cc1c(c(sc1C(=O)N/C=N/OCc2ccccc2F)C#N)c3ccccc3 6M-016 Cc1ccc(cc1)c2nnc3n2c4ccccc4nc3C(F)(F)F 6M-018 c1ccc2c(c1)nc(c(n2)NNS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F 6M-019 CO/N=C/Cc1c(sc(c1c2ccccc2)C#N)C#N 6M-021 CN(c1c(nc2ccccc2n1)C(F)(F)F)NC(=O)c3ccc(cc3)OC 6M-022 Cc1ccc(cc1)CO/N=C/NC(=O)c2c(c(c(s2)C#N)c3ccccc3)C 6M-023 Cc1ccc(cc1)C(=O)NN(C)c2c(nc3ccccc3n2)C(F)(F)F 6M-024 CN(c1c(nc2ccccc2n1)C(F)(F)F)NC(=O)c3ccco3 6M-025 CN(c1c(nc2ccccc2n1)C(F)(F)F)NC(=O)c3ccccc3 6M-026 Cc1ccc(cc1)CO/N=C/Cc2c(sc(c2c3ccccc3)C#N)C#N 6M-027 c1ccc(cc1)c2c(c(sc2C#N)C#N)C/C=N/OCc3ccccc3F 6M-029 Cc1ccc(cc1)C(=O)Nc2ncc3c(n2)cccc3Cl 6M-030 CN(c1c(nc2ccccc2n1)C(F)(F)F)NS(=O)(=O)c3ccc(cc3)OC 6M-031 CN(c1c(nc2ccccc2n1)C(F)(F)F)NS(=O)(=O)c3ccc(cc3)Cl 6M-032 CN(c1c(nc2ccccc2n1)C(F)(F)F)NS(=O)(=O)c3ccccc3 6M-033 CN(c1c(nc2ccccc2n1)C(F)(F)F)NS(=O)(=O)c3ccc(cc3)Br 6M-034 c1ccc(cc1)/C(=C/C(=O)[O-])/C#N.[K+] 6M-035 c1cc(ccc1C2=CC(=O)N(C2=O)Nc3ccc(cc3)F)Cl 6M-039 Cc1ccc(cc1)NN2C(=O)C=C(C2=O)c3ccc(cc3)Cl 6M-040 c1ccc(cc1)C2=CC(=O)OC2=O 6M-041 c1ccc(cc1)/C(=C/C(=O)O)/C(=O)O 6M-043 Cc1ccc(cc1)NN2C(=O)C=C(C2=O)c3ccccc3 6M-046 Cc1cc(cc(c1)NC(=O)c2ccccc2CC[N+](=O)[O-])C 6M-047 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)Nc2ccc(cc2)Br 6M-048 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)Nc2ccc(cc2)F 6M-049 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)Nc2cccc(c2)C(F)(F)F 6M-050 COC(=O)c1ccc(cc1)NC(=O)c2ccccc2CC[N+](=O)[O-] 6M-051 c1ccc(cc1)CSCc2cc(no2)c3ccc(cc3)Cl 6M-303S c1cc(cc(c1)Cl)SCc2cc(no2)c3ccc(cc3)Cl 6M-304S c1ccc2c(c1)n(c(=O)o2)CC(=O)NCc3ccc(cc3)Cl 6M-306S COc1ccc(cc1)c2cc(on2)CSc3ccccc3 6M-309S COc1ccc(cc1)c2cc(on2)CSc3ccc(cc3)Cl 6M-310S c1ccc(cc1)CS(=O)(=O)Cc2cc(no2)c3ccc(cc3)Cl 6M-311S c1cc(cc(c1)Cl)S(=O)(=O)Cc2cc(no2)c3ccc(cc3)Cl 6M-312S c1ccc2c(c1)n(c(=O)o2)CC(=O)N3CCCC3 6M-317S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2csc(n2)c3ccccc3 6M-318S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2csc(n2)c3ccccc3Cl 6M-319S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2csc(n2)c3ccc(cc3)Cl 6M-320S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2csc(n2)C 6M-321S c1ccc(cc1)S(=O)(=O)Cc2cc(no2)c3ccccc3Cl 6M-322S COc1ccc(cc1)c2cc(on2)CS(=O)(=O)c3ccccc3 6M-323S c1ccc(c(c1)N2CC(=O)N(C2=O)N)O 6M-324S CN(C)C(=O)Cn1c2ccccc2oc1=O 6M-327S C=CCNC(=O)Cn1c2ccccc2oc1=O 6M-328S c1ccc(c(c1)c2cc(on2)CN3C(=O)c4ccccc4C3=O)Cl 6M-329S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2csc(n2)c3cccnc3 6M-331S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2csc(n2)c3ccccn3 6M-332S Cc1ccc2c(c1)N(C(CO2)C(C)(C)C)C(=O)c3cccc(c3)C(F)(F)F 6M-333S Cc1ccc2c(c1)N(C(CO2)C(C)(C)C)C(=O)c3cccc(c3)OC 6M-334S CCOC(=O)c1c(nc2n1ccs2)C 6M-336S Cc1c(n2ccsc2n1)C(=O)O 6M-337S COc1ccc(cc1)c2cc(on2)CN3C(=O)c4ccccc4C3=O 6M-339S CC(C)C(=O)NCc1cc(no1)c2ccccc2Cl 6M-340S c1ccc(cc1)S(=O)(=O)NCc2cc(no2)c3ccccc3Cl 6M-341S COc1ccc(cc1)S(=O)(=O)NCc2cc(no2)c3ccccc3Cl 6M-342S c1cc(ccc1c2cc(on2)CN)Cl 6M-343S Cc1c(n2ccsc2n1)C(=O)Nc3ccc(cc3)OC 6M-345S c1ccc2c(c1)nc(c(=O)o2)N 6M-346S c1ccc(c(c1)c2cc(on2)CNS(=O)(=O)c3cc(ccc3Cl)Cl)Cl 6M-348S c1ccc(c(c1)c2cc(on2)CNS(=O)(=O)c3ccc(cc3)Cl)Cl 6M-349S CC(=O)NCc1cc(no1)c2ccc(cc2)OC 6M-350S COc1ccc(cc1)OCc2cc(no2)c3ccc(cc3)Cl 6M-351S COc1ccc(cc1)c2cc(on2)CN 6M-352S COc1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3ccccc3 6M-353S COc1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3ccc(cc3)F 6M-354S c1ccc(cc1)c2cc(on2)COc3ccccc3 6M-355S c1ccc(cc1)c2cc(on2)COc3ccc(cc3Cl)Cl 6M-356S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2csc(n2)c3ccncc3 6M-357S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)c2cnc(s2)c3ccc(cc3)OC 6M-358S Cc1cc(nc(c1S(=O)(=O)C)O)c2ccccc2 6M-359S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)Cl)c3ccccc3 6M-360S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)Cl)c3ccccc3 6M-361S Cc1ccc(cc1)Sc2c(c(cc(n2)c3ccccc3)C)S(=O)(=O)c4ccccc4 6M-362S Cc1ccc(cc1)Sc2c(c(cc(n2)C)C)S(=O)(=O)C 6M-363S c1ccc(cc1)c2cc(on2)COc3cccc(c3)C(F)(F)F 6M-364S c1ccc(cc1)c2cc(on2)COc3ccc(cc3)F 6M-365S c1ccc(cc1)S(=O)(=O)NCc2cc(no2)c3ccc(cc3)Cl 6M-366S Cc1ccc(cc1)S(=O)(=O)c2c(c(cc(n2)C)C)S(=O)(=O)C 6M-367S Cc1cc(nc(c1S(=O)(=O)C)Cl)c2ccccc2 6M-368S Cc1cc(nc(c1S(=O)(=O)C)SCc2ccc(cc2)OC)C 6M-369S c1cc(ccc1c2cc(on2)CNC(=O)C(F)(F)F)Cl 6M-370S c1cc(ccc1c2cc(on2)COc3cc(cc(c3)Cl)Cl)Cl 6M-371S c1ccc(cc1)OCc2cc(no2)c3ccc(cc3)Cl 6M-372S Cc1cccc(c1S(=O)(=O)NCc2cc(no2)c3ccc(cc3)Cl)Cl 6M-373S c1cc(ccc1c2cc(on2)CNS(=O)(=O)c3cc(ccc3Cl)Cl)Cl 6M-374S c1ccc(cc1)c2cc(on2)CN 6M-375S Cc1ccc(cc1)n2c(c(cn2)Cl)C(=O)NCC=C 6M-506S Cc1ccc(cc1)n2c(=O)c(c(cn2)Cl)Sc3ccc(cc3)Cl 6M-507S Cn1c(c(c(n1)c2ccccc2)CN3CCOCC3)Cl 6M-508S Cn1c(c(c(n1)c2ccccc2)CN(C)C)Cl 6M-509S Cc1ccc(cc1)n2c(=O)c(c(cn2)N3CCOCC3)Sc4ccc(cc4)Cl 6M-511S Cc1ccccc1C(=O)NCc2nnc(n2C(C)C)SCC=C 6M-512S Cc1ccccc1C(=O)NCc2nnc(n2C(C)C)SCc3ccc(cc3)OC 6M-513S COC(=O)C(CCSC)NS(=O)(=O)c1ccc(cc1)Cl 6M-516S COc1cc(c(cc1Cl)Cl)NC(=O)c2ccc(cc2)C(=O)C(F)(F)F 6M-518S Cn1c(cc(n1)OCC(CS(=O)(=O)Cc2ccccc2)O)C(F)(F)F 6M-527S Cn1c(cc(n1)OCC(CS(=O)(=O)Cc2ccc(cc2)OC)O)C(F)(F)F 6M-528S Cc1ccc(cc1)S(=O)(=O)NC(Cc2ccccc2)C(=O)OC 6M-538S Cn1c(cc(n1)OC(=O)Nc2cccc(c2)Cl)C(F)(F)F 6M-539S Cn1c(cc(n1)OC(=O)Nc2ccc(cc2)Cl)C(F)(F)F 6M-540S Cn1c(cc(n1)OC(=O)NC2CCCCC2)C(F)(F)F 6M-541S CCCNC(=O)Oc1cc(n(n1)C)C(F)(F)F 6M-542S Cc1cccc(c1NC(=O)Oc2cc(n(n2)C)C(F)(F)F)C 6M-543S Cn1c(cc(n1)OC(=O)Nc2ccc(cc2)F)C(F)(F)F 6M-545S Cn1c(cc(n1)OC(=O)NCC=C)C(F)(F)F 6M-546S c1cc(sc1)c2c(c(nc(n2)N)S)C#N 6M-547S CSc1c(c(nc(n1)N)c2cccs2)C#N 6M-548S Cc1ccc(cc1)n2c(c(cn2)Cl)C(=O)NC3CC3 6M-549S Cn1c2c(cc(s2)C(=O)OC)c(n1)c3ccccc3 6M-550S Cc1ccc(cc1)n2c(=O)c(c(cn2)N(C)C)Oc3ccc(cc3)OC 6M-552S c1cc(ccc1C(=O)NCCO)Br 6M-559S Cn1c2c(cc(s2)C(=O)O)c(n1)c3ccccc3 6M-560S c1cc(cc(c1)Cl)C(=O)NCCO 6M-565S c1cc(ccc1n2c(=O)c(c(cn2)Cl)Oc3ccc(cc3)Cl)F 6M-566S Cc1ccc(cc1)n2c(=O)c(c(cn2)Cl)Oc3ccc(cc3)Cl 6M-567S CNC(=O)c1c(cnn1c2ccc(cc2)F)Cl 6M-568S Cn1c(cnc1S(=O)(=O)Cc2c(cccc2Cl)Cl)CO 6M-626S COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccc(cc3)Br)Cl 6M-654S COc1ccc(cc1)Oc2c(cnn(c2=O)c3c(cc(cc3Cl)F)Cl)Cl 6M-655S CC(=O)Nc1cccc(c1)Oc2ccc3nnc(n3n2)C(F)(F)F 6M-700 Cc1c(nn(n1)c2ccc(cc2)F)C(=O)Nc3ccc(cc3)Br 6M-701 CC(C)(CNc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])SCc2cccc(c2)C(F)(F)F 6M-702 Cc1c(c(=O)ccn1c2ccc(cc2)OC)Cc3c(cccc3Cl)Cl 6M-703 c1ccn(c1)c2ccc3nnc(n3n2)C(F)(F)F 6M-704 Cc1ccc(cc1)C(=O)CSc2c(c(sn2)C)C#N 6M-705 Cc1c(c(ns1)SCC(=O)c2ccc(cc2)[N+](=O)[O-])C#N 6M-706 Cc1c2c(c(sc2ns1)C(=O)c3ccccc3)N 6M-710 c1cc(ccc1Oc2ccc3nnc(n3n2)C(F)(F)F)Cl 6M-711 COc1cccc(c1)Oc2ccc3nnc(n3n2)C(F)(F)F 6M-712 COC(=O)c1c2c([nH]c1C(=O)OC)-c3ccccc3CC2 6M-715 CN(C)/C=C/C(=O)C(Cc1c(cccc1Cl)Cl)C(=O)/C=C\N(C)C 6M-716 Cc1c(c(ns1)SCC(=O)c2ccccc2Cl)C#N 6M-717 Cc1c(c(ns1)SCC(=O)c2ccc(cc2Cl)Cl)C#N 6M-718 c1cc(ccc1Oc2ccc3nnc(n3n2)C(F)(F)F)F 6M-719 c1cc(nn2c1nnc2C(F)(F)F)n3ccnc3 6M-720 Cc1cc(c(c(c1)C)CSC(C)(C)CNC(=O)c2ccccc2C(F)(F)F)C 6M-721 Cc1cc(nc(n1)N2CCOCC2)C(=O)N 6M-722 CC(=O)C(Cc1c(cccc1Cl)F)C(=O)C 6M-724 CC(C)(CNS(=O)(=O)c1ccc(cc1)OC)SCc2ccc(cc2)Cl 6M-726 CC(=O)C(Cc1ccc(cc1Cl)Cl)(Cc2ccc(cc2Cl)Cl)C(=O)C 6M-727 CC(C)(CNS(=O)(=O)c1ccc(cc1)F)SCc2ccc(cc2)Cl 6M-728 CC(C)(CNc1ccc(cn1)[N+](=O)[O-])SCc2cccc(c2)C(F)(F)F 6M-729 CC(=O)/C(=C/Nc1ccc(cc1)Cl)/c2ccccc2 6M-730 CC(=O)/C(=C/Nc1cc(cc(c1)Cl)Cl)/c2ccccc2 6M-734 CN(C)/C=C/C(=O)C(Cc1c(cccc1Cl)F)C(=O)/C=C\N(C)C 6M-735 Cc1coc(=N)n1CC(=O)c2ccc(cc2)Cl 6M-738 c1cc(c(cc1Cl)Cl)n2cnc(n2)c3ncn(n3)c4ccc(cc4Cl)Cl 6M-739 CC(=O)/C(=C/Nc1ccc(cc1)OC)/c2ccccc2 6M-740 CC(=O)c1ccc(cc1)N/C=C(\c2ccccc2)/C(=O)C 6M-742 CC(=O)/C(=C/Nc1ccc(cc1)Oc2ccccc2)/c3ccccc3 6M-743 CC(=O)/C(=C/Nc1ccc(cc1)I)/c2ccccc2 6M-745 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)NCc3cccc(c3)C(F)(F)F 6M-900 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)NCCc3ccccc3 6M-901 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)NCCCOC 6M-902 c1ccc(cc1)C(=O)/C=C/c2ccsc2 6M-903 CC(=O)Nc1ccc(cn1)Sc2c(cccn2)C(=O)O 6M-904 CC(=O)Nc1ccc(cn1)Sc2c(cccn2)C(=O)Nc3ccc(cc3)F 6M-905 CC(=O)Nc1ccc(cn1)Sc2c(cccn2)C(=O)Nc3ccc(cc3)OC(F)(F)F 6M-906 CC(=O)Nc1ccc(cn1)Sc2c(cccn2)C(=O)Nc3ccc(cc3)OC 6M-907 CC(=O)Nc1ccc(cn1)Sc2c(cccn2)C(=O)Nc3cc(cc(c3)Cl)Cl 6M-908 Cc1cc(cc(c1)NC(=O)c2cccnc2Sc3ccc(nc3)NC(=O)C)C 6M-909 COc1ccc(cc1)C(=O)NCCONC(=O)c2ccc(cc2)OC 6M-910 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)N3CCCC3 6M-911 CC(=O)Nc1ccc(cn1)Sc2ccccc2C(=O)N3CCOCC3 6M-912 Cc1cc(n2c(c(nc2n1)C(=O)/N=C/NOCc3c(cccc3Cl)F)C#N)C 6M-913 Cc1cc(n2c(c(nc2n1)C(=O)N/C=N\OCc3ccc(cc3)Cl)C#N)C 6M-914 Cc1ccc(cc1)C(=O)NCCONC(=O)c2ccc(cc2)C 6M-915 C/[N+](=C\c1coc2ccccc2c1=O)/[O-] 6M-916 CN1C(C2C(O1)C(=O)N(C2=O)c3ccc(cc3)Cl)c4coc5ccccc5c4=O 6M-917 CN1C(C2C(O1)C(=O)N(C2=O)c3ccc(cc3Cl)Cl)c4coc5ccccc5c4=O 6M-920 c1ccc2c(c1)n3c(nnc3c4n2c(nn4)CCl)CCl 6M-922 COC(=O)Cc1nnc2n1c3ccccc3n4c2nnc4CC(=O)OC 6M-923 CN1C(C2C(O1)C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)c4coc5ccccc5c4=O 6M-924 CC(=O)CC(=O)Nc1ccc(cn1)I 6M-925 c1cc(ncc1I)NC(=O)CCl 6M-927 c1cc(ncc1I)NC(=O)CN2CCOCC2 6M-928 CC(C)(C)C(C(=O)NC)NC(=O)CCl 6N-002 COC(=O)C(CC1CCCCC1)NC(=O)CCl 6N-003 COc1ccc(cc1)C(=O)OCC(c2ccccc2)NC(=O)Nc3ccc(cc3)Cl 6N-004 Cc1c2c(nn(c2nc(c1Cl)C)c3ccccc3)c4ccccc4 6N-005 CCOC(=O)c1c2ccc(cc2n3c1cccc3)O 6N-008 C1c2c(c(c(nc2OC1C(F)(F)F)N)C#N)N 6N-009 COC(=O)C(CC1CCCCC1)NC(=O)CN2CCOCC2 6N-010 c1c(cc(cc1Cl)Cl)NC(=O)C(CC2CCCCC2)N3CCS(=O)(=O)CC3 6N-011 CC(C)(C)C(C(=O)OC)n1cccc1C=O 6N-012 CC(C)(C)C(C(=O)NC)NC(=O)CN1CCN(CC1)c2ccccc2 6N-013 CC(C)(C)C(C(=O)OC)n1cccc1C=C(C#N)C#N 6N-016 CC(C)c1ccc(cc1)n2cnn(c2=O)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 6N-017 CC(C)c1ccc(cc1)n2cnn(c2=O)c3c(cccn3)[N+](=O)[O-] 6N-018 c1cc(cc(c1)n2cnn(c2=O)CC#N)C(F)(F)F 6N-019 c1cc(ccc1C(=O)Nc2ncc(s2)[N+](=O)[O-])F 6N-020 c1cc(sc1)C(=O)Nc2ncc(s2)[N+](=O)[O-] 6N-021 c1ccc(cc1)OCC2Cc3c(c(c(nc3O2)N)C#N)N 6N-023 CC(C)(C)C(C(=O)NC)NC(=O)CN1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 6N-025 CCOC(=O)Cn1c(=O)n(cn1)c2ccccc2 6N-027 c1cc(c(nc1)n2c(=O)n(cn2)c3ccc(cc3)Br)[N+](=O)[O-] 6N-029 COC(=O)C(CC1CCCCC1)Nc2c(cccn2)[N+](=O)[O-] 6N-031 CC(C)(C)C(C(=O)OC)NS(=O)(=O)c1ccc(cc1)Br 6N-032 CC(C)(C)C(C(=O)OC)Nc1ccc(cc1[N+](=O)[O-])C(F)(F)F 6N-033 c1cc(cc(c1)[N+](=O)[O-])/C=N/O 6N-034 CC(C)c1ccc(cc1)n2cnn(c2=O)Cc3ccc(cc3)Cl 6N-036 Cc1ccc(cc1)Cn2c(=O)n(cn2)c3ccccc3 6N-037 CC(C)(C)C(C(=O)OC)/N=C/c1ccc(cc1)[N+](=O)[O-] 6N-038 c1ccn(c1)c2cnccn2 6N-039 Cc1cc(c(c(c1)C)Cn2c(=O)n(cn2)c3ccc(cc3)Br)C 6N-040 CC(C)(C)C(C(=O)NC)NC(=O)CON1C(=O)c2ccccc2C1=O 6N-041 c1cc(cc(c1)n2cnn(c2=O)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 6N-042 COc1cccc(c1)Cn2c(=O)n(cn2)c3ccc(cc3)Br 6N-044 c1cc(cc(c1)F)Cn2c(=O)n(cn2)c3cccc(c3)C(F)(F)F 6N-045 CCOC(=O)Cn1c(=O)n(cn1)c2ccc(cc2)Br 6N-046 COc1ccc(cc1)C(=O)N2CCCc3c2cccc3 6N-047 COc1ccc(cc1)N/C(=N\O)/c2cccc(c2)[N+](=O)[O-] 6N-048 Cc1cccc(c1)C(=O)N2CCCc3c2cccc3 6N-049 c1cc(ccc1n2cn[nH]c2=O)Oc3c(cc(cn3)C(F)(F)F)Cl 6N-051 Cc1ccc(cc1)n2cn[nH]c2=O 6N-052 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2ccnc3 6N-054 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)cccn3 6N-055 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2nccc3 6N-056 c1ccc(cc1)C(=O)NC(=S)Nc2cc3ccccc3nc2 6N-057 c1ccc(cc1)C(=O)N2CCCc3c2cccc3 6N-058 c1ccc2c(c1)ccc(n2)/C=N/Nc3ccc(cc3)C(=O)O 6N-059 c1ccc2c(c1)CCCN2C(=O)c3cc(cc(c3)Cl)Cl 6N-062 c1cc2cccnc2c(c1)NC(=S)N 6N-063 c1cc2cnccc2c(c1)NC(=S)N 6N-064 c1cc2cc(ccc2nc1)NC(=S)N 6N-065 Cc1ccc(cc1)n2cnn(c2=O)CC3CC3 6N-066 c1ccnc(c1)n2cnn(c2=O)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 6N-067 c1ccc2c(c1)cc(cn2)NC(=S)N 6N-068 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)/N=N/c3ccccc3 6N-069 c1ccc(cc1)/N=N/c2ccc(cc2)NC(=S)N 6N-070 Cc1ccc(cc1)Cn2c(=O)n(cn2)c3ccccn3 6N-071 c1ccc2c(c1)nc(c3n2ccc3)n4cccc4 6N-072 Cc1ccc(cc1)n2cnn(c2=O)c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 6N-073 COc1ccc(cc1)C(=O)NC2CCCCCC2 6N-074 c1cc(ccc1Oc2ccc(cc2)S(=O)(=O)N)S(=O)(=O)N 6N-076 c1ccc2c(c1)CCCN2C(=O)c3c(cccc3Cl)Cl 6N-077 COc1cc(ccc1O)/C=N/NC(=O)c2ccc(cc2)N3CCCC3=O 6N-078 c1ccc(cc1)C(=O)NC(=S)Nc2ccnc(n2)O 6N-080 c1cc(ccc1C(=O)NC2CCCCCC2)I 6N-082 c1cc(ccc1n2cn[nH]c2=O)OC(F)(F)F 6N-083 CN(C)S(=O)(=O)c1ccc(cc1)Oc2ccc(cc2)S(=O)(=O)N(C)C 6N-084 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)I)Oc3c(cc(cn3)C(F)(F)F)Cl 6N-085 c1cc(ccc1Oc2ccc(cc2)S(=O)(=O)N3CCOCC3)S(=O)(=O)N4CCOCC4 6N-086 c1cc(ccc1Cn2c(=O)n(cn2)c3ccc(cc3)OC(F)(F)F)C(F)(F)F 6N-087 c1cc(ccc1C(=O)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)I 6N-088 Cc1ccc(cc1)CS(=O)c2nc3c(c(n2)Cl)CCCC3 6N-301S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)Cl)CCCC3 6N-302S c1ccc(cc1)N(CC(=O)Oc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccccc3 6N-303S c1ccc(cc1)N(CC(=O)Oc2ccc(cc2Cl)Cl)S(=O)(=O)c3ccccc3 6N-304S CCC(=O)O/N=C/1\CCS(=O)(=O)c2c1ccs2 6N-306S c1cc(ncc1C(=O)O/N=C/2\CCS(=O)(=O)c3c2ccs3)Cl 6N-307S CCNc1c2c(nc(n1)SCc3ccc(cc3)C)CCCC2 6N-308S Cc1ccc(cc1)CSc2nc3c(c(n2)N4CC(OC(C4)C)C)CCCC3 6N-309S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)N(C)C)CCCC3 6N-310S Cc1ccc(cc1)CSc2nc3c(c(n2)Oc4ccc(cc4)C(C)(C)C)CCCC3 6N-311S Cc1ccc(cc1)CSc2nc3c(c(n2)Oc4ccc(cc4)C)CCCC3 6N-312S Cc1ccc(cc1)CSc2nc3c(c(n2)Oc4cc(c(cc4Cl)Cl)Cl)CCCC3 6N-313S Cc1ccc(cc1)CSc2nc3c(c(n2)Oc4ccc(cc4)Cl)CCCC3 6N-314S Cc1ccc(cc1)CSc2nc3c(c(n2)Oc4cccc(c4)Cl)CCCC3 6N-315S COc1ccc(cc1)C(=O)/C=C/c2ccc(cc2Cl)Cl 6N-316S Cc1cccc(c1OC(=O)CN(c2ccccc2)S(=O)(=O)c3ccccc3)C 6N-317S c1ccc(cc1)N(CC(=O)Oc2ccc3ccccc3c2)S(=O)(=O)c4ccccc4 6N-319S c1ccc(cc1)N(CC(=O)Oc2cc(ccc2Cl)Cl)S(=O)(=O)c3ccccc3 6N-320S c1ccc(cc1)N(CC(=O)Oc2ccc(c3c2cccc3)Cl)S(=O)(=O)c4ccccc4 6N-321S Cc1cc(=O)n(c2c1cccc2)C 6N-323S c1cc(ccc1C(=O)OC2CCS(=O)(=O)c3c2ccs3)F 6N-329S c1cc(c(c(c1)F)C(=O)OC2CCS(=O)(=O)c3c2ccs3)F 6N-330S Cc1cccc(c1)C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-331S CS(=O)(=O)N(CC(=O)O)c1ccc(cc1Cl)Cl 6N-336S Cc1c(snn1)NC(=O)OCC=C 6N-337S c1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2ccc(cc2F)F 6N-339S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)Cl 6N-342S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)Sc4ccc(cc4)C 6N-343S c1ccc(cc1)c2nc(cc(n2)Cl)N3CCOCC3 6N-344S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)N4CCOCC4 6N-345S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)Cl 6N-346S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)Oc4ccc(cc4)C 6N-347S Cc1cc(=O)n(c2c1cccc2)Cc3ccccc3 6N-348S Cc1cc(=O)n(c2c1cccc2)CC=C 6N-349S Cc1cc(=O)n(c2c1cccc2)Cc3ccc(cc3)Cl 6N-350S c1cc(ccc1C(=O)OC2CCS(=O)(=O)c3c2ccs3)Cl 6N-352S c1cc(cc(c1)C(F)(F)F)C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-353S COc1cccc(c1)C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-354S Cc1ccc(cc1)C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-355S c1cc(cc(c1)Cl)C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-358S c1cc(c(cc1Cl)Cl)C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-359S c1cc(ncc1C(=O)OC2CCS(=O)(=O)c3c2ccs3)Cl 6N-360S c1cc(sc1)C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-361S c1ccc(cc1)S(=O)(=O)N(CC(=O)Oc2ccc(cc2)Cl)c3cccc(c3)C(F)(F)F 6N-364S COc1ccc(cc1)OC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccccc3 6N-365S Cc1ccccc1C(=O)OC2CCS(=O)(=O)c3c2ccs3 6N-366S c1ccc(c(c1)C(=O)OC2CCS(=O)(=O)c3c2ccs3)Cl 6N-367S c1ccc(cc1)S(=O)(=O)N(CC(=O)Oc2ccc(cc2Cl)Cl)c3cccc(c3)C(F)(F)F 6N-368S c1ccc(cc1)S(=O)(=O)N(CC(=O)Oc2ccc(cc2)Cl)c3ccc(cc3F)F 6N-369S Cc1c(snn1)NC(=O)OCCCl 6N-370S Cc1c(snn1)NC(=O)OCc2ccc(cc2Cl)Cl 6N-371S Cc1c(snn1)NC(=O)OCc2ccccc2Cl 6N-372S c1ccc(cc1)S(=O)(=O)N(CC(=O)Oc2ccc(cc2Cl)Cl)c3ccc(cc3F)F 6N-374S COc1ccc(cc1)OC(=O)CN(c2ccc(cc2F)F)S(=O)(=O)c3ccccc3 6N-375S Cc1cccc(c1OC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccccc3)C 6N-376S c1ccc(cc1)S(=O)(=O)N(CC(=O)Oc2ccc3ccccc3c2)c4cccc(c4)C(F)(F)F 6N-377S Cc1cccc(c1OC(=O)CN(c2ccc(cc2F)F)S(=O)(=O)c3ccccc3)C 6N-378S c1ccc(cc1)S(=O)(=O)N(CC(=O)Oc2cccc3c2cccc3)c4ccc(cc4F)F 6N-379S CS(=O)(=O)N(CC(=O)Nc1ccc(cc1)Cl)c2ccc(cc2Cl)Cl 6N-383S Cc1cc(=O)n(c2c1cccc2)C(C)C 6N-389S Cc1cc(=O)n(c2c1cccc2)CC#C 6N-390S Cc1cccc2c1n(c(=O)cc2C)C 6N-391S Cc1cccc2c1n(c(=O)cc2C)Cc3ccccc3 6N-392S Cc1cccc2c1n(c(=O)cc2C)CC=C 6N-393S Cc1cccc2c1n(c(=O)cc2C)Cc3ccc(cc3)Cl 6N-394S Cc1cccc(c1)Cn2c(=O)cc(c3c2c(ccc3)C)C 6N-395S Cc1cccc2c1n(c(=O)cc2C)C(C)C 6N-396S CS(=O)(=O)N(CC(=O)Nc1ccc(c(c1)Cl)Cl)c2ccc(cc2Cl)Cl 6N-398S CS(=O)(=O)N(CC(=O)Nc1cccc(c1)C(F)(F)F)c2ccc(cc2Cl)Cl 6N-399S CN(c1ccccc1)C(=O)CN(c2ccc(cc2Cl)Cl)S(=O)(=O)C 6N-400S CS(=O)(=O)N(CC(=O)N1CCCCC1)c2ccc(cc2Cl)Cl 6N-401S CS(=O)(=O)N(CC(=O)N1CCOCC1)c2ccc(cc2Cl)Cl 6N-403S CS(=O)(=O)N(CC(=O)N1CCCC1)c2ccc(cc2Cl)Cl 6N-404S Cc1ccc(cc1)CSc2nc3c(c(n2)Oc4cc(cc(c4)C)C)CCCC3 6N-408S Cc1ccc(cc1)CSc2nc3c(c(n2)Oc4ccc(cc4F)F)CCCC3 6N-409S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccccc4)CCCC3 6N-410S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccc(cc4)Br)CCCC3 6N-411S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4cccc(c4)Cl)CCCC3 6N-413S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4cccc(c4)C)CCCC3 6N-414S Cc1ccc(cc1)CSc2nc3c(c(n2)SCC(=O)OC)CCCC3 6N-415S CSc1nc2ccsc2c(n1)O 6N-419S CSc1nc2ccsc2c(n1)Cl 6N-420S CSc1nc2ccsc2c(n1)NCC=C 6N-421S CSc1nc2ccsc2c(n1)N3CCCC3 6N-423S CNc1c2c(ccs2)nc(n1)SC 6N-424S COC(=O)c1ccccc1Sc2c3c(ccs3)nc(n2)SC 6N-425S CSc1nc2ccsc2c(n1)Sc3ccc(cc3Cl)Cl 6N-426S CSc1nc2ccsc2c(n1)N3CCOCC3 6N-427S CSc1nc2ccsc2c(n1)Sc3ccccc3 6N-428S CSc1nc2ccsc2c(n1)Sc3cccc(c3)C(F)(F)F 6N-429S CSc1nc2ccsc2c(n1)Sc3ccc(cc3)Br 6N-430S Cc1ccc(cc1)Sc2c3c(ccs3)nc(n2)SC 6N-431S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccccc4N)CCCC3 6N-432S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)C 6N-435S COc1cc(c(cc1Cl)Cl)N(CC(=O)Nc2ccc(cc2Cl)Cl)S(=O)(=O)C 6N-436S Cc1cc(ccc1NC(=O)CN(c2cc(c(cc2Cl)Cl)OC)S(=O)(=O)C)Cl 6N-437S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccccc4NC(=O)c5cccc(c5)C)CCCC3 6N-439S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccc(cc4Cl)Cl)CCCC3 6N-440S Cc1ccc(cc1)C(=O)n2c(cc(n2)COC(=O)c3ccc(cc3)F)C(F)(F)F 6N-441S COc1ccc(cc1)NC(=O)CN(c2cc(c(cc2Cl)Cl)OC)S(=O)(=O)C 6N-442S CN(c1ccccc1)C(=O)CN(c2cc(c(cc2Cl)Cl)OC)S(=O)(=O)C 6N-443S COc1cc(c(cc1Cl)Cl)N(CC(=O)N2CCOCC2)S(=O)(=O)C 6N-445S CCN(CC)C(=O)CN(c1cc(c(cc1Cl)Cl)OC)S(=O)(=O)C 6N-446S CO/N=C(/CN1CCN(CC1)c2ccccc2F)\c3ccc(cc3)F 6N-501S CO/N=C(/CN1CCN(CC1)C(c2ccccc2)c3ccccc3)\c4ccc(cc4)F 6N-502S CO/N=C(/CN1CCOCC1)\c2ccc(cc2)F 6N-503S CO/N=C(/CN1CCN(CC1)c2cccc(c2)Cl)\c3ccc(cc3)F 6N-504S Cc1ccc(cc1)N2C(C(C2=O)CN(C)C)c3ccccc3 6N-506S Cc1ccc(cc1)N2C(C(C2=O)CN3CCOCC3)c4ccccc4 6N-507S Cc1ccc(cc1)N2C(C(C2=O)CN3CCCC3)c4ccccc4 6N-508S Cc1ccc(cc1)N2C(C(C2=O)CN3CCCCC3)c4ccccc4 6N-509S COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCOCC2 6N-510S Cc1ccc(cc1)N2C(C(C2=O)CSc3ccc(cc3)Cl)c4ccccc4 6N-511S Cc1ccc(cc1)N2C(C(C2=O)CSc3ccc(cc3)Br)c4ccccc4 6N-512S COc1ccc(cc1)N2C(C(C2=O)CSc3ccccc3C(=O)OC)c4ccccc4 6N-513S Cc1ccc(cc1)N2C(C(C2=O)CSc3cccc(c3)OC)c4ccccc4 6N-514S CSc1nc2ccccc2c(n1)N3CCCC3 6N-515S COCCNc1c2ccccc2nc(n1)SC 6N-516S Cc1ccc(cc1)N2C(C(C2=O)CSc3cccc(c3)C(F)(F)F)c4ccccc4 6N-521S CO/N=C(/CNC(=O)c1ccc(cc1)F)\c2ccc(cc2)Cl 6N-523S CO/N=C(/CNC(=O)c1cccc(c1)Cl)\c2ccc(cc2)Cl 6N-525S CO/N=C(/CNC(=O)c1ccccc1Cl)\c2ccc(cc2)Cl 6N-526S CO/N=C(/CNC(=O)c1ccc(cc1Cl)Cl)\c2ccc(cc2)Cl 6N-527S CO/N=C(/CNC(=O)c1cccs1)\c2ccc(cc2)Cl 6N-528S COc1ccc(cc1)S(=O)(=O)NC/C(=N/OC)/c2ccc(cc2)Cl 6N-529S CN(C)S(=O)(=O)NC/C(=N/OC)/c1ccc(cc1)Cl 6N-530S CO/N=C(/CNS(=O)(=O)c1cccc(c1Cl)Cl)\c2ccc(cc2)Cl 6N-531S CO/N=C(/CNC(=O)C1CC1)\c2ccc(cc2)Cl 6N-533S CCOC(=O)c1cnc(nc1Cl)SC 6N-537S c1ccc(c(c1)C(=O)c2ccc(s2)Br)C(=O)O 6N-538S CCOC(=O)c1cnc(nc1Nc2ccc(cc2)Cl)SC 6N-539S Cc1c2c(nc(n1)N3CCOCC3)CCC2 6N-561S Cc1c2c(nc(n1)O)CCCC2 6N-562S Cc1c2c(nc(n1)N3CCCCC3)CCC2 6N-563S Cc1c2c(nc(n1)Sc3ccc(cc3)Cl)CCC2 6N-564S Cc1c2c(nc(n1)Oc3ccc(cc3)Cl)CCC2 6N-565S Cc1c2c(nc(n1)Sc3ccc(cc3)Br)CCC2 6N-566S Cc1c2c(nc(n1)N3CCN(CC3)Cc4ccccc4)CCC2 6N-567S Cc1c2c(nc(n1)N3CCCC3)CCC2 6N-571S Cc1c2c(nc(n1)Sc3ccccc3Cl)CCC2 6N-574S Cc1c2c(nc(n1)N3CC(OC(C3)C)C)CCC2 6N-575S Cc1c2c(nc(n1)N3CCN(CC3)C)CCC2 6N-576S CCCN(CCC)c1nc(c2c(n1)CCC2)C 6N-578S Cc1c2c(nc(n1)NC3CCCCC3)CCC2 6N-579S Cc1c2c(nc(n1)Sc3ccc(cc3)F)CCC2 6N-580S Cc1ccc(cc1)Sc2nc(c3c(n2)CCC3)C 6N-581S Cc1c2c(nc(n1)Sc3ccc(cc3Cl)Cl)CCC2 6N-583S Cc1c2c(nc(n1)S(=O)(=O)c3ccc(cc3)Br)CCC2 6N-584S Cc1c2c(nc(n1)S(=O)(=O)c3ccc(cc3)F)CCC2 6N-585S Cc1ccc(cc1)S(=O)(=O)c2nc(c3c(n2)CCC3)C 6N-586S Cc1c2c(nc(n1)S(=O)(=O)c3ccc(cc3Cl)Cl)CCC2 6N-587S c1ccc(c(c1)c2cc(no2)CO)Cl 6N-641S c1ccc(c(c1)c2cc(no2)COC(=O)c3ccc(cc3Cl)Cl)Cl 6N-642S c1ccc(cc1)c2cc(no2)CO 6N-643S Cc1ccc(cc1)NC(=O)OCc2cc(on2)c3ccccc3Cl 6N-644S c1ccc(c(c1)c2cc(no2)COC(=O)c3cccc(c3)C(F)(F)F)Cl 6N-645S c1ccc(c(c1)c2cc(no2)COC(=O)c3cccc(c3)Cl)Cl 6N-647S c1ccc(c(c1)c2cc(no2)COC(=O)Nc3cccc(c3)Cl)Cl 6N-648S c1ccc(c(c1)c2cc(no2)COC(=O)Nc3ccc(cc3)Cl)Cl 6N-649S c1ccc(cc1)NC(=O)OCc2cc(on2)c3ccccc3Cl 6N-650S c1ccc(c(c1)c2cc(no2)COC(=O)Nc3ccc(cc3Cl)Cl)Cl 6N-651S Cc1ccc(cc1)C(=O)OCc2cc(on2)c3ccccc3 6N-652S c1ccc(cc1)c2cc(no2)COC(=O)c3cccc(c3)Cl 6N-653S c1cc(ccc1C(=O)OCc2cc(on2)c3ccc(c(c3)Cl)Cl)F 6N-654S c1ccc(cc1)c2cc(no2)COC(=O)c3ccc(cc3Cl)Cl 6N-656S c1ccc(cc1)c2cc(no2)COC(=O)c3cccc(c3)C(F)(F)F 6N-657S c1ccc(cc1)c2cc(no2)COC(=O)c3ccc(c(c3)Cl)Cl 6N-658S c1ccc(cc1)c2cc(no2)COC(=O)Nc3ccc(cc3)Cl 6N-659S Cc1ccc(cc1)NC(=O)OCc2cc(on2)c3ccccc3 6N-660S Cc1ccc(cc1)NC(=O)OCc2cc(on2)c3ccc(c(c3)Cl)Cl 6N-661S c1cc(ccc1NC(=O)OCc2cc(on2)c3ccc(c(c3)Cl)Cl)Cl 6N-662S c1cc(c(cc1c2cc(no2)CN3CCCCC3)Cl)Cl 6N-663S c1cc(ccc1c2cc(no2)CCl)Cl 6N-665S c1cc(ccc1c2cc(no2)COC(=O)Nc3ccc(cc3)Cl)Cl 6N-668S c1ccc(cc1)NC(=O)OCc2cc(on2)c3ccc(cc3)Cl 6N-671S c1cc(ccc1c2cc(no2)CN3CCCCC3)Cl 6N-672S c1ccc(c(c1)N2CCN(CC2)Cc3cc(on3)c4ccc(cc4)Cl)F 6N-673S c1cc(ccc1c2cc(no2)CN3CCOCC3)Cl 6N-674S Cc1ccc(cc1)SCc2cc(on2)c3ccc(cc3)Cl 6N-675S c1cc(ccc1c2cc(no2)CSc3ccc(cc3)Cl)Cl 6N-676S c1cc(c(c(c1)Cl)/C=C/C(=N\Nc2ccc(cc2)F)/c3ccc(cc3)F)F 6N-700 Cc1ccc(cc1)C2CC(=NN2c3ccc(cc3)F)c4ccc(cc4)F 6N-701 c1ccc(cc1)C2CC(=NN2c3cccc(c3)[N+](=O)[O-])c4ccc(cc4)Cl 6N-702 c1cc(cc(c1)C(F)(F)F)C(=O)/C=C\c2ccc(cc2)Cl 6N-706 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)Cl)Cl 6N-707 CN1CC(C(C1)C(=O)c2cccc(c2)C(F)(F)F)c3ccc(cc3)Cl 6N-708 CN1CC(C(C1)C(=O)c2ccccc2)c3ccccc3 6N-710 c1ccc(cc1)NC(=S)NC(=N)N[N+](=O)[O-] 6N-711 CCNC(=S)NC(=N)N[N+](=O)[O-] 6N-712 c1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccccc4 6N-713 Cc1ccc(cc1)/C(=N\O)/CN2Cc3ccccc3CC2C(=O)NC(C)(C)C 6N-714 COc1ccc(cc1)c2cnc3nc(nn3c2N)SCCC(=C(F)F)F 6N-715 COc1cc(c(cc1OC)OC)C(=O)/C=C\c2ccc(cc2)Cl 6N-716 c1cc(sc1)C(=O)/C=C/c2ccc(cc2)Cl 6N-719 c1cc(ccc1c2cnc3nc(nn3c2N)SCCC(=C(F)F)F)F 6N-720 C=CCNC(=S)NC(=N)N[N+](=O)[O-] 6N-721 c1cc(ccc1NC(=S)NC(=N)N[N+](=O)[O-])Cl 6N-722 c1ccc(cc1)C(=O)/C=C/C(=O)c2ccccc2 6N-723 c1ccc2c(c1)ncc(n2)SCCC(=C(F)F)F 6N-725 CN1CC(C(C1)C(=O)c2ccccc2)C(=O)c3ccccc3 6N-726 CC(C)(C)NC(=S)NC(=N)N[N+](=O)[O-] 6N-728 CN1CC(C(C1)C(=O)c2ccccc2Cl)c3ccc(cc3)Cl 6N-730 CN1CC(C(C1)C(=O)c2cccs2)c3ccc(cc3)Cl 6N-731 Cc1cccc(c1)CSc2nccc(n2)c3cc(sc3Cl)Cl 6N-733 c1cnc(nc1)SCCC(=C(F)F)F 6N-735 C1CN=C([NH2+]1)SCCC(=C(F)F)F.[Br-] 6N-737 Cn1c(c2c(c1c3ccccc3)CN(C2)C)c4ccccc4 6N-738 COc1ccc(cc1)C(=O)C2CN(CC2c3ccc(cc3)Cl)c4ccccc4 6N-740 c1cc(sc1)/C=C\c2ccnc3n2nc(n3)SCCC(=C(F)F)F 6N-741 C=CCNc1nc(c(s1)C(=O)c2ccccc2)N 6N-742 c1ccc(cc1)C(=O)c2c(nc(s2)Nc3ccccc3)N 6N-743 c1cc2c(cc1Cl)nc(o2)SCCC(=C(F)F)F 6N-748 c1ccc(cc1)C(=O)C2CN(CC2c3ccc(cc3)Cl)c4ccccc4 6N-749 Cc1ccc(cc1)C2CN(CC2C(=O)c3ccc(cc3)F)c4ccccc4 6N-750 Cc1ccc(cc1)C(=O)C2CN(CC2C(=O)c3ccc(cc3)C)C 6N-752 COc1ccc(cc1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccc(cc4)C(F)(F)F 6N-756 c1ccc(cc1)C(=O)C2CN(CC2C(=O)c3ccccc3)c4ccccc4 6N-758 CC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 6N-760 c1ccc(c(c1)C(=O)O)SCCC(=C(F)F)F 6N-761 c1[nH]nc(n1)SCCC(=C(F)F)F 6N-762 Cc1ccc(cc1)S(=O)(=O)CCC(=C(F)F)F 6N-763 c1ccc(cc1)N2CC(C(C2)C(=O)c3ccc(cc3)Cl)c4ccccc4F 6N-764 c1ccc(cc1)N2CC(C(C2)C(=O)c3cccs3)c4ccc(cc4)Cl 6N-765 c1ccc(cc1)Cn2cnc(n2)SCCC(=C(F)F)F 6N-767 COc1cccc(c1)C(=O)C2CN(CC2c3ccc(cc3)Cl)c4ccccc4 6N-768 COc1ccc(cc1)NC(=O)c2ccccc2SCCC(=C(F)F)F 6N-769 Cc1ccc(cc1)C(=O)/C=C/C(=O)c2ccc(cc2)C 6N-770 CCOC(=O)C(n1cnc(n1)SCCC(=C(F)F)F)(F)F 6N-773 c1c(cnc(c1Cl)n2cnc(n2)SCCC(=C(F)F)F)C(F)(F)F 6N-776 c1cnc(nc1)n2cnc(n2)SCCC(=C(F)F)F 6N-777 COC(=O)c1ccsc1NC(=O)CBr 6N-801 COC(=O)c1ccsc1NC(=O)CC(C#N)C#N 6N-802 COc1ccc(cc1)OCC2CO2 6N-803 COC(=O)c1ccsc1n2cc(c(=O)n(c2=O)Cc3cccc(c3)C(F)(F)F)C#N 6N-804 COc1ccc(cc1)Cn2c(=O)c(cn(c2=O)c3c(ccs3)C(=O)OC)C#N 6N-805 COC(=O)c1ccsc1n2cc(c(=O)n(c2=O)Cc3ccccc3Cl)C#N 6N-806 COc1ccc(cc1)OCC2Cc3c(c(c(nc3O2)N)C#N)N 6N-808 Cc1cc(cc(c1)NC(=S)Nc2cc(c(cc2C#N)OC)OC)C 6N-809 COc1ccccc1NC(=S)Nc2cc(c(cc2C#N)OC)OC 6N-810 Cc1ccccc1OCC2Cc3c(c(c(nc3O2)N)C#N)N 6N-811 c1cc(ccc1/C=N/c2c(ccs2)C#N)[N+](=O)[O-] 6N-812 COc1cc(ccc1O)/C=N/c2c(ccs2)C#N 6N-813 COc1cc(c(cc1OC)NC(=S)Nc2ccc(cc2)F)C#N 6N-814 COCCNC(=S)Nc1cc(c(cc1C#N)OC)OC 6N-815 COc1cc(c(cc1OC)NC(=S)NC2CCCCC2)C#N 6N-816 COc1cc(c(cc1OC)NC(=S)NCc2cccc(c2)Cl)C#N 6N-817 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OC 6N-818 CN1CCN(CC1)c2ccc(cc2)NC(=S)Nc3cc(c(cc3C#N)OC)OC 6N-819 COc1cc(c(cc1OC)NC(=S)Nc2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl)C#N 6N-820 COc1ccc2ccccc2c1S(=O)Nc3ccc(cc3)Cl 6N-822 COc1ccc2ccccc2c1S(=O)Nc3ccccc3 6N-823 Cc1ccccc1OCC2Cc3c(c(c(nc3O2)n4cccc4)C#N)n5cccc5 6N-824 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4cccc(c4)Cl 6N-825 CCN(CC)S(=O)c1c2ccccc2ccc1OC 6N-826 COc1ccc2ccccc2c1S(=O)N 6N-827 CC(C)(C)C(C(=O)NC)n1cc(c(=O)[nH]c1=O)C#N 6N-900 Cc1cc2c(cco2)c(=O)n1N 6N-901 c1ccc(c(c1)c2c(cco2)C(=O)N3CCOCC3)O 6N-902 c1ccc(c(c1)c2c(cco2)C(=O)NN)O 6N-903 c1ccc(c(c1)c2c(cco2)C(=O)N/N=C/c3ccc(cc3)[N+](=O)[O-])O 6N-904 c1ccc(cc1)Oc2ccc(cc2)n3cnc(c3N)C#N 6P-002 CCOc1ccccc1n2cnc(c2N)C#N 6P-005 c1cc(ccc1CC#N)n2cnc(c2N)C#N 6P-006 CC(C)(C)OC(=O)n1cc(c2c1cccc2)CCC(=O)O 6P-010 COC(=O)c1c(ccs1)Nc2ccnc(c2)C(F)(F)F 6P-011 COc1ccc(cc1OC)N/C=N/C(=C(/C#N)\N)/C#N 6P-014 c1cc2c(cc1N/C=N/C(=C(/C#N)\N)/C#N)OCCO2 6P-015 COC(=O)c1ccc(cc1)N/C=N/C(=C(/C#N)\N)/C#N 6P-016 c1ccc(cc1)Oc2ccccc2N/C=N/C(=C(/C#N)\N)/C#N 6P-017 c1ccc(c(c1)/C(=N/O)/Nc2cccc(c2)Cl)Cl 6P-018 Cc1ccc2c(c1NC(=S)N)cccn2 6P-019 c1cc(ccc1COn2ccnc2C=O)F 6P-020 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3cn[nH]c3c2 6P-021 CCOc1ccccc1N/C=N/C(=C(/C#N)\N)/C#N 6P-025 c1cc(ccc1CC#N)N/C=N\C(=C(\C#N)/N)\C#N 6P-026 c1ccc(cc1)N/C(=N\O)/c2cccc(c2)[N+](=O)[O-] 6P-029 c1cc(ccc1COn2ccnc2C=O)C(F)(F)F 6P-030 c1cc2c(cc1n3cnc(c3N)C#N)OCCO2 6P-037 COc1ccc(cc1OC)n2cnc(c2N)C#N 6P-038 c1cc2cn[nH]c2cc1NC(=S)N 6P-044 CCOC(=O)C1C(C(C1N2CCCC2)(C)C)C(=O)OCC 6P-045 c1ccc(cc1)Oc2ccccc2n3cnc(c3N)C#N 6P-047 c1ccc(cc1)c2nnc(o2)S 6P-050 c1cc([n+](c(c1)Br)[O-])Br 6P-053 Cc1ccccc1COn2ccnc2C=O 6P-057 c1ccc(cc1)N2CCN(CC2)CC(C(F)(F)F)O 6P-058 COC(=O)C(CO)NC(=O)OCc1ccccc1 6P-062 COC(=O)C(COS(=O)(=O)C)NC(=O)OCc1ccccc1 6P-069 COc1ccccc1CNc2c3cc(c(cc3ncn2)OC)OC 6P-071 c1cc(ccc1C(=O)O)Oc2ccc(c(c2)F)Cl 6P-077 Cc1ccc(cc1NC(=S)NC(=O)c2ccccc2)C(F)(F)F 6P-079 COC(=O)C1CC(CN1CC(C(F)(F)F)O)O 6P-082 Cc1ccc(cc1NC(=S)N)C(F)(F)F 6P-083 c1cc(cc(c1)[N+](=O)[O-])/C(=N/O)/Nc2cccc(c2)Cl 6P-084 c1ccc(c(c1)C#N)Nc2ccnc(c2)C(F)(F)F 6P-085 c1ccnc(c1)NC(=O)c2c(nc3ccccn3c2=O)O 6P-087 Cc1c(c(n(n1)CCCF)C)[N+](=O)[O-] 6P-092 c1ccc2c(c1)CCN2CC(C(F)(F)F)O 6P-094 Cc1c(c(=O)n2c(n1)CCCC2)CCN3CCC(CC3)C(=O)c4ccc(cc4O)F 6P-096 C1CCCN(CC1)CC(C(F)(F)F)O 6P-097 c1ccc(cc1)N/C(=N\O)/c2cccc(c2)Cl 6P-098 c1cc(cc(c1)OCc2cccnc2)C(=O)O.Cl 6P-101 c1cc(cc(c1)[N+](=O)[O-])/C(=N/O)/Nc2ccc(cc2)Cl 6P-104 CN(c1ccnc(c1)C(F)(F)F)c2ccccc2C(=O)OC 6P-106 c1ccc2c(c1)n3c(=O)c(c(nc3s2)O)C(=O)Nc4ccc(cc4)Cl 6P-107 c1ccc(c(c1)N/C(=N\O)/c2cccc(c2)[N+](=O)[O-])Cl 6P-109 C1C(OC(S1)C(=O)O)O 6P-110 c1cc(cc(c1)Cl)/C(=N/O)/Nc2ccc(cc2)Cl 6P-111 c1ccc(cc1)C2NC(CS2)C(=O)O 6P-115 c1ccc2c(c1)CCCN2/C(=N\O)/c3cccc(c3)[N+](=O)[O-] 6P-116 C[Si](C)(C)OC(CN1CCc2ccccc2C1)C(F)(F)F 6P-118 c1ccc2c(c1)nc(s2)NC(=O)c3c(nc4n(c3=O)c5ccccc5s4)O 6P-120 c1cc(sc1)C2NC(CS2)C(=O)O 6P-124 c1cc(ccc1Cn2c(ccc(c2=O)C(=O)N3CCOCC3)C(F)(F)F)Cl 6P-301S c1ccc(cc1)CNC(=O)c2ccc(n(c2=O)Cc3ccc(cc3)Cl)C(F)(F)F 6P-302S c1cc(ccc1Cn2c(ccc(c2=O)C(=O)N3CCCC3)C(F)(F)F)Cl 6P-303S c1ccn(c1)c2ccsc2C(=O)NNC(=O)c3cccs3 6P-311S COc1ccccc1C(=O)NNC(=O)c2c(ccs2)n3cccc3 6P-312S c1ccn(c1)c2ccsc2C(=O)NNC(=O)c3cccc(c3Cl)Cl 6P-313S c1ccc(c(c1)C(=O)NNC(=O)c2c(ccs2)n3cccc3)C(F)(F)F 6P-314S c1ccc2c(c1)nc(s2)N3CCN(CC3)Cc4ccc(cc4)Cl 6P-315S Cc1c2c(ncnc2on1)N(C)Cc3ccccc3 6P-316S Cc1c2c(ncnc2on1)N3CCOCC3 6P-317S Cc1c2c(ncnc2on1)N3CCCCC3 6P-318S CCCNc1c2c(noc2ncn1)C 6P-319S Cc1c2c(ncnc2on1)N3CCN(CC3)c4ccc(cc4)F 6P-321S c1ccn(c1)c2ccsc2C(=O)NNC(=O)c3c(cccc3F)F 6P-322S c1ccn(c1)c2ccsc2C(=O)NNC(=O)c3cccc(c3)C(F)(F)F 6P-323S CCCC(=O)NNC(=O)c1c(ccs1)n2cccc2 6P-324S c1ccc(cc1)/C=N\NC(=O)c2c(ccs2)n3cccc3 6P-325S c1ccc(cc1)n2c(nnc2S)c3c(ccs3)n4cccc4 6P-326S Cc1c(sc2n1c3ccccc3n2)/C(=N/O)/C 6P-327S CS(=O)(=O)NNC(=O)c1c(ccs1)n2cccc2 6P-328S CC(C)(C)C(=O)NNC(=O)c1c(ccs1)n2cccc2 6P-329S Cc1ccc(cc1)NC(=O)NNC(=O)c2c(ccs2)n3cccc3 6P-330S c1ccn(c1)c2ccsc2C(=O)N/N=C\c3ccc(cc3)Cl 6P-331S Cc1c2c(ncnc2on1)N3CCN(CC3)C 6P-332S Cc1c2c(ncnc2on1)N3CCN(CC3)c4cccc(c4)Cl 6P-333S c1ccn(c1)c2ccsc2C(=O)NNC(=O)Nc3ccc(cc3)Cl 6P-336S c1ccn(c1)c2ccsc2C(=O)NNC(=O)Nc3cccc(c3)Cl 6P-337S Cc1cccc(c1)NC(=O)NNC(=O)c2c(ccs2)n3cccc3 6P-338S Cc1ccc(cc1)CO/N=C(\C)/c2c(n3c4ccccc4nc3s2)C 6P-339S Cc1cccc(c1NC(=O)NNC(=O)c2c(ccs2)n3cccc3)C 6P-344S c1ccn(c1)c2ccsc2C(=O)NNC(=O)Nc3cccc(c3)C(F)(F)F 6P-345S c1ccn(c1)c2ccsc2C(=O)NNC(=O)Nc3ccc(cc3)F 6P-346S c1ccc(cc1)C(=O)NNC(=O)c2ccccc2n3cccc3 6P-349S c1ccc(c(c1)C(=O)NNC(=O)c2cccc(c2)Cl)n3cccc3 6P-350S Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2ccccc2n3cccc3 6P-351S COc1cccc(c1C(=O)NNC(=O)c2ccccc2n3cccc3)OC 6P-352S c1ccc(c(c1)C(=O)NNC(=O)c2c(cccc2F)F)n3cccc3 6P-353S Cc1ccc(cc1)C(=O)NNC(=O)c2ccccc2n3cccc3 6P-354S c1ccc(c(c1)C(=O)NNC(=O)c2cccs2)n3cccc3 6P-355S c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2Cl)Cl)n3cccc3 6P-356S c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)Cl)n3cccc3 6P-357S c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)F)n3cccc3 6P-358S c1ccc(c(c1)C(=O)NNC(=O)c2cccc(c2)C(F)(F)F)n3cccc3 6P-359S COc1cccc(c1)C(=O)NNC(=O)c2ccccc2n3cccc3 6P-360S Cc1cccc(c1)C(=O)NNC(=O)c2ccccc2n3cccc3 6P-361S c1ccc(c(c1)C(=O)NNC(=O)c2ccc(c(c2)Cl)Cl)n3cccc3 6P-362S CCC(=O)NNC(=O)c1ccccc1n2cccc2 6P-363S Cc1c(sc2n1ncn2)/C(=N/OC)/CSc3ccccc3OC 6P-367S Cc1ccc(cc1)SC/C(=N\OC)/c2c(n3c(s2)ncn3)C 6P-368S Cc1c(sc2n1ncn2)/C(=N/OC)/CSc3c(cccc3Cl)Cl 6P-372S Cc1c(sc2n1ncn2)/C(=N/OC)/CSc3ccccc3Cl 6P-374S Cc1c(sc2n1ncn2)/C(=N/OC)/CSc3cccc(c3)OC 6P-375S Cc1c(sc2n1ncn2)/C(=N/OCc3ccc(cc3Cl)F)/CSc4ccc(cc4)Cl 6P-381S Cc1c(sc2n1c3ccccc3n2)/C(=N/OC)/C 6P-394S CCO/N=C(\C)/c1c(n2c3ccccc3nc2s1)C 6P-395S Cc1c(sc2n1c3ccccc3n2)/C(=N/OCc4cccc(c4)C(F)(F)F)/C 6P-396S Cc1c(sc2n1c3ccccc3n2)/C(=N/OCc4ccc(cc4)Cl)/C 6P-397S Cc1c(sc2n1c3ccccc3n2)/C(=N/OCc4ccccc4)/C 6P-398S Cc1c(sc2n1c3ccccc3n2)/C(=N/OCc4ccc(c(c4)Cl)Cl)/C 6P-400S c1ccc(c(c1)C(=O)NNS(=O)(=O)c2ccc(cc2)Br)n3cccc3 6P-401S COc1ccc(cc1)S(=O)(=O)NNC(=O)c2ccccc2n3cccc3 6P-402S c1ccc(c(c1)C(=O)NNS(=O)(=O)c2cc(cc(c2)Cl)Cl)n3cccc3 6P-403S c1ccc(c(c1)C(=O)NNS(=O)(=O)c2ccc(cc2)C(F)(F)F)n3cccc3 6P-404S c1ccc(c(c1)C(=O)NNS(=O)(=O)c2ccccc2F)n3cccc3 6P-405S COC(=O)c1ccccc1S(=O)(=O)NNC(=O)c2ccccc2n3cccc3 6P-406S c1ccc(cc1)S(=O)(=O)NNC(=O)c2ccccc2n3cccc3 6P-407S CS(=O)(=O)NNC(=O)c1ccccc1n2cccc2 6P-408S c1ccc(cc1)/C=N\NC(=O)c2ccccc2n3cccc3 6P-411S c1ccn(c1)c2ccsc2C(=O)N/N=C\c3ccco3 6P-413S c1ccn(c1)c2ccsc2C(=O)N/N=C\c3cccs3 6P-414S Cc1cccc(c1)/C=N\NC(=O)c2c(ccs2)n3cccc3 6P-415S c1ccn(c1)c2ccsc2C(=O)N/N=C\c3ccc(cc3Cl)Cl 6P-416S c1ccc(c(c1)C(=O)N/N=C\c2ccc(cc2Cl)Cl)n3cccc3 6P-419S c1ccc(c(c1)C(=O)N/N=C\c2ccc(cc2Cl)F)n3cccc3 6P-420S COc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccc(cc3)Cl 6P-502S COc1ccccc1NC(=O)c2c(=O)ccn(n2)c3cccc(c3)C(F)(F)F 6P-505S COc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccccc3 6P-506S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SC 6P-511S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SCC(=O)OC 6P-515S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SCc3ccc(cc3)Cl 6P-516S COc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccc(cc3)OC(F)(F)F 6P-518S COc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccc(c(c3)F)F 6P-519S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SCC(=O)c3ccc(cc3)Cl 6P-523S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SCC=C 6P-526S Cc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccc(cc3)Cl 6P-527S Cc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccccc3 6P-528S Cc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccc(c(c3)F)F 6P-532S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SCc3ccccc3 6P-533S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SCc3ccc(c(c3)Cl)Cl 6P-534S Cc1ccccc1NC(=O)c2c(=O)ccn(n2)c3cccc(c3)C(F)(F)F 6P-535S Cc1ccccc1NC(=O)c2c(=O)ccn(n2)c3ccc(cc3)C(=O)OC 6P-536S c1ccc(cc1)NC(=O)c2c(=O)ccn(n2)c3ccccc3 6P-538S c1ccc(cc1)NC(=O)c2c(=O)ccn(n2)c3cccc(c3)C(F)(F)F 6P-540S c1ccc(cc1)NC(=O)c2c(=O)ccn(n2)c3cccc(c3)Cl 6P-542S CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2nnc(s2)SCc3ccc(cc3)OC 6P-543S c1ccc(cc1)NC(=O)c2c(=O)ccn(n2)c3ccc(cc3)Cl 6P-545S c1ccc(cc1)c2cc3c(o2)ncnc3Oc4ccc(cc4Cl)F 6P-561S CC(C)(C)c1ccc(cc1)Oc2c3cc(oc3ncn2)c4ccccc4 6P-562S COc1ccccc1Oc2c3cc(oc3ncn2)c4ccccc4 6P-563S CN1CCN(CC1)c2c3cc(oc3ncn2)c4ccccc4 6P-568S Cc1c(snn1)SCCNC(=O)c2ccc(cc2)F 6P-574S Cc1c(snn1)SCCNC(=O)c2c(cccc2F)F 6P-575S Cc1c(snn1)SCCNC(=O)c2cccc(c2Cl)Cl 6P-576S Cc1ccc(cc1)C(=O)NCCSc2c(nns2)C 6P-577S COc1cccc(c1)c2nc(no2)c3cc(oc3n4cccc4)c5ccccc5 6P-578S Cc1c(snn1)SCCNC(=O)C(C)(C)C 6P-581S Cc1c(snn1)SCCNS(=O)(=O)c2ccc(cc2)Cl 6P-582S Cc1cccc(c1)C(=O)Nc2c(c3c(o2)cccn3)C#N 6P-586S c1cc(c(c(c1)F)C(=O)Nc2c(c3c(o2)cccn3)C#N)F 6P-590S Cc1ccc(cc1)n2ccc(=O)c(n2)C(=O)OC 6P-650S COC(=O)c1c(=O)ccn(n1)c2ccccc2 6P-651S Cc1ccc(cc1)n2ccc(=O)c(n2)C(=O)NC 6P-654S CNC(=O)c1c(=O)ccn(n1)c2ccccc2 6P-655S c1ccc(cc1)n2ccc(=O)c(n2)C(=O)O 6P-658S Cc1ccc(cc1)n2ccc(=O)c(n2)C(=O)O 6P-659S CCn1c(nnc1S)c2c(=O)ccn(n2)c3ccccc3 6P-660S CCn1c(nnc1S)c2c(=O)ccn(n2)c3ccc(cc3)C 6P-661S CCn1c(nnc1SCc2ccc(cc2)C)c3c(=O)ccn(n3)c4ccccc4 6P-665S CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3c(=O)ccn(n3)c4ccccc4 6P-666S CCn1c(nnc1SCc2ccc(cc2)F)c3c(=O)ccn(n3)c4ccccc4 6P-667S CCn1c(nnc1SCc2c(cccc2Cl)Cl)c3c(=O)ccn(n3)c4ccccc4 6P-669S CCn1c(nnc1SCc2ccc(cc2)Cl)c3c(=O)ccn(n3)c4ccccc4 6P-670S CCn1c(nnc1SC)c2c(=O)ccn(n2)c3ccccc3 6P-671S COC(=O)c1c(=O)ccn(n1)c2cccc(c2)C(F)(F)F 6P-673S COC(=O)c1c(=O)ccn(n1)c2cccc(c2)Cl 6P-674S c1cc(cc(c1)Cl)n2ccc(=O)c(n2)C(=O)O 6P-675S c1cc(cc(c1)n2ccc(=O)c(n2)C(=O)O)C(F)(F)F 6P-676S c1cc2c(cc1CNC(=O)Cc3c(cc(cn3)C(F)(F)F)Cl)OCO2 6P-702 c1cc(ccc1CNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cl 6P-703 c1cc(ccc1CCNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N 6P-704 c1cc(c(cc1Br)[N+](=O)[O-])Cl 6P-705 Cc1cccc(n1)n2cc(nc2)C(=O)NN 6P-707 CCOC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NCc2ccc(cc2)C 6P-708 CCOC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NCc2cccc(c2)OC 6P-709 CCOC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NCc2ccc(cc2)F 6P-710 Cc1ccc(cc1)CNC(=O)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCc3ccc(cc3)C 6P-711 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)n3ccc(c(c3=O)Cc4ccc(cc4Cl)Cl)O 6P-713 c1cc(cc(c1)C(F)(F)F)CNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 6P-714 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)(C#N)C#N 6P-715 C1C(CN(N1C=O)C=O)Br 6P-718 c1cc(ccc1CNC(=O)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCc3ccc(cc3)F)F 6P-719 Cc1c(no[n+]1[O-])/C=N/O 6P-721 c1cc(cnc1)CNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 6P-722 CN1C(=O)N(C(O1)CC(=O)NC2CCCC2)c3ccc(cc3)Cl 6P-724 CC(C)N(C(C)C)C(=O)CC1N(C(=O)N(O1)C)c2ccc(cc2)Cl 6P-725 c1cc2c(cc1I)NC(=O)C2=O 6P-727 COc1cc(ccc1C=O)OCC(=O)O 6P-728 c1ccc2c(c1)cccc2NCCn3ccc(c(c3=O)Cc4ccc(cc4Cl)Cl)O 6P-733 Cc1c(sc(n1)c2ccccc2)C(=O)C 6P-734 c1c(cnc(c1Cl)C(C(=O)NCCCN2CCOCC2)C(=O)NCCCN3CCOCC3)C(F)(F)F 6P-736 c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)CCCN3CCOCC3)O 6P-738 c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)CC(=O)N)O 6P-740 Cc1c(sc([nH+]1)c2ccccc2)C(=O)C.[Cl-] 6P-741 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)C 6P-742 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)C(F)(F)F)C 6R-0001 CCC(=O)NNc1cccc(n1)Cl 6R-0005 CC(C)(C)C(=O)NNc1cccc(n1)Cl 6R-0006 CC(C(=O)NNc1cccc(n1)Cl)Cl 6R-0007 COc1ccc(cc1)CN2C(C(CCC2=O)C(=O)O)c3ccccc3 6R-0008 CCc1nnc2n1c(ccc2)Cl 6R-0009 CC(C)(C)c1nnc2n1c(ccc2)Cl 6R-0010 c1cc2c(c(c1)C=O)NCC2 6R-0011 CN(C)CCC(c1cc(sc1Cl)Cl)O 6R-0012 c1cc(ccc1NC(=S)Nn2cnnc2)Cl 6R-0014 CC(C(CCN(C)C)O)Oc1ccc(cc1)F 6R-0015 c1ccc(cc1)NC(=S)Nn2cnnc2 6R-0017 c1ccc(cc1)COc2cc(on2)/C=C/C(=O)O 6R-0022 c1cc(cc(c1)Cl)NC(=O)Nn2cnnc2 6R-0023 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)C)Cl)C)C 6R-0024 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)c5ccccc5)C)C 6R-0025 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)C)Cc5cccc(c5)F)C)C 6R-0026 COC(=O)c1ccccc1NC(=S)NC(=O)c2ccccc2 6R-0027 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(c(s2)C(=O)C)C 6R-0029 CN(C)CCC(c1cccnc1)O 6R-0030 CCOC(=O)NC(c1ccccc1F)C2CCCCCC2=O 6R-0031 CCOC(=O)C1CCCC(C1=O)C(c2ccccc2F)NC(=O)OCC 6R-0032 c1cc(c(cc1)F)/C=C\2/C(=O)/C(=C/c3c(cccc3)F)/CC2 6R-0034 c1c(ccc(c1)F)/C=C\2/C(=O)/C(=C/c3ccc(cc3)F)/CCC2 6R-0035 CCOC(=O)NC(c1ccccc1F)C2CCCCCCC2=O 6R-0036 c1cc(ccc1N\2C(=O)CS/C2=N/n3cnnc3)Cl 6R-0037 c1ccc(cc1)N\2C(=O)C(S/C2=N\n3cnnc3)CC(=O)O 6R-0038 CC(C)(C)OC(=O)N1CCc2c1c(ccc2)C=O 6R-0040 c1cc(c(c(c1)I)[N+](=O)[O-])Cl 6R-0041 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)O)Cc5ccc(cc5Cl)Cl)C)C 6R-0042 CN(C)/C=C/C(=O)c1ccc(c(c1)OC)OC 6R-0043 CC(C)(C)c1ccc(cc1O)CCC(=O)OC 6R-0044 CCOC(=O)c1cnn(c1N)C(=O)c2ccc(cc2Cl)Cl 6R-0045 c1cc(c(cc1Cl)Cl)C(=O)n2c(c(cn2)C#N)N 6R-0046 c1ccc(cc1)NC(=O)Nn2cnnc2 6R-0047 CC/C(=N\NC(=O)/C(=C/N(C)C)/C#N)/CC(=O)C(F)(F)F 6R-0048 COc1ccc(cc1)C(=O)/C=C/N2CCN(CC2)C(c3ccccc3)c4ccccc4 6R-0049 CCOC(=O)c1cn(nc1C)C(=O)/C(=C/N(C)C)/C#N 6R-0050 c1ccc2c(c1)CCN(C2)/C=C/C(=O)c3ccccn3 6R-0051 CCOC(=O)C(=Nc1cc(n[nH]1)C)C(=O)OCC 6R-0052 CC(=O)c1ccn(c1)S(=O)(=O)c2ccccc2 6R-0053 c1cc2nnc(n2c(c1)Cl)c3ccc(cc3)Cl 6R-0054 c1ccc(cc1)C2C(CC(=O)N2C3CCCCC3)C(=O)O 6R-0055 c1cc(nc(c1)Cl)NNC(=O)c2ccc(cc2)Cl 6R-0056 c1cc(nc(c1)Cl)NNC(=O)CCl 6R-0057 CC(C)(C)OC(=O)N1CCc2c1c(ccc2)/C=C\C(=O)O 6R-0058 c1ccc(cc1)N\2C(=O)CS/C2=N\n3cnnc3 6R-0061 c1ccc2c(c1)CCN(C2)CCC(c3ccccn3)O 6R-0062 CCCc1c(nc2cc(nn2c1C)c3c(ccs3)n4c(ccc4C)C)C 6R-0063 CCOC(=O)NC(c1ccccc1F)C2CCc3ccccc3C2=O 6R-0064 CCOC(=O)NC(c1cccc(c1)Cl)C2CCCCC2=O 6R-0065 c1c(sc(n1)Cl)C(=O)O 6R-0067 COc1c(nnc(n1)c2ccccc2)C(=O)O 6R-0068 c1cc(c(c(c1)I)N)Cl 6R-0069 CCc1nnc2n1c(ccc2)OCC 6R-0071 CCOC(=O)NC(c1cccc(c1)Cl)C2CCCCCC2=O 6R-0072 CCOC(=O)NC(c1cccc(c1)Cl)C2CCCCCCC2=O 6R-0073 c1cc2nnc(n2c(c1)Cl)CCl 6R-0074 C/C(=N\NC(=O)/C(=C/N(C)C)/C#N)/CC(=O)C(F)(F)F 6R-0075 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3cccc(c3)Cl 6R-0076 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)COC)C 6R-0077 Cc1cc2nc(c(c(n2n1)C)Cl)C 6R-0078 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccccc3Cl 6R-0079 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc3ccccc3n2)C(=O)OC 6R-0080 Cc1cc2nc(cc(n2n1)O)COC 6R-0082 c1cc(ccc1C2CC(=CC(=O)C2)N)Cl 6R-0084 CC(C)(C)OC(=O)N1CCc2c1c(ccc2)/C=C\C(=O)N3CCN(CC3)c4ccc(cc4)F 6R-0086 CN(C)/C=C/C(=O)c1ccc(o1)c2ccc(cc2Cl)Cl 6R-0087 c1ccc(cc1)C2C(CCC(=O)N2C3CCCCC3)C(=O)NCc4ccc(cc4)Cl 6R-0088 COCCNC(=O)C1CCC(=O)N(C1c2ccccc2)C3CCCCC3 6R-0089 CN(C)/C=C/C(=O)c1ccn(c1)S(=O)(=O)c2ccccc2 6R-0090 CCOC(=O)NC(c1cccc(c1)Cl)C2COc3ccccc3C2=O 6R-0092 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc(cc5)F)C 6R-0093 CN(C)/C=C\1/C(=O)N(/C(=N/n2cnnc2)/S1)c3ccccc3 6R-0094 c1cc(nc(c1)Cl)NNC(=O)C2CC2 6R-0095 c1cc(nc(c1)Cl)NNC(=O)c2cccs2 6R-0096 CC(=O)NNc1cccc(n1)Cl 6R-0097 CCOc1ccc(cc1)C2C(CCC(=O)N2C3CCCCC3)C(=O)O 6R-0098 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc(cc5Cl)Cl)C 6R-0099 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccccc3Cl)Br 6R-0100 COc1ccccc1/C=C(/c2ccccc2)\C(=O)N3CCN(CC3)c4ccccc4 6R-0200 COc1ccc(cc1)CNC(=O)/C(=C\c2ccccc2OC)/c3ccccc3 6R-0201 Cc1ccc(cc1)CNC(=O)/C(=C\c2ccccc2OC)/c3ccccc3 6R-0202 CN(CCOc1ccc(cc1)c2ccn(n2)C(=O)c3ccc(cc3)F)c4ccccn4 6R-0203 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5cc(cc(c5)C(F)(F)F)C(F)(F)F 6R-0205 COc1ccccc1/C=C(/c2ccccc2)\C(=O)N3CCN(CC3)c4ccccc4F 6R-0206 COc1ccccc1/C=C(/c2ccccc2)\C(=O)N3CCN(CC3)Cc4ccccc4 6R-0207 c1ccc(cc1)CN2CCC(CC2)C(=O)NNC(=N)CC#N 6R-0208 COc1ccccc1/C=C(\c2ccccc2)/C(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 6R-0209 COc1ccccc1/C=C(\c2ccccc2)/C(=O)NCCCn3ccnc3 6R-0212 c1ccc(cc1)Cc2c(nc3ccccc3n2)NNC(=N)CC#N 6R-0213 COc1ccccc1/C=C(\c2ccccc2)/C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 6R-0214 COC(=O)/C=C/COc1ccccc1[N+](=O)[O-] 6R-0216 COc1ccccc1/C=C(\c2ccccc2)/C(=O)OC 6R-0218 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NNC(=O)c4ccc(cc4)Cl 6R-0219 Cc1ccc(cc1)C(=O)NNC(=O)C2Cc3c4ccccc4ccc3O2 6R-0220 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5ccc(cc5Cl)Cl 6R-0222 Cc1cccc(c1)CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)Cc5ccccc5)OC)OC 6R-0223 CN(C)/C=N/NC(=O)C1Cc2c3ccccc3ccc2O1 6R-0224 Cc1ccc(cc1)S(=O)(=O)NNC(=O)C2Cc3c4ccccc4ccc3O2 6R-0225 COc1ccccc1/C=C(\c2ccccc2)/C(=O)NCCc3ccccc3 6R-0226 c1cc(c(nc1)SCC(=O)O)C(=O)O 6R-0228 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCc5cccc(c5)Cl 6R-0231 COc1ccc(cc1)S(=O)(=O)NNC(=O)C2Cc3c4ccccc4ccc3O2 6R-0232 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NNS(=O)(=O)c4ccc(cc4F)F 6R-0233 CS(=O)(=O)NNC(=O)C1Cc2c3ccccc3ccc2O1 6R-0234 COc1cc2c(cc1OC)NC(=S)N3C2=NC(=O)C3CC4CCCCC4 6R-0236 CCCCOc1ccc(cc1)S(=O)(=O)NNC(=O)C2Cc3c4ccccc4ccc3O2 6R-0238 c1ccc(cc1)Cc2c(nc3ccccc3n2)N/N=C/c4ccc(cc4)F 6R-0240 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5c(cccc5Cl)F 6R-0241 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccccc5Cl 6R-0242 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccccc5 6R-0243 Cc1ccc(cc1)CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)CC5CCCCC5)OC)OC 6R-0244 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccc(cc5)Cl 6R-0245 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccc(cc5)C(F)(F)F 6R-0246 Cc1c(cccc1Cl)NC(=O)c2ccccc2 6R-0247 Cc1cc(ccc1NC(=O)c2ccccc2)Cl 6R-0248 CC(C)(CO)C(C(=O)N)O 6R-0249 CCOC(=O)/C=C/COc1ccc(cc1C=O)Br 6R-0252 c1cc(c(nc1)N2CCN(CC2)c3c(cccn3)[N+](=O)[O-])[N+](=O)[O-] 6R-0253 CN(CCOc1ccc(cc1)c2ccn(n2)S(=O)(=O)c3ccc(cc3)OC)c4ccccn4 6R-0254 CN(CCOc1ccc(cc1)c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl)c4ccccn4 6R-0255 CCOC(=O)/C=C/COc1c(cc(cc1OC)Br)C=O 6R-0256 CCOC(=O)/C=C/COc1c(cc(cc1Br)Br)C=O 6R-0257 COCCN1C(=O)/C(=C/c2ccc(cc2)Br)/C(=O)NC1=O 6R-0258 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCC(=O)OC 6R-0260 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNC(=O)C3CCN(CC3)Cc4ccccc4 6R-0261 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=O)C3CCN(CC3)Cc4ccccc4 6R-0262 COc1ccccc1/C(=C\c2ccccc2)/C(=O)O 6R-0263 c1ccc(cc1)c2cc3cc(ccc3[nH]2)Cl 6R-0264 c1ccc(cc1)CN2CCC(CC2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl 6R-0266 Cc1c(cccc1Cl)NC(=O)c2ccc(cc2)F 6R-0267 CN(CCOc1ccc(cc1)c2ccn(n2)C(=O)c3cccs3)c4ccccn4 6R-0268 CN(CCOc1ccc(cc1)c2ccn(n2)C(=O)c3cccc(c3)C(F)(F)F)c4ccccn4 6R-0269 Cc1cc(ccc1NC(=O)c2ccc(cc2)F)OC 6R-0270 Cc1cc(ccc1NC(=O)c2ccccc2)OC 6R-0271 COCCN1C(=O)/C(=C/c2cc3c(cc2Br)OCO3)/C(=O)NC1=O 6R-0272 CC1(OC(=O)C(C(=O)O1)CN(C)C)C 6R-0273 c1ccc(cc1)CN2CCC(CC2)C(=O)NNS(=O)(=O)c3ccc4ccccc4c3 6R-0275 Cc1cc(c(c(c1)C)S(=O)(=O)NNC(=O)C2CCN(CC2)Cc3ccccc3)C 6R-0276 CC(C(=O)OC)SC1=Nc2cc(c(cc2C3=NC(=O)C(N31)CC4CCCCC4)OC)OC 6R-0278 CN(CCOc1ccc(cc1)c2ccn(n2)C(=O)c3ccc(cc3)C(F)(F)F)c4ccccn4 6R-0280 Cc1ccc(cc1)NC(=O)NNC(=O)C2CC(=NO2)c3cccnc3 6R-0282 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5cccc(c5)Cl 6R-0283 Cc1cccc(c1)CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)CC5CCCCC5)OC)OC 6R-0284 Cc1ccccc1CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)CC5CCCCC5)OC)OC 6R-0285 c1ccc(cc1)CN2CCC(CC2)C(=O)NNC(=O)c3cccs3 6R-0287 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SC/C=C/c5ccccc5 6R-0289 CN(CCOc1ccc(cc1)c2ccn(n2)S(=O)(=O)c3cccc4c3cccc4)c5ccccn5 6R-0291 CC1=C(C(CC(=O)N1)c2ccc(cc2)Br)C(=O)C 6R-0295 c1ccc(cc1)CN2CCC(CC2)C(=O)NNC(=O)C3CC3 6R-0297 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)O 6R-0298 COc1ccc2c(c1)cc([nH]2)c3ccccc3 6R-0301 Cc1cc(c(c(c1)C)S(=O)(=O)n2ccc(n2)c3ccc(cc3)OCCN(C)c4ccccn4)C 6R-0302 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)C(Cl)(Cl)Cl 6R-0303 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)NCC(OC)OC 6R-0304 Cc1c(cccc1Cl)NC(=O)c2cccc(c2)C(F)(F)F 6R-0307 Cc1cc(ccc1NC(=O)c2ccccc2)Br 6R-0308 Cc1ccc(cc1NC(=O)c2ccccc2)F 6R-0309 Cc1cc(ccc1NC(=O)c2ccccc2)F 6R-0310 CN(CCOc1ccc(cc1)c2ccn(n2)S(=O)(=O)c3c(cccc3Cl)Cl)c4ccccn4 6R-0311 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)NCC4CCCO4 6R-0313 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)NCCCOC 6R-0314 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)NCCc4ccccn4 6R-0315 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)NC4CC4 6R-0316 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)NCc4ccco4 6R-0317 c1cc(ccc1CNC(=O)/C=C/c2cc3c(cc2Br)OCO3)F 6R-0318 CCC(C)NC(=O)/C=C/c1cc2c(cc1Br)OCO2 6R-0319 c1cc(sc1)CNC(=O)/C=C/c2cc3c(cc2Br)OCO3 6R-0320 COc1ccc(cc1)CNC(=O)/C=C/c2cc3c(cc2Br)OCO3 6R-0321 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5cccc(c5)F 6R-0322 COc1ccc(cc1)CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)CC5CCCCC5)OC)OC 6R-0323 COc1cccc(c1)CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)CC5CCCCC5)OC)OC 6R-0324 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccccc5C(F)(F)F 6R-0325 Cc1ccc(c(c1)CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)CC5CCCCC5)OC)OC)C 6R-0326 CCOC(=O)c1c2ccccn2cc1c3cccc(c3)N 6R-0327 c1ccc(cc1)COc2ccc(cc2)/C=C(\c3ccccc3)/C(=O)O 6R-0329 CCc1cc(=O)[nH]c(n1)SCCC(=C(F)F)F 6R-0332 CCc1cc(=O)[nH]c(n1)SCc2cc(cc(c2)C(F)(F)F)C(F)(F)F 6R-0333 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3cc([nH]c3)C(=O)NCCCN4CCOCC4 6R-0334 CCC(C)(C)NC(=O)c1cc(c[nH]1)C(=O)c2c(onc2c3c(cccc3Cl)Cl)C 6R-0335 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NCc4ccc(cc4)Cl 6R-0338 c1ccc(cc1)Oc2c(nc3cc(c(cc3n2)Cl)Cl)C(F)(F)F 6R-0339 CCc1cc(=O)[nH]c(n1)SCCCF 6R-0341 COCCCNC(=O)c1cc(c[nH]1)C(=O)c2cccc(c2)C(F)(F)F 6R-0342 c1ccc2c(c1)ccc3c2CC(O3)C(=O)N4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 6R-0343 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NCCCN4CCOCC4 6R-0344 c1ccc2c(c1)ccc3c2CC(O3)C(=O)N4CCN(CC4)c5ccccc5F 6R-0345 c1ccc(cc1)c2ccnc3c2c(n[nH]3)N 6R-0346 CN(CCOc1ccc(cc1)c2ccn(n2)C(=O)c3cccc(c3)OC)c4ccccn4 6R-0348 CCc1cc(=O)[nH]c(n1)SC(C)C(=O)OC 6R-0349 c1cc(cc(c1)C(F)(F)F)C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 6R-0350 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NCc4ccc(cc4)F 6R-0351 COCCNC(=O)C1Cc2c3ccccc3ccc2O1 6R-0352 COC(=O)C1CCN(CC1)Cc2ccc(c(c2)Cl)Cl 6R-0353 c1ccc(cc1)NC(=O)NNC(=O)C2CC(=NO2)c3cccnc3 6R-0355 c1cc(cnc1)C2=NOC(C2)C(=O)NNC(=O)NC3CCCCC3 6R-0356 c1cc(cnc1)C2=NOC(C2)C(=O)NNC(=O)Nc3ccc(cc3)Cl 6R-0357 Cc1cc(c(c(c1O)Br)C(C)C)Br 6R-0600 CCOc1c(ccc(n1)c2ccc(cc2)OC)C#N 6R-0601 c1cc(sc1)C(CC(=O)O)N 6R-0602 Cn1c2ccc(c(c2nn1)[N+](=O)[O-])/C=C/N(C)C 6R-0603 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCc3cnc(s3)Cl 6R-0606 c1ccc2c(c1)ccc(c2/C=N\c3ccc(cc3)Br)OCc4cnc(s4)Cl 6R-0607 c1ccc2c(c1)ccc(c2/C=N\NC(=O)c3ccc(cc3)C(F)(F)F)OCc4cnc(s4)Cl 6R-0608 Cc1c(c(no1)c2ccccc2Cl)C(=O)OCc3cnc(s3)Cl 6R-0609 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)OCc3cnc(s3)Cl 6R-0610 c1ccc2c(c1)ccc(c2C=C(C#N)C#N)OCc3cnc(s3)Cl 6R-0611 COc1ccc(cc1)NC(=O)c2ccc(cc2)N3CCS(=O)(=O)CC3 6R-0612 CC1CCN(CC1)Cc2cnc(s2)Cl 6R-0613 COC(=O)Cc1ccc(cc1)OCc2cnc(s2)Cl 6R-0614 c1cc(ccc1C(CC(=O)O)N)F 6R-0615 c1ccc(c(c1)N2CCN(CC2)C(=O)c3ccc(cc3)N4CCS(=O)(=O)CC4)F 6R-0616 CCOc1ccc(cc1)C(CC(=O)O)N 6R-0617 Cc1c(ccc(n1)Cl)C(=O)C 6R-0618 CC1CCCCN1Cc2cnc(s2)Cl 6R-0619 CC1CCCN(C1)Cc2cnc(s2)Cl 6R-0620 CCOc1c(ccc(n1)c2ccco2)C#N 6R-0621 CCOc1c(ccc(n1)c2ccco2)C(=O)N 6R-0622 c1ccc(c(c1)C(CC(=O)O)N)Cl 6R-0624 Cc1c(ccc(n1)Oc2ccc(cc2)OC)C(=O)C 6R-0625 C/C(=C/C(=O)c1ccccc1)/N 6R-0626 Cc1cc(n(n1)Cc2cnc(s2)N3CCOCC3)C 6R-0629 Cc1ccc(cc1)C(CC(=O)O)N 6R-0630 CCOC(=O)C1CCN(CC1)Cc2cnc(s2)Cl 6R-0632 c1cc(ccc1C(CC(=O)O)N)Br 6R-0633 c1cc(cc(c1)C(F)(F)F)C(CC(=O)O)N 6R-0634 Cc1cc(n(n1)Cc2cnc(s2)N3CCC(CC3)C)C 6R-0635 Cc1cc(c(cc1O)C(C)C)Br 6R-0636 c1cc(oc1)C(CC(=O)O)N 6R-0637 Cc1c(nc2cc(ccc2n1)NC(=S)NC(=O)c3ccccc3)C 6R-0639 c1cc(cc(c1)Cl)C(CC(=O)O)N 6R-0641 c1ccc(c(c1)C(CC(=O)O)N)F 6R-0642 CCOC(=O)c1cnn2c1nc(c(c2C)Cc3c(cccc3Cl)Cl)C 6R-0802 Cc1cc2nc(c(c(n2n1)C)Cc3c(cccc3Cl)Cl)C 6R-0803 Cc1csc(n1)Nc2nccc(n2)c3cnc(s3)c4ccc(cc4)Cl 6R-0804 Cc1csc(n1)Nc2nccc(n2)c3c(nc(s3)c4cccnc4)C 6R-0805 Cc1c(sc(n1)c2ccccc2)C(=O)C3C(C3(C#N)C#N)c4ccc(cc4)Cl 6R-0806 Cc1cc2nc(c(c(n2n1)O)CC(=O)OC)C 6R-0807 CCOC(=O)c1cnn2c1nc(c(c2C)Cc3cccc(c3)F)C 6R-0808 CC(=O)c1ccccc1N/C=C/C(=O)c2ccc(cc2)Oc3ccccc3 6R-0809 Cc1c2ccccc2ncc1C(=O)c3ccc(cc3)Oc4ccccc4 6R-0810 Cc1ccc(cc1)N/C=C/C(=O)c2c(nc(s2)c3ccccc3)C 6R-0811 Cc1ccc(cc1)N/C=C/C(=O)c2c(nc(s2)c3cccnc3)C 6R-0812 Cc1ccc(cc1)N/C=C/C(=O)c2cnc(s2)c3ccc(cc3)Cl 6R-0813 c1cc(c(nc1)Cl)NC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 6R-0815 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/NOCc3ccccc3 6R-0816 c1cc(ccc1c2ncc(s2)c3ccc(c(=O)[nH]3)C#N)Cl 6R-0817 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/Nc3ccc(cc3Cl)Cl 6R-0821 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/Nc3ccc(cc3)Br 6R-0822 CC(=O)c1ccccc1N/C=C/C(=O)c2ccc(cc2)c3ccccc3 6R-0824 Cc1c2ccccc2ncc1C(=O)c3ccc(cc3)c4ccccc4 6R-0825 COC(=O)c1ccccc1n2c(c(nn2)CO)CO 6R-0826 CN(C)C(=O)Oc1c(cnn1c2cccc(n2)Cl)n3cncn3 6R-0827 Cc1cc2nc(c(c(n2n1)C)Cc3cccc(c3)F)C 6R-0828 Cc1ccc(cc1)N/C=C/C(=O)c2c(nc(s2)c3ccc[n+](c3)C)C.[I-] 6R-0829 Cc1ccc(cc1)N/C=C/C(=O)c2c(nc(s2)c3ccc[n+](c3)Cc4ccc(cc4)Cl)C.[Cl-] 6R-0830 c1ccc2c(c1)c(c[nH]2)CCNc3c(cc(cn3)C(F)(F)F)Cl 6R-0833 Cc1cc2nc(c(c(n2n1)C)Cc3cccc(c3)C(F)(F)F)C 6R-0834 COC(=O)c1c(noc1c2cn(nn2)c3ccsc3C(=O)OC)c4ccccc4 6R-0835 CC(=O)c1cnc(s1)c2cccnc2 6R-0836 Cc1c2ccccc2nc(c1C(=O)C(F)(F)F)O 6R-0838 Cc1c(c(n2c(n1)ncn2)C)Cc3cccc(c3)C(F)(F)F 6R-0839 c1cc(c(cc1Cl)Cl)C2CC(=O)CC(=O)C2n3cncn3 6R-0840 Cc1c(c(n2c(n1)nc(n2)SC)C)Cc3cccc(c3)F 6R-0841 Cc1ccc(cc1)C(C(C(=O)c2ccc(c(c2)OC)OC)O)N3CCOCC3 6R-1000 CN1c2ccccc2/C(=C/c3ccc(c(c3)[N+](=O)[O-])Cl)/C1=O 6R-1002 c1ccc(cc1)CNC(=O)c2c(ccs2)n3cccc3 6R-1004 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)Cl)/C(=O)OC 6R-1005 Cc1c(sc(n1)c2ccc(cc2)Cl)C(C)O 6R-1006 Cc1cccc(c1N2C(=O)CCC2=O)C 6R-1007 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCOCC3 6R-1009 Cc1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccc(cc2)N3CCOCC3 6R-1010 c1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccc(cc2)N3CCOCC3 6R-1011 COc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCOCC3 6R-1012 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)F)N3CCOCC3 6R-1013 COC(=O)c1ccccc1SCC(=O)Nc2ccc(cc2)N3CCOCC3 6R-1014 c1ccc(c(c1)N)SCC(=O)Nc2ccc(cc2)N3CCOCC3 6R-1015 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3ccc(cc3)N4CCOCC4 6R-1016 c1ccc(cc1)S(=O)(=O)Nc2ccccc2SCC(=O)Nc3ccc(cc3)N4CCOCC4 6R-1017 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCOCC3 6R-1018 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Cl)N3CCOCC3 6R-1019 COc1ccc(cc1)C(=O)Nc2ccccc2SCC(=O)Nc3ccc(cc3)N4CCOCC4 6R-1020 CN1CCN(CC1)c2ccc(cc2F)[N+](=O)[O-] 6R-1021 COC(=O)COc1ccc(=O)n(n1)c2ccccc2 6R-1023 CN1CCN(CC1)c2ccc(cc2F)N 6R-1024 c1ccc(cc1)n2c(=O)ccc(n2)OCC(=O)O 6R-1025 Cc1ccc2c(c1)C(CCS2)(C)O 6R-1026 Cc1ccc(cc1)S(=O)(=O)NCCc2c[nH]c3c2cccc3 6R-1027 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(cc3)Cl 6R-1028 Cc1ccc(cc1)NC(=O)c2ccc(c(c2)F)N3CCN(CC3)C 6R-1029 c1ccc2c(c1)c(c[nH]2)C(C(F)(F)F)O 6R-1060 c1ccc2c(c1)c(c[nH]2)C(=O)C(F)(F)Cl 6R-1061 c1ccc2c(c1)nc(o2)SC[C@H](C(F)(F)F)O 6R-1062 COC(=O)c1c(ccs1)NC(=O)CCl 6R-1063 c1ccc(cc1)SC[C@H](C(F)(F)F)O 6R-1064 CS(=O)(=O)n1cc(c2c1cccc2)C(=O)C(F)(F)F 6R-1065 Cn1cc(c2c1cccc2)C(=O)C(F)(F)F 6R-1066 c1cc(ccc1CNC(=O)C(F)(F)Br)F 6R-1068 CC(=O)Cn1c2ccccc2nn1 6R-1070 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NC(=O)c3cccs3)SC 6R-1120 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NC(=O)c3ccc(cc3)Cl)SC 6R-1121 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NC(=O)c3ccc(cc3)C)SC 6R-1122 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NC(=O)c3ccc(c(c3)Cl)Cl)SC 6R-1123 CSc1c(cc2ccccc2n1)/C=C(\C#N)/c3cccc(c3)Cl 6R-1124 CSc1c(cc2ccccc2n1)/C=C(\C#N)/c3cccc(c3)C(F)(F)F 6R-1126 Cc1cccc(c1)/C(=C/c2cc3ccccc3nc2SC)/C#N 6R-1127 CSc1c(cc2ccccc2n1)/C=C(\C#N)/c3ccccc3 6R-1128 CSc1c(cc2ccccc2n1)/C=C(\C#N)/c3ccc(c(c3)Cl)Cl 6R-1129 CSc1c(cc2ccccc2n1)/C=C(\C#N)/c3ccc(cc3Cl)Cl 6R-1131 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)c3ccc(cc3)Cl)SC 6R-1132 CSc1c(cc2ccccc2n1)/C=C/C(=O)c3ccc(cc3)Cl 6R-1134 CSc1c(cc2ccccc2n1)/C=C/C(=O)c3ccc(cc3)F 6R-1136 COc1cccc(c1)C(=O)/C=C/c2cc3ccccc3nc2SC 6R-1137 c1ccc(cc1)/C(=C/c2cc3ccccc3nc2SCc4ccc(cc4)Cl)/C#N 6R-1139 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=C(\C#N)/c4cccc(c4)Cl 6R-1140 COc1ccc(cc1)C(=O)/C=C/c2cc3ccccc3nc2SCc4ccc(cc4)Cl 6R-1141 COc1ccc(cc1OC)/C(=C/c2cc3ccccc3nc2SC)/C#N 6R-1145 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NC(=O)c3cccc(c3)Cl)SC 6R-1149 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NC(=O)c3cccc(c3Cl)Cl)SC 6R-1151 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NC(=O)c3ccc(cc3)F)SC 6R-1152 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)CO 6R-1155 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=C(\C#N)/c4ccc(c(c4)Cl)Cl 6R-1159 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)c3ccc(cc3)C)SC 6R-1163 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)c3ccc(cc3)F)SC 6R-1164 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)c3ccc(cc3Cl)Cl)SC 6R-1165 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)c3ccc(cc3)OC)SC 6R-1166 COC(=O)c1cc2cc3ccccc3nc2s1 6R-1168 COc1cccc(c1)CSc2c(cc3ccccc3n2)C=O 6R-1169 c1ccc2c(c1)cc(c(n2)SCc3ccc(c(c3)Cl)Cl)C=O 6R-1170 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)c3ccccc3)SC 6R-1171 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)SC 6R-1172 CCOC(=O)c1cnc(nc1Oc2cccc(c2)NS(=O)(=O)C)SC 6R-1173 CCSc1c(cc2ccccc2n1)C=O 6R-1174 Cc1ccc(cc1)CSc2c(cc3ccccc3n2)C=O 6R-1175 CC(C)(C)c1ccc(cc1)CSc2c(cc3ccccc3n2)C=O 6R-1176 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/O 6R-1178 c1ccc(cc1)c2c(cnn2c3c(cc(cc3Cl)Cl)Cl)NC(=O)Nc4ccc(cc4)Cl 6R-1181 c1ccc(cc1)c2c(cnn2c3c(cc(cc3Cl)Cl)Cl)NC(=O)Nc4ccccc4 6R-1182 Cc1cc(cc(c1)NC(=O)Nc2cnn(c2c3ccccc3)c4c(cc(cc4Cl)Cl)Cl)C 6R-1183 c1ccc(cc1)c2c(cnn2c3c(cc(cc3Cl)Cl)Cl)NC(=O)Nc4ccc(cc4)Br 6R-1185 c1ccc(cc1)c2c(cnn2c3c(cc(cc3Cl)Cl)Cl)NC(=O)Nc4cccc(c4)[N+](=O)[O-] 6R-1186 CC(C)c1ccc(cc1)NC(=O)Nc2cnn(c2c3ccccc3)c4c(cc(cc4Cl)Cl)Cl 6R-1187 COc1ccc(cc1)NC(=O)Nc2cnn(c2c3ccccc3)c4c(cc(cc4Cl)Cl)Cl 6R-1188 Cc1ccc(cc1)C(C(C(=O)c2ccc(cc2)C)O)N3CCCCC3 6R-1195 Cc1c(sc(n1)c2ccc(cc2)Cl)C(C)OC(=O)Nc3ccccc3 6R-1200 c1ccc(cc1)C(C(C(=O)c2ccccc2)O)N3CCOCC3 6R-1203 Cc1c(sc(n1)c2cccnc2)C(C)OC(=O)Nc3cccc(c3)Cl 6R-1205 Cc1c(sc(n1)c2ccc(cc2)Cl)C(C)OC(=O)NC(C)C 6R-1209 Cc1c(sc(n1)c2ccc(cc2)Cl)C(C)OC(=O)c3ccc(cc3)Cl 6R-1210 C=CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)/C=C/c3ccccc3 6R-1250 CCn1c(nnc1SCC#N)/C=C/c2ccccc2 6R-1252 CCn1c(nnc1SCC(=O)N)/C=C/c2ccccc2 6R-1254 CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)/C=C/c3ccccc3 6R-1255 CCSc1nc2c3c(cc(nc3sc2c(n1)Cl)C)C 6R-1301 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccc(cc4)Cl)Cl)C 6R-1302 Cc1ccc(cc1)C(=O)ON=C2CC(N(C(C2)(C)C)C(=O)C)(C)C 6R-1305 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)Oc5ccccc5)C)C 6R-1306 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)Oc5cccc(c5)C(F)(F)F)C)C 6R-1307 Cc1ccc(cc1)CSc2nc3c4c(cc(nc4sc3c(n2)Oc5ccc6ccccc6c5)C)C 6R-1308 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCC=C)Oc4ccccc4)C 6R-1309 Cc1cccc(c1)Oc2c3c(c4c(cc(nc4s3)C)C)nc(n2)SCC=C 6R-1310 CCSc1nc2c3c(cc(nc3sc2c(n1)Oc4ccc(cc4)C)C)C 6R-1312 CCSc1nc2c3c(cc(nc3sc2c(n1)Oc4ccccc4C(=O)OC)C)C 6R-1313 CCSc1nc2c3c(cc(nc3sc2c(n1)NCC=C)C)C 6R-1315 CCSc1nc2c3c(cc(nc3sc2c(n1)Sc4ccccc4)C)C 6R-1316 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccc(cc4)Cl)NC(C)C)C 6R-1318 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccc(cc4)Cl)N5CCCC5)C 6R-1319 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccc(cc4)Cl)N5CCCCCC5)C 6R-1320 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccc(cc4)Cl)SCc5cccc(c5)C(F)(F)F)C 6R-1321 Cc1cc(nc2c1c3c(s2)c(nc(n3)SCc4ccc(cc4)Cl)Sc5ccc(cc5)F)C 6R-1322 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OC(=O)c4ccc(c(c4)Cl)Cl 6R-1352 Cc1cccc(c1)C(=O)Nc2ccc(cc2)N3CCN(CC3)C(C)C 6R-1363 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)Cn2c3ccccc3nc2C(F)(F)F 6R-1364 c1ccc2c(c1)nc(n2CC(=O)Oc3cccc(c3)C(F)(F)F)C(F)(F)F 6R-1365 CCN1CCN(CC1)c2ccc(cc2)NC(=O)c3ccc(cc3)C 6R-1372 Cc1ccc(cc1)NC(=O)C(C)n2c3ccccc3nc2C(F)(F)F 6R-1373 Cc1cccc(c1)NC(=O)C(C)n2c3ccccc3nc2C(F)(F)F 6R-1374 Cc1ccccc1NC(=O)C(C)n2c3ccccc3nc2C(F)(F)F 6R-1375 CCCCc1ccc(cc1)c2csc(n2)N 6R-1506 CCC(C)c1ccc(cc1)c2csc(n2)N 6R-1507 CCCCc1ccc(cc1)c2csc(n2)NC(=O)C 6R-1508 CCC(C)c1ccc(cc1)c2csc(n2)NC(=O)C 6R-1509 CCCCc1ccc(cc1)c2csc(n2)NC(=O)Cc3ccccc3 6R-1510 CCCCc1ccc(cc1)c2csc(n2)NC(=O)c3cccs3 6R-1511 CCCCc1ccc(cc1)c2csc(n2)NC(=O)c3cccc(c3)C(F)(F)F 6R-1514 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OCc4ccc(cc4)Cl 6R-1520 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OC(=O)c4ccc(cc4)F 6R-1521 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OC(=O)C4CC4 6R-1522 COc1ccc(cc1)CO/N=C/c2cc3ccccc3nc2SCc4ccc(cc4)Cl 6R-1523 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OC(=O)c4cccs4 6R-1524 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OC(=O)c4cccc(c4)Cl 6R-1525 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OC(=O)c4cccc(c4)C(F)(F)F 6R-1526 CC(C)(C)c1ccc(cc1)CO/N=C/c2cc3ccccc3nc2SCc4ccc(cc4)Cl 6R-1527 CCOC(=O)c1cnc(nc1Sc2ccccc2NC(=O)c3ccc(c(c3)Cl)Cl)SC 6R-1529 COC(=O)CSc1ccsc1C(=O)OC 6R-1532 Cc1ccc(cc1)Nc2ncc(s2)c3ccnc(n3)N 6R-9005 Cc1ccc(cc1)Nc2nc(c(s2)c3ccnc(n3)N)C 6R-9007 Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)c3ccnc(n3)N 6R-9008 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)c3ccnc(n3)N 6R-9009 Cc1ccc(cc1)c2nc(c(s2)c3ccnc(n3)N)C 6R-9010 Cc1c(sc(n1)c2ccc(cc2)F)c3ccnc(n3)N 6R-9013 Cc1c(sc(n1)c2cccc(c2Cl)Cl)c3ccnc(n3)N 6R-9014 Cc1c(sc(n1)c2ccc(cc2Cl)Cl)c3ccnc(n3)N 6R-9015 Cc1c(sc(n1)Nc2ccc(cc2)C(F)(F)F)c3ccncn3 6R-9035 c1cc(ccc1C(F)(F)F)Nc2ncc(s2)c3ccnc(n3)N 6R-9038 Cc1c(sc(n1)N(C)c2ccc(cc2)C(F)(F)F)c3ccnc(n3)N 6R-9040 Cc1c(sc(n1)Nc2cccc(c2Cl)Cl)c3ccnc(n3)N 6R-9059 c1cc(sc1)c2ccnc(n2)SCC#N 6T-0001 CN(C)/C=C/C(=O)c1cc2c3ccccc3ccc2o1 6T-0002 Cc1ccc(n1c2ccc(cc2)C(=O)/C=C/N(C)C)C 6T-0003 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)C=C(C#N)C#N 6T-0004 CN1C(=O)C(=Cc2cccn2c3ccc(cc3)OC(F)(F)F)C(=O)N(C1=O)C 6T-0005 c1ccc2c(c1)n3cc(nc3s2)C(=O)NN 6T-0006 c1cc(oc1)c2ccnc(n2)S 6T-0007 Cc1ccn2cc(nc2c1)C(=O)NN 6T-0010 c1ccc2c(c1)C(=O)N(C2=O)Cc3cnc(s3)Cl 6T-0011 CC(=O)c1cn(c2c1cccc2)Cc3cnc(s3)Cl 6T-0013 c1ccc2c(c1)n3cc(nc3s2)C(=O)O 6T-0014 CC(=O)C(C(=O)C)Sc1nccc(n1)c2cccs2 6T-0016 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)/C=N\NC(=S)N 6T-0018 Cc1ccc(n1c2nccc(n2)c3ccco3)C 6T-0025 COC(=O)c1cc2ccccc2n1Cc3cnc(s3)Cl 6T-0026 c1ccn(c1)c2nccc(n2)c3ccco3 6T-0029 CC(=O)c1ccc(cc1)NC(=O)/C=C/C(=O)O 6T-0030 c1ccc(c(c1)C#N)n2ccc(c2)C=O 6T-0031 c1cc(oc1)C(=O)C/C=N/OCc2ccc(cc2Cl)Cl 6T-0032 c1cc(sc1)C(=O)/C=C/Nc2ccc(cc2)Cl 6T-0033 CN1CCN(CC1)c2ncc(s2)CN3C(=O)c4ccccc4C3=O 6T-0034 c1cc(n(c1)c2nccc(n2)c3ccco3)C=O 6T-0037 COC(=O)/C=C/c1ccccc1F 6T-0039 COc1cc2c(cc1OC)C(CC2NC(=O)C(F)(F)F)O 6T-0047 COc1cc2c(cc1OC)C(=O)NCC2NC(=O)C(F)(F)F 6T-0048 c1ccc2c(c1)cc(s2)c3cc[nH]n3 6T-0052 CSc1nccc(n1)c2cccs2 6T-0053 CC(=O)c1ccc(cc1)N2C(=O)C=CC2=O 6T-0056 CCOC(=O)Cn1c(c(c(n1)C)C=O)Cl 6T-0061 Cc1c(c(nc(c1C#N)O)O)CN2CCN(CC2)c3ccc(cc3)OC 6T-0063 c1cc(n(c1)Cc2cnc(s2)Cl)C=O 6T-0065 c1ccc2c(c1)cc(s2)c3ccnc(n3)S 6T-0069 COC(=O)CSc1nccc(n1)c2ccco2 6T-0070 c1cc(oc1)c2ccnc(n2)SCC#N 6T-0071 Cc1cccc(c1C)N/C=C/C(=O)c2cccs2 6T-0072 c1ccc2c(c1)c(cn2Cc3cnc(s3)Cl)C=C(C#N)C#N 6T-0077 CCOC(=O)c1cnc2c(c1NCCCN(C)C)cnn2C 6T-0078 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCCCN(C)C 6T-0079 CCOC(=O)c1cnc2c(c1NCCC#N)cnn2C 6T-0080 CCOC(=O)c1cnc2c(c1NCCc3ccccc3)cnn2C 6T-0081 CCOC(=O)c1cnc2c(c1NCc3cccc(c3)C(F)(F)F)cnn2C 6T-0083 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCCc3ccccc3 6T-0084 COc1cccc(c1)N/C=C/C(=O)c2cccs2 6T-0087 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCc3cccc(c3)C(F)(F)F 6T-0088 CCOC(=O)c1cnc2c(c1NCc3ccc(cc3)OC)cnn2C 6T-0089 CCOC(=O)c1cnc2c(c1N)cnn2C 6T-0092 c1ccnc(c1)c2nccc(n2)c3cccs3 6T-0096 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCc3ccc(cc3)OC 6T-0099 Cc1ccc(cc1)C/N=C/c2cccn2c3ccc(cc3)OC(F)(F)F 6T-0101 c1cc(oc1)c2ccn(n2)CCO 6T-0102 CCOC(=O)c1cnc2c(c1NCCCN)cnn2C 6T-0103 CCSc1nc(cc(=O)n1c2ccccc2)C(F)(F)F 6T-0201 c1ccc(cc1)n2c(=O)cc(nc2SCC(=O)O)C(F)(F)F 6T-0202 COc1ccc(cc1)c2cc3c(nc(nc3nc2c4ccc(cc4)OC)N)N 6T-0203 Cc1cccc(c1)CSc2nc(cc(=O)n2c3ccccc3)C(F)(F)F 6T-0205 c1ccc(cc1)n2c(=O)cc(nc2SCC(=O)c3ccc(cc3)Cl)C(F)(F)F 6T-0206 Cc1ccccc1Cn2ccc(n2)c3ccc4c(c3)OCO4 6T-0207 c1cc(ccc1c2ccnc3n2ncc3C#N)n4cncn4 6T-0208 CSc1c(c2c(c(n1)c3cccc(c3)C(F)(F)F)CCCC2)C#N 6T-0210 CCOC(=O)C1CCN(CC1)c2ccc(cc2)N 6T-0212 c1cc(cc(c1)F)Cn2ccc(n2)c3ccc4c(c3)OCO4 6T-0214 Cc1cc([nH]n1)/N=C(\C)/C2CCOC2=O 6T-0216 c1cc(cc(c1)C(F)(F)F)c2c3c(c(c(n2)SCc4c(cccc4Cl)F)C#N)CCCC3 6T-0219 c1cc(cc(c1)C(F)(F)F)c2c3c(c(c(n2)SCc4ccc(cc4)[N+](=O)[O-])C#N)CCCC3 6T-0220 Cc1cccc(c1)CSc2c(c3c(c(n2)c4cccc(c4)C(F)(F)F)CCCC3)C#N 6T-0221 CC(C)(C)c1ccc(cc1)CSc2c(c3c(c(n2)c4cccc(c4)C(F)(F)F)CCCC3)C#N 6T-0222 c1cc(cc(c1)Cl)CSc2c(c3c(c(n2)c4cccc(c4)C(F)(F)F)CCCC3)C#N 6T-0223 Cc1nnc(n1Cc2ccccc2)c3cnn(c3N)C 6T-0224 c1cc2c(cc1c3ccn(n3)CCO)OCO2 6T-0225 Cc1nnc(n1Cc2ccc(cc2)F)c3cnn(c3N)C 6T-0226 c1cc(cc(c1)C(F)(F)F)CSc2c(c3c(c(n2)c4cccc(c4)C(F)(F)F)CCCC3)C#N 6T-0227 c1ccc2c(c1)c(cn2c3ccc(cc3)C=O)C=O 6T-0228 COc1cc(cc(c1OC)OC)C(=O)n2ccc(n2)c3ccc4c(c3)OCO4 6T-0229 Cc1nnc(n1Cc2ccc3c(c2)OCO3)c4cnn(c4N)C 6T-0230 c1ccc(cc1)/C=C/Cn2ccc(n2)c3ccc4c(c3)OCO4 6T-0231 c1cc2c(cc1N)OCC(=O)N2 6T-0236 c1cc(c(cc1N2CCC(CC2)C(=O)O)C(=O)N)[N+](=O)[O-] 6T-0237 c1cc(c(cc1Cn2ccc(n2)c3ccc4c(c3)OCO4)Cl)Cl 6T-0240 CCOC(=O)C1CCN(CC1)c2ccc3c(c2)nc(c(n3)c4ccccc4)c5ccccc5 6T-0241 CCc1c(nc2cc(ccc2n1)N3CCC(CC3)C(=O)OCC)CC 6T-0242 c1ccc(cc1)n2c(=O)cc(nc2O)C(F)(F)F 6T-0246 c1ccc(cc1)n2c(=O)cc(nc2SCCC(=O)O)C(F)(F)F 6T-0247 c1ccc2c(c1)c(cn2c3ccc(cc3)/C=C(\C#N)/c4ccccc4F)C=O 6T-0248 c1ccc2c(c1)c(cn2c3ccc(cc3)/C=C(\C#N)/c4cccnc4)C=O 6T-0250 c1ccc2c(c1)c(cn2c3ccc(cc3)/C=C(\C#N)/c4cccs4)C=O 6T-0251 CC(C)(C)c1ccc(cc1)Cn2ccc(n2)c3ccc4c(c3)OCO4 6T-0255 c1cc2c(cc1c3ccnc(n3)Cn4cncn4)OCO2 6T-0256 CS(=O)(=O)/C(=C\c1ccc(cc1)n2cc(c3c2cccc3)/C=C(/C#N)\S(=O)(=O)C)/C#N 6T-0257 Cn1cccc1/C(=C/c2ccc(cc2)n3cc(c4c3cccc4)C=O)/C#N 6T-0259 c1ccc(cc1)n2c(=O)cc(nc2SCc3ccc(c(c3)Cl)Cl)C(F)(F)F 6T-0261 c1ccc(cc1)/C=C/CSc2nc(cc(=O)n2c3ccccc3)C(F)(F)F 6T-0263 c1ccc(cc1)n2c(=O)cc(nc2SCc3cccc(c3)F)C(F)(F)F 6T-0264 COc1ccc(cc1)c2c(sc(n2)N)c3ccc(cc3)OC 6T-0265 c1ccc2c(c1)c(cn2c3ccc(cc3)/C=C(\C#N)/c4c(cccc4Cl)Cl)C=O 6T-0266 CCCCCCCc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)n3cnc4c3cccc4 6T-0271 c1cc(ccc1C(=O)/C=C/c2ccc3c(c2)OCO3)n4cncn4 6T-0272 Cc1c(c(n(n1)C)C)/C=C/C(=O)c2ccc(cc2)n3cncn3 6T-0273 Cc1cccc(c1)Cn2c(cc(=O)n(c2=O)c3ccc(cc3)Cl)C(F)(F)F 6T-0274 Cc1ccc(cc1)C(=O)CSc2nc(cc(=O)n2c3ccccc3)C(F)(F)F 6T-0275 c1ccc(cc1)n2c(=O)cc(nc2SCC(=O)c3ccc(cc3)Br)C(F)(F)F 6T-0276 CC(=O)CSc1nc(cc(=O)n1c2ccccc2)C(F)(F)F 6T-0278 c1ccc(cc1)CCC2C(c3cccc4c3N2CCC4)(C(F)(F)F)O 6T-0279 COc1ccc(cc1)c2c(sc(n2)c3cccnc3)c4ccc(cc4)OC 6T-0281 c1cc(ccc1OCc2nccc(n2)c3ccc4c(c3)OCO4)F 6T-0282 c1cc(ccc1c2ccnc(n2)COc3ccc(cc3)F)n4cncn4 6T-0283 Cc1cc2[nH]c(c(c(=O)n2n1)CCO)C 6T-0285 COc1cc(c(cc1OC)NC(=S)NCc2ccc(c(c2)Cl)Cl)C#N 6T-0288 CCn1c(=O)cc(nc1SCc2ccc(cc2)C)C(F)(F)F 6T-0292 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=S)Nc3cc(c(cc3C#N)OC)OC 6T-0297 Cn1c(=O)c2c(n(c1=O)C)OCC2=O 6T-0298 CN(C)S(=O)(=O)c1ccc(cc1)NC(=S)Nc2cc(c(cc2C#N)OC)OC 6T-0299 c1cc2c(cc1c3ccn(n3)CCOc4c(cc(cn4)C(F)(F)F)Cl)OCO2 6T-0301 CC(=C)C(=O)NCCCCCCCCCCC(=O)O 6T-0302 COc1cc(c(cc1OC)/N=C(/NCc2ccc(c(c2)Cl)Cl)\SC)C#N 6T-0303 COc1ccc(cc1Cl)CN/C(=N/c2cc(c(cc2C#N)OC)OC)/SC 6T-0304 Cn1c(=O)c2c(n(c1=O)C)O/C(=C/N(C)C)/C2=O 6T-0305 Cc1c(c(on1)n2cccc2)Cl 6T-0308 CCn1c(=O)cc(nc1SCC(=O)c2ccc(cc2)Br)C(F)(F)F 6T-0312 CCn1c(=O)cc(nc1SCC(=O)c2ccc(cc2)C)C(F)(F)F 6T-0313 Cn1c(c(c(=O)n(c1=O)C)C(=O)Cn2ccnc2)O 6T-0314 CCOC(=O)c1cc2c([nH]1)ccs2 6T-0315 CCn1c(=O)cc(nc1SCC(=O)c2ccc(cc2)Cl)C(F)(F)F 6T-0316 COc1ccc(cc1)CNC(=O)CSc2nc(cc(=O)n2c3ccccc3)C(F)(F)F 6T-0318 c1ccc(cc1)CCc2c(c3cccc4c3n2CCC4)C(F)(F)F 6T-0320 COc1cc(c(cc1OC)NC(=S)NCc2ccc(cc2)F)C#N 6T-0321 COc1ccccc1CNC(=S)Nc2cc(c(cc2C#N)OC)OC 6T-0322 CCOC(=O)C1CCN(CC1)c2ccc3c(c2)nccn3 6T-0323 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)Cc3ccccc3Cl 6T-0324 c1cc(c(nc1)Oc2ccc(cc2)C#N)C=O 6T-0327 CCOC(=O)c1c(sc2n1nc(c2C=O)C)SCc3ccccc3 6T-0331 CC(=O)Nc1ccc(cc1N)OC 6T-0332 COc1cc(c(cc1OC)/N=C(\NCc2ccc(cc2)F)/SC)C#N 6T-0333 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccccc3Cl)SC 6T-0334 c1cc(ccc1C(F)(F)F)Nc2ncc(s2)c3ccncn3 6T-0609 CCOC(=O)C1=C(N(C(=C(C1c2ccc(cc2Cl)Cl)C#N)N)c3ccc(cc3)Cl)C 6T-0629 c1cc(ccc1/C=N/c2c(c3c(s2)CCCC3)C#N)Cl 6T-0631 C1CCc2c(c(c(s2)NC(=O)CCl)C#N)C1 6T-0648 CCOC(=O)c1c2c(sc1NC(=O)CCl)CCCC2 6T-0649 c1ccc(cc1)c2csc(n2)n3cccn3 6T-0800 COc1ccc(cc1)c2csc(n2)n3cccn3 6T-0801 Cc1cc(n2c(n1)c(cn2)c3ccccn3)C(F)(F)Cl 6T-0802 COc1ccc(cc1)c2csc(n2)N=C(N)N 6T-0803 Cc1cc(n2c(n1)c(cn2)S(=O)(=O)c3ccccc3)C(F)(F)Cl 6T-0804 COC(=O)c1cnc2c(cnn2c1N)c3ccc(cc3)Cl 6T-0805 Cn1c(c(cn1)c2cc3nc(cc(n3n2)O)COC)C(F)(F)F 6T-0807 Cc1cc(n2c(n1)c(c(n2)c3cnn(c3C(F)(F)F)C)Cl)C(F)(F)F 6T-0810 Cc1cc(n2c(n1)c(c(n2)c3cnn(c3C(F)(F)F)C)Br)C(F)(F)F 6T-0811 CC(=O)c1ccc(s1)N2CCN(CC2)c3cccc(c3)Cl 6T-0812 CC(=O)c1c(cc(cc1N)C(F)(F)F)C(F)(F)F 6T-0816 c1cc(ccc1c2cnn3c2ncc(c3N)C(=O)O)Cl 6T-0818 c1cc(ccc1CC(=O)NCCN2CCN(CC2)C(=O)Cc3ccc(cc3)Cl)Cl 6T-0824 CC(=O)/C=C/c1cc(ccc1F)F 6T-0827 Cc1c(c(n2c(n1)c(cn2)c3ccc(cc3)F)N)c4ccc(cc4)OC 6T-0829 Cc1cc2nc(c(c(n2n1)N)c3ccc(cc3)OC)C 6T-0832 CC(C)(C)S(=O)(=O)c1cnc2c(cnn2c1N)c3ccc(cc3)OC 6T-0833 CC(=O)c1ccc(s1)N2CCN(CC2)c3ccc(cc3)OC 6T-0834 CC(C(=O)c1cn(nn1)c2ccc(c(c2)Cl)F)Oc3cccc(c3)C(F)(F)F 6T-0835 COCc1cc(n2c(n1)c(cn2)c3ccc(cc3)OC)O 6T-0838 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)N)c5ccc(cc5)OC)C)C 6T-0840 Cc1c(c(n2c(n1)cc(n2)c3cnn(c3C(F)(F)F)C)N)c4ccc(cc4)OC 6T-0842 Cc1cc(n(n1)c2nc(cs2)C(=O)N3CCN(CC3)Cc4ccccc4)C(F)(F)F 6T-0846 Cc1cc(n(n1)c2nc(cs2)C(=O)Nc3nccs3)C(F)(F)F 6T-0847 Cc1cc(n(n1)c2nc(cs2)C(=O)Nc3ccccc3OC)C(F)(F)F 6T-0848 Cc1c(c(n2c(n1)c(cn2)c3ccsc3)N)c4ccc(cc4)OC 6T-0849 Cc1c(c(n2c(n1)c(cn2)c3ccccn3)N)c4ccc(cc4)OC 6T-0850 CCOC(=O)c1cnc2c(cnn2c1C(F)(F)F)c3ccc(cc3)F 6T-0851 Cn1c2c(cn1)C(=O)N3CCc4cc(c(cc4C3C2)OC)OC 6T-0852 COc1cc2c(cc1OC)C3Cc4c(cn[nH]4)C(=O)N3CC2 6T-0853 COc1cc2c(cc1OC)C3CC(=O)C4=C(N3CC2)CCCC4 6T-0855 Cc1ccc(n1c2ccsc2c3cc4ncc5c(n4n3)CCN(C5)c6ccc(cc6)[N+](=O)[O-])C 6T-0857 Cc1cc2ncc3c(n2n1)CCN(C3)c4ccc(cc4)[N+](=O)[O-] 6T-0858 CCNC(=O)Nc1nnc(s1)SCc2cccc(c2)OC 6T-0859 c1ccc(cc1)C2=Nc3ccccc3OC2 6T-0861 c1ccc2cc(ccc2c1)c3ccnc4n3ncc4c5ccc(cc5)Cl 6T-0863 c1ccc(cc1)Oc2ccccc2NC(=O)Cc3c(cc(cn3)C(F)(F)F)Cl 6T-0867 CCNC(=O)Nc1nnc(s1)SCc2cccc(c2)F 6T-0868 CCNC(=O)Nc1nnc(s1)SCc2cccc(c2)C(F)(F)F 6T-0869 CC(=O)Nc1nnc(s1)SCc2cccc(c2)OC 6T-0872 c1ccc2c(c1)CCN2C(=O)CC(=O)C(=O)CC(=O)N3CCc4c3cccc4 6T-0873 c1ccc(cc1)c2ccc(cc2)c3ccnc4n3ncc4c5cccc(c5)Cl 6T-0876 c1ccc(cc1)c2ccc(cc2)c3ccnc4n3ncc4c5ccc(cc5)F 6T-0877 COc1cc2c(cc1OC)C3CC4=C(CCCN4)C(=O)N3CC2 6T-0878 c1ccc2c(c1)c(c[nH]2)CCNC=O 6T-0879 Cc1ccc(n1c2nc3nc(c(c(n3n2)C)C/C=C/c4ccccc4)C)C 6T-0881 CN(C)/C=C/C(=O)c1ccc(s1)N2CCN(CC2)c3cccc(c3)Cl 6T-0882 CN(C)/C=C/c1c(c(cc(n1)C(F)(F)F)C(F)(F)F)C(=O)OC 6T-0883 C/C(=N\O)/c1ccc(s1)N2CCN(CC2)c3cccc(c3)Cl 6T-0884 CC(C)(C)c1ccc(cc1)Oc2cccc(c2)/C=C/c3ccnc4n3ncc4c5ccc(cc5)Cl 6T-0885 c1ccc(cc1)Nc2c(cccn2)C(=O)O 6T-0887 CC(=O)Nc1nnc(s1)SCc2cccc(c2)F 6T-0888 CC(=O)Nc1nnc(s1)SCc2cccc(c2)C(F)(F)F 6T-0889 c1ccc2cc(ccc2c1)c3ccnc4n3ncc4c5ccc(cc5)F 6T-0890 COc1cc2c(cc1OC)CNCC2 6T-0892 Cc1cc2nccc(n2n1)c3ccco3 6T-0897 COc1ccc(cc1OC)S(=O)(=O)N2CCc3cc(c(cc3C2)OC)OC 6T-0901 c1cc2c(cc1O)SCCO2 6T-0906 COc1ccc(cc1)C2=Nc3ccccc3OC2 6T-0911 c1cc(oc1)c2ccnc3n2ncc3c4ccc(cc4)Cl 6T-0914 CC(=O)c1ccc(s1)N2CCN(CC2)c3cccc(c3)C(F)(F)F 6T-0915 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2c(cn[nH]2)c3ccc(cc3)Cl)/C#N 6T-0919 Cn1c(c(cn1)c2cc3ncc(c(n3n2)N)S(=O)(=O)c4ccccc4)C(F)(F)F 6T-0920 COCc1cc(n2c(n1)c(cn2)c3ccccn3)O 6T-0921 CCC(=O)c1cc([nH]c1)C(=O)NC 6T-0922 CNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2F)F 6T-0923 COc1ccc(cc1)c2cnn3c2ncc(c3N)S(=O)(=O)c4ccccc4 6T-0924 c1ccc2c(c1)c(c[nH]2)C(=O)N3CCOCC3 6T-1485 c1ccc(cc1)CNC(=O)c2c[nH]c3c2cccc3 6T-1487 CC(=O)Oc1cc(nn1C)c2ccccc2 6T-1489 COC(=O)C1CCN(CC1)c2cc(nc(n2)N)Cl 6W-0016 Cc1ccc(cc1)/C(=N\C(=C\C#N)\C)/C=C/c2cc(c(c(c2)OC)OC)OC 6W-0017 CCOC(=O)c1cccc(c1)Nc2cc(nc(n2)N)Cl 6W-0018 Cc1cc(c(c(c1)C(=O)O)NC(=O)OC(C)(C)C)C 6W-0019 c1cc(ccc1/C=N/NC(=O)Nc2ccncc2)[N+](=O)[O-] 6W-0023 C/C(=N/NC(=O)Nc1ccncc1)/c2ccc(c(c2)Cl)Cl 6W-0027 c1cc2c(c(c1)F)c(=O)oc(=O)[nH]2 6W-0030 c1ccc(cc1)CS(=O)c2ccc(cc2[N+](=O)[O-])Cl 6W-0033 c1cc(c(nc1)c2ccc3c(ccc[n+]3c2)C(=O)[O-])C(=O)O 6W-0040 Cc1c(c(=O)[nH]n1S(=O)(=O)c2cccc(c2)C(F)(F)F)CCO 6W-0200 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccc(cc2Cl)Cl)CCO 6W-0201 Cc1c(c(=O)[nH]n1S(=O)(=O)c2ccccc2)CCO 6W-0202 CC(C)(C)OC(=O)N1CCC2(CC1)c3ccccc3CC2=O 6W-0205 c1cc2c(cc1C3=NNC(=O)CC3)CCC2 6W-0206 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)c3nc(on3)c4ccco4 6W-0208 COc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3O 6W-0209 c1ccc(c(c1)C(=O)c2cnn(c2)c3ccc(cc3)Cl)O 6W-0210 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3O 6W-0211 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NCc3cccc(c3)Cl 6W-0212 c1ccc(c(c1)C(=O)c2ccc3c(c2)CCC3)C(=O)O 6W-0213 Cc1cc2[nH]c(=O)c3ccccc3n2n1 6W-0214 c1cc(oc1)/C=C\2/C(=O)NC(=S)S2 6W-0219 CC(C)(C)OCCOc1cccc(c1)[N+](=O)[O-] 6W-0221 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)/C=C\C(=O)c4cccc(c4)C(F)(F)F 6W-0225 COc1ccc(cc1OC)c2c(cn(n2)c3ccccc3)/C=C\C(=O)c4cccs4 6W-0226 CSC1=NC(=O)/C(=C/c2ccco2)/S1 6W-0228 c1cc(c(cc1S(=O)(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-])Cl 6W-0230 CCOC(=O)c1cnc2c(c1NCCOC)c(nn2c3ccc(cc3)C)C 6W-0231 CCOC(=O)c1cnc2c(c1NCc3cccc(c3)C(F)(F)F)c(nn2c4ccc(cc4)C)C 6W-0233 CCOC(=O)C(=CNc1cc(nn1c2ccc(cc2)Cl)C)C(=O)OCC 6W-0235 c1ccc2c(c1)C(OC2=O)c3ccc4c(c3)CCC4 6W-0239 c1cc(ccc1c2ccn3c(c2C#N)nc(n3)C(Cl)(Cl)Cl)Cl 6W-0240 c1ccc2c(c1)c(n[nH]c2=O)c3ccc4c(c3)CCC4 6W-0242 c1cc2c(cc1c3cc[nH]n3)CCC2 6W-0243 CCOC(=O)c1cnc2c(c1NCCN3CCOCC3)c(nn2c4ccc(cc4)C)C 6W-0245 c1cc(c(cc1S(=O)(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-])NN 6W-0246 c1cc(c(cc1S(=O)(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-])N3CCOCC3 6W-0247 C1CC(=C(C1)C(=O)O)C(=O)O 6W-0249 CCOC(=O)C1=C(SCC1=O)Nc2ccccc2 6W-0252 Cc1cc2nc(ccn2n1)c3ccc4c(c3)CCC4 6W-0254 c1cc(c(cc1S(=O)(=O)N2CCCC2C(=O)O)[N+](=O)[O-])NN 6W-0257 c1cc(c(cc1S(=O)(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-])N3CCCC3 6W-0258 CC1CN(CC(O1)C)c2ccc(cc2[N+](=O)[O-])S(=O)(=O)N3CCC(CC3)C(=O)O 6W-0259 Cc1ccc(cc1)Cn2c3cc(nn3c4ccccc4c2=O)C 6W-0260 Cc1cc2n(c(=O)c3ccccc3n2n1)Cc4cccc(c4)C(F)(F)F 6W-0261 c1cc(c(cc1S(=O)(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-])N3CCCC3C(=O)O 6W-0263 Cc1ccsc1/C=C\2/C(=O)NC(=S)S2 6W-0266 c1cc(c(nc1)n2c(c(cn2)C#N)N)N 6W-0268 Cc1cc2n(c(=O)c3ccccc3n2n1)C/C=C/c4ccccc4 6W-0269 c1cc(oc1)/C=C/2\C(=O)N=C(S2)NC(C3CCCCC3)C(=O)O 6W-0271 Cc1n[nH]c(=O)n1c2ccc(cc2)Oc3ccccc3 6W-0273 Cc1cc2n(c(=O)c3ccccc3n2n1)Cc4cccc(c4)OC 6W-0276 c1cc(ccc1c2nc(on2)CCC(=O)O)Cl 6W-0277 c1ccc(cc1)n2cc(c(n2)c3ccc4c(c3)CCC4)C=O 6W-0278 c1ccc2c(c1)ccc(c2O)C(=O)c3cnn(c3)c4ccc(cc4)F 6W-0279 COc1ccc(cc1)n2cc(cn2)C(=O)c3ccc4ccccc4c3O 6W-0280 Cc1ccc(cc1)n2cc(cn2)C(=O)c3ccc4ccccc4c3O 6W-0281 c1ccc2c(c1)ccc(c2O)C(=O)c3cnn(c3)c4ccc(cc4)Cl 6W-0282 c1cc2c(cc1c3ccn4c(n3)ncn4)CCC2 6W-0284 CCC(=O)c1ccc2c(c1)CCC2 6W-0285 c1cc2c(cc1c3ccn4c(n3)c(cn4)C#N)CCC2 6W-0286 CC1=NCCN1S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl 6W-0288 CC1=NCCN1S(=O)(=O)c2ccc(cc2)[N+](=O)[O-] 6W-0290 c1cc2c(cc1c3ccnc(n3)N)CCC2 6W-0293 CCOC(=O)C1=C(OCC1=O)Nc2ccccc2 6W-0294 CSc1nc2nc(ccn2n1)c3ccc4c(c3)CCC4 6W-0296 COC(=O)c1cc(ccc1Cl)[N+](=O)[O-] 6W-0299 Cc1ccc(cc1)COc2c3ccccc3ccc2C(=O)c4cnn(c4)C(C)(C)C 6W-0301 c1ccc(cc1)n2cc(c(n2)c3ccc4c(c3)CCC4)/C=C(\C#N)/c5ccc6c(c5)OCO6 6W-0302 CC1=NCCN1S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])N3CCCC3 6W-0303 c1cc(ccc1C2CCCCC2)C(=O)CC(=O)C(F)(F)F 6W-0305 c1cc(oc1)/C=C\2/C(=O)N=C(S2)NC(=N)N 6W-0306 c1cc(oc1)/C=C/2\C(=O)N=C(S2)N3CCC(CC3)C(=O)O 6W-0307 Cc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)N3CCN(CC3)C(=O)OC(C)(C)C 6W-0312 C/C(=N\c1cc(cc(c1)OC)OC)/N(C)CCNS(=O)(=O)c2ccc(cc2)[N+](=O)[O-].I 6W-0316 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)CNC(=O)c3cccc(c3)OC 6W-0319 Cc1ccsc1/C=C\2/C(=O)N=C(S2)SC 6W-0320 c1ccc(cc1)n2cc(cn2)C(=O)c3ccc4ccccc4c3O 6W-0322 C/C(=N\c1ccc(cc1)OC(F)(F)F)/N(C)CCNS(=O)(=O)c2ccc(cc2)[N+](=O)[O-].I 6W-0324 c1cc(oc1)/C=C\2/C(=O)N=C(S2)NC(CO)C(=O)O 6W-0327 CCOC(=O)c1cnc2c(c1Cl)c(nn2c3ccc(cc3)Cl)C 6W-0328 Cc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)N3CCNCC3 6W-0330 CC1=NCCN1S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3 6W-0331 CC(C)(C)n1cc(cn1)C(=O)c2ccc3ccccc3c2Oc4ccc(c(n4)Cl)C(F)(F)F 6W-0332 CC(C)(C)n1cc(cn1)C(=O)c2ccc3ccccc3c2OCCCF 6W-0333 c1cc(ncc1C(=O)O)N2CCCCC2 6W-0335 CCOC(=O)/C(=C/C(=O)c1cccc(c1)[N+](=O)[O-])/N 6W-0802 COC(=O)CC(c1ccccc1F)NC(=O)C(F)(F)F 6W-0805 Cc1c(sc(n1)n2cccc2)c3ccn[nH]3 6W-0806 Cc1c(sc(n1)n2cccc2)c3ccnc(n3)N 6W-0807 Cc1cc(nc2n1nnn2)C(F)(F)F 6W-0810 CCOC(=O)c1cc(nc2c1C(=O)CCC2)c3cccc(c3)[N+](=O)[O-] 6W-0813 Cc1cc2c(cc(nc2cc1NC(=O)C(F)(F)F)Cl)COC 6W-0814 CCOC(=O)c1cc(nc2c1c(=O)[nH]c(=O)[nH]2)c3cccc(c3)[N+](=O)[O-] 6W-0815 Cc1cc(n2cc(nc2n1)c3ccc(cc3)F)O 6W-0819 c1ccc(cc1)c2c(nnc(n2)Sc3ccc(cc3[N+](=O)[O-])C#N)c4ccccc4 6W-0820 c1ccc(cc1)c2c(nnc(n2)Sc3c(cccn3)[N+](=O)[O-])c4ccccc4 6W-0821 c1cc(c(cc1N=[N+]=[N-])Cl)Cl 6W-0822 CC(=O)O/N=C/c1cccn1Cc2ccccc2[N+](=O)[O-] 6W-0823 CSc1nc(c(nn1)c2ccccc2)c3ccccc3 6W-0825 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/C)\c3cnccn3 6W-0826 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)O/N=C(/C)\c3cnccn3 6W-0827 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(/C)\c3cnccn3 6W-0828 C/C(=N/OC(=O)c1c(cccc1F)F)/c2cnccn2 6W-0829 COc1cc(ccc1OCc2cccc(c2)C(F)(F)F)/C=N/NC(=O)c3ccc(cc3)C(F)(F)F 6W-0830 COc1cc(ccc1OCc2cccc(c2)C(F)(F)F)/C=C/3\c4ccccc4NC3=O 6W-0832 CN1C(=O)C(=Cc2ccc(c(c2)OC)OCc3cccc(c3)C(F)(F)F)C(=O)N(C1=O)C 6W-0833 C/C(=N\O)/c1nccs1 6W-0834 Cc1cc(n2cc(nc2n1)c3ccc(cc3)F)Cl 6W-0835 c1ccc2c(c1)C(=O)NC(=CO2)c3cccc(c3)[N+](=O)[O-] 6W-0838 Cc1ccnc(n1)SCc2ccc(cc2)Cl 6W-0839 C/C(=N/OC(=O)c1c(cccc1F)F)/c2nccs2 6W-0840 C/C(=N\OC(=O)c1ccccc1F)/c2nccs2 6W-0843 COc1cc(ccc1OCc2cccc(c2)C(F)(F)F)/C=N/NC(=S)N 6W-0844 COc1cc(ccc1OCc2cccc(c2)C(F)(F)F)C=C(C#N)C#N 6W-0845 Cc1ccc(n1c2nc3nccc(n3n2)c4cccc(c4)N5CC(C5=O)(C)C)C 6W-0847 COC(=O)c1c2c(ccn(c2=O)CC(F)(F)F)c3cc4c(cc3n1)OCO4 6W-0848 c1cc(c(cc1n2cc(nn2)C(=O)C3CCCCC3=O)Cl)Cl 6W-0849 CN1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F 6W-0851 COc1cc(ccc1OCc2cccc(c2)C(F)(F)F)C(CC(=O)O)N 6W-0852 c1ccc2c(c1)c(=O)[nH]c3n2ncc3c4[nH]nnn4 6W-0853 CC1(CC(=O)C(=CNc2ccc(cc2)OC(F)(F)F)C(=O)C1)C 6W-0854 CC1(CC(=O)C(=CNc2cccnc2)C(=O)C1)C 6W-0855 COc1cc(ccc1OCc2ccc(cc2)F)C(CC(=O)O)N 6W-0856 c1cc(c(cc1n2cc(nn2)C(=O)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl 6W-0857 COc1cc(ccc1OCc2cnc(s2)Cl)C(CC(=O)O)N 6W-0859 Cc1ccc(n1C(CC(=O)OC)c2ccc(cc2)F)C 6W-0860 Cc1cc(n2cc(nc2n1)c3ccc(cc3)F)N4CCOCC4 6W-0861 Cc1cc(n2cc(nc2n1)c3ccc(cc3)F)N4CCN(CC4)C 6W-0862 COC(=O)c1c(c2ccccc2[nH]1)Cl 6W-0863 CC1(CC(=O)C(=CNc2ccccc2F)C(=O)C1)C 6W-0864 Cc1cc(n2cc(nc2n1)c3ccc(cc3)F)OCc4ccc(cc4)Cl 6W-0865 CC(=O)c1c(cc(cn1)C(F)(F)F)n2cncn2 6W-0867 COc1cc(ccc1OCc2cccc(c2)C(F)(F)F)/C=C/C(=O)O 6W-0869 c1ccc2c(c1)/C(=C\c3cnc(s3)Cl)/C(=O)N2 6W-0871 CC1(CC(=O)C(=CNc2ccccc2)C(=O)C1)C 6W-0872 Cc1cc2c(cc(=O)[nH]c2cc1NC(=O)c3cccc(c3)OC)COC 6W-0875 COc1ccc(cc1)C2COc3ccccc3C(=O)N2 6W-0878 CN1C(=O)C(=Cc2cnc(s2)Cl)C(=O)N(C1=O)C 6W-0879 COc1cc(ccc1OCc2cnc(s2)Cl)/C=C/C(=O)O 6W-0881 COc1ccc(cc1)c2cn3cc(ccc3n2)C(=O)OC 6W-0882 Cc1cc(n2cc(nc2n1)c3ccc(cc3)F)N4CCCCC4 6W-0883 COc1ccccc1C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 6X-0051 COc1ccc(c(c1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)OC 6X-0052 Cc1ccc(cc1)c2nc(on2)c3cccc(c3)OC 6X-0058 CC(=O)Nc1ccc(cc1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 6X-0086 Cc1ccc(cc1)c2nc(on2)c3ccc(cc3)Cl 6X-0089 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)NC(=O)CCCCl 6X-0200 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)NC(=O)c4ccc(cc4)[N+](=O)[O-] 6X-0202 c1ccc(c(c1)/C=C\2/C(=O)N=C(S2)NOCc3c(cccc3Cl)Cl)C(F)(F)F 6X-0204 c1ccc(cc1)CONC2=NC(=O)/C(=C/c3ccccc3C(F)(F)F)/S2 6X-0205 c1ccc2c(c1)cc(s2)C(=O)Nc3nc(cs3)CCN4C(=O)c5ccccc5C4=O 6X-0214 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)/C(=C/c4cc(ccc4Cl)[N+](=O)[O-])/C#N 6X-0216 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)N=C(N)N 6X-0218 CCOC(=O)C1CN(c2cc(ccc2O1)S(=O)(=O)CC)S(=O)(=O)c3ccc(cc3)OC 6X-0220 CCOC(=O)C1CN(c2cc(ccc2O1)S(=O)(=O)CC)S(=O)(=O)C 6X-0221 c1ccc(c(c1)/C=C(\C#N)/c2ccc3c(c2)OCO3)Oc4ccc(cc4Cl)Cl 6X-0224 c1cc(cc(c1)C(F)(F)F)/C=C\2/C(=O)C3CCN2CC3 6X-0225 c1ccc(cc1)CNc2nc(cs2)CCN3C(=O)c4ccccc4C3=O 6X-0226 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)/C(=C\c4cc(ccc4Sc5ccccn5)[N+](=O)[O-])/C#N 6X-0229 c1ccc(cc1)CN(CC(=O)O)C2=NC(=O)/C(=C\c3cccc4c3cccc4)/S2 6X-0230 c1cc2c(cc1/C=C\3/C(=O)C4CCN3CC4)OCO2 6X-0231 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)O)S(=O)(=O)c3ccc(cc3)OC 6X-0234 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)O)S(=O)(=O)C 6X-0235 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCNCC3 6X-0237 c1cc(nc2c1cncc2)C(=O)NCC(=O)N 6X-0238 c1cc(cc(c1)[N+](=O)[O-])/C=C\2/C(=O)C3CCN2CC3 6X-0240 c1cc(cc(c1)C(F)(F)F)CN2CCC(CC2)c3cc([nH]n3)c4cccc(c4)C(F)(F)F 6X-0244 c1cc(nc2c1cncc2)C(=O)NCCc3c[nH]cn3 6X-0245 c1ccc2c(c1)cccc2/C=C\3/C(=O)C4CCN3CC4 6X-0246 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)CC#N 6X-0249 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)Cc4ccc(cc4)Br 6X-0250 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)Cc4c(cccc4Cl)F 6X-0251 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)Cc4ccc(cc4)[N+](=O)[O-] 6X-0252 c1cc(c(cc1[N+](=O)[O-])/C=C\2/C(=O)C3CCN2CC3)Cl 6X-0254 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCNCC4 6X-0258 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4cccc(c4)C(F)(F)F 6X-0259 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 6X-0260 COc1ccc(cc1S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4cccc(c4)C(F)(F)F)Cl 6X-0261 CN(CC(=O)O)c1ncc2c(n1)-c3ccccc3OC2 6X-0262 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)c4ccc(c(c4)C(F)(F)F)[N+](=O)[O-] 6X-0265 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)c4c(cccn4)[N+](=O)[O-] 6X-0266 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4cccc5c4cccc5 6X-0267 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCN(CC4)S(=O)(=O)c5cccc(c5)C(F)(F)F 6X-0268 CCOC(=O)C1CN(c2cc(ccc2O1)S(=O)(=O)CC)S(=O)(=O)c3ccc(cc3)Cl 6X-0269 CCOC(=O)C1CN(c2cc(ccc2O1)S(=O)(=O)CC)S(=O)(=O)c3ccccc3 6X-0270 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)C(=O)c4ccc(cc4)[N+](=O)[O-] 6X-0272 Cc1cc(c(c(c1)C)C(=O)N2CCC(CC2)c3cc([nH]n3)c4cccc(c4)C(F)(F)F)C 6X-0274 Cc1ccc(c(c1)CN2CCC(CC2)c3cc([nH]n3)c4cccc5c4cccc5)C 6X-0279 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCN(CC4)Cc5ccc(cc5)F 6X-0280 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCN(CC4)Cc5c(cccc5Cl)Cl 6X-0281 COc1ccc(cc1)[NH2+]c2nc(cs2)CCN3C(=O)c4ccccc4C3=O.[Br-] 6X-0282 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)[NH2+]c4cccc(c4)C(F)(F)F.[Br-] 6X-0283 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)O)S(=O)(=O)c3ccc(cc3)Cl 6X-0289 CCOC(=O)C1CN(c2cc(ccc2O1)S(=O)(=O)CC)S(=O)(=O)c3ccc(cc3)C 6X-0290 CCOC(=O)C1CN(c2cc(ccc2O1)S(=O)(=O)CC)S(=O)(=O)c3cccs3 6X-0291 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)O)S(=O)(=O)c3ccccc3 6X-0296 CCS(=O)(=O)c1ccc2c(c1)NCC(O2)C(=O)NN 6X-0298 COC(=O)CCN1CCC(CC1)c2cc([nH]n2)c3cccc(c3)C(F)(F)F 6X-0299 CCOC(=O)C1CNc2cc(ccc2O1)Cl 6X-0302 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)O)S(=O)(=O)c3cccs3 6X-0303 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)O)S(=O)(=O)c3ccc(cc3)C 6X-0304 c1cc(cc(c1)[N+](=O)[O-])c2cc(n[nH]2)C3CCN(CC3)Cc4cc(cc(c4)C(F)(F)F)C(F)(F)F 6X-0307 c1ccc2c(c1)cccc2/C=C(\C#N)/c3nc(cs3)CCN4C(=O)c5ccccc5C4=O 6X-0309 c1ccc2c(c1)C(=O)N(C2=O)CCc3csc(n3)/C(=C/c4ccc(cc4)OCc5cccc(c5)C(F)(F)F)/C#N 6X-0310 c1ccc(cc1)/C=C/C=C(\C#N)/c2nc(cs2)CCN3C(=O)c4ccccc4C3=O 6X-0311 c1cc(cc(c1)[N+](=O)[O-])c2cc(n[nH]2)C3CCN(CC3)Cc4ccc(cc4)C(F)(F)F 6X-0314 c1cc(cc(c1)[N+](=O)[O-])c2cc(n[nH]2)C3CCN(CC3)c4c(cccn4)C#N 6X-0315 c1cc(cc(c1)[N+](=O)[O-])c2cc(n[nH]2)C3CCN(CC3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 6X-0316 CCOC(CCl)(OCC)OCC 6X-0700 c1cc(ccc1C(=O)CO)[N+](=O)[O-] 6X-0701 c1cc2c(cc1[N+](=O)[O-])nc(o2)CCl 6X-0702 c1cc2c(cc1[N+](=O)[O-])oc(n2)CCl 6X-0703 c1ccc(cc1)CN2CCC(CC2)CO 6X-0704 c1ccc(cc1)CN2CCCC(C2)CO 6X-0705 Cc1ccc(n1c2ccc(cc2)C=C(C#N)C#N)C 6X-0707 Cc1ccc(n1c2ccc(cc2)CC(C#N)C#N)C 6X-0708 CCOC(=O)C1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(=O)C 6X-0709 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCCCC2 6X-0710 c1cc2c(cc1Cl)nc(o2)CCl 6X-0711 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCOCC2 6X-0712 CC(C)(C)OC(=O)Nc1ccc(cn1)C(=O)OC 6X-0713 Cc1ccc(cc1)S(=O)(=O)/N=c\2/ccc(c[nH]2)C(=O)OC 6X-0714 Cc1cc(c(n1c2ccc(cc2)Br)C)C(=O)C(F)(F)F 6X-0715 CC(=O)Nc1ccc(cn1)C(=O)OC 6X-0716 c1cc2c(cc1Br)cc(s2)C(=O)NN 6X-0720 Cc1cc(=O)c(co1)O 6X-0801 CSc1c(c2nc(cc(n2n1)C(F)(F)F)C(F)(F)F)C#N 6X-0805 CC(=O)c1c(cc(cn1)C(F)(F)F)c2ccc(cc2)OC 6X-0816 c1cc2c(cc1[N+](=O)[O-])nco2 6X-0817 Cc1cc(ccc1NC(=O)c2ccc3c(c2)OCO3)Br 6X-0819 Cc1ccc2c(c1)nco2 6X-0820 c1cc(c2c(c1)ocn2)[N+](=O)[O-] 6X-0821 Cc1nc2c(o1)cccn2 6X-0823 Cc1c(oc2c1c(ccc2OC)[N+](=O)[O-])C 6X-0826 c1cscc1C(CCO)N2CCS(=O)(=O)CC2 6X-0827 Cc1cc(n(n1)c2nc(cs2)Cn3cccn3)C(F)(F)F 6X-0828 c1ccc(c(c1)C(F)(F)F)NC(=O)c2ccc3c(c2)OCO3 6X-0829 c1ccc(cc1)OCC(CN2CCOCC2)O 6X-0830 c1cc(ncc1C(=O)C2CC2)C3CC3 6X-0832 CC(C#Cc1c(cc(cn1)C(F)(F)F)Cl)O 6X-0835 c1cc2c(cc1N)nco2 6X-0836 COc1ccc(cc1OCC#C)[N+](=O)[O-] 6X-0837 COC(=O)c1cccn2c1nc(c2Cl)c3ccc(cc3)F 6X-0838 c1cc(c2nc(cn2c1)c3ccc(cc3)F)C(=O)O 6X-0839 c1ccc(cc1)OCC(CN2CCN(CC2)c3ccc(c(c3)Cl)Cl)O 6X-0840 COc1ccc(cc1)N2CCN(CC2)CC(COc3ccccc3)O 6X-0841 c1cc(ccc1C2c3ccsc3CCN2)C(F)(F)F 6X-0842 COc1ccc(cc1)C2c3ccsc3CCN2 6X-0843 c1cc(ccc1C2c3ccsc3CCN2)OC(F)(F)F 6X-0844 CCCCCC(=O)NNC(=O)c1c(c2ccccc2[nH]1)Cl 6X-0845 c1ccc(cc1)S(=O)(=O)NNC(=O)c2c(c3ccccc3[nH]2)Cl 6X-0846 c1ccc2c(c1)c(c([nH]2)C(=O)NNS(=O)(=O)c3cccs3)Cl 6X-0847 c1ccc(c(c1)C2NCC(O2)c3ccc(cc3)[N+](=O)[O-])Cl 6X-0850 Cc1ccc(cc1[N+](=O)[O-])OCC2NCCS2 6X-0852 COc1ccc(cc1)c2ccc(cn2)C(=O)c3ccc(cc3)OC 6X-0856 Cn1c(c(c(=O)n(c1=O)C)Cc2cn(c3c2cc(cc3)OC)C(=O)c4cccs4)O 6X-0857 CC(C(=O)n1cc(c2c1ccc(c2)OC)Cc3c(n(c(=O)n(c3=O)C)C)O)Oc4ccccc4 6X-0860 Cn1c(c(c(=O)n(c1=O)C)Cc2cn(c3c2cc(cc3)OC)S(=O)(=O)c4ccccc4)O 6X-0861 c1cc(c2c(c1)ocn2)N 6X-0863 COC(=O)c1ccc2nc(cn2c1)c3ccc(cc3)S(=O)(=O)C 6X-0864 c1cc(sc1)S(=O)(=O)Nc2ccc3c(c2)nco3 6X-0866 c1ccc(cc1)NC(=O)Nc2ccc3c(c2)nco3 6X-0867 CCOC(=O)c1ccccc1c2cn3cc(ccc3n2)Cl 6X-0868 CCOC(=O)C(=CNc1ccc2c(c1)nco2)C(=O)OCC 6X-0869 COC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)COc3ccc(cc3Cl)Cl 6X-0870 COC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)Cn3cncn3 6X-0871 CS(=O)(=O)c1ccc(cc1)c2cn3cc(ccc3n2)C(=O)O 6X-0872 CC1CCN(CC1)CC(C(F)(F)F)O 6X-0874 c1cc2c(cc1NC(=S)NC3CCCCC3)nco2 6X-0876 c1cc(cc(c1)c2ccnc(n2)N)C#N 6X-0878 COC(=O)Cc1cn2cc(ccc2n1)Cl 6X-0879 c1ccc(cc1)CC(c2ccccc2)NCN3C(=O)c4ccccc4C3=O 6X-0880 c1cc(c2nc(cn2c1)c3ccc(cc3)Br)[N+](=O)[O-] 6X-0882 COc1ccccc1CNC(=O)c2ccccc2c3ccc(cc3)C(F)(F)F 6X-0885 COc1ccccc1CNCC(C(F)(F)F)O 6X-0886 CCOc1cccc2c1oc(=O)c(c2)C(=O)O 6X-0887 CC1=C(CC(=O)N1CCc2c[nH]c3c2cc(cc3)OC)C(=O)OC 6X-0889 Cc1c2cc3c(cc2ncc1C(=O)c4ccc(cc4)OC)OCO3 6X-0890 CC(=O)c1cc2c(cc1N/C=C/c3ccc(cc3)OC)OCO2 6X-0891 c1cc(cc(c1)OC(F)F)CNC(=O)Cn2cncn2 6X-0892 Cc1ccc(c(c1)S)NC 6X-0920 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)C)C)O 6X-0922 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)OCC)C)C 6X-0924 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)C)C)C 6X-0925 c1ccc(cc1)C(=O)CCC#N 6X-0926 c1ccc2c(c1)-c3c(cn(n3)c4ccc(cc4)Cl)CO2 6X-0929 c1ccc2c(c1)-c3c(cn(n3)C(=O)c4ccc(cc4)[N+](=O)[O-])CO2 6X-0930 c1ccc2c(c1)-c3c(cn(n3)C(=O)c4ccc(cc4)Cl)CO2 6X-0931 C[NH+](C)CCC(=O)c1ccc(cc1)Cl.[Cl-] 6X-0932 c1ccc2c(c1)-c3c(cn(n3)c4ccc(cc4)F)CO2 6X-0933 CCOC(=O)CSc1ccc(cc1)OC 6X-0937 CCOC(=O)CS(=O)(=O)c1ccc(cc1)OC 6X-0941 c1ccc(cc1)CN(CCO)CCO 6X-0943 COc1cc2c(cc1OC)C=CNC(=O)C2 6X-0944 c1cc(ccc1C(=O)CCC#N)Cl 6X-0945 Cn1cc(c(=O)c2c1cccc2)c3ccccc3C(=O)OC 6X-0948 CC(C)c1ccc(c(c1)S)NC 6X-0949 c1ccc(cc1)CN(CCCl)CCCl.Cl 6X-0950 c1ccc2c(c1)C3c4cccn4CCN3C2=O.O 6X-0953 CSC(=C(CC#N)C(=O)c1ccc(cc1)Cl)SC 6X-0955 Cc1ccc(cc1)S(=O)(=O)C(=O)C2CCOc3c2cccc3 6X-0958 CCOC(=O)C1(CCN(CC1)Cc2ccccc2)S(=O)(=O)c3ccc(cc3)OC 6X-0961 C[NH+](C)CCC(=O)c1ccc(cc1)OC.[Cl-] 6X-0962 c1cc(ccc1CN(CCO)CCO)Cl 6X-0963 CN(C)/C=C/c1ccc(cc1[N+](=O)[O-])Cl 6X-0965 c1ccc(cc1)c2cnnc(c2C#N)N 6X-0966 c1cc(ccc1C[NH+](CCCl)CCCl)Cl.[Cl-] 6X-0968 CC(C)(C)OC(=O)Nc1cccc(c1)C(=O)O 6X-5023 CC(C)(C)OC(=O)NC1CCNCC1 6X-5030 COCCNC(=O)c1cccc(c1)[N+](=O)[O-] 6X-5055 c1cc(cc(c1)[N+](=O)[O-])C(=O)NCCO 6X-5074 CNc1ccc(cc1)c2nc3ccccc3s2 6X-7042 CN(C)C(=O)c1cccc(c1)N 6X-9015 c1cc(cc(c1)N)C(=O)NCCO 6X-9020 CN1CCC(=CC1)c2c[nH]c3c2cc(cc3)OC 6Y-0001 CN1CCC(=CC1)c2c[nH]c3c2cc(cc3)C#N 6Y-0003 CC(C)(C)OC(=O)N1CCC(=CC1)c2c[nH]c3c2cc(cc3)Br 6Y-0006 c1ccc(cc1)c2ccc(nc2)C#N 6Y-0033 c1cc2cccnc2c(c1)OS(=O)(=O)C(F)(F)F 6Y-0201 CC(C)(C)OC(=O)N1CCC(CC1)Nc2ccccc2 6Y-0207 CC(C)c1ccc(cc1)NC2CCN(CC2)C(=O)OC(C)(C)C 6Y-0211 c1cc2c(cc1N)cns2 6Y-0252 CN(C(=O)c1ccc(c(c1)Cl)Cl)OC 6Y-0602 C1CNCC1CO 6Y-0603 Cc1ccnc(n1)SC 6Y-0605 CSc1nccc(n1)CC(=O)c2ccc(c(c2)Cl)Cl 6Y-0607 CC(C)(C(=O)OC)n1cncn1 6Y-0608 c1ccc(cc1)/C=N/NC(=O)N 6Y-0609 c1cc2c(cc1O)c(c(o2)C3CC3)C=O 6Y-0800 COc1ccc(cc1OC(c2ccccc2)C(=O)O)C=O 6Y-0802 c1cc(ccc1/C(=N/O)/N)Br 6Y-0803 c1cn[nH]c1c2ccsc2 6Y-0804 Cc1cc(n[nH]1)c2ccc(cc2)OC 6Y-0805 Cc1cc(n[nH]1)c2cccc(c2)C(F)(F)F 6Y-0806 Cc1cc(n[nH]1)c2ccc3c(c2)OCO3 6Y-0807 CC(=O)c1ccc(cc1)OC(c2ccccc2)C(=O)O 6Y-0808 c1c(c(c(s1)C(=O)CCl)Br)Br 6Y-0810 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])c4c5ccccc5c(=O)[nH]n4 6Y-0814 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCCCCC4 6Y-0815 c1cc(oc1)c2c(c3cc(ccc3o2)O)C=O 6Y-0818 c1cc(ccc1c2cc[nH]n2)[N+](=O)[O-] 6Y-0820 CN1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(=O)c3ccccc3C(=O)O 6Y-0824 c1ccc(c(c1)C(=O)c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)N4CCCCC4)C(=O)O 6Y-0825 CN1CCN(CC1)c2ccc(cc2[N+](=O)[O-])c3c4ccccc4c(=O)[nH]n3 6Y-0827 CC1CCN(CC1)c2ccc(cc2[N+](=O)[O-])c3c4ccccc4c(=O)[nH]n3 6Y-0828 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCSCC4 6Y-0831 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCC(CC4)N5CCCCC5 6Y-0832 c1cc(ccc1c2c(cnc(n2)N)C#N)Br 6Y-0837 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCCC4 6Y-0839 COC(c1c(c2cc(ccc2o1)O)C=O)OC 6Y-0841 c1cnc(nc1c2ccsc2)N 6Y-0842 CN(C(=O)c1cccc(c1)C(F)(F)F)OC 6Y-0843 CCS(=O)(=O)N1CCN(CC1)c2ccc(cc2[N+](=O)[O-])c3c4ccccc4c(=O)[nH]n3 6Y-0845 c1ccnc(c1)c2cc[nH]n2 6Y-0847 c1cc(ccc1c2ccnc(n2)N)[N+](=O)[O-] 6Y-0848 CSc1nccc(n1)CC(=O)c2cccc(c2)C(F)(F)F 6Y-0849 c1c(c(cs1)Br)C=O 6Y-0850 c1c(c(c(s1)C=O)Br)Br 6Y-0851 c1cc(c(c(c1)Cl)Cl)C(CC(=O)O)N 6Y-0854 COc1ccc2c(c1)c(c(o2)C3CC3)C=O 6Y-0858 Cc1cc(cc(c1)COc2ccc3c(c2)c(c(o3)C4CC4)C=O)C 6Y-0859 c1cc2c(cc1OCc3ccc(nc3)Cl)c(c(o2)C4CC4)C=O 6Y-0860 c1ccc2c(c1)/C(=C/c3cscc3Br)/C(=O)N2 6Y-0861 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCSCC2 6Y-0862 CC(=O)c1ccc(c(c1)F)OCc2ccc(cc2)[N+](=O)[O-] 6Y-0922 CC(=O)c1ccc(c(c1)F)OCc2cc(ccc2Br)OC 6Y-0926 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(CC(=O)O)c4ccc(cc4)Cl 6Y-0928 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCN(CC4)c5ccc(cc5)O 6Y-0930 CC(C)c1ccc(cc1)C(CC(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4.O 6Y-0933 CC(=O)c1ccc(c(c1)Cl)OCc2cccc(c2)OC 6Y-0934 c1cnc(c(c1C(=O)O)Cl)Cl 6Z-0225 c1cc(c(nc1)N2CCCCC2)C(=O)O 6Z-0233 c1cc(c(nc1)N2CCOCC2)C(=O)O 6Z-0242 CN(c1c(cccn1)C(=O)O)C2CCCCC2 6Z-0243 CCOC(=O)/C=C/c1ccc(cc1)C(C)C 6Z-0260 CC(C)c1ccc(cc1)/C=C/CO 6Z-0274 c1cc2c(cc1C(CC(=O)O)N3CCC4(CC3)OCCO4)OCO2 6Z-0276 CCOC(=O)/C=C/c1ccc(cc1)OC 6Z-0282 CCOC(=O)c1cc(n[nH]1)C(F)(F)F 6Z-0604 CCOC(=O)c1cn[nH]c1C 6Z-0609 c1(c(non1)N)C(=O)O 6Z-0700 c1cc(ccc1c2ccc(cc2C(=O)O)[N+](=O)[O-])Br 6Z-0702 CCOC(=O)c1cn2cc(ccc2n1)C#N 6Z-0705 c1cc(ccc1C=O)c2ccsc2 6Z-0706 c1cc(ccc1C=O)c2cnccn2 6Z-0709 c1cc(ccc1C=O)c2ccc3c(c2)OCO3 6Z-0711 CCOC(=O)Cc1csc(n1)c2cccc(c2)C(F)(F)F 6Z-0712 c1cc(cc(c1)C(F)(F)F)c2nc(cs2)CC(=O)O 6Z-0713 Cn1c(c(c(n1)C(F)(F)F)C=O)Oc2ccccc2C(F)(F)F 6Z-0715 c1ccc(cc1)C(=O)Nc2ccc(cc2)C3c4ccsc4CCN3 6Z-0800 c1csc(n1)C(=O)CBr.Br 6Z-0801 CC(C)(C)OC(=O)NCCCCO 6Z-0811 c1cc(ccc1Oc2ccc(cc2C=O)[N+](=O)[O-])Cl 6Z-0813 c1cc(ccc1Oc2ccc(cc2CO)[N+](=O)[O-])Cl 6Z-0814 c1cc(c(c(c1)C#N)N2CCOCC2)C#N 6Z-0818 COc1ccc2c(c1)c(cn2c3ncccn3)C=O 6Z-0825 c1ccc(cc1)COc2cnccc2C#N 6Z-5009 c1cc(ccc1n2c(c(nn2)C#N)N)Cl 7B-005 CN(C)/C=N/c1c(nnn1c2ccc(cc2)Cl)C#N 7B-006 CN(c1cccc(n1)Cl)N 7B-009 c1ccc(c(c1)CNC(=O)c2ccc(cc2)Cl)n3ccnc3 7B-010 c1cc(ccc1C(=O)c2ccc(cc2)n3ccnc3)n4ccnc4 7B-011 c1ccc2c(c1)c(=O)c3ccc(nc3o2)c4ccc(cc4)Cl 7B-012 c1ccc2c(c1)c(=O)c3ccc(nc3o2)c4cccnc4 7B-013 c1ccc(c(c1)CNS(=O)(=O)c2ccc(cc2)Cl)n3ccnc3 7B-014 C[n+]1ccn(c1)c2ccc(cc2)C(=O)c3ccc(cc3)n4cc[n+](c4)C.[I-].[I-] 7B-015 CN(C)/C=N/c1nc2ccccc2s1 7B-017 c1ccc2c(c1)c(=O)c3ccc(nc3o2)c4ccncc4 7B-018 CN(c1cccc(n1)Cl)NC(=O)c2ccc(cc2)Cl 7B-024 CC(=O)c1cnc2n(c1=O)c3ccccc3s2 7B-026 CN(C)/C=N/c1c(nnn1c2cccc(c2)C(F)(F)F)C#N 7B-029 CC(=O)CC(=O)Nc1ccsc1C(=O)OC 7B-030 CN(C)/C=C/C(=O)c1cnc2n(c1=O)c3ccccc3s2 7B-031 CC(=O)c1cnc2n(c1=O)ccs2 7B-032 CC(=O)c1cnc2n(c1=O)ncs2 7B-033 c1cc(ccc1C(c2ccc(cc2)n3ccnc3)O)n4ccnc4 7B-034 c1ccc2c(c1)n3c(=O)c(cnc3s2)c4ccn[nH]4 7B-035 c1ccc2c(c1)n3c(=O)c(cnc3s2)c4ccnc(n4)N 7B-036 Cn1c(c(c(n1)Cl)Cl)N(C)NC(=O)c2cccc(c2)C(F)(F)F 7B-038 c1ccc(cc1)/C=C/CSc2ccccc2 7B-041 CN(C)/C=C/C(=O)c1cnc2n(c1=O)ccs2 7B-043 c1ccc(cc1)/C=C/CS(=O)(=O)c2ccccc2 7B-044 c1cn[nH]c1c2cnc3n(c2=O)ccs3 7B-045 CN(C)/C=C(/C=C/c1ccccc1)\S(=O)(=O)c2ccccc2 7B-048 CO/N=C\C(/C=C/c1ccccc1)S(=O)(=O)c2ccccc2 7B-050 c1ccc(cc1)/C=C/C(/C=N\O)S(=O)(=O)c2ccccc2 7B-051 CNc1c2c(nn1C)CCCC2.C(=C/C(=O)O)\C(=O)O 7B-052 CC(=O)/C(=C/N(C)C)/C(=O)Nc1ccsc1C(=O)OC 7B-055 c1ccc(cc1)n2cc3c(=O)c4ccccc4oc3nc2=O 7B-056 c1ccc2c(c1)c(=O)c3cn(c(=O)nc3o2)c4ccc(cc4)Cl 7B-057 Cc1ccc(cc1)n2cc3c(=O)c4ccccc4oc3nc2=O 7B-058 CC(=O)c1cnc2n(c1=O)CCS2 7B-060 CC(=O)c1ccc(cc1)N2CCN(CC2)C 7B-061 CN(C)/C=C(\C#N)/c1nnc(o1)N(C)C 7B-063 COC(=O)c1c(ccs1)/N=C/NNc2ccc(cc2Cl)Cl 7B-064 CN(C)c1nnc(o1)c2cn[nH]c2N 7B-067 Cc1cc(nc(n1)O)C.Cl 7B-070 CN(C)c1nnc(o1)c2cnc(nc2N)N 7B-071 CC(c1ccc(cc1)n2ccnc2)O 7B-073 CC(=O)c1cnc2[nH]c3ccccc3n2c1=O 7B-075 Cn1c(c2c(n1)CCCC2)N(C)C(=O)Nc3ccccc3 7B-076 Cn1c(c2c(n1)CCCC2)N(C)C(=O)N 7B-078 Cn1c(c2c(n1)CCCC2)N(C)C(=O)c3ccc(cc3)Cl 7B-080 CN(C)/C=C/C(=O)c1cnc2n(c1=O)CCS2 7B-081 c1cn[nH]c1c2cnc3n(c2=O)CCS3 7B-086 c1cnc(nc1c2cnc3n(c2=O)CCS3)N 7B-087 CC(=O)c1cnc2n(c1=O)nc(s2)SC 7B-088 c1cc(c(nc1)Cl)C(=O)Nc2ccc(cc2F)F 7B-091 CN(C)/C=C/C(=O)c1cnc2n(c1=O)ncs2 7B-092 c1cc(ccc1N2CCCC2=O)Cl 7B-101 Cc1ccccc1C(=O)NNc2cccc(n2)Cl 7B-104 c1cc(nc(c1)Cl)NNC(=O)c2ccc(cc2Cl)Cl 7B-105 c1cc(c(c(c1)F)C(=O)NNc2cccc(n2)Cl)F 7B-106 c1cc(c(c(c1)Cl)C(=O)NNc2cccc(n2)Cl)Cl 7B-107 C/C(=N\Nc1cccc(n1)Cl)/c2ccc(cc2Cl)Cl 7B-108 Cc1ccc(cc1)N2CCCC2=O 7B-109 COc1ccc(cc1)N2CCCC2=O 7B-110 c1cc(c(c(c1)Cl)C(=O)NNc2c(cccn2)C(F)(F)F)Cl 7B-111 CN(c1cccc(n1)Cl)NC(=O)c2c(cccc2Cl)Cl 7B-114 c1ccnc(c1)SCC(=C(C#N)C#N)N 7C-003 c1ccc(cc1)CSC(=C(C#N)C#N)N 7C-007 Cc1c(c(ns1)SCC(=O)c2ccc(cc2)Cl)C#N 7C-009 Cc1c(c(ns1)S(=O)(=O)Cc2ccc(cc2Cl)Cl)C#N 7C-010 c1ccc(cc1)OCC(=C(C#N)C#N)N 7C-013 CC(=O)C1=C(C(NC1=O)(C)O)c2ccccc2 7C-014 CC1(C(=C(C(=O)N1)C(=O)/C=C/N(C)C)c2ccccc2)O 7C-015 c1cc(ccc1OCC#N)F 7C-016 CC1=C(C(=O)NC1(C)O)C(=O)C 7C-017 c1cc(ccc1OCC(=C(C#N)C#N)N)F 7C-019 c1cc(cc(c1)Cl)OCC(=C(C#N)C#N)N 7C-021 c1cc(cc(c1)OCC#N)C(F)(F)F 7C-024 c1cc(ccc1[N+](=O)[O-])OCC(=C(C#N)C#N)N 7C-025 c1cc(cc(c1)OCC(=C(C#N)C#N)N)C(F)(F)F 7C-026 COc1ccc(cc1)SCC(=C(C#N)C#N)N 7C-035 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)NC(C)(C)C 7C-039 CCN(CC)C(=O)c1cc2c(=O)c3cc(ccc3oc2nc1C)Cl 7C-040 CN1CCN(CC1)/C(=N/C#N)/SC 7C-042 CS/C(=N\C#N)/N1CCN(CC1)Cc2ccccc2 7C-043 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)NCc4ccncc4 7C-044 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)Nc4ccncc4 7C-045 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)Cl)C(=O)OCc4ccccc4 7C-046 c1ccc(cc1)C(=C(C#N)C#N)N 7C-047 c1c(cc(c(c1[N+](=O)[O-])N2CCNCC2)[N+](=O)[O-])C(F)(F)F 7C-048 COC(=O)c1c(nc(s1)N2CCN(CC2)Cc3ccccc3)N 7C-049 CC(=O)C(C(c1ccc(cc1)Cl)Br)Br 7C-050 Cc1c(c(on1)C)Cc2ccc(cc2)O 7C-052 CC(=O)/C(=C/c1ccc(cc1)Cl)/Br 7C-061 CS/C(=N\C#N)/N1CCN(CC1)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 7C-064 CN(C)c1c(cc(s1)C(=O)c2ccccc2)c3ccccc3 7C-066 CS/C(=C\[N+](=O)[O-])/N1CCN(CC1)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 7C-068 c1ccc(cc1)C(=O)c2ccnc(n2)N 7C-077 CC(=O)c1cc(c(s1)N(C)C)c2ccccc2 7C-085 CS/C(=C\[N+](=O)[O-])/N1CCN(CC1)Cc2ccccc2 7C-086 CS/C(=N\C#N)/N1CCN(CC1)c2ccc(cc2)Cl 7C-087 CN(C)c1c(cc(s1)C#N)c2ccccc2 7C-088 CS/C(=N\C#N)/N1CCN(CC1)c2cccc(c2)Cl 7C-089 COC(=O)c1c(nc(s1)N2CCN(CC2)c3ccc(cc3)Cl)N 7C-091 CN(C)/C=N/c1c(sc(n1)N2CCN(CC2)c3ccc(cc3)Cl)C(=O)OC 7C-094 Cc1cccc(c1N2CCN(CC2)/C(=N/C#N)/SC)C 7C-106 c1csc(c1Cl)C(=O)N 7C-110 CS/C(=N\C#N)/N1CCN(CC1)C(c2ccccc2)c3ccccc3 7C-111 c1c(cc(cc1Cl)Cl)N2CCCC2=O 7C-116 Cc1c(cc2c(=O)c3cc(ccc3oc2n1)F)C(=O)OCc4ccccc4 7C-124 c1ccc(cc1)/C=C(\c2ccnn2S(=O)(=O)c3ccc(cc3Cl)Cl)/Oc4ccc(cc4)Cl 7C-125 CS/C(=N\C#N)/N1CCN(CC1)c2ccccn2 7C-126 Cc1ccc(cc1C)N2CCCC2=O 7C-127 CS/C(=N\C#N)/N1CCN(CC1)/C(=N/C#N)/SC 7C-129 c1cc(ccc1C(F)(F)F)N2CCCC2=O 7C-131 COc1ccc(cc1)N2CCN(CC2)/C(=N/C#N)/SC 7C-132 c1ccc(cc1)/C=C(\c2ccnn2S(=O)(=O)c3ccccc3Cl)/Oc4ccc(cc4)Cl 7C-139 Cc1c(c(ns1)S(=O)(=O)Cc2c(cccc2Cl)F)C#N 7C-141 Cc1c(c(ns1)S(=O)(=O)Cc2ccc(cc2)Cl)C#N 7C-144 Cc1ccc(cc1)CS(=O)(=O)c2c(c(sn2)C)C#N 7C-145 C1CN(CCN1c2[nH]nc(n2)N)c3[nH]nc(n3)N 7C-146 c1cc(ccc1N2CCCC2=O)[N+](=O)[O-] 7C-147 CN(C)/C=C\1/CCN(C1=O)c2cc(cc(c2)Cl)Cl 7C-148 c1cc(ccc1N2CCCC2=O)OC(F)(F)F 7C-149 CN(C)/C=C\1/CCN(C1=O)c2ccc(cc2)C(F)(F)F 7C-150 CN(C)/C=C\1/CCN(C1=O)c2ccc(cc2)[N+](=O)[O-] 7C-151 c1cc(ccc1C2=C(C(=O)OC2)C#N)Cl 7D-002 CN(C)/C=C/1\C(=C(C(=O)O1)C#N)c2ccc(cc2)Cl 7D-004 Cc1c(c(nc(n1)N)Sc2ccc(cc2)Cl)Cl 7D-005 Cc1c(c(nc(n1)N)SCc2ccccc2Cl)Cl 7D-006 Cc1ccc(cc1)COc2ccsc2C(=O)OC 7D-007 COC(=O)c1c(ccs1)OCc2ccc(cc2Cl)Cl 7D-008 Cc1c(c(nc(n1)N)SCC(=O)NC)Cl 7D-009 c1ccc(cc1)COc2ccsc2C(=O)NN 7D-010 c1ccc(cc1)/C=C\2/C(=C(C(=O)O2)C#N)c3ccc(cc3)Cl 7D-011 Cc1ccc(cc1)COc2ccsc2C(=O)NN 7D-015 c1cc(c(cc1Cl)Cl)COc2ccsc2C(=O)NN 7D-019 CNC(=S)NNC(=O)c1c(ccs1)OCc2ccccc2 7D-020 Cc1ccc(cc1)COc2ccsc2C(=O)NNC(=S)NC 7D-021 c1ccc(cc1)Cc2c3ccccc3c(=O)[nH]n2 7D-022 CNC(=S)NNC(=O)c1c(ccs1)OCc2ccc(cc2Cl)Cl 7D-024 Cn1c(nnc1S)c2c(ccs2)OCc3ccccc3 7D-028 Cc1ccc(cc1)COc2ccsc2c3nnc(n3C)S 7D-029 Cc1ccc(cc1)COc2ccsc2C(=O)O 7D-030 CC(=O)C(=NNc1ccccc1)C(=O)C 7D-032 Cc1ccc(cc1)COc2ccsc2c3nnc(n3C)SC 7D-034 Cn1c(nnc1SC)c2c(ccs2)OCc3ccccc3 7D-035 CN(C)c1c(c(c(s1)C(=O)OC)N)C#N 7D-036 Cn1c(nnc1S)c2c(ccs2)OCc3ccc(cc3Cl)Cl 7D-037 CN(C)C(=C(C#N)C#N)Sc1cccc[nH+]1.[OH-] 7D-038 Cn1c(nnc1SC)c2c(ccs2)OCc3ccc(cc3Cl)Cl 7D-039 CN(C)c1nnnn1c2ccc(cc2)Oc3ccccc3 7D-040 CN(C)c1c(c(nc(n1)N)N)C#N 7D-043 c1ccc2c(c1)nc3n2cc(c(c3C#N)N)c4ccc(cc4)F 7D-045 Cc1ccc(cc1)COc2ccsc2C(=O)NNC(=S)N 7D-046 COC(=O)c1c(ccs1)OCc2cccc(c2)C(F)(F)F 7D-048 CN(C)/C=C(\C#N)/C(=O)N/N=C/c1ccc(cc1)Cl 7D-049 c1cc(ccc1Sc2c(n3ccsc3n2)[N+](=O)[O-])Cl 7D-050 c1cc(cc(c1)Sc2c(n3ccsc3n2)[N+](=O)[O-])C(F)(F)F 7D-051 Cc1c(c(nc(n1)NC(=O)C)Cl)Cl 7D-052 c1cc(cc(c1)C(F)(F)F)COc2ccsc2C(=O)NN 7D-053 CN(C)/C=C(\C#N)/C(=O)N/N=C/c1ccc(cc1)F 7D-054 c1cc(c(cc1Cl)Cl)COc2ccsc2C(=O)O 7D-058 CN(C)c1nnnn1c2ccc(cc2)Cl 7D-060 CN(C)CCCn1c(nnn1)N(C)C 7D-063 Cc1ccc(cc1)COc2ccsc2c3[nH]c(nn3)S 7D-066 CNC(=S)NNC(=O)c1c(ccs1)OCc2cccc(c2)C(F)(F)F 7D-067 Cn1c(nnc1S)c2c(ccs2)OCc3cccc(c3)C(F)(F)F 7D-068 CN(C)c1nnnn1C2CCCCC2 7D-070 COc1ccc(cc1)/C=N/NC(=O)CC#N 7D-071 c1cc(ccc1SC2=CCS(=O)(=O)C2)Cl 7D-073 CN(C)/C=C(\C#N)/C(=O)N/N=C/c1ccc(cc1Cl)Cl 7D-074 Cc1ccc(cc1)COc2cc(sc2C(=O)OC)OC 7D-075 c1cc(cc(c1)C(F)(F)F)COc2ccsc2C(=O)NNC(=S)N 7D-077 CN(C)/C=C(\C#N)/C(=O)N/N=C/c1ccc(cc1)OC 7D-078 CN(C)c1nnnn1c2ccc(cc2)S(=O)(=O)N(C)C 7D-079 CN(C)c1nnnn1c2ccc(cc2)OC 7D-080 Cn1c(nnc1SC)c2c(ccs2)OCc3cccc(c3)C(F)(F)F 7D-081 c1cc(c(cc1Cl)Cl)COc2ccsc2C(=O)NNC(=S)N 7D-082 c1cc(ccc1c2ncc(s2)C(=O)c3ccc(cc3)Br)Cl 7D-084 CN(C)/C=N/C(=S)Nc1ccccc1 7D-085 Cc1ccc(cc1)SC2=CCS(=O)(=O)C2 7D-086 c1ccc(cc1)C(=O)c2cnc(s2)Nc3ccccc3 7D-088 c1ccc(cc1)CSc2c(n3ccsc3n2)[N+](=O)[O-] 7D-089 c1cc(ccc1CSc2c(n3ccsc3n2)[N+](=O)[O-])Cl 7D-090 COC(=O)c1ccccc1Sc2c(n3ccsc3n2)[N+](=O)[O-] 7D-091 CC(C)Sc1c(n2ccsc2n1)[N+](=O)[O-] 7D-092 CC(C)(C)Sc1c(n2ccsc2n1)[N+](=O)[O-] 7D-093 c1ccc(c(c1)CSc2c(n3ccsc3n2)[N+](=O)[O-])Cl 7D-094 Cc1ccc(cc1)Sc2c(n3ccsc3n2)[N+](=O)[O-] 7D-095 c1ccc(cc1)Nc2ncc(s2)C(=O)c3ccc(cc3)Cl 7D-096 c1ccc(cc1)Nc2ncc(s2)C(=O)c3ccc(cc3)F 7D-098 CC(=O)c1cnc(s1)Nc2ccccc2 7D-099 c1ccc(cc1)Nc2ncc(s2)C(=O)c3ccc(cc3)Br 7D-105 c1cc(ccc1c2ncc(s2)C(=O)c3ccc(c(c3)Cl)Cl)Cl 7D-106 c1ccc(cc1)Nc2ncc(s2)C(=O)c3ccc(c(c3)Cl)Cl 7D-107 COC(=O)CSc1c(n2ccsc2n1)[N+](=O)[O-] 7D-108 c1csc2n1c(c(n2)N3CCOCC3)[N+](=O)[O-] 7D-109 c1ccc(cc1)Oc2c(n3ccsc3n2)[N+](=O)[O-] 7D-110 CCOC(=O)COc1ccsc1C(=O)OC 7D-111 CC(C)(C)C(=O)c1cnc(s1)Nc2ccccc2 7D-113 C[N+](=C/N=C(\Nc1ccccc1)/SC)C.[I-] 7D-116 c1cc(ccc1Oc2c(n3ccsc3n2)[N+](=O)[O-])Cl 7D-117 c1ccc(c(c1)Oc2c(n3ccsc3n2)[N+](=O)[O-])Cl 7D-118 c1cc(cc(c1)Oc2c(n3ccsc3n2)[N+](=O)[O-])C(F)(F)F 7D-119 c1cc(cc(c1)Cl)Oc2c(n3ccsc3n2)[N+](=O)[O-] 7D-120 c1cc(ccc1c2ncc(s2)C(=O)c3ccc(cc3Cl)Cl)Cl 7D-121 c1ccc(cc1)Nc2ncc(s2)C(=O)c3ccc(cc3Cl)Cl 7D-122 COc1ccc(cc1)Oc2c(n3ccsc3n2)[N+](=O)[O-] 7D-123 c1cc(ccc1[N+](=O)[O-])Oc2c(n3ccsc3n2)[N+](=O)[O-] 7D-124 c1ccc(cc1)CNc2c(n3ccsc3n2)[N+](=O)[O-] 7D-125 c1cc(ccc1CNc2c(n3ccsc3n2)[N+](=O)[O-])Cl 7D-126 c1ccc(cc1)Nc2[nH]ncn2 7D-127 c1ccc(c(c1)CNc2c(n3ccsc3n2)[N+](=O)[O-])Cl 7D-128 c1cc(cc(c1)Cl)CNc2c(n3ccsc3n2)[N+](=O)[O-] 7D-129 c1cc(ccc1c2ncc(s2)C(=O)c3ccc(cc3)F)Cl 7D-130 CNC(=S)/N=C/N(C)C 7D-131 c1cc(ccc1S(=O)(=O)C2=CCS(=O)(=O)C2)Cl 7D-132 c1ccc(cc1)c2ccc(cc2)C(=O)c3cnc(s3)c4ccc(cc4)Cl 7D-133 c1cc(c(cc1Cl)Cl)COc2ccsc2c3[nH]c(nn3)S 7D-134 CSc1[nH]c(nn1)c2c(ccs2)OCc3ccc(cc3Cl)Cl 7D-135 c1ccc(cc1)C2=C(C(=O)OC2)C#N 7D-136 Cc1ccc(cc1)S(=O)(=O)C2=CCS(=O)(=O)C2 7D-137 CNc1c(n2ccsc2n1)[N+](=O)[O-] 7D-138 CNc1ncc(s1)C(=O)c2ccc(cc2)Br 7D-139 c1ccc(cc1)c2ccc(cc2)C(=O)c3cnc(s3)c4ccccc4 7D-140 c1ccc(cc1)c2ncc(s2)C(=O)c3ccc(cc3)Br 7D-141 c1ccc(cc1)c2ncc(s2)C(=O)c3ccc(c(c3)Cl)Cl 7D-142 c1ccc(cc1)c2ncc(s2)C(=O)c3ccc(cc3Cl)Cl 7D-143 CN(C)S(=O)(=O)c1ccc(cc1)N/C=C\2/c3ccccc3C(=O)O2 7D-144 CN(C)S(=O)(=O)c1ccc(cc1)NCc2c3ccccc3c(=O)[nH]n2 7D-145 c1ccc(cc1)c2ccc(cc2)C(=O)c3cnc(s3)Nc4ccccc4 7D-146 c1ccc2c(c1)/C(=C/NC34CC5CC(C3)CC(C5)C4)/OC2=O 7D-147 CSc1nc([nH]n1)N/C=C\2/c3ccccc3C(=O)O2 7D-148 c1ccc2c(c1)/C(=C/N3CCN(CC3)c4ccc(cc4)Cl)/OC2=O 7D-149 c1cc2c(cc1[N+](=O)[O-])CS(=O)(=O)O2 7E-001 Cc1ccc(cc1)C(C#N)c2ccc(nn2)Cl 7E-003 c1ccc(c(c1)CC[N+](=O)[O-])C(=O)N 7E-005 Cc1cccc(c1)C(C#N)c2ccc(nn2)Cl 7E-007 c1cc(nc(c1)F)NNc2ncc(cn2)C#N 7E-009 Cc1cccc(c1)Cc2ccc(nn2)O 7E-010 c1cc(nnc1Nn2cnc3ccsc3c2=O)Cl 7E-011 CC(=O)c1ccccc1Oc2c(cc(cn2)C(F)(F)F)Cl 7E-012 CN(c1ccc(nn1)Cc2ccc(cc2Cl)Cl)N 7E-013 CSc1nc2nccc(n2n1)/C=C\c3cccs3 7E-015 Cc1cccc(c1)Cc2ccc(nn2)Cl 7E-016 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)/OC2=O 7E-017 Cc1ccc(cc1)Cc2ccc(nn2)O 7E-018 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl 7E-019 COc1ccc(cc1)S(=O)(=O)CS(=O)(=O)C(F)(F)F 7E-020 c1cc(c(cc1Cl)Cl)COn2cnc3ccsc3c2=O 7E-021 Cc1ccc(cc1)Cc2ccc(nn2)Cl 7E-023 CC(=O)c1cccc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl 7E-024 c1cc(ccc1CONc2ncc(cn2)C#N)Cl 7E-031 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3)O 7E-032 c1cc(cc(c1)Cl)C(C#N)c2ccc(nn2)Cl 7E-033 Cc1ccc(cc1)Cc2ccc(nn2)NN 7E-035 c1ccc(c(c1)C(C#N)c2ccc(nn2)Cl)Cl 7E-036 c1cc(ccc1CONc2ncc(cn2)C#N)[N+](=O)[O-] 7E-037 c1ccc2c(c1)/C(=C/Nc3ccccc3O)/OC2=O 7E-038 c1cc(c(cc1Cl)Cl)CONc2ncc(cn2)C#N 7E-039 COc1ccc(cc1)Oc2ncc(cn2)C#N 7E-042 c1cc(cc(c1)Cl)Cc2ccc(nn2)O 7E-045 c1cc(ccc1C(C#N)c2ccc(nn2)Cl)Cl 7E-046 c1ccc(c(c1)Cc2ccc(nn2)O)Cl 7E-047 c1cc(cc(c1)Cl)Cc2ccc(nn2)Cl 7E-048 c1cc(ccc1Cc2ccc(nn2)O)Cl 7E-049 c1ccc(c(c1)Cc2ccc(nn2)Cl)Cl 7E-050 c1cc(ccc1F)Sc2ncc(cn2)C#N 7E-052 c1cc(cc(c1)Cl)Cc2ccc(nn2)NN 7E-057 c1cc(ccc1Cc2ccc(nn2)Cl)Cl 7E-058 c1cc(c(c(c1)Cl)COn2cnc3ccsc3c2=O)Cl 7E-059 c1cc(ccc1COn2cnc3ccsc3c2=O)Cl 7E-060 c1ccc(c(c1)Cn2cc(ccc2=O)C(=O)O)Cl 7E-302S COC(=O)c1c(ccs1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3)Cl 7E-303S c1cc(ccc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)C(F)(F)F)C(F)(F)F 7E-304S c1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3ccc(cc3)C(F)(F)F 7E-305S c1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3c(cccc3Cl)Cl 7E-306S c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3F)F)Cl 7E-307S c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)Cl)Cl 7E-308S CN(C)CCNC(=O)c1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 7E-309S c1cc(cc(c1)NC(=O)c2ccc(=O)n(c2)Cc3c(cccc3Cl)Cl)C(F)(F)F 7E-310S c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)OC(F)(F)F)Cl 7E-311S c1ccc(cc1)CNC(=O)c2ccc(=O)n(c2)Cc3c(cccc3Cl)Cl 7E-312S c1cc(ccc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3F)F)C(F)(F)F 7E-313S c1cc(ccc1Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F 7E-314S COC(=O)c1ccc(=O)n(c1)Cc2ccccc2 7E-316S CN(C)CCCNC(=O)c1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 7E-317S c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)NCCN3CCOCC3)Cl 7E-318S CCCNC(=O)c1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 7E-319S CCN(CC)C(=O)c1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 7E-320S c1ccc(cc1)CNC(=O)c2cccn(c2=O)Cc3cccc(c3)Cl 7E-321S c1cc(cc(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3nccs3 7E-322S c1cc(cc(c1)Cl)Cn2cccc(c2=O)C(=O)Nc3cccnc3 7E-323S c1cc(ccc1Cn2cc(ccc2=O)C(=O)O)Cl 7E-327S c1ccc(cc1)NC(=O)c2ccc(=O)n(c2)Cc3cccc(c3)Cl 7E-328S c1cc(cc(c1)Cl)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3F)F 7E-329S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)O 7E-330S C=CCNC(=O)c1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 7E-332S c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)N3CCCC3)Cl 7E-333S c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)NC3CC3)Cl 7E-334S CONC(=O)c1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 7E-335S c1c(c[nH]c(=O)c1C(=O)O)Cl 7E-336S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)NCCN3CCOCC3 7E-338S CN(C)S(=O)(=O)Nc1ccncc1 7E-341S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)C(F)(F)F 7E-342S CN(c1ccccc1)C(=O)c2ccc(=O)n(c2)Cc3c(cccc3Cl)Cl 7E-343S c1cc(cc(c1)C(F)(F)F)CNC(=O)c2ccc(=O)n(c2)Cc3c(cccc3Cl)Cl 7E-344S COC(=O)c1cccn(c1=O)Cc2c(cccc2Cl)F 7E-347S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)Nc3ccccc3 7E-348S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3)OC(F)(F)F 7E-349S c1cc(c(c(c1)Cl)Cn2cccc(c2=O)C(=O)O)F 7E-350S COC(=O)c1cc(cn(c1=O)Cc2ccc(c(c2)Cl)Cl)Cl 7E-352S COC(=O)c1cc(c(=O)[nH]c1)Cl 7E-353S c1cc(c(cc1Cn2cc(cc(c2=O)C(=O)O)Cl)Cl)Cl 7E-355S C=CCNC(=O)c1ccc(=O)n(c1)Cc2ccccc2 7E-358S Cc1c(snn1)S(=O)(=O)c2ccc(cc2)Cl 7E-359S c1ccc(cc1)Cn2cc(ccc2=O)C(=O)Nc3ccc(cc3F)F 7E-362S c1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3ccc(c(c3)Cl)Cl)Cl 7E-364S c1cc(c(cc1Cn2cc(cc(c2=O)C(=O)Nc3ccc(cc3F)F)Cl)Cl)Cl 7E-365S c1cc(cc(c1)NC(=O)c2cc(cn(c2=O)Cc3ccc(c(c3)Cl)Cl)Cl)C(F)(F)F 7E-366S Cc1cccc(c1NC(=O)c2cc(cn(c2=O)Cc3ccc(c(c3)Cl)Cl)Cl)C 7E-367S Cc1c(snn1)S(=O)(=O)c2cccc(c2)C(F)(F)F 7E-368S CNC(=O)c1cc(cn(c1=O)Cc2ccc(c(c2)Cl)Cl)Cl 7E-369S c1cc(c(cc1Cn2cc(cc(c2=O)Cl)C(=O)O)Cl)Cl 7E-370S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3c(cccc3Cl)F 7E-372S CN(C)CCNC(=O)c1cc(cn(c1=O)Cc2ccc(c(c2)Cl)Cl)Cl 7E-374S Cc1c(snn1)S(=O)c2ccccc2Cl 7E-375S Cc1c(snn1)S(=O)(=O)c2ccccc2 7E-376S CN(C)S(=O)(=O)N1CCN(CC1)c2ccccc2 7E-377S CN(C)S(=O)(=O)N1CC[NH+](CC1)c2ccccc2Cl.[Cl-] 7E-378S CN(C)S(=O)(=O)N1CCN(CC1)c2cccc(c2)Cl 7E-379S c1cc(cc(c1)NC(=O)c2cccn(c2=O)Cc3c(cccc3Cl)F)C(F)(F)F 7E-380S c1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl 7E-381S CN(C)S(=O)(=O)N1CCN(CC1)c2ccc(cc2)Cl 7E-382S CN(C)S(=O)(=O)N1CCN(CC1)c2ccc(cc2)F 7E-383S CN(C)S(=O)(=O)N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 7E-384S CN(C)S(=O)(=O)N1CC[NH+](CC1)Cc2ccccc2.[Cl-] 7E-385S CN(C)S(=O)(=O)N1CCN(CC1)Cc2ccc3c(c2)OCO3 7E-386S CN(C)S(=O)(=O)N1CCN(CC1)c2ccccn2 7E-387S c1cc(c(cc1Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3F)F)Cl)Cl 7E-388S CN(C)CCNC(=O)c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)Cl 7E-389S CCN(CC)C(=O)c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)Cl 7E-390S CNC(=O)c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)Cl 7E-391S COC(=O)c1cc(cn(c1=O)Cc2c(cccc2Cl)Cl)Cl 7E-392S C[NH+]1CCN(CC1)S(=O)(=O)N(C)C.[Cl-] 7E-393S Cc1cccc(c1[NH+]2CCN(CC2)S(=O)(=O)N(C)C)C.[Cl-] 7E-394S CN(C)S(=O)(=O)N1CCN(CC1)c2ccc(cc2)OC 7E-395S c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)C(=O)O)Cl)Cl 7E-396S CN(C)S(=O)(=O)N1CCN(CC1)c2ncccn2 7E-397S c1ccc(cc1)CNC(=O)c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl 7E-398S c1cc(ccc1NC(=O)c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl)Cl 7E-399S COC(=O)c1cc(c(=O)n(c1)Cc2c(cccc2Cl)Cl)Cl 7E-400S Cc1c(snn1)S(=O)(=O)c2cccc(c2)Cl 7E-401S CN(c1ccccc1)C(=O)c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl 7E-402S c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)O)Cl 7E-405S Cc1c(snn1)S(=O)(=O)Cc2ccccc2Cl 7E-406S Cc1c(snn1)S(=O)(=O)Cc2ccccc2 7E-407S C=CCNC(=O)c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)Cl 7E-408S Cc1c(snn1)S(=O)(=O)Cc2ccc(cc2)Cl 7E-410S CNC(=O)c1cc(c(=O)n(c1)Cc2c(cccc2Cl)Cl)Cl 7E-411S c1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)Cl 7E-412S c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3F)F)Cl 7E-413S CN(C)S(=O)(=O)N1CCN(CC1)CCc2ccccc2C(F)(F)F 7E-414S COC(=O)Nc1ccc(=O)n(c1)Cc2c(cccc2Cl)Cl 7E-505 c1cc(c(cc1Cn2cc(ccc2=O)N)Cl)Cl 7E-508 c1cc(c(cc1Cn2cc(ccc2=O)NC(=O)c3ccc(c(c3)Cl)Cl)Cl)Cl 7E-510 c1cc(c(cc1Cn2cc(ccc2=O)NC(=O)c3ccc(cc3Cl)Cl)Cl)Cl 7E-511 c1ccc(c(c1)C(=O)Nc2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)[N+](=O)[O-] 7E-512 c1ccc(cc1)S(=O)(=O)Nc2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 7E-514 c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)N 7E-516 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 7E-517 c1cc(ccc1S(=O)(=O)Nc2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl 7E-518 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl 7E-520 c1ccc(c(c1)S(=O)(=O)Nc2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl 7E-521 c1cc(cc(c1)S(=O)(=O)Nc2ccc(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)C(F)(F)F 7E-522 c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)NC(=O)c3ccc(c(c3)Cl)Cl 7E-523 Cc1ccc(cc1)C(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 7E-525 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 7E-526 c1ccc(c(c1)C(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl)[N+](=O)[O-] 7E-528 COc1ccc(cc1)C(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 7E-529 c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)NC(=O)C3CC3 7E-531 CC(C)(C)C(=O)Nc1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 7E-532 c1ccc(cc1)S(=O)(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 7E-540 Cc1ccc(cc1)S(=O)(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl 7E-542 c1cc(c(=O)n(c1)Cc2ccc(c(c2)Cl)Cl)NS(=O)(=O)c3ccc(cc3)Cl 7E-543 c1cc(cc(c1)S(=O)(=O)Nc2cccn(c2=O)Cc3ccc(c(c3)Cl)Cl)C(F)(F)F 7E-544 C=CCNC(=S)Nc1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 7E-547 CCCCC(=O)Nc1cccn(c1=O)Cc2ccc(c(c2)Cl)Cl 7E-551 c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(F)(F)F)Cl 7E-558 c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)[N+](=O)[O-])C(F)(F)F)Cl 7E-559 Cc1ccc(cc1)C(=O)Oc2cccnc2I 7E-900 Cc1cc(c(c(=O)o1)/C(=N/Nc2ccccc2)/C)O 7E-901 Cc1cc(c(c(=O)o1)/C(=N/NC(=S)N)/C)O 7E-902 Cc1c(c(n(n1)c2ccccc2)O)C(=O)/C=C(\C)/O 7E-903 c1ccc(cc1)NC(=O)Oc2cccnc2I 7E-904 Cc1cc(n(n1)c2ccccc2)c3c(nn(c3O)c4ccccc4)C 7E-906 Cc1c(c(n(n1)c2nc(cs2)c3ccc(cc3)Cl)O)C(=O)/C=C(/C)\O 7E-909 c1cc(cc(c1)Cl)C(=O)Nc2cc3c(oc2=O)CCCC3=O 7E-910 Cc1cc([nH]n1)c2c(nn(c2O)c3ccccc3)C 7E-912 Cc1cc(n(n1)c2ccccc2)c3c(nn(c3O)c4nc(cs4)c5ccc(cc5)Cl)C 7E-913 Cc1c(cc(c(=O)o1)NC(=O)c2cccc(c2)Cl)C(=O)C 7E-914 Cc1c(cc(c(=O)o1)NC(=O)c2cccc(c2)Cl)C(=O)OC 7E-915 Cc1c(cc(c(=O)o1)NC(=O)c2cccc(c2)Cl)C(=O)c3ccccc3 7E-916 CCOC(=O)c1cc(c(=O)oc1c2ccccc2)NC(=O)c3cccc(c3)Cl 7E-917 Cc1ccc(cc1)C(=O)Nc2cc(c(oc2=O)C)C(=O)OC 7E-918 CCOC(=O)c1cc(c(=O)oc1c2ccccc2)NC(=O)c3ccc(cc3)C 7E-919 CN(C)C=C(C(=O)Nc1ccccc1)C(=O)Nc2ccccc2 7E-920 Cc1ccc(cc1)C(=O)Nc2cc(c(oc2=O)C)C(=O)C 7E-921 Cc1ccc(cc1)C(=O)Nc2cc3c(oc2=O)CCCC3=O 7E-923 c1ccc(cc1)NC(=O)C(/C=N/OCc2ccc(cc2Cl)Cl)C(=O)Nc3ccccc3 7E-929 CC(=O)Nc1ccc(cc1)NC(=O)CC2(C3CC4CC(C3)CC2C4)C 7E-933 c1ccc2c(c1)cc(o2)C(=O)Nc3cccc(c3)C(F)(F)F 7E-934 CC1(C2CC3CC(C2)CC1C3)CC(=O)Oc4ccccc4 7E-936 CC1(C2CC3CC(C2)CC1C3)CC(=O)OCc4ccccc4 7E-938 c1ccc2c(c1)c(ncn2)N/N=C/c3ccc(cc3Cl)Cl 7E-939 c1ccc2c(c1)c3nnc(n3cn2)c4ccc(cc4Cl)Cl 7E-942 CCOC(=O)c1cc(c(=O)oc1C(F)(F)F)NC(=O)c2ccc(cc2)C 7E-945 Cc1cc(c(c(=O)o1)/C(=N/Nc2nc(cs2)c3ccccc3)/C)O 7E-946 Cc1ccc(cc1)C(=O)Nc2cc3ccc(cc3oc2=O)O 7E-947 C/C(=N/Oc1c(cc(cn1)C(F)(F)F)Cl)/c2ccccc2 7F-001 Cc1cc(nc(n1)O/N=C(/C)\c2ccc(cc2)F)C 7F-002 c1cc(ccc1c2csc(n2)Cn3cncn3)Cl 7F-003 c1ncn(n1)CC(=S)N 7F-004 c1cc(c(cc1Cl)Cl)C(=O)O/N=C(/Cn2cncn2)\N 7F-006 CCOC1C(CCCO1)C(OCC)OCC 7F-009 CC(C)(c1nnc(n1C)SCc2ccc(cc2)Cl)n3cncn3 7F-010 COC(=O)c1c(ccs1)OCc2ccc(cc2)Cl 7F-011 CC(C)(C(=O)NNC(=S)NC)n1cncn1 7F-012 C1CC(=COC1)C=O 7F-013 Cn1cccc1/C(=C/c2ccc(cc2)Cl)/C#N 7F-014 c1cc(ccc1COc2ccsc2C(=O)NN)Cl 7F-015 CN(C)/C=C(\C#N)/c1ccc(cc1Cl)Cl 7F-017 c1cc(c(cc1Cl)Cl)/C(=C/O)/C#N 7F-018 Cn1c(c(c(c1C(=O)C(Cl)(Cl)Cl)C(=O)c2ccc(cc2Cl)Cl)C(=O)c3ccc(cc3Cl)Cl)CC#N 7F-020 CO/C(=C/c1ccc(o1)c2cccc(c2)Cl)/c3ccccc3 7F-022 CO/C(=C/c1ccc(o1)c2ccccc2Cl)/c3ccccc3 7F-023 COC(=O)Nc1c(ccs1)OCc2ccc(cc2)Cl 7F-026 c1ccc(cc1)COc2ccsc2NC(=O)Nc3ccccc3 7F-028 CO/C(=C/c1ccc(o1)c2ccccc2)/c3ccccc3 7F-029 COC(=O)c1c(ccs1)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 7F-030 c1ccnc(c1)C(=N)NNC(=O)c2c(ccs2)OCc3ccc(cc3Cl)Cl 7F-031 COC(=O)Nc1c(ccs1)OCc2cccc(c2)C(F)(F)F 7F-033 c1ccc(cc1)COc2ccsc2NC(=O)Nc3c(ccs3)OCc4ccccc4 7F-034 c1cc(c(cc1Cl)Cl)COc2ccsc2C(=O)NNC(=N)Cn3cncn3 7F-037 c1cc(c(cc1Cl)Cl)COc2ccsc2C(=O)N=N#N 7F-040 c1cc(ccc1COc2ccsc2C(=O)O)Cl 7F-042 c1cc(cc(c1)C(F)(F)F)COc2ccsc2C(=O)O 7F-044 CC(C)(c1nnc(n1C)Sc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)n4cncn4 7F-049 c1ccc(cc1)NC(=O)Nc2c(ccs2)OCc3ccc(cc3Cl)Cl 7F-050 CCOC(=O)Cc1[nH]c(nn1)c2ccc(cc2)Cl 7F-052 c1cc(cnc1)C(=N)NNC(=O)c2c(ccs2)OCc3ccc(cc3Cl)Cl 7F-054 CCOC(=O)C(CC(=O)c1ccc(cc1)Cl)(C(=O)OCC)O 7F-055 c1ccc2c(c1)nc(n2O)c3c(cccc3Cl)F 7F-301S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)Br)Cl)Cl)Cl 7F-302S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)C(F)(F)F)Cl)Cl)Cl 7F-303S c1cc(c(cc1CS(=O)(=O)CC(CN2CCCC2=O)O)Cl)Cl 7F-304S Cc1ccc(cc1)c2nc3ccccc3n2OCc4ccc(cc4Cl)Cl 7F-307S Cc1ccc(cc1)c2nc3ccccc3n2OCc4ccccc4Cl 7F-308S Cc1ccc(cc1)c2nc3ccccc3n2OCc4c(cccc4Cl)F 7F-309S COc1ccc(cc1)c2nc3ccccc3n2O 7F-311S COc1ccc(cc1)c2nc3ccccc3n2OCc4c(cccc4Cl)Cl 7F-312S COc1ccc(cc1)c2nc3ccccc3n2OCc4ccc(c(c4)Cl)Cl 7F-314S c1cc(ccc1c2c3ccc(cc3c(=O)n(n2)c4ccc(cc4)Br)F)F 7F-315S c1cc(ccc1c2c3ccc(cc3c(=O)n(n2)c4ccc(cc4)Cl)F)F 7F-316S c1cc(ccc1c2c3ccc(cc3c(=O)n(n2)c4ccc(cc4)OC(F)(F)F)F)F 7F-317S c1cc(ccc1c2c3ccc(cc3c(=O)n(n2)c4ccc(cc4)F)F)F 7F-318S c1cc(ccc1c2c3ccc(cc3c(=O)n(n2)c4ccc(cc4)C(F)(F)F)F)F 7F-319S COc1ccc(cc1)c2nc3ccccc3n2OCc4ccccc4Cl 7F-320S COc1ccc(cc1)c2nc3ccccc3n2OCc4cccc(c4)Cl 7F-321S COc1ccc(cc1)c2nc3ccccc3n2OCc4ccc(cc4)Cl 7F-322S COc1ccc(cc1)c2nc3ccccc3n2OCc4c(cccc4Cl)F 7F-324S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)F)Cl)Cl)F 7F-326S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)Cl)Cl)Cl)F 7F-327S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)OC(F)(F)F)Cl)Cl)F 7F-328S Cc1ccc(cc1)COn2c3ccccc3nc2c4ccc(cc4)OC 7F-329S Cc1cc(cc(c1)COn2c3ccccc3nc2c4ccc(cc4)OC)C 7F-330S COc1ccc(cc1)c2nc3ccccc3n2OCc4cccc(c4)C(F)(F)F 7F-331S c1ccc(c(c1)c2nc3ccccc3n2OCc4cccc(c4)Cl)Cl 7F-332S c1cc(ccc1c2c3cc(c(cc3c(=O)n(n2)c4ccc(cc4)C(F)(F)F)Cl)Cl)F 7F-333S CN(C)C(=O)On1c2ccccc2nc1c3ccc(cc3)OC 7F-335S c1ccc(cc1)c2nc3ccccc3n2OCC(=O)O 7F-337S c1cc(cc(c1)NC(=O)c2cc(cc(c2)Cl)Cl)C#N 7F-338S c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2ccc(cc2)Cl 7F-339S c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2cccc(c2)C(F)(F)F 7F-340S c1cc(cc(c1)NC(=N)c2cc(cc(c2)Cl)Cl)C#N 7F-341S c1cc(cc(c1)[N+](=O)[O-])C(=N)Nc2ccc(cc2)Cl 7F-342S c1ccc(c(c1)c2nc3ccccc3n2OCc4c(cccc4Cl)F)Cl 7F-343S c1cc(cc(c1)[N+](=O)[O-])C(=N)Nc2cccc(c2)C(F)(F)F 7F-344S c1ccc(cc1)COn2c3cccnc3nc2c4ccc(cc4)Cl 7F-345S c1cc2c(nc1)nc(n2O)c3ccc(cc3)Cl 7F-346S c1ccc(c(c1)COn2c3ccccc3nc2c4ccccc4Cl)Cl 7F-350S C/N=C(\c1cc(cc(c1)Cl)Cl)/Nc2cccc(c2)C#N 7F-351S c1cc(cc(c1)NC(=O)c2cccc(c2)C(F)(F)F)C#N 7F-352S c1cc(cc(c1)[N+](=O)[O-])C(=N)Nc2ccc(c(c2)Cl)Cl 7F-357S Cc1cc(cc(c1)C(=N)Nc2ccc(c(c2)Cl)Cl)C 7F-358S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2F)F)Sc3cccc(c3)C(F)(F)F 7F-360S c1ccc(c(c1)c2nc3ccccc3n2OCc4ccc(cc4Cl)Cl)Cl 7F-362S c1cc(cc(c1)C(F)(F)F)CNc2c(cccn2)[N+](=O)[O-] 7F-363S c1cc(cc(c1)C(F)(F)F)c2nc3c(n2O)cccn3 7F-364S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccc(c2)C(F)(F)F 7F-365S c1cc(cc(c1)Cl)COn2c3cccnc3nc2c4ccc(cc4)Cl 7F-366S c1cc(cc(c1)C(F)(F)F)COn2c3cccnc3nc2c4ccc(cc4)Cl 7F-367S Cc1ccc(cc1)CNc2c(cccn2)[N+](=O)[O-] 7F-368S Cc1ccc(cc1)c2nc3c(n2O)cccn3 7F-369S c1cc(cc(c1)NC(=N)c2cccc(c2)C(F)(F)F)C#N 7F-370S c1ccc(cc1)CNc2c(cccn2)[N+](=O)[O-] 7F-371S c1ccc(cc1)c2nc3c(n2O)cccn3 7F-372S c1ccc(cc1)COn2c3cccnc3nc2c4ccccc4 7F-373S Cc1ccc(cc1)COn2c3cccnc3nc2c4ccccc4 7F-374S c1cc(cc(c1)NC(=N)c2cccc(c2)[N+](=O)[O-])C#N 7F-375S COn1c2cccnc2nc1c3ccccc3 7F-377S c1ccc(cc1)c2nc3c(n2OCc4ccc(cc4)Cl)cccn3 7F-378S c1ccc(cc1)c2nc3c(n2OCc4ccc(cc4)Br)cccn3 7F-379S COc1ccc(cc1)COn2c3cccnc3nc2c4ccccc4 7F-380S C/N=C(\c1cc(cc(c1)Cl)Cl)/Nc2ccc(c(c2)Cl)Cl 7F-381S Cc1cc(cc(c1)/C(=N\C)/Nc2cccc(c2)C(F)(F)F)C 7F-382S c1ccc(cc1)c2nc3c(n2OCc4ccc(cc4Cl)Cl)cccn3 7F-383S c1ccc(cc1)c2nc3c(n2OCc4cccc(c4)C(F)(F)F)cccn3 7F-384S c1cc2c(nc1)nc(n2OCc3ccc(cc3Cl)Cl)c4ccc(cc4)Cl 7F-385S Cc1cc(cc(c1)COn2c3cccnc3nc2c4ccc(cc4)Cl)C 7F-386S COn1c2cccnc2nc1c3ccc(cc3)Cl 7F-387S C/N=C(\c1cc(cc(c1)Cl)Cl)/Nc2ccc(cc2)Cl 7F-388S CCOC(=O)c1ccccc1c2csc(n2)N 7F-900 CCOC(=O)c1ccccc1c2csc(n2)Nc3ccccc3 7F-901 CCOC(=O)c1ccccc1c2csc(n2)NC(=O)c3ccc(cc3)OC 7F-903 CCOC(=O)c1ccccc1c2csc(n2)c3ccccc3 7F-905 c1ccc(cc1)C(=O)OC2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 7F-907 Cc1ccc(cc1)C(=O)OC2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 7F-908 c1cc(ccc1C(=O)OC2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])Cl 7F-909 COc1ccc(cc1)C(=O)OC2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 7F-910 c1ccc(cc1)C(=O)ON=C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 7F-911 Cc1ccc(cc1)C(=O)ON=C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 7F-912 c1cc(ccc1C(=O)ON=C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])Cl 7F-913 COc1ccc(cc1)C(=O)ON=C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 7F-914 c1ccc-2c(c1)CCc3c2nc(nc3)NC(=O)c4ccc(cc4)Cl 7F-915 c1ccc(cc1)C2(C3CC4CC(C3)CC2C4)CC(=O)N5CCN(CC5)c6cccc(n6)Cl 7F-916 CCOC(=O)NC(=O)C(/C=N\OCCOc1cccc(c1)C(F)(F)F)C#N 7F-917 c1cc(cc(c1)OCCOn2cc(c(=O)[nH]c2=O)C#N)C(F)(F)F 7F-918 c1ccc(cc1)C2=N/C(=C/Nc3ncccn3)/C(=O)O2 7F-921 COC(=O)c1c(nc(s1)N)c2cccnc2 7F-922 CCOC(=O)c1ccccc1c2csc(n2)N/C=N/OCc3ccc(cc3)[N+](=O)[O-] 7F-924 c1ccnc(c1)N2CCN(CC2)C(=N)CC#N 7F-925 c1cc(ccc1N2CCC(=NO)CC2)[N+](=O)[O-] 7F-927 c1ccc(cc1)C2=N/C(=C/Nc3cnccn3)/C(=O)O2 7F-928 c1ccc(cc1)C(=O)c2cc(c([nH]2)N3CCN(CC3)c4ccccn4)C#N 7F-929 c1cc(ccc1NCc2c(snn2)Cl)Cl 7F-930 c1cc(ccc1C(F)(F)F)NCc2c(snn2)Cl 7F-931 Cc1ccnc(n1)/N=C/N(C)C 7F-933 Cc1ccnc(n1)N/C=C/2\C(=O)OC(=N2)c3ccccc3 7F-934 CCN(CC)C(=O)/C(=C\Nc1ncccn1)/NC(=O)c2ccccc2 7F-935 Cc1ccnc(n1)N/C=C(\C(=O)NN)/NC(=O)c2ccccc2 7F-936 c1ccc(cc1)C(=O)NCC(=O)Nc2ccsc2C(=O)O 7F-938 c1cc(ccc1NCc2c(snn2)Cl)OC(F)(F)F 7F-940 Cc1ccnc(n1)N/C=C(\C(=O)N/N=C\N(C)C)/NC(=O)c2ccccc2 7F-942 c1c(cnc(c1Cl)C(C(=O)N2CCOCC2)C(=O)N3CCOCC3)C(F)(F)F 7G-001 c1ccc(cc1)/C(=C(\c2ccccc2)/c3ccccc3Cl)/C#N 7G-002 Cc1cc(n(n1)c2nnc(nn2)NCCc3ccccc3)C 7G-003 c1cc(ccc1N/C=C/2\CCN(C2=O)c3c(cc(cn3)C(F)(F)F)Cl)Cl 7G-004 COC(=O)C1=C(c2c(cccc2F)C1(C#N)c3ccccc3)N 7G-005 CO/N=C/C1CCN(C1=O)c2c(cc(cn2)C(F)(F)F)Cl 7G-006 c1cc(ccc1C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NC(=O)Nc3ccc(cc3)Cl)Cl 7G-008 c1cc(ccc1C(=O)c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 7G-009 C/C(=C\C(=O)C(F)(F)F)/NCC(=O)c1ccccc1 7G-010 c1ccc(cc1)C2(CC(=O)c3c2cccc3F)C(=O)O 7G-011 c1ccc(cc1)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 7G-012 Cc1cc(c([nH]1)C(=O)c2ccccc2)C(F)(F)F 7G-013 c1ccc(cc1)C2CC(=O)c3c2cccc3F 7G-014 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)OC 7G-015 CN(C)/C=C(\C=O)/c1c(cc(cn1)C(F)(F)F)Cl 7G-016 c1ccc(cc1)NC(=O)c2cccnc2Cl 7G-017 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NN 7G-018 CN(C)/C=C\1/C(c2cccc(c2C1=O)F)c3ccccc3 7G-019 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)OCc2ccccc2 7G-021 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)OCc2ccccc2Cl 7G-022 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NC 7G-023 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NC2CC2 7G-024 c1cc(sc1)Cc2c(cc(cn2)C(F)(F)F)Cl 7G-025 c1cc(ccc1/C(=N\N)/c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 7G-026 c1ccnc(c1)Cc2c(cc(cn2)C(F)(F)F)Cl 7G-027 c1c(cnc(c1Cl)c2cnc(nc2)N)C(F)(F)F 7G-028 c1ccc(cc1)C(C#N)c2ccc(c(n2)Cl)C(F)(F)F 7G-029 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NNC(=S)Nc2ccccc2 7G-030 c1ccc(c(c1)C#N)C(C#N)n2cncn2 7G-031 CC(c1c(cc(cn1)C(F)(F)F)Cl)c2nnc(n2c3ccccc3)S 7G-033 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NNC(=S)NC 7G-034 c1ccc(cc1)C(=O)c2ccc(cc2)C(CCC#N)(C#N)c3ccccc3 7G-035 CC(c1c(cc(cn1)C(F)(F)F)Cl)c2nnc(n2c3ccccc3)SC 7G-036 CC(c1c(cc(cn1)C(F)(F)F)Cl)c2nnc(n2c3ccccc3)SCC=C 7G-037 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NCC#C 7G-038 CC(c1c(cc(cn1)C(F)(F)F)Cl)c2nnc(n2C)S 7G-039 CC(c1c(cc(cn1)C(F)(F)F)Cl)c2nnc(n2C)SC 7G-040 CC(c1c(cc(cn1)C(F)(F)F)Cl)c2nnc(n2C)SCC=C 7G-041 c1ccc(cc1)C(=O)c2ccc(cc2)C3(CCC(=O)NC3=O)c4ccccc4 7G-042 Cc1cc2ncc(cn2n1)C#N 7G-043 CN(C)/C=N/c1ncc(cn1)c2c(cc(cn2)C(F)(F)F)Cl 7G-044 Cc1c(c2ncc(cn2n1)C#N)Br 7G-045 COc1ccc(cc1)Cc2c(cc(cn2)C(F)(F)F)Cl 7G-046 c1cc(ccc1c2cn[nH]c2N)Cl 7G-047 CO/N=C/Nc1ncc(cn1)c2c(cc(cn2)C(F)(F)F)Cl 7G-052 c1c(cnc(c1Cl)N2CCC(C2=O)/C=N\O)C(F)(F)F 7G-053 COC(=O)CCC(C#N)(c1ccccc1)c2cccc(c2C#N)F 7G-054 c1cc(cc(c1)NC(=O)O/N=C(\c2c(cc(cn2)C(F)(F)F)Cl)/N)C(F)(F)F 7G-055 c1cc(ccc1CSc2c(cc(cn2)C#N)C#N)F 7G-056 c1c(cnc(c1Cl)NN/C=N/O)C(F)(F)F 7G-057 c1c(cnc(c1Cl)NNC#N)C(F)(F)F 7G-058 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)Cl 7G-060 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)O 7G-062 c1cc(cc(c1)Cl)Cc2c(cc(cn2)C(F)(F)F)Cl 7G-070 Cc1cccc(c1)Cc2c(cc(cn2)C(F)(F)F)Cl 7G-071 c1cc(ccc1F)SCCOc2ccc(cc2Cl)Cl 7G-301S Cc1ccc(cc1)SCCOc2ccc(cc2Cl)Cl 7G-302S CNC(=O)C(Oc1cccc(c1)C(F)(F)F)(F)F 7G-303S c1cc(cc(c1)OC(C(=O)Nc2cccnc2)(F)F)C(F)(F)F 7G-304S CCNc1nc(cc(n1)Cl)C(F)(F)F 7G-305S CCNc1nc(cc(n1)Sc2ccccc2)C(F)(F)F 7G-306S CCNc1nc(cc(n1)Sc2ccc(cc2)Cl)C(F)(F)F 7G-307S CCNc1nc(cc(n1)Sc2ccc(cc2)Br)C(F)(F)F 7G-308S c1ccc(cc1)S(=O)(=O)CCCS(=O)(=O)c2ccccc2 7G-310S Cc1ccc(cc1)S(=O)CCCS(=O)c2ccc(cc2)C 7G-311S Cc1ccc(cc1)S(=O)(=O)CCCS(=O)(=O)c2ccc(cc2)C 7G-312S Cc1ccc(cc1)C2=[N+](C(CC2)(C)C)[O-] 7G-313S CC1(CCC(=[N+]1[O-])c2ccc(cc2)F)C 7G-314S Cc1ccc(cc1)S(=O)CCOc2ccc(cc2Cl)Cl 7G-315S c1ccc(cc1)OCCCCSc2ccc(cc2)Cl 7G-316S Cc1c(c(nn1c2ccccc2)C(F)(F)F)O 7G-317S Cc1cc(ccc1OC(C(=O)Nc2ccccc2)(F)F)Cl 7G-319S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2)Cl)(F)F)Cl 7G-320S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2Cl)Cl)(F)F)Cl 7G-321S CCNc1nc(cc(n1)Oc2ccc(cc2)OC)C(F)(F)F 7G-322S CC(C)OC(=O)c1cccnc1N2CCN(CC2)c3cccc(c3)C(F)(F)F 7G-323S c1ccc(cc1)OCCCCS(=O)(=O)c2ccc(cc2)Cl 7G-324S Cc1cc(ccc1OC(C(=O)Nc2c(cccc2F)F)(F)F)Cl 7G-325S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2)OC(F)(F)F)(F)F)Cl 7G-326S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2)OC)(F)F)Cl 7G-327S Cc1c(c(nn1c2ccccc2)C(F)(F)F)OCc3ccc(cc3)Cl 7G-328S CCNc1nc(cc(n1)SCc2ccc(cc2)Cl)C(F)(F)F 7G-330S Cc1c(c(nn1c2ccccc2)C(F)(F)F)OCc3ccc(cc3Cl)Cl 7G-331S CCNc1nc(cc(n1)Oc2c(cccc2Cl)Cl)C(F)(F)F 7G-332S CCNc1nc(cc(n1)Sc2ccc(cc2)F)C(F)(F)F 7G-333S CCNc1nc(cc(n1)Sc2cccc(c2)Cl)C(F)(F)F 7G-334S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2)F)(F)F)Cl 7G-335S Cc1ccc(cc1Cl)NC(=O)C(Oc2ccc(cc2C)Cl)(F)F 7G-336S CC(C)Nc1nc(cc(n1)O)C(F)(F)F 7G-337S CCNc1nc(cc(n1)Sc2ccc(cc2Cl)Cl)C(F)(F)F 7G-338S CCNc1nc(cc(n1)Sc2ccc(cc2)C)C(F)(F)F 7G-341S c1ccc(cc1)SCCCSc2ccccn2 7G-343S CCNc1nc(cc(n1)SCc2ccc(c(c2)Cl)Cl)C(F)(F)F 7G-344S CCNc1nc(cc(n1)Sc2ccc(c(c2)Cl)Cl)C(F)(F)F 7G-345S c1ccc(cc1)c2c(=O)n(cc(n2)c3ccc(cc3)Cl)O 7G-347S CC(C)(C)c1ccc(cc1)Oc2cc(nc(n2)N(C)C)C(F)(F)F 7G-349S CNc1nc(cc(n1)OC(=O)N(C)C)C(F)(F)F 7G-350S c1ccc(cc1)c2c(=O)n(cc(n2)c3ccc(cc3)Br)O 7G-351S CCNc1nc(cc(n1)Oc2cc(cc(c2)Cl)Cl)C(F)(F)F 7G-352S CCNc1nc(cc(n1)Oc2ccc(cc2Cl)Cl)C(F)(F)F 7G-353S Cc1c(c(nn1c2ccccc2)C(F)(F)F)OCc3c(cccc3Cl)Cl 7G-354S CC(C)(C)c1ccc(cc1)CS(=O)(=O)CCOc2ccccc2 7G-355S CC(C)(C)c1ccc(cc1)CS(=O)(=O)CCCS(=O)(=O)c2ccccc2 7G-356S CCNc1nc(cc(n1)Oc2ccc(cc2)C#N)C(F)(F)F 7G-357S CC(C)Nc1nc(cc(n1)OC)C(F)(F)F 7G-359S CC(C)Nc1nc(cc(n1)Sc2ccc(cc2)F)C(F)(F)F 7G-360S CCNc1nc(cc(n1)SCc2ccc(cc2)C(C)(C)C)C(F)(F)F 7G-361S COC(=O)c1cccnc1N2CCN(CC2)c3ccccc3 7G-363S COC(=O)c1cccnc1N2CCN(CC2)c3cccc(c3)Cl 7G-365S COC(=O)c1cccnc1N2CCN(CC2)c3ccccc3Cl 7G-366S CC(C)OC(=O)c1ccc(nc1)N2CCN(CC2)c3ccccc3 7G-367S CC(C)OC(=O)c1ccc(nc1)N2CCN(CC2)c3ccc(cc3)F 7G-368S CC(C)OC(=O)c1ccc(nc1)N2CCN(CC2)c3ccccc3F 7G-369S CC(C)OC(=O)c1ccc(nc1)N2CCN(CC2)C(c3ccccc3)c4ccccc4 7G-370S CC(C)OC(=O)c1ccc(nc1)N2CCN(CC2)c3cccc(c3)Cl 7G-371S c1ccc(c(c1)N2CCN(CC2)c3ccc(cn3)C(=O)OCC(F)(F)F)F 7G-373S c1cc(ccc1N2CCN(CC2)c3ccc(cn3)C(=O)OCC(F)(F)F)F 7G-374S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ccc(cn4)C(=O)OCC(F)(F)F 7G-375S c1cc(cc(c1)Cl)N2CCN(CC2)c3ccc(cn3)C(=O)OCC(F)(F)F 7G-377S C=CCOC(=O)c1ccc(nc1)N2CCN(CC2)c3ccccc3F 7G-379S C=CCOC(=O)c1ccc(nc1)N2CCN(CC2)c3ccc(cc3)F 7G-380S C=CCOC(=O)c1ccc(nc1)N2CCN(CC2)c3cccc(c3)Cl 7G-381S C=CCOC(=O)c1ccc(nc1)N2CCN(CC2)c3ccccc3 7G-382S COC(=O)c1ccc(nc1)N2CCN(CC2)c3ccccc3 7G-383S COC(=O)c1ccc(nc1)N2CCN(CC2)c3ccccc3F 7G-384S COC(=O)c1ccc(nc1)N2CCN(CC2)c3ccccc3Cl 7G-386S COC(=O)c1ccc(nc1)N2CCN(CC2)c3cccc(c3)Cl 7G-387S CCNc1nc(cc(n1)Oc2ccc(cc2)F)C(F)(F)F 7G-389S CC(C)Nc1nc(cc(n1)Sc2ccc(cc2)Cl)C(F)(F)F 7G-392S Cc1c(c(nn1c2ccccc2)C(F)(F)F)OCC=C 7G-394S Cc1c(c(nn1c2ccccc2)C(F)(F)F)OCC#C 7G-395S Cc1c(c(nn1c2ccccc2)C(F)(F)F)OCc3ccccc3 7G-396S Cc1nnc(s1)SCCOc2ccccc2 7G-397S CC(C)Nc1nc(cc(n1)Oc2ccc(cc2)Cl)C(F)(F)F 7G-398S COc1ccc(cc1)c2nc3ccc(cc3n2OCC=C)Cl 7G-399S CC(C)Nc1nc(cc(n1)Oc2cc(cc(c2)Cl)Cl)C(F)(F)F 7G-400S CCOC(=O)c1c(cc(=O)n(n1)c2cccc(c2)Cl)O 7G-401S CN(C)S(=O)(=O)Oc1c(n(nc1C(F)(F)F)c2ccccc2)c3ccccc3 7G-402S c1ccc(cc1)c2c(c(nn2c3ccccc3)C(F)(F)F)OCc4ccc(cc4)Cl 7G-404S c1ccc(cc1)c2c(=O)n(cc(n2)c3ccc(cc3)F)O 7G-405S c1ccc(cc1)CN2CCN(CC2)c3c(cccn3)C(=O)Nc4ccc(cc4F)F 7G-407S c1cc(cc(c1)N2CCN(CC2)c3c(cccn3)C(=O)Nc4ccc(cc4F)F)C(F)(F)F 7G-409S c1cc(cc(c1)Cl)N2CCN(CC2)c3c(cccn3)C(=O)Nc4ccc(cc4F)F 7G-410S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4c(cccn4)C(=O)Nc5ccc(cc5F)F 7G-412S c1cc(cc(c1)NC(=O)c2cccnc2N3CCN(CC3)c4ccc(cc4)F)C(F)(F)F 7G-414S c1ccc(c(c1)N2CCN(CC2)c3c(cccn3)C(=O)Nc4ccc(cc4)Cl)F 7G-416S Cc1ccc(c(c1)N2CCN(CC2)c3ccc(cn3)C(=O)OCC=C)C 7G-417S c1ccc(cc1)CN2CCN(CC2)c3ccc(cn3)C(=O)OCC(F)(F)F 7G-418S Cc1ccc(c(c1)N2CCN(CC2)c3ccc(cn3)C(=O)OC)C 7G-420S CC(C)Nc1nc(cc(n1)Oc2ccc(cc2Cl)Cl)C(F)(F)F 7G-421S CC(C)Nc1nc(cc(n1)Oc2cccc(c2Cl)Cl)C(F)(F)F 7G-422S CC(C)Nc1nc(cc(n1)Oc2ccc(cc2)C#N)C(F)(F)F 7G-423S CC(C)Nc1nc(cc(n1)Sc2ccc(cc2)Br)C(F)(F)F 7G-424S CNc1nc(cc(n1)Sc2ccccc2)C(F)(F)F 7G-427S c1ccc(cc1)c2c(c(nn2c3ccccc3)C(F)(F)F)OCc4c(cccc4Cl)Cl 7G-428S Cc1ccc(cc1)Sc2cc(nc(n2)NC)C(F)(F)F 7G-430S CNc1nc(cc(n1)Sc2cccc(c2)C(F)(F)F)C(F)(F)F 7G-431S c1ccc(cc1)c2c(c(nn2c3ccccc3)C(F)(F)F)OCc4ccc(cc4Cl)Cl 7G-432S CC(C)(C)c1ccc(cc1)CSc2cc(nc(n2)NC)C(F)(F)F 7G-433S COc1ccc(cc1)NC(=O)c2ccc(nc2)Cl 7G-434S C=CCOc1c(n(nc1C(F)(F)F)c2ccccc2)c3ccccc3 7G-435S c1ccc(cc1)c2c(c(nn2c3ccccc3)C(F)(F)F)OCc4ccc(cc4)[N+](=O)[O-] 7G-436S CNc1nc(cc(n1)Sc2ccccc2Cl)C(F)(F)F 7G-437S Cn1c(=O)cc(nc1N)C(F)(F)F 7G-438S CCOC(=O)CSc1ccc(cn1)C(=O)OC 7G-439S c1ccc(cc1)COc2c(n(nc2C(F)(F)F)c3ccccc3)c4ccccc4 7G-441S COC(=O)c1ccc(cc1)COc2c(n(nc2C(F)(F)F)c3ccccc3)c4ccccc4 7G-442S c1cc(ccc1[N+](=O)[O-])Sc2ccc(cc2)F 7G-445S C#CCOc1c(n(nc1C(F)(F)F)c2ccccc2)c3ccccc3 7G-446S CC(C)Sc1ccc(cn1)C(=O)Nc2ccc(cc2)OC 7G-447S c1cc(ccc1N)Sc2ccc(cc2)F 7G-448S CC(C)(C)Sc1ccc(cn1)C(=O)O 7G-449S CCOC(=O)COc1c(n(nc1C(F)(F)F)c2ccccc2)c3ccccc3 7G-450S c1ccc(cc1)c2c(c(nn2c3ccccc3)C(F)(F)F)Oc4ccc(cc4)[N+](=O)[O-] 7G-451S CC(C)Sc1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 7G-452S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)Sc3ccc(cc3)F 7G-453S C(C(=O)NO)N 7G-455S c1ccc(cc1)c2cn(c(=O)c(n2)c3ccccc3)O 7G-457S c1cc(c(cc1F)F)NC(=O)c2ccc(nc2)Cl 7G-458S c1ccc2c(c1)nc(s2)c3cccc(c3)CSc4cccc(c4)C(F)(F)F 7G-462S c1cc(ccc1c2cn(c(=O)cn2)O)Cl 7G-463S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)Sc3ccc(cc3)F 7G-464S COC(=O)c1c(cc(=O)n(n1)c2cccc(c2)Cl)Cl 7G-465S c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)N3CCC(=O)CC3 7G-902 CN1CCOC12CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 7G-903 c1cc(cc(c1)N2C(=O)C3C4COCCN4OC3C2=O)C(F)(F)F 7G-904 CN1[C@@H]([C@@H]2[C@H](O1)C(=O)N(C2=O)c3ccc(cc3Cl)Cl)c4ccccc4 7G-905 c1cc(c(cc1Cl)Cl)C(=O)N2CCOC23CCN(CC3)c4ccc(nn4)Cl 7G-908 COc1ccc(cc1)C(=O)N2CCOC23CCN(CC3)c4ccc(nn4)Cl 7G-909 CN1CCC2(CC1)N(CCO2)C(=O)Nc3ccccc3 7G-910 CCOC(=O)C1=NOC2C1C(=O)N(C2=O)c3ccc(cc3Cl)Cl 7G-911 COC(=O)C1(C2C(C(=O)N(C2=O)c3ccc(cc3Cl)Cl)ON1)C(=O)OC 7G-912 c1ccc(cc1)C(C(C(=O)c2ccccc2)Br)Br 7G-914 c1ccc(cc1)CN2[C@@H]([C@@H]3[C@H](O2)C(=O)N(C3=O)c4ccc(cc4)Cl)c5ccccc5 7G-915 COC(=O)c1ccccc1N2C(=O)C3C4COCCN4OC3C2=O 7G-916 c1cc(ccc1N2C(=O)C3C4COCCN4OC3C2=O)Cl 7G-918 COc1ccc(cc1)C(=O)N2CCOC23CCN(CC3)c4ccc(cc4)[N+](=O)[O-] 7G-922 c1cc(ccc1N2CCC3(CC2)N(CCO3)C(=O)c4ccc(cc4Cl)Cl)[N+](=O)[O-] 7G-923 c1ccc(cc1)CN2[C@@H]([C@@H]3[C@H](O2)C(=O)N(C3=O)Cc4ccccc4)c5ccccc5 7G-926 c1cnc(nc1)N2CCC3(CC2)N(CCO3)C(=O)c4ccc(cc4Cl)Cl 7G-927 COc1ccc(cc1)C(=O)N2CCOC23CCN(CC3)c4ncccn4 7G-928 CN1[C@@H]([C@@H]2[C@H](O1)C(=O)N(C2=O)c3ccccc3)c4ccc(cc4)OC 7G-929 COC(=O)c1ccc(cc1)CON2C(=O)c3ccccc3C2=O 7G-934 COc1ccc(cc1)C(=O)N2CCOC23CCN(CC3)c4ncc(cn4)C#N 7G-935 c1cc(c(cc1Cl)Cl)C(=O)N2CCOC23CCN(CC3)c4ncc(cn4)C#N 7G-936 c1cc2c(cc1Cl)n3c(c(n2)N4CCC(=O)CC4)nnc3C(F)(F)F 7G-937 COC(=O)c1ccc(cc1)CON.Cl 7G-944 c1ccc(cc1)C[n+]2cccc(c2)O.[Br-] 7G-945 CC1(CC(=O)C(=NO)C(=O)C1)C 7G-947 CCOC(=O)c1nc(on1)N(C)C 7G-948 CCOC(=O)c1c(non1)C(=O)OCC 7G-949 CC1(CC(=O)C2(C3C(C(=O)N(C3=O)c4ccccc4)ON2)C(=O)C1)C 7G-950 CC1(CC(=O)C2(C3C(C(=O)N(C3=O)c4cccc(c4)C(F)(F)F)ON2)C(=O)C1)C 7G-951 c1ccc2c(c1)ccc3c2[C@H]([C@H](CO3)CO)NC(=S)Nc4cccc(c4)C(F)(F)F 7G-954 Cc1ccc(cc1)C(=O)NNC(=O)c2ccc(cc2)CONC(=O)c3ccc(cc3)C 7G-959 CNC(=S)N[C@@H]1c2c3ccccc3ccc2OC[C@@H]1CO 7G-960 c1ccc(cc1)CN2C(C(CO2)S(=O)(=O)c3ccccc3)c4ccccc4 7G-961 CN([C@H]1c2cccc(c2OC[C@H]1CO)OC)C(=O)Nc3ccc(cc3)Cl 7G-964 COc1cc(c(c(c1)OCC=C)/C=N/O)OC 7G-965 c1ccn(c1)c2nc3nccc(n3n2)/C=C/c4cccs4 7H-001 c1cc(c(cc1Cl)Cl)Oc2c(cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)C#N 7H-003 COc1ccc(cc1)Oc2c(cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)C#N 7H-004 c1ccc(cc1)Oc2c(cc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)C#N 7H-005 Cc1nc(c(s1)C(=O)NC(c2ccc(cc2)Cl)C(C)C)C(F)(F)F 7H-008 CN(C)/C=C(\C#N)/C(=O)C(F)(F)F 7H-009 CO/N=C/CC#N 7H-010 Cn1c(cnc1Sc2ccc(nn2)Sc3ncc(n3C)C(=O)OC)C(=O)OC 7H-011 c1ccnc(c1)C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3 7H-012 c1ccnc(c1)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 7H-014 c1ccc(cc1)c2c(n3ccsc3n2)/C=C/c4ccnc(n4)N 7H-015 CO/N=C/C(=C/c1ccc(cc1)Cl)/C#N 7H-016 CO/N=C/C(=C/c1ccccc1O)/C#N 7H-017 c1ccc(cc1)c2c(n3ccsc3n2)/C=C/c4ccn[nH]4 7H-018 CC(=O)c1cc(n(c1)C)C(=O)O 7H-020 CN(C)/C=C(\C=N\OC)/C#N 7H-022 c1ccc2c(c1)CCN(C2CC#N)C(=O)Nc3cccc(c3)C(F)(F)F 7H-023 c1ccc2c(c1)CCN(C2CC#N)C(=O)Nc3ccc(cc3Cl)Cl 7H-024 c1ccc2c(c1)CCN(C2CC#N)C(=O)Nc3ccc(cc3)C(F)(F)F 7H-025 CO/N=C/C(=N/Nc1ccc(cc1)Cl)/C#N 7H-026 c1ccc(cc1)n2c3c(cn2)C(=O)N4CCc5ccccc5C4C3 7H-027 c1ccc2c(c1)CCN3C2Cc4c(cnn4c5ccc(cc5)Cl)C3=O 7H-028 c1ccc2c(c1)CCN3C2Cc4c(cnn4c5c(cc(cn5)C(F)(F)F)Cl)C3=O 7H-029 c1ccc2c(c1)CCN3C2Cc4c(cnn4c5ccccc5Cl)C3=O 7H-030 c1ccc2c(c1)CCN3C2Cc4c(cnn4c5cccc(c5)Cl)C3=O 7H-031 c1cc(cc(c1)Cl)NC(=O)CC(=O)O 7H-034 c1ccc2c(c1)CCNC2CC(=O)Nc3cccc(c3)Cl 7H-036 c1ccc(c(c1)NC(=O)CC(=O)O)Cl 7H-037 CSc1nc2ncc3c(n2n1)CC4c5ccccc5CCN4C3=O 7H-038 COc1c(cc(cn1)c2c(cc(cn2)C(F)(F)F)Cl)C#N 7H-039 COc1ccc(cc1)N\2C(=O)C=C(/C2=C/Nc3ccc(c(c3)Cl)Cl)c4ccc(cc4)F 7H-040 c1ccc2c(c1)CCNC2CC(=O)Nc3ccccc3Cl 7H-041 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 7H-042 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)N3CCOCC3 7H-043 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)OC(F)(F)F 7H-046 COc1ccc(cc1)NC(=O)O/N=C(\c2ccccc2)/c3c(cc(cn3)C(F)(F)F)Cl 7H-047 Cc1nc(c(s1)C(=O)NNC(=N)c2ccccn2)C(F)(F)F 7H-048 Cc1nc(c(s1)C(=O)NNC(=N)c2cccnc2)C(F)(F)F 7H-049 c1ccc2c(c1)CCN3C2CC(=O)C(C3=O)/C=N/OCc4ccc(cc4Cl)Cl 7H-051 c1ccc(cc1)N/C=C/2\C(=O)CC3c4ccccc4CCN3C2=O 7H-052 Cc1nc(c(s1)c2[nH]c(nn2)c3ccccn3)C(F)(F)F 7H-053 Cc1nc(c(s1)c2[nH]c(nn2)c3cccnc3)C(F)(F)F 7H-054 c1ccc2c(c1)CCN3C2Cc4c(cnc5n4ncc5C#N)C3=O 7H-055 c1ccc2c(c1)CCN3C2CC(=O)/C(=C\Nc4cccc(c4)Oc5c(cc(cn5)C(F)(F)F)Cl)/C3=O 7H-056 c1ccc2c(c1)CCN3C2Cc4c(cnc5n4ncn5)C3=O 7H-057 c1cc(ccc1CSc2nc([nH]n2)N)Cl 7H-058 c1ccc(c(c1)CSc2nc([nH]n2)N)Cl 7H-059 c1cc(cc(c1)Cl)CSc2nc([nH]n2)N 7H-060 c1ccc2c(c1)CCN3C2Cc4c(cnc5n4nc(n5)SCc6ccccc6Cl)C3=O 7H-061 c1ccc2c(c1)CCN3C2Cc4c(cnc5n4nc(n5)SCc6cccc(c6)Cl)C3=O 7H-062 c1ccc2c(c1)CCN3C2Cc4c(cnc5n4nc(n5)SCc6ccc(cc6)Cl)C3=O 7H-063 c1ccc(cc1)CSc2nc3ncc4c(n3n2)CC5c6ccccc6CCN5C4=O 7H-064 c1cc(ccc1C(=O)CSc2ncc(cn2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 7H-065 c1ccc(cc1)C(=O)CSc2ncc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 7H-066 c1cc(cc(c1)C(F)(F)F)C(=O)CSc2ncc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 7H-067 CN(C)/C=C(\C#N)/C(C(F)(F)F)(NNc1c(cc(cn1)C(F)(F)F)Cl)O 7H-068 CN(C)/C=C(\C#N)/C(C(F)(F)F)(NN)O 7H-070 CO/N=C/C(C#N)c1c(cc(cn1)C(F)(F)F)Cl 7H-071 c1ccc2c(c1)CCN(C2Cc3c(cc(cn3)C(F)(F)F)Cl)C(=O)c4ccc(cc4)Cl 7H-072 c1c(cnc(c1Cl)n2c(c(cn2)C#N)C(F)(F)F)C(F)(F)F 7H-073 c1ccc(c(c1)N)Oc2c(cc(cn2)C(F)(F)F)Cl 7H-074 c1c(c(n[nH]1)C(F)(F)F)C#N 7H-076 c1ccc(cc1)c2cc(c(c(n2)N)C#N)c3ccc(cc3)F 7H-301S Cc1c(c(c(nc1c2ccc(cc2)Cl)N)C#N)c3ccccc3 7H-302S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2ccccc2Cl 7H-304S COc1ccc(cc1)c2ccc(s2)C(=O)Nc3ccc(cc3)Cl 7H-305S COc1ccc(cc1)c2ccc(s2)C(=O)Nc3ccc(cc3)OC 7H-306S CNC(=O)c1ccc(s1)c2ccc(cc2)OC 7H-307S CN(c1ccccc1)C(=O)c2ccc(s2)c3ccc(cc3)OC 7H-308S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2cccc(c2)Cl 7H-309S c1cc(ccc1CN2C(=O)CS(=O)CC2=O)F 7H-311S c1cc(ccc1CN2C(=O)CS(=O)(=O)CC2=O)F 7H-312S Cc1c(c(c(nc1c2ccc(cc2)Cl)N)C#N)c3ccccc3Cl 7H-313S Cc1c(nc(c(c1c2ccccc2Cl)C#N)N)C 7H-314S c1ccc(cc1)c2cc(c(c(n2)N)C#N)c3ccccc3Cl 7H-315S CN(C)S(=O)(=O)Oc1ccsc1C(=O)Nc2cccc(c2Cl)Cl 7H-316S CC(C)(C)c1cc(c(c(n1)N)C#N)c2ccccc2Cl 7H-317S COc1ccc(cc1)NC(=O)CSc2cccc(c2)Cl 7H-319S c1cc(ccc1C(=O)O)NC(=O)CSCC(=O)O 7H-320S c1cc(ccc1C(=O)O)NC(=O)CS(=O)CC(=O)O 7H-321S Cc1ccc(cc1)CN2C(=O)CSC(C2=O)C 7H-325S c1cc(ccc1C(=O)O)NC(=O)CS(=O)(=O)CC(=O)O 7H-326S c1cc(ccc1C(=O)O)N2C(=O)CSCC2=O 7H-327S c1cc(ccc1C(=O)O)N2C(=O)CS(=O)CC2=O 7H-328S c1cc(ccc1F)S(=O)(=O)CC(=O)c2ccc(cc2Cl)Cl 7H-329S c1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)Cl 7H-330S Cc1ccc(cc1)CN2C(=O)CS(=O)(=O)C(C2=O)C 7H-331S COc1ccc(cc1)NC(=O)CS(=O)c2cccc(c2)Cl 7H-332S c1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)F 7H-334S CN(C)/C=C(/C(=O)c1ccc(cc1)Cl)\S(=O)(=O)c2ccccc2 7H-337S CC1C(=O)N(C(=O)CS1)c2ccc(cc2F)F 7H-338S CC1C(=O)N(C(=O)CS1=O)c2ccc(cc2F)F 7H-339S c1ccc(cc1)n2c(c(cn2)S(=O)(=O)c3ccccc3)c4ccc(cc4)Cl 7H-342S CC1C(=O)N(C(=O)CS1)c2ccc(cc2)C#N 7H-343S CC1C(=O)N(C(=O)CS1)c2c(cccc2Cl)Cl 7H-344S c1ccc(cc1)S(=O)(=O)c2cnn(c2c3ccc(cc3)Cl)c4ccc(c(c4Cl)Cl)Cl 7H-345S c1ccc(cc1)S(=O)(=O)c2cnn(c2c3ccc(cc3)Cl)c4c(cc(cc4Cl)C(F)(F)F)Cl 7H-346S CN(C)/C=C(/C(=O)c1ccc(cc1Cl)Cl)\S(=O)(=O)c2ccc(cc2)F 7H-347S CC1C(=O)N(C(=O)CS1)c2cccc(c2)Cl 7H-348S CC1C(=O)N(C(=O)CS1)c2ccccc2Cl 7H-349S CCOC(=O)/C(=N/Nc1ccccc1)/C(=O)c2ccccc2 7H-350S c1ccc(cc1)S(=O)(=O)c2cnn(c2c3ccc(cc3)Cl)c4ccc(cc4Cl)Cl 7H-352S CC1C(=O)N(C(=O)CS1=O)Cc2ccc(cc2Cl)Cl 7H-354S c1ccc(cc1)S(=O)(=O)c2cnn(c2c3ccc(cc3)Cl)c4ccc(cc4F)F 7H-355S CC1C(=O)N(C(=O)CS1=O)c2c(cccc2Cl)Cl 7H-356S c1cc(ccc1C(=O)CSc2ccc(cc2)F)F 7H-357S CC1C(=O)N(C(=O)CS1)c2cc(ccc2Cl)Cl 7H-358S CC1C(=O)N(C(=O)CS1)c2ccc(cc2)F 7H-359S CC1C(=O)N(C(=O)CS1)c2ccc(cc2)OC 7H-360S CC1C(=O)N(C(=O)CS1)c2ccc(cc2)Br 7H-361S CC1C(=O)N(C(=O)CS1)c2cccc(c2)C(F)(F)F 7H-362S CC1C(=O)N(C(=O)CS1)c2ccc(cc2)C(F)(F)F 7H-363S c1cc(ccc1C(=O)CS(=O)(=O)c2ccc(cc2)F)F 7H-364S COc1ccc(cc1)C(=O)CS(=O)(=O)c2ccccc2 7H-365S COc1ccc(cc1)n2c(c(cn2)S(=O)(=O)c3ccccc3)c4ccc(cc4)Cl 7H-366S c1ccc(cc1)S(=O)(=O)c2cnn(c2c3ccc(cc3)Cl)c4ccc(c(c4)Cl)Cl 7H-367S Cc1cccc(c1C)n2c(c(cn2)S(=O)(=O)c3ccccc3)c4ccc(cc4)Cl 7H-368S CC1C(=O)N(C(=O)CS1)c2ccccc2C(F)(F)F 7H-369S c1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(c(c2)Cl)Cl 7H-370S c1ccc(cc1)S(=O)(=O)CC(=O)c2ccccc2Cl 7H-371S CN(C)/C=C(/C(=O)c1ccc(cc1)OC)\S(=O)(=O)c2ccccc2 7H-372S CN(C)/C=C(/C(=O)c1ccc(cc1)F)\S(=O)(=O)c2ccccc2 7H-373S Cc1ccc(cc1)N2C(=O)CSC(C2=O)C 7H-376S CN(C)/C=C(/C(=O)c1ccc(cc1)F)\S(=O)(=O)c2ccc(cc2)F 7H-377S COc1ccc(cc1)c2c(cnn2c3ccccc3)S(=O)(=O)c4ccccc4 7H-378S c1ccc(cc1)n2c(c(cn2)S(=O)(=O)c3ccccc3)c4ccc(cc4)F 7H-379S CN(C)/C=C(/C(=O)c1ccc(c(c1)Cl)Cl)\S(=O)(=O)c2ccccc2 7H-380S c1ccc(cc1)S(=O)(=O)c2cnn(c2c3ccc(cc3)F)c4cc(ccc4Cl)Cl 7H-381S CN(C)/C=C(/C(=O)c1ccccc1Cl)\S(=O)(=O)c2ccccc2 7H-382S Cc1cccc(c1)N2C(=O)CSC(C2=O)C 7H-383S Cc1ccccc1N2C(=O)CSC(C2=O)C 7H-384S CC(C)S(=O)(=O)CC(=O)c1ccc(cc1)Cl 7H-385S c1ccc(c(c1)NC(=O)CS(=O)CC(=O)O)Cl 7H-386S c1cc(cc(c1)Cl)NC(=O)CS(=O)CC(=O)O 7H-387S c1cc(ccc1C(F)(F)F)NC(=O)CS(=O)CC(=O)O 7H-388S Cc1ccccc1NC(=O)CS(=O)CC(=O)O 7H-389S c1cc(c(cc1Cl)C(F)(F)F)NC(=O)CS(=O)CC(=O)O 7H-390S Cc1ccc(cc1)CNC(=O)CS(=O)CC(=O)O 7H-391S c1ccc(cc1)n2c(c(cn2)S(=O)(=O)c3ccccc3)c4ccc(c(c4)Cl)Cl 7H-392S c1ccc(cc1)S(=O)(=O)c2cnn(c2c3ccc(c(c3)Cl)Cl)c4ccc(cc4)F 7H-393S COc1ccc(cc1)C(=O)CS(=O)(=O)C 7H-396S c1ccc(c(c1)NC(=O)CS(=O)(=O)CC(=O)O)Cl 7H-397S c1cc(cc(c1)Cl)NC(=O)CS(=O)(=O)CC(=O)O 7H-398S c1cc(ccc1C(F)(F)F)NC(=O)CS(=O)(=O)CC(=O)O 7H-399S Cc1ccccc1NC(=O)CS(=O)(=O)CC(=O)O 7H-400S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)OC 7H-401S COc1ccsc1C(=O)OC 7H-402S CC(C)n1c(nnc1S)CSCc2ccc(cc2)Cl 7H-404S CC(C)(C)c1ccc(cc1)CSc2nnc(n2C)C3CCCN3S(=O)(=O)c4ccc(cc4)Br 7H-406S Cn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])C3CCCN3S(=O)(=O)c4ccc(cc4)Br 7H-407S CC(C)n1c(nnc1SCc2ccc(cc2)Br)CSCc3ccc(cc3)Cl 7H-408S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)O 7H-409S COC(=O)c1c(ccs1)OCc2c(cccc2Cl)Cl 7H-410S COc1ccsc1C(=O)O 7H-411S c1ccc(cc1)/C(=N/OCc2ccc(cc2Cl)Cl)/CSc3ccc(cc3)Cl 7H-413S CCn1c(nnc1S)CSCc2ccc(cc2)Cl 7H-415S CCn1c(nnc1SCc2ccc(cc2)Br)CSCc3ccc(cc3)Cl 7H-419S CCn1c(nnc1SCc2ccc(cc2)Cl)CSCc3ccc(cc3)Cl 7H-422S CCn1c(nnc1SCc2ccc(cc2)F)CSCc3ccc(cc3)Cl 7H-423S CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)CSCc3ccc(cc3)Cl 7H-424S CCn1c(nnc1SCc2ccc(cc2)C(F)(F)F)CSCc3ccc(cc3)Cl 7H-425S CCn1c(nnc1SCc2ccc(cc2Cl)Cl)CSCc3ccc(cc3)Cl 7H-426S CCn1c(nnc1SCc2c(cccc2Cl)Cl)CSCc3ccc(cc3)Cl 7H-427S CCn1c(nnc1SCc2ccc(cc2)C)CSCc3ccc(cc3)Cl 7H-429S c1ccc(cc1)n2c(nnc2S)CSCc3ccc(cc3)Cl 7H-430S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)C(F)(F)F)CSCc4ccc(cc4)Cl 7H-431S c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)Cl)CSCc4ccc(cc4)Cl 7H-432S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Br)CSCc4ccc(cc4)Cl 7H-433S Cc1ccc(cc1)CSc2nnc(n2c3ccccc3)CSCc4ccc(cc4)Cl 7H-434S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)[N+](=O)[O-])CSCc4ccc(cc4)Cl 7H-435S c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)F)CSCc4ccc(cc4)Cl 7H-436S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)CSCc4ccc(cc4)Cl 7H-437S c1cc(c(c(c1)Cl)CSCC(=O)NN)Cl 7H-438S CCn1c(nnc1S)CSCc2c(cccc2Cl)Cl 7H-439S c1ccc(cc1)n2c(nnc2S)CSCc3c(cccc3Cl)Cl 7H-440S CCn1c(nnc1SCc2cccc(c2)F)CSCc3ccc(cc3)Cl 7H-442S c1cc(c(c(c1)Cl)COc2ccsc2C(=O)Nc3ccc(c(c3)Cl)Cl)Cl 7H-443S c1cc(c(c(c1)Cl)COc2ccsc2C(=O)Nc3ccc(cc3F)F)Cl 7H-444S c1cc(c(c(c1)Cl)COc2ccsc2C(=O)Nc3ccc(c(c3)F)F)Cl 7H-445S CCn1c(nnc1SCc2cc(ccc2Cl)Cl)CSCc3ccc(cc3)Cl 7H-446S c1ccc(c(c1)NC(=O)c2c(ccs2)OCc3c(cccc3Cl)Cl)Cl 7H-449S c1cc(c(c(c1)Cl)Cl)NC(=O)c2c(ccs2)OCc3c(cccc3Cl)Cl 7H-450S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3Cl)Cl)CSCc4ccc(cc4)Cl 7H-451S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)F)CSCc4ccc(cc4)Cl 7H-452S c1cc(c(c(c1)Cl)COc2ccsc2C(=O)Nc3ccc(cc3)[N+](=O)[O-])Cl 7H-453S c1cc(c(c(c1)Cl)COc2ccsc2C(=O)Nc3ccc(cc3)Br)Cl 7H-454S c1cc(c(c(c1)Cl)COc2ccsc2C(=O)Nc3ccc(cc3)C(F)(F)F)Cl 7H-455S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(c(c3)Cl)Cl 7H-457S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3F)F 7H-458S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(c(c3)F)F 7H-459S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3ccccc3Cl 7H-461S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3cccc(c3Cl)Cl 7H-463S CCn1c(nnc1SCc2ccc(cc2)Cl)CSCc3c(cccc3Cl)Cl 7H-464S CCn1c(nnc1SCc2ccc(cc2)Br)CSCc3c(cccc3Cl)Cl 7H-465S CCn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])CSCc3c(cccc3Cl)Cl 7H-466S CCn1c(nnc1SCc2c(cccc2Cl)Cl)CSCc3c(cccc3Cl)Cl 7H-467S CCn1c(nnc1SCc2c(cccc2Cl)F)CSCc3c(cccc3Cl)Cl 7H-468S c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)Cl)CSCc4c(cccc4Cl)Cl 7H-469S c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)F)CSCc4c(cccc4Cl)Cl 7H-470S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Br)CSCc4c(cccc4Cl)Cl 7H-471S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)CSCc4c(cccc4Cl)Cl 7H-472S Cc1ccc(cc1)CSc2nnc(n2c3ccccc3)CSCc4c(cccc4Cl)Cl 7H-473S COC(=O)c1ccc(cc1)CSc2nnc(n2c3ccccc3)CSCc4c(cccc4Cl)Cl 7H-474S c1ccc(cc1)n2c(nnc2SCc3cccc(c3)C(F)(F)F)CSCc4c(cccc4Cl)Cl 7H-475S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)[N+](=O)[O-])CSCc4c(cccc4Cl)Cl 7H-476S Cn1c(nnc1S)CS(=O)Cc2c(cccc2Cl)Cl 7H-477S Cn1c(nnc1SCc2ccc(cc2)Cl)CS(=O)Cc3c(cccc3Cl)Cl 7H-478S Cn1c(nnc1SCc2c(cccc2Cl)Cl)CS(=O)Cc3c(cccc3Cl)Cl 7H-479S Cn1c(nnc1SCc2c(cccc2Cl)F)CS(=O)Cc3c(cccc3Cl)Cl 7H-480S Cn1c(nnc1SCc2ccc(cc2)C(=O)OC)CS(=O)Cc3c(cccc3Cl)Cl 7H-481S c1cc(c(cc1Cl)Cl)CSCC(=O)NN 7H-483S c1cc(c(cc1Cl)Cl)CS(=O)CC(=O)NN 7H-484S Cn1c(nnc1S)CS(=O)Cc2ccc(cc2Cl)Cl 7H-485S CCn1c(nnc1S)CS(=O)Cc2ccc(cc2Cl)Cl 7H-486S Cc1ccc(cc1)CSc2nnc(n2C)CS(=O)Cc3ccc(cc3Cl)Cl 7H-487S Cn1c(nnc1SCc2ccc(cc2)C(=O)OC)CS(=O)Cc3ccc(cc3Cl)Cl 7H-488S Cn1c(nnc1SCc2c(cccc2Cl)F)CS(=O)Cc3ccc(cc3Cl)Cl 7H-489S Cn1c(nnc1SCc2ccc(cc2)C(F)(F)F)CS(=O)Cc3ccc(cc3Cl)Cl 7H-490S CCn1c(nnc1SCc2c(cccc2Cl)Cl)CS(=O)Cc3ccc(cc3Cl)Cl 7H-491S CCn1c(nnc1SCc2c(cccc2Cl)F)CS(=O)Cc3ccc(cc3Cl)Cl 7H-492S CCn1c(nnc1SCc2ccc(cc2)Br)CS(=O)Cc3ccc(cc3Cl)Cl 7H-493S CCn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])CS(=O)Cc3ccc(cc3Cl)Cl 7H-494S CC(C)n1c(nnc1S)CSCc2ccc(cc2Cl)Cl 7H-495S c1ccc(cc1)n2c(nnc2S)CSCc3ccc(cc3Cl)Cl 7H-496S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3)Br 7H-497S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3)[N+](=O)[O-] 7H-498S CC(C)(C)c1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3)C(F)(F)F 7H-499S c1cc(cc(c1)C(F)(F)F)COc2ccsc2C(=O)Nc3ccc(c(c3)Cl)Cl 7H-500S c1cc(cc(c1)C(F)(F)F)COc2ccsc2C(=O)Nc3ccc(cc3F)F 7H-501S c1cc(cc(c1)C(F)(F)F)COc2ccsc2C(=O)Nc3ccc(cc3)Br 7H-502S c1ccc(c(c1)NC(=O)c2c(ccs2)OCc3cccc(c3)C(F)(F)F)Cl 7H-504S Cn1c(nnc1SCc2ccc(cc2)Br)CS(=O)Cc3c(cccc3Cl)Cl 7H-505S Cc1ccc(cc1)CSc2nnc(n2C)CS(=O)Cc3c(cccc3Cl)Cl 7H-506S COc1ccsc1C(=O)Nc2ccc(cc2F)F 7H-507S COc1ccsc1C(=O)Nc2ccc(c(c2)F)F 7H-508S c1ccc(cc1)n2c(nnc2SCc3ccc(c(c3)Cl)Cl)CSCc4ccc(cc4)Cl 7H-509S CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)CSCc3ccc(cc3)Cl 7H-510S COc1ccsc1C(=O)Nc2ccc(cc2[N+](=O)[O-])Cl 7H-511S COc1ccsc1C(=O)Nc2ccccc2Br 7H-512S CCn1c(nnc1SCc2ccc(cc2)F)CSCc3c(cccc3Cl)Cl 7H-514S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)F)CSCc4c(cccc4Cl)Cl 7H-515S CCn1c(nnc1SCc2c(cccc2Cl)F)CSCc3ccc(cc3)Cl 7H-516S COc1ccc(c(c1)NC(=O)c2ccc(cc2)c3cccs3)OC 7H-517S COc1ccc(cc1OC)NC(=O)c2ccc(cc2)c3cccs3 7H-518S CCn1c(nnc1SCc2nnc(n2c3ccccc3)S)CSCc4ccc(cc4)Cl 7H-519S CC(C)n1c(nnc1SCc2ccc(cc2)Cl)CSCc3ccc(cc3Cl)Cl 7H-520S CC(C)n1c(nnc1SCc2ccc(cc2)C(=O)OC)CSCc3ccc(cc3Cl)Cl 7H-521S c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)Cl)CSCc4ccc(cc4Cl)Cl 7H-522S COC(=O)c1ccc(cc1)CSc2nnc(n2c3ccccc3)CSCc4ccc(cc4Cl)Cl 7H-523S CSc1nnc(n1c2ccccc2)CSCc3ccc(cc3Cl)Cl 7H-524S c1ccc(cc1)n2c(nnc2SCc3cccc(c3)C(F)(F)F)CSCc4ccc(cc4Cl)Cl 7H-525S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)CSCc4ccc(cc4Cl)Cl 7H-526S Cc1ccc(cc1)CSc2nnc(n2c3ccccc3)CSCc4ccc(cc4Cl)Cl 7H-527S c1ccc(cc1)n2c(nnc2S)CS(=O)Cc3ccc(cc3)Br 7H-529S CCn1c(nnc1S)CS(=O)Cc2ccc(cc2)Br 7H-530S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Br)CS(=O)Cc4ccc(cc4)Br 7H-531S c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)Cl)CS(=O)Cc4ccc(cc4)Br 7H-532S c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)F)CS(=O)Cc4ccc(cc4)Br 7H-533S COC(=O)c1ccc(cc1)CSc2nnc(n2c3ccccc3)CS(=O)Cc4ccc(cc4)Br 7H-535S c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)CS(=O)Cc4ccc(cc4)Br 7H-536S CCn1c(nnc1SCc2c(cccc2Cl)Cl)CS(=O)Cc3ccc(cc3)Br 7H-537S CCn1c(nnc1SCc2ccc(cc2)C)CS(=O)Cc3ccc(cc3)Br 7H-538S CCn1c(nnc1SCc2ccc(cc2)Cl)CS(=O)Cc3ccc(cc3)Br 7H-539S CCn1c(nnc1SCc2ccc(cc2)C(F)(F)F)CS(=O)Cc3ccc(cc3)Br 7H-540S CCn1c(nnc1SCc2ccc(cc2)F)CS(=O)Cc3ccc(cc3)Br 7H-541S c1ccc(cc1)C(C(=O)Nc2ccc(cc2)Cl)SCC(=O)O 7H-544S c1cc(c(cc1Cl)C(F)(F)F)NC(=O)CS(=O)(=O)CC(=O)O 7H-570S Cc1ccc(cc1)CNC(=O)CS(=O)(=O)CC(=O)O 7H-571S CS(=O)(=O)CC(=O)c1ccc(c(c1)Cl)Cl 7H-572S CS(=O)(=O)CC(=O)c1ccc(cc1)Cl 7H-573S CCOC(=O)C1=C(Nc2ccccc2S1)C 7H-574S CN(C)/C=C(/C(=O)c1ccc(cc1)Cl)\S(=O)(=O)C 7H-577S CN(C)/C=C(/C(=O)c1ccc(cc1)OC)\S(=O)(=O)C 7H-578S CN(C)/C=C(/C(=O)c1ccc(c(c1)Cl)Cl)\S(=O)(=O)C 7H-579S CC1=C(Sc2ccccc2N1)C(=O)C 7H-580S CN(C)/C=C/C(=O)c1ccc2c(c1)c(on2)c3ccccc3 7H-900 C/C(=N/OCc1ccc(cc1)OC)/c2ccc3c(c2)c(on3)c4ccccc4 7H-901 COc1ccc(cc1)N/C=C/C(=O)c2ccc3c(c2)c(on3)c4ccccc4 7H-902 Cn1c(cnc1SCc2c(cccc2Cl)Cl)CS(=O)(=O)c3ccccc3 7H-903 c1cc(ccc1C2OCCO2)[N+](=O)[O-] 7H-904 c1ccc(cc1)c2c3cc(ccc3no2)C4OCCO4 7H-906 Cn1c(cnc1SCc2c(cccc2Cl)Cl)/C(=C/N(C)C)/S(=O)(=O)c3ccccc3 7H-907 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)CC(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl 7H-908 Cc1cc2c(n1c3cccc(c3)OC)CC(CC2=O)(C)C 7H-909 c1cc(cc(c1)NC(=S)N2CC(CO2)O)C(F)(F)F 7H-910 c1ccc(cc1)c2c3cc(ccc3no2)C=O 7H-911 Cc1cc(on1)N 7H-912 c1ccc(c(c1)N2CCN(CC2)C(=N)CC#N)Cl 7H-913 C1CCC(CC1)NC(=O)N2CC(CO2)O 7H-914 c1ccc(cc1)c2c3cc(ccc3no2)/C=N\Nc4c(cc(cn4)C(F)(F)F)Cl 7H-915 c1cc(cc(c1)NC(=O)N2CC(CO2)O)C(F)(F)F 7H-916 c1ccc(c(c1)N2CCN(CC2)/C(=C(\C=C(C#N)C#N)/C#N)/N)Cl 7H-918 c1cc(nc(c1)Cl)N2CCN(CC2)CC(=O)N3CC(CO3)O 7H-919 c1c(cnc(c1Cl)N2CCN(CC2)CC(=O)N3CC(CO3)O)C(F)(F)F 7H-920 Cc1ccc(cc1)c2c3cc(ccc3no2)C4OCCO4 7H-921 c1cc(ccc1c2c3cc(ccc3no2)C4OCCO4)Cl 7H-922 Cc1ccc(cc1)c2c3cc(ccc3no2)C=O 7H-923 c1cc(ccc1c2c3cc(ccc3no2)C=O)Cl 7H-924 c1cc(ccc1c2c3cc(ccc3no2)/C=N\O)Cl 7H-926 c1cc(ccc1c2c3cc(ccc3no2)C#N)Cl 7H-927 Cc1ccc(cc1)c2c3cc(ccc3no2)/C=C/C(=O)O 7H-928 CC1(NC(=O)N(N1)c2c(cc(cn2)C(F)(F)F)Cl)C3=NOC(C3)CNc4c(cc(cn4)C(F)(F)F)Cl 7H-929 CC1(NC(=O)N(N1)c2ccc(cc2)F)C3=NOC(C3)CNc4c(cc(cn4)C(F)(F)F)Cl 7H-930 C/C(=N\OC)/C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 7H-931 c1cc(ccc1N/C=C/C(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)OC(F)(F)F 7H-933 c1cc(c(cc1Cl)Cl)N/C=C/C(=O)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 7H-934 c1cnc(nc1C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)N 7H-935 c1cn(nc1C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)c4c(cc(cn4)C(F)(F)F)Cl 7H-936 Cc1cc(c(nc1)N/N=C(/C)\c2c(cc(oc2=O)C)O)Cl 7H-937 Cc1cc(=O)c(c(o1)C)C(=O)O 7H-938 Cc1cc(cc(=O)o1)O 7H-939 COc1cccc(c1)NC=C2C(=O)CCCC2=O 7H-940 c1ccc(cc1)c2nccc(n2)C3=NOC(C3)CNc4c(cc(cn4)C(F)(F)F)Cl 7H-942 CCOC(=O)c1c(c2ccccc2[nH]1)n3cccc3 7H-943 c1cc(ccc1n2ccc(n2)C3=NOC(C3)CNc4c(cc(cn4)C(F)(F)F)Cl)F 7H-944 Cc1cc(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)c3c(nn(c3O)c4ccccc4)C 7H-945 Cc1nccc(n1)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 7H-946 c1ccnc(c1)N2CCN(CC2)CC(=O)N3CC(CO3)O 7H-947 Cc1c2c(con2)c(nn1)c3ccc(cc3)OC 7H-948 CCOC(=O)c1c(c2ccccc2n1Cc3ccc(cc3)C)n4cccc4 7H-949 Cc1cc2ccccc2n1c3c(cc(cn3)C(F)(F)F)Cl 7H-950 Cc1c(c2ccccc2[nH]1)c3c(cc(cn3)C(F)(F)F)Cl 7H-951 Cc1c(c2ccccc2n1c3c(cc(cn3)C(F)(F)F)Cl)Br 7H-952 c1ccc(cc1)c2cn(cc2[N+](=O)[O-])c3c(cc(cn3)C(F)(F)F)Cl 7H-953 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC3CC(=NO3)C(=O)C 7H-954 CC(=O)c1c(con1)C#N 7H-955 CN(/C=C\1/c2ccccc2NC1=O)O 7H-956 c1ccc2c(c1)C(C(=O)N2)/C=N\OCc3c(snn3)Cl 7H-957 CC(=C(C#N)C#N)C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 7H-958 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)Br 7H-960 Cc1ccc(cc1)Cn2c(c(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl)C 7H-961 c1ccc2c(c1)c(c(n2c3c(cc(cn3)C(F)(F)F)Cl)CBr)Br 7H-962 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N3CCOCC3 7J-002 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl 7J-004 CN1CCN(CC1)S(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 7J-005 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N3CCCC3 7J-007 c1ccnc(c1)c2ncc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 7J-008 c1cnccc1c2ncc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 7J-009 c1ccc(cc1)CNS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 7J-010 COCCCNS(=O)(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 7J-011 c1cc(cnc1)CNS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl 7J-012 CN(C)CCCNS(=O)(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 7J-013 c1cc(cnc1)c2ncc(cn2)c3c(cc(cn3)C(F)(F)F)Cl 7J-014 c1c(cn2cnnc2c1Cl)C(F)(F)F 7J-015 CCOC(=O)C(=CNc1cccc(c1C)C)C(=O)OCC 7J-016 CCOC(=O)c1cnc2c(c(ccc2c1O)C)C 7J-017 CCOC(=O)c1cnc2c(c(ccc2c1Cl)C)C 7J-018 CCN(CC)S(=O)(=O)c1ccc(s1)Cc2c(cc(cn2)C(F)(F)F)Cl 7J-019 CCOC(=[NH2+])COc1ccc(cc1)F.[Cl-] 7J-020 c1cc(ccc1OCC(=N)N)F.Cl 7J-021 CCN(CC)S(=O)(=O)c1ccc(s1)/C(=C\N(C)C)/c2c(cc(cn2)C(F)(F)F)Cl 7J-023 CCN(CC)S(=O)(=O)c1ccc(s1)C(/C=N/OC)c2c(cc(cn2)C(F)(F)F)Cl 7J-024 CCOC(=O)N(c1c(cccn1)[N+](=O)[O-])OC 7J-025 CCN(CC)S(=O)(=O)c1ccc(s1)C(/C=N/O)c2c(cc(cn2)C(F)(F)F)Cl 7J-028 CCN(CC)S(=O)(=O)c1ccc(s1)/C(=C\Nc2ccc(cc2)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 7J-029 CCN(CC)S(=O)(=O)c1ccc(s1)C(/C=N\OCc2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl 7J-030 Cc1cc([nH]c(=O)c1S(=O)(=O)c2ccccc2F)C 7J-301S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2)C)C 7J-302S Cc1ccccc1S(=O)(=O)c2c(cc(nc2OCC(=C)C)c3ccccc3)C 7J-303S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2OC)CC(=C)C)C 7J-304S Cc1ccc(cc1)S(=O)(=O)c2c(cc(n(c2=O)CC(=C)C)C)C 7J-305S Cc1cc(n(c(=O)c1S(=O)(=O)c2ccccc2Cl)CC(=C)C)C 7J-306S Cc1cc(n(c(=O)c1S(=O)(=O)c2cccc(c2)Cl)CC(=C)C)C 7J-307S Cc1cccc(c1)S(=O)(=O)c2c(cc(n(c2=O)CC(=C)C)C)C 7J-309S CCn1c(cc(c(c1=O)S(=O)(=O)c2ccccc2Cl)C)C 7J-310S Cc1cc2c(cc1C)nc([nH]2)c3cccnc3Cl 7J-317S CCOC(=O)Cn1c2cc(c(cc2nc1c3cccnc3Cl)C)C 7J-318S Cc1cccc(c1)Cn2c3cc(c(cc3nc2c4cccnc4Cl)C)C 7J-319S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccc(cc4)Cl 7J-320S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccccc4Cl 7J-321S Cc1ccccc1S(=O)(=O)c2c(cc(n(c2=O)C)C)C 7J-323S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccc(cc4Cl)Cl 7J-324S CCCn1c2cc(c(cc2nc1c3cccnc3Cl)C)C 7J-325S Cc1cc(cc(c1O)C)C(=O)CCl 7J-328S Cc1cc(cc(c1O)C)C(=O)CSc2ccc(cc2)Cl 7J-331S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)CC=C 7J-333S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)CC#C 7J-334S CCSc1ccc(c(c1Cl)Cl)C(=O)C 7J-335S Cc1cc(cc(c1O)C)C(=O)CS(=O)(=O)c2ccc(cc2)Cl 7J-336S Cc1cc(cc(c1O)C)C(=O)CS(=O)c2ccc(cc2)Cl 7J-337S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CSc2ccc(cc2)Cl 7J-338S Cc1cc(cc(c1O)C)C(=O)CSc2cccc(c2)C(F)(F)F 7J-340S CCCCn1c(cc(c(c1=O)S(=O)(=O)c2ccccc2C)C)C 7J-341S Cc1ccccc1S(=O)(=O)c2c(cc(n(c2=O)CC(C)C)C)C 7J-342S Cc1ccccc1S(=O)(=O)c2c(cc(n(c2=O)C(C)C)C)C 7J-343S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccc(cc4)F 7J-346S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccc(c(c4)Cl)Cl 7J-347S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)C 7J-348S Cc1cc(cc(c1OC(=S)N(C)C)C)C(=O)CSc2ccc(cc2)Cl 7J-349S Cc1cc(cc(c1O)C)C(=O)CS(=O)(=O)c2cccc(c2)C(F)(F)F 7J-350S Cc1cc(cc(c1OC(=S)N(C)C)C)C(=O)CSc2cccc(c2)C(F)(F)F 7J-351S c1ccc2c(c1)[nH]c(n2)CCl 7J-352S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccc(cc4)C(C)(C)C 7J-353S Cc1ccccc1Cn2c3cc(c(cc3nc2c4cccnc4Cl)C)C 7J-354S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)CC(=C)C 7J-355S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccccc4F 7J-356S Cc1ccc(cc1)SCc2[nH]c3ccccc3n2 7J-357S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CSc2cccc(c2)C(F)(F)F 7J-358S CCS(=O)(=O)c1ccc(c(c1Cl)Cl)C(=O)O 7J-359S Cc1cc(cc(c1O)C)C(=O)CS(=O)c2cccc(c2)C(F)(F)F 7J-360S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4ccc(cc4)[N+](=O)[O-] 7J-361S Cc1ccc(cc1)SCC(=O)c2cc(c(c(c2)C)O)C 7J-362S Cc1ccc(cc1)S(=O)CC(=O)c2cc(c(c(c2)C)O)C 7J-364S Cc1ccc(cc1)SCc2nc3ccccc3n2CC(=O)Nc4ccccc4 7J-365S Cc1ccc(cc1)S(=O)(=O)CC(=O)c2cc(c(c(c2)C)O)C 7J-366S c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C#N 7J-511S c1ccc(cc1)C(=O)CC(C#N)c2cccc(c2)Cl 7J-515S COC(=O)C(CC(=O)c1ccccc1)c2cccc(c2)Cl 7J-516S c1ccc(cc1)C(=O)CC(c2cccc(c2)Cl)C(=O)O 7J-517S c1ccc(cc1)C(=O)CC(C#N)c2ccc(cc2Cl)Cl 7J-519S Cc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Cl 7J-522S Cc1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C#N 7J-523S Cc1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C(=O)OC 7J-524S Cc1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C(=O)O 7J-525S c1cc(cc(c1)Cl)C(CC(=O)c2ccc(cc2)Cl)C#N 7J-527S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2cccc(c2)Cl 7J-528S c1cc(cc(c1)Cl)C(CC(=O)c2ccc(cc2)Cl)C(=O)O 7J-529S c1cc(c(c(c1)Cl)Cl)C(CC(=O)c2ccc(cc2)Cl)C#N 7J-531S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2cccc(c2Cl)Cl 7J-532S c1cc(c(c(c1)Cl)Cl)C(CC(=O)c2ccc(cc2)Cl)C(=O)O 7J-533S COc1cccc(c1)C(=O)CC(C#N)c2ccc(cc2)F 7J-535S COc1cccc(c1)C(=O)CC(c2ccc(cc2)F)C(=O)OC 7J-536S COc1cccc(c1)C(=O)CC(c2ccc(cc2)F)C(=O)O 7J-537S c1cc(ccc1C(=O)CC(C#N)c2ccc(cc2Cl)Cl)Cl 7J-539S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2ccc(cc2Cl)Cl 7J-540S c1cc(ccc1C(=O)CC(c2ccc(cc2Cl)Cl)C(=O)O)Cl 7J-541S CCc1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C(=O)OC 7J-544S CCc1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C(=O)O 7J-545S c1cc(ccc1C(CC(=O)c2ccc(cc2)Cl)C#N)F 7J-547S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2ccc(cc2)F 7J-548S c1cc(ccc1C(CC(=O)c2ccc(cc2)Cl)C(=O)O)F 7J-549S c1cc(c(c(c1)Cl)C(CC(=O)c2ccc(cc2)Cl)C#N)Cl 7J-551S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2c(cccc2Cl)Cl 7J-552S c1cc(cc(c1)F)C(CC(=O)c2ccc(cc2)Cl)C#N 7J-555S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2cccc(c2)F 7J-556S c1cc(cc(c1)F)C(CC(=O)c2ccc(cc2)Cl)C(=O)O 7J-557S c1ccc(cc1)C(=O)CC(C#N)c2ccc(cc2)Cl 7J-558S COC(=O)C(CC(=O)c1ccccc1)c2ccc(cc2)Cl 7J-559S c1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)C(=O)O 7J-560S c1cc(ccc1C(CC(=O)c2ccc(cc2)Cl)C#N)Cl 7J-561S c1cc(ccc1C(CC(=O)c2ccc(cc2)Cl)C(=O)O)Cl 7J-563S c1ccc(cc1)C(=O)CC(C#N)c2c(cccc2Cl)Cl 7J-565S COC(=O)C(CC(=O)c1ccccc1)c2c(cccc2Cl)Cl 7J-566S Cc1cccc(c1)C(=O)CC(C#N)c2ccc(cc2)Cl 7J-569S Cc1cccc(c1)C(=O)CC(c2ccc(cc2)Cl)C(=O)OC 7J-570S Cc1cccc(c1)C(=O)CC(c2ccc(cc2)Cl)C(=O)O 7J-571S Cc1cccc(c1)C(=O)CC(C#N)c2ccc(cc2Cl)Cl 7J-573S Cc1cccc(c1)C(=O)CC(c2ccc(cc2Cl)Cl)C(=O)OC 7J-574S CC(C)c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Cl 7J-576S CC(C)c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C(=O)OC 7J-578S CC(C)c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)C(=O)O 7J-579S c1cc(c(c(c1)Cl)C(CC(=O)c2ccc(cc2)Cl)C#N)F 7J-581S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2c(cccc2Cl)F 7J-582S c1cc(c(c(c1)Cl)C(CC(=O)c2ccc(cc2)Cl)C(=O)O)F 7J-583S c1cc(cc(c1)Br)C(CC(=O)c2ccc(cc2)Cl)C#N 7J-585S COC(=O)C(CC(=O)c1ccc(cc1)Cl)c2cccc(c2)Br 7J-586S c1cc(cc(c1)Br)C(CC(=O)c2ccc(cc2)Cl)C(=O)O 7J-587S c1cc(ccc1C(CC(=O)c2ccc(cc2)Br)C#N)Cl 7J-589S c1cc(ccc1c2cnc(nc2)S)Cl 7J-591S CSc1ncc(cn1)c2ccc(cc2)Cl 7J-592S C#CCSc1ncc(cn1)c2ccc(cc2)Cl 7J-593S COC(=O)CSc1ncc(cn1)c2ccc(cc2)Cl 7J-594S CCOC(=O)C(C)Sc1ncc(cn1)c2ccc(cc2)Cl 7J-595S c1ccc(cc1)CSc2ncc(cn2)c3ccc(cc3)Cl 7J-596S c1cc(ccc1CSc2ncc(cn2)c3ccc(cc3)Cl)Cl 7J-597S c1cc(ccc1CSc2ncc(cn2)c3ccc(cc3)Cl)F 7J-598S c1cc(ccc1c2cnc(nc2)SCc3ccc(c(c3)Cl)Cl)Cl 7J-599S c1cc(cc(c1)Cl)c2cnc(nc2)S 7J-600S C=CCSc1ncc(cn1)c2ccc(cc2)Cl 7J-601S c1cc(cc(c1)C(F)(F)F)CSc2ncc(cn2)c3ccc(cc3)Cl 7J-602S c1cc(cc(c1)Cl)CSc2ncc(cn2)c3ccc(cc3)Cl 7J-603S c1cc(ccc1CSc2ncc(cn2)c3ccc(cc3)Cl)[N+](=O)[O-] 7J-604S c1cc(ccc1c2cnc(nc2)SCc3ccc(cc3Cl)Cl)Cl 7J-605S CCOC(=O)C(C)Sc1ncc(cn1)c2cccc(c2)Cl 7J-606S CCOC(=O)CSc1ncc(cn1)c2cccc(c2)Cl 7J-607S C#CCSc1ncc(cn1)c2cccc(c2)Cl 7J-608S C=CCSc1ncc(cn1)c2cccc(c2)Cl 7J-609S c1ccc(cc1)c2cnc(nc2)S 7J-610S CSc1ncc(cn1)c2ccccc2 7J-611S C#CCSc1ncc(cn1)c2ccccc2 7J-612S CCOC(=O)CSc1ncc(cn1)c2ccccc2 7J-613S CCOC(=O)C(C)Sc1ncc(cn1)c2ccccc2 7J-614S C=CCSc1ncc(cn1)c2ccccc2 7J-615S c1ccc(cc1)c2cnc(nc2)SCc3ccc(c(c3)Cl)Cl 7J-616S c1ccc(cc1)c2cnc(nc2)SCc3ccc(cc3)Cl 7J-617S c1ccc(cc1)c2cnc(nc2)SCc3ccc(cc3)F 7J-618S c1cc(ccc1C(CC(=O)c2ccc(cc2)Br)C(=O)O)Cl 7J-620S c1cc(ccc1/C=C/C(=O)c2ccc(c(c2)Cl)Cl)Cl 7J-621S c1cc(ccc1C(CC(=O)c2ccc(c(c2)Cl)Cl)C#N)Cl 7J-622S c1cc(ccc1C(CC(=O)c2ccc(c(c2)Cl)Cl)C(=O)O)Cl 7J-624S Cc1ccc(cc1)C(CC(=O)c2ccc(c(c2)Cl)Cl)C#N 7J-626S Cc1ccc(cc1)C(CC(=O)c2ccc(c(c2)Cl)Cl)C(=O)O 7J-628S CCc1ccc(cc1)C(CC(=O)c2ccc(c(c2)Cl)Cl)C#N 7J-630S c1cc(ccc1C(CC(=O)c2ccc(cc2)Br)C#N)F 7J-634S Cc1ccc(cc1)C2CC(=NNC2=O)c3ccc(cc3)Cl 7J-637S c1cc(cc(c1)Cl)C2CC(=NNC2=O)c3ccc(cc3)Cl 7J-640S COc1cccc(c1)C2=NNC(=O)C(C2)c3ccc(cc3)F 7J-641S CCc1ccc(cc1)C2CC(=NNC2=O)c3ccc(cc3)Cl 7J-642S c1cc(ccc1C2CC(=NNC2=O)c3ccc(cc3)Cl)F 7J-645S Cc1cccc(c1)C2=NNC(=O)C(C2)c3ccc(cc3)Cl 7J-646S CC(C)c1ccc(cc1)C2CC(=NNC2=O)c3ccc(cc3)Cl 7J-647S c1cc(ccc1C2=NNC(=O)C(C2)c3ccc(cc3Cl)Cl)Cl 7J-648S c1cc(c(c(c1)Cl)C2CC(=NNC2=O)c3ccc(cc3)Cl)Cl 7J-649S c1cc(c(c(c1)Cl)C2CC(=NNC2=O)c3ccc(cc3)Cl)F 7J-650S c1ccc(cc1)C2=NNC(=O)C(C2)c3ccc(cc3Cl)Cl 7J-651S Cc1cccc(c1)C2=NNC(=O)C(C2)c3ccc(cc3Cl)Cl 7J-652S c1cc(ccc1C2CC(=NNC2=O)c3ccc(c(c3)Cl)Cl)Cl 7J-653S c1ccc(cc1)c2c3ccccc3[nH]c2c4ccccc4 7J-655S c1ccc(cc1)C2CC(=NNC2=O)c3ccc(cc3)Br 7J-657S CCc1ccc(cc1)C2CC(=NNC2=O)c3ccc(c(c3)Cl)Cl 7J-658S c1cc(ccc1C2CC(=NNC2=O)c3ccc(cc3)Br)Cl 7J-659S c1cc(cc(c1)Br)C2CC(=NNC2=O)c3ccc(cc3)Cl 7J-660S c1cc(cc(c1)Cl)CN2C(=O)C(CC(=N2)c3ccc(cc3)Cl)c4cccc(c4Cl)Cl 7J-662S Cc1ccc(cc1)CN2C(=O)C(CC(=N2)c3ccc(cc3)Cl)c4cccc(c4Cl)Cl 7J-663S COC(=O)c1ccc(cc1)CN2C(=O)C(CC(=N2)c3ccc(cc3)Cl)c4cccc(c4Cl)Cl 7J-664S c1cc(cc(c1)C(F)(F)F)c2cnc(nc2)S 7J-666S CSc1ncc(cn1)c2cccc(c2)Cl 7J-668S c1cc(cc(c1)Cl)c2cnc(nc2)SCc3ccc(c(c3)Cl)Cl 7J-669S CSc1ncc(cn1)c2cccc(c2)C(F)(F)F 7J-670S Cn1c(cc(nc1=S)C(F)(F)F)O 7J-672S Cn1c(=O)cc(nc1SCc2ccc(c(c2)Cl)Cl)C(F)(F)F 7J-673S COC(=O)C1CSC(N1C(=O)Nc2ccc(c(c2)Cl)Cl)C(=O)OC 7J-900 CCOC(=O)/C=C(\N)/N1CCN(CC1)c2cccc(n2)Cl 7J-901 CCOC(=O)/C=C(/NC(=O)Nc1cccc(c1)C(F)(F)F)\NN(C)c2c(cc(cn2)C(F)(F)F)Cl 7J-902 c1cc(nc(c1)Cl)N2CCN(CC2)c3cc(n(c(=O)n3)C4CCCCC4)O 7J-905 c1cc(cc(c1)n2c(cc(nc2=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)O)C(F)(F)F 7J-906 CN(c1c(cc(cn1)C(F)(F)F)Cl)Nc2cc(n(c(=O)n2)c3cccc(c3)C(F)(F)F)O 7J-907 Cc1cc(nc(n1)NC(=O)c2c(onc2C(=O)O)C)C 7J-908 c1cn[nH]c1c2c(ccs2)Cl 7J-911 c1ccc(cc1)NC(=O)n2c(ccn2)c3c(ccs3)Cl 7J-912 c1ccc(cc1)S(=O)(=O)n2c(ccn2)c3c(ccs3)Cl 7J-913 c1cc(cc(c1)N/C=C/C(=O)c2c(ccs2)Cl)C(F)(F)F 7J-914 c1csc(c1Cl)C(=O)C/C=N/OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 7J-915 c1csc(c1Cl)C(=O)C/C=N/OCc2c(snn2)Cl 7J-916 COC(=O)C1CSC(N1C(=O)Nc2ccccc2)C(=O)OC 7J-917 Cc1ccc(cc1)c2ccccc2C#N 7J-918 COC(=O)C1CSC(N1C(=O)CN2CCN(CC2)c3ccc(c(c3)Cl)Cl)C(=O)OC 7J-919 COC(=O)C1CSC(N1C(=O)CN2CCN(CC2)C(c3ccccc3)c4ccccc4)C(=O)OC 7J-920 COC(=O)C1CSC(N1C(=O)CN2CCN(CC2)c3ccccc3)C(=O)OC 7J-921 Cc1c(c(no1)C(=O)O)C(=O)Nc2cccc(c2)C(F)(F)F 7J-922 c1cnn(c1c2c(ccs2)Cl)S(=O)(=O)C(F)(F)F 7J-923 c1cc(c(c(c1)Cl)c2c(con2)C(=O)c3c(ccs3)Cl)Cl 7J-924 COC(=O)C1CSC(N1C(=O)CN2CCN(CC2)c3ccccn3)C(=O)OC 7J-925 c1cc(ccc1CCc2c(cc(cn2)C(F)(F)F)Cl)N 7K-001 COc1ccc(cc1OC)C(C#N)c2ccc(cc2)C(=O)c3ccccc3 7K-002 c1ccc(cc1)C(C#N)c2cccc(c2C#N)C(C#N)c3ccccc3 7K-003 CO/N=C/NC(=O)C(c1ccc(cc1)C(=O)c2ccccc2)c3ccc(cc3)Cl 7K-004 Cc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)OC 7K-005 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2c4[nH]c(nn4)S 7K-006 CSc1[nH]c(nn1)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4cccs4 7K-007 Cc1ccc(cc1)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)F 7K-008 COc1ccc(cc1OC)C(C#N)c2cccc(c2C#N)F 7K-009 Cc1ccc(cc1C)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)F 7K-010 Cc1ccc(cc1C)N/N=C(\C=N\OC)/C(=O)c2ccc(cc2)OC 7K-011 c1ccc(c(c1)C(C#N)c2cccc(c2C#N)F)Cl 7K-012 c1ccc(cc1)C(=O)c2ccc(cc2)C(C#N)c3cccs3 7K-015 COc1cnc(o1)c2cc(ccc2Cl)Cl 7K-016 c1cc(oc1)C=C(C#N)C#N 7K-021 CC1CC(CC(C1)(CC(=O)Nc2cc(cc(c2)Cl)Cl)C(=O)O)(C)C 7K-025 CC1CC(CC2(C1)CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl)(C)C 7K-026 Cn1c(c(c(n1)c2ccccc2)CSc3c(cccc3Cl)Cl)Sc4ccc(cc4)Cl 7K-301S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)O 7K-303S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)Cl 7K-304S c1cc(ccc1C(=O)/C=N/O)Cl 7K-310S Cc1ccc(cc1)Sc2c(nnc(n2)c3ccccc3)c4ccccc4 7K-315S COc1c(nnc(n1)c2ccccc2)c3ccccc3 7K-316S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)N4CCOCC4 7K-318S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)Oc4ccc(cc4Cl)Cl 7K-319S Cc1ccc(cc1)Sc2c(cc3ccccc3n2)c4ccccc4 7K-320S c1ccc(cc1)c2cc3ccccc3nc2Sc4ccc(cc4)Br 7K-321S CS(=O)(=O)c1ccc(nn1)Nc2ccccc2 7K-325S COc1ccc(cc1)Nc2ccc(nn2)S(=O)(=O)C 7K-326S CS(=O)(=O)c1ccc(nn1)Nc2cccc(c2)C(F)(F)F 7K-327S CS(=O)(=O)c1ccc(nn1)Nc2ccc(cc2)F 7K-328S CS(=O)(=O)c1ccc(nn1)Nc2ccc(cc2)Cl 7K-329S CN(C)c1c(nnc(n1)c2ccccc2)c3ccccc3 7K-332S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)Sc4c(cccc4Cl)Cl 7K-333S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)Sc4cccc(c4)C(F)(F)F 7K-336S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)Sc4ccc(cc4)F 7K-337S c1ccc2c(c1)cc(c(n2)Cl)c3ccc(cc3)Cl 7K-338S CC1CN(CC(O1)C)c2c(nnc(n2)c3ccccc3)c4ccccc4 7K-339S CS(=O)(=O)c1ccc(nn1)Nc2ccc(cc2)OC(F)(F)F 7K-342S COc1ccc(c(c1)Nc2ccc(nn2)S(=O)(=O)C)OC 7K-344S CC(C)Nc1c(nnc(n1)c2ccccc2)c3ccccc3 7K-349S Cc1ccc(cc1)Sc2c(cc3ccccc3n2)c4ccc(cc4)Cl 7K-350S c1ccc2c(c1)cc(c(n2)Sc3ccc(cc3)Cl)c4ccc(cc4)Cl 7K-351S c1ccc2c(c1)cc(c(n2)Sc3ccc(cc3)F)c4ccc(cc4)Cl 7K-352S c1ccc2c(c1)cc(c(n2)Sc3c(cccc3Cl)Cl)c4ccc(cc4)Cl 7K-353S Cc1c(nc(nn1)c2ccccc2)O 7K-355S Cc1c(nc(nn1)c2ccccc2)Cl 7K-356S COc1ccc(cc1)Sc2c(cc3ccccc3n2)c4ccc(cc4)Cl 7K-357S c1ccc2c(c1)cc(c(n2)Sc3cccc(c3)Cl)c4ccc(cc4)Cl 7K-358S c1ccn2c(c1)ncc2C(=O)c3ccc(cc3)Cl 7K-361S c1ccn2c(c1)ncc2C(=O)c3ccc(cc3Cl)Cl 7K-362S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)Oc4ccc(cc4)C#N 7K-363S c1ccc(cc1)c2c(nc(nn2)c3ccccc3)Oc4cccc(c4)C(F)(F)F 7K-364S Cc1c(nc(nn1)c2ccccc2)N(C)C 7K-365S Cc1c(nc(nn1)c2ccccc2)N3CCOCC3 7K-366S COc1ccc(cc1)S(=O)(=O)N(CC(=O)O)c2ccccc2 7K-367S Cc1c(nc(nn1)c2ccccc2)Sc3ccccc3Cl 7K-374S CCOC(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(cc2)Cl 7K-375S COc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccc(cc2Cl)Cl)c3ccccc3 7K-376S Cc1ccc(cc1)c2nc(c(nn2)C)O 7K-377S Cc1ccc(cc1)c2nc(c(nn2)C)N3CCCC3 7K-382S Cc1ccc(cc1)c2cc3ccccc3[nH+]c2Cl.OS(=O)(=O)[O-] 7K-383S Cc1ccccc1Sc2c(cc3ccccc3n2)c4ccc(cc4)Cl 7K-384S c1ccc2c(c1)cc(c(n2)Sc3ccccc3Cl)c4ccc(cc4)Cl 7K-386S CN(C)C(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(cc2)OC 7K-387S CC(C)(C#C)NC(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(cc2)OC 7K-388S c1ccc2c(c1)cc(c(n2)N3CCOCC3)c4ccc(cc4)Cl 7K-390S Cc1ccc(cc1)c2nc(c(nn2)C)Sc3c(cccc3Cl)Cl 7K-391S Cc1ccc(cc1)c2nc(c(nn2)C)Sc3cccc(c3)C(F)(F)F 7K-392S COc1ccc(cc1)S(=O)(=O)N(CC(=O)Nc2ccccc2)c3ccccc3 7K-393S c1ccc(cc1)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)Cl 7K-394S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccccc3 7K-501S CCOC(=O)c1c(nc(nn1)c2ccccc2)N3CC(OC(C3)C)C 7K-502S CCOC(=O)c1c(nc(nn1)c2ccccc2)N3CCSCC3 7K-503S CCOC(=O)c1c(nc(nn1)c2ccccc2)NC 7K-505S CCOC(=O)c1c(nc(nn1)c2ccccc2)NOC 7K-510S CCOC(=O)c1c(nc(nn1)c2ccccc2)N(C)c3ccccc3 7K-511S CCOC(=O)c1c(nc(nn1)c2ccccc2)NCc3ccccc3 7K-512S CCOC(=O)c1c(nc(nn1)c2ccccc2)NCc3ccc(cc3)Cl 7K-513S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccc(cc3)C 7K-514S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccc(cc3Cl)Cl 7K-515S CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)Cl 7K-518S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccccc3C 7K-519S CCOC(=O)n1c2ccccc2n(c1=O)Cc3cccc(c3)C 7K-520S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccc(c(c3)Cl)Cl 7K-521S CCOC(=O)n1c2ccccc2n(c1=O)Cc3c(cccc3Cl)Cl 7K-522S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccccc3Cl 7K-523S CCOC(=O)n1c2ccccc2n(c1=O)Cc3cccc(c3)F 7K-526S CCOC(=O)n1c2ccccc2n(c1=O)C 7K-527S CCOC(=O)n1c2cc(ccc2[nH]c1=O)Br 7K-528S c1ccc2c(c1)cc(c(n2)Cl)c3cccc(c3)C(F)(F)F 7K-530S CCOC(=O)n1c2cc(ccc2n(c1=O)C)Br 7K-533S CCOC(=O)n1c2cc(ccc2n(c1=O)CC=C)Br 7K-534S CCOC(=O)n1c2cc(ccc2n(c1=O)Cc3ccc(c(c3)Cl)Cl)Br 7K-535S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccc(cc3)OC 7K-538S CCOC(=O)n1c2ccccc2n(c1=O)Cc3ccc(cc3)F 7K-539S CCOC(=O)n1c2cc(ccc2n(c1=O)C)Cl 7K-542S CCOC(=O)n1c2cc(ccc2n(c1=O)CC=C)Cl 7K-543S Cc1cccc(c1)C(=O)NNC(=O)c2ccccc2SC 7K-544S Cc1cccc(c1)c2nnc(o2)c3ccccc3SC 7K-545S Cc1cccc(c1)C(=O)CC(c2ccc(cc2)Br)C(=O)OC 7K-557S Cc1cccc(c1)C2=NNC(=O)C(C2)c3ccc(cc3)Br 7K-558S Cc1ccc(cc1)C2=NNC(=O)C(C2)c3ccc(cc3)Cl 7K-567S c1ccc(cc1)c2cc3ccccc3nc2Sc4ccccc4 7K-569S c1ccc(cc1)c2cc3ccccc3nc2Sc4ccc(cc4)Cl 7K-571S c1cc(ccc1SCC(=O)Nc2nnc(s2)C(F)(F)F)Br 7K-574S c1cc(ccc1SCC(=O)Nc2nnc(s2)C(F)(F)F)Cl 7K-575S c1ccc(c(c1)SCC(=O)Nc2nnc(s2)C(F)(F)F)Cl 7K-576S COc1ccc(cc1)SCC(=O)Nc2nnc(s2)C(F)(F)F 7K-577S c1cc(cc(c1)Cl)SCC(=O)Nc2nnc(s2)C(F)(F)F 7K-578S c1cc(c(c(c1)Cl)Cl)SCC(=O)Nc2nnc(s2)C(F)(F)F 7K-579S Cc1ccccc1SCC(=O)Nc2nnc(s2)C(F)(F)F 7K-580S COC(=O)c1ccccc1SCC(=O)Nc2nnc(s2)C(F)(F)F 7K-581S c1ccc(c(c1)C2=NNC(=O)C(C2)c3ccc(cc3)Cl)F 7K-585S Cc1cc(ccc1Cl)C(=O)CC(C#N)c2ccc(cc2)Cl 7K-587S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)N3CCSCC3 7K-591S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)N3CCCC3 7K-592S c1ccc(cc1)c2cc3ccccc3nc2Sc4ccc(cc4)F 7K-599S COc1ccccc1Sc2c(cc3ccccc3n2)c4ccccc4 7K-600S c1ccc(cc1)c2cc3ccccc3nc2Sc4cccc(c4)Cl 7K-602S c1ccc(cc1)c2cc3ccccc3nc2Sc4cc(ccc4Cl)Cl 7K-603S COc1ccc(cc1)Sc2c(cc3ccccc3n2)c4ccccc4 7K-606S c1ccc(cc1)c2cc3ccccc3nc2Sc4ccc(cc4Cl)Cl 7K-609S COc1ccc(cc1)S(=O)(=O)CC(=O)Nc2nnc(s2)C(F)(F)F 7K-610S c1cc(ccc1S(=O)(=O)CC(=O)Nc2nnc(s2)C(F)(F)F)Br 7K-611S c1cc(cc(c1)Cl)S(=O)(=O)CC(=O)Nc2nnc(s2)C(F)(F)F 7K-612S Cc1ccc(cc1)S(=O)(=O)CC(=O)Nc2nnc(s2)C(F)(F)F 7K-613S c1ccc(cc1)SCC(=O)Nc2nnc(s2)C(F)(F)F 7K-614S c1cc(c(cc1Cl)SCC(=O)Nc2nnc(s2)C(F)(F)F)Cl 7K-615S CSc1ccccc1c2nnc(o2)c3ccc(c(c3)Cl)Cl 7K-619S COc1ccc(cc1)c2nnc(o2)c3ccccc3SC 7K-621S CSc1ccccc1c2nnc(o2)c3ccc(cc3)F 7K-623S CSc1ccccc1c2nnc(o2)c3ccccc3 7K-625S CCOC(=O)c1c(nc(nn1)c2cccs2)N3CCOCC3 7K-626S CCOC(=O)c1c(nc(nn1)c2cccs2)N3CC(OC(C3)C)C 7K-627S CCOC(=O)c1c(nc(nn1)c2cccs2)N3CCSCC3 7K-628S CCOC(=O)c1c(nc(nn1)c2cccs2)N3CCCC3 7K-629S CCOC(=O)c1c(nc(nn1)c2cccs2)NCC=C 7K-631S CCOC(=O)c1c(nc(nn1)c2cccs2)NCc3ccccc3 7K-632S Cc1ccc(cc1)S(=O)(=O)C/C(=N/O)/N 7K-633S CCOC(=O)c1c(nc(nn1)c2cccs2)NC3CCCCC3 7K-636S CCOC(=O)c1c(nc(nn1)c2cccs2)Oc3ccc(cc3)Cl 7K-638S CSc1ccccc1c2nnc(o2)c3ccc(cc3)Cl 7K-641S Cc1ccc(cc1)c2nnc(o2)c3ccccc3SC 7K-643S CSc1ccccc1c2nnc(o2)c3ccc(cc3Cl)Cl 7K-645S CS(=O)(=O)c1ccccc1c2nnc(o2)c3ccc(c(c3)Cl)Cl 7K-649S COc1ccc(cc1)c2nnc(o2)c3ccccc3S(=O)(=O)C 7K-650S CS(=O)(=O)c1ccccc1c2nnc(o2)c3ccc(cc3)Cl 7K-657S c1ccc(cc1)CSc2ccccc2C(=O)O 7K-659S c1cc(sc1)c2nnc(o2)c3cccs3 7K-661S CSc1ccccc1c2nnc(o2)c3ccc(cc3)Br 7K-663S c1ccc(cc1)c2nc(cc(n2)O)CSc3ccccc3 7K-664S c1ccc2cc(ccc2c1)C(=O)CBr 7K-900 c1ccc2cc(ccc2c1)C(=O)C[N+]34CN5CN(C3)CN(C5)C4.[Br-] 7K-901 COC(=O)c1ccc(cc1)C[P+](c2ccccc2)(c3ccccc3)c4ccccc4.[Br-] 7K-902 c1ccc2cc(ccc2c1)C(=O)CN.Cl 7K-903 c1ccc2cc(ccc2c1)C(CN)O 7K-904 c1ccc2cc(ccc2c1)C(CNC(=O)c3c(cccc3F)F)O 7K-905 c1ccc2cc(ccc2c1)C(CNC(=O)c3c(cccc3F)F)Cl 7K-906 COC(=O)C(COC(=O)c1c(cccc1F)F)NC(=O)c2c(cccc2F)F 7K-907 CC1(C2NC(=S)N(N2C(=S)N1)c3ccccc3)c4ccc(cc4)OC 7K-911 c1c(=O)[nH]c(=O)[nH]c1Cl 7K-912 c1ccc(c(c1)N)Sc2c[nH]c(=O)[nH]c2=O 7K-913 Cc1c(c(c(c(n1)/C=C/N(C)C)C#N)c2ccccc2OC)C#N 7K-914 CCCCCCCCCCC/C=C/c1ccc(cc1)C(=O)OC 7K-915 CCCCCCCCCCC/C=C/c1ccc(cc1)C(=O)O 7K-916 COC(=O)c1c(noc1c2cn(nc2C(F)(F)F)c3ccc(cc3)F)c4c(cccc4Cl)Cl 7L-001 c1cc(ccc1/C=C\2/C(=O)C3CCN2CC3)Cl 7L-002 CN(C)/C=C/C(=O)c1ccc2ccccc2c1 7L-003 CCOC(=O)C(=O)/C(=C\N(C)C)/c1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC 7L-004 COc1ccc(cc1)N/C=C/C(=O)c2ccc3ccccc3c2 7L-005 c1ccc2cc(ccc2c1)C(=O)/C=C/Nc3ccc(cc3)I 7L-006 c1ccc2cc(ccc2c1)C(=O)/C=C/Nc3ccc(cc3)Cl 7L-007 CCOC(=O)c1c(cn(n1)c2ccc(cc2)C)c3c(c(no3)c4ccccc4Cl)C(=O)OC 7L-008 c1cc(ccc1/C=C\2/C(=O)C3CCN2CC3)F 7L-009 Cc1c(c(on1)C=O)[N+](=O)[O-] 7L-011 Cc1ncc(c(n1)C(F)(F)F)c2c(c(no2)c3c(cccc3Cl)Cl)C(=O)OC 7L-012 c1ccc2c(c1)C(=O)N(C2=O)OCc3ccc(cc3)[N+](=O)[O-] 7L-013 c1cc(ccc1CON)[N+](=O)[O-].Cl 7L-014 c1cc(ccc1c2cc(n[nH]2)C3CCNCC3)Cl 7L-015 c1ccc(cc1)C(=O)c2ccc(s2)CC(=O)O 7L-016 c1cc(c(cc1Cl)Cl)C(=O)c2ccc(s2)CC#N 7L-017 c1cc(c(cc1Cl)Cl)C(=O)c2ccc(s2)CC(=O)O 7L-018 c1cc(ccc1NC(=O)CCCCl)Oc2c(cc(cn2)C(F)(F)F)Cl 7L-019 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)CCCCl 7L-020 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)CCCCl 7L-021 c1ccc(c(c1)n2cccc2)O 7L-022 CC(C(=O)C)Oc1ccccc1Oc2c(cc(cn2)C(F)(F)F)Cl 7L-023 CC(C(=O)C)Oc1ccccc1n2cccc2 7L-024 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2CCCC2=O 7L-025 c1csc(n1)NC(=O)CCCCl 7L-027 CCNC(=O)Oc1ccccc1n2cccc2 7L-028 c1csc(n1)N2CCCC2=O 7L-029 c1cc(ncc1Cl)NC(=O)CCCCl 7L-030 Cc1cc2c(cc1C(=O)OCc3ccccc3)c(=O)c4ccccc4o2 7L-056 Cc1nnc(s1)Nc2cc(c(cc2Cl)Cl)OCCOC 7L-303S c1cc(ccc1C(C(=O)O)N)Cl 7L-304S c1cc(cc(c1)C(F)(F)F)C(=O)C/N=C/c2ccc(nc2)Oc3cccc(c3)C(F)(F)F 7L-307S c1cc(cc(c1)F)CO/N=C/c2ccc(nc2)Oc3ccc(cc3)C#N 7L-308S COc1cccc(c1)C(C(=O)O)N 7L-312S c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C/c2ccc(nc2)Oc3ccc(cc3)C#N 7L-313S c1cc(ccc1C#N)Oc2ccc(cn2)/C=N/OC(=O)c3ccc(cc3Cl)Cl 7L-314S COc1cc(c(cc1Cl)Cl)n2c(=O)c3ccc(cc3nc2S)Cl 7L-317S Cc1ccc2c(c1)c(=O)n(c(n2)S)c3cc(c(cc3Cl)Cl)OC 7L-318S CO/N=C/c1ccc(nc1)Sc2ccccc2Cl 7L-320S c1ccc(c(c1)Sc2ccc(cn2)/C=N/OCc3ccc(cc3Cl)Cl)Cl 7L-321S Cc1c(oc(n1)c2ccccc2)C(=O)NC 7L-322S CCOC(=O)Oc1cc(c(cc1Cl)Cl)N 7L-324S CC(=O)NC(C#N)c1ccc(cc1)Cl 7L-325S CC(C(=O)O)NC(=O)c1ccc(cc1)Cl 7L-326S Cc1ccc(cc1)C2=N/C(=C/N(C)C)/C(=O)O2 7L-327S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)O 7L-328S CC(C)Oc1cc(c(cc1Cl)Cl)N2C(=O)CSCC2=O 7L-329S COc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)O 7L-330S COCCOc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)O 7L-331S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)CSCC(=O)O 7L-333S CC(=O)NC(C#N)c1cccc(c1)OC 7L-337S c1ccc(cc1)C(CC(=O)O)N 7L-339S Cc1nnc(s1)Nc2cc(c(cc2Cl)Cl)OC 7L-340S Cc1nnc(s1)Nc2cc(c(cc2Cl)Cl)OC(C)C 7L-341S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)n3c(=O)c4ccccc4nc3SCc5ccccc5 7L-344S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)O 7L-345S CCOC(=O)COc1cc(c(cc1Cl)Cl)N2C(=O)CSCC2=O 7L-346S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)N3C(=O)CSCC3=O 7L-347S COc1cc(c(cc1Cl)Cl)N2C(=O)CSCC2=O 7L-348S COCCOc1cc(c(cc1Cl)Cl)N2C(=O)CSCC2=O 7L-349S CCOC(=O)c1nc(n(n1)c2cc(c(cc2Cl)Cl)OC)C 7L-351S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)O 7L-352S COc1ccc(cc1)S(=O)(=O)NC(c2cccs2)C(=O)O 7L-354S Cc1c(oc(n1)c2ccc(cc2)Cl)C(=O)OC 7L-355S Cc1ccc(cc1)c2nc(no2)C(=O)OC 7L-356S COCCOc1cc(c(cc1Cl)Cl)Nc2nnc(s2)C(F)(F)F 7L-360S Cc1ccc(cc1)c2nc(no2)C(=O)O 7L-361S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3ccccc3nc2S 7L-365S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3ccc(cc3)Br 7L-367S Cc1c(cccc1Cl)NC(=O)c2nc(n(n2)c3cc(c(cc3Cl)Cl)OC)C 7L-368S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3ccccc3OC 7L-369S CCOC(=O)COc1cc(c(cc1Cl)Cl)n2c(=O)c3ccccc3nc2S 7L-371S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3cccc(c3)C(F)(F)F 7L-372S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3ccc(cc3)Oc4ccccc4 7L-373S c1ccc(cc1)c2nc(cs2)CC(=O)O 7L-375S COc1cc(c(cc1Cl)Cl)n2c(=O)c3ccc(cc3nc2SC)Cl 7L-376S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3ccc(cc3C(F)(F)F)Cl 7L-380S Cc1ccc(cc1)NC(=O)OCc2ccccc2S(=O)C 7L-502S CS(=O)c1ccccc1COC(=O)Nc2cccc(c2)Cl 7L-503S COc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccccc3[N+](=O)[O-] 7L-505S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccccc3[N+](=O)[O-] 7L-506S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3c(ccs3)Oc4ccccc4[N+](=O)[O-] 7L-507S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccccc3[N+](=O)[O-] 7L-508S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccccc3[N+](=O)[O-] 7L-509S COc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-] 7L-510S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-] 7L-511S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3c(ccs3)Oc4ccc(cc4)[N+](=O)[O-] 7L-512S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-] 7L-513S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3)[N+](=O)[O-] 7L-514S COC(=O)c1ccccc1SCc2ccccc2SC 7L-515S CSc1ccccc1CSc2c(cccc2Cl)Cl 7L-516S CSc1ccccc1CSc2ccc(cc2)Br 7L-517S CSc1ccccc1c2nnc(o2)SCc3ccc(c(c3)Cl)Cl 7L-518S CSc1ccccc1c2nnc(o2)SCC#C 7L-519S CCSc1nnc(o1)c2ccccc2SC 7L-521S CSc1ccccc1CSc2ccc(cc2)Cl 7L-523S CCn1c(nnc1SCc2c(cccc2Cl)Cl)c3ccccc3SC 7L-524S Cc1ccc(cc1)CSc2nnc(o2)c3ccccc3SC 7L-525S c1ccc(cc1)c2c(nc(nn2)c3ccccn3)Oc4cccc(c4)C(F)(F)F 7L-526S CCOC(=O)CSc1nnnn1c2cc(c(cc2Cl)Cl)OC 7L-527S COc1cc(c(cc1Cl)Cl)n2c(nnn2)SCC=C 7L-528S COc1cc(c(cc1Cl)Cl)n2c(nnn2)SCC#C 7L-529S CNc1c(nnc(n1)c2ccccn2)c3ccccc3 7L-530S CSc1ccccc1c2nnc(o2)SCc3ccccc3 7L-532S CSc1ccccc1c2nnc(o2)SCc3ccc(cc3)F 7L-533S CSc1ccccc1c2nnc(o2)SCc3cccc(c3)Cl 7L-534S CC(C)(C)c1ccc(cc1)CSc2nnc(o2)c3ccccc3SC 7L-535S CSc1ccccc1c2nnc(n2c3ccccc3)S 7L-536S CSc1ccccc1c2nnc(n2c3ccccc3)SC 7L-537S CCOC(=O)CSc1nnc(n1c2ccccc2)c3ccccc3SC 7L-538S c1ccc(cc1)CNc2c(nnc(n2)c3ccccn3)c4ccccc4 7L-539S CN(C)c1c(nnc(n1)c2ccccn2)c3ccccc3 7L-540S Cc1ccc(cc1)CSc2nnc(n2c3ccccc3)c4ccccc4SC 7L-541S CSc1ccccc1c2nnc(n2c3ccccc3)SCc4ccc(c(c4)Cl)Cl 7L-542S c1ccc(cc1)c2c(nc(nn2)c3ccccn3)Oc4ccccc4 7L-543S COc1cc(c(cc1Cl)Cl)n2c(=O)c3ccccc3nc2SCC=C 7L-545S COCCOc1cc(c(cc1Cl)Cl)n2c(=O)c3cc(c(cc3c(n2)c4ccc(cc4)Cl)Cl)Cl 7L-546S COCCOc1cc(c(cc1Cl)Cl)n2c(=O)c3ccccc3c(n2)c4ccc(cc4)Cl 7L-547S COc1cc(c(cc1Cl)Cl)n2c(=O)c3ccccc3c(n2)c4ccc(cc4)Cl 7L-548S COc1cc(c(cc1Cl)Cl)n2c(=O)c3cc(c(cc3c(n2)c4ccc(cc4)Cl)Cl)Cl 7L-549S CSc1ccccc1CSc2ccccc2C(=O)O 7L-551S CSc1ccccc1c2nc(no2)c3ccc(cc3)Cl 7L-552S C=CCNc1c(nnc(n1)c2ccccn2)c3ccccc3 7L-553S COc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 7L-554S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 7L-555S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3c(ccs3)Oc4ccc(cc4F)[N+](=O)[O-] 7L-556S CCOC(=O)COc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 7L-557S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3F)[N+](=O)[O-] 7L-558S CSc1ccccc1c2nc(no2)c3cccc(c3)Cl 7L-559S CSc1ccccc1c2nc(no2)c3cccc(c3)C(F)(F)F 7L-560S c1ccc(cc1)c2c(nc(nn2)c3ccccn3)NC4CCCCC4 7L-563S CS(=O)c1ccccc1c2nc(no2)c3cccc(c3)C(F)(F)F 7L-564S CS(=O)c1ccccc1c2nc(no2)c3cccc(c3)Cl 7L-565S CS(=O)c1ccccc1c2nc(no2)c3ccc(cc3)Cl 7L-566S COc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F 7L-567S CC(C)Oc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F 7L-568S c1ccc(cc1)COc2cc(c(cc2Cl)Cl)NC(=O)c3c(ccs3)Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F 7L-569S c1ccc(cc1)C2=NNC(=O)CC2 7L-571S CS(=O)(=O)c1ccccc1c2nc(no2)c3cccc(c3)Cl 7L-572S CS(=O)(=O)c1ccccc1c2nc(no2)c3cccc(c3)C(F)(F)F 7L-573S CC(C)C(=O)Nc1cccn2c1nnc2C(F)(F)F 7L-576S CC(C)(C)C(=O)Nc1cccn2c1nnc2C(F)(F)F 7L-577S c1cc(c2nnc(n2c1)C(F)(F)F)NC(=O)C3CC3 7L-579S c1ccc(cc1)C2=NN(CCC2)C(=O)c3ccc(c(c3)Cl)Cl 7L-581S CSc1ccccc1c2nc(no2)c3ccc(cc3)[N+](=O)[O-] 7L-583S COc1ccc(cc1)C(=O)N2CCCC(=N2)c3ccccc3 7L-584S CC(CSc1c(cccc1Cl)Cl)(C(=O)Nc2cc(c(cc2Cl)Cl)OCCOC)O 7L-585S Cc1ccc(cc1)C(=O)N2CCCC(=N2)c3ccccc3 7L-587S c1ccc(cc1)C2=NN(CCC2)C(=O)c3ccc(cc3)Cl 7L-589S CS(=O)c1ccccc1c2nc(no2)c3ccc(cc3)[N+](=O)[O-] 7L-590S CS(=O)(=O)c1ccccc1c2nc(no2)c3ccc(cc3)[N+](=O)[O-] 7L-591S Cc1c(snn1)C(=O)Nc2ccc(cc2Cl)Cl 7L-592S CSc1ccccc1c2nc(no2)c3ccccn3 7L-593S CCOC(=O)C1=C(N(C(=O)CC1c2ccc(cc2)Cl)CC#N)C 7L-703 c1cc(ccc1/C=N/NC(=O)CC#N)Cl 7L-704 Cc1ccsc1/C=N/NC(=O)CC#N 7L-706 CN(C)c1ccc(cc1)/C=N\NC(=O)CC#N 7L-707 COC(=O)c1c(noc1c2cnc(nc2C(F)(F)F)c3ccccc3)c4ccccc4 7L-712 CN(C)/C=C/c1ccc2ccccc2c1[N+](=O)[O-] 7L-714 COc1ccc(cc1)/C=C/2\C(=O)C3CCN2CC3 7L-715 Cc1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N 7L-716 CCOC(=O)c1c(cn(n1)c2ccc(cc2)F)c3c(c(no3)c4c(cccc4Cl)F)C(=O)OC 7L-717 CCOC(=O)c1c(cn(n1)c2ccc(cc2Cl)Cl)c3c(c(no3)c4ccccc4Cl)C(=O)OC 7L-719 CCOC(=O)c1c(cn(n1)c2ccccc2Cl)c3c(c(no3)c4c(cccc4Cl)Cl)C(=O)OC 7L-720 c1cc(ccc1C=C(C#N)C#N)Cl 7L-721 CO/N=C/NC(=O)c1c(cc(=O)n(n1)c2ccccc2)O 7L-722 CCOC(=O)c1c(cn(n1)c2ccc(cc2)C)c3c(c(no3)c4ccccc4)C(=O)OC 7L-723 CCOC(=O)c1c(cn(n1)c2cccc(c2)Cl)c3c(c(no3)c4c(cccc4Cl)Cl)C(=O)OC 7L-724 c1cc(ccc1N/C=C(/C=C/C#N)\C#N)F 7L-730 c1cc(oc1)/C=C/2\C(=O)C3CCN2CC3 7L-732 CCOC(=O)c1c(c(c(=O)n(c1N)N)C#N)c2ccc(cc2)Cl 7L-733 c1cc(ccc1N/C=C(/C=C/C#N)\C#N)I 7L-734 c1cc(c(cc1Cl)Cl)/C=C\2/C(=O)C3CCN2CC3 7L-735 Cc1ccc(cc1)N/C=C/c2ccc3ccccc3c2[N+](=O)[O-] 7L-736 c1cc(ccc1CN2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)Cl)Cl 7L-737 CCOC(=O)c1c(c(c(=O)n(c1N)N)C#N)c2ccc(cc2)OC 7L-738 c1ccc2c(c1)ccc(c2[N+](=O)[O-])C/C=N/O 7L-739 c1ccc(c(c1)/C=N/NC(=O)CC#N)C(F)(F)F 7L-740 CCOC(=O)c1c(c(c(=O)n(c1N)N)C#N)c2ccc(cc2)N(C)C 7L-741 Cc1ccc(cc1)CN2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)Cl 7L-742 CC(C)(CCl)C(=O)Nc1ccc(cc1)C(F)(F)F 7L-743 c1ccc2c(c1)ccc(c2[N+](=O)[O-])CC#N 7L-744 CC1(CN(C1=O)c2ccc(cc2)C(F)(F)F)C 7L-745 CC(=O)c1ccc(cc1)NC(=O)C(C)(C)CCl 7L-746 CC(=O)c1ccc(cc1)N2CC(C2=O)(C)C 7L-747 C1SC(=[NH2+])NC(=N)S1.[I-] 7L-800 CCOC(=O)c1c(nc(s1)NC(=O)Nc2ccccc2)c3ccccc3 7L-801 CCOC(=O)C(=CNc1nc(cs1)c2ccc(cc2)Cl)C(=O)OCC 7L-802 c1ccc2c(c1)CCN(C2)c3cc(nc(n3)N)Cl 7L-803 Cc1ccc(cc1Cl)Nc2cc(nc(n2)N)Cl 7L-804 c1ccc(c(c1)/C=N/NC(=O)Nc2ccncc2)O 7L-805 CSc1nc(c(c(n1)O)/N=N/c2ccc(cc2F)F)O 7L-806 c1cc(ccc1F)Sc2cc(nc(n2)N)Cl 7L-807 c1ccc2c(c1)CCCN2c3cc(nc(n3)N)Cl 7L-808 CSc1nc(cc(n1)Cl)Sc2ccc(cc2)F 7L-809 c1ccc2c(c1)c(c[nH]2)/C=N/Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F 7L-810 c1ccc(cc1)CNc2cc(nc(n2)N)Cl 7L-811 COC(=O)CCSc1cc(nc(n1)N)Cl 7L-812 COc1ccc(cc1OC)Nc2cc(nc(n2)N)Cl 7L-813 c1ccc(cc1)Oc2ccc(cc2)Nc3cc(nc(n3)N)Cl 7L-814 Cc1cccc(c1C)N2CCN(CC2)c3cc(nc(n3)N)Cl 7L-815 c1cc(ccc1CCNc2cc(nc(n2)N)Cl)O 7L-816 c1cc(ccc1Sc2cc(nc(n2)N)N3CCCCC3)Cl 7L-817 c1ccc(cc1)Sc2cc(nc(n2)N)Cl 7L-818 CC(C)Sc1cc(nc(n1)N)Cl 7L-819 c1ccc(cc1)c2csc3n2c4cc(ccc4n3)OC(F)F 7L-820 CN(C)c1ccc(cc1)/C=N\NC(=O)OC 7L-821 Cc1ccc(cc1)SCc2ccc(cc2)CSc3ccc(cc3)C 7L-823 c1cc(sc1)Sc2cc(nc(n2)N)Cl 7L-824 COc1cccc(c1O)/C=N/NC(=O)OCCO 7L-826 CC(C)(C)c1c(sc([nH+]1)N)Br.[Br-] 7L-827 CC(C)(C)c1c(sc(n1)N)SC#N 7L-828 c1ccc(cc1)Nc2cc(nc(n2)N)Cl 7L-829 CCCN(CCC)c1cc(nc(n1)N)Cl 7L-830 c1cc(ccc1Nc2cc(nc(n2)N)Cl)Cl 7L-831 COc1ccc(cc1)Nc2cc(nc(n2)N)Cl 7L-832 CCOc1ccccc1N2CCN(CC2)c3cc(nc(n3)N)Cl 7L-833 CCN(CC)c1cc(nc(n1)N)Cl 7L-834 c1c(nc(nc1Cl)N)N2CCOCC2 7L-836 c1c(nc(nc1Cl)N)N2CCCCC2 7L-837 c1cc(ccc1N)Sc2cc(nc(n2)N)Cl 7L-838 c1cc(ccc1Sc2cc(nc(n2)N)N3CCOCC3)Cl 7L-839 C[NH+]1CCN(CC1)c2cc(nc(n2)SC)Cl.[Cl-] 7L-840 CSc1nc(cc(n1)Cl)N2CCOCC2 7L-841 CSc1nc(cc(n1)Cl)Nc2ccc(cc2)F 7L-842 COc1ccc2c(c1)n(c(=S)[nH]2)CC(=O)c3ccccc3 7L-843 CCOC(=O)C(=CNc1nc(cs1)C(C)(C)C)C(=O)OCC 7L-844 CC(=O)c1cc(c(cc1NC(=O)Nc2ccccc2)OC)OC 7L-845 c1cc(ccc1/N=N/c2c(nc(nc2O)N)N)Cl 7L-847 c1ccc2c(c1)c3ccccc3n2c4ccc(cc4[N+](=O)[O-])C(F)(F)F 7L-848 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=N\NC(=O)Nc2ccccc2 7L-849 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)[N+](=O)[O-] 7L-850 c1cc(c(cc1F)F)/N=N/c2c(nc(nc2O)N)O 7L-851 c1cc(c(cc1F)F)/N=N/c2c(nc(nc2O)O)O 7L-852 c1ccc(cc1)/N=N/c2c(ncnc2O)O 7L-853 c1c(cnc(c1Cl)NCC(CC#N)OC(=O)C2CC2)C(F)(F)F 7L-900 C1COCN2N1CN3COCCN3C2 7L-901 C1CC2N3CCOC4N3C(CCC4)N5N2C(C1)OCC5 7L-902 Cn1cc(c2c1cccc2)CC(=O)O 7L-904 c1ccc2c(c1)c(cn2Cc3ccc(cc3)F)CC(=O)O 7L-905 c1ccc2c(c1)c(cn2c3ccc(nn3)Cl)CC(=O)O 7L-906 C/C(=N/Nc1ccccc1)/c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 7L-907 CC(=O)c1cn(c(=O)[nH]c1=O)CC=C 7L-908 c1ccc2c(c1)c(cn2Cc3cccc(c3)Cl)CC(=O)O 7L-909 C/C(=N/OC/C=C/Cl)/c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 7L-910 c1cc(cc(c1)C(F)(F)F)C(=O)OC(CC#N)CNc2c(cc(cn2)C(F)(F)F)Cl 7L-911 Cc1ccc(cc1)C(=O)O/C(=C(\C#N)/C(=O)Nc2cccc(c2)C(F)(F)F)/C 7L-913 C/C(=N/N(C)c1c(cc(cn1)C(F)(F)F)Cl)/c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 7L-914 COC(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 7L-915 COC(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)N 7L-916 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)NN)Cl 7L-917 COC(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)n3cccc3 7L-918 c1cc(cc(c1)NC(=O)NNC(=O)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-])C(F)(F)F 7L-919 c1cc(nc(c1)F)N2CCC(=NNC(=O)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-])CC2 7L-920 CN(C)c1ccc(cc1)/C=N/NC(=O)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 7L-921 C=CCNC(=O)c1ccccc1Cl 7L-922 c1cc(cc(c1)[N+](=O)[O-])C(=O)OC(CC#N)CNc2c(cc(cn2)C(F)(F)F)Cl 7L-923 c1ccc2c(c1)C(=O)N(C2=O)OCC3CC3 7L-924 c1cc(oc1)C(=O)OC(CC#N)CNc2c(cc(cn2)C(F)(F)F)Cl 7L-925 CC(=O)c1cn(c(=O)[nH]c1=O)CC2CC(N(O2)C)c3ccc(cc3)OC 7L-926 COC(=O)CCCNc1ncccn1 7L-927 c1cc(c(cc1Cl)Cl)C(=O)OC(CC#N)CNc2c(cc(cn2)C(F)(F)F)Cl 7L-928 c1ccc2c(c1)ncc(n2)SCC(=O)c3ccc(s3)Cc4c(cc(cn4)C(F)(F)F)Cl 7M-001 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)C(=O)CSc3nc[nH]n3 7M-002 c1cc[n+](c(c1)SCC(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl)[O-] 7M-003 c1ccc(cc1)NC(=O)c2ccccc2CC[N+](=O)[O-] 7M-004 c1cc(cnc1)c2nnc(o2)SCC(=O)c3ccc(s3)Cc4c(cc(cn4)C(F)(F)F)Cl 7M-005 CCOC(=O)c1ccc(cc1)NC(=O)c2ccccc2CC[N+](=O)[O-] 7M-006 COc1cc(cc(c1OC)OC)NC(=O)c2ccccc2CC[N+](=O)[O-] 7M-007 c1cc(ncc1C(F)(F)F)SCC(=O)c2ccc(s2)Cc3c(cc(cn3)C(F)(F)F)Cl 7M-008 c1cc(sc1)/C(=C/C(=O)[O-])/C#N.[K+] 7M-009 COc1ccc(cc1)/C(=C/C(=O)[O-])/C#N.[K+] 7M-010 c1ccc(cc1)/C(=C/C(=O)NNc2ccccc2)/C(=O)O 7M-011 c1ccc(cc1)/C(=C/C(=O)NNc2ccc(cc2Cl)Cl)/C(=O)O 7M-012 Cc1c(cccc1Cl)NC(=O)c2ccccc2CC[N+](=O)[O-] 7M-014 CC(=O)Nc1ccc(cc1)NC(=O)c2ccccc2CC[N+](=O)[O-] 7M-015 c1cc(ccc1C2=CC(=O)N(C2=O)Nc3ccc(cc3Cl)Cl)Cl 7M-016 c1ccc(cc1)C2=CC(=O)N(C2=O)Nc3ccccc3 7M-017 c1ccc(cc1)C2=CC(=O)N(C2=O)Nc3ccc(cc3Cl)Cl 7M-018 c1cc(sc1)/C(=C\C(=O)O)/C(=O)O 7M-019 COc1ccc(cc1)/C(=C\C(=O)O)/C(=O)O 7M-020 Cc1cc(nc2c1c(c(s2)C(=O)c3ccc(s3)Cc4c(cc(cn4)C(F)(F)F)Cl)N)C 7M-021 c1cc(sc1)C2=CC(=O)OC2=O 7M-022 c1ccc(cc1)NN2C(=O)C=C(C2=O)c3ccc(cc3)Cl 7M-025 COc1ccnc(c1C#N)Oc2ccc(cc2)F 7M-026 COc1ccc(cc1)Oc2c(c(ccn2)OC)C#N 7M-027 COc1ccnc(c1C#N)Oc2ccccc2 7M-028 COc1ccc(cc1)C2=CC(=O)OC2=O 7M-030 COc1ccc(cc1)/C(=C\C(=O)NNc2ccccc2)/C(=O)O 7M-031 COc1ccc(cc1)/C(=C\C(=O)NNc2ccc(cc2Cl)Cl)/C(=O)O 7M-032 COc1ccc(cc1)/C(=C/C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)/C(=O)O 7M-033 Cc1c(c(on1)N)Cl 7M-034 COc1ccc(cc1)C2=CC(=O)N(C2=O)Nc3ccc(cc3Cl)Cl 7M-035 COc1ccc(cc1)C2=CC(=O)N(C2=O)Nc3ccccc3 7M-036 COc1ccc(cc1)C2=CC(=O)N(C2=O)Nc3c(cc(cn3)C(F)(F)F)Cl 7M-037 CC(=O)Nc1ccc(cc1)Oc2c(c(ccn2)OC)C#N 7M-040 Cc1ccc(c(c1)C)Oc2c(c(ccn2)OC)C#N 7M-041 CCSc1nnc(n1C)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 7M-043 CN(C)/C=N/C(=O)c1c(ccnc1Oc2ccc(cc2)Cl)OC 7M-044 COc1ccnc(c1c2nc[nH]n2)Oc3ccc(cc3)Cl 7M-045 COc1ccnc(c1C#N)Oc2ccc3ccccc3c2 7M-046 COc1ccnc(c1C#N)Oc2cc(cc(c2)Cl)Cl 7M-047 Cc1ccc(cc1)Oc2c(c(ccn2)OC)C#N 7M-048 COc1ccnc(c1C#N)N2CCN(CC2)c3ccc(cc3)Cl 7M-049 Cc1cc2c(cc1Cc3cc4c(cc3C)OCO4)OCO2 7M-050 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)Cl 7M-051 c1cc(ccc1c2cc(on2)CNS(=O)(=O)c3ccc(cc3)Cl)Cl 7M-301S CC(C)C(=O)NCc1cc(no1)c2ccc(cc2)Cl 7M-302S COc1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3cc(ccc3Cl)Cl 7M-303S CC(=O)Nc1ccc(cc1)S(=O)(=O)NCc2cc(no2)c3ccc(cc3)OC 7M-304S Cc1cc(nc(c1S(=O)(=O)C)S(=O)Cc2ccc(cc2)OC)C 7M-305S Cc1cc(nc(c1S(=O)(=O)C)S(=O)(=O)Cc2ccc(cc2)OC)C 7M-306S c1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3ccccc3 7M-307S CC(C)C(=O)NCc1cc(no1)c2ccccc2 7M-308S c1ccc(cc1)c2cc(on2)COc3ccc(c(c3)Cl)Cl 7M-309S COc1ccccc1OCc2cc(no2)c3ccccc3 7M-310S Cc1cccc(c1C)OCc2cc(no2)c3ccccc3 7M-311S Cc1cc(ccc1OCc2cc(no2)c3ccccc3)Cl 7M-312S COc1cc2c(cc1OC)C(OCC2)c3ccc(cc3)[N+](=O)[O-] 7M-313S Cc1c(n2ccsc2n1)C(=O)Nc3ccc(cc3)Cl 7M-314S Cc1c(cccc1Cl)NC(=O)c2c(nc3n2ccs3)C 7M-315S Cc1c(n2ccsc2n1)C(=O)Nc3cccc(c3)C(F)(F)F 7M-316S CCCSc1c(c(cc(n1)C)C)S(=O)(=O)C 7M-317S CCCS(=O)c1c(c(cc(n1)C)C)S(=O)(=O)C 7M-318S CCCS(=O)(=O)c1c(c(cc(n1)C)C)S(=O)(=O)C 7M-319S c1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3ccccc3Cl 7M-320S c1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3ccc(cc3)Cl 7M-321S Cc1cc(nc(c1S(=O)(=O)C)Sc2ccc(cc2)Cl)C 7M-322S Cc1c(n2ccsc2n1)C(=O)NN 7M-324S c1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3cccc(c3Cl)Cl 7M-325S COc1ccc(c(c1)S(=O)(=O)NCc2cc(no2)c3ccccc3)OC 7M-326S COc1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3cc(ccc3OC)OC 7M-327S COc1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl 7M-328S c1ccc(cc1)c2cc(on2)CNS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl 7M-329S Cc1c(n2ccsc2n1)C(=O)NC(C)C 7M-331S Cc1cc(nc(c1)NC(=O)c2c(nc3n2ccs3)C)C 7M-332S Cc1c(n2ccsc2n1)C(=O)Nc3ccsc3C(=O)OC 7M-333S Cc1cc(nc(c1S(=O)(=O)C)S(=O)c2ccc(cc2)Cl)C 7M-334S Cc1cc(nc(c1S(=O)(=O)C)S(=O)(=O)c2ccc(cc2)Cl)C 7M-335S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)N3CCOCC3)C 7M-336S c1ccc(c(c1)c2cc(on2)COc3cc(c(cc3Cl)Cl)Cl)Cl 7M-337S Cc1cccc(c1C)OCc2cc(no2)c3ccc(cc3)Cl 7M-341S Cc1c(n2ccsc2n1)C(=O)NC 7M-344S c1ccc(cc1)c2cc(on2)COc3cc(c(cc3Cl)Cl)Cl 7M-346S COc1ccc(cc1)c2cc(on2)COc3cc(c(cc3Cl)Cl)Cl 7M-347S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)Sc3cccc(c3)C(F)(F)F)C 7M-348S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)Sc3ccc(cc3)Cl)C 7M-349S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)S(=O)c3ccc(cc3)Cl)C 7M-350S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)N(C)C)C 7M-353S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)N3CCN(CC3)C)C 7M-354S c1cc(ccc1c2cc(on2)COc3cc(c(cc3Cl)Cl)Cl)Cl 7M-355S COC(=O)c1ccc(cc1)OCc2cc(no2)c3ccc(cc3)Cl 7M-356S COc1ccc(cc1)c2cc3ccc(cc3s2)OC 7M-358S COc1ccc(cc1)c2cc(on2)COc3ccccc3 7M-359S COc1ccc(cc1)c2cc(on2)COc3ccc(c(c3)Cl)Cl 7M-360S COc1ccc(cc1)c2c(c3ccc(cc3s2)OC)Br 7M-361S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)NCc3ccc(cc3)OC)C 7M-362S Cc1cc(nc(c1S(=O)(=O)C)Sc2ccc(cc2)Cl)c3ccccc3 7M-363S Cc1cc(ccc1OCc2cc(no2)c3ccc(cc3)OC)Cl 7M-366S COc1ccc(cc1)c2cc3c(cccc3s2)OC 7M-367S Cc1cc(nc(c1S(=O)(=O)C)S(=O)c2ccc(cc2)Cl)c3ccccc3 7M-369S Cc1cc(nc(c1S(=O)(=O)C)S(=O)(=O)c2ccc(cc2)Cl)c3ccccc3 7M-370S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2OS(=O)(=O)c3ccc(cc3)C)C)C 7M-371S c1cc(ccc1CS(=O)(=O)CC#N)Cl 7M-372S c1ccc(cc1)c2cc(on2)CNC(=O)C(F)(F)F 7M-373S CC(=O)NCc1cc(no1)c2ccccc2 7M-374S CC(=O)NCc1cc(no1)c2ccc(cc2)Cl 7M-375S Cc1c(n2ccsc2n1)c3nnc(o3)SC(C)C 7M-377S Cc1cc(nc(c1S(=O)(=O)C)N2CCOCC2)c3ccccc3 7M-381S Cc1cc(nc(c1S(=O)(=O)C)N2CCCCC2)c3ccccc3 7M-383S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Cl)c3ccccc3)C 7M-385S c1ccc(cc1)NC(=O)OCCNC(=O)c2cccc(c2)Cl 7M-501S CCOC(=O)c1cc2c(nn(c2s1)C)CSc3ccccc3 7M-502S Cn1c(c(c(n1)c2ccccc2)CN3CCN(CC3)c4ncccn4)Cl 7M-504S c1cc(ccc1C(=O)C(F)(F)F)C(=O)N2CCOCC2 7M-507S c1cc(ccc1CNC(=O)c2ccc(cc2)C(=O)C(F)(F)F)Cl 7M-508S CC(C)NC(=O)c1ccc(cc1)C(=O)C(F)(F)F 7M-509S CN1CCN(CC1)C(=O)c2ccc(cc2)C(=O)C(F)(F)F 7M-510S Cn1c(c(c(n1)c2ccccc2)CN3CCN(CC3)c4ccccc4)Cl 7M-511S C/C(=N\O)/c1cc(no1)c2ccc(cc2)Cl 7M-512S c1cc(cc(c1)Cl)C(=O)NCCOC(=O)Nc2ccc(c(c2)Cl)Cl 7M-514S Cc1ccc(cc1)n2c(=O)c(c(cn2)Br)Oc3ccc(cc3)OC 7M-515S c1cc(ccc1n2c(=O)c(c(cn2)N3CCOCC3)Oc4ccc(cc4)Cl)F 7M-518S Cc1ccc(cc1)n2c(c(cn2)Br)C(=O)NC 7M-521S Cc1ccc(cc1)n2c(c(cn2)Br)C(=O)NCC=C 7M-522S Cc1ccc(cc1)n2c(=O)c(c(cn2)N3CCCCC3)Oc4ccc(cc4)OC 7M-524S CCOC(=O)/C(=N/Nc1cccc(c1)C(F)(F)F)/C(=O)C(F)(F)F 7M-527S C/C(=N\OC(=O)c1ccccc1)/c2cc(no2)c3ccc(cc3)Cl 7M-530S CC(C)CC(=O)O/N=C(/C)\c1cc(no1)c2ccc(cc2)Cl 7M-531S C/C(=N/OC(=O)C1CC1)/c2cc(no2)c3ccc(cc3)Cl 7M-532S c1ccc(cc1)NC(=O)OCCNC(=O)c2cccc(c2)Br 7M-533S c1cc(cc(c1)Br)C(=O)NCCOC(=O)Nc2ccc(cc2)Cl 7M-534S Cn1c(c(c(n1)c2ccccc2)CN3CCN(CC3)C)Cl 7M-536S Cn1c2c(cc(s2)C(=O)O)c(n1)CSc3ccccc3 7M-537S C/C(=N\OC(=O)c1cccc(c1)C(F)(F)F)/c2cc(no2)c3ccc(cc3)Cl 7M-538S Cc1ccc(cc1)n2c(c(cn2)Cl)C(=O)NCc3ccccc3 7M-539S CCCNC(=O)c1c(cnn1c2ccc(cc2)C)Cl 7M-540S Cc1c(nc(nn1)c2cccs2)O 7M-541S Cc1c(nc(nn1)c2ccc(cc2)Cl)O 7M-542S Cc1c(nc(nn1)c2cccc(c2)Cl)O 7M-543S c1ccc(cc1)CC(C(=O)NN)NC(=O)c2ccc(cc2)F 7M-544S Cc1ccc(cc1)n2c(=O)c(c(cn2)Cl)Sc3ccc(cc3)C 7M-549S c1ccc(cc1)c2cc(on2)C(=O)CSCc3cccc(c3)C(F)(F)F 7M-550S c1cc(cc(c1)C(F)(F)F)c2cc(ncn2)O 7M-551S c1cc(cc(c1)N/N=C(\C(=O)C(F)(F)F)/C(=O)O)C(F)(F)F 7M-552S c1cc(ccc1NC(=O)OCCNS(=O)(=O)c2ccc(cc2)Cl)Cl 7M-553S Cc1ccc(cc1)n2c(=O)c(c(cn2)NCC=C)Sc3ccc(cc3)C 7M-554S Cc1ccc(cc1)n2c(=O)c(c(cn2)NC)Sc3ccc(cc3)C 7M-555S c1ccc(cc1)CC(c2nnc(n2c3ccccc3)SCc4ccc(cc4)F)NC(=O)c5ccc(cc5)F 7M-557S COc1ccc(cc1)CSc2nnc(n2c3ccccc3)C(Cc4ccccc4)NC(=O)c5ccc(cc5)F 7M-558S CC(C)(C)c1ccc(cc1)CSc2nnc(n2c3ccccc3)C(Cc4ccccc4)NC(=O)c5ccc(cc5)F 7M-559S c1ccc(cc1)CC(c2nnc(n2c3ccccc3)SCc4ccc(c(c4)Cl)Cl)NC(=O)c5ccc(cc5)F 7M-560S Cn1c2c(cc(s2)C(=O)Nc3ccc(cc3)OC)c(n1)c4ccccc4 7M-561S C/C(=C\C(=O)c1ccccc1)/N(C)C 7M-562S Cn1c2c(cc(s2)C(=O)NCC=C)c(n1)c3ccccc3 7M-564S CNC(=O)c1cc2c(nn(c2s1)C)c3ccccc3 7M-565S Cn1c2c(cc(s2)C(=O)N3CCOCC3)c(n1)c4ccccc4 7M-566S Cn1c2c(cc(s2)C(=O)Nc3cccc(c3)C(F)(F)F)c(n1)c4ccccc4 7M-567S Cc1ccc(cc1)n2c(=O)c(c(cn2)N3CCOCC3)Sc4ccc(cc4)C 7M-569S COc1ccc(cc1)NC(=O)/C(=N/Nc2cccc(c2)C(F)(F)F)/C(=O)C(F)(F)F 7M-574S c1cc(cc(c1)N/N=C(\C(=O)C(F)(F)F)/C(=O)Nc2ccc(cc2)F)C(F)(F)F 7M-575S CCOC(=O)c1c(cc(=O)n(n1)c2cccc(c2)C(F)(F)F)C(F)(F)F 7M-576S Cn1c(c(c(n1)CSc2ccccc2)COC(=O)Nc3ccc(c(c3)Cl)Cl)Cl 7M-577S Cn1c(c(c(n1)CSc2ccccc2)COC(=O)Nc3ccc(cc3)Cl)Cl 7M-578S Cc1cc(oc(=O)c1NC(=O)c2ccccc2)c3ccccc3 7M-579S Cc1cc(oc(=O)c1NC(=O)c2ccccc2)c3ccc(cc3)Cl 7M-580S c1c(cc(c2c1c(=O)n(c(n2)C(F)(F)F)O)Cl)Cl 7M-581S Cc1c(sc2n1ncn2)C(=O)C 7M-582S c1cc(ccc1c2ccnc(c2C#N)O)Cl 7M-584S Cn1c2c(cc(s2)c3nnc(n3C)S)c(n1)c4ccccc4 7M-585S Cc1c(sc2n1ncn2)C(=O)CBr.Br 7M-587S Cn1c2c(cc(s2)c3nnc(n3C)SC)c(n1)c4ccccc4 7M-589S c1cc(cc(c1)NC(=O)/C(=N\Nc2cccc(c2)C(F)(F)F)/C(=O)C(F)(F)F)C(F)(F)F 7M-591S c1cc(cc(c1)N/N=C(/C(=O)C(F)(F)F)\C(=O)Nc2ccc(cc2F)F)C(F)(F)F 7M-592S c1cc(cc(c1)N/N=C(/C(=O)C(F)(F)F)\C(=O)Nc2cccc(c2Cl)Cl)C(F)(F)F 7M-593S c1cc(cc(c1)N/N=C(/C(=O)C(F)(F)F)\C(=O)Nc2cc(cc(c2)Cl)Cl)C(F)(F)F 7M-594S CN(c1ccccc1)C(=O)/C(=N/Nc2cccc(c2)C(F)(F)F)/C(=O)C(F)(F)F 7M-595S Cc1ccc(cc1)n2c(=O)c(c(cn2)Cl)Oc3ccc4ccccc4c3 7M-596S C/C(=C\C(=O)c1ccc(cc1)Br)/N(C)C 7M-599S c1ccc(cc1)CSc2c(c(nc(n2)N)c3cccs3)C#N 7M-600S c1cc(sc1)c2c(c(nc(n2)N)SCc3ccc(cc3)Cl)C#N 7M-601S COc1ccc(cc1)NC(=O)c2c(cc(=O)n(n2)c3cccc(c3)C(F)(F)F)C(F)(F)F 7M-603S Cc1cc(oc(=O)c1NC(=O)c2ccccc2)c3ccc(cc3)Br 7M-604S Cc1ccc(cc1)C(=O)Nc2c(cc(oc2=O)c3ccc(cc3)Br)C 7M-605S Cc1ccc(cc1)C(=O)Nc2c(cc(oc2=O)c3ccccc3)C 7M-606S Cc1ccc(cc1)C(=O)Nc2c(cc(oc2=O)c3ccc(cc3)Cl)C 7M-607S c1cc(ccc1S(=O)(=O)NCCOC(=O)Nc2ccc(c(c2)Cl)Cl)Cl 7M-609S Cn1c2c(cc(s2)c3nnc(n3C)SCC=C)c(n1)c4ccccc4 7M-610S CC(C)Sc1c(c(nc(n1)N)c2cccs2)C#N 7M-611S CCSc1c(c(nc(n1)N)c2cccs2)C#N 7M-612S CCCSc1c(c(nc(n1)N)c2cccs2)C#N 7M-613S c1cc(cc(c1)C(F)(F)F)CSc2c(c(nc(n2)N)c3cccs3)C#N 7M-614S COc1ccc(cc1)CSc2c(c(nc(n2)N)c3cccs3)C#N 7M-615S Cc1c(sc2n1ncn2)c3csc(n3)N 7M-618S c1cc(ccc1c2csc(n2)NC(=N)N)Cl 7M-619S Cn1c2c(cc(s2)c3nnc(n3C)SCc4nc5cc(ccc5s4)F)c(n1)c6ccccc6 7M-620S Cn1c2c(cc(s2)c3nnc(n3C)SCC(=O)c4ccc(cc4)Cl)c(n1)c5ccccc5 7M-621S c1ccc(cc1)c2ccnc(c2C#N)O 7M-622S COc1ccc(cc1)Cn2ccc(c(c2=O)C#N)c3ccccc3 7M-624S c1c(c(c(=O)[nH]n1)Br)Br 7M-627S c1cc(ccc1C(F)(F)F)NC(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/C(=O)C(F)(F)F 7M-630S CCOC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)C(F)(F)F)C(F)(F)F 7M-631S CCCNc1nc(cs1)c2c(n3c(s2)ncn3)C 7M-632S Cc1c(sc2n1ncn2)c3csc(n3)NC(=N)N 7M-633S Cc1c(sc2n1ncn2)c3csc(n3)c4ccccc4 7M-634S Cc1c(sc2n1ncn2)c3csc(n3)C#N 7M-635S Cn1ccc(c(c1=O)C#N)c2ccccc2 7M-660S Cc1c(c(ns1)SCC(=O)c2ccc(cc2)F)C#N 7M-700 Cc1c(c(ns1)SCC(=O)c2ccc(cc2)Br)C#N 7M-701 Cc1c(c(ns1)SCC(=O)c2ccc(cc2)OC)C#N 7M-703 Cc1coc2n1cc(n2)c3ccc(cc3)Cl 7M-704 CC(=O)/C(=C\Nc1ccsc1C(=O)OC)/c2ccccc2 7M-705 CC(=O)/C(=C/Nc1cccc(c1)[N+](=O)[O-])/c2ccccc2 7M-706 CC(=O)/C(=C/Nc1cccc(c1)C(=O)OC)/c2ccccc2 7M-707 Cc1c(c(=O)ccn1c2cc(cc(c2)OC)OC)Cc3c(cccc3Cl)Cl 7M-708 CC(=O)/C(=C\Nc1ccc(cc1)OCc2ccccc2)/c3ccccc3 7M-709 CC(=O)/C(=C\Nc1cc(cc(c1)OC)OC)/c2ccccc2 7M-710 Cc1ccc(cc1)C(=O)Cn2c(coc2=N)C 7M-712 Cc1ccc(cc1)C(=O)c2c(c3c(snc3s2)C)N 7M-713 CC(=O)/C(=C\Nc1ccc(cc1)C(F)(F)F)/c2ccccc2 7M-714 Cc1c(c(=O)ccn1c2ccc(cc2)OCc3ccccc3)Cc4c(cccc4Cl)Cl 7M-715 Cc1c(cccc1Cl)N/C=C(\c2ccccc2)/C(=O)C 7M-716 Cc1c2c(c(sc2ns1)C(=O)c3ccc(cc3)Br)N 7M-717 CC(=O)/C(=C\Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/c2ccccc2 7M-719 CC(=O)/C(=C\Nc1ccc(cc1)/N=N/c2ccccc2)/c3ccccc3 7M-721 Cc1c(c(=O)ccn1c2ccc(cc2)C(C)(C)C)Cc3c(cccc3Cl)Cl 7M-722 Cc1c(c(=O)ccn1c2ccc(cc2)N(C)C)Cc3c(cccc3Cl)Cl 7M-723 Cc1c(c(=O)ccn1Cc2ccc(cc2)OC)Cc3c(cccc3Cl)Cl 7M-724 c1c([nH]nc1C(=O)O)C(=O)O 7M-725 Cc1ccc(cc1C)N/C=C(\c2ccc(c(c2)OC)OC)/C(=O)C 7M-727 CC(=O)/C(=C/Nc1ccc(cc1Cl)Cl)/c2ccc(c(c2)OC)OC 7M-728 CCOC(=O)c1ccc(cc1)N/C=C(/c2ccc(c(c2)OC)OC)\C(=O)C 7M-729 COC(=O)c1cc(n[nH]1)C(=O)OC 7M-731 Cc1c2c(c(sc2ns1)C(=O)c3ccc(cc3)F)N 7M-733 Cc1c2c(c(sc2ns1)C(=O)c3ccc(cc3)Cl)N 7M-734 Cc1c2c(c(sc2ns1)C(=O)c3ccc(cc3)OC)N 7M-735 Cc1c(cccc1Cl)N/C=C(/c2ccc(c(c2)OC)OC)\C(=O)C 7M-736 CC(=O)/C(=C\Nc1ccc(cc1)Oc2ccccc2)/c3ccc(c(c3)OC)OC 7M-737 CC(=O)/C(=C\Nc1ccc(cc1)C(F)(F)F)/c2ccc(c(c2)OC)OC 7M-738 CC(=O)/C(=C\Nc1cccc(c1)Br)/c2ccc(c(c2)OC)OC 7M-739 c1ccc(c(c1)C(=O)c2cc(c3nc4ccccc4n3c2)C#N)O 7M-740 COc1ccc(cc1)CNC(=O)N 7M-741 c1cc(cnc1)CNC(=O)N 7M-742 c1ccc(cc1)CNC(=O)N 7M-744 c1cc(cnc1)CNc2ccc3nnc(n3n2)C(F)(F)F 7M-745 c1cc(ccc1CON2C(=O)C(=O)NC2=O)Cl 7M-746 CC(=O)/C(=C\Nc1ccc(c(c1)OC)OC)/c2ccc(c(c2)OC)OC 7M-747 Cc1ccc(cc1)CNC(=O)N 7M-748 c1cc(ccc1CNC(=O)N)F 7M-749 Cc1c(c(=O)ccn1c2ccc(cc2)C(=O)OC)Cc3c(cccc3Cl)Cl 7M-750 CC(=O)c1cc(sc1Cl)Cl 7M-751 Cc1ccc(c(c1)C(=O)c2cc(c3nc4ccccc4n3c2)C#N)O 7M-752 c1cc(sc1)CNC(=O)N 7M-753 CC(=O)c1ccc(cc1)N/C=C(/c2ccc(c(c2)OC)OC)\C(=O)C 7M-754 Cc1ccc(cc1)CN2C(=O)C(=O)NC2=O 7M-755 c1cc(ccc1CN2C(=O)C(=O)NC2=O)F 7M-756 c1ccc(c(c1)CNC(=O)N)Cl 7M-757 COc1ccc(cc1OC)CNC(=O)N 7M-758 Cc1c(c(=O)ccn1N(C)c2c(cc(cn2)C(F)(F)F)Cl)Cc3c(cccc3Cl)Cl 7M-760 c1cc(ccc1CNC(=O)N)Cl 7M-761 c1cc(ccc1Sc2ccc3nnc(n3n2)C(F)(F)F)Cl 7M-762 COc1ccc(cc1)CN2C(=O)C(=O)NC2=O 7M-763 COC(=O)c1cc(n(n1)CCBr)C(=O)OC 7M-764 c1ccc(c(c1)CN2C(=O)C(=O)NC2=O)Cl 7M-765 COc1ccc(cc1OC)CN2C(=O)C(=O)NC2=O 7M-766 c1cc(ccc1CN2C(=O)C(=O)NC2=O)Cl 7M-767 Cc1c(c(=O)ccn1Cc2cccc(c2)C(F)(F)F)Cc3c(cccc3Cl)Cl 7M-768 COc1ccc(cc1)Sc2ccc3nnc(n3n2)C(F)(F)F 7M-771 CN(C)/C=C/C(=O)c1cc(sc1Cl)Cl 7M-772 c1cc(ccc1CONC(=O)N)F 7M-773 c1ccc(c(c1)CONC(=O)N)F 7M-774 c1cc(c(cc1F)Cl)CONC(=O)N 7M-775 c1cc(c(c(c1)Cl)CONC(=O)N)F 7M-776 c1cc(c(c(c1)Cl)Cc2c(ccc(c2O)/C=N/Cc3ccc(cc3)Cl)O)F 7M-777 Cc1c(c(=O)ccn1c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cc4c(cccc4Cl)Cl 7M-778 CC(C)(CNC(=O)c1ccc(cc1)[N+](=O)[O-])SCc2cccc(c2)C(F)(F)F 7M-779 Cc1c(c(=O)ccn1Cc2cccnc2)Cc3c(cccc3Cl)Cl 7M-780 CSc1nc(cc(n1)Cl)N2CCCC2 7M-800 CCCCNc1cc(nc(n1)N)Cl 7M-801 C[NH+]1CCN(CC1)c2cc(nc(n2)N)Cl.[Cl-] 7M-802 Cc1ccc(cc1)Sc2cc(nc(n2)N)Cl 7M-803 c1cc(sc1)Sc2cc(nc(n2)N)Sc3cccs3 7M-804 c1ccc(cc1)CCNc2cc(nc(n2)N)Cl 7M-805 c1c(nc(nc1Cl)N)N2CCC(CC2)C(=O)N 7M-806 CC(C)Sc1cc(nc(n1)NC(=O)Nc2ccccc2)Cl 7M-807 CC(C)(C)c1csc(n1)NC(=O)Nc2ccccc2 7M-808 CCOc1ccccc1N2CCN(CC2)c3cc(nc(n3)N)Sc4ccc(cc4)Cl 7M-809 c1ccc2c(c1)CCN(C2)c3cc(nc(n3)N)Sc4ccc(cc4)F 7M-810 CCOc1ccccc1N2CCN(CC2)c3cc(nc(n3)SC)Cl 7M-811 CCNc1cc(nc(n1)SC)Sc2ccc(cc2)F 7M-812 c1ccc2cc(ccc2c1)Sc3cc(nc(n3)N)Cl 7M-813 CSc1nc(cc(n1)Cl)Sc2ccc(cc2)Cl 7M-814 CSc1nc(cc(n1)N2CCOCC2)N3CCOCC3 7M-815 CSc1nc(cc(n1)Cl)N2CCN(CC2)c3ccc(cc3)F 7M-816 Cc1ccc(cc1)Sc2cc(nc(n2)SC)Cl 7M-817 Cc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)O 7M-818 CCCN(CCC)c1cc(nc(n1)SC)Cl 7M-819 CSc1nc(cc(n1)Cl)Nc2ccccc2N 7M-820 CSc1nc(cc(n1)Cl)N2CCN(CC2)c3ccccc3Cl 7M-821 CCOC(=O)N1CCN(CC1)c2cc(nc(n2)SC)Cl 7M-822 CSc1nc(cc(n1)Sc2ccc(cc2)F)N3CCOCC3 7M-823 Cc1cc(nc(n1)SCCS(=O)(=O)O)O 7M-824 CSc1nc(cc(n1)Cl)N2CCN(CC2)c3cc(nc(n3)SC)Cl 7M-825 Cc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)N3CCOCC3 7M-826 c1ccc(cc1)Sc2cc(nc(n2)N)Sc3ccccc3 7M-827 CCNc1cc(nc(n1)SC)Cl 7M-828 CSc1nc(cc(n1)Cl)N2CCCc3c2cccc3 7M-829 c1cc(ccc1F)Sc2cc(nc(n2)N)N3CCCC3 7M-830 CCOc1ccccc1N2CCN(CC2)c3cc(nc(n3)N)Sc4ccc(cc4)C 7M-831 Cc1cc(nc(n1)SCc2ccc(cc2)Cl)O 7M-832 CSc1nc(cc(n1)Cl)N(CCO)Cc2ccccc2 7M-833 CSc1nc(cc(n1)Cl)NN 7M-834 CSc1nc(cc(n1)Cl)N(CCO)CCO 7M-835 CCOC(=O)N1CCN(CC1)c2cc(nc(n2)SC)Sc3ccc(cc3)F 7M-836 CSc1nc(cc(n1)Cl)N2CCC(CC2)C(=O)N 7M-837 CSc1nc(cc(n1)N2CCN(CC2)C(=O)N)N3CCN(CC3)c4ccccc4 7M-838 CCOC(=O)N1CCN(CC1)c2cc(nc(n2)SC)N3CCN(CC3)C(=O)N 7M-839 c1ccc(cc1)N2CCN(CC2)c3cc(nc(n3)N)N4CCCC4 7M-840 CSc1nc(cc(n1)N2CCN(CC2)c3ccccc3)N=[N+]=[N-] 7M-841 CSc1nc(cc(n1)N2CCN(CC2)c3ccccc3)N4CCN(CC4)c5ccccc5 7M-842 c1ccc(cc1)NC(=O)Nc2nc(cc(n2)Cl)N3CCCCC3 7M-843 CSc1nc(cc(n1)Cl)NNC(=O)Nc2ccccc2 7M-844 CSc1nc(cc(n1)Cl)N/N=C/c2ccccc2 7M-845 CCCCC/C(=C/c1ccccc1)/C=N/Nc2cc(nc(n2)SC)Cl 7M-846 c1ccc2c(c1)C(=O)N(C2=O)OCC(=O)Nc3ccc(cn3)I 7M-900 c1cc(ncc1I)NC(=O)CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 7M-901 c1cc(ncc1I)NC(=O)CON.Cl 7M-903 c1cc(ccc1C(=O)C/C=N/OCC(=O)Nc2ccc(cn2)I)F 7M-904 Cc1ccc(cc1)C(=O)C/C=N/OCC(=O)Nc2ccc(cn2)I 7M-905 C/C(=C/C(=O)Nc1ccc(cn1)I)/N2CCCC2 7M-906 COC(=O)c1c2ccc3ccc4ccc5c(c(c(n5c4c3n2c(c1C(=O)OC)C(=O)OC)C(=O)OC)C(=O)OC)C(=O)OC 7M-907 c1ccc(cc1)c2ccc(cc2)C(=O)C/C=N/OCC(=O)Nc3ccc(cn3)I 7M-908 c1c(cnc(c1Cl)n2c3c(cn2)c(=O)[nH]c(=O)[nH]3)C(F)(F)F 7M-909 Cc1c(c(no1)C(=O)C)C(=O)Nc2ccc(cn2)I 7M-910 CCOC(=O)c1c(c(on1)C)C(=O)Nc2ccc(cn2)I 7M-911 c1ccc(cc1)n2c3c(cn2)c(=O)[nH]c(=O)[nH]3 7M-912 Cc1c(c(no1)C(=O)N2CCCC2)C(=O)Nc3ccc(cn3)I 7M-914 Cc1c(c(no1)/C(=N/OC)/C)C(=O)Nc2ccc(cn2)I 7M-915 c1ccc2c(c1)nc(o2)c3c[nH]nc3 7M-916 c1ccc2c(c1)nc(o2)c3cnn(c3)c4ccc(cc4Cl)Cl 7M-918 c1ccc2c(c1)nc(o2)c3cnn(c3)C(=O)c4ccc(cc4)F 7M-919 c1ccc2c(c1)nc(o2)c3cnn(c3)C4CCS(=O)(=O)C4 7M-922 c1ccc(cc1)n2cc(cn2)c3nc4ccccc4o3 7M-923 CCOC(=O)NC(=O)/C(=C(/C)\N(C)C)/C#N 7M-924 c1ccc(cc1)C(=O)/C=C/c2ccc[nH]2 7M-928 c1cc(oc1)/C=C/C(=O)c2ccc(cc2)C(F)(F)F 7M-929 CC(=O)/C(=N/Nc1ccc(cc1)F)/C(=O)OC 7M-930 Cc1c(c(=O)n(nc1C(=O)OC)c2ccc(cc2)F)C#N 7M-931 c1cc(cc(c1)C(=O)/C=C/c2occc2)C(=O)/C=C/c3occc3 7M-933 c1ccc(cc1)C(=O)/C=C/c2c[nH]c3c2cccc3 7M-934 c1ccc(cc1)/C=C/C(=O)/C=C/c2ccco2 7M-935 c1ccc(cc1)C(=O)/C=C/C=C/c2ccco2 7M-936 Cc1ccc(c(c1)C)N/N=C(/C(=O)C)\C(=O)OC 7M-937 CC(=O)/C(=N/Nc1ccc(cc1)OC)/C(=O)OC 7M-938 CC(=O)/C(=N/Nc1cccc(c1)C(F)(F)F)/C(=O)OC 7M-939 Cc1c(c(=O)n(nc1C(=O)OC)c2ccc(cc2)OC)C#N 7M-943 c1ccc2c(c1)CCCN2C(=O)c3ccccc3C(F)(F)F 7N-002 c1cc(ccc1n2cnn(c2=O)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])OC(F)(F)F 7N-003 c1cc(oc1)CNC(=O)c2ccc(cc2)I 7N-004 c1cc(ccc1NC(=O)C2CC2)I 7N-005 CS(=O)(=O)NCc1ccc(cc1)Cl 7N-006 COc1ccc(cc1)OCc2cnc(s2)Cl 7N-007 c1cc(ccc1Oc2ccc(cc2)S(=O)(=O)N3CCCCC3)S(=O)(=O)N4CCCCC4 7N-008 CC(C)(C)OC(=O)N(Cc1ccc(cc1)Cl)S(=O)(=O)C 7N-009 c1ccc(cc1)C(=O)Nc2ncc(s2)[N+](=O)[O-] 7N-010 Cc1ccc(cc1)CNS(=O)(=O)/C=C/c2ccc(cc2)OC 7N-011 c1cc(ccc1Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)I 7N-013 c1ccc(cc1)OCc2cnc(s2)Cl 7N-014 CS(=O)(=O)NCc1ccccc1 7N-015 c1ccn(c1)c2ncc(s2)[N+](=O)[O-] 7N-016 Cc1ccc(cc1)CNS(=O)(=O)/C=C/c2ccc3c(c2)OCO3 7N-017 c1cc(ccc1n2cnn(c2=O)CC(=O)O)Br 7N-018 Cc1cccc(c1)C(=O)Nc2ncc(s2)[N+](=O)[O-] 7N-019 CC(=O)Nc1ccc(cc1)OCc2cnc(s2)Cl 7N-020 c1cc(ccc1[N+](=O)[O-])OCc2cnc(s2)Cl 7N-021 c1cc(c(cc1Cl)Cl)OCc2cnc(s2)Cl 7N-022 c1cc(oc1)C(=O)Nc2ncc(s2)[N+](=O)[O-] 7N-023 c1cc(ccc1C(=O)Nc2ccc(cc2)I)I 7N-024 Cc1cccc(c1)OCc2cnc(s2)Cl 7N-025 c1cc(ccc1CNS(=O)(=O)/C=C/c2ccc(cc2)Br)Cl 7N-027 c1cc(oc1)C(=O)NC2CCCCCCC2 7N-028 c1cc(ccc1C#N)OCc2cnc(s2)Cl 7N-029 c1cc(ccc1OCc2cnc(s2)Cl)F 7N-030 CC(C)(C)OC(=O)N(Cc1ccccc1)S(=O)(=O)C 7N-031 CS(=O)(=O)NCc1cccs1 7N-033 CC(C)(C)c1ccc(cc1)OCc2cnc(s2)Cl 7N-034 c1c(sc(n1)NC(=O)C2CC2)[N+](=O)[O-] 7N-035 c1cc(cnc1)CNC(=O)c2ccc(cc2)I 7N-037 c1cc(ccc1CNS(=O)(=O)/C=C/c2ccc(cc2)[N+](=O)[O-])Cl 7N-038 c1cc(sc1)CNS(=O)(=O)c2ccc(cc2)I 7N-040 CS(=O)(=O)NCc1ccc2c(c1)OCO2 7N-041 c1cc(ccc1CNS(=O)(=O)/C=C/c2ccc3c(c2)OCO3)Cl 7N-042 CC(C)(C)OC(=O)N(Cc1cccs1)S(=O)(=O)C 7N-044 c1cc(cnc1)CNS(=O)(=O)c2ccc(cc2)I 7N-045 COc1cc(ccc1OCc2cnc(s2)Cl)C=O 7N-046 c1ccc2c(c1)C(=O)N(C2=O)OCc3cnc(s3)Cl 7N-047 COc1cccc(c1)CNS(=O)(=O)C 7N-048 c1cc(cc(c1)OCc2cnc(s2)Cl)C(F)(F)F 7N-050 CC(C)(C)OC(=O)N(Cc1ccc2c(c1)OCO2)S(=O)(=O)C 7N-051 COc1cc(ccc1OCc2cnc(s2)Cl)/C=N/NC(=O)c3ccncc3 7N-052 c1cc(sc1)CNS(=O)(=O)/C=C/c2ccc3c(c2)OCO3 7N-053 c1cc(sc1)CNS(=O)(=O)/C=C/c2ccc(o2)c3ccc(cc3)Cl 7N-054 c1ccc2c(c1)c(nc(n2)C(F)(F)F)Oc3ccc(cc3)I 7N-055 c1cc(ccc1C(=O)NC2CCCCCCC2)I 7N-056 COc1cc(ccc1OCc2cnc(s2)Cl)/C=N/Nc3ccc(cc3)C(=O)O 7N-057 c1c(sc(n1)Cl)CSc2nc[nH]n2 7N-058 c1cc(sc1)CNS(=O)(=O)/C=C/c2ccc(cc2Cl)Cl 7N-059 c1cc(ccc1C(=O)Nc2ncc(s2)[N+](=O)[O-])Cl 7N-060 c1cnc(nc1)Oc2ccc(cc2)N 7N-061 c1ccc(cc1)CNS(=O)(=O)/C=C/c2ccc(cc2)Cl 7N-062 CC(C)(C)OC(=O)N(Cc1cccc(c1)OC)S(=O)(=O)C 7N-063 COc1ccc(cc1OC)/C=C/S(=O)(=O)NCc2ccccc2 7N-064 c1ccc2c(c1)CCCN2C(=O)c3cccs3 7N-066 COc1cc(ccc1C=O)Oc2c3ccccc3nc(n2)C(F)(F)F 7N-067 c1cnc(nc1)Oc2ccc(cc2)I 7N-068 c1cc(ccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])I 7N-069 COc1ccc(cc1)NS(=O)(=O)C 7N-070 c1cc(c(nc1)Oc2ccc(cc2)I)[N+](=O)[O-] 7N-072 c1cc(ccc1C(=O)NC2CCCCCC2)F 7N-073 Cc1cccc(c1)C(=O)NC2CCCCCC2 7N-074 c1ccc(cc1)CNS(=O)(=O)/C=C/c2ccccc2 7N-075 Cc1cccc(c1)C(=O)NC2CCCCCCC2 7N-076 c1cc(cc(c1)Cl)C(=O)NC2CCCCCCC2 7N-077 c1cc(ccc1C(=O)NC2CCCCCCC2)F 7N-078 c1cc(cc(c1)Cl)C(=O)NC2CCCCCC2 7N-079 c1ccc2c(c1)nc(s2)SCc3cnc(s3)Cl 7N-080 CC(C)(C)OC(=O)N(c1ccc(cc1)OC)S(=O)(=O)C 7N-081 c1ccc(cc1)CNS(=O)(=O)/C=C/c2ccc3ccccc3c2 7N-082 CS(=O)(=O)NC1CCCCCC1 7N-083 CC(=O)c1ccc(cc1)Oc2ncccn2 7N-084 c1cc(sc1)CNS(=O)(=O)/C=C/c2ccncc2 7N-085 CN(C)c1ccc(cc1)/C=C/S(=O)(=O)NCc2ccccc2 7N-086 c1ccc2c(c1)nc(s2)S(=O)(=O)Cc3cnc(s3)Cl 7N-087 CC(=O)OCc1cnc(s1)Cl 7N-088 COc1ccc(cc1)NS(=O)(=O)/C=C/c2ccc(c(c2)OC)OC 7N-089 CN(C)/C=C/C(=O)c1ccc(cc1)Oc2ncccn2 7N-090 c1ccc(cc1)CNS(=O)(=O)/C=C/c2ccc(cc2Cl)Cl 7N-091 c1cc(ccc1OCc2cnc(s2)Cl)S(=O)(=O)Cl 7N-092 c1cc(sc1)/C=C/S(=O)(=O)NCc2ccc3c(c2)OCO3 7N-093 COc1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)Oc3ncccn3 7N-094 c1cc2c(cc1CNS(=O)(=O)/C=C/c3ccncc3)OCO2 7N-095 COc1ccc(cc1)/C=C/S(=O)(=O)NCc2ccc3c(c2)OCO3 7N-096 c1cc(oc1)/C=C/S(=O)(=O)NCc2ccc3c(c2)OCO3 7N-097 c1c(sc(n1)Cl)CO 7N-099 Cc1ccsc1/C=C/S(=O)(=O)NCc2ccc3c(c2)OCO3 7N-100 COc1cccc(c1)CNS(=O)(=O)/C=C/c2ccc(c(c2)OC)OCc3ccc(cc3)Cl 7N-101 Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)N4CCCC4 7N-302S CCOC(=O)Cn1c2ccccc2c(cc1=O)C 7N-308S CCOC(=O)Cn1c(=O)cc(c2c1c(ccc2)C)C 7N-309S Cc1cccc(c1)Cn2cnc(n2)SCc3ccc(cc3)Cl 7N-312S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)N4CCOCC4 7N-313S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)Sc4ccc(cc4)C 7N-314S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)Oc4cccc(c4)C(F)(F)F 7N-315S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)N4CCCC4 7N-316S Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccc3)Sc4ccccc4C(=O)OC 7N-317S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)N4CCOCC4 7N-318S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)Oc4cccc(c4)C(F)(F)F 7N-319S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)S(=O)(=O)c4ccccc4C(=O)OC 7N-320S CC(C)C(=O)OC1CCS(=O)(=O)c2c1ccs2 7N-322S c1ccc(cc1)N/N=C(\C(=O)C2CC2)/C(=O)C(F)(F)F 7N-323S Cc1ccc(cc1)CSc2nc3c(c(n2)SCC(=O)O)CCCC3 7N-326S Cc1ccc(cc1)CSc2nc3c(c(n2)Sc4ccccc4Cl)CCCC3 7N-327S Cc1ccc(cc1)CSc2nc3c(c(n2)SC4CCCCC4)CCCC3 7N-328S CS(=O)(=O)N(CC(=O)Nc1cccc(c1)C(F)(F)F)c2cc(ccc2Cl)C(F)(F)F 7N-330S CS(=O)(=O)N(CC(=O)Nc1ccc(cc1Cl)Cl)c2cc(ccc2Cl)C(F)(F)F 7N-331S CS(=O)(=O)N(CC(=O)Nc1ccc(cc1F)F)c2cc(ccc2Cl)C(F)(F)F 7N-332S Cc1cc(ccc1NC(=O)CN(c2cc(ccc2Cl)C(F)(F)F)S(=O)(=O)C)Cl 7N-333S CSc1nc2ccsc2c(n1)Oc3ccc(cc3)Cl 7N-334S Cc1cccc(c1C)Oc2c3c(ccs3)nc(n2)SC 7N-335S CSc1nc2ccsc2c(n1)Oc3ccccc3 7N-336S CSc1nc2ccsc2c(n1)Oc3ccc4ccccc4c3 7N-337S CSc1nc2ccsc2c(n1)Oc3ccc(cc3F)F 7N-338S COc1ccc(cc1)Oc2c3c(ccs3)nc(n2)SC 7N-339S CSc1nc2ccsc2c(n1)NC3CCCCC3 7N-340S COc1ccc(cc1)NC(=O)CN(c2cc(ccc2Cl)C(F)(F)F)S(=O)(=O)C 7N-341S c1ccc(cc1)CSc2nc3ccsc3c(n2)O 7N-342S c1ccc(cc1)CSc2nc3ccsc3c(n2)Cl 7N-343S C=CCNc1c2c(ccs2)nc(n1)SCc3ccccc3 7N-344S CCN(CC)c1c2c(ccs2)nc(n1)SCc3ccccc3 7N-345S c1ccc(cc1)CSc2nc3ccsc3c(n2)N4CCCC4 7N-346S c1ccc(cc1)CSc2nc3ccsc3c(n2)N4CCOCC4 7N-348S c1ccc(cc1)CSc2nc3ccsc3c(n2)NC4CCCCC4 7N-349S COc1cccc(c1)Sc2c3c(ccs3)nc(n2)SCc4ccccc4 7N-350S c1ccc(cc1)CSc2nc3ccsc3c(n2)Sc4ccc(cc4Cl)Cl 7N-351S c1ccc(cc1)CSc2nc3ccsc3c(n2)SCc4cccc(c4)C(F)(F)F 7N-352S Cc1ccc(cc1)Sc2c3c(ccs3)nc(n2)SCc4ccccc4 7N-354S c1ccc(cc1)CSc2nc3ccsc3c(n2)Oc4ccccc4 7N-356S COc1ccc(cc1)Oc2c3c(ccs3)nc(n2)SCc4ccccc4 7N-357S c1ccc(cc1)CSc2nc3ccsc3c(n2)Oc4ccc(cc4Cl)Cl 7N-359S c1ccc(cc1)CSc2nc3ccsc3c(n2)Oc4ccc(cc4F)F 7N-360S Cc1ccc(cc1)Oc2c3c(ccs3)nc(n2)SCc4ccccc4 7N-361S CCCC(=O)OC1CCS(=O)(=O)c2c1ccs2 7N-362S CCCCC(=O)OC1CCS(=O)(=O)c2c1ccs2 7N-363S CC(C)(C)C(=O)OC1CCS(=O)(=O)c2c1ccs2 7N-364S c1csc2c1C(CCS2(=O)=O)OC(=O)C3CC3 7N-365S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)S(=O)(=O)c4ccccc4)CCCC3 7N-366S Cc1cccc(c1C)Oc2c3c(nc(n2)SCc4ccc(cc4)Cl)CCCC3 7N-367S CC(=O)Nc1ccc(cc1)Oc2c3c(nc(n2)SCc4ccc(cc4)Cl)CCCC3 7N-368S c1csc2c1C(CCS2(=O)=O)Cl 7N-369S c1cc(cc(c1)Oc2c3c(nc(n2)SCc4ccc(cc4)Cl)CCCC3)C(F)(F)F 7N-377S Cc1ccc(cc1)Oc2c3c(nc(n2)SCc4ccc(cc4)Cl)CCCC3 7N-379S COc1ccc(cc1)Oc2c3c(nc(n2)SCc4ccc(cc4)Cl)CCCC3 7N-380S Cc1ccc(cc1)CS(=O)c2nc3c(c(n2)N4CCOCC4)CCCC3 7N-383S Cc1ccc(cc1)CS(=O)c2nc3c(c(n2)NCC=C)CCCC3 7N-384S Cc1ccc(cc1)CS(=O)c2nc3c(c(n2)N4CCN(CC4)C)CCCC3 7N-385S c1cc(ccc1SC2CCS(=O)(=O)c3c2ccs3)Cl 7N-396S CS(=O)(=O)N(CC(=O)Oc1cccc(c1)C(F)(F)F)c2cc(ccc2Cl)C(F)(F)F 7N-398S CS(=O)(=O)N(CC(=O)Oc1ccc(cc1)Cl)c2cc(ccc2Cl)C(F)(F)F 7N-400S CS(=O)(=O)N(CC(=O)Oc1ccc(cc1)Cl)c2ccc(cc2)Cl 7N-411S Cc1cccc(c1)N(CC(=O)Oc2ccc(cc2)Cl)S(=O)(=O)C 7N-412S CS(=O)(=O)N(CC(=O)Oc1cccc(c1)C(F)(F)F)c2ccc(cc2)Cl 7N-413S Cc1cccc(c1OC(=O)CN(c2ccc(cc2)Cl)S(=O)(=O)C)C 7N-414S CS(=O)(=O)N(CC(=O)Oc1ccc2ccccc2c1)c3ccc(cc3)Cl 7N-416S C=CCNc1c2c(nc(n1)SCc3ccc(cc3)Cl)CCCC2 7N-418S c1cc(ccc1CSc2nc3c(c(n2)N4CCOCC4)CCCC3)Cl 7N-419S c1cc(ccc1CSc2nc3c(c(n2)SC4CCCCC4)CCCC3)Cl 7N-420S c1cc(ccc1CSc2nc3c(c(n2)Sc4ccc(cc4)Cl)CCCC3)Cl 7N-421S CC(C)(C)Sc1c2c(nc(n1)SCc3ccc(cc3)Cl)CCCC2 7N-423S c1ccc(cc1)SC2CCS(=O)(=O)c3c2ccs3 7N-424S Cc1ccc(cc1)SC2CCS(=O)(=O)c3c2ccs3 7N-425S c1cc(c(cc1Cl)Cl)SC2CCS(=O)(=O)c3c2ccs3 7N-426S c1cc(cc(c1)SC2CCS(=O)(=O)c3c2ccs3)C(F)(F)F 7N-427S Cc1cccc(c1C)Oc2c3c(nc(n2)S(=O)(=O)Cc4ccc(cc4)Cl)CCCC3 7N-428S CSc1nc2c(c(n1)Cl)CCCC2 7N-430S c1ccc(cc1)S(=O)(=O)c2c(cc(=O)n(n2)c3cccc(c3)C(F)(F)F)C(F)(F)F 7N-432S c1ccc(cc1)n2c(=O)cc(c(n2)S(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F 7N-433S CC(C)(C)c1ccc(cc1)COC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)C 7N-437S COc1ccc(cc1)COC(=O)CN(c2cccc(c2)C(F)(F)F)S(=O)(=O)C 7N-438S Cc1cccc(c1)SC2CCS(=O)(=O)c3c2ccs3 7N-440S c1cc(ccc1SC2CCS(=O)(=O)c3c2ccs3)Br 7N-441S c1cc(c(cc1Cl)SC2CCS(=O)(=O)c3c2ccs3)Cl 7N-442S Cc1cccc(c1)Oc2c3c(nc(n2)SCc4ccccc4Cl)CCCC3 7N-444S c1cc(c(c(c1)Cl)SC2CCS(=O)(=O)c3c2ccs3)Cl 7N-448S CC(C)c1ccc(cc1)SC2CCS(=O)(=O)c3c2ccs3 7N-449S c1ccc(c(c1)SC2CCS(=O)(=O)c3c2ccs3)Cl 7N-450S c1cc(cc(c1)Cl)SC2CCS(=O)(=O)c3c2ccs3 7N-451S COc1cccc(c1)SC2CCS(=O)(=O)c3c2ccs3 7N-456S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)Sc4ccc(cc4)Cl 7N-459S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)Oc4ccc(cc4F)F 7N-460S c1ccc(cc1)c2nc(cc(n2)N3CCOCC3)N4CCCC4 7N-461S COc1cccc(c1)Sc2cc(nc(n2)c3ccccc3)N4CCOCC4 7N-462S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3)Cl)N4CCOCC4 7N-463S c1cc(ccc1CSC2CCS(=O)(=O)c3c2ccs3)Cl 7N-464S CNc1c2c(nc(n1)SCc3ccccc3Cl)CCCC2 7N-467S C=CCNc1c2c(nc(n1)SCc3ccccc3Cl)CCCC2 7N-468S c1ccc(c(c1)CSc2nc3c(c(n2)Oc4ccc(cc4F)F)CCCC3)Cl 7N-469S C=CCSc1nc2ccsc2c(n1)O 7N-470S C=CCSc1nc2ccsc2c(n1)Cl 7N-471S Cc1ccc(cc1)Sc2c3c(ccs3)nc(n2)SCC=C 7N-475S C=CCSc1nc2ccsc2c(n1)Sc3ccccc3 7N-476S C=CCNc1c2c(ccs2)nc(n1)SCC=C 7N-478S CCN(CC)c1c2c(ccs2)nc(n1)SCC=C 7N-479S C=CCSc1nc2ccsc2c(n1)N3CCCC3 7N-480S CNc1c2c(ccs2)nc(n1)SCC=C 7N-481S C=CCSc1nc2ccsc2c(n1)N3CCOCC3 7N-482S C=CCSc1nc2ccsc2c(n1)NC3CCCCC3 7N-483S C=CCSc1nc2ccsc2c(n1)Oc3ccccc3 7N-484S COc1ccc(cc1)Oc2c3c(ccs3)nc(n2)SCC=C 7N-485S C=CCSc1nc2ccsc2c(n1)Oc3ccc4ccccc4c3 7N-486S C=CCSc1nc2ccsc2c(n1)Oc3ccc(cc3Cl)Cl 7N-487S Cc1ccc(cc1)Oc2c3c(ccs3)nc(n2)SCC=C 7N-488S COC(=O)c1ccccc1Oc2c3c(ccs3)nc(n2)SCC=C 7N-489S COc1ccc(cc1)Oc2c3c(nc(n2)SCc4ccccc4Cl)CCCC3 7N-490S CC(C)(C)c1ccc(cc1)Oc2c3c(nc(n2)SCc4ccccc4Cl)CCCC3 7N-491S COC(=O)CSc1c2c(nc(n1)SCc3ccccc3Cl)CCCC2 7N-492S c1ccc(c(c1)CSc2nc3c(c(n2)SCC(=O)O)CCCC3)Cl 7N-493S c1ccc(cc1)c2nc(cc(n2)Oc3ccc(cc3F)F)N4CCOCC4 7N-494S Cc1ccc(cc1)Sc2c3c(nc(n2)SCc4ccccc4Cl)CCCC3 7N-497S c1ccc(c(c1)CSc2nc3c(c(n2)Sc4ccc(cc4)Cl)CCCC3)Cl 7N-498S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)Sc4ccc(cc4)C)CCCC3 7N-499S CCOC(=O)c1cnc(nc1Nc2ccc(c(c2)Cl)Cl)SC 7N-501S CCOC(=O)c1cnc(nc1Nc2ccc(cc2)C(F)(F)F)SC 7N-502S CCOC(=O)c1cnc(nc1Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)SC 7N-503S CCOC(=O)c1cnc(nc1Nc2ccc(cc2)OC(F)(F)F)SC 7N-504S CCOC(=O)c1cnc(nc1Nc2cc(ccc2Cl)C(F)(F)F)SC 7N-505S Cn1cncc1COC(=O)c2ccc(cc2)Cl 7N-509S CCOC(=O)c1cnc(nc1N2CCOCC2)SC 7N-510S CCOC(=O)c1cnc(nc1N2CCCCC2)SC 7N-511S CCOC(=O)c1cnc(nc1NC)SC 7N-512S CCOC(=O)c1cnc(nc1NCC=C)SC 7N-513S CCOC(=O)c1cnc(nc1Sc2cc(ccc2Cl)Cl)SC 7N-514S CCOC(=O)c1cnc(nc1Sc2ccc(cc2)Br)SC 7N-515S CCOC(=O)c1cnc(nc1Sc2ccccc2)SC 7N-516S CCOC(=O)c1cnc(nc1Sc2ccc(cc2Cl)Cl)SC 7N-517S CCOC(=O)c1cnc(nc1Sc2ccc(cc2)F)SC 7N-518S CCOC(=O)c1cnc(nc1Sc2ccc(cc2)C)SC 7N-519S CCOC(=O)c1cnc(nc1N2CCN(CC2)c3ccccc3F)SC 7N-520S CCOC(=O)c1cnc(nc1N2CCCC2)SC 7N-521S CCOC(=O)c1cnc(nc1N(C)C)SC 7N-522S CCOC(=O)c1cnc(nc1Sc2ccccc2Cl)SC 7N-523S CCOC(=O)c1cnc(nc1Sc2cccc(c2)C(F)(F)F)SC 7N-524S CSc1nc(cc(n1)Cl)C(F)(F)F 7N-527S CCOC(=O)c1cnn(c1N)c2ccccc2 7N-528S CSc1ncc2c(=O)[nH]c(nc2n1)c3ccccc3 7N-530S CSc1nc(cc(n1)N2CCOCC2)C(F)(F)F 7N-531S CSc1nc(cc(n1)N2CCN(CC2)C(c3ccccc3)c4ccccc4)C(F)(F)F 7N-532S CSc1nc(cc(n1)N2CCCCC2)C(F)(F)F 7N-533S CSc1nc(cc(n1)NCC=C)C(F)(F)F 7N-534S CNc1cc(nc(n1)SC)C(F)(F)F 7N-535S CSc1nccc(n1)c2ccc(cc2)Cl 7N-538S CCOC(=O)c1cnc(nc1NCCOC)SC 7N-541S Cc1c2c(nc(n1)N3CCOCC3)CCCC2 7N-562S Cc1c2c(nc(n1)N3CCCC3)CCCC2 7N-563S Cc1ccc(cc1)Sc2nc(c3c(n2)CCCC3)C 7N-564S Cc1c2c(nc(n1)S(=O)(=O)c3ccccc3)CCC2 7N-567S Cc1c2c(nc(n1)S(=O)(=O)c3cccc(c3)OC)CCC2 7N-569S CCOC(=O)CS(=O)(=O)c1nc(c2c(n1)CCC2)C 7N-573S Cc1c2c(nc(n1)S(=O)(=O)c3ccc(cc3)Cl)CCC2 7N-574S Cc1c2c(nc(n1)S(=O)(=O)c3cccc(c3)Cl)CCC2 7N-575S Cc1c2c(nc(n1)S(=O)(=O)c3cccc(c3)C(F)(F)F)CCC2 7N-576S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2O)c3ccccc3 7N-585S c1ccc(cc1)c2ncc(c(n2)N3CCCC3)S(=O)(=O)c4ccccc4 7N-590S Cc1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)OC 7N-592S c1ccc(cc1)c2ncc(c(n2)Sc3ccc(cc3)Cl)S(=O)(=O)c4ccccc4 7N-594S CN1CCN(CC1)c2c(cnc(n2)c3ccccc3)S(=O)(=O)C 7N-595S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2N(C)Cc3ccccc3)c4ccccc4 7N-596S CC(C)(C)c1ccc(cc1)SCc2cc(on2)c3ccc(c(c3)Cl)Cl 7N-644S c1ccc(cc1)SCc2cc(on2)c3ccc(c(c3)Cl)Cl 7N-645S c1ccc(c(c1)c2cc(no2)CCl)Cl 7N-646S c1ccc(c(c1)c2cc(no2)CSc3ccc(cc3)Cl)Cl 7N-647S c1ccc(c(c1)c2cc(no2)CSc3cc(ccc3Cl)Cl)Cl 7N-648S c1ccc(cc1)c2cc(no2)CCl 7N-651S c1ccc2cc(ccc2c1)OCc3cc(on3)c4ccc(cc4)Cl 7N-654S c1ccc(cc1)c2cc(no2)CN3CCN(CC3)c4ccccc4F 7N-657S c1ccc(cc1)c2cc(no2)CSc3ccc(cc3)Cl 7N-658S c1ccc(cc1)c2cc(no2)CSc3ccc(cc3)Br 7N-659S c1ccc(c(c1)c2cc(no2)COc3cc(ccc3Cl)Cl)Cl 7N-660S c1ccc2cc(ccc2c1)OCc3cc(on3)c4ccccc4Cl 7N-661S c1ccc(c(c1)c2cc(no2)CN3CCN(CC3)c4ccccc4F)Cl 7N-662S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)Cc4cc(on4)c5ccccc5Cl 7N-663S c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCCCC3 7N-664S c1cc(c(c(c1)F)C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCCCC3)F 7N-665S Cc1ccc(cc1)C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCCCC3 7N-666S c1cc(cc(c1)Cl)C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCCCC3 7N-669S c1cc(c(cc1/C=N\OC(=O)c2ccc(cc2Cl)Cl)[N+](=O)[O-])N3CCCCC3 7N-670S c1cc(sc1)C(=O)O/N=C/c2ccc(c(c2)[N+](=O)[O-])N3CCCCC3 7N-671S c1cc(cc(c1)OCc2cc(on2)c3ccc(c(c3)Cl)Cl)C(F)(F)F 7N-672S c1ccc(cc1)OCc2cc(on2)c3ccc(c(c3)Cl)Cl 7N-673S COC(=O)c1c(ccs1)OCc2cc(on2)c3ccc(c(c3)Cl)Cl 7N-674S COC(=O)c1c(ccs1)OCc2cc(on2)c3ccccc3 7N-675S c1cc(ccc1C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)F 7N-676S Cc1ccc(cc1)C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3 7N-677S c1ccc(c(c1)C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)Cl 7N-680S c1cc(c(cc1/C=N\OC(=O)C2CC2)[N+](=O)[O-])N3CCOCC3 7N-682S c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C\c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3 7N-683S c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCC(=O)N 7N-701 c1ccc2c(c1)nc(s2)SC(=O)c3cccnc3SCCC(=C(F)F)F 7N-704 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OC(=O)Nc3ccc(c(c3)Cl)Cl 7N-707 c1cc(c(nc1)n2cnc(n2)SCCC(=C(F)F)F)[N+](=O)[O-] 7N-708 c1ccc(cc1)C(=O)/C=C/C(=O)O 7N-710 c1cc(ccc1C(=O)/C=C/C(=O)c2ccc(cc2)Cl)Cl 7N-711 C=CCNc1nc(c(s1)C(=O)c2ccc(cc2)Br)N 7N-712 C=CCNc1nc(c(s1)C(=O)c2ccc(cc2)Cl)N 7N-713 CN1CC(C(C1)C(=O)c2ccc(cc2)Cl)C(=O)c3ccc(cc3)Cl 7N-714 COC(=O)/C=C/C(=O)c1ccccc1 7N-715 Cc1ccc(cc1)C(=O)C2CN(CC2C(=O)c3ccc(cc3)C)c4ccccc4 7N-716 CCOC(=O)C1CN(CC1C(=O)c2ccccc2)C 7N-717 C=CCNc1nc(c(s1)C(=O)c2ccc(cc2)F)N 7N-719 CCOC(=O)/C=C/C(=O)c1ccccc1 7N-720 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)Cc4c(cc(cn4)C(F)(F)F)Cl 7N-723 COC(=O)Cc1c(c(sc1C(=O)OC)N(C(=O)Nc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)Cl)C(=O)OC 7N-724 c1ccc(cc1)/N=N\c2ccc(cc2)NC(=O)c3ccccc3SCCC(=C(F)F)F 7N-725 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)SCCC(=C(F)F)F 7N-729 C=CCNc1nc(c(s1)C(=O)c2cccc(c2)[N+](=O)[O-])N 7N-730 c1cc(ccc1C(=O)/C=C/C(=O)O)Cl 7N-732 C=CCNc1nc(c(s1)C(=O)c2cccc(c2)C(F)(F)F)N 7N-733 c1cc(cc(c1)C#N)COc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 7N-734 Cc1ccc(cc1)C(=O)COc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 7N-735 CN1CC(C(C1)C(=O)c2ccc(cc2)OC)C(=O)c3ccc(cc3)OC 7N-736 c1ccc(cc1)C(=O)c2c(nc(s2)Nc3ccc(cc3)Cl)N 7N-737 COC(=O)Cc1c(c(sc1C(=O)OC)N(C(=O)Nc2ccccc2)C(=O)Nc3ccccc3)C(=O)OC 7N-739 c1ccc(c(c1)C(=O)Nc2nccs2)SCCC(=C(F)F)F 7N-740 c1cc(cc(c1)C(F)(F)F)C(=O)c2c(nc(s2)Nc3ccc(cc3)Cl)N 7N-741 c1cc(ccc1C(=O)c2c(nc(s2)Nc3ccc(cc3)Cl)N)Cl 7N-742 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCC(=O)c3ccc(cc3)Br 7N-743 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)O 7N-744 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 7N-745 Cc1ccc(cc1)/C(=N\OCc2ccc(cc2Cl)Cl)/COc3ccc(cc3)Cc4c(cc(cn4)C(F)(F)F)Cl 7N-746 COC(=O)C1CN(CC1C(=O)c2ccccc2)c3ccccc3 7N-747 COC(=O)/C=C/C(=O)c1ccc(cc1)Cl 7N-749 c1cc(ccc1Nc2nc(c(s2)C(=O)c3ccc(cc3Cl)Cl)N)Cl 7N-750 c1cc(ccc1C(=O)c2c(nc(s2)Nc3ccc(cc3)Cl)N)Br 7N-752 c1cc(ccc1N(c2ccnc(c2)C(F)(F)F)c3c(cc(cn3)C(F)(F)F)Cl)Cl 7N-753 COC(=O)c1c(c(sc1C(=O)OC)N(C(=O)NC2CCCCC2)C(=O)NC3CCCCC3)C(=O)OC 7N-754 c1cc(c(c(c1)Cl)F)CO/N=C(/COc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl)\c4ccc(cc4)Br 7N-755 COC(=O)CS(=O)(=O)CCC(=C(F)F)F 7N-758 COc1ccc(cc1)C(=O)/C=C/C(=O)c2ccc(cc2)OC 7N-759 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCC(=O)c3ccc(cc3)F 7N-760 Cc1ccc(cc1)C(=O)/C=C/C(=O)O 7N-761 c1[nH]c2c(n1)c(ncn2)SCCC(=C(F)F)F 7N-762 Cc1ccc(cc1)C2C(C(CN2C)C(=O)c3ccccc3)C(=O)c4ccccc4 7N-763 c1ccc2c(c1)c(=O)[nH]c(n2)SCCC(=C(F)F)F 7N-764 Cc1ccc(n1c2c(c(c(s2)C(=O)OC)CC(=O)OC)C(=O)OC)C 7N-767 c1cc(ccc1C(=O)c2c(nc(s2)Nc3ccc(cc3)Cl)N)F 7N-768 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OC/C(=N\O)/c3ccc(cc3)F 7N-769 CSc1nccc(n1)c2cc(sc2Cl)Cl 7N-770 Cc1ccc(cc1)C2=NNC(C2)C(=O)O 7N-771 CC(C)(C)Nc1nc(c(s1)C(=O)c2ccc(cc2)Cl)N 7N-773 c1cc(cc(c1)C(=O)N)COc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 7N-774 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCC(=O)NC(=O)Nc3ccc(c(c3)Cl)Cl 7N-775 Cc1ccc(cc1)C(=O)c2c(nc(s2)NC(C)(C)C)N 7N-776 Cc1ccc(cc1)C(=O)C2CN(CC2C(=O)OC)c3ccccc3 7N-778 CC(C)(C)Nc1nc(c(s1)C(=O)c2ccccc2)N 7N-779 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)NC2CCCCCCC2 7N-781 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)NCc2ccco2 7N-782 CC(C)(C)Nc1nc(c(s1)C(=O)c2ccc(cc2)Br)N 7N-783 c1ccc(cc1)n2ccnc2SCCC(=C(F)F)F 7N-784 CN1CC(C(C1c2ccc(cc2)Cl)C(=O)c3ccccc3)C(=O)c4ccccc4 7N-785 Cc1ccc(cc1)NC(=O)Oc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 7N-788 Cc1c(c(=O)cco1)Cc2ccc(cc2)Cl 7N-792 c1cc(ccc1Cc2c(ccc(c2O)C=O)O)Cl 7N-793 c1cnc(nc1)SCCC(C(F)(F)Br)(F)Br 7N-796 c1cc(cc(c1)[N+](=O)[O-])C(=O)c2c(nc(s2)Nc3ccc(cc3)Cl)N 7N-797 COC(=O)c1c(cc(=O)n(n1)c2ccccc2)Oc3ccc(cc3)Cc4c(cc(cn4)C(F)(F)F)Cl 7N-798 COc1cnc(nc1O)SCCC(=C(F)F)F 7N-799 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4ccc(cc4)[N+](=O)[O-] 7N-801 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4ccc(cc4)C 7N-802 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4cccc(c4)C(F)(F)F 7N-803 COc1ccc(cc1)NS(=O)c2c3ccccc3ccc2OC 7N-804 CCOC(=O)c1c2ccc(cc2n3c1cccc3)Oc4c(cc(cn4)C(F)(F)F)Cl 7N-805 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4c5ccccc5oc4C(=O)c6ccccc6 7N-806 COc1ccc2ccccc2c1S(=O)NCc3ccccc3 7N-807 COc1ccc2ccccc2c1S(=O)NC3CCCCC3 7N-808 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC#N 7N-809 CCOC(=O)COc1ccc2c(c1)n3ccccc3c2C(=O)OCC 7N-810 COc1ccc2ccccc2c1S(=O)N3CCOCC3 7N-811 COc1ccc2ccccc2c1S(=O)N3CCN(CC3)Cc4ccccc4 7N-812 CCOC(=O)c1c2ccc(cc2n3c1cccc3)Oc4c(nns4)c5ccccc5 7N-814 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4c5ccccc5oc4C(=O)c6ccc(cc6)Cl 7N-815 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4c(cccc4Cl)Cl 7N-816 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4ccc(cc4)F 7N-817 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)O 7N-818 Cc1cc(cc(c1)NS(=O)c2c3ccccc3ccc2OC)C 7N-819 COc1ccc2ccccc2c1S(=O)Nc3cccc(c3)C(F)(F)F 7N-820 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)NN 7N-821 Cn1c(c(c(n1)C(F)(F)F)C#N)N(C)N(S(=O)(=O)C)S(=O)(=O)C 7N-822 COc1ccc2ccccc2c1S(=O)N3CCN(CC3)c4ccc(cc4)Cl 7N-823 COc1ccc2ccccc2c1S(=O)N3CCN(CC3)c4ccccc4F 7N-824 CN1CCN(CC1)S(=O)c2c3ccccc3ccc2OC 7N-825 COc1ccc2ccccc2c1S(=O)N3CCN(CC3)c4ccccn4 7N-826 COc1ccc2ccccc2c1S(=O)N3CCN(CC3)c4cccc(c4)C(F)(F)F 7N-827 COc1ccc2ccccc2c1S(=O)NCc3ccc(cc3)Cl 7N-828 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCc4c(cccc4Cl)F 7N-829 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)N/N=C/c4ccc(cc4)C 7N-831 COc1ccc2ccccc2c1S(=O)S(=O)(=O)c3ccccc3 7N-832 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)NNC(=O)Nc4ccccc4 7N-833 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)NNC(=S)NC 7N-834 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)N/N=C/c4ccc(cc4)Cl 7N-835 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)N/N=C/c4ccccc4C(F)(F)F 7N-836 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)N/N=C/c4cccc(c4)[N+](=O)[O-] 7N-837 COc1ccc2ccccc2c1S(=O)Nc3ccncc3 7N-838 COc1ccc2ccccc2c1S(=O)O 7N-839 CCNC(=S)NNC(=O)COc1ccc2c(c1)n3ccccc3c2C(=O)OCC 7N-840 CCOC(=O)c1c(c2cccc3c2n(c1=O)CCC3)O 7N-901 COc1ccc(cc1OC)NC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O 7N-903 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C(=O)NN)O 7N-904 c1cc(cc(c1)Cl)CNC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O 7N-905 CC(=O)CC(c1cc(cc(c1OCc2ccccc2)Cl)Cl)O 7N-907 C/C(=[N+](/C)\[O-])/CC(c1cc(cc(c1OCc2ccccc2)Cl)Cl)O 7N-908 c1cc(oc1)C(=O)N/N=C/c2cnc(s2)Cl 7P-001 c1cc(ccc1C(=O)N/N=C/c2cnc(s2)Cl)C(F)(F)F 7P-002 CCOC(=O)CCC(=O)N1Cc2ccccc2NC1c3cccs3 7P-005 c1ccc2c(c1)CCN2/C(=N\O)/c3cccc(c3)[N+](=O)[O-] 7P-006 CN(Cc1ccccc1)/C(=N/O)/c2cccc(c2)Cl 7P-010 c1ccc(c(c1)C(=O)O)Nc2ccnc(c2)C(F)(F)F 7P-011 c1csc(n1)NC(=O)c2c(nc3n(c2=O)ccs3)O 7P-014 c1cc(ccc1Oc2ncc(s2)C=O)Br 7P-015 COc1ccccc1C2NC(CS2)C(=O)O 7P-016 c1cc(ccc1C2NC(CS2)C(=O)O)F 7P-017 c1ccc(cc1)CN/C(=N/O)/c2cccc(c2)Cl 7P-020 c1ccc(c(c1)/C(=N/O)/Nc2ccc(cc2)Cl)Cl 7P-022 COC(=O)c1ccc(cc1)Oc2ccc(cc2)C#N 7P-023 c1cc(ccc1C2NC(CS2)C(=O)O)Br 7P-024 Cc1ccc(cc1)/C(=C\C#N)/N 7P-028 c1cc(ccc1C2NC(CS2)C(=O)O)[N+](=O)[O-] 7P-029 c1ccc(cc1)/C=C/C2NC(CS2)C(=O)O 7P-030 c1ccc(c(c1)C2NC(CS2)C(=O)O)C(F)(F)F 7P-031 c1cc(cc(c1)[N+](=O)[O-])C2NC(CS2)C(=O)O 7P-032 c1cc2c(cc1C3NC(CS3)C(=O)O)OCO2 7P-033 CCCCCCC1NC(CS1)C(=O)O 7P-035 Cc1ccc(cc1)COn2ccnc2/C=C/3\C(=O)NC(=O)S3 7P-036 c1ccc(cc1)CCNCC(C(F)(F)F)O 7P-037 c1ccc(cc1)CCC2NC(CS2)C(=O)O 7P-038 Cc1ccc(cc1)c2c(c(cc(n2)c3cccs3)C(F)(F)F)C#N 7P-040 CC1(NC(CS1)C(=O)O)c2ccc(cc2)OC 7P-041 C/C(=C\C(=O)C(F)(F)F)/Nc1ccccc1c2ccccc2 7P-044 CCOC(=O)c1c(onc1C(=O)C)C 7P-048 c1cc(ccc1/C(=C\C#N)/N)Cl 7P-049 CN(C)/C=C/C(=C/C(=O)C(F)(F)F)/Nc1ccccc1c2ccccc2 7P-050 c1ccc(cc1)N/C(=N\O)/c2ccccc2Cl 7P-054 c1ccc2c(c1)c(c[nH]2)/C=N/O 7P-055 c1cc(c(cc1[N+](=O)[O-])Br)F 7P-057 c1ccc(cc1)CCNCC(c2ccccc2)O 7P-058 CN(c1ccccc1)NC(=S)N 7P-060 c1cc(ccc1/C(=C\C#N)/N)Br 7P-061 c1ccc(cc1)c2ccccc2Nc3ccnc(c3)C(F)(F)F 7P-063 Cc1ccc(cc1)n2c(cc(n2)c3ccc(cc3)Br)N 7P-064 c1cc(sc1)c2cc(c(c(n2)c3ccc(cc3)Cl)C#N)C(F)(F)F 7P-065 c1ccc(cc1)c2cc(c(c(n2)c3ccc(cc3)Cl)C#N)C(F)(F)F 7P-066 c1cc(ccc1/C(=C/C#N)/N)C(F)(F)F 7P-068 CONC(=O)C1CCN(CC1)C(=O)OCc2ccccc2 7P-069 c1cc(sc1)c2cc(c(c(n2)c3ccc(cc3)Br)C#N)C(F)(F)F 7P-071 c1ccc(cc1)c2cc(c(c(n2)c3ccc(cc3)Br)C#N)C(F)(F)F 7P-074 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)NCCCl 7P-079 Cc1cccc(c1C)NC(=O)C 7P-080 Cc1[nH]c2cccc(c2n1)Cl 7P-082 c1cc(cc(c1)C(F)(F)F)CNCC(C(F)(F)F)O 7P-085 Cn1cccc1/C=N/O 7P-087 Cc1ccc(c(c1)NC(=O)C)C 7P-092 c1ccc(cc1)N/C(=N\O)/c2cccnc2 7P-093 C1CSCCN1CC(C(F)(F)F)O 7P-095 c1cc(ccc1c2c(c(c(c(n2)N)C#N)C#N)C#N)Br 7P-097 c1cc(ccc1c2c(c(c(c(n2)N)C#N)C#N)C#N)Cl 7P-098 C1COCCN1CC(C(F)(F)F)O 7P-100 c1cc(ccc1c2c(c(c(c(n2)N)C#N)C#N)C#N)C(F)(F)F 7P-101 c1ccnc(c1)CCNCC(C(F)(F)F)O 7P-102 CN(C)/C=N/c1c(c(c(c(n1)c2ccc(cc2)Cl)C#N)C#N)C#N 7P-103 c1cc(cc(c1)C(F)(F)F)/C=N/O 7P-105 c1ccnc(c1)/C(=C/C#N)/N 7P-106 c1cc(cc(c1)Oc2ccc(cc2)/C(=C/C#N)/N)C(F)(F)F 7P-108 CCO/C=C(\C#N)/S(=O)(=O)c1ccccc1 7P-109 c1ccnc(c1)c2c(c(c(c(n2)N)C#N)C#N)C#N 7P-112 c1ccc2c(c1)nc(s2)Sc3ncc(s3)C=O 7P-115 Cc1ccccc1/C=N\NC(=O)c2c(ccs2)n3cccc3 7P-301S CN(C)c1ccc(cc1)/C=N/NC(=O)c2c(ccs2)n3cccc3 7P-302S C/C(=N\NC(=O)c1c(ccs1)n2cccc2)/c3cccs3 7P-303S Cc1c(sc2n1c3ccccc3n2)/C(=N/OCC=C)/C 7P-304S Cc1c(sc2n1c3ccccc3n2)/C(=N/OC(C)C)/C 7P-305S Cc1cccc(c1)/C=N\NC(=O)c2ccccc2n3cccc3 7P-307S COc1cccc(c1)/C=N\NC(=O)c2ccccc2n3cccc3 7P-308S COc1ccc(cc1)/C=N/NC(=O)c2c(ccs2)n3cccc3 7P-309S C/C(=N\NC(=O)c1c(ccs1)n2cccc2)/c3ccc(cc3)Cl 7P-311S Cc1c(sc2n1ncn2)/C(=N/OC(C)C)/CSc3ccc(cc3)Cl 7P-313S Cc1ccc(cc1)CO/N=C(\CSc2ccc(cc2)Cl)/c3c(n4c(s3)ncn4)C 7P-314S Cc1c(sc2n1ncn2)/C(=N/OCc3cccc(c3)Cl)/CSc4ccc(cc4)Cl 7P-315S Cc1c(sc2n1ncn2)/C(=N/OCc3ccccc3Cl)/CSc4ccc(cc4)Cl 7P-316S Cc1c(sc2n1ncn2)/C(=N/OCc3ccc(cc3)C(F)(F)F)/CSc4ccc(cc4)Cl 7P-320S Cc1c(sc2n1ncn2)/C(=N/OCc3ccc(cc3)OC)/CSc4ccc(cc4)Cl 7P-321S c1ccc(c(c1)/C=N\NC(=O)c2ccccc2n3cccc3)F 7P-323S c1ccc(c(c1)C(=O)N/N=C/c2c(cccc2Cl)F)n3cccc3 7P-324S c1ccc(c(c1)C(=O)N/N=C\c2cccc(c2)Br)n3cccc3 7P-325S C/C(=N\NC(=O)c1c(ccs1)n2cccc2)/c3ccc(cc3)OC 7P-326S C/C(=N\NC(=O)c1c(ccs1)n2cccc2)/c3cccc(c3)C(F)(F)F 7P-327S c1ccc\2c(c1)CCC/C2=N\NC(=O)c3c(ccs3)n4cccc4 7P-328S Cc1c(sc2n1c3ccccc3n2)/C(=N/OC(=O)c4cccc(c4)OC)/C 7P-331S Cc1ccc(cc1)C(=O)NCc2c(c(n(c2n3cccc3)Cc4ccccc4)C)C 7P-332S c1ccc2c(c1)nc(s2)N3CCN(CC3)Cc4ccc(c(c4)Cl)Cl 7P-333S c1ccc2c(c1)nc(s2)N3CCN(CC3)Cc4ccc(cc4)[N+](=O)[O-] 7P-334S COc1ccc(cc1)CN2CCN(CC2)c3nc4ccccc4s3 7P-335S Cc1ccccc1CN2CCN(CC2)c3nc4ccccc4s3 7P-336S c1ccc2c(c1)nc(s2)N3CCN(CC3)Cc4cccc(c4)C(F)(F)F 7P-337S c1ccc2c(c1)nc(s2)N3CCN(CC3)Cc4c(cccc4Cl)F 7P-338S c1ccc(cc1)CN2CCN(CC2)c3nc4ccccc4s3 7P-339S Cc1ccc(cc1)C(=O)N2CCN(CC2)c3nc4ccccc4s3 7P-340S c1ccc2c(c1)nc(s2)N3CCN(CC3)C(=O)c4cccc(c4)C(F)(F)F 7P-341S c1ccc2c(c1)nc(s2)N3CCN(CC3)C(=O)c4ccc(cc4)Cl 7P-353S c1ccc(cc1)C(=O)N2CCN(CC2)c3nc4ccccc4s3 7P-354S COc1cccc(c1)C(=O)N2CCN(CC2)c3nc4ccccc4s3 7P-355S CCC(=O)N1CCN(CC1)c2nc3ccccc3s2 7P-356S c1ccc2c(c1)nc(s2)N3CCN(CC3)C(=O)C4CC4 7P-357S COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3nc4ccccc4s3 7P-358S CC(C)(C)C(=O)Nc1c(cccn1)C(=O)c2ccccc2 7P-360S c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3nc4ccccc4s3 7P-361S CS(=O)(=O)N1CCN(CC1)c2nc3ccccc3s2 7P-362S Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3nc4ccccc4s3 7P-363S c1ccc2c(c1)nc(s2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 7P-364S c1ccc2c(c1)nc(s2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)[N+](=O)[O-] 7P-365S c1ccc2c(c1)nc(s2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Br 7P-366S Cc1c(sc2n1c3ccccc3n2)/C(=N/OC(=O)c4ccccc4)/C 7P-367S COC(=O)c1c(c2ccccc2s1)N 7P-368S CN(C)c1ccc(cc1)/C=N\NC(=O)c2ccccc2n3cccc3 7P-370S c1ccc(c(c1)C(=O)N/N=C\c2cccs2)n3cccc3 7P-373S Cc1ccccc1/C=N\NC(=O)c2ccccc2n3cccc3 7P-375S c1ccc(c(c1)/C=N\NC(=O)c2ccccc2n3cccc3)Cl 7P-376S Cc1c(n(c(c1CNC(=O)c2ccc(cc2)F)n3cccc3)Cc4ccccc4)C 7P-378S Cc1c(n(c(c1CNC(=O)c2cccc(c2)OC)n3cccc3)Cc4ccccc4)C 7P-379S Cc1c(n(c(c1CNC(=O)c2c(cccc2F)F)n3cccc3)Cc4ccccc4)C 7P-380S Cc1c(n(c(c1CNC(=O)c2cccs2)n3cccc3)Cc4ccccc4)C 7P-381S CSc1nnc(o1)c2c(ccs2)n3cccc3 7P-382S c1ccc(cc1)CSc2nnc(o2)c3c(ccs3)n4cccc4 7P-383S Cc1c(n(c(c1CNC(=O)c2ccccc2Cl)n3cccc3)Cc4ccccc4)C 7P-384S CCC(=O)NCc1c(c(n(c1n2cccc2)Cc3ccccc3)C)C 7P-385S Cc1c(n(c(c1CNC(=O)C2CC2)n3cccc3)Cc4ccccc4)C 7P-386S Cc1c(n(c(c1CNC(=O)c2cccc(c2)Cl)n3cccc3)Cc4ccccc4)C 7P-391S Cc1c(n(c(c1CNC(=O)c2cccc(c2)C(F)(F)F)n3cccc3)Cc4ccccc4)C 7P-393S c1cc(c[n+](c1)[O-])CC#N 7P-396S Cc1ccc(cc1)S(=O)(=O)NCc2c(c(n(c2n3cccc3)Cc4ccccc4)C)C 7P-397S CCNC(=O)NCc1c(c(n(c1n2cccc2)Cc3ccccc3)C)C 7P-398S Cc1c(n(c(c1CNS(=O)(=O)c2ccccc2)n3cccc3)Cc4ccccc4)C 7P-399S Cc1c(n(c(c1CNS(=O)(=O)c2ccc(cc2)Cl)n3cccc3)Cc4ccccc4)C 7P-400S Cc1c(n(c(c1CNS(=O)(=O)c2ccc(cc2)Br)n3cccc3)Cc4ccccc4)C 7P-401S Cc1c(n(c(c1CNS(=O)(=O)c2cc(cc(c2)Cl)Cl)n3cccc3)Cc4ccccc4)C 7P-402S CSc1nc2c3ccccc3sc2c(n1)O 7P-403S CSc1nc2c3ccccc3sc2c(n1)Cl 7P-404S Cc1ccc(cc1)NC(=O)NCc2c(c(n(c2n3cccc3)Cc4ccccc4)C)C 7P-407S Cc1c(n(c(c1CNC(=O)Nc2ccc(cc2)Cl)n3cccc3)Cc4ccccc4)C 7P-408S CC(C)(C)c1cc2cccnc2[nH]1 7P-418S COc1ccc(cc1)CSc2nnc(o2)c3c(ccs3)n4cccc4 7P-419S c1ccn(c1)c2ccsc2c3nnc(o3)SCc4ccc(cc4)Cl 7P-420S c1ccn(c1)c2ccsc2c3nnc(o3)SCc4c(cccc4Cl)Cl 7P-421S c1ccn(c1)c2ccsc2c3nnc(o3)SCc4ccc(cc4)F 7P-422S CC(C)(C)c1cc2cccnc2n1Cc3ccccc3 7P-425S c1ccn(c1)c2ccsc2c3nnc(o3)SCc4cccc(c4)C(F)(F)F 7P-430S c1ccn(c1)c2ccsc2c3nnc(o3)SCc4cccc(c4)Cl 7P-431S c1ccn(c1)c2ccsc2c3nnc(o3)SCC(=O)c4ccc(cc4)Cl 7P-432S Cc1cccc(c1)C(=O)NCc2c(c(n(c2n3cccc3)Cc4ccccc4)C)C 7P-492S c1ccc2c(c1)C(=O)/C(=C/NC(=O)N)/C(=O)O2 7P-503S c1ccc(cc1)N/C=C\2/C(=O)c3ccccc3OC2=O 7P-504S c1ccc2c(c1)C(=O)/C(=C/Nc3cccc(c3)Cl)/C(=O)O2 7P-505S c1ccc(cc1)C(=O)N2CCC(CC2)c3nc4ccccc4s3 7P-506S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)c4cccs4 7P-507S c1ccc2c(c1)C(=O)/C(=C/Nc3cccc(c3)C(F)(F)F)/C(=O)O2 7P-509S c1ccc2c(c1)C(=O)/C(=C/Nc3ccc(cc3)C(F)(F)F)/C(=O)O2 7P-510S Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F 7P-512S COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F 7P-513S c1cc(c(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F 7P-514S c1ccc2c(c1)C(=O)/C(=C/Nc3ccc(cc3)Br)/C(=O)O2 7P-516S c1ccc2c(c1)C(=O)/C(=C/Nc3ccc(c(c3)Cl)Cl)/C(=O)O2 7P-517S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)c4cccc(c4)Cl 7P-519S CCOC(=O)/C(=N\OC)/CN1CCOCC1 7P-521S COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F 7P-522S c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)Br 7P-523S c1cc(ncc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl 7P-524S CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F 7P-526S CN(C)S(=O)(=O)N1CCN(CC1)c2ccc(cn2)C(F)(F)F 7P-527S c1ccc(cc1)c2ccc(nn2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)F 7P-528S c1ccc(cc1)c2ccc(nn2)N3CCN(CC3)S(=O)(=O)c4cc(cc(c4)Cl)Cl 7P-529S CCOC(=O)/C(=N\OC)/CN1CCN(CC1)c2ccc(cc2)F 7P-530S CCOC(=O)/C(=N\OC)/CN1CCCCC1 7P-531S c1ccc(cc1)c2cc(c(o2)n3cccc3)c4nc(on4)c5ccc(cc5)F 7P-567S c1ccc(cc1)c2cc(c(o2)n3cccc3)c4nc(on4)c5ccccc5Cl 7P-578S c1ccc(cc1)c2cc(c(o2)n3cccc3)c4nc(on4)c5c(cccc5F)F 7P-579S Cc1c(snn1)SCCNC(=O)Nc2ccccc2 7P-580S Cc1c(snn1)SCCNC(=O)Nc2ccc(cc2)Cl 7P-581S Cc1cccc(c1NC(=O)NCCSc2c(nns2)C)C 7P-582S Cc1c(snn1)SCCNC(=O)NC2CCCCC2 7P-583S Cc1c(snn1)SCCNS(=O)(=O)c2ccc(cc2)OC 7P-584S CCn1c(nnc1SCC=C)c2c(=O)ccn(n2)c3ccc(cc3)Cl 7P-642S CCn1c(nnc1SC)c2c(=O)ccn(n2)c3ccc(cc3)Cl 7P-643S CCn1c(nnc1SC=C=C)c2c(=O)ccn(n2)c3ccc(cc3)Cl 7P-644S CCn1c(nnc1SCC(=O)OC)c2c(=O)ccn(n2)c3ccc(cc3)Cl 7P-645S CCn1c(nnc1SCc2cccc(c2)C(F)(F)F)c3c(=O)ccn(n3)c4ccc(cc4)Cl 7P-646S CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)c3c(=O)ccn(n3)c4ccc(cc4)Cl 7P-647S COc1ccc(cc1)n2ccc(=O)c(n2)C(=O)OC 7P-649S Cc1ccc(cc1)n2ccc(=O)c(n2)c3ccnc(n3)SC 7P-653S COc1ccc(cc1)n2ccc(=O)c(n2)C(=O)O 7P-655S Cc1ccc(cc1)n2ccc(=O)c(n2)c3ccnc(n3)SCc4ccc(cc4Cl)Cl 7P-656S Cc1ccc(cc1)n2ccc(=O)c(n2)c3ccnc(n3)SCc4cccc(c4)Cl 7P-657S CCSc1nccc(n1)c2c(=O)ccn(n2)c3ccc(cc3)C 7P-658S Cc1ccc(cc1)n2ccc(=O)c(n2)c3ccnc(n3)SCC=C 7P-661S Cc1ccc(cc1)n2ccc(=O)c(n2)c3ccnc(n3)SCC#C 7P-662S CN(C(=O)c1c(=O)ccn(n1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)OC 7P-666S CN(C(=O)c1c(=O)ccn(n1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)[N+](=O)[O-] 7P-668S c1cc(ccc1CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)I)C#N 7P-700 Cc1c(sc([nH+]1)c2cccnc2)C(=O)C.[Cl-] 7P-701 Cc1c(sc([nH+]1)c2ccncc2)C(=O)C.[Cl-] 7P-702 COc1cccc(c1)CNC(=O)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCc3cccc(c3)OC 7P-703 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/N(C)C 7P-704 Cc1cccc(n1)n2cc(nc2)C(=O)N/N=C\c3ccc(cc3)Br 7P-705 Cc1cccc(n1)n2cc(nc2)C(=O)N/N=C\c3ccc(cc3)[N+](=O)[O-] 7P-706 c1csc2c1c(ncn2)Cl 7P-707 Cc1c(sc(n1)c2ccncc2)C(=O)C 7P-712 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/N(C)C 7P-713 Cc1cccc(n1)n2cc(nc2)C(=O)NNC(=O)Nc3ccc(cc3)Cl 7P-714 Cc1cccc(n1)n2cc(nc2)C(=O)NNC(=S)Nc3ccccc3 7P-715 Cc1ccc(cc1)C(=O)NNC(=O)c2cn(cn2)c3cccc(n3)C 7P-716 Cc1cccc(n1)n2cc(nc2)C(=O)NNS(=O)(=O)c3ccc(cc3)OC 7P-717 Cc1cc(ccc1NC(=O)CC2N(C(=O)N(O2)C)c3ccc(cc3)Cl)[N+](=O)[O-] 7P-719 Cc1ccc(cc1)/C=C\2/C(=O)N(/C(=N/n3cnnc3)/S2)c4ccccc4 7R-0001 CCOC(=O)CN\1C(=O)CS/C1=N\n2cnnc2 7R-0002 Cc1cc(c(n1n2cnnc2)C)/C=C/C(=O)O 7R-0003 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2)F)C(=O)C 7R-0008 CC1=NN(C(=O)C1)C(C)(C)C 7R-0012 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)Br 7R-0014 Cc1ccc(n1c2c(ccs2)C(=O)OC)C 7R-0015 Cc1cc2nc(c(c(n2n1)O)Cl)C 7R-0016 c1ccc(cc1)N\2C(=O)/C(=C/c3cccs3)/S/C2=N\n4cnnc4 7R-0017 CC(=O)Nc1ccc(cc1)/C=C\2/C(=O)N(/C(=N/n3cnnc3)/S2)c4ccccc4 7R-0018 c1cc(ccc1c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F)Br 7R-0019 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)O)Cl)C)C 7R-0020 Cc1cc2nc(c(c(n2n1)O)C)C 7R-0021 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3OCCOCCOc4cc(ccc4OC)/C=C\c5cc(c(c(c5)OC)OC)OC 7R-0023 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)O)C/C=C/c5ccccc5)C)C 7R-0025 CCC(=O)CC(C)(Nc1cc(n[nH]1)c2c(ccs2)n3c(ccc3C)C)O 7R-0026 Cc1cc2nc(cc(n2n1)O)CCl 7R-0027 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)C(F)(F)F)c5cccc(c5)Cl)C 7R-0030 CC(CC(=O)Nc1ccc(cc1)C(F)(F)F)N2CCCC2 7R-0032 CN(C)/C=C(/C#N)\c1ccc(s1)C(=O)c2ccc(cc2)Cl 7R-0034 CC1=C(C(C(=C(N1)C)C(=O)OCc2ccccc2)c3ccc(cc3)Br)C(=O)OC 7R-0036 CC(CC(=O)Nc1ccccn1)N2CCCC2 7R-0038 CC(CC(=O)Nc1cccc(c1)C(F)(F)F)N2CCCC2 7R-0039 CCNC(=S)Nn1cnnc1 7R-0040 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)O)C)C)C 7R-0041 c1cc(c(cc1[N+](=O)[O-])F)C(=O)O 7R-0042 Cc1ccc(n1c2c(ccs2)C(=O)O)C 7R-0044 c1nncn1/N=C\2/N(C(=O)CS2)CC(=O)O 7R-0045 CCN\1C(=O)CS/C1=N\n2cnnc2 7R-0046 c1ccc(cc1)N\2C(=O)/C(=C/c3ccc(nc3)Cl)/S/C2=N\n4cnnc4 7R-0047 Cc1ccc(n1c2c(ccs2)C(=O)CC#N)C 7R-0048 CC(CC(=O)Nc1cccc(c1)Cl)N2CCCC2 7R-0049 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)C(F)(F)F)C#N)C 7R-0050 Cc1cc2ncc(c(n2n1)C(F)(F)F)C#N 7R-0052 Cc1cc2nc(cc(n2n1)O)CSc3ccccc3 7R-0053 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc(cc5)c6ccccc6)C 7R-0056 CCN\1C(=O)/C(=C/c2ccc(nc2)Cl)/S/C1=N\n3cnnc3 7R-0057 Cc1ccc(n1c2c(ccs2)c3cc4nc(cc(n4n3)C)C)C 7R-0061 CCN\1C(=O)/C(=C/c2ccc(cc2)F)/S/C1=N\n3cnnc3 7R-0063 CCN\1C(=O)/C(=C/c2cccs2)/S/C1=N\n3cnnc3 7R-0064 CCN\1C(=O)/C(=C/c2ccco2)/S/C1=N/n3cnnc3 7R-0065 CCN\1C(=O)/C(=C/c2ccc(cc2)O)/S/C1=N\n3cnnc3 7R-0066 CCN\1C(=O)/C(=C/c2ccc(cc2)NC(=O)C)/S/C1=N\n3cnnc3 7R-0067 CN(C)/C=C(\C#N)/C(=O)N/N=C(\CC(=O)C(F)(F)F)/c1ccco1 7R-0069 CC(CC(=O)Nc1ccc(cc1)OC)N2CCCC2 7R-0070 Cc1ccc(cc1)NC(=O)CC(C)N2CCCC2 7R-0071 CC(CC(=O)Nc1ccc(cc1)F)N2CCCC2 7R-0072 Cc1cc2ncc(c(n2n1)c3ccccc3)n4cncn4 7R-0074 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)c5ccccc5)n6cncn6)C 7R-0075 COc1ccc(cc1)CCC(c2ccccn2)O 7R-0076 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NCCCn4ccnc4 7R-0200 CCCCCCCNC(=O)c1cc(c[nH]1)C(=O)c2cccc(c2)C(F)(F)F 7R-0202 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)c2cccc(c2)C(F)(F)F 7R-0203 c1cc(cc(c1)F)NC(=O)NNC(=O)C2CC(=NO2)c3cccnc3 7R-0204 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 7R-0205 c1ccc(c(c1)NC(=O)NNC(=O)C2CC(=NO2)c3cccnc3)Cl 7R-0206 c1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)c3cccc(c3)C(F)(F)F 7R-0207 c1cc(cc(c1)C(F)(F)F)C(=O)c2cc([nH]c2)C(=O)NCc3ccc(cc3)F 7R-0208 c1ccc(c(c1)NC(=O)NNC(=O)C2CC(=NO2)c3cccnc3)F 7R-0209 COc1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)c3cccc(c3)C(F)(F)F 7R-0210 COc1ccc(cc1)NC(=O)NNC(=O)C2CC(=NO2)c3cccnc3 7R-0211 c1ccc(cc1)N2CCN(CC2)C(=O)C3Cc4c5ccccc5ccc4O3 7R-0213 c1cc(c(cc1CN2CCC(CC2)C(=O)NN)Cl)Cl 7R-0214 CCOC(=O)c1cc2c3ccccc3ccc2o1 7R-0215 c1cc(cc(c1)C(F)(F)F)C(=O)c2cc([nH]c2)C(=O)NCC3CCCO3 7R-0216 c1ccnc(c1)CCNC(=O)c2cc(c[nH]2)C(=O)c3cccc(c3)C(F)(F)F 7R-0217 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccnc3 7R-0218 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3cc4c(cc3Br)OCO4 7R-0219 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCC3CCCO3 7R-0220 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCc3ccccn3 7R-0221 c1cc(cc(c1)C(F)(F)F)C(=O)c2cc([nH]c2)C(=O)NCc3cccnc3 7R-0222 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccs3 7R-0223 CCC(C)(C)NC(=O)/C=C/c1cc2c(cc1Br)OCO2 7R-0224 c1ccc(c(c1)CNC(=O)/C=C/c2cc3c(cc2Br)OCO3)Cl 7R-0225 c1ccc(c(c1)N2CCN(CC2)C(=O)/C=C/c3cc4c(cc3Br)OCO4)F 7R-0226 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)/C=C/c3cc4c(cc3Br)OCO4)C(F)(F)F 7R-0227 c1ccc(cc1)C(=O)CNC(=O)C2Cc3c4ccccc4ccc3O2 7R-0229 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NCCCl 7R-0230 c1ccc2c(c1)ccc3c2CC(O3)C(=O)Nc4[nH]c5ccccc5n4 7R-0231 c1ccc2c(c1)ccc3c2CC(O3)C(=O)NCc4cccc(c4)C(F)(F)F 7R-0232 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCOC 7R-0233 Cc1ccc(cc1)C(=O)NNC(=O)C2CCN(CC2)Cc3ccc(c(c3)Cl)Cl 7R-0234 CC(C)(C)c1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)Cc3ccc(c(c3)Cl)Cl 7R-0235 c1cc(ccc1CNC(=O)/C=C/c2cc3c(cc2Br)OCO3)Cl 7R-0238 c1cc(sc1)C(=O)NNC(=O)C2CCN(CC2)Cc3ccc(c(c3)Cl)Cl 7R-0239 c1cc(c(cc1CN2CCC(CC2)C(=O)NNC(=O)C3CC3)Cl)Cl 7R-0240 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3ccco3 7R-0241 Cc1ccc(cc1)NC(=S)N 7R-0242 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)OC 7R-0246 c1ccc(cc1)S(=O)(=O)NNC(=O)C2CC(=NO2)c3cccnc3 7R-0248 Cc1ccc(cc1)Nc2nc(c(s2)C(=O)C)C 7R-0250 CCCCN(CCCC)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)C(C)(C)C 7R-0252 CCNC(=O)NNC(=O)C1CC(=NO1)c2cccnc2 7R-0254 COc1ccc(cc1)CNC(=O)/C(=C/c2cccs2)/c3ccccc3 7R-0255 COc1ccc(cc1)S(=O)(=O)NNC(=O)C2CC(=NO2)c3cccnc3 7R-0256 c1cc(cnc1)C2=NOC(C2)C(=O)NNS(=O)(=O)c3ccc(cc3)F 7R-0257 COc1ccccc1CNC(=O)/C=C/c2cc3c(cc2Br)OCO3 7R-0259 c1cc(ccc1N2CCN(CC2)C(=O)/C=C/c3cc4c(cc3Br)OCO4)Cl 7R-0260 COc1cccc(c1)N2CCN(CC2)C(=O)/C(=C/c3cccs3)/c4ccccc4 7R-0261 c1ccc(cc1)C(=O)CNC(=O)/C(=C/c2cccs2)/c3ccccc3 7R-0262 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)/C(=C/c2cccs2)/c3ccccc3 7R-0263 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCC(=O)OC 7R-0264 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SC/C=C/c5ccccc5 7R-0265 COC(=O)/C=C/c1cc2cc(ccc2o1)Cl 7R-0268 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl)F 7R-0269 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3 7R-0270 COCCCNC(=O)N 7R-0274 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 7R-0276 CCc1cc(=O)[nH]c(n1)SCc2ccc(cc2)C 7R-0277 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCOC 7R-0278 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3Cc4ccccc4)SCC(=O)N 7R-0279 Cc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 7R-0280 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3)F 7R-0284 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3)F 7R-0285 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)O 7R-0286 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)NC34CC5CC(C3)CC(C5)C4 7R-0287 c1cc(sc1)C2=NOC(C2)C(=O)NN 7R-0289 COCCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)F 7R-0290 c1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)F 7R-0291 COc1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)F 7R-0292 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)NCC3CCCO3)F 7R-0293 c1cc(sc1)CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)F 7R-0294 COC(=O)/C(=C/c1cccs1)/c2ccccc2 7R-0295 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)NCc3cccs3 7R-0299 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)NCc3ccc(cc3)F 7R-0300 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)N 7R-0302 CCN(CC)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)C(C)(C)C 7R-0303 Cc1cccc(c1)Nc2nc(c(s2)C(=O)C)C 7R-0304 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 7R-0305 COc1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)C/C=C/c3ccccc3 7R-0306 Cc1ccc(cc1)Nc2ncc(s2)C(=O)C 7R-0307 Cc1cccc(c1)Nc2ncc(s2)C(=O)C 7R-0308 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3ccc(cc3)OC 7R-0309 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCN(C)C 7R-0310 CS(=O)(=O)O/N=C/1\CCCCC1c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] 7R-0311 c1ccc(cc1)S(=O)(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 7R-0312 COc1ccc(cc1)S(=O)(=O)O/N=C/2\CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 7R-0313 c1cc(ccc1CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)F)F 7R-0315 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)/N=C/N(C)C 7R-0316 CC(C)N(C(C)C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)F 7R-0317 CC(C)C1C(=O)N=C2N1C(=S)Nc3c2cc(c(c3)OC)OC 7R-0318 c1cc(cnc1)CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)F 7R-0319 CC(C)(C)c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccc(c3)C(F)(F)F 7R-0320 CCC(C)(C)NC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)C 7R-0321 Cc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccnc3 7R-0322 Cc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 7R-0323 CCOC(=O)/C=C/COc1ccccc1[N+](=O)[O-] 7R-0325 c1cc(oc1)CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)F 7R-0326 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)F 7R-0327 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2cccc(c2)OC 7R-0328 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)NCc3ccco3 7R-0329 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)C 7R-0331 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)NCC3CCCO3 7R-0332 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)NCc3ccco3 7R-0333 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)/C(=C/c4cccs4)/c5ccccc5 7R-0334 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)NCc3cccc(c3)C(F)(F)F 7R-0335 c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)F 7R-0336 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)NCc3cccnc3 7R-0337 COCCNC(=O)c1cc(c[nH]1)C(=O)c2cccc(c2)OC 7R-0341 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)NCc3ccccc3 7R-0342 COC(=O)C1CCN(CC1)Cc2cccc(c2)F 7R-0345 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN=C(C=C3)C(F)(F)F 7R-0346 COC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)F 7R-0348 COc1ccc(cc1Cl)CN.Cl 7R-0349 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4cccc(c4)F 7R-0350 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4cc(cc(c4)C(F)(F)F)C(F)(F)F 7R-0351 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4c(cccc4Cl)F 7R-0352 Cc1ccc(cc1)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F 7R-0353 Cc1ccc(cc1)C(=O)N2CCN=C(C=C2)C(F)(F)F 7R-0354 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)NCC3CCCO3 7R-0355 c1ccc(c(c1)CO/N=C/c2cc3c(cc2Br)OCO3)F 7R-0356 CN1C(=O)C(=Cc2cc3c(cc2Br)OCO3)C(=O)N(C1=O)C 7R-0357 c1c(c(cc2c1OCO2)Br)C=C3C(=O)NC(=O)NC3=O 7R-0358 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4ccc(cc4)C(F)(F)F 7R-0359 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)NCc3cccs3 7R-0360 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4cccc(c4)Cl 7R-0361 c1cc(cc(c1)F)CN2CCC(CC2)C(=O)NN 7R-0362 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F 7R-0363 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN=C(C=C3)C(F)(F)F 7R-0364 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)NCCCN3CCOCC3 7R-0365 Cc1ccccc1CSc2[nH]c(=O)cc(n2)C(C)(C)C 7R-0366 c1cc(cc(c1)F)CN2CCC(CC2)C(=O)NNC(=O)C3CC3 7R-0367 c1cc(cc(c1)F)CN2CCC(CC2)C(=O)NNC(=O)c3cccs3 7R-0368 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNC(=O)C3CCN(CC3)Cc4cccc(c4)F 7R-0369 c1ccc(cc1)/C=C/CN2CCC(CC2)C(=O)NNC(=O)c3cccs3 7R-0371 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 7R-0372 COc1ccc(cc1)OC(=O)/C=C/c2cc3c(cc2Br)OCO3 7R-0373 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 7R-0376 CN1C(=O)C(=Cc2c3ccccc3ccc2OCc4cnc(s4)Cl)C(=O)N(C1=O)C 7R-0600 c1ccc(c(c1)C(CC(=O)O)N)O 7R-0601 Cc1cc(n(n1)Cc2cnc(s2)N3CCN(CC3)C)C 7R-0602 CC(C)(C)OC(=O)COc1ccc(cc1)O 7R-0603 COc1ccc(cc1OC)C(CC(=O)O)N 7R-0605 c1cc2c(cc1C(CC(=O)O)N)OCO2 7R-0606 c1cc(cc(c1)F)C(CC(=O)O)N 7R-0608 c1cc(cc(c1)Br)C(CC(=O)O)N 7R-0609 COc1ccc(cc1OC)/C=C/C(=O)O 7R-0613 c1cnn(c1)Cc2cnc(s2)N3CCOCC3 7R-0614 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccs1 7R-0615 COc1ccc(cc1OC)C(CC(=O)O)N2Cc3ccccc3C2=O 7R-0616 COC(=O)CC(c1ccc(cc1)Br)N 7R-0617 c1ccc(c(c1)C(CC(=O)O)N)Br 7R-0619 c1cc(c(cc1C(CC(=O)O)N)Cl)Cl 7R-0620 c1ccc(cc1)CN2CCN(CC2)c3ncc(s3)Cn4cccn4 7R-0621 c1c(sc(n1)Cl)C#N 7R-0622 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1)Br 7R-0623 COc1ccc(cc1)C(CC(=O)O)N 7R-0624 CC(C)c1ccc(cc1)C(CC(=O)O)N 7R-0625 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1)F 7R-0626 CCOc1ccc(cc1)C(CC(=O)O)NC(=O)OC(C)(C)C 7R-0627 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(c(c1)OC)OC 7R-0628 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3cccs3 7R-0629 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc4c(c3)OCO4 7R-0630 CC(C)c1ccc(cc1)C(CC(=O)O)N2Cc3ccccc3C2=O 7R-0631 COc1cccc(c1)C(CC(=O)O)N 7R-0632 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc(c1)F 7R-0633 COC(=O)CC(c1cccs1)N 7R-0635 CC(C)(C)C(=O)n1cc(c2c1cccc2)CCN3CCS(=O)(=O)CC3 7R-0637 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(c(c1)Cl)Cl 7R-0639 CC(C)c1ccc(cc1)C(CC(=O)O)NC(=O)OC(C)(C)C 7R-0640 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(cc3)Br 7R-0641 CN1CCN(CC1)c2ncc(s2)CN3CCN(CC3)c4ccccc4 7R-0642 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc3c(c2)nccn3 7R-0643 c1cc(oc1)C(=O)Nc2ccc3c(c2)nccn3 7R-0644 c1ccc(cc1)CC(=O)Nc2ccc3c(c2)nccn3 7R-0645 c1cc(ccc1F)S(=O)(=O)Nc2ccc3c(c2)nccn3 7R-0646 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc(c1)Cl 7R-0648 c1cc2c(cc1NC(=S)Nc3ccc(cc3F)Br)nccn2 7R-0649 Cc1ccsc1/C=C/C(=O)O 7R-0651 Cc1ccccc1C(CC(=O)O)N 7R-0653 Cc1cccc(c1)C(CC(=O)O)N 7R-0654 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccccc1Cl 7R-0655 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3ccc4c(c3)OCO4 7R-0800 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)CC(c3ccccc3[N+](=O)[O-])O 7R-0801 COC(=O)c1cn(c(=O)c2c1cccc2)CCc3c[nH]c4c3cccc4 7R-0802 CC(=O)c1cccc(c1)NC(=O)C(C)(C)CCl 7R-0803 CC(=O)c1cccc(c1)N2CC(C2=O)(C)C 7R-0804 CC1(CN(C1=O)c2cccc(c2)C(=O)/C=C/N(C)C)C 7R-0805 Cc1c(sc(n1)c2cccs2)C(=O)C 7R-0806 c1cc(ccc1c2ccnc(n2)NCCCC(C(=O)O)N)F 7R-0807 Cc1c(cccc1[N+](=O)[O-])/N=C/c2ccc(cc2)N(C)C 7R-0809 c1cc(nnc1n2c(c(cn2)n3cncn3)O)Cl 7R-0810 c1ccc(cc1)CCNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 7R-0811 Cc1c(sc(n1)c2cc[n+](cc2)C)C(=O)C.[I-] 7R-0812 Cc1c(sc(n1)c2cccs2)C(=O)/C=C/N(C)C 7R-0813 c1cc(cc(c1)Cl)n2c(c(cn2)n3cncn3)O 7R-0814 COc1ccc(cc1OC)CCn2ccc(c(c2=O)CC(=O)OC)O 7R-0815 CC1=C(CC(=O)N1CCc2ccc(c(c2)OC)OC)C(=O)OC 7R-0816 CC1=C(/C(=C/N(C)C)/C(=O)N1CCc2ccc(c(c2)OC)OC)C(=O)OC 7R-0818 COc1ccc(cc1OC)CCNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 7R-0819 CC(=O)c1cnc(s1)c2ccncc2 7R-0820 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)C#N)N)CSc3ccccc3 7R-0821 COc1ccc(cc1OC)CCn2ccc(c(c2=O)Cc3ccc(cc3Cl)Cl)O 7R-0824 COC(=O)c1c(ccs1)n2cc(nn2)C(=O)c3ccc(cc3)c4ccccc4 7R-0825 CN(C)/C=C/C(=O)c1cnc(s1)c2cccnc2 7R-0826 Cc1c(sc(n1)c2cccs2)c3ccnc(n3)N 7R-0827 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)OC)C#N)N)CSc3ccccc3 7R-0829 Cc1c(sc(n1)c2ccncc2)c3ccnc(n3)NC 7R-0830 Cc1ccc(cc1)c2nc(c(s2)C(=O)C)C 7R-0832 Cc1c(sc(n1)c2ccc(cc2Cl)Cl)C(=O)C 7R-0833 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/c3cccnc3 7R-0834 c1ccc(cc1)n2c(=O)ccc(n2)OCC(=O)N3CCOCC3 7R-1002 CNC(=O)COc1ccc(=O)n(n1)c2ccccc2 7R-1003 c1ccc(cc1)n2c(=O)ccc(n2)OCC(=O)NC3CC3 7R-1004 c1cc(c(cc1[N+](=O)[O-])F)N2CCNCC2 7R-1005 Cc1ccc2c(c1)C(CCS2)(c3ccccc3)O 7R-1006 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cc3F)[N+](=O)[O-])Cl 7R-1008 CC1CN(CC(O1)C)C(=O)COc2ccc(=O)n(n2)c3ccccc3 7R-1009 C=CCNC(=O)COc1ccc(=O)n(n1)c2ccccc2 7R-1010 c1ccc(cc1)n2c(=O)ccc(n2)OCC(=O)N3CCCCCC3 7R-1011 CN(C)C(=O)COc1ccc(=O)n(n1)c2ccccc2 7R-1012 c1cc(cc(c1)Cl)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 7R-1014 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 7R-1015 c1cc(ccc1NC(=O)CN2CCOCC2)N3CCOCC3 7R-1017 c1cc(ccc1NC(=O)CN2CCCCC2)N3CCOCC3 7R-1018 CC(=O)Nc1ccc(c(c1)F)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 7R-1019 CC(C)CC(=O)Nc1ccc(c(c1)F)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 7R-1020 CCCCC(=O)Nc1ccc(c(c1)F)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 7R-1021 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cc3F)NC(=O)C4CC4)Cl 7R-1023 c1cc(ccc1NC(=O)CN2CCC(CC2)(C(=O)N)N3CCCCC3)N4CCOCC4 7R-1024 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3F)[N+](=O)[O-] 7R-1025 CS(=O)(=O)N1CCN(CC1)c2ccc(cc2F)[N+](=O)[O-] 7R-1026 CS(=O)(=O)N1CCN(CC1)c2ccc(cc2F)N 7R-1030 c1ccc2c(c1)c(c[nH]2)C(C(F)(F)Cl)O 7R-1060 Cn1cc(c2c1cccc2)C(C(F)(F)F)O 7R-1061 Cn1cc(c2c1cccc2)C(C(F)(F)F)OC(=O)c3cccs3 7R-1063 Cn1cc(c2c1cccc2)C(C(F)(F)F)OC(=O)C3CC3 7R-1065 C1CN(CCC12OCCO2)C[C@H](C(F)(F)F)O 7R-1066 COC(=O)c1ccccc1SC[C@H](C(F)(F)F)O 7R-1067 c1ccc(c(c1)N)SC[C@@H](C(F)(F)F)O 7R-1068 Cn1cc(c2c1cccc2)C(=O)C(F)(F)Cl 7R-1069 Cn1cc(c2c1cccc2)C(C(F)(F)Cl)O 7R-1073 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OCc4ccc(cc4Cl)Cl 7R-1120 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OCc4ccc(c(c4)Cl)Cl 7R-1121 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OCc4ccc(cc4)F 7R-1122 Cc1ccc(cc1)C(=O)O/N=C/c2cc3ccccc3nc2SCc4ccc(cc4)Cl 7R-1123 Cc1cccc(c1)C(=O)O/N=C/c2cc3ccccc3nc2SCc4ccc(cc4)Cl 7R-1124 COC(=O)CSc1c(cc2ccccc2n1)C=O 7R-1125 c1ccc2c(c1)cc(c(n2)SCCCF)C=O 7R-1126 CCOC(=O)c1cnc(nc1Sc2ccccc2NC(=O)c3ccc(cc3)F)SC 7R-1127 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NN 7R-1128 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OCc4c(cccc4Cl)Cl 7R-1129 c1ccc2c(c1)cc(c(n2)SCc3ccc(cc3)Cl)/C=N/OCc4c(cccc4Cl)F 7R-1130 c1ccc2c(c1)cc3cc(sc3n2)C(=O)O 7R-1131 Cc1ccc(cc1)C(=O)NNC(=O)c2cc3cc4ccccc4nc3s2 7R-1133 c1ccc2c(c1)cc3cc(sc3n2)C(=O)N4CCOCC4 7R-1134 CC(C)NC(=O)c1cc2cc3ccccc3nc2s1 7R-1135 c1ccc(cc1)c2cc(n(n2)c3ccccc3)c4ccccc4 7R-1136 c1ccc2c(c1)cc3cc(sc3n2)C(=O)N4CCCC4 7R-1137 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NC4CC4 7R-1138 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NC4CCCCC4 7R-1139 COc1ccc(cc1)NC(=O)c2cc3cc4ccccc4nc3s2 7R-1141 CC(C)c1ccc(cc1)NC(=O)c2cc3cc4ccccc4nc3s2 7R-1142 c1ccc2c(c1)cc3cc(sc3n2)C(=O)Nc4cccc(c4)C(F)(F)F 7R-1143 c1ccc2c(c1)cc3cc(sc3n2)C(=O)Nc4ccc(cc4)F 7R-1144 c1ccc2c(c1)cc3cc(sc3n2)C(=O)N4CCCCC4 7R-1146 c1ccc2c(c1)cc3cc(sc3n2)C(=O)N4CCc5ccccc5C4 7R-1147 CC(C)C(C)NC(=O)c1cc2cc3ccccc3nc2s1 7R-1148 COCCNC(=O)c1cc2cc3ccccc3nc2s1 7R-1149 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc3cc4ccccc4nc3s2 7R-1150 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NNC(=O)C4CC4 7R-1151 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NNC(=O)c4cccc(c4)Cl 7R-1152 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NNC(=O)c4cccc(c4)C(F)(F)F 7R-1153 Cn1c(c(c(n1)C(F)(F)F)/C=C(\C#N)/c2ccc(c(c2)Cl)Cl)Cl 7R-1157 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NNC(=O)c4ccc(cc4)F 7R-1158 Cc1cccc(c1)C(=O)NNC(=O)c2cc3cc4ccccc4nc3s2 7R-1160 Cc1ccc(cc1)c2nnc(o2)c3cc4cc5ccccc5nc4s3 7R-1161 c1ccc(cc1)S(=O)(=O)NNC(=O)c2cc3cc4ccccc4nc3s2 7R-1162 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NNS(=O)(=O)c4ccc(cc4)F 7R-1163 Cn1c(c(c(n1)C(F)(F)F)/C=C(\C#N)/c2ccc(c(c2)OC)OC)Cl 7R-1164 Cc1cccc(c1)c2nnc(o2)c3cc4cc5ccccc5nc4s3 7R-1168 Cn1c(c(c(n1)C(F)(F)F)/C=N/c2ccc(cc2)OC)Cl 7R-1169 CS(=O)(=O)NNC(=O)c1cc2cc3ccccc3nc2s1 7R-1171 COc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc3cc4ccccc4nc3s2 7R-1172 c1ccc2c(c1)cc3cc(sc3n2)C(=O)NNS(=O)(=O)c4ccc(cc4)Cl 7R-1173 Cn1c(c(c(n1)C(F)(F)F)CNc2ccc(cc2)OC)Cl 7R-1174 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)[N+](=O)[O-] 7R-1182 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)N 7R-1183 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)c4ccc(cc4)Cl 7R-1184 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 7R-1185 C[NH+]1CCN(CC1)c2ccc(cc2F)NC(=O)c3ccc(cc3)Cl.[Cl-] 7R-1186 Cc1cccc(c1)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)C 7R-1190 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)c4ccc(cc4)F 7R-1193 Cc1cccc(c1)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 7R-1194 COc1ccc(cc1)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 7R-1195 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)C4CC4 7R-1196 c1ccc(cc1)CC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 7R-1197 c1cc(c(cc1N)F)N2CCOCC2 7R-1199 COc1ccc(cc1)C(=O)Nc2ccc(c(c2)F)N3CCOCC3 7R-1200 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)F)N3CCOCC3 7R-1201 c1cc(cc(c1)Cl)C(=O)Nc2ccc(c(c2)F)N3CCOCC3 7R-1202 CN1CCN(CC1)c2ccc(cc2F)NC(=O)C3CC3 7R-1203 CC(C)C(=O)Nc1ccc(c(c1)F)N2CCN(CC2)C 7R-1205 CCCCC(=O)Nc1ccc(c(c1)F)N2CCOCC2 7R-1209 c1cc(sc1)C(=O)Nc2ccc(c(c2)F)N3CCOCC3 7R-1212 c1cc(c(cc1NC(=O)C2CC2)F)N3CCOCC3 7R-1213 C=CCn1c(nnc1SCc2ccc(cc2)F)/C=C/c3ccccc3 7R-1240 c1ccc(cc1)S(=O)(=O)CC(COc2ccccc2C#N)O 7R-1244 CCn1c(nnc1SCc2cccc(c2)[N+](=O)[O-])/C=C/c3ccccc3 7R-1245 c1ccc(c(c1)C#N)OCC(CS(=O)(=O)c2ccc(cc2)Cl)O 7R-1246 Cc1ccc(cc1)S(=O)(=O)CC(COc2ccccc2C#N)O 7R-1247 c1cc(ccc1C#N)OCC2CO2 7R-1251 c1cc(ccc1S(=O)(=O)CC(COc2ccc(cc2Cl)F)O)Cl 7R-1253 c1cc(ccc1C#N)OCC(CS(=O)(=O)c2ccc(cc2)Cl)O 7R-1254 c1ccc(c(c1)OCC(CS(=O)(=O)c2ccc(cc2)Cl)O)Cl 7R-1257 c1ccc(cc1)S(=O)(=O)CC(COc2ccc(cc2)C#N)O 7R-1261 Cc1ccc(cc1)S(=O)(=O)CC(COc2ccc(cc2)C#N)O 7R-1262 COc1ccccc1S(=O)(=O)CC(COc2ccc(cc2)C#N)O 7R-1263 Cc1ccc(c(c1)C)S(=O)(=O)CC(COc2ccc(cc2)C#N)O 7R-1264 c1cc(ccc1C#N)OCC(CS(=O)(=O)c2ccc(cc2)F)O 7R-1265 c1cc(ccc1F)S(=O)(=O)CC(COc2ccc(cc2Cl)F)O 7R-1266 Cc1ccc(cc1)S(=O)(=O)CC(COc2ccc(cc2Cl)F)O 7R-1267 Cc1ccc(c(c1)C)S(=O)(=O)CC(COc2ccc(cc2Cl)F)O 7R-1269 COc1ccccc1S(=O)(=O)CC(COc2ccc(cc2Cl)F)O 7R-1270 c1ccc(cc1)S(=O)(=O)CC(COc2ccccc2Cl)O 7R-1271 COc1ccccc1S(=O)(=O)CC(COc2ccccc2Cl)O 7R-1273 c1ccc(c(c1)OCC(CS(=O)(=O)c2ccc(cc2)F)O)Cl 7R-1275 CC(=O)N1C(CC(=NOC(=O)c2ccccc2)CC1(C)C)(C)C 7R-1300 CC(=O)N1C(CC(=NOC(=O)c2ccc(cc2)F)CC1(C)C)(C)C 7R-1301 CC(=O)N1C(CC(=NOC(=O)c2ccc(cc2)OC)CC1(C)C)(C)C 7R-1302 CC(=O)N1C(CC(=NOC(=O)c2cccs2)CC1(C)C)(C)C 7R-1303 CC(=O)N1C(CC(=NOC(=O)c2cccc(c2)C(F)(F)F)CC1(C)C)(C)C 7R-1305 c1ccc(cc1)c2[nH]c(=O)c3c(n2)ccs3 7R-1306 CC(=O)N1C(CC(=NOS(=O)(=O)c2ccccc2)CC1(C)C)(C)C 7R-1307 CC(=O)N1C(CC(=NOS(=O)(=O)c2ccc(cc2)OC)CC1(C)C)(C)C 7R-1308 CC(=O)N1C(CC(=NOS(=O)(=O)c2ccc(cc2)Cl)CC1(C)C)(C)C 7R-1309 c1ccc(cc1)c2nc3ccsc3c(n2)Cl 7R-1316 c1ccc(cc1)c2nc3ccsc3c(=O)o2 7R-1320 c1ccc(cc1)c2nc3ccsc3c(n2)O 7R-1324 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)N3CCOCC3 7R-1325 c1ccc(cc1)c2nc3ccsc3c(n2)N4CCOCC4 7R-1327 COC(=O)c1c(ccs1)NC(=O)c2ccc(cc2)F 7R-1329 Cc1ccc(cc1)C(=O)Nc2ccsc2C(=O)OC 7R-1330 COC(=O)c1c(ccs1)NC(=O)c2ccccc2Cl 7R-1331 Cc1ccc(cc1)C(=O)Nc2ccsc2C(=O)O 7R-1333 c1ccc(c(c1)C(=O)Nc2ccsc2C(=O)O)Cl 7R-1334 c1cc(ccc1c2nc3ccsc3c(=O)o2)F 7R-1337 Cc1ccc(cc1)c2nc3ccsc3c(=O)o2 7R-1338 c1ccc(c(c1)c2nc3ccsc3c(=O)o2)Cl 7R-1339 CC(C(=O)Nc1ccc(cn1)Cl)n2c3ccccc3nc2C(F)(F)F 7R-1360 Cc1cc(nc(c1)NC(=O)C(C)n2c3ccccc3nc2C(F)(F)F)C 7R-1361 CC(C(=O)Nc1ncccn1)n2c3ccccc3nc2C(F)(F)F 7R-1362 CC(C(=O)NC(C)(C)C)n1c2ccccc2nc1C(F)(F)F 7R-1363 CC(C(=O)Nc1ccccc1C(=O)OC)n2c3ccccc3nc2C(F)(F)F 7R-1365 Cc1cc(n(n1)c2ccc(cc2)[N+](=O)[O-])O 7R-1366 CC(C(=O)NCc1cccnc1)n2c3ccccc3nc2C(F)(F)F 7R-1367 CC(C(=O)NCc1ccncc1)n2c3ccccc3nc2C(F)(F)F 7R-1368 CC(C(=O)Nc1cccc(c1)C(F)(F)F)n2c3ccccc3nc2C(F)(F)F 7R-1371 CC(C(=O)Nc1ccc(cc1F)F)n2c3ccccc3nc2C(F)(F)F 7R-1372 CC(C(=O)Nc1ccccc1C(=O)O)n2c3ccccc3nc2C(F)(F)F 7R-1373 c1ccc2c(c1)nc(n2CCO)C(F)(F)F 7R-1374 COC(=O)c1c(=O)ccn(n1)c2ccc(cc2)Cl 7R-1423 c1cc(ccc1C#N)Oc2cnns2 7R-1502 Cn1c2c(cn1)c(c(cn2)CO)NCc3ccc(cc3)OC 7T-0001 c1ccnc(c1)c2nccc(n2)c3ccco3 7T-0002 c1ccc2c(c1)cc(s2)c3ccnc(n3)c4ccccn4 7T-0003 c1ccc2c(c1)ccc3c2cc(o3)c4ccnc(n4)N 7T-0004 COc1ccc(cc1)NC(=O)Nc2cccc(c2)c3cnc4ccccc4n3 7T-0007 CNC(=S)Nc1cccc(c1)c2cnc3ccccc3n2 7T-0009 COc1cccc2c1oc(c2)c3ccnc(n3)c4ccncc4 7T-0010 c1ccc2c(c1)ccc3c2cc(o3)c4ccn[nH]4 7T-0011 c1cc(sc1)c2ccn3cnnc3n2 7T-0012 c1ccc2c(c1)ncc(n2)c3cccc(c3)NC(=O)c4ccco4 7T-0013 c1ccc2c(c1)ncc(n2)c3cccc(c3)NS(=O)(=O)c4cccs4 7T-0014 c1ccc2c(c1)ncc(n2)c3cccc(c3)NC(=O)C4CC4 7T-0015 c1cc(n(c1)Cc2cnc(s2)Cl)C=C(C#N)C#N 7T-0016 c1ccc2c(c1)c(cn2Cc3cnc(s3)Cl)/C=N/NC(=S)N 7T-0019 CC1(OC(=O)C(=Cc2cn(c3c2cccc3)Cc4cnc(s4)Cl)C(=O)O1)C 7T-0020 CN1C(=O)C(=Cc2cn(c3c2cccc3)Cc4cnc(s4)Cl)C(=O)N(C1=O)C 7T-0021 CS(=O)(=O)Nc1cccc(c1)c2cnc3ccccc3n2 7T-0022 Cc1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccc(cc4)n5cccc5 7T-0023 COc1cccc2c1oc(c2)c3ccnc(n3)S 7T-0024 CC(C)C(CC(=O)O)N 7T-0026 c1cc(n(c1)Cc2cnc(s2)Cl)/C=N/NC(=O)c3ccncc3 7T-0027 Cc1ccc(cc1)NC(=O)OC2CC(c3c2cc(c(c3)OC)OC)NC(=O)C(F)(F)F 7T-0028 c1ccc(cc1)C(=O)/C(=C/c2cccn2Cc3cnc(s3)Cl)/C#N 7T-0029 c1c2c(cc3c1OCO3)C(CC2NC(=O)C(F)(F)F)O 7T-0031 c1cc(ccc1C=C(C#N)C#N)OCc2cnc(s2)Cl 7T-0032 c1cc(n(c1)Cc2cnc(s2)Cl)C=C3C(=O)NC(=O)NC3=O 7T-0033 COc1ccccc1/C=C/C(=O)c2cccs2 7T-0034 c1cc(cc(c1)Cl)/C=C/C(=O)c2cccs2 7T-0035 c1ccc2c(c1)c(cn2Cc3cnc(s3)Cl)/C=N/Cc4ccc5c(c4)OCO5 7T-0043 COc1cc(ccc1OCc2cnc(s2)Cl)/C=C\3/C(=O)NC(=O)S3 7T-0044 c1c(sc(n1)Cl)CN2C(=O)CSC2=O 7T-0045 c1ccc2c(c1)c(cn2Cc3cnc(s3)Cl)/C=C/4\c5ccccc5NC4=O 7T-0049 COC(=O)C(c1ccc(cc1)[N+](=O)[O-])C(=O)OC 7T-0054 c1cc(n(c1)Cc2cnc(s2)Cl)/C=N/O 7T-0058 Cc1cc(nc2c1c(nn2C)NC(=O)c3cccs3)C 7T-0059 c1cc(oc1)c2ccnc(n2)c3ccncc3 7T-0061 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cccc(c3)c4cnc5ccccc5n4 7T-0066 C1(C(=O)NC(=O)S1)Br 7T-0067 c1cc(cc(c1)NC(=N)NCc2ccc(cc2)Cl)C(F)(F)F 7T-0069 CC(c1ccc(cc1)[N+](=O)[O-])(C(=O)OC)C(=O)OC 7T-0070 c1cc(sc1)C(=O)OC2CC(c3c2cc4c(c3)OCO4)NC(=O)C(F)(F)F 7T-0072 CC(=O)c1cccc(c1)NC(=O)c2ccccc2C(=O)O 7T-0073 CC(=O)c1ccc(cc1)NC(=O)CCC(=O)O 7T-0074 c1ccc(c(c1)/C(=N/O)/N)n2cccc2 7T-0075 CN1C(=O)C(=Cc2ccc(c(c2)OC)OCc3cnc(s3)Cl)C(=O)N(C1=O)C 7T-0076 COc1cc(ccc1OCc2cnc(s2)Cl)C=C(C#N)C#N 7T-0077 c1ccc2c(c1)n3cc(nc3s2)c4ccc(c(c4)Cl)Cl 7T-0078 COc1cc(ccc1/C=C\2/c3ccccc3NC2=O)OCc4cnc(s4)Cl 7T-0079 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCCc3c[nH]cn3 7T-0080 c1ccc2c(c1)ncc(n2)c3cccc(c3)n4cccc4 7T-0084 c1ccc(cc1)N2CCN(CC2)c3ncc(s3)CN4C(=O)c5ccccc5C4=O 7T-0086 c1ccc2c(c1)ccc3c2cc(o3)c4cn5cc(ccc5n4)Cl 7T-0087 Cc1cc(nc2c1c(nn2C)NC(=O)C3CC3)C 7T-0088 Cc1cc(nc2c1c(nn2C)NS(=O)(=O)C)C 7T-0089 Cc1cc(n(c(=O)c1C#N)CC=C)C 7T-0091 CC(=O)c1ccc(cc1)N2C(=O)CCC2=O 7T-0092 CC(=O)c1cccc(c1)N2C(=O)c3ccccc3C2=O 7T-0093 CN1C(=O)CSC1=O 7T-0094 c1ccc2c(c1)ccc3c2cc(o3)c4ccnc(n4)n5cccc5 7T-0095 COc1ccccc1C2CC(=Nc3ccccc3S2)c4cccs4 7T-0097 CC(c1ccc(cc1)[N+](=O)[O-])C(=O)O 7T-0098 c1cc(sc1)C=C(C#N)C#N 7T-0099 Cn1c2c(cn1)c(c(cn2)C(=O)O)NCCn3cccc3 7T-0102 COc1ccc(cc1O)/C=C/2\C(=O)NC(=O)S2 7T-0106 CCOC(=O)c1cnc2c(c1NCCC(C(F)(F)F)O)cnn2C 7T-0108 C1CCC(CC1)C(CC(=O)O)N 7T-0112 Cc1cc(nc2c1c(nn2C)NC(=S)NC)C 7T-0113 Cc1cc(nc2c1c(nn2C)NC(=O)CCl)C 7T-0114 Cc1cc(nc2c1c(nn2C)NC(=S)NC(=O)c3ccccc3)C 7T-0115 Cc1cc(n(c(=O)c1C#N)C)C 7T-0120 CS(=O)(=O)N1C(=O)CSC1=O 7T-0121 CC(C)(C)c1ccc(cc1)N/C=C\2/C(=O)N(C(=O)S2)C 7T-0125 Cc1cc(n(c(=O)c1C#N)Cc2cccc(c2)C(F)(F)F)C 7T-0127 CN1C(=O)/C(=C\N2CCOCC2)/SC1=O 7T-0128 CCOC(=O)c1c(n2c3ccccc3sc2n1)Br 7T-0129 Cc1ccc(n1c2c3c(cc(nc3n(n2)C)C)C)C 7T-0131 Cc1cc(nc2c1c(nn2C)NC(=O)C)C 7T-0132 Cc1ccc(cc1)CSC2=Nc3c(ccs3)C4=NC(=O)CN42 7T-0202 c1ccn(c1)c2cc(c(cc2F)Cl)O 7T-0203 CC(=O)c1ccc(cc1)NC(=O)Oc2ccccc2 7T-0204 c1c(c(cc(c1Cl)Cl)[N+](=O)[O-])CC(=O)O 7T-0205 CC(=O)c1ccc(cc1)NC(=O)N2CCc3ccccc3C2 7T-0206 c1cc(ccc1COc2cc(c(cc2Cl)F)[N+](=O)[O-])F 7T-0212 c1ccc(cc1)OC(=O)Nc2ccc3c(c2)OCO3 7T-0217 COc1cc(c(cc1OC)NC(=S)Nc2ccc3c(c2)OCO3)C#N 7T-0218 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)Oc2ccccc2 7T-0219 CCNc1[nH]c2ccccc2n1 7T-0223 CC(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 7T-0224 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)Oc3ccccc3 7T-0225 c1ccnc(c1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCO4 7T-0226 c1ccc(cc1)CN2CCN(CC2)C(=O)Nc3ccc4c(c3)OCO4 7T-0227 c1ccc(cc1)CN(Cc2ccccc2)C(=O)Nc3ccc4c(c3)OCO4 7T-0228 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCO4 7T-0229 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCOCC2 7T-0230 c1cnc(cn1)/C(=N\OC(=O)CCl)/N 7T-0231 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3Cl 7T-0232 c1cc2c(cc1NC(=O)NCCCn3ccnc3)OCO2 7T-0234 Cc1ccc(c(n1)C(C(F)(F)F)O)O 7T-0235 CN(C)/C=C/C(=O)C1CC1 7T-0237 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)N3CCc4ccccc4C3 7T-0238 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)N3CCc4c3cccc4 7T-0239 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N(C)C2CCCCC2 7T-0240 COc1cc(c(cc1Cl)F)[N+](=O)[O-] 7T-0245 c1ccc(c(c1)c2ccnc3n2c4ccccc4n3)OCc5ccc(cc5)Cl 7T-0248 CCCCCC1CCC(CC1)c2ccc(cc2)n3cccc3 7T-0249 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 7T-0250 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3 7T-0251 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccn3 7T-0252 CCCCCC1CCC(CC1)c2ccc(cc2)/C=C/C(=O)OC 7T-0254 CCNc1nc2ccccc2n1Cc3ccc(cc3Cl)Cl 7T-0260 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cc3)OC 7T-0261 c1cnc2ncnn2c1C3CC3 7T-0262 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCCN(CC2)C(=O)Nc3ccc(cc3)S(=O)(=O)N(C)C 7T-0264 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 7T-0265 c1cc2c(cc1NC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)OCO2 7T-0269 c1cc(cc(c1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCO4)C(F)(F)F 7T-0270 COc1ccc(cc1Cl)CNC(=O)Oc2ccccc2 7T-0271 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 7T-0272 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)N2CCN(CC2)c3cccc(c3)C(F)(F)F 7T-0273 CN(C)/C=C/c1c(c(c2c(n1)-c3ccccc3C2=O)c4ccccc4F)C#N 7T-0275 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)N3CCOCC3 7T-0277 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)N(C)C3CCCCC3 7T-0278 c1cc2c(cc1CN3CCN(CC3)C(=O)Nc4ccc5c(c4)OCO5)OCO2 7T-0279 CCNc1nc2ccccc2n1Cc3cc(ccc3C)C 7T-0284 CCNc1nc2ccccc2n1Cc3cccc(c3)C(F)(F)F 7T-0285 CCNc1nc2ccccc2n1Cc3ccc(cc3)C(C)(C)C 7T-0286 COc1ccc(cc1Cl)CNC(=O)N2CCN(CC2)c3cccc(c3)C(F)(F)F 7T-0287 COc1ccc(cc1Cl)CNC(=O)N2CCc3ccccc3C2 7T-0288 c1cc2c(cc1NC(=O)N3CCC(CC3)C(=O)O)OCO2 7T-0289 c1cc2c(cc1NC(=O)N3CCCC3C(=O)O)OCO2 7T-0290 Cn1c(=O)c2c3c(cn(n3)CCO)oc2n(c1=O)C 7T-0293 Cc1c(c(n(n1)C)OC)C=O 7T-0295 Cc1ccc2c(c1)oc3cccc(c3c2=O)NCCN 7T-0296 c1cc(ccc1COc2cc(c(cc2Cl)F)N)F 7T-0297 c1cnc2c(cnn2c1C3CC3)C#N 7T-0298 CN1C(=O)C(=C2CCCO2)C(=O)N(C1=O)C 7T-0300 Cc1ccc(cc1)NC(=O)Nc2c(c(no2)C)Cl 7T-0301 COc1ccc(cc1)N2CCN(CC2)C(=O)NCc3ccc(c(c3)Cl)OC 7T-0303 Cc1cnn2c1nccc2C3CC3 7T-0305 c1ccc(c(c1)c2ccn(n2)CCO)OCc3ccc(cc3)F 7T-0306 COc1ccc(c(c1)[N+](=O)[O-])n2cccc2 7T-0307 c1ccc(cc1)OC(=O)Nc2ccc3c(c2)NC(=O)CO3 7T-0310 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)C)C 7T-0311 COc1ccc(cc1Cl)CNC(=O)N2CCN(CC2)c3ccccc3Cl 7T-0313 COC(=O)Cc1cc(c(cc1[N+](=O)[O-])Cl)Cl 7T-0315 Cc1nnc(n1CCN2CCCCC2)c3cnn(c3N)C 7T-0316 Cc1ccc(cc1)NC(=O)CCCCCCCCCCNC(=O)C(=C)C 7T-0317 Cc1cc(cc(c1)N/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccccc5F)C#N)C 7T-0319 Cc1ccc(n1c2ccc(cc2)C(=O)O)C 7T-0322 c1ccc(cc1)N/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccccc5F)C#N 7T-0323 COc1cccc(c1)N/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccccc5F)C#N 7T-0324 C1CCc2c(c(c(s2)NC(=O)CO)C#N)C1 7T-0610 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3c(c4c(s3)CCCC4)C#N 7T-0611 CCOC(=O)c1c2c(sc1NC(=O)CN3CCN(CC3)c4ccccc4)CCCC2 7T-0612 c1cc(ccc1NC(=O)C2C(C2(C#N)C#N)c3ccc(cc3Cl)Cl)F 7T-0614 CC(C(=O)O)NCC(=O)O.Cl 7T-0622 Cc1cc(n(n1)CC(=O)C)C 7T-0800 c1ccc(cc1)S(=O)(=O)c2cnn3c2nccc3c4ccco4 7T-0802 c1ccc(cc1)S(=O)(=O)c2cnn3c2nccc3c4cccs4 7T-0803 CC(C)(C)S(=O)(=O)c1cnc2c(cnn2c1N)c3cccs3 7T-0804 c1ccc(cc1)S(=O)(=O)c2cnc3c(cnn3c2N)c4cccs4 7T-0805 Cc1c(nc2c(cnn2c1C)c3cccs3)C 7T-0806 CSc1cccc(c1)O 7T-0807 Cc1cc(n2c(n1)c(cn2)c3cccs3)C(F)(F)Cl 7T-0808 Cc1ccc(cc1)S(=O)(=O)c2cnc3cc(nn3c2N)c4cnn(c4C(F)(F)F)C 7T-0809 Cn1c(c(cn1)c2cc3ncc(c(n3n2)C(F)(F)F)C#N)C(F)(F)F 7T-0810 C/C(=N\O)/c1c(cc(cn1)C(F)(F)F)Cl 7T-0813 Cn1c(c(cn1)c2c(c3ncc(c(n3n2)C(F)(F)F)C#N)Cl)C(F)(F)F 7T-0815 COc1cc(cc(c1OC)OC)C(=O)N2CCc3cc(c(cc3C2)OC)OC 7T-0816 C/C(=N\OC)/c1c(cc(cn1)C(F)(F)F)Cl 7T-0819 Cc1c(nnn1c2ccsc2C(=O)OC)C(=O)OCc3ccccc3 7T-0821 C/C(=C\C(=O)c1c(cc(cn1)C(F)(F)F)Cl)/N(C)C 7T-0828 CC(=O)CC(=O)c1c(cc(cn1)C(F)(F)F)Cl 7T-0829 C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)Cl 7T-0830 C/C(=N/O)/c1ccc(s1)N2CCN(CC2)c3ccc(cc3)OC 7T-0832 C/C(=N\OCc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)Cl 7T-0836 C/C(=N\OCc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)Oc3cccc(c3)C(F)(F)F 7T-0837 COc1ccc(cc1)c2cnn3c2ncc(c3)c4cccc(c4)Cl 7T-0838 Cc1ccc(cc1)c2cnc3c(cnn3c2)c4ccc(cc4)F 7T-0839 Cc1ccc(cc1)S(=O)(=O)c2cnc3c(cnn3c2N)c4ccccn4 7T-0840 Cc1ccc(n1c2ccsc2c3cc4ncc(cn4n3)c5cccc(c5)Cl)C 7T-0841 COCc1cc(n2c(n1)c(cn2)c3ccsc3)O 7T-0843 Cc1cc2ncc(cn2n1)c3cccc(c3)Cl 7T-0844 Cc1c(c2ncc(cn2n1)c3cccc(c3)Cl)Cl 7T-0845 Cc1c(c2ncc(cn2n1)c3cccc(c3)Cl)Br 7T-0846 c1ccc(cc1)S(=O)(=O)c2cnn3c2nc(cc3C(F)(F)F)c4ccc(cc4)F 7T-0847 COc1ccc(cc1)CNC(=O)c2c[nH]c3c2cccc3 7T-1481 c1ccc2c(c1)c(c[nH]2)C(=O)NCc3ccc(c(c3)Cl)Cl 7T-1482 c1ccc2c(c1)c(c[nH]2)C(=O)NCc3ccc(cc3)Cl 7T-1483 CC(c1ccccc1)NC(=O)c2c[nH]c3c2cccc3 7T-1484 Cc1cccc(c1NC(=O)c2c[nH]c3c2cccc3)C 7T-1485 COc1ccccc1NC(=O)c2c[nH]c3c2cccc3 7T-1486 c1ccc2c(c1)c(c[nH]2)C(=O)N3CCCC3 7T-1487 c1ccc(cc1)N2CCN(CC2)C(=O)c3c[nH]c4c3cccc4 7T-1488 c1ccc(c(c1)CNC(=O)c2c[nH]c3c2cccc3)Cl 7T-1489 c1ccc(cc1)CN2CCN(CC2)C(=O)c3c[nH]c4c3cccc4 7T-1490 Cn1cc(c2c1cccc2)C(=O)O 7T-1500 COC(=O)c1c[nH]c2c1cccc2 7T-1502 c1ccc(cc1)CSc2ccccc2[N+](=O)[O-] 7W-0001 c1ccc(c(c1)CSc2ccccc2[N+](=O)[O-])Cl 7W-0002 c1ccc(c(c1)CSc2cc(ccc2[N+](=O)[O-])C(F)(F)F)Cl 7W-0007 c1ccc(cc1)CSc2cc(ccc2[N+](=O)[O-])C(F)(F)F 7W-0008 c1ccc(c(c1)CSc2ccc(cc2)[N+](=O)[O-])Cl 7W-0016 c1ccc(cc1)CSc2ccc(cc2)[N+](=O)[O-] 7W-0017 c1ccc(cc1)CS(=O)c2ccccc2[N+](=O)[O-] 7W-0020 CCOc1c(c(nn1C)C(F)(F)F)C#N 7W-0026 Cn1c(c(c(n1)C(F)(F)F)C#N)Oc2ccccc2 7W-0027 c1ccc(c(c1)CS(=O)c2ccccc2[N+](=O)[O-])Cl 7W-0039 c1ccc(cc1)/C=C\2/c3c(cccc3Cl)NC2=O 7W-0050 c1ccc(c(c1)CS(=O)(=O)c2cc(ccc2[N+](=O)[O-])C(F)(F)F)Cl 7W-0052 Cc1ccc(cc1)C(=O)NCc2cn(nc2c3ccc4ccccc4c3)c5ccccc5 7W-0200 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)CNC(=O)C5CCCCC5 7W-0202 COC(=O)c1cc(ccc1N2CCNCC2)[N+](=O)[O-] 7W-0206 c1cc(c(cc1S(=O)(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-])N3CCC(CC3)C(=O)O 7W-0207 c1c(c2nc(c(cn2n1)CCCO)C(F)(F)F)C#N 7W-0210 CCOC(=O)c1cnc(nc1C(F)(F)F)c2ccccn2 7W-0211 Cc1cc(cc(c1)/N=C(\C)/N(C)CCNS(=O)(=O)c2ccc(cc2)[N+](=O)[O-])C.I 7W-0213 c1cc2c(cc(=O)oc2cc1O)CCl 7W-0215 COc1ccc(cc1)CNC(=O)c2ccccc2C(=O)c3ccc4c(c3)CCC4 7W-0216 CN(Cc1ccccc1)c2ccc(cc2[N+](=O)[O-])S(=O)(=O)N3CCC(CC3)C(=O)O 7W-0218 c1ccc(cc1)n2cc(c(n2)c3ccc4ccccc4c3)CNC(=O)c5c(cccc5F)F 7W-0220 c1cc2c(cc1c3ccn(n3)CCO)CCC2 7W-0221 c1cc(oc1)/C=C\2/C(=O)N=C(S2)N3CCCC3C(=O)O 7W-0222 Cc1cc(cc(c1)/N=C(\C)/N(C)CCN(CC=C)S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])C 7W-0223 CC(C)c1ccc(cc1)/N=C(\C)/N(C)CCNS(=O)(=O)c2ccc(cc2)[N+](=O)[O-].I 7W-0224 C/C(=C\1/CCOC1=O)/Nc2ccc(cc2)OC(F)(F)F 7W-0227 c1cc(c(cc1S(=O)(=O)N2CCC(CC2)C(=O)O)[N+](=O)[O-])N3CCC(CC3)O 7W-0231 c1ccc(c(c1)C(=O)c2ccc3c(c2)CCC3)C(=O)NCc4cccc(c4)C(F)(F)F 7W-0234 Cc1ccc2c(c1)NC(=O)C(O2)CCO 7W-0235 c1cc2c(cc1[N+](=O)[O-])NC(=O)C(O2)CCO 7W-0236 c1cc(oc1)/C=C/2\C(=O)N=C(S2)N3CCCCC3CCO 7W-0237 c1cc(c(cc1S(=O)(=O)N2CCOCC2)[N+](=O)[O-])Cl 7W-0241 CCCCCC1CCC(CC1)Cc2nnc(n2C)S 7W-0242 CCOC(=O)c1cnc2c(c1NCCN3CCOCC3)c(nn2c4ccc(cc4)Cl)C 7W-0243 CCOC(=O)c1cnc2c(c1NCc3cccc(c3)C(F)(F)F)c(nn2c4ccc(cc4)Cl)C 7W-0244 Cn1c(c(c(n1)C(F)(F)F)CNC(=O)c2ccc(cc2)C(F)(F)F)N3CCOCC3 7W-0245 CCCCCC(=O)NCc1c(nn(c1N2CCOCC2)C)C(F)(F)F 7W-0246 CC(C)(CCl)C(=O)NCc1c(nn(c1N2CCOCC2)C)C(F)(F)F 7W-0247 c1ccc(c(c1)C(=O)c2ccc3c(c2)CCC3)C(=O)NCc4ccco4 7W-0251 C/C(=C\1/CCOC1=O)/Nc2ccccc2Oc3ccccc3 7W-0252 c1ccc2c(c1)c(nn(c2=O)CCN3C(=O)c4ccccc4C3=O)c5ccc6c(c5)CCC6 7W-0255 Cc1cc(cc(c1)/N=C(\C)/N(C)CCN(Cc2ccc(cc2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)[N+](=O)[O-])C 7W-0257 Cc1cc(cc(c1)/N=C(\C)/N(C)CCN(CCCF)S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])C 7W-0258 COC(=O)c1ccc2nc(cn2c1)c3ccc(cc3)F 7W-0262 Cc1cc2n(c(=O)c3ccccc3n2n1)CCc4ccccc4 7W-0264 Cc1c(c(c2cc(ccc2n1)OC(F)(F)F)Cl)CCCl 7W-0266 CN1CCN(CC1)CCC2C(=O)Nc3cc(ccc3O2)[N+](=O)[O-] 7W-0267 COc1ccccc1CNC(=O)c2ccccc2C(=O)c3ccc4c(c3)CCC4 7W-0271 c1cc(ncc1C(=O)O)N2CCCC2 7W-0272 Cn1c(c(c(n1)C(F)(F)F)CNS(=O)(=O)c2cccs2)N3CCOCC3 7W-0274 c1cc2c(cc1S(=O)(=O)N3CCOCC3)NC(=O)C4N2CCC4 7W-0276 c1cc(ccc1c2cn3cc(cc(c3n2)Cl)C(F)(F)F)F 7W-0280 CC1(CN(C1=O)Cc2c(nn(c2N3CCOCC3)C)C(F)(F)F)C 7W-0281 Cc1c2c(c3cc(ccc3n1)OC(F)(F)F)SCC2 7W-0282 CN1CCN(CC1)S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl 7W-0283 COc1ccc(cc1)c2c(n3cc(ccc3n2)C(=O)OC)Br 7W-0284 c1cc(ccc1N2CCN(CC2)CCC3C(=O)Nc4cc(ccc4O3)[N+](=O)[O-])[N+](=O)[O-] 7W-0285 CCOC(=O)c1cnc(nc1C(F)(F)F)c2ccncc2 7W-0286 c1ccc(c(c1)C(=O)c2ccc3c(c2)CCC3)C(=O)NCc4cccc(c4)Cl 7W-0288 c1ccc2c(c1)c(nnc2Cl)c3ccc4c(c3)CCC4 7W-0289 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)c3c(n2)CCCC3)CCO 7W-0294 COc1ccc(cc1)N2CCN(CC2)CCC3C(=O)Nc4cc(ccc4O3)[N+](=O)[O-] 7W-0295 c1cc2c(cc1[N+](=O)[O-])NC(=O)C(O2)CCN3CCOCC3 7W-0297 c1ccc(c(c1)/C=C/c2c3c(c4cc(ccc4n2)OC(F)(F)F)SCC3)Cl 7W-0301 c1ccc(c(c1)/C=C/c2c3c(c4cc(ccc4n2)OC(F)(F)F)SCC3)F 7W-0302 c1cc2c(cc1OC(F)(F)F)c3c(c(n2)/C=C/c4ccc(cc4Cl)Cl)CCS3 7W-0303 c1cc(ccc1/C=C/c2c3c(c4cc(ccc4n2)OC(F)(F)F)SCC3)[N+](=O)[O-] 7W-0304 COC(=O)CCc1nc2c(c(ccn2n1)c3ccc(cc3)Cl)C#N 7W-0305 c1ccc(cc1)CNC(=O)c2cnc(nc2C(F)(F)F)c3ccccc3 7W-0306 COc1ccc(cc1)c2cn3cc(ccc3n2)C(=O)O 7W-0307 c1cc(ccc1c2c(n3cc(cc(c3n2)Cl)C(F)(F)F)Br)F 7W-0308 c1ccc2c(c1)c(nn(c2=O)CCN)c3ccc4c(c3)CCC4 7W-0309 c1cc(oc1)/C=C/2\C(=O)N=C(S2)N3CCC(CC3)O 7W-0311 COc1ccc(c(c1C=O)[N+](=O)[O-])OC 7W-0313 CCOC(=O)c1cnc(nc1C(F)(F)F)C 7W-0316 c1ccnc(c1)c2ncc(c(n2)C(F)(F)F)C(=O)O 7W-0317 CC(C)(C)c1cc(n(n1)C)C(=O)O 7W-0319 CCOC(=O)c1c(c(sc1Nc2ccccc2)C=O)Cl 7W-0320 c1ccc(c(c1)NS(=O)(=O)CCN2CCOCC2)[N+](=O)[O-] 7W-0321 c1cc(sc1)/C=C/c2c3c(c4cc(ccc4n2)OC(F)(F)F)SCC3 7W-0323 c1ccc2c(c1)cccc2/C=C/c3c4c(c5cc(ccc5n3)OC(F)(F)F)SCC4 7W-0324 c1cc(ccc1/C=C/c2c3c(c4cc(ccc4n2)OC(F)(F)F)SCC3)F 7W-0325 c1cc(ccc1c2ccn3c(c2C#N)nc(n3)CCC(=O)O)Cl 7W-0326 Cc1cc(=O)n([nH]1)C(=N)N 7W-0329 c1cc(oc1)/C=C/c2c3c(c4cc(ccc4n2)OC(F)(F)F)SCC3 7W-0330 Cc1c(c(c2cccc(c2n1)Oc3ccccc3)Cl)CCCl 7W-0331 COC(=O)c1ccc2nc(c(n2c1)Br)c3ccc(cc3)F 7W-0332 CCOC(=O)C1CCN(CC1)c2ccc(cc2C(=O)OC)[N+](=O)[O-] 7W-0333 COC(=O)c1cc(ccc1N2CCN(CC2)Cc3ccccc3)[N+](=O)[O-] 7W-0334 CCOC(=O)C1CCN(CC1)c2ccc(cc2C(=O)O)[N+](=O)[O-] 7W-0335 COC(=O)c1cc(c(nc1)Cl)Br 7W-0337 c1c(c[nH]c(=O)c1Br)C(=O)O 7W-0338 COC(=O)c1cc(c(=O)[nH]c1)Br 7W-0339 CCOC(=O)c1cnc([nH]c1=O)n2c(=O)c(c([nH]2)C)CCO 7W-0341 CCOC(=O)c1cnc([nH]c1=O)n2c(=O)cc([nH]2)C 7W-0342 CCOC(=O)c1cnc2c(c1NCc3ccco3)c(nn2c4ccc(cc4)Cl)C 7W-0345 CCOc1ccccc1/C=C/c2c3c(c4cc(ccc4n2)OC(F)(F)F)SCC3 7W-0346 Cc1c2c(c3cccc(c3n1)Oc4ccccc4)SCC2 7W-0347 COc1ccc(cc1)CNc2c3ccccc3c(nn2)c4ccc5c(c4)CCC5 7W-0348 CSc1[nH]c(=O)c2ccccc2n1 7W-0349 c1cc(ccc1c2cn3cc(ccc3n2)C(=O)O)F 7W-0351 COC(=O)c1ccc2nc(cn2c1)c3cccc(c3)[N+](=O)[O-] 7W-0352 COC(=O)c1ccc2nc(cn2c1)c3ccc(cc3)Br 7W-0354 COc1cccc(c1)CNC(=O)c2cnc(nc2C(F)(F)F)c3ccccn3 7W-0355 COC(=O)c1cc(ccc1Oc2cccc(c2)C=O)[N+](=O)[O-] 7W-0357 CCOC(=O)c1cnc2c(c1NCc3ccc(cc3)OC)c(nn2c4ccc(cc4)Cl)C 7W-0360 c1ccc(cc1)Oc2cccc3c2nc(c4c3SCC4)/C=C/c5ccc(cc5)[N+](=O)[O-] 7W-0362 c1ccc(cc1)Oc2cccc3c2nc(c4c3SCC4)/C=C/c5ccc(cc5Cl)Cl 7W-0363 c1ccc(cc1)Oc2cccc3c2nc(c4c3SCC4)/C=C/c5ccccc5F 7W-0364 c1ccc(cc1)Oc2cccc3c2nc(c4c3SCC4)/C=C/c5ccc(cc5)F 7W-0365 COc1ccc(cc1)NC(=O)c2ccc(cc2)Cl 7W-0366 CCOC(=O)C1=C(SCC1=O)Nc2ccccc2C 7W-0368 Cn1c(c(c(n1)C(F)(F)F)CN)N2CCOCC2 7W-0370 Cc1cnc(nc1c2ccc(c(c2)F)OC)n3c(=O)c(c([nH]3)C)CCO 7W-0371 c1ccc(cc1)n2cc(c(n2)c3ccc4c(c3)CCC4)/C=C(\C#N)/c5cccc(c5)C(F)(F)F 7W-0378 c1ccc2c(c1)c(nnc2NCc3ccco3)c4ccc5c(c4)CCC5 7W-0379 COc1ccc(cc1)Oc2c3ccccc3c(nn2)c4ccc5c(c4)CCC5 7W-0380 CCOc1ccccc1/C=C/c2c3c(c4cccc(c4n2)Oc5ccccc5)SCC3 7W-0381 c1ccc(cc1)Oc2cccc3c2nc(c4c3SCC4)/C=C/c5ccccc5Cl 7W-0382 c1ccc(cc1)Oc2cccc3c2nc(c4c3SCC4)/C=C/c5cccs5 7W-0383 c1cc(ccc1c2cn3cc(cc(c3n2)Cl)C(F)(F)F)Br 7W-0386 c1cc(ccc1c2cn3cc(ccc3n2)C(=O)O)Br 7W-0388 c1ccc(cc1)N2CCN(CC2)CCC3C(=O)Nc4ccc(cc4O3)[N+](=O)[O-] 7W-0389 c1cc2c(cc1[N+](=O)[O-])OC(C(=O)N2)CCN3CCOCC3 7W-0390 Cc1cc(=O)[nH]c(n1)n2c(=O)c(c([nH]2)C)CCO 7W-0391 CN1CCN(CC1)CCC2C(=O)Nc3ccc(cc3O2)[N+](=O)[O-] 7W-0392 Cc1c(c(=O)n([nH]1)C(=N)N)Cc2ccccc2 7W-0394 COC(=O)c1cc(cnc1Cl)Cl 7W-0397 COC(=O)c1cc(c[nH]c1=O)Cl 7W-0398 c1c(cnc(c1C(=O)O)Cl)Cl 7W-0399 CC(C)(C)OC(=O)N1CCC(CC1)N2CC(CC2=O)C(=O)OC 7W-0612 CC(C)(C)OC(=O)N1CCC(CC1)N2CC(CC2=O)C(=O)O 7W-0625 CCCCCCC(C(=O)/C=C/N(C)C)C(=O)OC 7W-0800 CCCCCCc1c(ccn(c1=O)CCc2c[nH]c3c2cccc3)O 7W-0801 c1ccc2c(c1)NCCC(=O)N2 7W-0803 CN1CCN(CC1)c2ccc(cc2NO)C(F)(F)F 7W-0804 c1ccc(c(c1)Cn2cccc2C#N)[N+](=O)[O-] 7W-0805 CCOC(=O)c1cc([nH]n1)c2cccc(c2)N 7W-0806 CC1(Cc2c3ccccc3ncc2C(=O)C1)C 7W-0808 Cc1cc(nc(n1)n2c(c(nn2)CO)CO)C(F)(F)F 7W-0809 c1ccc2c(c1)ccc(c2C=O)OCc3cccc(c3)C(F)(F)F 7W-0811 Cc1cc(n(n1)c2nc(c(s2)C)C(=O)C)C(F)(F)F 7W-0812 c1cc(c(cc1C(F)(F)F)N)NCCC(=O)O 7W-0813 COC(=O)c1c(c2ccccc2[nH]1)Br 7W-0815 Cc1cc(n(n1)c2nc(c(s2)C)c3ccc4ccccc4n3)C(F)(F)F 7W-0816 Cc1cc(n(n1)c2nc(c(s2)C)c3ccc4cc(cc(c4n3)Br)Br)C(F)(F)F 7W-0819 Cn1c(cc(=O)n(c1=O)C)N2CCCCC2 7W-0820 c1ccc(cc1)c2c(nnc(n2)Sc3c(cc(cn3)C(F)(F)F)Cl)c4ccccc4 7W-0821 Cc1ccnc(n1)S(=O)(=O)Cc2ccc(cc2)Cl 7W-0823 c1ccn(c1)C(CC(=O)N/N=C/c2ccc3c(c2)OCO3)c4cccc(c4)Cl 7W-0824 c1ccc(cc1)c2c(nnc(n2)SCCOc3ccccc3)c4ccccc4 7W-0825 CN1CCN(CC1)c2ccc(cc2N)C(F)(F)F 7W-0827 c1cc(cc(c1)[N+](=O)[O-])C(=O)/C=C(/CO)\N 7W-0828 Cn1c(cc(=O)n(c1=O)C)N2CCOCC2 7W-0830 c1cc(c(cc1CC(=O)N2CCOCC2)Cl)Cl 7W-0831 COc1cccc(c1)NC(=O)Cc2ccccc2 7W-0834 c1cc2c(cc1C(F)(F)F)NC(=O)CCN2 7W-0837 c1cc(sc1)c2cc([nH]n2)C(F)(F)F 7W-0838 CN1CCN(CC1)c2ccc(cc2NC(=O)Nc3ccccc3)C(F)(F)F 7W-0840 COC(=O)c1ccc2c(c1)OCO2 7W-0842 c1ccc2c(c1)c(=O)c3c([nH]2)cc(cc3O)O 7W-0843 Cn1c(cc(=O)n(c1=O)C)N2CCN(CC2)Cc3ccc4c(c3)OCO4 7W-0844 CN1CCN(CC1)c2ccc(cc2NC(=O)c3ccco3)C(F)(F)F 7W-0845 COc1ccc(cc1)N2CCN(CC2)C(=O)Cc3ccc(c(c3)Cl)Cl 7W-0847 c1ccc(c(c1)Cn2cccc2C#N)N 7W-0849 CC\1(Cc2c3ccccc3ncc2C(=O)/C1=C\Nc4ccccc4)C 7W-0851 CC1=Nc2ccccc2NC(C1)(C)C 7W-0852 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2N3CCN(CC3)C)C(F)(F)F 7W-0853 CNc1nc2c(s1)CCCC2 7W-0854 Cn1c(cc(n1)c2cccs2)C(F)(F)F 7W-0855 c1nc2n(n1)c3c(s2)CCCC3 7W-0856 Cc1cc2c(cc(nc2cc1N)Cl)COC 7W-0857 COc1ccc(cc1)C2COc3ccccc3C(=O)N2C(=O)c4ccco4 7W-0858 Cc1ccc(n1c2nccs2)C 7W-0860 CN(c1nc2c(s1)CCCC2)S(=O)(=O)C 7W-0861 CN(c1nc2c(s1)CCCC2)C(=O)c3ccc(cc3)OC 7W-0862 CN(c1nc2c(s1)CCCC2)C(=O)c3ccco3 7W-0863 Cn1c(cc(=O)n(c1=O)C)N2CCN(CC2)C 7W-0864 COc1cccc(c1)C(=O)N2CCC(=O)Nc3c2cccc3 7W-0865 COc1ccc2cc(c(=O)[nH]c2c1)c3ccccc3 7W-0866 Cc1ccn2cc(nc2c1)C(=O)O 7W-0867 Cc1cc2c(cc(nc2cc1NC(=O)C(F)(F)F)N3CCN(CC3)c4ccccc4)COC 7W-0868 C1CC2=C(CCC(=O)N2)C(=O)C1 7W-0869 COC(=O)NNC(=O)Nc1ccccc1 7W-0870 c1ccc2c(c1)-c3c(cc4c(n3)CCCC4=O)C(O2)O 7W-0871 c1ccc2c(c1)NC(=O)CCN2C(=O)c3ccco3 7W-0873 CC1(CC(=O)C(=CNc2ccccc2N)C(=O)C1)C 7W-0874 c1ccc(cc1)n2c(=O)[nH][nH]c2=O 7W-0875 c1c(cc(c(c1[N+](=O)[O-])O)Cl)c2c(cc(cn2)C(F)(F)F)Cl 7W-0876 c1c(cc(c(c1[N+](=O)[O-])O)Br)c2c(cc(cn2)C(F)(F)F)Cl 7W-0877 c1c(cc(c(c1[N+](=O)[O-])O)[N+](=O)[O-])c2c(cc(cn2)C(F)(F)F)Cl 7W-0878 Cc1c(sc2n1cc(n2)c3ccc(cc3)Br)C(=O)C 7W-0879 c1cc2c(cc1C(=O)NN)OCO2 7W-0880 C=CCNC(=S)NNC(=O)c1ccc2c(c1)OCO2 7W-0881 C=CCn1c(nnc1S)c2ccc3c(c2)OCO3 7W-0882 c1ccc2c(c1)c3c([nH]2)C(=O)CCC3 7W-0883 CC1CN(CCN1Cc2ccc(cc2)F)C(=O)OC(C)(C)C 7W-1362 COc1ccc(c(c1)/C=C\2/C(=O)C3CCN2CC3)OC 7X-0016 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(=O)O 7X-0049 c1cc(cc(c1)C(F)(F)F)CN2CCC(CC2)c3cc([nH]n3)c4ccc(cc4Cl)Cl 7X-0055 c1ccc(c(c1)C(=O)O)OCc2cnc(s2)Cl 7X-0056 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)NN)S(=O)(=O)C 7X-0203 CCOC(=O)C1CN(c2cc(ccc2O1)Cl)S(=O)(=O)C 7X-0209 CCOC(=O)C1CNc2cc(ccc2O1)CC(=O)OC 7X-0210 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCN(CC4)Cc5cccc(c5)Cl 7X-0216 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCN(CC4)C(=O)CCl 7X-0217 c1ccc(cc1)/C=C/C(=O)N2CCC(CC2)c3cc([nH]n3)c4cccc5c4cccc5 7X-0218 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCN(CC4)Cc5ccccc5F 7X-0219 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)NCc3ccccc3OC)S(=O)(=O)C 7X-0220 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)NCc3cccc(c3)Cl)S(=O)(=O)C 7X-0221 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)NN3CCOCC3)S(=O)(=O)C 7X-0222 CCOC(=O)C1(C(=O)Nc2cc(ccc2O1)S(=O)(=O)CC)C 7X-0223 Cc1ccc(cc1)c2nc(on2)c3ccc(cc3)C#N 7X-0226 CS(=O)(=O)N1CC(Oc2c1cc(cc2)Cl)C(=O)O 7X-0227 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)NCCOC)S(=O)(=O)C 7X-0234 CCS(=O)(=O)c1ccc2c(c1)N(CC(O2)C(=O)NC3CC3)S(=O)(=O)C 7X-0235 CCOC(=O)C1CN(c2cc(ccc2O1)CC(=O)OC)S(=O)(=O)C 7X-0236 c1cc2c(cc1Cl)NCC(O2)C(=O)NN 7X-0240 CCS(=O)(=O)c1ccc2c(c1)NC(=O)C(O2)(C)C(=O)O 7X-0241 CCOC(=O)C1CN(c2cc(ccc2O1)CC(=O)OC)S(=O)(=O)c3ccc(cc3)OC 7X-0242 CS(=O)(=O)N1CC(Oc2c1cc(cc2)CC(=O)O)C(=O)O 7X-0247 CCOC(=O)C1CN(c2cc(ccc2O1)Cl)S(=O)(=O)c3ccc(cc3)OC 7X-0248 c1cc(c(cc1Cl)Cl)C2C3=C(C4CCN3CC4)NC(=S)N2 7X-0254 COc1ccc(cc1)S(=O)(=O)N2CC(Oc3c2cc(cc3)CC(=O)O)C(=O)O 7X-0255 CCOC(=O)C1CN(c2cc(ccc2O1)Cl)S(=O)(=O)Cc3ccccc3[N+](=O)[O-] 7X-0256 CCOC(=O)C1CN(c2cc(ccc2O1)Cl)S(=O)(=O)c3ccc(cc3)Cl 7X-0257 COC(=O)Cc1ccc2c(c1)NC(=O)C(O2)CCO 7X-0258 COc1ccc(cc1)S(=O)(=O)N2CC(Oc3c2cc(cc3)Cl)C(=O)O 7X-0265 CCOC(=O)C1CN(c2cc(ccc2O1)Cl)S(=O)(=O)c3cccc(c3)C(F)(F)F 7X-0266 CCOC(=O)C1CN(c2cc(ccc2O1)Cl)S(=O)(=O)c3ccc(cc3)C(C)(C)C 7X-0267 c1ccc(c(c1)CS(=O)(=O)N2CC(Oc3c2cc(cc3)Cl)C(=O)O)[N+](=O)[O-] 7X-0272 c1cc(ccc1S(=O)(=O)N2CC(Oc3c2cc(cc3)Cl)C(=O)O)Cl 7X-0273 CC1=C(C(C2=C(N1)C3CCN2CC3)c4ccc(cc4Cl)Cl)C#N 7X-0276 COc1ccccc1NC(=S)NNC(=O)C2CCN(CC2)Cc3ccccc3 7X-0280 CCNC(=S)NNC(=O)C1CCN(CC1)Cc2ccccc2 7X-0281 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CC(Oc3c2cc(cc3)Cl)C(=O)O 7X-0282 c1cc(cc(c1)S(=O)(=O)N2CC(Oc3c2cc(cc3)Cl)C(=O)O)C(F)(F)F 7X-0283 COC(=O)Cc1ccc2c(c1)NC(=O)C(O2)CCCl 7X-0284 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4cccc(c4)C(F)(F)F 7X-0290 Cc1c(n(c(c1S(=O)(=O)C)N)Cc2ccccc2)C 7X-0291 c1cc(c(cc1Cl)Cl)C2C(C(=S)NC3=C2N4CCC3CC4)C#N 7X-0293 Cc1c(c(=O)nc2n1CCS2)CCO 7X-0301 CCn1c(nnc1S)C2CCN(CC2)Cc3ccccc3 7X-0305 CCOC(=O)C1CN(c2cc(ccc2O1)CC(=O)OC)S(=O)(=O)c3cccc(c3)C(F)(F)F 7X-0306 c1cc(cc(c1)F)CN2CCC(CC2)c3cc([nH]n3)c4cccc(c4)C(F)(F)F 7X-0307 CCOC(=O)C1CN(c2ccc(cc2O1)CC(=O)OC)S(=O)(=O)c3cccs3 7X-0310 CS(=O)(=O)N1CC(Oc2c1cc(cc2)Cl)C(=O)NN 7X-0311 C=CCOc1ccc2ccccc2c1C=C(C#N)C#N 7X-0312 COc1ccccc1n2c(nnc2S)C3CCN(CC3)Cc4ccccc4 7X-0313 C=CCOc1ccc2ccccc2c1/C=C(\C#N)/C(=S)N 7X-0314 COc1cc(cc(c1OC)OC)/C=N/NC(=O)C2CN(c3cc(ccc3O2)Cl)S(=O)(=O)C 7X-0324 CS(=O)(=O)N1CC(Oc2c1cc(cc2)Cl)C(=O)N/N=C/c3ccc(cc3)[N+](=O)[O-] 7X-0325 c1cc(cc(c1)C(F)(F)F)c2cc(n[nH]2)C3CCN(CC3)C(=O)c4ccc(c(c4)Cl)Cl 7X-0332 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4ccc5c(c4)OCO5 7X-0341 c1cc(ccc1S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4ccc5c(c4)OCO5)I 7X-0344 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4ccc5c(c4)OCO5 7X-0345 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4ccc5c(c4)OCO5 7X-0346 C=CCOc1ccc2ccccc2c1/C=N/OCc3c(cccc3Cl)Cl 7X-0351 c1cc(sc1)S(=O)(=O)N2CC(Oc3c2cc(cc3)CC(=O)O)C(=O)O 7X-0352 c1cc(cc(c1)S(=O)(=O)N2CC(Oc3c2cc(cc3)CC(=O)O)C(=O)O)C(F)(F)F 7X-0353 CS(=O)(=O)N1CC(Oc2c1cc(cc2)Cl)c3nnc(o3)c4ccc(cc4)Cl 7X-0354 Cn1cccc1C(=O)OC 7X-0419 Cn1cc(cc1C(=O)OC)C=O 7X-0420 Cc1c(nc(nc1O)N)C 7X-0601 CC(=O)c1ccc(c(c1)N)N2CCOCC2 7X-0700 c1cc(ccc1C(=O)N2CCOCC2)[N+](=O)[O-] 7X-0701 CC(=O)c1ccc(c(c1)N)N2CCCCC2 7X-0702 c1cc(ccc1C(=O)N2CCOCC2)N 7X-0704 c1cocc1C(=O)Cl 7X-0706 COC(=O)c1cc2cc(ccc2s1)Br 7X-0709 COC(=O)Cc1csc(n1)N 7X-0710 C#CCOc1ccc2ccccc2c1C=O 7X-0711 CCOC(=O)COc1ccc2ccccc2c1C=O 7X-0712 COC(=O)C(c1ccc(cc1)Br)N.Cl 7X-0715 c1ccc(cc1)Cn2cc(cc(c2=O)C(=O)O)Br 7X-0716 c1cc(cc(c1)F)Cn2cc(cc(c2=O)C(=O)O)Br 7X-0719 c1cc(oc1)CNCC(C(F)(F)F)O 7X-0800 Cc1cccc(c1N2CCN(CC2)CC(C(F)(F)F)O)C 7X-0801 CCOC(=O)N1CCN(CC1)CC(C(F)(F)F)O 7X-0802 c1ccc2c(c1)c(c[nH]2)CCNCC(C(F)(F)F)O 7X-0803 c1cc(c(nc1)N)OCc2ccc(cc2)Br 7X-0805 c1ccc(cc1)c2cc(n(n2)c3nc(cs3)c4ccc(cc4)F)c5ccccc5 7X-0806 c1ccc(cc1)OCC(CN2CCN(CC2)c3ncccn3)O 7X-0807 c1ccc(cc1)OCC(CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])O 7X-0808 c1cc2nc(cn2cc1Cl)CC(=O)O 7X-0811 c1cc(cc2c1cc(c(=O)o2)C(=O)O)O 7X-0812 c1cc(cc(c1)C(F)(F)F)COc2cccnc2N 7X-0814 c1ccc(cc1)c2c(nnc(n2)O)c3ccccc3 7X-0815 Cc1cc(n(n1)C(=O)c2ccc(c(c2)OC)O)C 7X-0816 c1cn(cn1)CCCNCC(C(F)(F)F)O 7X-0819 C1COCCN1NCC(C(F)(F)F)O 7X-0820 COC(=O)c1cc2ccc(cc2oc1=O)O 7X-0821 Cc1cc(n(n1)Cc2ccc(cc2)C(=O)OC)C 7X-0822 COC(=O)/C(=C\Nc1ccc(c(c1F)F)F)/c2c(cc(cn2)C(F)(F)F)Cl 7X-0824 c1c(cnc(c1Cl)c2c[nH]c3c(c2=O)cc(c(c3F)F)F)C(F)(F)F 7X-0825 c1cc(oc1)c2ccc(cn2)C(=O)c3ccco3 7X-0827 COc1ccc(cc1OC)CNC(=O)Cn2cncn2 7X-0828 CC1=C(/C(=C/c2ccc3c(c2)OCO3)/C(=O)N1CCc4c[nH]c5c4cc(cc5)OC)C(=O)OC 7X-0829 Cc1cc(n(n1)C(=O)C)C 7X-0830 Cc1cccn2c1ncc2 7X-0831 C1CC(OC1)CNCC(C(F)(F)F)O 7X-0833 c1cc2c(cc1CN3CCN(CC3)CC(C(F)(F)F)O)OCO2 7X-0834 c1ccc(cc1)CC2CCN(CC2)CC(C(F)(F)F)O 7X-0835 c1c(c(cc(c1Br)F)F)[N+](=O)[O-] 7X-0836 c1ccc(c(c1)c2cn3cc(ccc3n2)Cl)C(=O)O 7X-0837 Cc1c(n2cc(ccc2n1)Cl)C(=O)/C=C/N(C)C 7X-0839 CC(C(=O)O)Oc1ccc2cc(ccc2c1)Br 7X-0841 CC(CCC(=O)O)(c1ccc(c(c1)[N+](=O)[O-])O)c2ccc(c(c2)[N+](=O)[O-])O 7X-0843 Cc1cc(cnc1N)Br 7X-0844 Cc1cccn2c1ncc2Br 7X-0845 c1ccc2cc3c(cc2c1)OC(O3)C(=O)O 7X-0849 c1ccc2c(c1)c3cccc(c3s2)C(=O)O 7X-0850 c1ccc(cc1)NC(=S)NCC(=O)O 7X-0851 C1CCC(CC1)NC(=O)/C=C/C(=O)O 7X-0852 CN1CCN(CC1)c2cc(c(cc2[N+](=O)[O-])Br)F 7X-0853 COc1ccc(cc1OC)n2cccc2C=O 7X-0856 COC(=O)c1ccc2nccn2c1 7X-0857 c1ccc(cc1)OCC(CNCc2cc(cc(c2)F)F)O 7X-0858 c1ccc(cc1)CCCNC(=O)Cn2cncn2 7X-0859 CN1CCN(CC1)c2ccc(cc2)C(=O)c3cn(nn3)c4ccc(c(c4)Cl)F 7X-0860 Cc1ccc2ncc(n2c1)Br 7X-0861 Cc1ccc2ncc(n2c1)[N+](=O)[O-] 7X-0862 c1ccc(c(c1)C(CCO)N2CCS(=O)(=O)CC2)F 7X-0863 Cc1cc(n2c(n1)nc(n2)SCC(=O)N(C)c3ccccc3)C 7X-0864 CCOC(=O)[C@H](CC(C)C)NS(=O)(=O)c1ccc(cc1)CBr 7X-0866 c1cc2nccn2cc1C(=O)O 7X-0867 c1cc2nccn2cc1C(=O)NN 7X-0868 Cc1ccn2cc(nc2c1)CC(=O)O 7X-0869 c1ccc2c(c1)ccc(c2CC(=O)O)O 7X-0870 CC(=O)Nc1cc(ccc1C#N)N 7X-0871 c1cc(cnc1)CNc2nc[nH]n2 7X-0872 CC1(C(=S)NC(N1)(C)C)C 7X-0873 COc1ccc(cc1OC)n2cccc2 7X-0874 Cc1cc(cn2c1ncc2)Br 7X-0875 CCOC(=O)c1c(n(nn1)c2nc(cc(n2)C(F)(F)F)C)C(=O)OCC 7X-0877 c1cc(c(cc1n2cc(nn2)C(=O)C3CC3)Cl)Cl 7X-0878 c1cc(ccc1c2ccc(cn2)C(=O)c3ccc(cc3)F)F 7X-0879 CS(=O)(=O)c1ccc2c(c1)sc3n2cc(n3)c4ccc(cc4)Br 7X-0880 c1ccc(c(c1)CNCC(C(F)(F)F)O)Br 7X-0881 COc1ccc(cc1)N2CCN(CC2)CC(C(F)(F)F)O 7X-0882 COC(=O)c1ccc2ncc(n2c1)Cl 7X-0883 COC(=O)c1c(n(nn1)c2ccc(c(c2)Cl)Cl)C(=O)OC 7X-0884 CC(=O)c1cn(nn1)c2ccc(c(c2)Cl)Cl 7X-0885 c1ccc2c(c1)CCNC2C3=C(C(C(CC3=O)c4ccc(cc4)F)n5cncn5)O 7X-0886 COC(=O)c1ccc2ncc(n2c1)Br 7X-0887 Cc1cccn2c1ncc2[N+](=O)[O-] 7X-0888 Cc1c(n2cc(ccc2n1)Cl)/C(=N/O)/C 7X-0890 c1cc2nccn2cc1I 7X-0891 c1cc2nccn2cc1Cl 7X-0892 CCOC(=O)[C@H](CC(C)C)NS(=O)(=O)c1ccc(cc1)CSc2nc3nc(cc(n3n2)C)C 7X-0893 COc1ccc(cc1)OCC(CN2CCN(CC2)c3ccc(cc3)F)O 7X-0894 CCCSc1nc2nc(cc(n2n1)C)C 7X-0895 CN1CCN(CC1)c2ccc(cc2)C(=O)c3ccc(nc3)c4ccc(cc4)F 7X-0898 c1cc(ccc1CO/N=C(/c2cn(nn2)c3ccc(c(c3)Cl)Cl)\C4CC4)Cl 7X-0899 c1cc(c(cc1n2c(c(nn2)CO)CO)Cl)Cl 7X-0900 COC(=O)C(=Cc1cn(nn1)c2ccc(c(c2)Cl)Cl)C(=O)OC 7X-0901 c1cc2nccn2cc1Br 7X-0903 Cc1cc(cn2c1nc(c2)C(=O)O)Br 7X-0905 Cc1cc(cn2c1nc(c2)C(=O)NN)Br 7X-0906 CCOC(=O)c1c(n2cc(nc2s1)c3ccc(cc3)OC)C 7X-0907 Cc1c2cc3c(cc2ncc1C(=O)C4CC4)OCO3 7X-0909 c1cc(oc1)C(=O)c2cc(cc(c2)C(=O)c3ccco3)C(=O)c4ccco4 7X-0910 c1ccn2cc(nc2c1)CC(=O)O 7X-0911 c1ccc(c(c1)C(CCOC(=O)c2ccco2)N3CCS(=O)(=O)CC3)F 7X-0912 Cc1c2c(cc(nc2n(n1)c3cccc(c3)F)c4cccs4)C(F)(F)F 7X-0916 Cc1cc(n2c(n1)nc(n2)SCCCCOc3ccccc3)C 7X-0917 Cc1cc(n2c(n1)nc(n2)SCCCc3ccccc3)C 7X-0918 Cc1cc(n2c(n1)nc(n2)SC)C 7X-0919 COC(=O)n1cc2c(n1)-c3ccccc3OC2 7X-0921 CCOC(=O)C1(CCN(CC1)Cc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)OC 7X-0922 COc1ccc(cc1)C(=O)CCC#N 7X-0923 CCOC(=O)CSc1ccc(cc1)C 7X-0925 Cc1ccc(cc1)C(=O)CC[NH+](C)C.[Cl-] 7X-0926 Cn1cc(c(=O)c2c1ccc(c2)Cl)c3ccccc3C(=O)O 7X-0927 COc1cc2c(cc1OC)C=CN(C(=O)C2)Cc3ccc(cc3)Br 7X-0928 Cn1cc(c(=O)c2c1ccc(c2)Cl)c3ccccc3C(=O)N 7X-0929 Cc1ccc(cc1)C(=O)CCC#N 7X-0934 Cc1cc(=O)n(c(=S)[nH]1)N 7X-0936 COc1cc2c(cc1OC)C=CN(C(=O)C2)Cc3ccc(cc3)[N+](=O)[O-] 7X-0938 COc1cc2c(cc1OC)C=CN(C(=O)C2)Cc3c(cccc3Cl)F 7X-0939 Cc1cc(=O)n2c(n1)sc(n2)c3ccc(cc3)C(F)(F)F 7X-0942 Cc1cc(=O)n2c(n1)sc(n2)c3ccccc3OC 7X-0943 CCOC(=O)CS(=O)(=O)c1ccc(cc1)C 7X-0944 c1cc(ccc1c2cnnc(c2C#N)N)Br 7X-0945 CCn1c2ccccc2c3c(c1=O)c(cc(=O)o3)O 7X-0948 Cc1cc(=O)n2c(n1)sc(n2)S 7X-0951 CCOc1nn2c(=O)cc(nc2s1)C 7X-0952 COC(=O)/C=C(\C(=O)OC)/Nc1ccc(cc1)[N+](=O)[O-] 7X-0954 Cn1c2ccccc2c3c(c1=O)c(cc(=O)o3)O 7X-0958 CCn1c2ccccc2c(c(c1=O)c3cc(=O)[nH][nH]3)O 7X-0960 CCn1c2ccccc2c3c(c1=O)c(c(c(=O)o3)Cc4ccccc4)O 7X-0961 c1ccc2c(c1)-c3c(c(c(c(n3)/C=C/c4cccc(c4)[N+](=O)[O-])C#N)c5ccc6c(c5)OCO6)C2=O 7X-0967 c1ccc2c(c1)-c3c(c(cc(n3)/C=C/c4ccc(cc4)Cl)c5ccc6c(c5)OCO6)C2=O 7X-0968 c1ccc(c(c1)/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccc6c(c5)OCO6)C#N)Cl 7X-0969 c1ccc2c(c1)-c3c(c(c(c(n3)/C=C/c4ccc(cc4)F)C#N)c5ccc6c(c5)OCO6)C2=O 7X-0970 c1ccc(cc1)Cn2c3ccccc3c4c(c2=O)c(cc(=O)o4)O 7X-0971 CCn1c2ccc(cc2cc1C(=O)OCC)NC(=O)c3ccccc3c4ccc(cc4)C(F)(F)F 7X-5020 c1ccc(c(c1)C(=O)N2CCOCC2)[N+](=O)[O-] 7X-5058 c1cc(cc(c1)[N+](=O)[O-])C(=O)N2CCOCC2 7X-5087 CCCCc1nc2cc(c(cc2o1)[N+](=O)[O-])Cl 7X-5092 CCCCc1nc2ccc(cc2o1)[N+](=O)[O-] 7X-5093 CCCCc1nc2cc(ccc2o1)[N+](=O)[O-] 7X-5094 c1cc(cc(c1)n2c(=O)c3c([nH]2)CCCC3)C(=O)O 7Y-0017 c1ccc(c(c1)C(=O)c2cnn(c2)c3cccc(c3)C(=O)O)O 7Y-0027 Cc1c(c(=O)n([nH]1)c2cccc(c2)C(=O)O)CCO 7Y-0028 c1cc(ccc1C=O)N2CCC3(CC2)OCCO3 7Y-0047 COc1ccc(cc1F)c2nc3cc(cc(c3o2)Br)OC 7Y-0058 Cc1c(c(=O)n([nH]1)c2ccc(cc2)Br)CCO 7Y-0201 COC(=O)C(=O)C(C(=O)c1ccccc1)Br 7Y-0606 CC(=O)C(C(=O)C)C(C)(C)C 7Y-0608 COc1ccc(cc1)C(=O)CC(=O)C(=O)OC 7Y-0613 CC(C)(C)OC(=O)NCC(=O)N1CCOCC1 7Y-0617 COC(=O)C(=O)CC(=O)c1cccc(c1)[N+](=O)[O-] 7Y-0618 CC(C)(C)OC(=O)NCC(=O)N(C)C 7Y-0621 C1COCCN1C(=O)CN.Cl 7Y-0622 CN(C)C(=O)CN.Cl 7Y-0624 c1csc2n1c(c(n2)Cl)CO 7Y-0700 c1ccc(c(c1)C(=O)O)Oc2ccc(cc2)N 7Y-0701 Cc1ccc(cc1)C(=O)CC(=O)CCCO 7Y-0702 c1cc(c(cc1N)C(=O)O)N2CCOCC2 7Y-0703 c1ccc(cc1)c2c(n3ccsc3n2)CO 7Y-0704 CCCCc1nc2cc(ccc2o1)N 7Y-0705 CCCCc1nc2ccc(cc2o1)N 7Y-0706 c1cc(c(cc1C(F)(F)F)N)NCCCC(=O)O 7Y-0707 COC(=O)c1cc(ccc1N2CCCC2)[N+](=O)[O-] 7Y-0709 c1cc(c(cc1[N+](=O)[O-])C(=O)O)N2CCCC2 7Y-0712 COC(=O)CCNc1ccc(cc1[N+](=O)[O-])C(F)(F)F 7Y-0713 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCC(=O)O 7Y-0714 Cc1cc(cc(c1O)C(=O)O)Br 7Y-0800 COC(=O)c1ccc(c(c1)N)N2CCSCC2 7Y-0802 CCOc1ccccc1NC(=S)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 7Y-0803 Cc1cc(cc(c1OC)C(=O)OC)Br 7Y-0806 c1cc(c(cc1C(=O)NN)[N+](=O)[O-])N2CCSCC2 7Y-0807 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3cccc(c3Cl)Cl 7Y-0810 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=S)NCc3ccco3 7Y-0811 Cc1cc(n[nH]1)C(=O)NN 7Y-0813 CC(C(=O)OC)Oc1ccc2c(c1)c(c(o2)C3CC3)C=O 7Y-0814 c1cc(c(c(c1)Cl)COc2ccc3c(c2)c(c(o3)C4CC4)C=O)F 7Y-0815 CCOC(=O)c1ccc(cc1)c2ccc(cc2)OC 7Y-0816 COC(=O)c1ccc(c(c1)n2cccc2)N3CCSCC3 7Y-0825 CCS(=O)(=O)N1CCN(CC1)C(=O)CCCl 7Y-0826 Cc1cc(n[nH]1)c2ccc(cc2)c3ccccc3 7Y-0829 C/C(=C\C(=O)c1ccsc1)/N(C)C 7Y-0830 CC(=O)Nc1cccc(c1)C#C 7Y-0831 c1c(sc(n1)Cl)CN2CCC(CC2)N3CCCCC3 7Y-0836 c1cc(ccc1C(=O)N/N=C/c2cscc2Br)C(F)(F)F 7Y-0837 CN1C(=O)C(=Cc2cscc2Br)C(=O)N(C1=O)C 7Y-0838 c1cc(ccc1NS(=O)(=O)NCCCl)Br.c1cc(ccc1N2CCNS2(=O)=O)Br 7Y-0839 CC(CC(=O)NC)NNC(=O)OC(C)(C)C 7Y-0927 CC(=O)c1ccc(c(c1)F)OC 7Y-0947 CC(=O)Oc1ccc(c(c1)F)OCc2cc(ccc2Br)OC 7Y-0950 Cc1cccc(c1C)n2c(c(cn2)C#N)N 7Y-0951 COc1ccc(cc1)/C=C/CO 7Z-0200 c1ccc2c(c1)NC(=O)CC(S2)c3cccs3 7Z-0202 c1cc(ccc1/C=C/CO)Br 7Z-0205 c1ccc2c(c1)NC(=O)CC(S2)c3cc(ccc3Cl)Cl 7Z-0210 Cc1ccc(cc1)S(=O)(=O)OCCN2CCOC2=O 7Z-0220 c1cc(c(cc1N)I)N 7Z-0702 c1cc(ccc1c2ccc3c(c2)OCO3)C(=O)O 7Z-0706 c1cc(ccc1S(=O)(=O)CCl)Cl 7Z-0708 Cn1c(nnc1S)c2c(ccs2)n3cccc3 7Z-0806 COc1ccc2c(c1)c(cn2c3ncccn3)CO 7Z-0807 CN(C)Cc1cnc2n1cc(cc2)Br.Cl 7Z-0808 Cc1ccc(c(c1)[N+](=O)[O-])n2cccc2 7Z-0812 Cc1ccc(cc1n2cccc2)[N+](=O)[O-] 7Z-0813 Cc1c(c(n[nH]1)C(=O)OC)Br 7Z-0815 Cc1cc(c(c(c1)Br)N)[N+](=O)[O-] 7Z-0817 c1cc2ncc(n2cc1Cl)C[NH2+]C34CC5CC(C3)CC(C5)C4.[Cl-] 7Z-0818 CN(C)/C=C/C(=O)c1ccc2c(c1)Nc3ccccc3S2 7Z-0819 Cc1ccc(c(c1)N)n2cccc2 7Z-0821 COc1ccccc1N2CCN(CC2)Cc3cnc4n3cc(cc4)Cl 7Z-0822 c1ccc2c(c1)Nc3cc(ccc3S2)c4cc[nH]n4 7Z-0823 CC(c1ccc(cn1)N)(C(=O)OC)C(=O)OC 7Z-0825 Cc1ccc(cc1n2cccc2)N 7Z-0827 c1ccc(cc1)OCCNc2c(cccc2C#N)C#N 7Z-0828 Cc1c(c(n[nH]1)C(=O)NN)Br 7Z-0829 Cc1c(c(n[nH]1)C(=O)O)Br 7Z-0830 c1cn2c(cc(cc2n1)C(F)(F)F)C(F)(F)F 7Z-0834 CN(C)/C=C/C(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCOCC2 7Z-0837 c1cc(c(cc1c2ccn[nH]2)[N+](=O)[O-])N3CCOCC3 7Z-0839 COc1ccc(cc1)c2cc(cnc2OC)C(F)(F)F 7Z-5023 Cc1ccn(n1)c2ccc(c(c2)Cl)C(=O)O 7Z-5041 COc1ccc(cc1)Cn2c(=O)cc([nH]c2=O)C(=O)OC 7Z-7003 COC(=O)c1cc(=O)n(c(=O)[nH]1)Cc2cccc3c2nsn3 7Z-7004 CC(C)(C)OC(=O)N1CCN(CC1)c2ccccc2C(=O)O 7Z-7046 c1cc(c(cc1F)F)N2CCCC2=O 8B-005 CN(C)/C=C\1/CCN(C1=O)c2ccc(cc2)Cl 8B-006 CN(C)c1nnc(o1)CC(=O)N 8B-008 c1cc(ncc1C(F)(F)F)n2ccnc2 8B-017 c1cc(c(nc1)NN)Cl 8B-018 Cc1c(c[nH]n1)C(=O)Nc2ccsc2C(=O)OC 8B-020 c1cc(c(c(c1)Cl)C(=O)NNc2c(cccn2)Cl)Cl 8B-022 c1cc(c(c(c1)n2ccnc2)C#N)n3ccnc3 8B-024 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])n2ccnc2 8B-029 c1cc(ccc1N/C=C\2/CCN(C2=O)c3ccc(cc3)Cl)F 8B-030 COC(=O)c1ccc(cc1)N/C=C\2/CCN(C2=O)c3ccc(cc3)Cl 8B-031 COC(=O)Cc1ccccc1C(=O)OC 8B-035 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)O 8B-038 C/C(=N\O)/c1ccccc1O 8B-041 CS(=O)(=O)c1cc(cc(c1O)Br)Br 8B-042 CS(=O)(=O)c1cc(cc(c1O)I)I 8B-043 CS(=O)(=O)c1cc(cc(c1OCC(=O)O)I)I 8B-045 C[n+]1ccn(c1)c2cccc(c2C#N)n3cc[n+](c3)C.[I-].[I-] 8B-046 c1ccc2c(c1)c(=O)c3cc(c(nc3o2)C(F)(F)F)C(=O)Nc4ccc(cc4)Cl 8B-047 Cc1c(cnc(n1)N)C(=O)Nc2ccsc2C(=O)OC 8B-048 CCC(=O)Oc1c(cc(cc1I)I)S(=O)(=O)C 8B-054 Cc1c(cnn1c2ccccc2)C(=O)Nc3ccsc3C(=O)OC 8B-055 CCCCCC(=O)Oc1c(cc(cc1I)I)S(=O)(=O)C 8B-056 COC(=O)c1ccc(cc1)NC=C2C=NNC2=O 8B-059 COc1ccccc1NC=C2C=NNC2=O 8B-060 COc1cccc(c1)NC=C2C=NNC2=O 8B-061 c1cc(c(cc1Cl)Cl)NC=C2C=NNC2=O 8B-062 c1cc(c(cc1F)F)NC=C2C=NNC2=O 8B-063 c1ccc(cc1)NC(=O)c2cc3c(=O)c4ccccc4oc3nc2C(F)(F)F 8B-066 c1ccc(cc1)CNC(=O)c2cc3c(=O)c4ccccc4oc3nc2C(F)(F)F 8B-067 c1ccn(c(=O)c1)CC(=O)c2ccc(cc2)Cl 8B-068 CC(c1ccccc1)NC(=O)c2cc3c(=O)c4ccccc4oc3nc2C(F)(F)F 8B-070 CNC1=C(CC(=C(N1C)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl)[N+](=O)[O-])[N+](=O)[O-] 8B-071 CNC1=C(CC(=C(N1C)N2CCN(CC2)C(=O)Nc3cccc(c3)C(F)(F)F)[N+](=O)[O-])[N+](=O)[O-] 8B-072 Cc1c(cn(n1)C(=O)Nc2ccccc2)C(=O)Nc3ccsc3C(=O)OC 8B-073 c1cc(ccc1NC=C2C=NNC2=O)[N+](=O)[O-] 8B-074 c1ccc(c(c1)C#N)NC=C2C=NNC2=O 8B-075 c1cc(c(cc1Cl)NC=C2C=NNC2=O)O 8B-076 Cc1c(cn(n1)C(=O)c2ccc(cc2)Cl)C(=O)Nc3ccsc3C(=O)OC 8B-077 c1ccc(c(c1)NC=C2C=NNC2=O)O 8B-079 COC(=O)c1c(ccs1)NC=C2C=NNC2=O 8B-080 C1=NNC(=O)C1/C=N/O 8B-081 CNC1=C(CC(=C(N1C)N2CCN(CC2)C(=O)c3ccccc3)[N+](=O)[O-])[N+](=O)[O-] 8B-082 c1cc(ccc1c2c(c[nH]n2)N3C=CCCC3=O)Cl 8B-084 CNC1=C(CC(=C(N1C)N2CCN(CC2)S(=O)(=O)c3ccccc3)[N+](=O)[O-])[N+](=O)[O-] 8B-085 CC(=O)N1CCN(CC1)C2=C(CC(=C(N2C)NC)[N+](=O)[O-])[N+](=O)[O-] 8B-086 CNC1=C(CC(=C(N1C)N2CCN(CC2)S(=O)(=O)C)[N+](=O)[O-])[N+](=O)[O-] 8B-087 c1ccnc(c1)CC(=S)N2CCOCC2 8B-088 CN(C)/C=C/c1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] 8B-089 CC1=NNC(=O)C1=CN(C)C 8B-091 CC1=NNC(=O)C1=CNc2ccc(cc2)Cl 8B-093 CN(C)C=C1C(=NNC1=O)C(F)(F)F 8B-094 c1ccn(c(=O)c1)c2cnc(nc2c3ccc(cc3)Cl)N 8B-096 CC1=NNC(=O)C1=CNc2ccccc2 8B-098 Cc1ccc(cc1)NC=C2C(=NNC2=O)C 8B-099 CC1=NNC(=O)C1=CNc2ccc(cc2)OC 8B-100 CC1=NNC(=O)C1=CNc2cccc(c2)C(F)(F)F 8B-101 CC1=NNC(=O)C1=CNc2cc(ccc2O)Cl 8B-102 c1ccc(cc1)NC=C2C(=NNC2=O)C(F)(F)F 8B-103 c1ccc(c(c1)NC=C2C(=NNC2=O)C(F)(F)F)Cl 8B-104 c1cc(cc(c1)Cl)NC=C2C(=NNC2=O)C(F)(F)F 8B-105 c1cc(ccc1NC=C2C(=NNC2=O)C(F)(F)F)Cl 8B-106 c1cc(cc(c1)NC=C2C(=NNC2=O)C(F)(F)F)C(F)(F)F 8B-107 c1ccc(cc1)CN2CCN(CC2)c3[nH]nc(n3)N 8C-002 Cc1c(c(ns1)S(=O)(=O)Cc2cccc(c2)Cl)C#N 8C-011 CN(C)/C=C\1/CCN(C1=O)c2ccc(cc2)OC(F)(F)F 8C-012 Cc1c(c(ns1)SCc2ccccc2Cl)C#N 8C-013 Cc1c(c(ns1)S(=O)(=O)Cc2ccccc2Cl)C#N 8C-016 Cc1c(c(ns1)S(=O)(=O)CC#N)C#N 8C-019 CS/C(=N\C#N)/N1CCN(CC1)c2ccccc2Cl 8C-022 c1cc(ccc1/C=C(\c2ccn[nH]2)/Oc3ccc(cc3)Cl)Cl 8C-038 c1cc(ccc1N2CCCC2=O)Br 8C-039 CC(C(=O)C)Oc1ccc(cc1)Cl 8C-042 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1)Cl 8C-045 CC(c1ccnc(n1)N)Oc2ccc(cc2)Cl 8C-047 CC(c1ccn[nH]1)Oc2ccc(cc2)Cl 8C-048 Cc1c(c(ns1)S(=O)(=O)Cc2c(cccc2Cl)Cl)C#N 8C-051 CC(c1ccnn1S(=O)(=O)c2ccc(cc2)Cl)Oc3ccc(cc3)Cl 8C-053 CN1CC/C(=C/N(C)C)/C1=S 8C-055 CN(C)/C=C\1/CCN(C1=O)c2ccc(cc2)Br 8C-057 c1cc(ccc1/C=C(/c2ccnn2S(=O)(=O)c3ccc(cc3)Cl)\Oc4ccc(cc4)Cl)Cl 8C-064 Cc1c(c(ns1)SCc2ccc(cc2)F)C#N 8C-075 Cc1c(c(ns1)S(=O)(=O)Cc2ccc(cc2)F)C#N 8C-076 c1ccc(cc1)/C=C(\c2ccnn2S(=O)(=O)c3cccc(c3)Cl)/Oc4ccc(cc4)Cl 8C-079 c1cc(ccc1N2CCCC2=O)F 8C-080 CO/N=C/CC(=O)c1ccc(cc1)Cl 8C-082 CN1/C(=C/[N+](=O)[O-])/SC(C1=O)C2c3ccccc3C(=O)O2 8C-084 c1ccc2c(c1)/C(=N/Nc3ccc(cc3)Cl)/C(=O)OC2=O 8C-088 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)O 8C-090 c1ccc2c(c1)/C(=N\Nc3ccc(cc3)F)/C(=O)OC2=O 8C-097 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)F)C(=O)O 8C-098 c1ccc2c(c1)/C(=N/Nc3ccc(cc3Cl)Cl)/C(=O)OC2=O 8C-099 c1ccc(cc1)N/N=C\2/c3ccccc3C(=O)OC2=O 8C-101 CC1=C(C(=O)NC1(C)O)C(=O)/C=C/N(C)C 8C-106 c1cc(ccc1N2CCN(CC2)c3[nH]nc(n3)N)Cl 8C-107 c1ccc(c(c1)/C(=N/Nc2ccc(cc2Cl)Cl)/C(=O)O)C(=O)O 8C-108 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)O 8C-111 c1ccc2c(c1)/C(=N/Nc3cccc(c3)C(F)(F)F)/C(=O)OC2=O 8C-112 c1ccc(cc1)CN2Cc3ccccc3C2=O 8C-113 Cc1cc(c2c(c1)occ(c2=O)C=O)C 8C-118 Cc1cccc(c1N2CCN(CC2)c3[nH]nc(n3)N)C 8C-121 COc1ccc(cc1)N/N=C\2/c3ccccc3C(=O)OC2=O 8C-122 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4[nH]nc(n4)N 8C-123 c1ccc2c(c1)c(nn(c2=O)c3cccc(c3)C(F)(F)F)C(=O)O 8C-124 COc1ccc(cc1)N2CCN(CC2)c3[nH]nc(n3)N 8C-127 c1ccc(c(c1)N2CCN(CC2)c3[nH]nc(n3)N)Cl 8C-128 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)O 8C-132 c1ccnc(c1)N2CCN(CC2)c3[nH]nc(n3)N 8C-133 CS/C(=N\C#N)/N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] 8C-134 CN(C)C(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)Cl 8C-137 c1cc(ccc1N2CCN(CC2)c3[nH]nc(n3)N)[N+](=O)[O-] 8C-138 CN(C)C(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)F 8C-140 CNC(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)F 8C-144 COC(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)Cl 8C-146 c1ccc(cc1)NC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(cc4)F 8C-147 COC(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)F 8C-148 c1ccc(cc1)OC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(cc4)F 8C-149 c1ccc(c(c1)[N+](=O)[O-])Oc2c(n3ccsc3n2)[N+](=O)[O-] 8D-001 COc1ccc(cc1)CNc2c(n3ccsc3n2)[N+](=O)[O-] 8D-002 c1ccc2c(c1)c(n[nH]c2=O)CN3CCN(CC3)c4ccc(cc4)Cl 8D-003 CSc1[nH]nc(n1)NCc2c3ccccc3c(=O)[nH]n2 8D-004 c1ccc(cc1)N2CCN(CC2)c3c(n4ccsc4n3)[N+](=O)[O-] 8D-006 CNc1ncc(s1)C(=O)c2ccc(cc2)Cl 8D-007 CNc1ncc(s1)C(=O)c2ccc(cc2)F 8D-008 c1ccc2c(c1)c(n[nH]c2=O)CNC34CC5CC(C3)CC(C5)C4 8D-009 CNc1ncc(s1)C(=O)c2ccc(cc2Cl)Cl 8D-010 CNc1ncc(s1)C(=O)c2ccc(cc2)c3ccccc3 8D-011 c1cc(ccc1C(=O)C/C=N/OCc2ccc(cc2Cl)Cl)Cl 8D-012 c1ccc2c(c1)/C(=C/Nc3[nH]nc(n3)SCc4c(cccc4Cl)Cl)/OC2=O 8D-013 CN(C)/C=N/C(=S)Nc1ccccc1Cl 8D-014 c1ccc(cc1)c2cnc(sc2=O)c3ccccc3 8D-015 CNc1ncc(s1)C(=O)c2ccc(c(c2)Cl)Cl 8D-016 CNc1ncc(s1)C(=O)c2ccccc2 8D-017 c1ccc(cc1)CN2CCN(CC2)c3c(n4ccsc4n3)[N+](=O)[O-] 8D-018 c1csc2n1c(c(n2)N3CCCCC3)[N+](=O)[O-] 8D-019 c1csc2n1c(c(n2)N3CCCC3)[N+](=O)[O-] 8D-020 c1ccc(c(c1)Nc2ncc(s2)C(=O)c3ccc(cc3)Cl)Cl 8D-021 c1ccc(cc1)Nc2ncnc(n2)N 8D-023 CC(C)(C)C(=O)c1cnc(s1)NC 8D-024 CC(=O)c1cnc(s1)NC 8D-026 c1ccc(cc1)COc2ccsc2C(=O)NNC(=S)N 8D-027 c1ccc(cc1)C(=O)c2cnc(s2)Nc3ccccc3Cl 8D-028 CC(=O)c1cnc(s1)Nc2ccccc2Cl 8D-031 c1ccc(cc1)c2ccc(cc2)C(=O)c3cnc(s3)Nc4ccccc4Cl 8D-032 c1ccc(c(c1)Nc2ncc(s2)C(=O)c3ccc(cc3)Br)Cl 8D-033 c1ccc(c(c1)Nc2ncc(s2)C(=O)c3ccc(c(c3)Cl)Cl)Cl 8D-034 CC(C)(C)C(=O)c1cnc(s1)Nc2ccccc2Cl 8D-035 c1csc2n1c(c(n2)S)[N+](=O)[O-] 8D-036 CNC(=O)CSc1c(n2ccsc2n1)[N+](=O)[O-] 8D-038 c1csc2n1c(c(n2)SCC(=O)O)[N+](=O)[O-] 8D-039 c1ccc(cc1)COc2ccsc2c3[nH]c(nn3)S 8D-040 Cc1ccc(cc1)COc2ccsc2c3[nH]c(nn3)SC 8D-041 c1c(ccc(c1)Cl)C(=C(/C=N/OCc2c(cc(cc2)Cl)Cl)/C=N/OCc3c(cc(cc3)Cl)Cl)O 8D-044 c1cc(ccc1/C=[N+]/2\CCC(=O)[N-]2)Cl 8D-045 c1ccc2c(c1)/C(=C/NOCc3ccc(cc3Cl)Cl)/OC2=O 8D-047 c1ccc(c(c1)Nc2ncc(s2)C(=O)c3ccc(cc3)F)Cl 8D-049 c1ccnc(c1)c2nnc(o2)S 8D-050 c1ccnc(c1)c2nn(c(=S)o2)CN3CCOCC3 8D-053 c1cc(cnc1)c2nnc(o2)S 8D-054 c1cc(sc1)c2nnc(o2)S 8D-055 c1c(nc(n(c1=O)N)N)C(F)(F)F 8D-056 c1cc(cnc1)c2nn(c(=S)o2)CN3CCOCC3 8D-060 c1cc(sc1)c2nn(c(=S)o2)CN3CCOCC3 8D-061 c1csc2n1c(c(n2)Cl)C=O 8D-062 CC(=O)C1=C(CS(=O)(=O)C1)Sc2ccc(cc2)Cl 8D-064 c1ccc(cc1)Sc2c(n3ccsc3n2)C=O 8D-068 c1cc(ccc1Sc2c(n3ccsc3n2)C=O)Cl 8D-069 CN(C)/C=N/C(=S)Nc1ccc(c(c1)Cl)Cl 8D-070 Cc1ccc(cc1)SC2=C(CS(=O)(=O)C2)C(=O)C 8D-071 c1ccc(cc1)Sc2c(n3ccsc3n2)/C=N\O 8D-073 c1cc(ccc1Sc2c(n3ccsc3n2)/C=N\O)Cl 8D-074 CO/N=C\c1c(nc2n1ccs2)Sc3ccccc3 8D-075 CO/N=C\c1c(nc2n1ccs2)Sc3ccc(cc3)Cl 8D-076 c1cc(cc(c1)Sc2c(n3ccsc3n2)C=O)C(F)(F)F 8D-077 Cc1ccc(cc1)Sc2c(n3ccsc3n2)C=O 8D-078 c1ccc(cc1)Sc2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl 8D-079 c1cc(ccc1Sc2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl)Cl 8D-080 Cc1cc(n(n1)C(=S)N)C 8D-081 c1ccc(cc1)Sc2c(n3ccsc3n2)/C=N/OCc4c(cccc4Cl)Cl 8D-082 c1cc(c(c(c1)Cl)CO/N=C/c2c(nc3n2ccs3)Sc4ccc(cc4)Cl)Cl 8D-083 Cc1ccc(cc1)Sc2c(n3ccsc3n2)/C=N\OC 8D-084 Cc1ccc(cc1)Sc2c(n3ccsc3n2)/C=N/OCc4ccc(c(c4)Cl)Cl 8D-085 c1cc(cc(c1)Sc2c(n3ccsc3n2)/C=N/O)C(F)(F)F 8D-086 Cc1ccc(cc1)Sc2c(n3ccsc3n2)/C=N\O 8D-087 c1cc(ccc1C(=O)c2cnc(s2)Nc3ccc(c(c3)Cl)Cl)F 8D-090 c1cc(ccc1C(=O)c2cnc(s2)Nc3ccc(c(c3)Cl)Cl)Cl 8D-091 CN(C)C(=C(C#N)C#N)Sc1ccc(cn1)C(F)(F)F 8D-092 c1cc(nc(c1)Cl)NNC(=O)C(F)(F)F 8D-093 CN(C)C(=C(C#N)C#N)N1CCN(CC1)c2ccccc2 8D-096 Cc1ccc(cc1)Sc2c(n3ccsc3n2)/C=N/OCc4c(cccc4Cl)Cl 8D-097 CN(C)C(=C(C#N)C#N)N1CCN(CC1)Cc2ccccc2 8D-101 c1cc(ccc1C(=O)c2cnc(s2)Nc3ccc(c(c3)Cl)Cl)Br 8D-102 c1ccc(cc1)C(=O)c2cnc(s2)Nc3ccc(c(c3)Cl)Cl 8D-103 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)N 8D-104 c1cc(c(cc1C(=O)c2cnc(s2)Nc3ccc(c(c3)Cl)Cl)Cl)Cl 8D-109 c1cc(ccc1CSc2c(n3ccsc3n2)C=O)Cl 8D-110 c1cc(c(cc1Nc2ncc(s2)C(=O)c3ccc(cc3Cl)Cl)Cl)Cl 8D-111 c1ccnc(c1)c2cc(sc2N3CCOCC3)C(=O)c4ccc(cc4)Cl 8D-112 CO/N=C/c1c(nc2n1ccs2)Sc3cccc(c3)C(F)(F)F 8D-113 Cc1ccc(cc1)S(=O)(=O)C2=C(CS(=O)(=O)C2)C(=O)C 8D-114 c1ccnc(c1)c2cc(sc2N3CCOCC3)C(=O)c4ccc(c(c4)Cl)Cl 8D-116 c1ccc(cc1)C(=O)c2cc(c(s2)N3CCOCC3)c4ccccn4 8D-117 c1cc(ccc1CSc2c(n3ccsc3n2)/C=N/O)Cl 8D-119 CO/N=C/c1c(nc2n1ccs2)SCc3ccc(cc3)Cl 8D-120 c1cc(c(c(c1)Cl)CO/N=C/c2c(nc3n2ccs3)SCc4ccc(cc4)Cl)Cl 8D-121 c1ccnc(c1)c2cc(sc2N3CCOCC3)C(=O)c4ccc(cc4)Br 8D-122 CN(C)C(=C(C#N)C#N)N1CCN(CC1)c2ccc(cc2)Cl 8D-123 c1ccc(cc1)NC(=O)CC(=O)O 8D-126 COC(=O)c1c(ccs1)c2ccc(o2)C=O 8D-127 c1ccc2c(c1)c(n[nH]c2=O)CNOCc3ccc(cc3Cl)Cl 8D-128 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)OC(F)(F)F)/OC2=O 8D-129 c1cc(ccc1SC2=CS(=O)(=O)CC2)Cl 8D-134 CN(C)C(=C(C#N)C#N)N1CCN(CC1)c2ccc(c(c2)Cl)Cl 8D-135 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3)OC(F)(F)F 8D-136 c1ccc2c(c1)/C(=C/NOCc3ccc(cc3)Cl)/OC2=O 8D-138 c1ccc2c(c1)/C(=C/NOCc3c(cccc3Cl)Cl)/OC2=O 8D-139 c1ccc2c(c1)/C(=C/NOCc3ccc(c(c3)Cl)Cl)/OC2=O 8D-140 COc1ccc(c(c1)OC)n2cc3ccsc3c2 8E-003 c1cc(ccc1C(F)(F)F)S(=O)(=O)CS(=O)(=O)C(F)(F)F 8E-006 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3ccc(cc3)F)/[N+](=O)[O-] 8E-009 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3ccc(cc3Cl)Cl)/[N+](=O)[O-] 8E-010 c1ccc2c(c1)C(OC2=O)/C(=C\Nc3ccc(cc3)[N+](=O)[O-])/[N+](=O)[O-] 8E-011 COc1ccc(cc1)N/C=C(\C2c3ccccc3C(=O)O2)/[N+](=O)[O-] 8E-012 Cc1ccccc1C(C#N)c2ccc(nn2)Cl 8E-014 CC(C)(C)c1ccc(cc1)N/C=C(\C2c3ccccc3C(=O)O2)/[N+](=O)[O-] 8E-015 c1ccc(cc1)NC(=O)C(F)(F)F 8E-016 Cc1ccccc1Cc2ccc(nn2)O 8E-017 Cc1ccccc1Cc2ccc(nn2)Cl 8E-020 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)N 8E-021 CN(C)/C=N/C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 8E-022 Cc1nc(cn1C)[N+](=O)[O-] 8E-023 c1cc(c(cc1Cl)Cl)CO/N=C\NC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3Cl)Cl 8E-024 Cc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)O 8E-025 CN(C)/C=C/C(=O)c1cccc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl 8E-026 Cc1ccccc1Cc2ccc(nn2)NN 8E-027 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)c3cc[nH]n3 8E-028 c1cc(ccc1C#N)Oc2c(cc(cn2)C(F)(F)F)Cl 8E-031 c1cc(ccc1C(=O)N)Oc2c(cc(cn2)C(F)(F)F)Cl 8E-033 CN(C)/C=N/C(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 8E-034 CO/N=C\NC(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 8E-035 Cc1c(cccc1C#N)C#N 8E-036 c1cc(ccc1NC(=O)N)Oc2c(cc(cn2)C(F)(F)F)Cl 8E-037 c1cc(ccc1c2cc[nH]n2)Oc3c(cc(cn3)C(F)(F)F)Cl 8E-038 Cc1ccc(cc1)C(C#N)c2ccc(nn2)NN 8E-039 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)N/C=N\OCc3ccc(cc3Cl)Cl 8E-041 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)N 8E-044 c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)C(=O)Nc3ccc(cc3F)F)Cl)Cl 8E-301S CNC(=O)c1cc(cn(c1=O)Cc2c(cccc2Cl)Cl)Cl 8E-302S C=CCNC(=O)c1cc(c(=O)n(c1)Cc2c(cccc2Cl)Cl)Cl 8E-303S c1cc(cc(c1)NC(=O)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)Cl)C(F)(F)F 8E-304S c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3)Cl)Cl 8E-305S COc1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3ccc(c(c3)Cl)Cl)Cl 8E-306S CCN(CC)C(=O)c1cc(cn(c1=O)Cc2c(cccc2Cl)Cl)Cl 8E-307S c1ccc(cc1)CNC(=O)c2cc(cn(c2=O)Cc3c(cccc3Cl)Cl)Cl 8E-308S c1cnccc1c2nc(cc(n2)O)C(F)(F)F 8E-309S Cc1c(snn1)S(=O)(=O)Cc2ccccc2C(F)(F)F 8E-310S COC(=O)c1cc(c(=O)n(c1)Cc2cccc(c2)C(F)(F)F)Cl 8E-311S c1ccc(cc1)CNC(=O)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)Cl 8E-312S CN(c1ccccc1)C(=O)c2cc(c(=O)n(c2)Cc3c(cccc3Cl)Cl)Cl 8E-313S c1cc(cc(c1)NC(=O)c2cc(cn(c2=O)Cc3c(cccc3Cl)Cl)Cl)C(F)(F)F 8E-314S c1cc(cnc1)c2nc(cc(n2)O)C(F)(F)F 8E-317S CCN(CC)C(=O)c1cc(c(=O)n(c1)Cc2c(cccc2Cl)Cl)Cl 8E-318S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)Cl)C(=O)O 8E-319S COC(=O)c1cc(cn(c1=O)Cc2cccc(c2)C(F)(F)F)Cl 8E-320S c1ccc(cc1)Cn2cc(cc(c2=O)C(=O)O)Cl 8E-321S Cc1ccccc1CS(=O)(=O)c2c(nns2)C 8E-322S c1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)C(F)(F)F)Cl 8E-324S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3)Cl 8E-325S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 8E-326S COC(=O)c1cc(cn(c1=O)Cc2ccc(cc2)Cl)Cl 8E-328S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3F)F 8E-329S CNC(=O)c1cc(c(=O)n(c1)Cc2cccc(c2)C(F)(F)F)Cl 8E-330S c1ccc(cc1)CNC(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)C(F)(F)F)Cl 8E-331S COC(=O)c1cc(c(=O)n(c1)Cc2ccccc2)Cl 8E-332S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)C(=O)O)Cl 8E-333S c1cc(ccc1Cn2cc(cc(c2=O)C(=O)O)Cl)Cl 8E-334S C=CCNC(=O)c1cc(c(=O)n(c1)Cc2cccc(c2)C(F)(F)F)Cl 8E-335S CN(C)CCNC(=O)c1cc(c(=O)n(c1)Cc2cccc(c2)C(F)(F)F)Cl 8E-336S c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C(=O)O 8E-337S c1cnccc1c2nc(cc(n2)Cl)C(F)(F)F 8E-339S c1cc(cnc1)c2nc(cc(n2)Cl)C(F)(F)F 8E-340S CN(c1ccccc1)C(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)C(F)(F)F)Cl 8E-342S COC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)Cl 8E-343S c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3)Cl 8E-344S c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccccc3 8E-345S c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C(=O)Nc3cccc(c3)C(F)(F)F 8E-346S CNC(=O)c1cc(c(=O)n(c1)Cc2ccccc2)Cl 8E-350S c1cc(ccc1Cn2cc(cc(c2=O)Cl)C(=O)O)Cl 8E-351S c1ccc(cc1)CNC(=O)c2cc(c(=O)n(c2)Cc3ccccc3)Cl 8E-358S c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3F)F 8E-359S CN(c1ccccc1)C(=O)c2cc(cn(c2=O)Cc3ccccc3)Cl 8E-365S CN(C)CCNC(=O)c1cc(c(=O)n(c1)Cc2ccccc2)Cl 8E-366S c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C(=O)N3CCOCC3 8E-367S CN1CCN(CC1)C(=O)c2cc(c(=O)n(c2)Cc3ccccc3)Cl 8E-368S c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C(=O)Nc3cc(cc(c3)Cl)Cl 8E-370S COC(=O)c1ccc(=O)n(c1)CC(=O)c2ccc(cc2)Cl 8E-373S c1cc(ccc1Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3)Cl)Cl 8E-374S c1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)Cl 8E-375S COC(=O)c1cccn(c1=O)CC(=O)c2ccc(cc2)Cl 8E-376S COC(=O)c1cccn(c1=O)CC(=O)c2ccc(cc2Cl)Cl 8E-379S COC(=O)c1cc(c(=O)n(c1)Cc2cccc(c2)Cl)Cl 8E-382s CN(C)CCNC(=O)c1cc(cn(c1=O)Cc2ccc(cc2)Cl)Cl 8E-383S c1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)Cl)Cl 8E-384S CNC(=O)c1cc(cn(c1=O)Cc2ccc(cc2)Cl)Cl 8E-386S c1cc(cc(c1)NC(=O)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)Cl)C(F)(F)F 8E-387S c1cc(nc(c1C(=O)N)O)C(F)(F)F 8E-389S CNC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)Cl 8E-390S c1ccc(cc1)CNC(=O)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)Cl 8E-391S c1cc(ccc1Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3F)F)Cl 8E-392S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)O 8E-393S CN(C)CCNC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)Cl 8E-396S C=CCNC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)Cl 8E-397S CN(c1ccccc1)C(=O)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)Cl 8E-398S c1cc(ccc1Cn2cc(cc(c2=O)Cl)C(=O)N3CCOCC3)Cl 8E-399S CN1CCN(CC1)C(=O)c2cc(c(=O)n(c2)Cc3ccc(cc3)Cl)Cl 8E-400S c1cc(ccc1Cn2cc(cc(c2=O)Cl)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl 8E-401S COc1cc(cn(c1=O)Cc2c(cccc2Cl)Cl)C(F)(F)F 8E-501 c1ccc(cc1)Cn2cc(cc(c2=O)[N+](=O)[O-])C(F)(F)F 8E-502 c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)[N+](=O)[O-])C(F)(F)F 8E-503 COC(c1cc(c(=O)n(c1)Cc2ccccc2)Cl)(OC)OC 8E-505 COC(c1cc(c(=O)n(c1)Cc2cccc(c2)Cl)Cl)(OC)OC 8E-506 COC(=O)c1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-508 COC(=O)c1ccc(cc1)Cn2cc(cc(c2=O)[N+](=O)[O-])C(F)(F)F 8E-509 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)C(=O)O 8E-510 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)C(=O)Nc3ccc(cc3)Cl 8E-513 c1cc(ccc1CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F)Cl 8E-514 c1ccc(cc1)CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-515 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 8E-517 CC(C)(C)NC(=O)c1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-518 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)C(=O)Nc3ccc(cc3)OC(F)(F)F 8E-519 C=CCNC(=O)c1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-520 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)C(=O)NCc3ccncc3 8E-521 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)C(=O)NCC3CC3 8E-523 c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)N)C(F)(F)F)Cl 8E-525 c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)NC(=O)c3ccc(cc3Cl)F)C(F)(F)F)Cl 8E-532 CC(C)Oc1ccc(cc1)C(=O)Nc2cc(cn(c2=O)Cc3c(cccc3Cl)Cl)C(F)(F)F 8E-533 c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)NC(=O)C(Cl)(Cl)Cl)C(F)(F)F)Cl 8E-534 CC(C)CC(=O)Nc1cc(cn(c1=O)Cc2c(cccc2Cl)Cl)C(F)(F)F 8E-535 c1cc(cnc1)CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-539 c1ccnc(c1)CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-540 Cc1cccc(c1)NC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-541 COc1ccccc1NC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-542 Cc1c(cccc1Cl)NC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-544 c1cc(sc1)CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-545 CCCNC(=O)c1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-546 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)C(=O)Nc3ccc(cc3)[N+](=O)[O-] 8E-547 c1cc(cc(c1)C(F)(F)F)CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-548 COC(=O)c1ccc(cc1)NC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-549 c1ccc(c(c1)CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F)Cl 8E-550 COc1ccccc1CNC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-551 c1ccc(cc1)NC(=O)c2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-552 COC(=O)Nc1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-555 CNC(=O)Nc1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-556 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)NC(=O)N3CCOCC3 8E-557 CC(C)(C)NC(=O)Nc1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-558 c1ccc(cc1)NC(=O)Nc2ccc(cc2)Cn3cc(ccc3=O)C(F)(F)F 8E-559 c1cc(ccc1Cn2cc(ccc2=O)C(F)(F)F)NC(=O)Nc3ccc(cc3)OC(F)(F)F 8E-561 COC(=O)CSC(=O)Nc1ccc(cc1)Cn2cc(ccc2=O)C(F)(F)F 8E-563 Cc1c(c(n(n1)c2nc(cs2)c3ccccc3)O)C(=O)/C=C(/C)\O 8E-902 C=CCNC(=S)Nc1ccccc1 8E-903 Cc1cc(n(n1)c2ccc(cc2)Cl)c3c(nn(c3O)c4nc(cs4)c5ccccc5)C 8E-904 c1ccc(c(c1)/C=N/Nc2c3ccccc3ncn2)F 8E-906 c1ccc2c(c1)c(ncn2)N/N=C/c3cccc(c3)Cl 8E-907 c1ccc2c(c1)c3nnc(n3cn2)c4ccccc4F 8E-908 c1ccc2c(c1)c(nc(n2)Cl)N/N=C/c3ccc(cc3Cl)Cl 8E-909 c1ccc2c(c1)c(ncn2)N/N=C/c3ccc(c(c3)Cl)Cl 8E-910 c1ccc2c(c1)c(ncn2)N/N=C/c3ccc(cc3)Br 8E-911 c1ccc2c(c1)c3nnc(n3cn2)c4cccc(c4)Cl 8E-912 c1ccc2c(c1)c3nnc(n3cn2)c4ccc(c(c4)Cl)Cl 8E-913 c1ccc2c(c1)c3nnc(n3cn2)c4ccc(cc4)Br 8E-914 COC(=O)/C(=C\Nc1ccccc1N)/NC(=O)c2ccccc2 8E-915 COC(=O)/C(=C/n1c2ccccc2nn1)/NC(=O)c3ccccc3 8E-916 c1ccc2c(c1)c(nc(n2)Cl)N/N=C/c3ccc(cc3)Br 8E-917 c1ccc(cc1)/C=N/Nc2c3ccccc3ncn2 8E-918 c1ccc2c(c1)c3nnc(n3c(n2)Cl)c4ccc(cc4)Br 8E-919 c1ccc2c(c1)c(nc(n2)Cl)N/N=C/c3cccc(c3)Cl 8E-920 c1ccc(c(c1)/C=N/Nc2c3ccccc3nc(n2)Cl)F 8E-921 c1ccc2c(c1)c(nc(n2)Cl)N/N=C/c3ccc(c(c3)Cl)Cl 8E-922 CN1CCN(CC1)c2nc3ccccc3c4n2c(nn4)c5ccc(cc5)Br 8E-923 c1ccc2c(c1)c3nnc(n3c(n2)Cl)c4ccc(cc4Cl)Cl 8E-924 c1ccc2c(c1)c3nnc(n3c(n2)Cl)c4ccc(c(c4)Cl)Cl 8E-925 c1ccc2c(c1)c3nnc(n3c(n2)Cl)c4ccccc4F 8E-926 c1ccc2c(c1)c3nnc(n3c(n2)N4CCCCC4)c5ccc(cc5)Br 8E-927 c1ccc2c(c1)c3nnc(n3c(n2)N4CCOCC4)c5ccc(cc5)Br 8E-928 C=CCNC(=S)Nc1ccc(cc1)Cl 8E-930 COc1ccc(cc1)NC(=S)NCC=C 8E-931 COc1nc2ccccc2c3n1c(nn3)c4ccc(cc4)Br 8E-932 C=CCNC(=S)Nc1cccc(c1)C(F)(F)F 8E-934 c1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccc(cc5)Br 8E-936 c1ccc2c(c1)c3nnc(n3c(n2)O)c4cccc(c4)Cl 8E-937 CNc1nc2ccccc2c3n1c(nn3)c4ccc(cc4)Br 8E-938 COc1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccc(cc5)Br 8E-940 c1ccc(cc1)C(C#N)c2ccc(nn2)Sc3ccccc3 8F-001 CCOC(=O)Cc1[nH]c(nn1)c2ccccc2 8F-002 CCOC(=O)C(CC(=O)c1ccc(cc1Cl)Oc2ccc(cc2)Cl)(C(=O)OCC)O 8F-003 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)Sc3nc([nH]n3)N 8F-004 Cc1c(nc(s1)c2c(cccc2F)F)OCc3ccccc3 8F-005 Cc1c(nc(s1)c2c(cccc2F)F)OCc3ccc(cc3)C(F)(F)F 8F-007 c1cc(c(cc1Cl)Cl)/C(=C/Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)/C#N 8F-009 CCOC(=O)c1c(nc(s1)C)C(F)(F)F 8F-011 CC(C)(c1nnc(n1C)SCC=C)n2cncn2 8F-012 CCOc1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F 8F-013 CC(C)(c1nnc(n1C)SCC(=O)OC)n2cncn2 8F-014 Cc1nc(c(s1)C(=O)O)C(F)(F)F 8F-015 c1ccc(cc1)Sc2ccc(nn2)C(C#N)c3ccc(cc3Cl)Cl 8F-016 Cc1nc(c(s1)C(=O)N)C(F)(F)F 8F-017 Cc1nc(c(s1)C#N)C(F)(F)F 8F-018 CCOC(=O)Cc1csc(n1)Cn2cncn2 8F-019 CN(C)/C=C/c1nc(c(s1)C#N)C(F)(F)F 8F-020 c1cc(ccc1N/C=C/c2nc(c(s2)C#N)C(F)(F)F)Cl 8F-021 c1cc(cc(c1)C(F)(F)F)COc2ccsc2C(=O)NNC(=N)COc3ccc(cc3)Cl 8F-022 Cc1nc(c(s1)C(=O)OCC(=O)c2ccc(cc2)Cl)C(F)(F)F 8F-024 c1ccc(cc1)C(C#N)c2ccc(nn2)Sc3ccc(cc3)Cl 8F-026 c1cc(ccc1CO/N=C\Cc2nc(c(s2)C#N)C(F)(F)F)Cl 8F-027 c1ccc(cc1)Sc2ccc(nn2)C(c3ccc(cc3Cl)Cl)C(=O)N 8F-028 CC(C)(c1nnc(n1C)Sc2c(cc(cn2)C(F)(F)F)Cl)n3cncn3 8F-029 c1ccc(cc1)Nc2ccc(nn2)C(C#N)c3ccc(cc3Cl)Cl 8F-030 COc1ccc(cc1)N/C=C/c2nc(c(s2)C#N)C(F)(F)F 8F-032 c1cc(c(c(c1)Cl)CON/C=C/c2nc(c(s2)C#N)C(F)(F)F)Cl 8F-034 c1ccc(cc1)Cc2c3ccccc3c(nn2)Oc4ccc(cc4Cl)Cl 8F-035 c1cc(ccc1C(=O)N/C=N/OCc2ccc(cc2Cl)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 8F-036 c1cc(ccc1Sc2ccc(nn2)C(C#N)c3ccc(cc3Cl)Cl)Cl 8F-037 c1cc(cc(c1)OC(=O)c2ccc(cc2)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 8F-039 c1ccc(c(c1)S(=O)(=O)Oc2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl 8F-040 CCOC(=O)c1c(nc(s1)/C=C/N(C)C)C(F)(F)F 8F-042 Cc1ccc(cc1)Sc2c3ccccc3c(nn2)Cc4ccccc4 8F-043 c1ccc(c(c1)COn2c3cccnc3nc2c4ccc(cc4)Cl)Cl 8F-301S c1ccc(c(c1)COn2c3cccnc3nc2c4cccc(c4)C(F)(F)F)Cl 8F-302S Cc1ccc(cc1)c2nc3c(n2OCc4ccccc4)cccn3 8F-303S Cc1ccc(cc1)c2nc3c(n2OCc4cccc(c4)C(F)(F)F)cccn3 8F-304S Cc1cc(cc(c1)C(=N)Nc2cccc(c2)C#N)C 8F-305S c1ccc(cc1)CNc2ccc(cc2[N+](=O)[O-])Cl 8F-306S c1ccc(cc1)c2nc3ccc(cc3n2O)Cl 8F-307S Cc1ccc(cc1)c2nc3c(n2OCc4cccc(c4)Cl)cccn3 8F-308S COc1ccc(cc1)CNc2c(cccn2)[N+](=O)[O-] 8F-309S COc1ccc(cc1)c2nc3c(n2O)cccn3 8F-310S Cc1ccc(cc1)c2nc3c(n2OC)cccn3 8F-311S C/N=C(\c1cccc(c1)[N+](=O)[O-])/Nc2ccc(cc2)Cl 8F-312S c1cc(cc(c1)C(F)(F)F)C(=N)Nc2cccc(c2)C(F)(F)F 8F-313S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(cc2)Cl 8F-314S Cc1ccc(cc1)c2nc3c(n2OCc4ccc(cc4Cl)Cl)cccn3 8F-315S Cc1ccc(cc1)c2nc3c(n2OCc4ccccc4Cl)cccn3 8F-316S C/N=C(\c1cccc(c1)[N+](=O)[O-])/Nc2ccc(c(c2)Cl)Cl 8F-317S Cc1ccc(cc1)c2nc3c(n2OCc4ccc(cc4)OC)cccn3 8F-318S COc1ccc(cc1)c2nc3c(n2OCc4ccccc4)cccn3 8F-319S COc1ccc(cc1)c2nc3c(n2OCc4ccccc4Cl)cccn3 8F-320S c1ccc2c(c1)c(nn(c2=O)Cc3ccc(cc3)Cl)CC(=O)O 8F-321S COc1ccc(cc1)c2nc3c(n2OCc4cccc(c4)C(F)(F)F)cccn3 8F-322S CCOc1ccc(cc1)NC(=O)c2cccn(c2=O)CC=C 8F-323S C=CCn1cccc(c1=O)C(=O)Nc2ccc(cc2)F 8F-324S Cc1ccc(cc1)NC(=O)c2cccn(c2=O)CC=C 8F-325S C=CCn1cccc(c1=O)C(=O)Nc2ccc(cc2)Cl 8F-326S COc1ccc(cc1Cl)NC(=O)c2cccn(c2=O)CC=C 8F-327S Cc1ccc(cc1Cl)NC(=O)c2cccn(c2=O)CC=C 8F-328S Cc1ccc(cc1C)NC(=O)c2cccn(c2=O)CC=C 8F-329S CSc1ccc(cc1)NC(=O)c2cccn(c2=O)CC=C 8F-330S C=CCn1cccc(c1=O)C(=O)Nc2ccc(c(c2)Cl)Cl 8F-331S CN(C)c1ccc(cc1)NC(=O)c2cccn(c2=O)CC=C 8F-332S CC(=O)Nc1ccc(cc1)NC(=O)c2cccn(c2=O)CC=C 8F-334S C/N=C(\c1cccc(c1)[N+](=O)[O-])/Nc2cccc(c2)C(F)(F)F 8F-335S Cc1ccc(cc1)COn2c3cccnc3nc2c4ccc(cc4)OC 8F-336S COc1ccc(cc1)c2nc3c(n2OCc4ccc(cc4)Br)cccn3 8F-337S COc1ccc(cc1)c2nc3c(n2OCc4cccc(c4)Cl)cccn3 8F-340S COc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-341S COc1ccccc1NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-342S COc1ccc(cc1OC)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-343S Cc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-344S Cc1ccccc1NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-345S Cc1ccc(cc1C)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-346S Cc1cccc(c1)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-347S CCc1cccc(c1NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F)CC 8F-348S Cc1ccc(c(c1)C)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-349S CC(C)(C)c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3cccc(c3)C(F)(F)F 8F-350S CCCn1cccc(c1=O)C(=O)Nc2ccc(cc2)OC 8F-352S COc1ccc(cc1)c2nc3c(n2OCc4ccc(cc4Cl)Cl)cccn3 8F-354S c1ccc(c(c1)CNc2c(cccn2)[N+](=O)[O-])Cl 8F-355S c1ccc(c(c1)c2nc3c(n2O)cccn3)Cl 8F-356S C/C=C/Cn1cccc(c1=O)C(=O)Nc2ccc(cc2)OC 8F-357S COc1ccc(cc1)NC(=O)c2cccn(c2=O)CC3CC3 8F-358S c1cc2c(nc1)nc(n2O)c3ccc(cc3Cl)Cl 8F-359S CC(=CCn1cccc(c1=O)C(=O)Nc2ccc(cc2)OC)C 8F-361S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2cccc(c2)C#N 8F-362S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2ccc(c(c2)Cl)Cl 8F-363S COc1ccc(cc1)NC(=O)c2cccn(c2=O)CC#C 8F-364S COc1ccc(cc1)NC(=O)c2cccn(c2=O)CC=C(Cl)Cl 8F-365S C/N=C(\c1cccc(c1)C(F)(F)F)/Nc2cccc(c2)C(F)(F)F 8F-366S Cc1ccc(cc1)Cn2cc(cc(c2=O)C(=O)Nc3ccccc3)Cl 8F-367S Cc1cc(cc(c1)Cn2cc(cc(c2=O)C(=O)Nc3ccccc3)Cl)C 8F-368S CCOC(=O)Cn1cc(cc(c1=O)C(=O)Nc2ccccc2)Cl 8F-369S C#CCn1cc(cc(c1=O)C(=O)Nc2ccccc2)Cl 8F-370S Cn1cc(cc(c1=O)C(=O)Nc2ccccc2)Cl 8F-371S C=CCn1cc(cc(c1=O)C(=O)Nc2ccccc2)Cl 8F-372S c1ccc(c(c1)COn2c3cccnc3nc2c4ccccc4Cl)Cl 8F-373S c1ccc(c(c1)c2nc3c(n2OCc4ccc(cc4Cl)Cl)cccn3)Cl 8F-374S c1ccc(c(c1)c2nc3c(n2OCc4c(cccc4Cl)Cl)cccn3)Cl 8F-375S c1ccc(c(c1)c2nc3c(n2OCc4ccc(c(c4)Cl)Cl)cccn3)Cl 8F-376S c1ccc(c(c1)c2nc3c(n2OCc4ccc(cc4)Br)cccn3)Cl 8F-377S c1cc(ccc1Nc2nc(c(s2)N)C#N)[N+](=O)[O-] 8F-900 Cc1ccnc(n1)N/C=C(/C(=O)OC)\NC(=O)c2ccccc2 8F-901 CCOC(=O)C(=CNc1cn(c(c1C(=O)c2ccccc2)C)Cc3ccc(cc3Cl)Cl)C(=O)OCC 8F-902 CCOC(=O)c1cnc2c(c(n(c2c1O)Cc3ccc(cc3Cl)Cl)C)C(=O)c4ccccc4 8F-903 CC(=O)N(/C=C/1\C(=O)OC(=N1)c2ccccc2)OCc3ccc(cc3)Cl 8F-904 c1ccc2c(c1)CCC(C2=O)(COC(=O)c3ccc(cc3Cl)Cl)COC(=O)c4ccc(cc4Cl)Cl 8F-905 c1ccc2c(c1)C(=O)C(CO2)(COC(=O)c3ccc(cc3Cl)Cl)COC(=O)c4ccc(cc4Cl)Cl 8F-906 c1ccc2c(c1)C(=O)C(CS2)(COC(=O)c3ccc(cc3Cl)Cl)COC(=O)c4ccc(cc4Cl)Cl 8F-907 COc1ccc(cc1)C(=O)OCC2(CSc3ccccc3C2=O)COC(=O)c4ccc(cc4)OC 8F-908 COc1ccc(cc1)C(=O)OCC2(COc3ccccc3C2=O)COC(=O)c4ccc(cc4)OC 8F-909 c1ccc2c(c1)C(=O)C3(COC(OC3)c4cccc(c4)C(F)(F)F)CS2 8F-910 COc1ccc(cc1)C2OCC3(CO2)CSc4ccccc4C3=O 8F-911 c1ccc2c(c1)C(=O)C3(CO2)COC(OC3)c4cccc(c4)C(F)(F)F 8F-912 COc1ccc(cc1)C(=O)OCC2(CCc3ccccc3C2=O)COC(=O)c4ccc(cc4)OC 8F-913 COC(=O)/C(=C\Nc1ncccn1)/NC(=O)c2ccccc2 8F-914 CC1=CC(=O)C23C1(C2)C(=O)C=C3C 8F-915 CC1=CC(=O)C2CC1C(=CC2=O)C 8F-916 c1cc(ccc1Nc2nc3c(ncnc3s2)N)[N+](=O)[O-] 8F-918 c1cc(cc(c1)Nc2nc(c(s2)N)C#N)C(F)(F)F 8F-920 Cc1cc2c(cc1C)N=C3C=C(C4CC3C(=N2)C=C4C)C 8F-923 Cc1c([nH][nH]c1=O)C 8F-924 CCOC(=O)c1cc([nH]c1Nc2ccc(cc2)Cl)C(=O)c3ccccc3 8F-925 c1ccc(cc1)CC(=O)NCCO 8F-926 c1ccc(cc1)CC(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl 8F-927 c1c(cnc(c1Cl)N2CCNCC2)C(F)(F)F 8F-928 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)N)C(F)(F)F 8F-929 c1cc(c(cc1Cl)Cl)C(=O)NCCO 8F-930 CN(C)/C=N/C(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 8F-931 Cc1cc(n(n1)CCO)C 8F-932 Cc1cccnc1N/C=C(\C(=O)OC)/NC(=O)c2ccccc2 8F-933 Cc1cc(n(n1)CCOc2c(cc(cn2)C(F)(F)F)Cl)C 8F-934 CN(C)c1nc2c(c(nn2c3ccc(cc3)OC)N)c(=O)o1 8F-935 Cc1ccc(cc1)CON/C=N/C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 8F-936 c1cc(ccc1CON/C=N/C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 8F-937 Cc1cc(nc(n1)/N=C/N(C)C)C 8F-938 c1c(cnc(c1Cl)N2CCC(=O)CC2)C(F)(F)F 8F-941 c1ccc(cc1)c2ncc3c(n2)CCN(C3)c4ccc(cc4)[N+](=O)[O-] 8F-942 CN(C)/C=C(\C#N)/C(=O)N/C=N/OCc1ccc(cc1)Cl 8F-943 CN(C)/C=N/Nc1c(cc(cn1)C(F)(F)F)Cl 8G-001 c1cc(c(c(c1)F)C#N)C(C#N)c2ccc(cc2)Cl 8G-002 CN(C)/C=C(\C=O)/c1c(c(no1)c2ccccc2Cl)C#N 8G-003 c1cc(ccc1SCS(=O)(=O)c2ccc(cc2)Cl)Cl 8G-004 COc1ccc(cc1)c2cnn(c2N)C3CCS(=O)(=O)C3 8G-005 COC(=O)CC(=O)/C(=N\Nc1cccc(c1)Cl)/C(=O)OC 8G-006 Cc1c(c(on1)/C(=C/N(C)C)/C=O)[N+](=O)[O-] 8G-007 COC(=O)C1=C(c2c(cccc2F)C(C1)(C#N)c3ccccc3)N 8G-008 c1cc(ccc1c2cnn(c2N)C3CCS(=O)(=O)C3)Cl 8G-009 c1cc(c(nc1)Cl)C(=O)N2CCOCC2 8G-010 c1cc(cc(c1)Cl)n2c(=O)cc(c(n2)C(=O)O)O 8G-011 c1c(cnc(c1C#N)O)c2c(cc(cn2)C(F)(F)F)Cl 8G-012 COC(=O)C1=C(c2c(cccc2F)C1(C#N)c3ccc(cc3)Cl)N 8G-013 c1cc(ccc1c2cnn(c2N)C3CCS(=O)(=O)C3)F 8G-014 c1ccc(cc1)/C=C/c2ccnn2C3CCS(=O)(=O)C3 8G-015 c1ccc(cc1)C(C#N)N2CCOCC2 8G-016 c1cc(sc1Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N 8G-019 COC(=O)CCCC(C#N)(c1ccccc1)c2ccccc2C#N 8G-020 c1c(cnc(c1Cl)c2cnc(nc2)O)C(F)(F)F 8G-021 c1cc(ccc1N2C(=O)C3C(C2=O)ON=C3c4c(cc(cn4)C(F)(F)F)Cl)Cl 8G-022 c1ccc(cc1)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 8G-023 c1ccc(cc1)C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3 8G-024 c1c(cnc(c1C#N)Cl)c2c(cc(cn2)C(F)(F)F)Cl 8G-026 COC(=O)c1c(cc(=O)n(n1)c2cccc(c2)Cl)O 8G-027 COC(=O)/C=C/CC(C#N)(c1ccccc1)c2ccccc2C#N 8G-028 c1c(cn2c(n1)c(cn2)C#N)C#N 8G-029 CSc1nc2ncc(cn2n1)C#N 8G-030 COC(=O)/C=C/C1=C(c2ccccc2C1(C#N)c3ccccc3)N 8G-031 c1cc(ccc1CC#N)Oc2c(cc(cn2)C(F)(F)F)Cl 8G-032 Cc1nc(c(s1)C(=O)NC(=O)NNc2ccc(cc2Cl)Cl)C(F)(F)F 8G-035 c1ccc(c(c1)C(C#N)N2CCOCC2)Cl 8G-038 c1ccc(cc1)C(C#N)(c2cccc(c2C#N)F)N3CCOCC3 8G-040 CCOC(=O)/C=C(\C(F)(F)F)/NC(=O)C(F)(F)F 8G-041 c1ccc(cc1)C(=O)c2cccc(c2C#N)F 8G-042 c1c(cnc(c1Cl)N2CCC(C2=O)C#N)C(F)(F)F 8G-046 c1cc(c(cc1Cl)F)N2C(=O)C=CC2=O 8G-047 c1c(cnc(c1Cl)CONC(=O)N/C=N/O)C(F)(F)F 8G-048 c1ccc(cc1)CN2C(=O)C3C(C2=O)ON=C3c4c(cc(cn4)C(F)(F)F)Cl 8G-049 CC(c1ccc(c(n1)O)C#N)Oc2ccc(cc2)Cl 8G-051 c1ccc(cc1)C(CCC#N)(C#N)c2c(cc(cn2)C(F)(F)F)Cl 8G-057 CN(C)/C=N/c1c(cc(cn1)C(F)(F)F)Cl 8G-059 Cc1c(c(n(n1)C)Cl)S(=O)(=O)N 8G-062 c1ccc2c(c1)c(c(nc2Br)N)c3ccc(cc3)Cl 8G-063 c1cc(c(c(c1)Cl)CON/C=N/OCc2c(cccc2Cl)Cl)Cl 8G-064 c1ccc(cc1)C2(CCC(=O)NC2=O)c3c(cc(cn3)C(F)(F)F)Cl 8G-065 CCOC(=O)/C=C(\C(F)(F)F)/NC(=O)c1ccc(cc1)C 8G-066 CCOC(=O)CSc1ccc(cn1)C(=O)Nc2ccc(cc2)OC 8G-301S CCOC(=O)CSc1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-302S CCOC(=O)C(C)Sc1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-303S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)F 8G-304S COc1cc(=O)n(nc1C(=O)O)c2cccc(c2)Cl 8G-305S CCOC(=O)c1c(cc(=O)n(n1)c2ccccc2)O 8G-306S c1cc(cc(c1)NC(=O)c2ccc(nc2)Cl)C(F)(F)F 8G-307S CCCSc1ccc(cn1)C(=O)Nc2ccc(cc2F)F 8G-308S CCOC(=O)C(C)Sc1ccc(cn1)C(=O)O 8G-309S CC(C)Sc1ccc(cn1)C(=O)Nc2ccc(cc2F)F 8G-310S CCOC(=O)c1c(cc(=O)n(n1)c2ccccc2)Cl 8G-312S CNC(=O)c1c(cc(=O)n(n1)c2cccc(c2)Cl)OC 8G-313S CC(C(=O)NO)N 8G-314S Cc1c(=O)n(cc(n1)c2ccccc2)O 8G-315S c1ccc(cc1)c2c(=O)n(cc(n2)c3cccc(c3)Cl)O 8G-317S Cc1c(=O)n(cc(n1)c2ccc(cc2)Cl)O 8G-318S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2)C(=O)OC)(F)F)Cl 8G-319S CCc1cccc(c1NC(=O)C(Oc2ccc(cc2C)Cl)(F)F)CC 8G-320S CCOC(=O)CSc1ccc(cn1)C(=O)Nc2ccc(cc2F)F 8G-323S CCCSc1ccc(cn1)C(=O)Nc2cccc(c2)C(F)(F)F 8G-324S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)O)Cl 8G-325S CCOC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)O 8G-329S c1ccc2c(c1)nc(s2)c3ccc(cc3)CSc4cccc(c4)C(F)(F)F 8G-333S c1ccc2c(c1)nc(s2)c3ccc(cc3)CSc4ccc(cc4)Br 8G-340S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)N 8G-341S CCOC(=O)c1c(cc(=O)n(n1)c2ccccc2)N(C)C 8G-342S CCOC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)Cl)Cl 8G-344S CCOC(=O)c1c(cc(=O)n(n1)c2cc(cc(c2)Cl)Cl)O 8G-345S c1cc(ccc1[N+](=O)[O-])Sc2ccc(cc2)Br 8G-348S CCOC(=O)c1c(cc(=O)n(n1)c2cc(cc(c2)Cl)Cl)Cl 8G-349S Cc1cc(ccc1OC(C(=O)Nc2ccc(c(c2)OC)OC)(F)F)Cl 8G-350S CCCSc1cc(=O)n(nc1C(=O)OCC)c2ccc(cc2)Cl 8G-352S c1cc(ccc1n2c(=O)cc(c(n2)C(=O)O)Cl)Cl 8G-353S c1cc(ccc1N)Sc2ccc(cc2)Br 8G-354S c1c(cc(cc1Cl)Cl)n2c(=O)cc(c(n2)C(=O)O)Cl 8G-356S CCCSc1cc(=O)n(nc1C(=O)O)c2ccc(cc2)Cl 8G-358S CCC(C)Sc1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-359S CCCSc1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-360S CC(C)S(=O)(=O)c1ccc(cn1)C(=O)Nc2ccc(cc2F)F 8G-361S COc1cccc(c1)C(=O)Nc2ccc(cc2)Sc3ccc(cc3)Br 8G-362S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)Sc3ccc(cc3)Br 8G-363S c1cc(cc(c1)Cl)C(=O)Nc2ccc(cc2)Sc3ccc(cc3)Br 8G-364S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)Sc3ccc(cc3)Br 8G-365S CCOC(=O)c1c(cc(=O)n(n1)c2ccccc2)SC(C)C 8G-367S CCOC(=O)c1c(cc(=O)n(n1)c2ccccc2)SC3CCCCC3 8G-368S COc1cccc(c1)C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)Br 8G-369S CCCCSc1cc(=O)n(nc1C(=O)OCC)c2ccccc2 8G-370S CCC(C)Sc1cc(=O)n(nc1C(=O)OCC)c2ccccc2 8G-371S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)Br 8G-372S c1cc(cc(c1)Cl)C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)Br 8G-373S Cc1cc(ccc1OC(C(=O)NC2CCCCC2)(F)F)Cl 8G-374S Cc1cc(ccc1OC(C(=O)O)(F)F)Cl 8G-375S Cc1ccc(cc1)Sc2ccc(cc2)N 8G-376S CCCSc1cc(=O)n(nc1C(=O)OCC)c2ccccc2 8G-377S CCCSc1cc(=O)n(nc1C(=O)O)c2ccccc2 8G-378S CCCCSc1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-379S Cc1cc(ccc1OC(C(=O)NC(C)C)(F)F)Cl 8G-380S CCC(C)S(=O)(=O)c1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-381S C=CCNC(=O)c1c(cc(=O)n(n1)c2ccccc2)Cl 8G-382S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)Nc3ccc(cc3)F)Cl 8G-383S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)Nc3cccc(c3)C(F)(F)F)Cl 8G-384S c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)Nc3ccc(cc3F)F)Cl 8G-385S CCCS(=O)(=O)c1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-386S CCOC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)F)O 8G-387S Cc1cc(ccc1OC(C(=O)Nc2cc(cc(c2)OC)OC)(F)F)Cl 8G-388S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)c3ccc(cc3)Cl 8G-389S CCCCS(=O)(=O)c1ccc(cn1)C(=O)Nc2ccc(cc2)Cl 8G-390S CCOC(=O)c1c(cc(=O)n(n1)c2ccc(cc2)F)Cl 8G-391S CCCSc1cc(=O)n(nc1C(=O)Nc2cccc(c2)Cl)c3ccccc3 8G-392S CCCSc1cc(=O)n(nc1C(=O)Nc2ccc(cc2)Cl)c3ccccc3 8G-393S c1ccc2c(c1)nc(s2)c3cccc(c3)CSc4ccc(cc4)Br 8G-395S c1ccc2c(c1)nc(s2)c3cccc(c3)CSc4ccc(cc4)Cl 8G-397S c1ccc2c(c1)nc(s2)c3cccc(c3)CSc4cccc(c4)Cl 8G-398S c1ccc2c(c1)nc(s2)c3cccc(c3)CSc4ccccc4Cl 8G-399S Cc1ccccc1SCc2cccc(c2)c3nc4ccccc4s3 8G-400S c1ccc2c(c1)nc(s2)c3cccc(c3)COc4cc(cc(c4)Cl)Cl 8G-402S c1ccc2c(c1)nc(s2)c3cccc(c3)COc4ccc(cc4Cl)Cl 8G-403S c1ccc2c(c1)nc(s2)c3cccc(c3)COc4cccc(c4Cl)Cl 8G-404S c1ccc2c(c1)nc(s2)c3cccc(c3)COc4ccc(cc4)F 8G-405S c1ccc2c(c1)nc(s2)c3cccc(c3)COc4ccc(cc4)Cl 8G-406S c1ccc2c(c1)nc(s2)c3ccc(cc3)COc4cc(cc(c4)Cl)Cl 8G-408S c1ccc(cc1)OCc2cccc(c2)c3nc4ccccc4s3 8G-410S CC(C)(C)c1ccc(cc1)OCc2cccc(c2)c3nc4ccccc4s3 8G-411S Cc1cccc(c1)SCc2cccc(c2)c3nc4ccccc4s3 8G-412S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)c3cccc(c3)C(F)(F)F 8G-413S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)C 8G-414S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl 8G-415S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)c3c(cccc3F)F 8G-416S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)c3ccc(cc3Cl)S(=O)(=O)C 8G-417S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)C(Cl)Cl 8G-418S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)c3ccc(cc3)F 8G-419S c1cc(ccc1n2c(=O)cc(c(n2)C(=O)O)Cl)F 8G-421S CCCSc1cc(=O)n(nc1C(=O)OCC)c2ccc(cc2)F 8G-422S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2)Br)(F)F)Cl 8G-423S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)c3cccc(c3)OC 8G-424S Cc1ccc(cc1)Sc2ccc(cc2)NC(=O)c3cccnc3Cl 8G-425S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)NC(=O)c3cccc(c3)C(F)(F)F 8G-426S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)NC(=O)c3c(cccc3F)F 8G-427S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)NC(=O)C 8G-428S CCCSc1cc(=O)n(nc1C(=O)O)c2ccc(cc2)F 8G-429S CC(=O)Nc1ccc(cc1)Sc2ccc(cc2)F 8G-430S c1cc(ccc1C(=O)Nc2ccc(cc2)Sc3ccc(cc3)F)F 8G-431S c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)Sc3ccc(cc3)F 8G-432S Cc1cccc(c1)NC(=O)CC(=O)Nc2cccc(c2)C 8G-902 Cc1ccc(c(c1)C)NC(=O)CC(=O)Nc2ccc(cc2C)C 8G-903 c1cc(ccc1C(F)(F)F)NC(=O)CC(=O)Nc2ccc(cc2)C(F)(F)F 8G-904 c1ccc(c(c1)NC(=O)CC(=O)Nc2ccccc2Cl)Cl 8G-905 c1cc(ccc1NC(=O)CC(=O)Nc2ccc(cc2)Cl)Cl 8G-906 c1c(cc(cc1Cl)Cl)NC(=O)CC(=O)Nc2cc(cc(c2)Cl)Cl 8G-908 C/[N+](=C\c1cc(ccc1OCC=C)Br)/[O-] 8G-909 Cc1cccc(c1)NC(=O)C(/C=N/OC)C(=O)N(C)c2cccc(c2)C 8G-910 c1ccc(c(c1)C(F)(F)F)NC(=O)CC(=O)Nc2ccccc2C(F)(F)F 8G-911 Cc1ccc(c(c1)C)NC(=O)C(/C=N/OC)C(=O)Nc2ccc(cc2C)C 8G-913 CN(C)C=C(C(=O)Nc1ccccc1Cl)C(=O)Nc2ccccc2Cl 8G-914 CO/N=C/C(C(=O)Nc1ccccc1Cl)C(=O)Nc2ccccc2Cl 8G-916 CO/N=C/C(C(=O)Nc1ccc(cc1)Cl)C(=O)Nc2ccc(cc2)Cl 8G-917 CO/N=C/C(C(=O)Nc1ccccc1C(F)(F)F)C(=O)Nc2ccccc2C(F)(F)F 8G-919 c1ccc(cc1)CON2C(=O)c3ccccc3C2=O 8G-920 CN([C@H]1c2c3ccccc3ccc2OC[C@H]1CO)C(=S)Nc4ccc(cc4)[N+](=O)[O-] 8G-921 CNC(=S)N(C)[C@H]1c2c3ccccc3ccc2OC[C@H]1CO 8G-922 c1ccc(c(c1)CON2C(=O)c3ccccc3C2=O)Cl 8G-923 c1c(cc(cc1C(F)(F)F)NC(=O)CC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F 8G-924 CN(C)C=C(C(=O)Nc1cc(cc(c1)Cl)Cl)C(=O)Nc2cc(cc(c2)Cl)Cl 8G-925 CN(C)C=C(C(=O)Nc1ccc(cc1)C(F)(F)F)C(=O)Nc2ccc(cc2)C(F)(F)F 8G-929 CO/N=C/C(C(=O)Nc1cc(cc(c1)Cl)Cl)C(=O)Nc2cc(cc(c2)Cl)Cl 8G-930 c1cc(c(cc1F)F)NC(=O)CC(=O)Nc2ccc(cc2F)F 8G-932 c1ccc(c(c1)CON)Cl.Cl 8G-933 CN(C)C=C(C(=O)Nc1ccc(cc1F)F)C(=O)Nc2ccc(cc2F)F 8G-934 CO/N=C/C(C(=O)Nc1ccc(cc1F)F)C(=O)Nc2ccc(cc2F)F 8G-935 c1ccc(cc1)CON=C2CCN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 8G-937 CN([C@H]1c2c3ccccc3ccc2OC[C@H]1CO)C(=S)Nc4cccc(c4)C(F)(F)F 8G-940 Cc1c(c(n(n1)C)OCC=C)C=O 8G-941 CCON1C(=O)c2ccccc2C1=O 8G-942 c1cc(ccc1CO[NH3+])C(=O)O.[Cl-] 8G-943 COC(=O)c1c2c(sc1N)CN(CC2)c3ccc4c(cc(nc4n3)C(F)(F)F)C(F)(F)F 8G-949 CN1C2c3c(cc(cc3OC)OC)OCC2CO1 8G-951 c1c(cnc(c1Cl)NCCNC(=O)/C=C/C(=O)O)C(F)(F)F 8G-954 c1cc(nc(c1)F)N2CCC(=O)CC2 8G-955 Cc1cccc(c1)NC(=O)C(/C=N/OC)C(=O)Nc2cccc(c2)C 8G-958 CN1[C@H]2c3c4ccccc4ccc3OC[C@H]2COC1c5cccc(c5)OC 8G-959 c1c(cnc(c1Cl)NCCN2C(=O)C=CC2=O)C(F)(F)F 8G-962 C[N+]1([C@H]2c3c4ccccc4ccc3OC[C@H]2CO1)Cc5ccccc5.[Br-] 8G-964 c1ccc(cc1)Cn2c(=O)ccn(c2=O)c3c(cc(cn3)C(F)(F)F)Cl 8G-965 c1c(cnc(c1Cl)NCCNC(=O)CCl)C(F)(F)F 8G-966 CCOC(=O)C1=NOC2C1C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 8G-967 c1ccc(cc1)N2CCN(CC2)C(=O)CCl 8G-969 c1ccc(cc1)N2CCN(CC2)C(=O)CON3C(=O)c4ccccc4C3=O 8G-970 c1cc(nc(c1)F)N2CCC3(CC2)N(CCO3)C(=S)Nc4ccc(cc4)[N+](=O)[O-] 8G-972 CN1C(C(CO1)S(=O)(=O)c2ccccc2)c3ccccc3 8G-973 CN(C=C(C(=O)Nc1ccc(cc1Cl)Cl)C(=O)Nc2ccc(cc2Cl)Cl)O 8G-974 Cc1ccc(c(c1)C)NC(=O)C(/C=[N+](/C)\[O-])C(=O)Nc2ccc(cc2C)C 8G-975 c1cc(ccc1NC(=O)CCl)Cl 8G-976 c1ccc(cc1)N2CCN(CC2)C(=O)CON.Cl 8G-977 C/[N+](=C\CC(=O)c1ccc(cc1)[N+](=O)[O-])/[O-] 8G-978 c1ccc2c(c1)C(=O)N(C2=O)OCC(=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl 8G-979 C/[N+](=C\CC(=O)/C=C\c1ccc(cc1)Cl)/[O-] 8G-980 CN1[C@H]2c3cc(ccc3OC[C@H]2CO1)Br 8G-981 CC(C(=O)C)Oc1ccsc1C(=O)OC 8H-003 c1c(c(nc(n1)N)C(F)(F)F)C#N 8H-006 COC(=O)C1CC(=O)NNC1 8H-007 c1ccc2c(c1)CCN3C2CC(=O)/C(=C\Nc4ccccc4Oc5c(cc(cn5)C(F)(F)F)Cl)/C3=O 8H-009 Cn1c(cnc1Sc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)Nc3ccc(cc3)Cl 8H-010 COC(=O)C1CC(=O)NN(C1)C(=O)Nc2ccc(cc2)Cl 8H-011 COC(=O)C1CC(=O)NN(C1)S(=O)(=O)c2ccc(cc2)Cl 8H-012 COC(=O)C1CC(=O)NN(C1)S(=O)(=O)C 8H-014 COC(=O)C1CC(=O)NN(C1)C(=O)N 8H-016 c1ccc2c(c1)C(=O)N(C2=O)OCc3ccc(cc3)C(F)(F)F 8H-019 COc1ccc(cc1)N\2C(=O)C=C(/C2=C/Nc3ccccc3Cl)c4ccc(cc4)F 8H-020 COc1ccc(cc1)N\2C(=O)C=C(/C2=C/Nc3cccc(c3)Cl)c4ccc(cc4)F 8H-021 COc1ccc(cc1)N\2C(=O)C=C(/C2=C/Nc3ccccc3)c4ccc(cc4)F 8H-022 c1cc(ccc1NC(=O)n2cc(c(n2)C(F)(F)F)C#N)Cl 8H-023 c1cc(ccc1CSc2ncc(c(n2)C(F)(F)F)C#N)Cl 8H-027 c1cc(ccc1CON)C(F)(F)F.Cl 8H-028 c1cc(ccc1C(C#N)(c2ccc(nn2)C(C#N)(c3ccc(cc3)Cl)N4CCOCC4)N5CCOCC5)Cl 8H-029 c1cc(ccc1CO/N=C/CC#N)Cl 8H-030 c1cn(ccc1=O)Nc2c(cc(cn2)C(F)(F)F)Cl 8H-031 c1cc(ccc1C(=O)c2ccc(nn2)C(=O)c3ccc(cc3)Cl)Cl 8H-032 c1ccc(cc1)S(=O)(=O)C(C2c3ccccc3CCN2C(=O)c4cccc(c4)C(F)(F)F)[N+](=O)[O-] 8H-034 CN(C)/C=C(\C#N)/C(=O)CCl 8H-035 CC(C(=O)/C=C/N(C)C)Oc1ccsc1C(=O)OC 8H-036 c1ccc(c(c1)C(C#N)N2CCOCC2)F 8H-037 CC(c1ccnc2n1nc(n2)N)Oc3ccsc3C(=O)OC 8H-040 CO/N=C/C(c1nnc(cc1)C(C#N)/C=N/OC)C#N 8H-041 c1ccc(c(c1)C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3)F 8H-042 c1ccc(c(c1)C(=O)c2c(cc(cn2)C(F)(F)F)Cl)F 8H-043 CC(C(=O)C)Oc1ccc(cc1)F 8H-045 CC(C(=O)/C=C\N(C)C)Oc1ccc(cc1)F 8H-046 CC(c1ccnc2n1nc(n2)N)Oc3ccc(cc3)F 8H-047 c1cc(ccc1N/C=C(/C#N)\C(=O)CCl)Cl 8H-048 CCOC(=O)C(=O)C(=CN(C)C)C#N 8H-049 CCOC(=O)c1c(cnn1c2c(cc(cn2)C(F)(F)F)Cl)C#N 8H-051 c1ccc2c(c1)CCN3C2CC(=O)C(C3=O)/C=N/OCc4ccc(cc4)C(F)(F)F 8H-052 c1c(c(n[nH]1)C(=O)NN)C#N 8H-053 CCOC(=O)c1c(cnn1c2cccc(c2)Cl)C#N 8H-054 CCOC(=O)C(=O)/C(=C/Nc1ccc(cc1)Cl)/C#N 8H-055 COc1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)no2 8H-056 c1cc(c(cc1Cl)Cl)C(C#N)N2CCOCC2 8H-057 CS(=O)(=O)CC(=O)c1ccc(cc1Cl)Cl 8H-301S CC1C(=O)N(C(=O)CS1=O)c2ccc(cc2)Br 8H-304S CC1C(=O)N(C(=O)CS1=O)c2ccc(cc2)OC 8H-305S Cc1ccc(cc1)N2C(=O)CS(=O)C(C2=O)C 8H-306S Cc1ccccc1N2C(=O)CS(=O)C(C2=O)C 8H-307S CS(=O)(=O)c1cnn(c1c2ccc(c(c2)Cl)Cl)c3ccccc3 8H-308S CS(=O)(=O)CC(=O)c1cccc(c1)C(F)(F)F 8H-309S COc1ccc(cc1)NC(=O)CS(=O)(=O)c2cccc(c2)Cl 8H-310S COc1ccc(cc1)NC(=O)CSc2ccc(cc2)F 8H-311S COc1ccc(cc1)NC(=O)CS(=O)c2ccc(cc2)F 8H-312S COc1ccc(cc1)NC(=O)CS(=O)(=O)c2ccc(cc2)F 8H-313S CS(=O)(=O)CC(=O)c1cc(c(cc1Cl)F)F 8H-314S CS(=O)(=O)c1cnn(c1c2ccc(c(c2)Cl)Cl)c3c(cc(cc3Cl)C(F)(F)F)Cl 8H-316S CS(=O)(=O)c1cnn(c1c2ccc(c(c2)Cl)Cl)c3c(cc(cc3Cl)Cl)Cl 8H-317S COc1ccc(cc1)NC(=O)CSc2ccccc2Cl 8H-318S COc1ccc(cc1)NC(=O)CSc2ccc(c(c2)Cl)Cl 8H-319S COc1ccc(cc1)NC(=O)CS(=O)c2ccccc2Cl 8H-320S COc1ccc(cc1)NC(=O)CS(=O)(=O)c2ccccc2Cl 8H-321S COc1ccc(cc1)NC(=O)CSCc2ccc(cc2)Cl 8H-322S COc1ccc(cc1)NC(=O)CS(=O)(=O)c2ccc(c(c2)Cl)Cl 8H-323S COc1ccc(cc1)NC(=O)CS(=O)c2ccc(c(c2)Cl)Cl 8H-324S COc1ccc(cc1)NC(=O)CSc2cccc(c2)C(F)(F)F 8H-325S COc1ccc(cc1)NC(=O)CS(=O)c2cccc(c2)C(F)(F)F 8H-326S COc1ccc(cc1)NC(=O)CS(=O)(=O)c2cccc(c2)C(F)(F)F 8H-327S CN(C)/C=C(/C(=O)c1cc(c(cc1Cl)F)F)\S(=O)(=O)C 8H-328S CN(C)/C=C(/C(=O)c1cccc(c1)[N+](=O)[O-])\S(=O)(=O)C 8H-329S COc1ccc(cc1)NC(=O)CSc2ccc(cc2)Br 8H-330S COc1ccc(cc1)NC(=O)CS(=O)c2ccc(cc2)Br 8H-331S COc1ccc(cc1)NC(=O)CS(=O)(=O)c2ccc(cc2)Br 8H-332S COc1ccc(cc1)NC(=O)CS(=O)Cc2ccc(cc2)Cl 8H-333S CS(=O)(=O)CC(=O)c1ccccc1Cl 8H-335S CN(C)/C=C(/C(=O)c1cc(c(cc1Cl)F)F)\S(=O)(=O)c2ccccc2 8H-336S c1ccc(cc1)C(=O)/C=N/Nc2ccc(cc2Cl)Cl 8H-338S CS(=O)(=O)c1cnn(c1c2ccc(c(c2)Cl)Cl)c3ccc(cc3Cl)C(F)(F)F 8H-339S CS(=O)(=O)c1cnn(c1c2ccc(c(c2)Cl)Cl)c3ccc(cc3)OC(F)(F)F 8H-340S CS(=O)(=O)c1cnn(c1c2ccc(c(c2)Cl)Cl)c3ccc(c(c3Cl)Cl)Cl 8H-341S CN(C)c1ncc(c(n1)c2ccc(cc2)Cl)S(=O)(=O)c3ccccc3 8H-342S C=CCNC(=O)CSc1ccc(cc1)F 8H-343S C=CCNC(=O)CSc1ccc(c(c1)Cl)Cl 8H-344S C=CCNC(=O)CSc1ccc(cc1)Br 8H-345S C=CCNC(=O)CSc1c(cccc1Cl)Cl 8H-346S C=CCNC(=O)CSc1ccccc1Cl 8H-347S CCOC(=O)CCn1ccnc1C 8H-348S C=CCNC(=O)CSCc1ccc(cc1)Cl 8H-349S COc1ccc(cc1)SCC(=O)NCC=C 8H-350S c1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2Cl)Cl)/CN3CCCCC3 8H-351S CC(C)N(C(C)C)C(=O)CSc1ccc(c(c1)Cl)Cl 8H-353S CN(Cc1ccccc1)C(=O)CSc2ccccc2Cl 8H-354S CC(C)N(C(C)C)C(=O)CS(=O)(=O)c1ccc(c(c1)Cl)Cl 8H-355S COc1ccc(cc1)NC(=O)CS(=O)(=O)Cc2ccc(cc2)Cl 8H-357S c1cc(cc(c1)NC(=O)CSCc2ccc(cc2)Cl)C(F)(F)F 8H-358S c1cc(cc(c1)NC(=O)CSc2cccc(c2)Cl)C(F)(F)F 8H-359S COc1ccc(cc1)SCC(=O)Nc2cccc(c2)C(F)(F)F 8H-360S c1cc(ccc1F)SCC(=O)N2CCOCC2 8H-361S c1cc(ccc1SCC(=O)N2CCOCC2)Br 8H-362S c1ccc(c(c1)SCC(=O)N2CCOCC2)Cl 8H-363S c1ccc(c(c1)NC(=O)CSc2cccc(c2)Cl)Cl 8H-364S COc1ccc(cc1)SCC(=O)Nc2ccccc2Cl 8H-365S c1ccc(c(c1)NC(=O)CSc2ccc(cc2)F)Cl 8H-366S c1cc(cc(c1)NC(=O)CS(=O)Cc2ccc(cc2)Cl)C(F)(F)F 8H-367S COc1ccc(cc1)S(=O)CC(=O)Nc2cccc(c2)C(F)(F)F 8H-369S c1cc(cc(c1)NC(=O)CS(=O)c2cccc(c2)Cl)C(F)(F)F 8H-370S c1cc(ccc1F)S(=O)(=O)CC(=O)N2CCOCC2 8H-371S c1cc(ccc1S(=O)(=O)CC(=O)N2CCOCC2)Br 8H-372S c1ccc(c(c1)S(=O)(=O)CC(=O)N2CCOCC2)Cl 8H-373S c1ccc(c(c1)NC(=O)CSc2ccc(c(c2)Cl)Cl)Cl 8H-374S c1ccc(c(c1)NC(=O)CSc2cccc(c2)C(F)(F)F)Cl 8H-375S c1ccc(c(c1)CSCC(=O)Nc2ccccc2Cl)Cl 8H-376S COc1ccc(cc1)S(=O)CC(=O)Nc2ccccc2Cl 8H-377S c1cc(c(cc1F)F)NC(=O)c2c(ccs2)OCc3ccc(cc3Cl)Cl 8H-402S c1cc(c(cc1NC(=O)c2c(ccs2)OCc3ccc(cc3Cl)Cl)Cl)Cl 8H-403S c1cc(ccc1NC(=O)c2c(ccs2)OCc3ccc(cc3Cl)Cl)Br 8H-405S c1cc(ccc1NC(=O)c2c(ccs2)OCc3ccc(cc3Cl)Cl)[N+](=O)[O-] 8H-406S c1cc(ccc1C(F)(F)F)NC(=O)c2c(ccs2)OCc3ccc(cc3Cl)Cl 8H-407S c1cc(c(cc1Cl)Cl)COc2ccsc2C(=O)Nc3ccc(cc3C(F)(F)F)Cl 8H-409S c1cc(c(cc1Cl)Cl)COc2ccsc2C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 8H-410S CCOC(=O)C1=C(N(c2ccccc2S1)Cc3ccc(cc3Cl)Cl)C 8H-414S CCOC(=O)C1=C(N(c2ccccc2S1)Cc3c(cccc3Cl)Cl)C 8H-421S CCOC(=O)C1=C(N(c2ccccc2S1)Cc3c(cccc3Cl)F)C 8H-422S CCOC(=O)C1=C(N(c2ccccc2S1)Cc3ccccc3Cl)C 8H-423S CCOC(=O)C1=C(N(c2ccccc2S1)Cc3cc(ccc3Cl)Cl)C 8H-424S COc1ccc(cc1)COc2ccsc2C(=O)OC 8H-426S COc1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(c(c3)Cl)Cl 8H-427S COc1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3)[N+](=O)[O-] 8H-428S COc1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3)Br 8H-429S c1ccc(cc1)C2C(=O)N(C(=O)CS2)c3ccc(cc3)Cl 8H-430S COc1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3)Cl 8H-434S COc1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3F)F 8H-437S COc1ccc(cc1)COc2ccsc2C(=O)Nc3ccc(cc3)C(F)(F)F 8H-438S COc1ccc(cc1)COc2ccsc2C(=O)Nc3cccc(c3)C(F)(F)F 8H-439S c1ccc(cc1)C(C(=O)Nc2ccc(cc2)Br)SCC(=O)O 8H-440S c1ccc(cc1)C2C(=O)N(C(=O)CS2)c3ccc(cc3)Br 8H-441S COc1ccc(cc1)COc2ccsc2C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 8H-446S CC1(CC(=C(C(=O)C1)CS(=O)(=O)c2ccccc2)O)C 8H-900 Cn1c(cnc1SCc2ccc(c(c2)Cl)Cl)CO 8H-901 Cc1c(c[nH]n1)C(=O)N(Cc2ccc(cc2)F)C(=O)NN(C)c3c(cc(cn3)C(F)(F)F)Cl 8H-902 c1cc(ccc1N2CCC3(CC2)OCC=CCO3)[N+](=O)[O-] 8H-903 c1ccc(cc1)S(=O)(=O)CC2C(=O)CCCC2=O 8H-904 c1ccc(cc1)S(=O)(=O)CC2C(=O)CC(CC2=O)c3ccc(cc3)Cl 8H-905 Cc1ccc(cc1)C(=O)OC2=C(C(=O)CC(C2)(C)C)CS(=O)(=O)c3ccccc3 8H-906 CC1(CC(=C(C(=O)C1)CS(=O)(=O)c2ccccc2)Cl)C 8H-907 c1cnoc1C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl 8H-909 c1ccc(cc1)S(=O)(=O)CC2=C(CC(CC2=O)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl 8H-911 CC1CN(C(ON1C)c2ccccc2)C(=O)NC3CCCCC3 8H-912 CC(=O)C1=NOC2C1COC3(CCN(CC3)c4ccc(cc4)[N+](=O)[O-])OC2 8H-913 Cc1c(cn(n1)C)C(=O)NC(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl 8H-915 CC(=O)CC(=O)c1cnn(c1O)c2ccccc2 8H-916 c1cc(c(cc1Cl)Cl)C2OCC=CCO2 8H-917 C1CN2CCN3C2C(N1)N4CCN5C4C3NCC5 8H-918 Cn1c(cnc1SCc2ccc(c(c2)Cl)Cl)CON3C(=O)c4ccccc4C3=O 8H-920 CC(=O)C(CS(=O)(=O)c1ccccc1)C(=O)C 8H-921 Cc1c(c(n(n1)c2ccccc2)C)CS(=O)(=O)c3ccccc3 8H-922 CC(=O)C(CS(=O)(=O)c1ccccc1)C(=O)C(F)(F)F 8H-923 Cc1c(c(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)C)CS(=O)(=O)c3ccccc3 8H-925 Cc1c(c(n[nH]1)C)CS(=O)(=O)c2ccccc2 8H-927 Cc1c(c(n(n1)C(=O)Nc2ccc(cc2)Cl)C)CS(=O)(=O)c3ccccc3 8H-928 CCOC(=O)c1c(c2ccccc2n1Cc3cccc(c3)Cl)n4cccc4 8H-929 CCOC(=O)c1c(c2ccccc2n1Cc3ccccc3Cl)n4cccc4 8H-930 CCOC(=O)c1c(c2ccccc2n1Cc3ccc(cc3)Cl)n4cccc4 8H-931 CCOC(=O)c1c(c2ccccc2n1Cc3ccccc3)n4cccc4 8H-932 CCOC(=O)c1c(c2ccccc2n1c3c(cc(cn3)C(F)(F)F)Cl)n4cccc4 8H-935 CCOC(=O)c1c(c2ccccc2[nH]1)N/C=C(/C#N)\C(=O)NC(=O)OCC 8H-936 CCOC(=O)c1c(c2ccccc2[nH]1)n3cc(c(=O)[nH]c3=O)C#N 8H-937 CCOC(=O)c1c(c2ccccc2n1Cc3ccc(cc3)C)n4cc(c(=O)n(c4=O)Cc5ccc(cc5)C)C#N 8H-938 CC(=O)c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 8H-939 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)O 8H-940 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)Nc4ccc(cc4)OC(F)(F)F 8H-942 COC(=O)Cc1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 8H-944 CC(=O)c1cn(c2c1cccc2)C 8H-945 CN(C)/C=C/C(=O)c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl 8H-946 CN(C)/C=C/C(=O)c1c[nH]c2c1cccc2 8H-947 Cc1c(c(n(n1)S(=O)(=O)c2ccc(cc2)Cl)C)CS(=O)(=O)c3ccccc3 8H-948 c1c(cc(c(c1[N+](=O)[O-])N2CCC3(CC2)OCC=CCO3)[N+](=O)[O-])C(F)(F)F 8H-949 c1ccc2c(c1)c(cn2c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)NN 8H-950 CN(C)/C=C(/c1cn(c2c1cccc2)c3c(cc(cn3)C(F)(F)F)Cl)\C(=O)OC 8H-951 c1cnc(nc1)N2CCC3(CC2)OCC=CCO3 8H-952 c1cc(ccc1C(=O)O)NCCN.Cl.Cl 8H-953 Cc1c(c(n(n1)C(=O)c2ccccc2)C)CS(=O)(=O)c3ccccc3 8H-954 c1ccc(cc1)NC(=S)NNC(=O)Cc2cn(c3c2cccc3)c4c(cc(cn4)C(F)(F)F)Cl 8H-955 CCOC(=O)c1c(c2ccccc2n1C)n3cc(c(=O)n(c3=O)C)C#N 8H-956 CCOC(=O)c1c(nc(s1)c2ccc(cc2)Cl)C 8J-003 CCOC(=O)/N=C/c1c(cc(cn1)C(F)(F)F)Cl 8J-004 CCOC(=O)C(=CNc1ccc(cc1C(=O)c2ccccc2)Cl)C(=O)OCC 8J-006 c1ccnc(c1)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 8J-010 c1cc(cnc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)O 8J-011 CCOC(=O)c1cnc2c(c1O)cc(cc2C(=O)c3ccccc3)Cl 8J-012 CCOC(=O)c1cnc2ccc(cc2c1c3ccccc3)Cl 8J-013 CCOC(=O)c1cnc2c(c1Cl)cc(cc2C(=O)c3ccccc3)Cl 8J-014 CCOC(=O)C(=CNc1ccc(cc1)C(=O)C)C(=O)OCC 8J-015 c1ccnc(c1)c2nnc3n2cc(cc3Cl)C(F)(F)F 8J-017 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 8J-018 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl 8J-019 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)NCC=C 8J-020 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)NNc3cccc(n3)Cl 8J-022 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)N 8J-023 c1cc(cnc1)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 8J-024 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)N3CCN(CC3)c4ccccc4 8J-025 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 8J-026 c1cc(cnc1)c2nnc3n2cc(cc3Cl)C(F)(F)F 8J-028 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)/N=C/N(C)C 8J-029 c1cc(ccc1NC=C(C(=O)C(F)(F)F)C(=O)C(F)(F)F)Oc2c(cc(cn2)C(F)(F)F)Cl 8J-030 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)c2cc([nH]c2)C(=O)N/C=N/OC 8J-031 COC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3ccccn3 8J-032 c1c(cnc(c1Cl)Cn2cncn2)C(F)(F)F 8J-033 c1ccnc(c1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)O 8J-035 c1cnccc1C(C#N)(c2c(cc(cn2)C(F)(F)F)Cl)N3CCOCC3 8J-037 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)O 8J-038 c1cc(sc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)N 8J-040 CCOC(=O)C(=CNc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl)C(=O)OCC 8J-041 c1cc(sc1)c2csc3c2ncc(c3)C(F)(F)F 8J-044 CCOC(=O)c1cnc2ccc(cc2c1O)Oc3c(cc(cn3)C(F)(F)F)Cl 8J-045 COCCCNC(=O)CCc1c(cc(cn1)C(F)(F)F)Cl 8J-047 c1ccc(cc1)C(=O)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl 8J-048 c1ccc(cc1)C(=O)c2nnc3n2cc(cc3Cl)C(F)(F)F 8J-049 CCOC(=O)c1cnc2ccc(cc2c1Cl)Oc3c(cc(cn3)C(F)(F)F)Cl 8J-051 Cc1ccc(cc1)SCC(=O)c2cc(c(c(c2)C)OC(=O)N(C)C)C 8J-301S Cc1ccc(cc1)SCC(=O)c2cc(c(c(c2)C)OC(=S)N(C)C)C 8J-302S c1ccc2c(c1)[nH]c(n2)CSc3ccc(cc3)Cl 8J-305S Cc1ccc(cc1)SCc2nc3ccccc3n2CC(=O)Nc4ccc(cc4)OC 8J-306S Cc1ccc(cc1)SCc2nc3ccccc3n2CC(=O)Nc4ccc(cc4)Cl 8J-307S Cc1ccc(cc1)SCc2nc3ccccc3n2CC(=O)Nc4c(cccc4C)C 8J-308S Cc1ccc(cc1)S(=O)(=O)Cc2nc3ccccc3n2CC(=O)Nc4ccc(cc4)OC 8J-309S CN(c1ccccc1)C(=O)Cn2c3ccccc3nc2CSc4ccc(cc4)Cl 8J-310S c1ccc(cc1)SCc2[nH]c3ccccc3n2 8J-311S CN(c1ccccc1)C(=O)Cn2c3ccccc3nc2CS(=O)(=O)c4ccc(cc4)Cl 8J-312S CN(c1ccccc1)C(=O)Cn2c3ccccc3nc2CS(=O)c4ccc(cc4)Cl 8J-313S Cc1cc(cc(c1O)C)C(=O)CSc2ccc(cc2)F 8J-314S Cc1cc(cc(c1O)C)C(=O)CS(=O)(=O)c2ccc(cc2)F 8J-317S Cc1cc(cc(c1O)C)C(=O)CS(=O)c2ccc(cc2)F 8J-318S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CSc2ccc(cc2)F 8J-319S Cc1cc(cc(c1OC(=S)N(C)C)C)C(=O)CSc2ccc(cc2)F 8J-320S c1ccc(cc1)SCc2nc3ccccc3n2CC(=O)Nc4cccc(c4)C(F)(F)F 8J-321S c1ccc(cc1)SCc2nc3ccccc3n2CC(=O)Nc4ccc(cc4Cl)Cl 8J-322S Cc1cc(cc(c1O)C)C(=O)CSc2ccc(cc2)OC 8J-324S Cc1cc(cc(c1O)C)C(=O)CS(=O)(=O)c2ccc(cc2)OC 8J-326S Cc1cc(cc(c1O)C)C(=O)CS(=O)c2ccc(cc2)OC 8J-327S Cc1cc(cc(c1O)C)C(=O)CS(=O)(=O)c2ccccc2 8J-328S Cc1cc(cc(c1O)C)C(=O)CS(=O)c2ccccc2 8J-329S c1ccc(cc1)SCc2nc3ccccc3n2CC(=O)Nc4ccccc4F 8J-330S c1ccc(cc1)NC(=O)Cn2c3ccccc3nc2CSc4ccccc4 8J-331S Cc1ccc(cc1Cl)NC(=O)Cn2c3ccccc3nc2CSc4ccccc4 8J-332S COc1ccc(cc1)NC(=O)Cn2c3ccccc3nc2CSc4ccccc4 8J-333S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)C 8J-334S c1ccc(cc1)NC(=O)Cn2c3ccccc3nc2CS(=O)c4ccccc4 8J-335S COc1ccc(cc1)NC(=O)Cn2c3ccccc3nc2CS(=O)c4ccccc4 8J-336S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4cccc(c4)Cl 8J-337S c1ccc(cc1)NC(=O)Cn2c3ccccc3nc2CSc4ccc(cc4)Cl 8J-338S c1ccc2c(c1)nc(n2CC(=O)Nc3ccc(cc3)Cl)CSc4ccc(cc4)Cl 8J-339S Cc1cc(cc(c1OC(=S)N(C)C)C)C(=O)CSc2ccc(cc2)OC 8J-340S Cc1ccc(cc1)S(=O)(=O)CC(=O)c2cc(c(c(c2)C)OC(=O)N(C)C)C 8J-341S Cc1ccc(cc1)S(=O)CC(=O)c2cc(c(c(c2)C)OC(=O)N(C)C)C 8J-342S c1ccc2c(c1)nc(n2CC(=O)Nc3ccc(cc3Cl)Cl)CSc4ccc(cc4)Cl 8J-344S Cc1cccc(c1NC(=O)Cn2c3ccccc3nc2CSc4ccc(cc4)Cl)C 8J-345S c1ccc2c(c1)nc(n2CC(=O)Nc3cccc(c3)C(F)(F)F)CSc4ccc(cc4)Cl 8J-346S c1ccc2c(c1)[nH]c(n2)CSc3ccccc3Cl 8J-347S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CSc2ccccc2 8J-348S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CS(=O)(=O)c2ccccc2 8J-349S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CS(=O)c2ccccc2 8J-350S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)Cl)C 8J-351S Cc1cc(nc(c1S(=O)(=O)c2ccccc2)OC)C 8J-352S CN(c1ccccc1)C(=O)Cn2c3ccccc3nc2CSc4ccccc4Cl 8J-353S c1ccc(cc1)NC(=O)Cn2c3ccccc3nc2CSc4ccccc4Cl 8J-354S c1ccc2c(c1)nc(n2CC(=O)Nc3cccc(c3)C(F)(F)F)CSc4ccccc4Cl 8J-355S Cc1ccc(cc1Cl)NC(=O)Cn2c3ccccc3nc2CSc4ccccc4Cl 8J-356S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4c(cccc4Cl)Cl 8J-357S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4c(cccc4Cl)F 8J-358S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4cccc(c4)C(F)(F)F 8J-359S Cc1cc2c(cc1C)n(c(n2)c3cccnc3Cl)Cc4cccc(c4)OC 8J-360S C=CCSc1ncc(cn1)c2cccc(c2)C(F)(F)F 8J-501S CCOC(=O)CSc1ncc(cn1)c2cccc(c2)C(F)(F)F 8J-502S CCOC(=O)C(C)Sc1ncc(cn1)c2cccc(c2)C(F)(F)F 8J-503S Cn1c(=O)cc(nc1SCc2ccc(cc2)Cl)C(F)(F)F 8J-504S Cn1c(=O)cc(nc1SCc2cccc(c2)Cl)C(F)(F)F 8J-505S Cn1c(=O)cc(nc1SCc2ccccc2Cl)C(F)(F)F 8J-506S Cn1c(=O)cc(nc1SCc2ccccc2)C(F)(F)F 8J-507S Cn1c(=O)cc(nc1SCc2ccc(cc2Cl)Cl)C(F)(F)F 8J-508S Cn1c(=O)cc(nc1SCc2c(cccc2Cl)Cl)C(F)(F)F 8J-509S Cn1c(=O)cc(nc1SCc2nc3c(cccc3s2)F)C(F)(F)F 8J-510S CC(C)(C)c1ccc(cc1)CSc2nc(cc(=O)n2C)C(F)(F)F 8J-511S Cc1ccc(cc1)CSc2nc(cc(=O)n2C)C(F)(F)F 8J-512S Cc1cccc(c1)CSc2nc(cc(=O)n2C)C(F)(F)F 8J-513S Cc1ccccc1CSc2nc(cc(=O)n2C)C(F)(F)F 8J-514S Cn1c(=O)cc(nc1SCc2ccc(cc2)F)C(F)(F)F 8J-515S Cn1c(=O)cc(nc1SCc2ccccc2F)C(F)(F)F 8J-516S c1cc(cc(c1)C(F)(F)F)c2cnc(nc2)SCc3ccc(cc3)Cl 8J-518S c1cc(cc(c1)C(F)(F)F)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F 8J-519S Cn1c(=O)cc(nc1SCc2ccc(cc2)C(=O)OC)C(F)(F)F 8J-520S Cn1c(=O)cc(nc1SCc2ccccc2C#N)C(F)(F)F 8J-521S Cn1c(=O)cc(nc1SCc2cccc(c2)C#N)C(F)(F)F 8J-522S Cn1c(=O)cc(nc1SCc2cccc(c2)C(F)(F)F)C(F)(F)F 8J-523S Cn1c(=O)cc(nc1SCc2c(cccc2Cl)F)C(F)(F)F 8J-524S c1ccc(cc1)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F 8J-525S Cc1cccc(c1)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F 8J-526S c1cc(cc(c1)C(F)(F)F)c2cnc(nc2)SCc3c(cccc3Cl)Cl 8J-527S COc1cccc(c1)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F 8J-529S c1cc(cc(c1)C(F)(F)F)c2cnc(nc2)SCc3ccc(c(c3)Cl)Cl 8J-530S CC(=C)CSc1ncc(cn1)c2cccc(c2)C(F)(F)F 8J-532S CC(C)CSc1ncc(cn1)c2cccc(c2)C(F)(F)F 8J-533S c1cc(cc(c1)F)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F 8J-535S Cn1c(=O)cc(nc1SC)C(F)(F)F 8J-537S CCOC(=O)CSc1nc(cc(=O)n1C)C(F)(F)F 8J-538S Cn1c(=O)cc(nc1SCC=C)C(F)(F)F 8J-539S c1ccc(c(c1)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F)Cl 8J-541S c1cc(cc(c1)Cl)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F 8J-542S c1cc(cc(c1)C(F)(F)F)c2cnc(nc2)SCc3ccc(cc3)F 8J-543S Cc1ccc(cc1)CSc2ncc(cn2)c3cccc(c3)C(F)(F)F 8J-544S COc1cccc(c1)C(=O)CC(c2ccc(cc2)Cl)C(=O)O 8J-550S Cc1cc(cc(c1O)C)C(=O)CSc2ccccc2 8J-552S c1ccc(cc1)CNc2c(cccn2)c3nc4cc(ccc4o3)Cl 8J-553S c1cc(cc(c1)C(F)(F)F)CNc2c(cccn2)c3nc4cc(ccc4o3)Cl 8J-554S Cc1ccc(cc1)CNc2c(cccn2)c3nc4cc(ccc4o3)Cl 8J-556S c1cc(c(nc1)NCc2ccc(cc2)Cl)c3nc4cc(ccc4o3)Cl 8J-557S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)Cl)CSC2 8J-559S COc1cccc(c1)Cn2c3ccccc3nc2c4ccc[nH]c4=O 8J-560S CC(C)(C)C(=O)NNC(=S)N 8J-562S CN(C)C(=O)c1ccc(cc1)n2cc(cn2)c3cccc(c3)C(F)(F)F 8J-565S c1cc(cc(c1)C(F)(F)F)c2cnn(c2)c3ccc(cc3)S(=O)(=O)N 8J-566S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)Cl)CS(=O)C2 8J-578S COC(=O)c1c2n(c(c1C(=O)OC)c3ccccc3)CSC2 8J-581S c1cc(cc(c1)C(F)(F)F)c2cnn(c2)c3cccc(c3)C(=O)O 8J-583S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)Cl)CS(=O)(=O)C2 8J-586S c1ccc(cc1)CO/N=C/CC(=O)c2c(ccs2)Cl 8J-900 c1cc(ccc1n2c(ccn2)c3c(ccs3)Cl)Cl 8J-902 COC(=O)C1CSC(N1C(=O)CN2CCOCC2)C(=O)OC 8J-903 C/C(=C/C(=O)OCc1ccccc1)/N2CCCC2 8J-904 COC(=O)C1N2C(CS1)C(=O)N(CC2=O)CCc3ccccc3 8J-906 CN1CCN(CC1)CC(=O)N2C(CSC2C(=O)OC)C(=O)OC 8J-907 C=CC(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 8J-908 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)C2CC(N(O2)c3ccccc3)c4ccccc4 8J-909 COC(=O)C1N2C(CS1)C(=O)N(CC2=O)Cc3ccc(cc3)Cl 8J-910 CC(=O)c1c(con1)C(=O)c2c(ccs2)Cl 8J-911 CCOC(=O)c1c(con1)C(=O)c2c(ccs2)Cl 8J-912 COC(=O)C1N2C(CS1)C(=O)N(CC2=O)Cc3ccccc3 8J-913 COC(=O)C1N2C(CS1)C(=O)N(CC2=O)CCc3ccccn3 8J-914 c1ccc(cc1)C2CC(ON2c3ccccc3)C(=O)N4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 8J-915 CCOC(=O)/C=C(\C)/NCCNc1c(cc(cn1)C(F)(F)F)Cl 8J-918 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C3C4c5ccccc5C(C3C2=O)(c6c4cccc6)O 8J-919 CCOC(=O)C1=C(N(C(=O)CC1)CCNc2c(cc(cn2)C(F)(F)F)Cl)C 8J-920 COC(=O)c1c(onc1c2ccccc2)/C=C/c3cnc(c4c3onc4c5ccccc5)Oc6ccc(cc6)Cl 8K-003 c1cc(sc1)CC(C#N)(C#N)c2c(cc(cn2)C(F)(F)F)Cl 8K-006 c1cc(sc1)CCc2c(cc(cn2)C(F)(F)F)Cl 8K-007 COc1ccc(cc1)S(=O)(=O)N(CC(=O)N2CCCC2)c3ccccc3 8K-301S Cc1ccc(cc1)c2cc3ccccc3nc2Sc4ccc(cc4)C 8K-303S Cc1ccc(cc1)c2cc3ccccc3nc2Sc4ccc(cc4)Cl 8K-304S Cc1ccc(cc1)c2cc3ccccc3nc2Sc4c(cccc4Cl)Cl 8K-305S Cc1ccc(cc1)c2nc(c(nn2)C)Sc3ccc(cc3)OC 8K-306S Cc1ccc(cc1)c2cc3ccccc3nc2Sc4ccc(cc4)F 8K-307S Cc1ccc(cc1)c2cc3ccccc3nc2Sc4cccc(c4)Cl 8K-309S Cc1ccc(cc1)c2cc3ccccc3nc2N4CCOCC4 8K-310S c1ccc(cc1)c2cc3ccccc3nc2N4CCOCC4 8K-311S CCOC(=O)CN(c1ccccc1)S(=O)(=O)c2ccccc2 8K-312S CN(C)C(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(cc2)Cl 8K-313S C=CCNC(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(cc2)Cl 8K-314S c1ccc(cc1)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl 8K-316S c1ccc(cc1)N(CC(=O)Nc2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)Cl 8K-317S c1ccc2c(c1)cc(c(n2)Sc3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl 8K-320S Cc1ccc(cc1)c2cc3ccccc3nc2Sc4cccc(c4)C(F)(F)F 8K-321S c1ccc2c(c1)cc(c(n2)N3CCCCC3)c4ccc(cc4)Cl 8K-323S Cc1ccc(cc1)c2cc3ccccc3nc2N4CCCCC4 8K-324S Cc1ccc(cc1)c2nc(c(nn2)c3ccccc3)Sc4ccc(cc4)Br 8K-325S c1ccc(cc1)N(CC(=O)O)S(=O)(=O)c2ccccc2 8K-326S c1ccc(cc1)N(CC(=O)O)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F 8K-327S CCOC(=O)CN(c1ccccc1)S(=O)(=O)c2cc(ccc2Cl)Cl 8K-328S CCOC(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(cc2)F 8K-329S Cc1ccc(cc1)c2nc(c(nn2)c3ccccc3)N4CCOCC4 8K-330S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)O 8K-335S c1ccc(cc1)c2cc3ccccc3nc2N4CCCC4 8K-336S Cc1ccc(cc1)c2cc3ccccc3nc2N4CCCC4 8K-337S c1ccc2c(c1)cc(c(n2)N3CCCC3)c4ccc(cc4)Cl 8K-338S c1ccc(cc1)N(CC(=O)O)S(=O)(=O)c2cc(ccc2Cl)Cl 8K-340S CC1CN(CC(O1)C)c2c(cc3ccccc3n2)c4ccccc4 8K-341S CC1CN(CC(O1)C)c2c(cc3ccccc3n2)c4ccc(cc4)Cl 8K-342S Cc1ccc(cc1)c2cc3ccccc3nc2N4CC(OC(C4)C)C 8K-343S c1ccc(cc1)N(CC(=O)Nc2ccc(cc2)F)S(=O)(=O)c3ccccc3 8K-346S c1ccc(cc1)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3ccccc3 8K-347S c1ccc(cc1)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)S(=O)(=O)c3ccccc3 8K-348S c1ccc(cc1)NC(=O)CN(c2ccccc2)S(=O)(=O)c3ccccc3 8K-349S c1ccc(cc1)N(CC(=O)Nc2ccc(cc2F)F)S(=O)(=O)c3ccccc3 8K-350S c1ccc(cc1)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)F 8K-351S c1ccc(cc1)NC(=O)Cc2cccc(c2)C(F)(F)F 8K-352S COC(=O)c1ccccc1Sc2c(cc3ccccc3n2)c4ccc(cc4)Cl 8K-354S c1ccc(cc1)N(CC(=O)N2CCCC2)S(=O)(=O)c3ccccc3 8K-357S C=CCNC(=O)CN(c1ccccc1)S(=O)(=O)c2ccccc2 8K-358S CN(C)C(=O)CN(c1ccccc1)S(=O)(=O)c2ccccc2 8K-359S c1cnccc1/C(=N\O)/N 8K-361S c1ccnc(c1)c2nc(on2)c3ccc(cc3)F 8K-367S c1ccc(cc1)c2nc(no2)c3ccccn3 8K-368S c1ccnc(c1)c2nc(on2)c3ccc(cc3Cl)Cl 8K-369S c1ccnc(c1)c2nc(on2)c3c(cccc3F)F 8K-370S c1ccc(c(c1)c2nc(no2)c3ccccn3)Cl 8K-371S c1ccnc(c1)c2nc(on2)c3cc(cc(c3)Cl)Cl 8K-372S CN(C)C(=O)CN(c1ccccc1)S(=O)(=O)c2cc(ccc2Cl)Cl 8K-374S c1ccc(cc1)N(CC(=O)N2CCCC2)S(=O)(=O)c3cc(ccc3Cl)Cl 8K-375S c1ccc(cc1)N(CC(=O)Nc2ccc(cc2F)F)S(=O)(=O)c3cc(ccc3Cl)Cl 8K-376S c1ccc(cc1)N(CC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)c3cc(ccc3Cl)Cl 8K-377S c1ccc(cc1)N(CC(=O)O)S(=O)(=O)c2ccc(cc2Cl)Cl 8K-378S c1ccc(cc1)N(CC(=O)O)S(=O)(=O)c2ccccc2Cl 8K-379S c1ccc2c(c1)cc(c(n2)Sc3ccc(cc3)Cl)c4cccc(c4)C(F)(F)F 8K-381S c1ccc2c(c1)cc(c(n2)Sc3ccccc3Cl)c4cccc(c4)C(F)(F)F 8K-382S c1ccc2c(c1)cc(c(n2)Sc3c(cccc3Cl)Cl)c4cccc(c4)C(F)(F)F 8K-383S c1ccc2c(c1)cc(c(n2)Sc3cccc(c3)C(F)(F)F)c4cccc(c4)C(F)(F)F 8K-384S COC(=O)c1ccccc1Sc2c(cc3ccccc3n2)c4cccc(c4)C(F)(F)F 8K-385S CN(C)C(=O)CN(c1ccccc1)S(=O)(=O)c2ccc(cc2)F 8K-386S c1ccc(cc1)N(CC(=O)N2CCCC2)S(=O)(=O)c3ccc(cc3)F 8K-387S c1ccc(cc1)N(CC(=O)N2CCOCC2)S(=O)(=O)c3ccc(cc3)F 8K-388S c1ccc(cc1)N(CC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)F 8K-389S c1ccc(cc1)N(CC(=O)Nc2cc(cc(c2)Cl)Cl)S(=O)(=O)c3ccc(cc3)F 8K-390S COc1ccc(cc1)NC(=O)CN(c2ccccc2)S(=O)(=O)c3ccc(cc3)F 8K-391S c1ccc(cc1)N(CC(=O)N2CCOCC2)S(=O)(=O)c3ccccc3 8K-392S COc1ccc(cc1)NC(=O)CN(c2ccccc2)S(=O)(=O)c3ccccc3 8K-393S c1ccc(cc1)CNC(=O)CN(c2ccccc2)S(=O)(=O)c3ccccc3 8K-394S c1ccc2c(c1)cc(c(n2)N3CCOCC3)c4cccc(c4)C(F)(F)F 8K-396S c1ccc2c(c1)cc(c(n2)N3CCCC3)c4cccc(c4)C(F)(F)F 8K-398S c1ccc2c(c1)cc(c(n2)Sc3ccc(cc3)F)c4cccc(c4)C(F)(F)F 8K-400S c1ccc2c(c1)cc(c(n2)Sc3ccc(cc3)Br)c4cccc(c4)C(F)(F)F 8K-401S c1cc(ccc1C(=O)c2cnc3n2cc(cc3)Cl)Cl 8K-404S c1ccnc(c1)c2nc(on2)c3cccc(c3)Cl 8K-406S c1ccnc(c1)c2nc(on2)c3cccc(c3)C(F)(F)F 8K-407S Cc1ccc2ncc(n2c1)C(=O)c3ccc(cc3)Cl 8K-408S Cc1ccc2ncc(n2c1)C(=O)c3ccc(cc3)OC 8K-409S c1ccc(cc1)Oc2c(cc3ccccc3n2)c4ccc(cc4)Cl 8K-410S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)NCC=C 8K-412S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)NC(C)(C)C 8K-413S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)N3CCOCC3 8K-414S c1ccc(cc1)S(=O)(=O)Nc2nnc(s2)C(F)(F)F 8K-417S Cc1ccn2c(c1)ncc2C(=O)c3ccc(cc3)Cl 8K-420S Cc1ccc(cc1)S(=O)(=O)Nc2nnc(s2)C(F)(F)F 8K-421S c1cc(ccc1F)S(=O)(=O)Nc2nnc(s2)C(F)(F)F 8K-422S c1cc(ccc1S(=O)(=O)Nc2nnc(s2)C(F)(F)F)Cl 8K-423S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccc(cc3)Br 8K-430S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)Sc3ccccc3C(=O)OC 8K-431S c1cc(cc(c1)S(=O)(=O)Nc2nnc(s2)C(F)(F)F)C(F)(F)F 8K-436S CN(c1c(nns1)c2ccccc2)N 8K-441S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)Oc3cc(c(cc3Cl)Cl)Cl 8K-444S Cc1c(nc(nn1)c2cccc(c2)C(F)(F)F)Oc3ccc(cc3)C#N 8K-445S Cc1ccc(cc1)c2nc(c(nn2)C)N3CCOCC3 8K-447S c1ccc(cc1)c2nc(cc(n2)Cl)CSc3ccccc3 8K-501S c1ccc(cc1)c2nc(cc(n2)Sc3ccc(cc3)Br)CSc4ccccc4 8K-503S c1ccc(cc1)CSc2ccccc2c3nnc(o3)c4ccccc4 8K-509S c1ccc(c(c1)C(=O)O)SCc2ccc(cc2)Cl 8K-511S Cc1ccc(cc1)CSc2ccccc2C(=O)O 8K-513S c1ccc(cc1)c2nnc(o2)c3ccccc3SCc4ccc(cc4)Cl 8K-516S Cc1ccc(cc1)C(=O)NNC(=O)c2ccccc2SCc3ccc(cc3)Cl 8K-517S Cc1ccc(cc1)c2nnc(o2)c3ccccc3SCc4ccc(cc4)Cl 8K-518S c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)SCc4ccc(cc4)Cl 8K-520S c1ccc(cc1)CS(=O)(=O)c2ccccc2c3nnc(o3)c4ccccc4 8K-521S Cc1ccc(cc1)CSc2ccccc2c3nnc(o3)c4ccccc4 8K-524S Cc1ccc(cc1)CSc2ccccc2c3nnc(o3)c4ccc(cc4)C 8K-526S Cc1ccc(cc1)CSc2ccccc2c3nnc(o3)c4ccc(cc4)Cl 8K-528S c1ccc(cc1)c2nnc(o2)c3ccccc3S(=O)(=O)Cc4ccc(cc4)Cl 8K-530S c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)S(=O)(=O)Cc4ccc(cc4)Cl 8K-531S Cc1ccc(cc1)c2nnc(o2)c3ccccc3S(=O)(=O)Cc4ccc(cc4)Cl 8K-532S CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccccc3 8K-533S c1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F 8K-534S c1cc(ccc1c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F)Cl 8K-535S Cc1ccc(cc1)CS(=O)c2ccccc2c3nnc(o3)c4ccccc4 8K-537S Cc1ccc(cc1)CS(=O)(=O)c2ccccc2c3nnc(o3)c4ccccc4 8K-538S Cc1ccc(cc1)CS(=O)(=O)c2ccccc2c3nnc(o3)c4ccc(cc4)Cl 8K-539S CNC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)Cl 8K-546S Cc1ccc(cc1)CNC(=O)c2cnn(c2C(F)(F)F)c3nc(cs3)c4ccc(cc4)Cl 8K-548S CCOC(=O)c1c(nc(nn1)c2cccs2)NC(C)C 8K-549S CCOC(=O)c1c(nc(nn1)c2cccs2)NCc3ccc(cc3)Cl 8K-552S CCOC(=O)c1c(nc(nn1)c2cccs2)NCc3ccc(cc3)C 8K-553S c1cc(ccc1CNC(=O)c2cnn(c2C(F)(F)F)c3nc(cs3)c4ccc(cc4)Cl)Cl 8K-554S c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cnn(c2C(F)(F)F)c3nc(cs3)c4ccc(cc4)Cl 8K-555S C=CCNC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)Cl 8K-556S CC(C)NC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)Cl 8K-557S c1ccc(cc1)c2nc(no2)c3ccncc3 8K-558S COc1ccc(cc1)c2nc(no2)c3ccncc3 8K-559S c1cc(ccc1c2nc(no2)c3ccncc3)F 8K-560S c1cc(cc(c1)C(F)(F)F)c2nc(no2)c3ccncc3 8K-561S Cc1ccc(cc1)c2nc(no2)c3ccncc3 8K-562S c1ccc(c(c1)c2nc(no2)c3ccncc3)Cl 8K-563S c1ccc(c(c1)c2nc(no2)c3ccncc3)C(F)(F)F 8K-567S c1cc(c(c(c1)Cl)c2nc(no2)c3ccncc3)F 8K-568S c1cc(c(c(c1)F)c2nc(no2)c3ccncc3)F 8K-569S COc1cccc(c1)c2nc(no2)c3ccncc3 8K-570S CCOC(=O)c1c(nc(nn1)c2ccc(cc2)C)NCc3ccc(cc3)Cl 8K-572S CNC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccccc3 8K-574S C=CCNC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccccc3 8K-575S c1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)NCc4cccc(c4)C(F)(F)F)C(F)(F)F 8K-576S c1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)NCc4ccc(cc4)Cl)C(F)(F)F 8K-577S c1(nc(=S)ss1)N 8K-579S c1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)NCc4ccc(c(c4)Cl)Cl)C(F)(F)F 8K-580S c1ccc(cc1)c2nc(c(nn2)C#N)N3CCOCC3 8K-585S CCOC(=O)c1c(noc1C)C 8K-591S c1ccc(cc1)c2c3cc(ccc3n(c2C(=O)N)Cc4ccc(cc4)[N+](=O)[O-])Cl 8K-900 c1ccc(cc1)c2c3cc(ccc3n(c2C#N)Cc4ccc(cc4)[N+](=O)[O-])Cl 8K-901 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)c3ccncc3C2=O 8K-902 c1cc(cc(c1)Cl)CN2C(=O)c3ccncc3C2=O 8K-903 COc1ccc(cc1OC)CCN2C(=O)c3ccncc3C2=O 8K-904 Cc1ccc(cc1)NCC(=O)c2ccc(cc2)Cl 8K-905 c1ccc2cc(ccc2c1)C(CNC(=O)C34CC5CC(C3)CC(C5)C4)O 8K-908 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)C34CC5CC(C3)CC(C5)C4)C(F)(F)F 8K-909 c1ccc2c(c1)ccc3c2C4C(CO3)CON4C(=O)C56CC7CC(C5)CC(C7)C6 8K-910 Cc1ccc(cc1)S(=O)(=O)N(CC=C)CC=C 8K-911 c1cc(sc1)CNC(=O)C23CC4CC(C2)CC(C4)C3 8K-912 c1c(cnc(c1Cl)OCC23CC4CC(C2)CC(C4)C3)C(F)(F)F 8K-913 Cc1ccccc1NC(=O)Oc2ccccc2n3cccc3 8L-001 CC(c1ccnc(n1)N)Oc2ccccc2n3cccc3 8L-002 Cc1ccc(cc1)C(=O)Oc2ccccc2n3cccc3 8L-003 c1cc(ccc1C(=O)c2ccc(s2)CC(=O)O)Cl 8L-005 c1cc(ccc1C(=O)c2ccc(s2)CC(=O)O)F 8L-006 COc1ccc(cc1)C(=O)c2ccc(s2)CC(=O)O 8L-007 c1ccc(cc1)C(=O)c2ccc(s2)CC(=O)N 8L-008 c1ccc(c(c1)C(=O)c2ccc(s2)CC(=O)O)F 8L-009 c1cc(ccc1C(=O)c2ccc(s2)CC(=O)N)Cl 8L-010 c1cc(sc1)C(=O)c2ccc(s2)CC#N 8L-011 c1ccc(c(c1)C(=O)c2ccc(s2)CC(=O)N)F 8L-012 c1cc(ccc1C(=O)c2ccc(s2)CC(=O)N)F 8L-013 c1cc(oc1)C(=O)c2ccc(s2)CC#N 8L-014 c1cc(sc1)C(=O)c2ccc(s2)CC(=O)N 8L-015 CC(C)C(C(=O)O)N1Cc2ccccc2C1=O 8L-016 CC(C(=O)O)N1Cc2ccccc2C1=O 8L-017 c1ccc(cc1)CC(C(=O)O)N2Cc3ccccc3C2=O 8L-018 c1ccc2c(c1)CN(C2=O)CC(=O)O 8L-019 Cc1c(cccc1Cl)NC(=O)c2nc(n(n2)c3cc(c(cc3Cl)Cl)OC(C)C)C 8L-301S CCOC(=O)COc1cc(c(cc1Cl)Cl)n2c(=O)c3cc(c(cc3nc2S)OC)OC 8L-303S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3ccc(cc3nc2S)Cl 8L-309S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3cc(ccc3nc2S)Cl 8L-310S CC(=O)NC(C#N)c1cccc(c1)F 8L-312S CSCCC(C(=O)O)NC(=O)c1ccccc1 8L-313S Cc1c(oc(n1)c2ccc(cc2)Cl)C(=O)NC 8L-315S Cc1c(oc(n1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)Cl 8L-316S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3ccc(cc3nc2SC)Cl 8L-320S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3ccc(cc3nc2SCc4ccccc4)Cl 8L-321S CCOC(=O)CSc1nc2cc(ccc2c(=O)n1c3cc(c(cc3Cl)Cl)OC(C)C)Cl 8L-322S c1cc(ccc1c2nc(cs2)CC(=O)O)Cl 8L-323S COc1ccc(cc1)c2nc(cs2)CC(=O)O 8L-324S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3cc(ccc3Cl)Cl 8L-325S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3ccc(cc3Cl)Cl 8L-326S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OCCOC)C(=O)Nc3ccccc3OC 8L-327S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3cc(ccc3nc2SC)Cl 8L-328S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3cc(ccc3nc2SCc4ccccc4)Cl 8L-329S CC(C)Oc1cc(c(cc1Cl)Cl)n2c(=O)c3cc(ccc3nc2SCC#C)Cl 8L-330S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OCCOC)C(=O)Nc3ccc(cc3)Br 8L-333S Cc1c(cccc1Cl)NC(=O)c2nc(n(n2)c3cc(c(cc3Cl)Cl)OCCOC)C 8L-334S C#CCOc1cc(c(cc1Cl)Cl)NC(=O)CSCC(=O)O 8L-335S C#CCOc1cc(c(cc1Cl)Cl)N2C(=O)CSCC2=O 8L-336S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3cccc(c3Cl)Cl 8L-337S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3ccc(c(c3)Cl)Cl 8L-338S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3ccc(cc3F)F 8L-339S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3ccccc3F 8L-340S Cc1ccc(c(c1)C)NC(=O)c2nc(n(n2)c3cc(c(cc3Cl)Cl)OC)C 8L-341S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F 8L-342S CCc1cccc(c1NC(=O)c2nc(n(n2)c3cc(c(cc3Cl)Cl)OC)C)CC 8L-343S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3ccc(cc3F)F 8L-344S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3cc(cc(c3)Cl)Cl 8L-345S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3cccc(c3)Cl 8L-346S Cc1ccc(c(c1)C)NC(=O)c2nc(n(n2)c3cc(c(cc3Cl)Cl)OC(C)C)C 8L-352S Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3cccc(c3)C(F)(F)F 8L-353S CSc1ccccc1c2nc(no2)c3ccncc3 8L-501S CSc1ccccc1c2nc(no2)c3ccc(cc3)C(F)(F)F 8L-502S CSc1ccccc1c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F 8L-503S CC(C)(C)c1ccc(cc1)c2nc(on2)c3ccccc3SC 8L-504S Cc1c(snn1)/C(=N/c2ccc(cc2Cl)Cl)/Oc3cccc(c3)C(F)(F)F 8L-505S COc1ccc(cc1)C(=O)NCCSc2ccc(cc2)Br 8L-507S CC(C)(C)c1ccc(cc1)c2nc(on2)c3ccccc3S(=O)C 8L-508S CC(C)(C)c1ccc(cc1)c2nc(on2)c3ccccc3S(=O)(=O)C 8L-509S CS(=O)c1ccccc1c2nc(no2)c3ccc(cc3)C(F)(F)F 8L-510S CS(=O)(=O)c1ccccc1c2nc(no2)c3ccc(cc3)C(F)(F)F 8L-511S CS(=O)c1ccccc1c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F 8L-512S CS(=O)(=O)c1ccccc1c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F 8L-513S Cn1c(c(c(n1)c2ccccc2)C#N)Cl 8L-515S c1cc(ccc1C2=NNC(=O)CC2)Cl 8L-516S CC(CSc1ccc(cc1)Cl)(C(=O)Nc2cc(c(cc2Cl)Cl)OCCOC)O 8L-517S CC(CSc1ccccc1C(=O)OC)(C(=O)Nc2cc(c(cc2Cl)Cl)OCCOC)O 8L-518S c1ccc(cc1)c2c(c(nc(n2)S)O)C#N 8L-519S Cc1c(c(on1)C)CSc2ccc(cc2)Br 8L-520S Cn1c(c(c(n1)c2ccccc2)C#N)Sc3ccc(cc3)Br 8L-521S Cn1c(c(c(n1)c2ccccc2)C#N)Sc3ccccc3C(=O)OC 8L-522S COCCOc1cc(c(cc1Cl)Cl)NC(=O)c2c(ccs2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F 8L-526S Cn1c(c(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)C(F)(F)F)Cl 8L-529S CC(C)(C)c1ccc(cc1)O/C(=N\c2cccc(c2)C(F)(F)F)/c3c(nn(c3Cl)C)C(F)(F)F 8L-530S COc1ccc(cc1)C(=O)NCCSc2ccc(cc2)Cl 8L-533S c1cc(ccc1C(=O)NCCSc2ccc(cc2)Cl)Cl 8L-534S Cc1ccccc1C(=O)NCCSc2ccc(cc2)Cl 8L-539S c1ccc(cc1)C(=O)NCCSc2ccc(cc2)Cl 8L-540S CCOC(=O)c1c(n(c(=S)s1)c2ccccc2)SC 8L-542S CCOC(=O)C/C(=N\Nc1cc(c(cc1Cl)Cl)OCCOC)/C(F)(F)F 8L-543S c1cc(ccc1SCCNC(=O)c2ccc(cc2Cl)Cl)Cl 8L-545S c1cc(ccc1C2=NN(CCC2)C(=O)c3ccc(c(c3)Cl)Cl)Cl 8L-546S CCOC(=O)c1c(n(c(=S)s1)c2ccc(cc2)Cl)SC 8L-547S COc1cccc(c1)C(=O)N2CCCC(=N2)c3ccc(cc3)Cl 8L-550S c1cc(cc(c1)Cl)C(=O)N2CCCC(=N2)c3ccc(cc3)Cl 8L-551S COc1ccc(cc1)C(=O)N2CCCC(=N2)c3ccc(cc3)Cl 8L-552S Cc1ccc(cc1)C(=O)N2CCCC(=N2)c3ccc(cc3)Cl 8L-553S CCOC(=O)c1c(n(c(=S)s1)c2cccc(c2)C(F)(F)F)SC 8L-554S C/C(=N\NC(=O)N)/C(=O)OC 8L-556S COC(=O)c1csnn1 8L-557S Cn1c(c(c(n1)C(F)(F)F)/C(=N/c2cccc(c2)C(F)(F)F)/Oc3ccc(cc3Cl)Cl)Cl 8L-558S COc1ccc(cc1)Oc2nc(cc(n2)OC)OC 8L-559S COc1ccc(cc1)C(=O)NCCSc2ccccc2 8L-561S c1ccc(cc1)SCCNC(=O)c2ccc(c(c2)Cl)Cl 8L-562S CC(C)(CCl)C(=O)Nc1ccc(cc1Cl)Cl 8L-700 CC1(CN(C1=O)c2ccc(cc2Cl)Cl)C 8l-701 CN(C)/C=C(/c1ccc2ccccc2c1[N+](=O)[O-])\C(=O)C(F)(F)F 8L-703 c1ccc(c(c1)/C=N/c2ccccc2N)[N+](=O)[O-] 8L-706 COc1ccc(cc1)c2cc(n[nH]2)C3CCNCC3 8L-707 c1ccc2c(c1)c3c(nc4ccccc4n3)nn2 8L-708 CC(C)(CCl)C(=O)Nc1ccsc1C(=O)OC 8L-709 CC1(CN(C1=O)c2ccsc2C(=O)OC)C 8L-710 Cc1ccc(cc1)n2cc(c(n2)C(F)(F)F)c3ccc4ccccc4c3[N+](=O)[O-] 8L-711 COc1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N 8L-712 CC1(CN(C1=O)c2ccc(cc2)C(=O)/C=C/N(C)C)C 8L-713 CC(C)(CCl)C(=O)Nc1cccc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl 8L-714 CC1(CN(C1=O)c2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl)C 8L-715 c1ccc(c(c1)/C=N/n2c(=O)cc(nc2N)C(F)(F)F)[N+](=O)[O-] 8L-716 Cc1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)n4cccc4)C#N 8L-717 c1cc(ccc1CN2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)Cl)[N+](=O)[O-] 8L-718 c1ccc(cc1)COc2ccc(cc2)/C=N/NC(=O)CC#N 8L-719 c1ccc(cc1)C/C=N/NC(=O)CC#N 8L-720 c1ccc2c(c1)ccc(c2[N+](=O)[O-])c3cn(nc3C(F)(F)F)c4ccc(cc4)Cl 8L-721 CC(C)(CCl)C(=O)Nc1ccccc1C(=O)c2ccccc2 8L-722 CC1(CN(C1=O)c2ccc(cc2)C(=O)c3ccccc3)C 8L-723 c1ccc2c(c1)ccc(c2[N+](=O)[O-])c3cn(nc3C(F)(F)F)c4ccccc4F 8L-724 c1cc(c(cc1Cl)Cl)c2cc([nH]n2)C3CCNCC3 8L-725 c1ccc2c(c1)ccc(c2[N+](=O)[O-])c3cn(nc3C(F)(F)F)c4ccc(cc4)F 8L-726 c1cc(oc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N 8L-727 CO/N=C/Cc1ccc2ccccc2c1[N+](=O)[O-] 8L-728 COc1ccc(cc1)CN2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)OC 8L-729 COc1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)n4cccc4)C#N 8L-730 c1cc(c(c(c1)Cl)CN2CCC(CC2)c3cc([nH]n3)c4ccc(cc4Cl)Cl)Cl 8L-731 CCOC(=O)c1c(c(c(=O)n(c1N)N)C#N)c2ccc(cc2)OCc3ccccc3 8L-732 c1ccc2c(c1)ccc(c2[N+](=O)[O-])c3cn(nc3C(F)(F)F)c4cccc(c4)[N+](=O)[O-] 8L-733 CCOC(=O)C1=C(Nc2c(cnn2c3ccc(cc3)F)C1c4ccc(cc4)Cl)C 8L-734 c1cc([nH]c1)/C=N/NC(=O)CC#N 8L-736 CC1(CN(C1=O)c2ccc(cc2)c3ccnn3c4ccc(cc4)Cl)C 8L-737 c1ccc2c(c1)/C(=N\Nc3ccc(c(c3)C(F)(F)F)Cl)/C(=O)OC2=O 8L-738 c1ccc2c(c1)/C(=N\Nc3ccc(c(c3)C(=O)O)Cl)/C(=O)OC2=O 8L-739 CCOC(=O)C1=C(Nc2c(cnn2c3c(cc(cn3)C(F)(F)F)Cl)C1c4ccc(cc4)Cl)C 8L-740 CC(C)(CCl)C(=O)Nc1ccc(cc1)I 8L-741 CC1(CN(C1=O)c2ccc(cc2)I)C 8L-742 CC(C)(CCl)C(=O)Nc1ccccc1C(=O)OC 8L-743 CC1(CN(C1=O)c2ccccc2C(=O)OC)C 8L-744 CCOC(=O)C1=C(Nc2c(cnn2c3ccc(cc3)Cl)C1c4ccc(cc4)Cl)C 8L-745 CC(C)(CCl)C(=O)Nc1cccnc1Cl 8L-747 CC1(CN(C1=O)c2cccnc2Cl)C 8L-748 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)C=O)Sc3ccc(cc3)Cl)C 8L-749 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)Cc4ccc(cc4)[N+](=O)[O-] 8L-751 Cc1c(snn1)/C(=N/c2ccc(cc2Cl)Cl)/Sc3cccc(c3)C(F)(F)F 8L-804S CCOC(=O)C1=NOC(C1)CNC(=O)c2ccccc2Cl 8L-900 CCOC(=O)C1=NOC(C1)Cn2cc(c(=O)[nH]c2=O)C(=O)C 8L-901 CCOC(=O)c1c(con1)c2ccc3c(c2)C(=O)c4ccccc4C3=O 8L-902 c1ccc(c(c1)C(=O)NCC2CC(=NO2)C(=O)O)Cl 8L-903 c1ccc(c(c1)C(=O)NCC(CC#N)O)Cl 8L-905 c1cc(ccc1N/C=C/2\C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)I 8L-906 c1ccc(cc1)Oc2ccc(cc2)N/C=C/3\C(=O)NC(=O)N(C3=O)CCNc4c(cc(cn4)C(F)(F)F)Cl 8L-907 c1cc(c(c(c1)Cl)CO/N=C/C2C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)F 8L-908 c1cc(ccc1N/C=C/2\C(=O)NC(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl 8L-909 c1c(cnc(c1Cl)NCCN2C(=O)C(C(=O)NC2=O)/C=N/Nc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 8L-910 Cc1c(c(n[nH]1)N)C(=O)Nc2cccc(c2)C(F)(F)F 8L-911 COC(=O)CCCNc1c(cccn1)[N+](=O)[O-] 8L-912 c1c(cnc(c1Cl)ON2C(=O)CCC2=O)C(F)(F)F 8L-913 C/C(=C\1/C(=O)NC(=O)N(C1=O)CCNc2c(cc(cn2)C(F)(F)F)Cl)/N(C)C 8L-914 COC(=O)CCCNc1ccc(cc1[N+](=O)[O-])C(F)(F)F 8L-915 c1ccc(cc1)c2ncc3c(n2)-c4ccccc4CC3 8L-916 c1cc(c(nc1)NCCCC(=O)O)[N+](=O)[O-] 8L-917 c1c(cnc(c1Cl)NCCN2C(=O)C3C4CC(C3C2=O)C=C4)C(F)(F)F 8L-918 COC(=O)CCCNc1ccc(cc1N)C(F)(F)F 8L-919 c1ccc-2c(c1)CCc3c2nn(c3)C(=O)c4ccc(cc4)F 8L-921 c1ccc-2c(c1)CCc3c2nn(c3)c4c(cc(cn4)C(F)(F)F)Cl 8L-922 c1ccc-2c(c1)CCc3c2nn(c3)C(=O)Nc4ccc(cc4)Cl 8L-923 COC(=O)c1ccncc1C(=O)O 8L-924 Cc1ccc(cc1)C(=O)n2cc3c(n2)-c4ccccc4CC3 8L-925 c1ccc-2c(c1)CCc3c2nn(c3)S(=O)(=O)c4ccc(cc4)F 8L-926 COc1ccc(cc1)NC(=O)c2cnccc2C(=O)OC 8L-927 COC(=O)c1ccncc1C(=O)Nc2ccc(cc2)F 8L-928 COC(=O)c1ccncc1C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 8L-929 CCOC(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 8L-930 c1cc2c(cc1N/N=C/3\CCCCC3=O)OCCO2 8L-932 c1c2c(cc3c1OCCO3)[nH]c4c2CCCC4=O 8L-933 COC(=O)CCCNc1ccc(cc1NC(=O)Nc2ccc(cc2)Cl)C(F)(F)F 8L-934 COC(=O)CCCNc1ccc(cc1NC(=O)c2ccc(cc2)Cl)C(F)(F)F 8L-937 c1cc2c(c(c1)N)C(=O)N(C2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl 8L-938 CCOC(=O)C1=NOC2C1C3CC2C4C3C(=O)N(C4=O)CCNc5c(cc(cn5)C(F)(F)F)Cl 8L-939 c1cc(cc(c1)NC(=O)Nc2cccc3c2C(=O)N(C3=O)CCNc4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 8L-940 c1ccn(c1)c2cccc3c2C(=O)N(C3=O)CCNc4c(cc(cn4)C(F)(F)F)Cl 8L-941 c1c(cnc(c1Cl)NCCN2C(=O)C3C4CC(C3C2=O)C5C4C(=NO5)C(=O)N6CCCC6)C(F)(F)F 8L-942 c1c(cnc(c1Cl)NCCN2C(=O)C3C4CC(C3C2=O)C5C4C(=NO5)C(=O)O)C(F)(F)F 8L-943 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)N3CCCC3)Cl 8L-944 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2N)C(=O)N3CCCC3)Cl 8L-945 c1c(cnc(c1Cl)NCCN2C(=O)C3C4CC(C3C2=O)C(C4C#N)O)C(F)(F)F 8L-946 c1cc(ccc1NC(=O)Nc2ccc(cc2CS(=O)(=O)c3ccc(cc3)Cl)C(=O)N4CCCC4)Cl 8L-947 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2NC(=O)C(F)(F)F)C(=O)N3CCCC3)Cl 8L-948 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)N)Cl 8L-949 c1ccn(c1)c2ccc(cc2CS(=O)(=O)c3ccc(cc3)Cl)C(=O)N4CCCC4 8L-950 c1cc(ccc1C(=O)Nc2ccc(cc2CS(=O)(=O)c3ccc(cc3)Cl)C(=O)N4CCCC4)F 8L-951 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C#N)Cl 8L-952 c1ccc(c(c1)C(=O)NCC(CC#N)OC(=O)c2cccc(c2)C(F)(F)F)Cl 8L-953 Cc1c(cccc1Cl)N/C=C/C(=C(C#N)C#N)N(C)C 8M-001 Cc1ccc(c(c1)N/C=C/C(=C(C#N)C#N)N(C)C)C 8M-002 Cc1c(cccc1Cl)Nc2c(c(ccn2)N(C)C)C#N 8M-003 COc1ccnc(c1C#N)N2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 8M-004 COc1ccnc(c1C#N)N2CCN(CC2)C(c3ccccc3)c4ccccc4 8M-005 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)Br 8M-006 Cc1cccc(c1)N/C=C/C(=C(C#N)C#N)N(C)C 8M-007 COc1ccnc(c1C(=O)N/C=N/OC)Oc2ccc(cc2)Cl 8M-008 COc1ccnc(c1C(=O)N/C=N/OCc2ccc(cc2)Cl)Oc3ccc(cc3)Cl 8M-009 Cc1ccc(c(c1)Nc2c(c(ccn2)N(C)C)C#N)C 8M-011 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)Br 8M-012 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)[N+](=O)[O-] 8M-013 Cc1ccccc1N/C=C/C(=C(C#N)C#N)N(C)C 8M-014 Cc1ccccc1Nc2c(c(ccn2)N(C)C)C#N 8M-015 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)[N+](=O)[O-] 8M-016 Cc1cccc(c1)Nc2c(c(ccn2)N(C)C)C#N 8M-017 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccccc1F 8M-018 CN(C)c1ccnc(c1C#N)Nc2ccccc2F 8M-019 CN(C)C(=C(C#N)C#N)/C=C/Nc1cccc(c1)Br 8M-020 CN(C)C(=C(C#N)C#N)/C=C/Nc1cc(cc(c1)Cl)Cl 8M-022 COc1ccnc(c1C#N)N/C=N/OC 8M-023 COc1ccnc(c1C#N)N/C=N/OCc2ccc(cc2)Cl 8M-024 COc1ccnc(c1C#N)N/C=N/OCc2cccc(c2)C(F)(F)F 8M-025 Cc1ccc(cc1)CO/N=C/Nc2c(c(ccn2)OC)C#N 8M-026 COc1ccnc(c1C#N)N/C=N/OCCOc2cccc(c2)C(F)(F)F 8M-027 COc1ccnc(c1C#N)N/C=N/OCc2ccc(cc2)F 8M-028 COc1ccnc(c1C#N)Oc2ccc(cc2)S(=O)(=O)N3CCOCC3 8M-029 COc1ccnc(c1C#N)N/C=N/OCc2cccc(c2Cl)Cl 8M-030 COc1ccnc(c1C#N)N/C=N/OCc2ccc(cc2Cl)F 8M-031 CN(C)c1ccnc(c1C#N)Nc2cc(cc(c2)Cl)Cl 8M-032 COc1ccnc(c1C#N)N2CCN(CC2)c3cccc(c3)C(F)(F)F 8M-033 CN(C)c1ccnc(c1C#N)Nc2cccc(c2)Br 8M-035 CN(C)C(=C(C#N)C#N)/C=C/Nc1cccc(c1)[N+](=O)[O-] 8M-037 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccccc1OC 8M-038 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccccc1 8M-039 COc1ccnc(c1C(=O)N)Oc2ccccc2 8M-040 CN(C)c1ccnc(c1C#N)Nc2ccccc2OC 8M-041 CN(C)C(=C(C#N)C#N)/C=C/Nc1cc(ccc1Cl)C(F)(F)F 8M-042 CN(C)C(=C(C#N)C#N)/C=C/Nc1ccc(cc1)I 8M-043 CN(C)c1ccnc(c1C#N)Nc2ccccc2 8M-044 CN(C)c1ccnc(c1C#N)Nc2cccc(c2)[N+](=O)[O-] 8M-045 CN(C)c1ccnc(c1C#N)Nc2cc(ccc2Cl)C(F)(F)F 8M-047 CN(C)c1ccnc(c1C#N)Nc2ccc(cc2)I 8M-048 CN(C)C(=C(C#N)C#N)C/C=N/OCc1ccc(cc1)Cl 8M-049 CC(C)(C)NS(=O)(=O)c1ccc(cc1)Oc2c(c(ccn2)OC)C#N 8M-050 COc1ccnc(c1C#N)NCc2cccnc2 8M-051 Cc1ccc(cc1)CNc2c(c(ccn2)OC)C#N 8M-052 CN(C)C(=C(C#N)C#N)C/C=N/OCc1ccc(cc1Cl)F 8M-053 CN(C)C(=C(C#N)C#N)C/C=N/OCC(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 8M-054 COc1ccnc(c1C#N)NCc2cccc(c2)C(F)(F)F 8M-055 CN(C)C(=C(C#N)C#N)C/C=N/OCC(=O)N1CCN(CC1)c2ccccc2 8M-056 CN(C)C(=C(C#N)C#N)C/C=N/OCc1cccc(c1)Cl 8M-057 CN(C)C(=C(C#N)C#N)C/C=N/OCc1c(cccc1Cl)Cl 8M-058 CN(C)C(=C(C#N)C#N)C/C=N/OCCOc1cccc(c1)C(F)(F)F 8M-059 CN(C)C(=C(C#N)C#N)C/C=N/OCc1ccc(cc1)F 8M-060 CN(C)C(=C(C#N)C#N)C/C=N/OCc1ccccc1F 8M-061 CN(C)C(=C(C#N)C#N)C/C=N/OCc1cccc(c1Cl)Cl 8M-062 CN(C)C(=C(C#N)C#N)C/C=N/Nc1ccc(cc1Cl)Cl 8M-063 CN(C)C(=C(C#N)C#N)C/C=N/OCc1ccccc1Cl 8M-064 COc1ccnc(c1C#N)n2cccc2/C=N/OCc3c(cccc3Cl)F 8M-066 COc1ccnc(c1C#N)n2cccc2/C=N/OCc3ccc(cc3Cl)Cl 8M-067 Cc1ccc(cc1)CO/N=C/c2cccn2c3c(c(ccn3)OC)C#N 8M-068 COc1cccc(c1)CO/N=C/c2cccn2c3c(c(ccn3)OC)C#N 8M-069 COc1ccnc(c1C#N)n2cccc2/C=N/OCc3cccc(c3)C(F)(F)F 8M-070 Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2N3CCOCC3)C)C 8M-301S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)NCc3ccc(cc3)OC)c4ccccc4 8M-302S CCSc1nnc(o1)c2c(nc3n2ccs3)C 8M-303S Cc1c(n2ccsc2n1)c3nnc(o3)SC=C=C 8M-304S Cc1c(n2ccsc2n1)c3nnc(o3)SCc4cccc(c4)C(F)(F)F 8M-305S Cc1c2c(c(=O)[nH]nc2c3ccccc3)no1 8M-309S CCOC(=O)c1cc(on1)c2ccccc2 8M-311S Cn1c2c(cc(s2)c3nnc(o3)SCC=C)c(n1)C(F)(F)F 8M-315S Cc1c2c(c(=O)n(nc2c3ccccc3)CC=C)no1 8M-317S Cc1cccc(c1)CSc2nnc(o2)c3cc4c(nn(c4s3)C)C(F)(F)F 8M-319S Cn1c2c(cc(s2)c3nnc(o3)SCc4ccc(cc4)OC)c(n1)C(F)(F)F 8M-320S Cn1c2c(cc(s2)c3nnc(o3)SCc4ccc(cc4)Cl)c(n1)C(F)(F)F 8M-321S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)SC3CCCCC3)c4ccccc4 8M-322S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)C3CCCCC3)c4ccccc4 8M-323S Cn1c2c(cc(s2)c3nnc(o3)SC)c(n1)C(F)(F)F 8M-324S Cn1c2c(cc(s2)c3nnc(o3)SCc4ccc(cc4)F)c(n1)C(F)(F)F 8M-325S Cn1c2c(cc(s2)c3nnc(o3)SCc4c(cccc4Cl)F)c(n1)C(F)(F)F 8M-326S COC(=O)C1CC(=NO1)c2ccc(cc2)Cl 8M-327S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)NCc3ccccc3Cl)c4ccccc4 8M-328S Cc1ccccc1Oc2c(c(cc(n2)c3ccccc3)C)S(=O)(=O)c4ccc(cc4)Cl 8M-329S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)Oc3ccc(cc3)C(C)(C)C)c4ccccc4 8M-330S Cc1cc(nc(c1S(=O)(=O)Cc2ccc(cc2)Cl)O)c3ccccc3 8M-331S Cc1cc(nc(c1S(=O)(=O)Cc2ccc(cc2)Cl)Cl)c3ccccc3 8M-332S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)Oc3cccc(c3)C(F)(F)F)c4ccccc4 8M-333S c1ccc(cc1)c2ccn(c(=O)c2C#N)Cc3ccc(cc3)Cl 8M-502S Cc1ccc(cc1)Cn2ccc(c(c2=O)C#N)c3ccccc3 8M-503S c1ccc(cc1)c2ccn(c(=O)c2C#N)Cc3ccccc3Cl 8M-504S c1ccc(cc1)c2ccn(c(=O)c2C#N)Cc3cccc(c3)Cl 8M-505S c1ccc(cc1)c2ccn(c(=O)c2C#N)Cc3cccc(c3)C(F)(F)F 8M-506S c1ccc(cc1)c2ccnc(c2C#N)Cl 8M-510S CCn1ccc(c(c1=O)C#N)c2ccccc2 8M-512S CCOC(=O)Cn1ccc(c(c1=O)C#N)c2ccccc2 8M-513S Cc1c(sc2n1ncn2)c3csc(n3)NC 8M-515S Cc1c(sc2n1ncn2)c3csc(n3)c4ccc(cc4)Cl 8M-516S Cc1c(sc2n1ncn2)c3csc(n3)c4ccc(cc4)OC 8M-517S Cc1c(sc2n1ncn2)c3csc(n3)C 8M-518S CNc1c(c(ccn1)c2ccccc2)C#N 8M-519S c1ccc(cc1)c2ccnc(c2C#N)N3CCOCC3 8M-520S Cc1c(sc2n1ncn2)c3csc(n3)Nc4ccccc4 8M-521S Cc1c(sc2n1ncn2)c3csc(n3)Nc4ccc(cc4)Cl 8M-522S Cc1ccccc1Cn2ccc(c(c2=O)C#N)c3ccc(cc3)Cl 8M-526S Cc1cccc(c1)Cn2ccc(c(c2=O)C#N)c3ccc(cc3)Cl 8M-527S c1cc(cc(c1)C(F)(F)F)Cn2ccc(c(c2=O)C#N)c3ccc(cc3)Cl 8M-528S C=CCn1ccc(c(c1=O)C#N)c2ccccc2 8M-529S COC(=O)Cn1ccc(c(c1=O)C#N)c2ccc(cc2)Cl 8M-530S CNc1c(c(ccn1)c2ccc(cc2)Cl)C#N 8M-531S c1cc(ccc1c2ccnc(c2C#N)N3CCOCC3)Cl 8M-532S COc1c(c(ccn1)c2ccc(cc2)Cl)C#N 8M-533S c1cc(ccc1COn2c(=O)c3cc(cc(c3nc2C(F)(F)F)Cl)Cl)Cl 8M-534S Cc1c(sc2n1ncn2)C(=O)CSc3ccc(cc3)Cl 8M-536S Cc1c(sc2n1ncn2)/C(=N/O)/C 8M-537S Cc1cccc(c1C)Oc2c(c(ccn2)c3ccccc3)C#N 8M-539S COc1ccc(cc1)Oc2c(c(ccn2)c3ccccc3)C#N 8M-540S c1ccc(cc1)/C=C(/C#N)\C(=S)N 8M-542S COc1cnn(c(=O)c1Cl)c2ccccc2 8M-543S COc1c(cnn(c1=O)c2ccccc2)Cl 8M-544S COc1ccc(cc1)Sc2c(c(ccn2)c3ccc(cc3)Cl)C#N 8M-545S c1cc(cc(c1)Sc2c(c(ccn2)c3ccc(cc3)Cl)C#N)C(F)(F)F 8M-546S c1cc(ccc1c2ccnc(c2C#N)Oc3ccc(c(c3)Cl)Cl)Cl 8M-547S c1cc(cc(c1)Oc2c(c(ccn2)c3ccc(cc3)Cl)C#N)C(F)(F)F 8M-548S c1ccc(cc1)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl 8M-549S COc1c(cnn(c1=O)c2ccc(c(c2)Cl)Cl)Cl 8M-550S COc1cnn(c(=O)c1Cl)c2ccc(c(c2)Cl)Cl 8M-551S Cc1ccc(cc1)n2c(=O)c(c(cn2)Cl)OC 8M-552S Cc1ccc(cc1)n2c(=O)c(c(cn2)OC)Cl 8M-553S COc1ccc(cc1)c2csc(n2)/C(=C/c3ccccc3)/C#N 8M-554S c1cc(oc1)/C=C(\C#N)/C(=S)N 8M-555S COc1ccc(cc1OC)/C=C(/C#N)\C(=S)N 8M-556S c1cc(ccc1/C=C(/C#N)\C(=S)N)F 8M-557S COC(=O)c1ccccc1Sc2c(c(ccn2)c3ccc(cc3)Cl)C#N 8M-558S COc1ccc(cc1)CSc2c(c(ccn2)c3ccc(cc3)Cl)C#N 8M-559S Cc1c(sc2n1ncn2)/C(=N/OCc3ccc(cc3)Cl)/C 8M-560S Cc1c(sc2n1ncn2)/C(=N\O)/CSc3ccc(cc3)Cl 8M-561S c1cc(ccc1c2ccnc(c2C#N)Oc3ccc(cc3)F)Cl 8M-562S Cc1ccc(cc1)n2c(=O)c(c(cn2)Br)Br 8M-564S CCOc1cnn(c(=O)c1Cl)c2ccccc2 8M-565S CCOc1c(cnn(c1=O)c2ccccc2)Cl 8M-566S CCOc1cnn(c(=O)c1Cl)c2ccc(cc2)C 8M-567S CCOc1c(cnn(c1=O)c2ccc(cc2)C)Cl 8M-568S CCOc1cnn(c(=O)c1Cl)c2ccc(c(c2)Cl)Cl 8M-569S Cc1c(sc(n1)/C(=C/c2ccco2)/C#N)C(=O)C 8M-573S c1cc(oc1)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)F 8M-574S COc1ccc(cc1OC)/C=C(\C#N)/c2nc(cs2)c3ccccc3 8M-576S COc1ccc(cc1)c2csc(n2)/C(=C/c3ccc(cc3)F)/C#N 8M-577S CCOC(=O)Cc1csc(n1)N 8M-580S COc1ccc(cc1)Oc2c(c(ccn2)c3ccc(cc3)Cl)C#N 8M-582S Cc1c(sc2n1ncn2)C(C)O 8M-584S Cc1csc(n1)/C(=C/c2ccccc2)/C#N 8M-590S c1ccc(cc1)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)F 8M-591S c1ccc(cc1)/C=C(\C#N)/c2nc(cs2)c3ccccc3 8M-592S CC(C)Oc1c(cnn(c1=O)c2ccccc2)Cl 8M-593S CCOC(=O)c1c(nc(s1)N)C 8M-594S Cc1ccc(cc1)n2c(=O)c(c(cn2)OC)Br 8M-595S COc1cnn(c(=O)c1Br)c2ccc(cc2)F 8M-596S COc1c(cnn(c1=O)c2ccc(cc2)F)Br 8M-597S c1ccc(c(c1)C(=O)O)Sc2ccc(cn2)C(F)(F)F 8M-605S c1cc(oc1)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl 8M-606S COc1ccc(cc1)c2csc(n2)/C(=C/c3ccco3)/C#N 8M-607S c1ccc(cc1)c2csc(n2)/C(=C/c3ccco3)/C#N 8M-609S COc1ccc(cc1OC)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl 8M-610S COc1ccc(cc1)c2csc(n2)/C(=C/c3ccc(c(c3)OC)OC)/C#N 8M-611S Cc1c(nc(s1)/C(=C/c2ccc(c(c2)OC)OC)/C#N)C(=O)C 8M-612S COc1ccc(cc1OC)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)F 8M-613S c1cc(ccc1/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl)F 8M-614S c1cc(ccc1/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)F)F 8M-616S c1ccc(cc1)c2csc(n2)/C(=C/c3ccc(cc3)F)/C#N 8M-617S Cc1ccc(cc1)n2c(=O)c(c(cn2)Br)OC 8M-621S CCOc1c(cnn(c1=O)c2ccc(cc2)C)Br 8M-622S CCOc1cnn(c(=O)c1Br)c2ccc(cc2)C 8M-623S CCOc1c(cnn(c1=O)c2ccc(cc2)F)Br 8M-624S Cc1c(sc2n1ncn2)C(C)OC(=O)Nc3ccc(cc3)Cl 8M-626S c1cc(ccc1C(=O)On2c(=O)c3cc(cc(c3nc2C(F)(F)F)Cl)Cl)Cl 8M-628S Cc1cc(n[nH]1)c2ccc(cc2)Br 8M-635S Cc1c(c(=O)ccn1c2ccc(cc2)/N=N/c3ccccc3)Cc4c(cccc4Cl)Cl 8M-700 c1ccc2cc(ccc2c1)Sc3ccc4nnc(n4n3)C(F)(F)F 8M-701 COc1ccc(cc1)N/C=C/C(=O)c2cc(sc2Cl)Cl 8M-702 c1cc(cc(c1)Cl)CONC(=O)N 8M-704 c1cc(c(cc1Cl)Cl)CON2C(=O)C(=O)NC2=O 8M-705 c1cc(c(c(c1)Cl)CON2C(=O)C(=O)NC2=O)Cl 8M-706 c1cc(ccc1CON2C(=O)C(=O)NC2=O)F 8M-707 c1ccc(c(c1)CON2C(=O)C(=O)NC2=O)F 8M-708 c1cc(cc(c1)C(F)(F)F)CNC(=O)N 8M-709 c1cc(c(cc1F)Cl)CON2C(=O)C(=O)NC2=O 8M-711 c1cc(c(c(c1)Cl)CON2C(=O)C(=O)NC2=O)F 8M-712 Cc1c(c(=O)ccn1Cc2cccc(c2)Cl)Cc3c(cccc3Cl)Cl 8M-713 c1cc(cc(c1)Cl)CON2C(=O)C(=O)NC2=O 8M-715 CC(C)(CNC(=O)Nc1ccc(cc1)Cl)SCc2cccc(c2)C(F)(F)F 8M-717 CON1C(=O)C(=O)NC1=O 8M-718 CCOC(=O)CNC(=O)N 8M-719 c1cc(cc(c1)C(F)(F)F)CN2C(=O)C(=O)NC2=O 8M-720 C/C(=N\O)/c1cc(sc1Cl)Cl 8M-721 CC(C)(CNC(=O)Nc1ccccc1)SCc2cccc(c2)C(F)(F)F 8M-723 CC(C)(CNC(=O)N)SCc1cccc(c1)C(F)(F)F 8M-724 Cc1c(c(=O)cco1)Cc2c(cccc2Cl)Cl 8M-726 CCOC(=O)CN1C(=O)C(=O)NC1=O 8M-728 CC(C)(CNS(=O)(=O)c1ccc(cc1)OC)SCc2ccc(cc2)F 8M-731 CC(C)(CNS(=O)(=O)c1ccc(cc1)Br)SCc2ccc(cc2)F 8M-732 Cc1c(c(=O)ccn1Cc2cccs2)Cc3c(cccc3Cl)Cl 8M-734 Cc1ccc(cc1)Cn2ccc(=O)c(c2C)Cc3c(cccc3Cl)Cl 8M-735 CC(C)(CNc1c(cccn1)[N+](=O)[O-])SCc2ccc(cc2)F 8M-736 CC(C)(CNS(=O)(=O)c1cc(ccc1Cl)Cl)SCc2ccc(cc2)F 8M-737 Cc1c(c(=O)ccn1CC(=O)OC)Cc2c(cccc2Cl)Cl 8M-738 CC(C)(CNC(=O)c1ccc(c(c1)Cl)Cl)SCc2cccc(c2)C(F)(F)F 8M-739 CC(C)(CNc1ccc(nn1)Cl)SCc2ccc(cc2)F 8M-740 Cc1ccc(cc1)S(=O)(=O)CC(=O)OC 8M-741 CC(C)(CNS(=O)(=O)c1ccc2ccccc2c1)SCc3ccc(cc3)F 8M-742 c1c2n(cn1)C(=O)NCC2 8M-743 CC(C)(CNS(=O)(=O)c1ccc(cc1)Cl)SCc2ccc(cc2)F 8M-744 c1ccc2c(c1)c3c(c(=O)o2)C(CO3)O 8M-746 Cc1cc(c(o1)C)C(=O)/C=C/c2ccoc2 8M-900 c1ccc(cc1)C(=O)NC(=S)n2c3ccccc3nn2 8M-901 C=CCn1c(nnc1S)CNS(=O)(=O)c2ccc(cc2)F 8M-902 CCOC(=O)NC(=O)/C(=C\Nc1ccc(cc1)OC)/C(=O)C 8M-903 CCOC(=O)NC(=O)/C(=C/Nc1ccc(cc1)F)/C#N 8M-904 CC(=O)c1cn(c(=O)[nH]c1=O)c2ccc(cc2)OC 8M-905 c1ccc(cc1)C(=O)/C=C/c2sc(cc2)/C=C/C(=O)c3ccccc3 8M-906 c1ccc2c(c1)c(=O)[nH]nn2 8M-907 c1ccc(cc1)C(=O)/C=C/c2ccc(o2)CO 8M-908 c1ccc(cc1)C(=O)/C=C/c2ccc(o2)C=O 8M-909 Cc1cc(cc(c1)N/C(=N\O)/c2cccc(c2)[N+](=O)[O-])C 8N-001 COc1ccc(cc1)COc2ccc(cc2OC)/C=C/S(=O)(=O)NCc3cccs3 8N-002 COc1ccc(cc1)/C=C/S(=O)(=O)NCc2cccs2 8N-003 COc1cccc(c1)CNS(=O)(=O)/C=C/c2ccc(c(c2)OC)OCc3ccc(cc3)F 8N-004 c1cc(c(nc1)OCc2cnc(s2)Cl)[N+](=O)[O-] 8N-005 CC(=O)c1cccc(c1)OCc2cnc(s2)Cl 8N-006 c1ccn(c1)c2ccc(cc2)Oc3ncccn3 8N-007 CC(=O)Nc1ccc(cc1)Oc2ncccn2 8N-008 c1c(sc(n1)Cl)CN2CCCCC2 8N-010 COc1ccc(cc1)NS(=O)(=O)/C=C\c2ccc(c(c2)OC)OCc3ccc(cc3)F 8N-012 COc1cccc(c1)CNS(=O)(=O)/C=C/c2ccc(c(c2)OC)OC 8N-013 CC(=O)c1ccc(cc1)OCc2cnc(s2)Cl 8N-014 COc1cccc(c1)CNS(=O)(=O)/C=C/c2ccc3c(c2)OCO3 8N-015 CN(c1ccccc1)C(=O)C(=O)OC 8N-016 c1cc(cc(c1)N/C=C/C(=O)c2ccc(cc2)Oc3ncccn3)C(F)(F)F 8N-017 c1cnc(nc1)Oc2ccc(cc2)C(=O)/C=C/Nc3ccc(cc3)F 8N-018 c1cnc(nc1)Oc2ccc(cc2)c3cc[nH]n3 8N-020 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])OCc2cnc(s2)Cl 8N-021 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])OCc2cnc(s2)Cl 8N-022 CS(=O)(=O)Nc1ccc(cc1)Oc2ncccn2 8N-023 COC(=O)C(=O)Nc1ccc(cc1)C(F)(F)F 8N-024 Cc1cccc(c1)Oc2ccc(cc2[N+](=O)[O-])C(=O)OC 8N-025 COc1ccc(cc1)OCc2cnc(s2)OCc3ccccc3 8N-026 COc1ccc(c(c1)[N+](=O)[O-])NC(=O)C(=O)OC 8N-027 CS(=O)(=O)NCc1ccc(cc1)F 8N-029 Cc1ccc(cc1)NS(=O)(=O)/C=C/c2ccc(c(c2)OC)OC 8N-032 c1ccc2cc(ccc2c1)Oc3ccc(cc3)[N+](=O)[O-] 8N-034 c1ccc(cc1)OCc2cnc(s2)OCc3cc(ccc3Cl)Cl 8N-035 COc1ccc(cc1)OCc2cnc(s2)OCc3ccc(c(c3)Cl)Cl 8N-036 COc1ccc(cc1)/C=C/S(=O)(=O)NCc2ccc(cc2)F 8N-037 Cc1ccc(cc1)NS(=O)(=O)/C=C/c2ccc(c(c2)OC)OCc3ccc(cc3)OC 8N-038 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(=O)OC 8N-039 COc1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)Oc4ncccn4 8N-040 CS(=O)(=O)n1ccc(n1)c2ccc(cc2)Oc3ncccn3 8N-041 Cc1ccc(cc1)NS(=O)(=O)/C=C/c2cccn2c3c(cc(cn3)C(F)(F)F)Cl 8N-042 c1c(sc(n1)Cl)CN2CCOCC2 8N-043 c1ccc(c(c1)Oc2ccc(cc2[N+](=O)[O-])/C=C/S(=O)(=O)NCc3ccc(cc3)F)Cl 8N-044 CS(=O)(=O)NCCNc1c(cc(cn1)C(F)(F)F)Cl 8N-045 CC(C)(C)OC(=O)N(CCNc1c(cc(cn1)C(F)(F)F)Cl)S(=O)(=O)C 8N-046 Cc1ccc(cc1)/C=C/S(=O)(=O)NCc2ccc(cc2)F 8N-048 c1ccc2c(c1)c(ccc2Cl)OCc3cnc(s3)Cl 8N-049 COC(=O)c1ccc(cc1)OCc2cnc(s2)Cl 8N-050 CC(C)(C)c1ccc(cc1)COc2ncc(s2)COc3ccccc3 8N-051 c1cnc(nc1)Oc2ccc(cc2)c3ccn(n3)C(=O)c4ccc(cc4)I 8N-052 COc1ccc(cc1)COc2ccc(cc2OC)/C=C/S(=O)(=O)NCc3ccc(cc3)F 8N-053 COc1ccc(cc1OC)NS(=O)(=O)c2ccc(cc2)OCc3cnc(s3)Cl 8N-054 COc1ccc(cc1OC)/C=C/S(=O)(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl 8N-055 c1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccc(cc3)Oc4ncccn4 8N-056 Cc1ccc(cc1)/C=C/S(=O)(=O)Nc2ccc(cc2)C 8N-057 c1cnc(nc1)Oc2ccc(cc2)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Br 8N-058 c1ccc(cc1)C(=O)n2ccc(n2)c3ccc(cc3)Oc4ncccn4 8N-059 Cc1cccc(c1)C(=O)n2ccc(n2)c3ccc(cc3)Oc4ncccn4 8N-060 c1cc(ccc1OCc2cnc(s2)Cl)S(=O)(=O)N3CCOCC3 8N-062 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)OCc3cnc(s3)Cl 8N-063 c1cc2c(cc1/C=C/S(=O)(=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl)OCO2 8N-064 CC(=O)c1cccc(c1)Oc2ncccn2 8N-068 COC(=O)C(Cc1ccc(cc1)O)Nc2ccccc2C(=O)c3ccccc3 8N-069 COc1cc(ccc1OCc2ccc(cc2)Cl)/C=C/S(=O)(=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl 8N-070 COc1cc(ccc1OCc2ccc(cc2)F)/C=C/S(=O)(=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl 8N-074 CC(C)(C)OC(=O)N(c1ccc(cc1)F)S(=O)(=O)C 8N-076 COC(=O)c1c(ccs1)Oc2ncccn2 8N-079 CN(C)/C=C/C(=O)c1cccc(c1)Oc2ncccn2 8N-081 COc1ccc(cc1OC)/C=C/S(=O)(=O)Nc2ccccc2 8N-085 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)OCc3cnc(s3)Cl)OC(F)(F)F 8N-087 c1cc(cc(c1)Br)NS(=O)(=O)c2ccc(cc2)OCc3cnc(s3)Cl 8N-088 COc1ccc(cc1)C(=O)C/C=N/OCc2cnc(s2)Cl 8N-090 c1cnc(nc1)Oc2ccc(cc2)CC#N 8N-091 c1ccc(c(c1)c2nc3ccsc3c(n2)O)Cl 8N-1311 Cc1ccc(cc1)S(=O)(=O)c2cc(nc(n2)c3ccccc3)S(=O)(=O)c4ccc(cc4)C 8N-301S Cc1ccc(cc1)S(=O)(=O)c2cc(nc(n2)c3ccccc3)N4CCOCC4 8N-302S Cc1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)S(=O)(=O)c4ccc(cc4)Cl 8N-303S Cc1ccc(cc1)S(=O)(=O)c2cc(nc(n2)c3ccccc3)Oc4cccc(c4)C(F)(F)F 8N-304S Cc1ccc(cc1)S(=O)(=O)c2cc(nc(n2)c3ccccc3)N4CCCC4 8N-305S c1csc2c1C(=O)NCCS2 8N-326S CN1CCSc2c(ccs2)C1=O 8N-331S CC(C)Sc1nc2ccsc2c(n1)O 8N-342S c1cc(ccc1CSc2nc3ccsc3c(n2)O)Cl 8N-343S Cn1c(=O)c2c(ccs2)nc1SCc3ccc(cc3)Cl 8N-345S c1cc(ccc1CS(=O)(=O)c2nc[nH]n2)Cl 8N-353S c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)c2nc[nH]n2 8N-354S COc1ccc(cc1)CS(=O)(=O)c2nc[nH]n2 8N-355S Cc1ccc2c(c1)C(=O)CCS2 8N-356S c1cc(ccc1CN2CCSc3c(ccs3)C2=O)Cl 8N-357S COC(=O)c1c(ccs1)NC(=O)c2ccccc2 8N-360S c1cc(ccc1CSc2nc[nH]n2)[N+](=O)[O-] 8N-361S c1cc(ccc1CS(=O)(=O)c2nc[nH]n2)[N+](=O)[O-] 8N-362S c1cc(ccc1C(=O)CSc2nc[nH]n2)Cl 8N-363S c1cc(ccc1C(=O)CS(=O)(=O)c2nc[nH]n2)Cl 8N-364S c1cc(c(c(c1)Cl)CSc2nc[nH]n2)F 8N-365S c1cc(c(c(c1)Cl)CS(=O)(=O)c2nc[nH]n2)F 8N-366S Cc1cccc(c1)CSc2nc[nH]n2 8N-367S Cc1cccc(c1)CS(=O)(=O)c2nc[nH]n2 8N-368S Cc1ccc2c(c1)/C(=N/O)/CCS2 8N-370S c1ccc(cc1)CN2CCSc3c(ccs3)C2=O 8N-371S c1cc(ccc1CN2CCSc3c(ccs3)C2=O)F 8N-372S c1cc(c(cc1Cl)Cl)CN2CCSc3c(ccs3)C2=O 8N-373S Cc1ccc(cc1)CN2CCSc3c(ccs3)C2=O 8N-378S c1cc(cc(c1)C(F)(F)F)CN2CCSc3c(ccs3)C2=O 8N-379S COc1ccc(cc1)CN2CCSc3c(ccs3)C2=O 8N-380S c1cc(cc(c1)F)CN2CCSc3c(ccs3)C2=O 8N-381S Cc1ccc2c(c1)NC(=O)CCS2 8N-382S Cc1ccc2c(c1)C(=O)/C(=C/N(C)C)/CS2 8N-387S Cc1ccc(cc1)Sc2nccc(n2)c3ccc(cc3)Cl 8N-501S c1cc(ccc1c2ccnc(n2)Sc3cc(ccc3Cl)Cl)Cl 8N-503S c1cc(ccc1c2ccnc(n2)Sc3ccc(cc3)Cl)Cl 8N-504S c1cc(cc(c1)Sc2nccc(n2)c3ccc(cc3)Cl)C(F)(F)F 8N-505S c1ccc(cc1)Sc2nccc(n2)c3ccc(cc3)Cl 8N-506S c1cc(ccc1c2ccnc(n2)Oc3cc(cc(c3)Cl)Cl)Cl 8N-507S c1cc(ccc1c2ccnc(n2)Oc3cc(ccc3Cl)Cl)Cl 8N-508S Cc1ccc(cc1)Oc2nccc(n2)c3ccc(cc3)Cl 8N-509S COc1ccc(cc1)Oc2nccc(n2)c3ccc(cc3)Cl 8N-511S c1cc(ccc1c2ccnc(n2)Oc3ccc(cc3)F)Cl 8N-512S c1ccc2cc(ccc2c1)Oc3nccc(n3)c4ccc(cc4)Cl 8N-513S c1cc(cnc1)Oc2nccc(n2)c3ccc(cc3)Cl 8N-514S Cc1c2ccccc2nc(c1C(=O)C)N3CCOCC3 8N-520S c1ccc(cc1)C(=NNC(=O)CN2CCOCC2)c3ccccc3 8N-522S Cc1c2ccccc2nc(c1C(=O)C)N3CCCCC3 8N-523S Cc1ccc(cc1)Sc2c(cnc(n2)c3ccccc3)S(=O)(=O)c4ccc(cc4)C 8N-562S CS(=O)(=O)c1cnc(nc1N2CCCC2)c3ccccc3 8N-563S COc1ccc(cc1)Oc2c(cnc(n2)c3ccccc3)S(=O)(=O)c4ccccc4 8N-564S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2Oc3ccccc3)c4ccccc4 8N-566S CS(=O)(=O)c1cnc(nc1Oc2ccc(cc2)F)c3ccccc3 8N-568S CN(C)c1ncc(c(n1)N2CCCC2)S(=O)(=O)c3ccc(cc3)Cl 8N-570S COc1ccc(cn1)n2c(=O)cc(c(n2)C(=O)c3ccccc3)C(F)(F)F 8N-572S Cc1ccc(cc1)Oc2c(cnc(n2)c3ccccc3)S(=O)(=O)c4ccc(cc4)C 8N-575S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2N3CCCCC3)c4ccccc4 8N-576S COc1cccc(c1)Sc2c(cnc(n2)c3ccccc3)S(=O)(=O)C 8N-577S CN(C)c1ncc(c(n1)Oc2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)Cl 8N-578S CS(=O)(=O)c1cnc(nc1N(Cc2ccccc2)c3ccccc3)c4ccccc4 8N-579S CS(=O)(=O)c1cnc(nc1Oc2ccc(cc2)Cl)c3ccccc3 8N-580S Cc1ccc(cc1)Oc2c(cnc(n2)c3ccccc3)S(=O)(=O)C 8N-581S CS(=O)(=O)c1cnc(nc1Sc2ccc(cc2)F)c3ccccc3 8N-582S Cc1ccc(c(c1)C)Sc2c(cnc(n2)c3ccccc3)S(=O)(=O)C 8N-583S CS(=O)(=O)c1cnc(nc1Sc2ccc(cc2)Cl)c3ccccc3 8N-584S Cc1cc(ccc1Oc2c(cnc(n2)c3ccccc3)S(=O)(=O)C)Cl 8N-585S CN(C)c1c(cnc(n1)c2ccccc2)S(=O)(=O)C 8N-586S c1ccc(cc1)c2ncc(c(n2)N3CCCCC3)S(=O)(=O)c4ccccc4 8N-587S CN(C)c1c(cnc(n1)N(C)C)S(=O)(=O)c2ccc(cc2)Cl 8N-588S CN(C)c1ncc(c(n1)Sc2cccc(c2)OC)S(=O)(=O)c3ccc(cc3)Cl 8N-589S COc1cccc(c1)Sc2c(cnc(n2)c3ccccc3)S(=O)(=O)c4ccccc4 8N-590S CC(C)(C)c1ccc(cc1)Sc2c(cnc(n2)c3ccccc3)S(=O)(=O)c4ccccc4 8N-591S Cc1cccc(c1Oc2c(cnc(n2)c3ccccc3)S(=O)(=O)c4ccccc4)C 8N-592S c1ccc(cc1)c2ncc(c(n2)Oc3ccc(cc3F)F)S(=O)(=O)c4ccccc4 8N-593S CN(C)c1c(cnc(n1)c2ccccc2)S(=O)(=O)c3ccccc3 8N-595S CN1CCN(CC1)c2c(cnc(n2)c3ccccc3)S(=O)(=O)c4ccccc4 8N-596S c1ccc(cc1)c2ncc(c(n2)Sc3cccc(c3)C(F)(F)F)S(=O)(=O)c4ccccc4 8N-597S c1ccc(cc1)c2ncc(c(n2)Sc3ccc(cc3)F)S(=O)(=O)c4ccccc4 8N-598S CSc1nc2c(cnn2c3ccccc3)c(n1)O 8N-644S CSc1nc2c(cnn2c3ccccc3)c(n1)Cl 8N-645S CSc1nc2c(cnn2c3ccccc3)c(n1)N4CCOCC4 8N-646S CSc1nc2c(cnn2c3ccccc3)c(n1)N4CCCCC4 8N-647S CSc1nc2c(cnn2c3ccccc3)c(n1)N4CCCC4 8N-648S CNc1c2cnn(c2nc(n1)SC)c3ccccc3 8N-649S COc1c2cnn(c2nc(n1)SC)c3ccccc3 8N-654S Cn1c(=S)n(cn1)c2ccccc2 8N-659S CN(C(=S)Nc1cccc(c1)C(F)(F)F)N 8N-661S COC(=O)c1c(ccs1)Oc2c3cnn(c3nc(n2)SC)c4ccccc4 8N-669S CSc1nc2c(cnn2c3ccccc3)c(n1)Oc4ccc5ccccc5c4 8N-670S Cn1c(=S)n(cn1)c2ccc(cc2)Cl 8N-673S Cn1c(=S)n(cn1)c2cccc(c2)C(F)(F)F 8N-678S Cc1nn(c(=S)n1c2ccc(cc2)Cl)C 8N-680S Cc1ccc(cc1)n2c3c(cn2)c(nc(n3)SC)N4CCOCC4 8N-682S Cc1ccc(cc1)n2c3c(cn2)c(nc(n3)SC)N4CCCCC4 8N-683S c1cnccc1c2nnc(o2)SCCC(=C(F)F)F 8N-700 CC(=O)C1CN(CC1c2ccc(cc2)OC)c3ccccc3 8N-701 CCC(C(=O)NCC(=O)O)SCCC(=C(F)F)F 8N-702 c1cnc(nc1c2cc(sc2Cl)Cl)SCC#N 8N-703 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OC(=O)c3ccc(c(c3)Cl)Cl 8N-705 C=CCSc1nccc(n1)c2cc(sc2Cl)Cl 8N-708 Cc1ccc(cc1)C(=O)C2CN(C(C2C(=O)c3ccc(cc3)C)c4cccs4)C 8N-710 Cc1ccc(c(c1)/C=C/C(=O)OC)C 8N-711 c1ccc(cc1)c2ccc(cc2)C(=O)COc3ccc(cc3)Cc4c(cc(cn4)C(F)(F)F)Cl 8N-712 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)Oc2ccc3c(c2)oc(=O)s3 8N-715 c1ccc(cc1)c2ccc(cc2)/C(=N/OCCOc3cccc(c3)C(F)(F)F)/COc4ccc(cc4)Cc5c(cc(cn5)C(F)(F)F)Cl 8N-716 Cc1ccc(cc1)C(=O)C2CN(C(C2C(=O)c3ccc(cc3)C)c4ccc(cc4Cl)Cl)C 8N-717 c1cc(cc(c1)C(F)(F)F)COc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 8N-718 CC(C)(C)Nc1nc(c(s1)C(=O)c2ccc(cc2Cl)Cl)N 8N-719 CC(C)(C)Nc1nc(c(s1)C(=O)c2ccc(cc2)F)N 8N-720 CN(C)/C=C(/c1c(cc(cn1)C(F)(F)F)Cl)\C(=O)OC 8N-723 COC(=O)C1(CC1)S(=O)(=O)CCC(=C(F)F)F 8N-724 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)OCC(=O)c3ccc(o3)c4ccc(cc4Cl)Cl 8N-727 COc1ccc(cc1)N2CC2c3ccncc3 8N-728 Cc1ccc(cc1)C(=O)C2CN(C(C2C(=O)c3ccc(cc3)C)c4cccc(c4)[N+](=O)[O-])C 8N-729 c1cc(c(cc1Cl)Cl)/C=C/c2[nH]ccn2 8N-733 Cc1c2ccccc2oc(=O)c1C#N 8N-735 CN(C)/C=C/c1c2ccccc2oc(=O)c1C#N 8N-737 c1ccc2c(c1)nc(o2)c3ccc(cc3)NC(=O)c4ccc(cc4)Cl 8N-738 c1c(cnc(c1Cl)SCCC(C(F)(F)Br)(F)Br)C(F)(F)F 8N-740 c1cc(ccc1/C=C/c2[nH]ccn2)Br 8N-741 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)Nc2ccc3c(c2)OCO3 8N-752 c1ccc(cc1)Oc2ccc(cc2)NC(=O)c3cccnc3SCCC(=C(F)F)F 8N-753 c1cc(c(c(c1)Cl)Cc2c(ccc(c2O)C=O)O)Cl 8N-754 c1ccc2c(c1)nc(o2)c3ccc(cc3)NC(=O)c4ccc(cc4)C(F)(F)F 8N-755 c1ccc2c(c1)nc(o2)c3ccc(cc3)N 8N-757 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)Nc2ccc(cc2)F 8N-763 c1ccc(cc1)CNC(=O)c2cccnc2SCCC(=C(F)F)F 8N-764 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)Nc2ccc(cc2)I 8N-765 COCCn1ccc(c(c1=O)Cc2ccccc2)O 8N-766 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)N2CCCCC2 8N-767 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)N2CCOCC2 8N-768 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cccnc3SCCC(=C(F)F)F 8N-769 c1ccc2c(c1)nc(o2)c3ccc(cc3)NC(=O)c4cccc(c4)Cl 8N-770 CC(=O)C(Cc1c(cccc1Cl)F)(Cc2c(cccc2Cl)F)C(=O)C 8N-771 CC(=O)Nc1ccc(cc1)C(=O)O 8N-772 CCn1c(nnc1S)COc2ccc3c(c2)n4ccccc4c3C(=O)OCC 8N-801 CCNC(=O)NNC(=O)COc1ccc2c(c1)n3ccccc3c2C(=O)OCC 8N-802 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)NNC(=S)NCC=C 8N-803 c1ccn2c(c1)c(c3c2cc(cc3)O)C#N 8N-804 COc1ccc2ccccc2c1S(=O)NC3CC3 8N-805 COc1ccc2ccccc2c1S(=O)NCc3cccs3 8N-806 CCOS(=O)c1c2ccccc2ccc1OC 8N-807 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)N 8N-808 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)Nc4ccc(cc4)[N+](=O)[O-] 8N-809 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)NCc4ccco4 8N-810 CN(C)S(=O)(=O)c1ccc(cc1)NS(=O)c2c3ccccc3ccc2OC 8N-811 CN1CCN(CC1)c2ccc(cc2)NS(=O)c3c4ccccc4ccc3OC 8N-812 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)Nc4ccc(cc4)Cl 8N-815 c1ccn2c(c1)c(c3c2cc(cc3)OCc4ccc(cc4)[N+](=O)[O-])C#N 8N-817 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)Nc4ccc(cc4)OC 8N-818 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)Nc4ccc(cc4F)F 8N-819 CCOC(=O)c1c2ccc(cc2n3c1cccc3)OCC(=O)Nc4cccc(c4)C(F)(F)F 8N-820 c1ccn2c(c1)c(c3c2cc(cc3)OCC(=O)N)C#N 8N-821 CCOC(=O)COc1ccc2c(c1)n3ccccc3c2C#N 8N-822 c1ccn2c(c1)c(c3c2cc(cc3)OCC#N)C#N 8N-823 COc1ccc2ccccc2c1SSc3c4ccccc4ccc3OC 8N-824 Cc1c(ccc(c1OC)S(=O)N)OC 8N-826 c1cc(ccc1OCCCF)Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 8P-004 c1cc(sc1)CN(CC(C(F)(F)F)O)CC(C(F)(F)F)O 8P-006 Cc1ccc(cc1)c2c(c(c(c(n2)N)C#N)C#N)C#N 8P-007 c1ccc(cc1)c2cc(c(c(n2)C3CC3)C#N)C(F)(F)F 8P-008 c1c(cnc(n1)N)Cl 8P-009 COc1ccc(cc1)Oc2ncc(s2)C=O 8P-010 Cc1ccc(cc1)c2c(c(c(c(n2)/N=C/N(C)C)C#N)C#N)C#N 8P-011 CN1C(=O)/C(=C\Nc2ccc(cc2)Br)/SC1=O 8P-012 c1cn(cn1)Cc2cnc(s2)Cl 8P-013 Cc1ccc(cc1)S(=O)(=O)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)C 8P-015 COC(=O)c1cc(ccc1N)Cl 8P-016 c1cc([nH]c1)/C=N/O 8P-018 COc1ccc(cc1)C(=O)Nc2ncc(cn2)Br 8P-019 COc1cccc2c1oc(c2)C(=O)N 8P-023 c1cnn(c1)Cc2cnc(s2)Cl 8P-025 COc1cccc2c1oc(c2)C#N 8P-026 c1c(sc(n1)Cl)CN2CCN(CC2)Cc3cnc(s3)Cl 8P-028 c1cc(c(cc1Cl)Cl)CNCC(C(F)(F)F)O 8P-029 c1cc(ccc1CNCC(C(F)(F)F)O)Cl 8P-030 C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1C(=O)OC)Cl 8P-031 CN(C)/C=C/C(=C\C(=O)C(F)(F)F)/Nc1ccc(cc1C(=O)OC)Cl 8P-035 Cn1c2c(c(=O)n(c1=O)C)[nH]c(n2)C3CC=CC3 8P-036 c1ccc(c(c1)CNCC(C(F)(F)F)O)C(F)(F)F 8P-040 CN(C)/C=N/c1c(c(c(c(n1)c2ccc(cc2)Br)C#N)C#N)C#N 8P-042 COc1ccc(c(c1)C=O)OCC#N 8P-046 c1c(sc(n1)Cl)Cn2cncn2 8P-047 c1ccc(c(c1)CNCC(C(F)(F)F)O)Cl 8P-050 c1ccc(cc1)CN(Cc2ccccc2)CC(C(F)(F)F)O 8P-051 C1CN(CCC1O)CC(C(F)(F)F)O 8P-052 c1cc(ccc1/C(=C/C#N)/N)Oc2ccc(c(c2)F)Cl 8P-056 c1cc(cc(c1)Oc2ccc(cc2)C3=C(CCC(=O)N3)C#N)C(F)(F)F 8P-057 CC(C)(C)OC(=O)NC(CO)C(=O)O 8P-058 c1c[nH]c2c1C(=O)CCC2 8P-059 COc1ccc(cc1)Oc2ccc(cc2)/C(=C/C#N)/N 8P-061 C1CC1C2=C(CCC(=O)N2)C#N 8P-062 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2CCCC3=O 8P-063 Cn1c2c(c(=O)n(c1=O)C)[nH]c(n2)C3CCC(C3)O 8P-064 CC(C(=O)OC)Oc1ccc(cc1)C=O 8P-065 c1cc(ccc1C2=C(CCC(=O)N2)C#N)Br 8P-067 c1cc(ccc1c2c(c(c(c(n2)N)C#N)C#N)C#N)Oc3ccc(c(c3)F)Cl 8P-068 CCc1ccc(nc1)CCO 8P-069 COc1ccc(cc1)Oc2ccc(cc2)c3c(c(c(c(n3)N)C#N)C#N)C#N 8P-070 C1CCCN(CC1)CCCN 8P-071 c1ccc(cc1)Cc2[nH]nnn2 8P-072 c1cc(ccc1C2=C(CCC(=O)N2)C#N)Cl 8P-073 Cc1cccnc1NC(=O)C(F)(F)F 8P-307S Cc1cccc(c1)Cn2c(cc3c2nccc3)C(C)(C)C 8P-308S CC(C)(C)c1cc2cccnc2n1Cc3ccc(cc3)OC 8P-309S CC(C)(C)c1cc2cccnc2n1Cc3cccc(c3)F 8P-310S CC(C)(C)c1cc2cccnc2n1C 8P-311S Cc1ccc2c(c1)-c3c4ccccc4nc(c3CS2)N5CCN(CC5)C 8P-318S Cc1ccc(cc1)Cn2c(cc3c2nccc3)C(C)(C)C 8P-320S CC(C)(C)c1cc2cccnc2n1Cc3ccc(cc3Cl)Cl 8P-322S CC(C)(C)c1cc2cccnc2n1Cc3cccc(c3)Cl 8P-323S CC(C)(C)c1cc2cccnc2n1Cc3cccc(c3)C(F)(F)F 8P-324S c1ccc(cc1)CSc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 8P-331S Cc1c(sc2n1ncn2)C(=O)CSc3c(cccc3Cl)Cl 8P-333S Cc1c(sc2n1ncn2)C(=O)CSc3cccc(c3Cl)Cl 8P-334S Cc1c(sc2n1ncn2)C(=O)CSc3ccc(cc3)Br 8P-336S Cc1c(sc2n1ncn2)C(=O)CSc3cccc(c3)C(F)(F)F 8P-337S Cc1c(sc2n1ncn2)C(=O)CSc3ccccc3Cl 8P-338S Cc1c(sc2n1ncn2)C(=O)CSc3ccc(cc3)OC 8P-340S Cc1c(sc2n1ncn2)C(=O)CSc3cccc(c3)OC 8P-341S Cc1ccc(cc1)SCC(=O)c2c(n3c(s2)ncn3)C 8P-344S Cc1c(sc2n1ncn2)C(=O)CSc3ccc(cc3F)F 8P-345S CCSc1c(c(c(s1)C(=O)c2ccccc2)N)C#N 8P-355S Cc1ccc2c(c1)-c3c4ccccc4nc(c3CS2)N5CCOCC5 8P-378S Cc1ccc2c(c1)-c3c4ccccc4nc(c3CS2)N5CCN(CC5)Cc6ccccc6 8P-379S c1ccc(cc1)C(=O)c2c(c(c(s2)SCc3ccc(cc3Cl)Cl)C#N)N 8P-381S c1ccc(cc1)C(=O)c2c(c(c(s2)SCc3ccc(c(c3)Cl)Cl)C#N)N 8P-382S COc1ccc(cc1)CSc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 8P-383S Cc1ccccc1CSc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 8P-384S c1ccc(cc1)C(=O)CSc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 8P-385S c1ccc(cc1)C(=O)c2c(c3c(c(sc3s2)C(=O)c4ccccc4)N)N 8P-387S c1ccc(cc1)C(=O)c2c(c(c(s2)SCc3cccc(c3)F)C#N)N 8P-388S c1ccc(cc1)C(=O)c2c(c(c(s2)SCc3ccc(cc3)F)C#N)N 8P-389S Cc1ccc(cc1)CSc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 8P-390S c1ccc(cc1)C(=O)c2c(c(c(s2)SCc3cccc(c3)Cl)C#N)N 8P-391S c1ccc(cc1)C(=O)c2c(c(c(s2)SCc3ccc(cc3)Cl)C#N)N 8P-392S c1ccc(cc1)C(=O)c2c(c(c(s2)SCc3ccccc3Cl)C#N)N 8P-393S CC(C)(C)c1ccc(cc1)CSc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 8P-394S c1ccc(cc1)C(=O)c2c(c(c(s2)SCC(=O)c3ccc(cc3)F)C#N)N 8P-395S Cc1c(c(no1)c2ccccc2)C(=O)O 8P-396S CSc1c(c(c(s1)C(=O)c2ccccc2)N)C#N 8P-397S CC(C)Sc1c(c(c(s1)C(=O)c2ccccc2)N)C#N 8P-398S C#CCSc1c(c(c(s1)C(=O)c2ccccc2)N)C#N 8P-399S C=CCSc1c(c(c(s1)C(=O)c2ccccc2)N)C#N 8P-400S Cc1c(c(no1)c2ccc(cc2)Cl)C(=O)O 8P-401S c1cc(sc1)c2ccc(nn2)O 8P-501S c1cc(sc1)c2ccc(nn2)Cl 8P-502S Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cc(c4cccc(c4n3)C)C 8P-504S Cc1cccc2c1nc(cc2C)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)F 8P-505S Cn1cc(c(n1)C(F)(F)F)C(=O)NNC(=O)c2ccccc2 8P-506S Cc1ccc(cc1)C(=O)NNC(=O)c2cn(nc2C(F)(F)F)C 8P-507S Cn1cc(c(n1)C(F)(F)F)C(=O)NNC(=O)c2cccs2 8P-508S Cn1cc(c(n1)C(F)(F)F)c2nnc(o2)c3cccs3 8P-509S Cn1cc(c(n1)C(F)(F)F)c2nnc(o2)c3ccccc3 8P-510S Cc1ccc(cc1)c2nnc(o2)c3cn(nc3C(F)(F)F)C 8P-511S Cc1cccc2c1nc(cc2C)N3CCN(CC3)c4ccc(cn4)C(=O)OC 8P-512S Cc1cccc2c1nc(cc2C)N3CCN(CC3)S(=O)(=O)c4ccccc4 8P-514S Cc1cccc2c1nc(cc2C)N3CCN(CC3)S(=O)(=O)Cc4ccccc4 8P-515S Cc1cccc2c1nc(cc2C)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Br 8P-517S Cc1cccc2c1nc(cc2C)N3CCN(CC3)c4ncccn4 8P-521S Cc1cc(nc(c1C#N)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)F)C 8P-522S Cc1cc(nc(c1C#N)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Br)C 8P-523S Cc1cc(nc(c1C#N)N2CCN(CC2)S(=O)(=O)Cc3ccccc3)C 8P-524S Cc1ccc(cc1)NC(=O)N2CCC(CC2)c3nc4ccccc4s3 8P-526S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)Nc4ccc(cc4)F 8P-527S c1cc(sc1)c2ccc(nn2)N3CCN(CC3)c4ncccn4 8P-528S Cc1cccc(c1)NC(=O)N2CCC(CC2)c3nc4ccccc4s3 8P-530S c1ccc(cc1)NC(=O)N2CCC(CC2)c3nc4ccccc4s3 8P-531S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)Nc4cccc(c4)Cl 8P-532S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)Nc4ccc(cc4)Cl 8P-533S Cc1cc(nc(c1C#N)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)F)C 8P-534S Cc1cc(nc(c1C#N)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)Br)C 8P-535S Cc1cc(nc(c1C#N)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)NC(=O)C)C 8P-536S Cc1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3c(c(cc(n3)C)C)C#N 8P-537S Cc1cc(nc(c1C#N)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3Cl)Cl)C 8P-538S Cc1cc(nc(c1C#N)N2CCCN(CC2)S(=O)(=O)Cc3ccccc3)C 8P-539S CCNC(=O)N1CCC(CC1)c2nc3ccccc3s2 8P-540S C=CCNC(=O)N1CCC(CC1)c2nc3ccccc3s2 8P-541S CCCNC(=O)N1CCC(CC1)c2nc3ccccc3s2 8P-542S CC(C)NC(=O)N1CCC(CC1)c2nc3ccccc3s2 8P-543S c1ccc2c(c1)c(=O)c3cc(ccc3s2)N 8P-567S COC(=O)c1ccc(o1)[N+](=O)[O-] 8P-568S COc1cccc(c1)C(=O)Nc2ccc3c(c2)c(=O)c4ccccc4s3 8P-569S c1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4ccc(cc4)F 8P-570S Cc1cccn2c1nc(c2/C=N/OC(=O)c3cccs3)c4ccc(cc4)Cl 8P-647S Cc1ccn2c(c1)nc(c2/C=N/OC)c3ccc(cc3)Cl 8P-649S Cc1ccn2c(c1)nc(c2/C=N/OCc3ccc(cc3Cl)Cl)c4ccc(cc4)Cl 8P-650S Cc1cccc(c1)NC(=O)O/N=C/c2c(nc3n2ccc(c3)C)c4ccc(cc4)Cl 8P-659S Cc1ccn2c(c1)nc(c2/C=N/OC(=O)C3CC3)c4ccc(cc4)Cl 8P-660S Cc1ccn2c(c1)nc(c2/C=N/OC(=O)c3ccc(cc3)F)c4ccc(cc4)Cl 8P-662S Cc1ccn2c(c1)nc(c2/C=N/OC(=O)c3cccc(c3)OC)c4ccc(cc4)Cl 8P-663S Cc1cccc(c1)CO/N=C/c2c(nc3n2cc(cc3)Cl)c4ccccc4 8P-664S Cc1ccc(cc1)C(=O)O/N=C/c2c(nc3n2cc(cc3)Cl)c4ccccc4 8P-665S c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)/C=N/OC(=O)c4ccc(cc4)Cl 8P-666S c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)/C=N/OC(=O)c4cccs4 8P-667S c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)/C=N/OCc4ccc(cc4Cl)Cl 8P-668S c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)/C=N/OCc4ccc(cc4)F 8P-670S c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)/C=N/OCc4cccc(c4)F 8P-671S Cc1ccn2c(c1)nc(c2/C=N/OCc3ccc(cc3)F)c4ccc(cc4)Cl 8P-676S Cc1ccn2c(c1)nc(c2/C=N/OCc3cccc(c3)F)c4ccc(cc4)Cl 8P-677S Cc1cccc(c1)CO/N=C/c2c(nc3n2ccc(c3)C)c4ccc(cc4)Cl 8P-678S Cc1cccc(c1)CO/N=C/c2c(nc3n2cccc3C)c4ccc(cc4)Cl 8P-679S Cc1cccn2c1nc(c2/C=N/OCc3cccc(c3)F)c4ccc(cc4)Cl 8P-680S Cc1cccn2c1nc(c2/C=N/OCc3ccc(cc3)F)c4ccc(cc4)Cl 8P-681S Cc1ccn2c(c1)nc(c2/C=N/OCc3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl 8P-682S Cc1cccn2c1nc(c2/C=N/OC(=O)C3CC3)c4ccc(cc4)Cl 8P-683S c1c(cnc(c1Cl)c2c(nc3cc(c(cc3n2)Cl)Cl)O)C(F)(F)F 8P-701 Cc1c(sc(n1)c2ccccn2)C(=O)C.Cl 8P-702 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccc(c(=O)[nH]3)C(=O)N 8P-703 Cc1cccc(n1)n2cc(nc2)C(=O)N/N=C/c3ccccc3 8P-705 Cc1cccc(n1)n2cc(nc2)C(=O)N/N=C/c3ccc(c(c3)OC)O 8P-706 CC(=O)C(Cc1ccc(cc1)Cl)Cc2ccc(cc2)Cl 8P-708 CN(C)/C=C/C(=O)C(Cc1ccc(cc1)Cl)Cc2ccc(cc2)Cl 8P-709 Cc1c(sc(n1)c2ccccn2)C(=O)C 8P-710 Cc1c(sc(n1)c2ccncc2)C(=O)/C=C/N(C)C 8P-711 c1cc(c(cc1Cl)Cl)Cc2c(ccn(c2=O)C3CCCC3)O 8P-714 Cc1cccc(n1)n2cc(nc2)C(=O)NNS(=O)(=O)c3ccc4ccccc4c3 8P-717 Cc1cccc(n1)n2cc(nc2)C(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F 8P-718 Cc1c(sc(n1)c2ccc(c(c2)OC)OC)C(=O)C 8P-719 Cc1c(sc(n1)c2cccnc2)C(=O)/C=C/N(C)C 8P-724 CCOC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NCc2ccc(o2)C 8P-727 Cc1ccc(o1)CNC(=O)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCc3ccc(o3)C 8P-728 C/[N+](=C/c1ccc(c(c1O)Cc2c(cccc2Cl)F)O)/[O-] 8P-729 Cc1c(sc(n1)c2ccncc2)c3ccc(c(=O)[nH]3)C(=O)N 8P-730 C[NH+]1CCOCC1.c1ccc(cc1)C2CC(=O)NC(=C2C#N)[C-](C#N)C#N 8P-731 c1cc(cc(c1)Cl)COCCO 8P-733 CCOC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)NCCc2c[nH]c3c2cccc3 8P-736 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C(c3c(cc(cn3)C(F)(F)F)Cl)C(=O)NCCc4c[nH]c5c4cccc5 8P-737 CC(C)(C)c1cc(cc(c1/C=N/Nc2cccc3c2nccc3)C(C)(C)C)O 8P-800 C/C(=N\Nc1cccc2c1[nH+]ccc2)/C(=O)O.[Cl-] 8P-801 C/C(=N\Nc1cccc2c1nccc2)/c3ccccc3O 8P-802 c1ccc(cc1)C(=NNc2cccc3c2nccc3)c4ccccc4 8P-803 C/C(=N\Nc1cccc2c1nccc2)/c3cccc4c3cccc4 8P-804 C/C(=N\Nc1cccc2c1nccc2)/c3ccc(cc3)N 8P-805 c1cc2ccc[nH+]c2c(c1)N[NH3+].[Cl-].[Cl-] 8P-806 Cc1csc2c1nc[nH]c2=O 8P-807 CCOC(=O)C(=CNc1nc(cs1)c2ccc(cc2)C)C(=O)OCC 8P-808 c1cc(ccc1CSc2ccc(cc2)F)CSc3ccc(cc3)F 8P-809 Cc1nc(cs1)c2ccccc2 8P-810 CCOC(=O)/C(=C/Nc1nc(cs1)c2ccc3ccccc3c2)/C#N 8P-811 c1cc(cc(c1)N[NH3+])C#N.[Cl-] 8P-812 Cc1ccc(cc1)c2csc(n2)NC(=O)Nc3ccc(cc3)Cl 8P-813 Cc1ccc(cc1)c2csc(n2)NC(=O)Nc3ccccc3 8P-814 CSc1nc(cc(n1)Cl)Nc2ccc(cc2)O 8P-815 COc1ccc(cc1)Sc2cc(nc(n2)SC)Cl 8P-816 CN(Cc1ccccc1)c2cc(nc(n2)SC)Cl 8P-817 CN(c1ccccc1)c2cc(nc(n2)SC)Cl 8P-818 Cc1cccc(c1C)N2CCN(CC2)c3cc(nc(n3)N)Sc4ccc5ccccc5c4 8P-819 c1ccc(cc1)NC(=O)Nc2nc(cs2)c3ccc(cc3)F 8P-820 CCOC(=O)c1c(nc(s1)n2cccc2)c3ccccc3 8P-821 c1cc(ccc1F)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F 8P-822 CCOC(=O)c1c(nn(c1C)c2cccc3c2nccc3)C 8P-823 CCOC(=O)c1c(sc(n1)N)C(=O)OCC 8P-824 CCOC(=O)CC1C(=O)NCCN1C(=O)Nc2ccc(cc2)Cl 8P-825 c1ccc(cc1)NC(=O)Nc2nc(cs2)c3ccc4ccccc4c3 8P-826 CSc1nc(cc2n1nnn2)Cl 8P-827 CSc1nc(cc(n1)Sc2ccccc2)Sc3ccccc3 8P-828 C[n+]1ccc(cc1)C(=O)NNC(=O)c2cc[n+](cc2)C.[I-].[I-] 8P-829 c1cc(ccc1CSc2cc(nc(n2)N)Cl)CSc3cc(nc(n3)N)Cl 8P-830 CC(C)(C)c1c(sc(n1)NC(=O)Nc2ccccc2)Br 8P-831 c1ccc2c(c1)c(c[nH]2)/C=N/Nc3cccc4c3nccc4 8P-832 c1ccc2c(c1)cccc2c3csc(n3)NC(=O)Nc4ccc(cc4)Cl 8P-834 Cc1csc(c1NC(=O)Nc2ccccc2)C(=O)OC 8P-835 c1ccc(cc1)NC(=O)NC2=NC(=O)CS2 8P-836 CSc1nc(cc(n1)Sc2ccccc2)N3CCCc4c3cccc4 8P-837 COc1cccc(c1O)/C=N/Nc2cccc3c2[nH+]ccc3.[Cl-] 8P-838 Cc1nccn1c2cc(nc(n2)SC)Cl 8P-839 COC(=O)N/N=C\c1cccc(c1)O 8P-840 CSc1nc(cc(n1)Cl)NCCNc2cc(nc(n2)SC)Cl 8P-841 c1ccc(cc1)CSc2cc(nc(n2)N)Cl 8P-842 CC(C)(C)c1c(sc(n1)N)C(=O)OC 8P-843 c1cnccc1C(=O)NNC(=O)c2ccncc2 8P-844 CCOC(=O)C(=CNc1nc(cs1)c2ccc3ccccc3c2)C(=O)OCC 8P-845 C/C(=N/Nc1cccc2c1[nH+]ccc2)/c3ccc(cc3)Cl.[Cl-] 8P-847 Cc1ccc(cc1)/C(=N/Nc2cccc3c2nccc3)/C 8P-848 Cc1cc(c(s1)C)/C(=N\Nc2cccc3c2nccc3)/C 8P-849 c1ccc(c(c1)/C=N/Nc2cccc3c2[nH+]ccc3)Cl.[Cl-] 8P-850 c1ccc(cc1)/C=N/Nc2cccc3c2nccc3 8P-851 CSc1nc(cc(n1)Cl)NCc2ccco2 8P-852 CCNc1cc(nc(n1)SC)N2CCOCC2 8P-853 CNc1cc(nc(n1)SC)Cl 8P-854 c1cc2cccnc2c(c1)N/N=C/c3cccc(c3Cl)Cl 8P-855 c1ccc(c(c1)/C=N/Nc2cccc3c2[nH+]ccc3)O.[Cl-] 8P-856 c1cc2ccc[nH+]c2c(c1)N/N=C/c3ccc(cc3)[N+](=O)[O-].[Cl-] 8P-857 c1cc2cccnc2c(c1)N/N=C/c3cccc(c3)O 8P-858 C/C(=N\Nc1cccc2c1[nH+]ccc2)/c3ccc(cc3)F.[Cl-] 8P-859 c1ccc(c(c1)N2CCN(CC2)CC(C(F)(F)F)O)F 8P-901 C1CCCN(CC1)C(=O)C(F)(F)Cl 8P-902 c1ccn(c1)c2ncc(cn2)Br 8P-903 c1ccc(cc1)CN2CCN(CC2)C(=O)C(F)(F)Cl 8P-904 c1ccc2c(c1)ccn2Cc3cnc(s3)Cl 8P-905 c1cc2cn[nH]c2c(c1)[N+](=O)[O-] 8P-906 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(C(F)(F)F)O 8P-908 c1cc(cc(c1)N2CCN(CC2)CC(C(F)(F)F)O)C(F)(F)F 8P-909 c1cc(ccc1N2CCN(CC2)CC(C(F)(F)F)O)[N+](=O)[O-] 8P-910 CCOC(=O)C1CCN(CC1)CC(C(F)(F)F)O 8P-916 COc1cccc(c1OCC#N)C=O 8P-917 CC(=O)c1cc2cccc(c2o1)OC 8P-918 c1cc2ccn(c2nc1)Cc3cnc(s3)Cl 8P-919 c1ccc2c(c1)CCCN2Cc3cnc(s3)Cl 8P-920 c1ccc(cc1)CNC(=O)C(F)(F)Cl 8P-923 c1ccc2c(c1)CCN(C2)C(=O)C(F)(F)Cl 8P-924 C1CN(CCC1O)C(=O)C(F)(F)Cl 8P-925 c1ccc(cc1)CN(CC(C(F)(F)F)O)C(=O)Nc2ccccc2 8P-926 Cc1ccc(n1c2ncc(cn2)Br)C 8P-927 c1ccc(cc1)C(CO)NC(=O)C(F)(Br)Br 8P-929 c1ccc(cc1)NC(=O)N(Cc2ccc(cc2)Cl)CC(C(F)(F)F)O 8P-932 c1ccc(cc1)c2nnc(n2N)c3ccccc3 8P-933 c1cc(cc(c1)F)NC(=O)N(Cc2ccc(cc2)Cl)CC(C(F)(F)F)O 8P-934 c1cc(cc(c1)NC(=S)N(Cc2ccc(cc2Cl)Cl)CC(C(F)(F)F)O)C(F)(F)F 8P-936 Cc1ccc(n1c2c(ccs2)c3cc4nc(cc(n4n3)C(F)(F)F)C(F)(F)F)C 8R-0001 CCOC(=O)c1ccc(cc1)n2c(ccc2C)C 8R-0002 Cc1cc2nccc(n2n1)c3ccc(cc3)F 8R-0003 CCOC(=O)c1ccc(cc1)n2c(cc(c2C)C=O)C 8R-0004 Cc1cc(c(n1n2cnnc2)C)C=C(C#N)C#N 8R-0005 CC(CC(=O)Nc1ccccc1C(F)(F)F)N2CCCC2 8R-0006 Cc1ccc(n1c2c(ccs2)c3cc4nccc(n4n3)c5ccc(cc5)F)C 8R-0007 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3cccs3 8R-0008 CCN\1C(=O)/C(=C/c2ccc(cc2)OC)/S/C1=N\n3cnnc3 8R-0009 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccccc3 8R-0010 Cc1ccc(n1c2c(ccs2)c3cc4nc(cc(n4n3)O)C)C 8R-0011 Cc1cc2nccc(n2n1)c3ccc(cc3Cl)Cl 8R-0012 COc1ccc(cc1)/C=C\2/C(=O)N(/C(=N/n3cnnc3)/S2)c4ccccc4 8R-0017 Cc1ccc(n1c2c(ccs2)c3cc4nc(c(c(n4n3)C)Cl)C)C 8R-0018 Cc1ccc(n1c2c(ccs2)c3cc4nc(c(c(n4n3)O)Cl)C)C 8R-0019 Cc1ccc(n1c2c(ccs2)c3cc4nccc(n4n3)c5ccc(cc5Cl)Cl)C 8R-0020 Cc1cc(c2nncn2n1)OC(=O)C 8R-0021 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccccc5)C 8R-0023 Cc1ccc(n1c2ccsc2c3cc4nc(c(c(n4n3)C)Cc5c(cccc5Cl)F)C)C 8R-0024 Cc1cc2nccc(n2n1)c3ccccc3 8R-0025 CC(=O)CC(=O)Nc1cc(ccc1OC)OC 8R-0028 Cc1ccc(cc1)c2ccnn2c3nc(cs3)c4ccc(cc4)Br 8R-0029 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccco3 8R-0034 c1cc(c(nc1)Sc2ccc(cc2)Cl)/C=C/C(=O)O 8R-0036 c1cc(ccc1c2csc(n2)NN)Br 8R-0038 CCN1C(S/C(=C\N(C)C)/C1=O)Nn2cnnc2 8R-0039 Cc1ccc(n1c2c(ccs2)c3cc4nc(cc(n4n3)O)COC)C 8R-0040 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)CSc5ccccc5)C 8R-0041 c1cc(ccc1c2ccnn2c3nc(cs3)c4ccc(cc4)Br)F 8R-0042 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)Br)C 8R-0045 COC(=O)c1cc2ccccc2o1 8R-0046 CC1=C(C(C(=C(N1)C)C(=O)OCc2ccccc2)c3ccc(cc3Cl)Cl)C(=O)OC 8R-0049 CC1=C(C(C(=C(N1)C)C(=O)OCc2ccccc2)c3ccc(cc3)F)C(=O)C 8R-0051 Cc1ccc(cc1)c2ccnc3n2nc(c3)c4c(ccs4)n5c(ccc5C)C 8R-0052 Cc1c(c2nccc(n2n1)c3ccc(cc3)F)Br 8R-0053 CC1=C(C(C(=C(N1)C)C(=O)OCc2ccccc2)c3ccc(cc3)[N+](=O)[O-])C(=O)C 8R-0054 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)CCl)C 8R-0055 Cc1c(c2nccc(n2n1)c3ccc(cc3)F)Cl 8R-0056 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)CN5CCCCC5)C 8R-0058 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)C)C 8R-0059 Cc1ccc(cc1)c2ccnc3n2nc(c3)C 8R-0060 Cc1cc2nccc(n2n1)c3cccnc3 8R-0066 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5cccnc5)C 8R-0067 Cc1cc(n(n1)c2nc(cs2)c3ccc(c(c3)Cl)Cl)C 8R-0074 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)/C=C/c5ccc(cc5Cl)Cl)C 8R-0075 Cc1cc2nccc(n2n1)/C=C/c3ccc(cc3Cl)Cl 8R-0076 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)C)c5ccc(c(c5)OC)OC)C 8R-0077 Cc1c(c(n(n1)c2nc(c(s2)Cl)c3ccc(c(c3)Cl)Cl)C)Cl 8R-0078 Cc1c(c(n(n1)c2nc(c(s2)Br)c3ccc(c(c3)Cl)Cl)C)Br 8R-0082 c1cc(cc(c1)F)CN2CCC(CC2)C(=O)NNC(=O)c3cccc(c3)Cl 8R-0200 c1c(c(cc2c1OCO2)Br)C#N 8R-0201 c1cc(c(cc1F)F)OC(=O)/C=C/c2cc3c(cc2Br)OCO3 8R-0202 c1cc(ccc1OC(=O)/C=C/c2cc3c(cc2Br)OCO3)F 8R-0203 c1cc(c(cc1OC(=O)/C=C/c2cc3c(cc2Br)OCO3)Cl)Cl 8R-0204 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 8R-0207 CC(C)(C)c1ccc(cc1)S(=O)(=O)NNC(=O)C2CCN(CC2)Cc3cccc(c3)F 8R-0208 c1cc(cc(c1)F)CN2CCC(CC2)C(=O)NNS(=O)(=O)c3ccc(cc3)F 8R-0209 CC(C)CC(=O)c1cc([nH]c1)C(=O)C(Cl)(Cl)Cl 8R-0211 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCCCN2CCOCC2 8R-0212 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCC2CCCO2 8R-0213 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCc2ccccc2 8R-0214 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCCCN(C)C 8R-0215 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCC3CCCO3 8R-0216 CC(C)C(C(=O)OC)NC(=O)/C(=C/c1cccs1)/c2ccccc2 8R-0217 c1c(cc(cc1Cl)Cl)OC(=O)/C=C/c2cc3c(cc2Br)OCO3 8R-0218 c1cc(cc(c1)F)OC(=O)/C=C/c2cc3c(cc2Br)OCO3 8R-0219 c1cc(cc(c1)F)CN2CCC(CC2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl 8R-0221 c1ccc(cc1)NC(=O)NNC(=O)C2CC(=NO2)c3cccs3 8R-0222 c1cc(sc1)C2=NOC(C2)C(=O)NNC(=O)NC3CCCCC3 8R-0223 Cc1ccc(cc1)NC(=O)NNC(=O)C2CC(=NO2)c3cccs3 8R-0224 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 8R-0225 c1cc(sc1)C2=NOC(C2)C(=O)NNC(=O)Nc3ccc(cc3)Cl 8R-0226 CCNC(=O)NNC(=O)C1CC(=NO1)c2cccs2 8R-0227 COCCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)OC 8R-0228 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCc2ccccc2OC 8R-0229 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCc2cccs2 8R-0230 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCc2cccc(c2)C(F)(F)F 8R-0231 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)N)F 8R-0232 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCCCn2ccnc2 8R-0233 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCCc2ccccn2 8R-0237 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3ccco3 8R-0238 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3 8R-0239 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCCOC 8R-0240 CC(C)CC(=O)c1cc([nH]c1)C(=O)N2CCN(CC2)Cc3ccccc3 8R-0241 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCc2cccnc2 8R-0243 CCC(C)c1ccc(cc1)OC(=O)/C=C/c2cc3c(cc2Br)OCO3 8R-0245 c1cc(c(cc1OC(=O)/C=C/c2cc3c(cc2Br)OCO3)Cl)Br 8R-0246 c1cc(cc(c1)Cl)OC(=O)/C=C/c2cc3c(cc2Br)OCO3 8R-0248 CCC(=O)c1cc([nH]c1)C(=O)NCc2ccco2 8R-0252 CCC(=O)c1cc([nH]c1)C(=O)NCc2cccc(c2)C(F)(F)F 8R-0253 CCC(=O)c1cc([nH]c1)C(=O)NCCOC 8R-0254 CCC(=O)c1cc([nH]c1)C(=O)NCCCN2CCOCC2 8R-0255 CCC(=O)c1cc([nH]c1)C(=O)NCc2cccnc2 8R-0256 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccs3 8R-0257 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccnc3 8R-0258 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCc2ccc(cc2)F 8R-0260 c1cc2c(cc1N)NC3C2CCCC3 8R-0261 CC(C)N(C(C)C)C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)OC 8R-0263 CCC(C)(C)c1ccc(c(c1)C(C)(C)CC)OCCCCNC(=O)c2cc(c[nH]2)C(=O)CC(C)C 8R-0264 CC(C)CC(=O)c1cc([nH]c1)C(=O)NCC#C 8R-0265 COc1ccc(cc1Cl)CNC(=O)c2cccc(c2)[N+](=O)[O-] 8R-0266 COc1ccc(cc1Cl)CNC(=O)c2cccc(c2)C(F)(F)F 8R-0267 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCc3ccc(c(c3)Cl)OC 8R-0268 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCc3ccc(c(c3)Cl)OC 8R-0269 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3ccccc3 8R-0270 CC(C(=O)O)SC1=Nc2cc(c(cc2C3=NC(=O)C(N31)CC4CCCCC4)OC)OC 8R-0271 COc1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)c3ccc(cc3)OC 8R-0272 CC(C)CC(=O)c1cc([nH]c1)C(=O)OC 8R-0273 CCC(=O)c1cc([nH]c1)C(=O)NCC2CCCO2 8R-0274 CCC(=O)c1cc([nH]c1)C(=O)NCCCn2ccnc2 8R-0275 CCC(=O)c1cc([nH]c1)C(=O)NCc2ccccc2OC 8R-0276 COC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 8R-0277 c1cc(cc(c1)Br)C(=O)c2cc([nH]c2)C(=O)C(Cl)(Cl)Cl 8R-0278 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)CC 8R-0279 CCC(=O)c1cc([nH]c1)C(=O)NCCc2ccccn2 8R-0280 CCC(=O)c1cc([nH]c1)C(=O)NCc2ccc(cc2)OC 8R-0281 CCOC(=O)CC1COc2ccccc2N1C(=O)c3ccc(cc3)C 8R-0283 COC(=O)c1ccc[nH]1 8R-0284 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3cccc(c3)C(F)(F)F 8R-0285 CC(C)CC(=O)c1cc([nH]c1)C(=O)O 8R-0286 CCCC(=O)c1cc([nH]c1)C(=O)C(Cl)(Cl)Cl 8R-0290 COC(=O)C1CCN(CC1)Cc2cnc(s2)Cl 8R-0291 C1CC1C(=O)N2CCN=C(C=C2)C(F)(F)F 8R-0293 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F)C 8R-0295 CCCC(=O)c1cc([nH]c1)C(=O)NCc2cccc(c2)C(F)(F)F 8R-0296 CCCC(=O)c1cc([nH]c1)C(=O)NCCc2ccccn2 8R-0297 CCCC(=O)c1cc([nH]c1)C(=O)NCc2ccc(cc2)F 8R-0298 CCCC(=O)c1cc([nH]c1)C(=O)NCc2cccs2 8R-0299 CCCC(=O)c1cc([nH]c1)C(=O)NCCCN(C)C 8R-0300 CCC(=O)c1cc([nH]c1)C(=O)NCc2cccs2 8R-0302 c1cc(ccc1C=O)OCC#N 8R-0303 CCCC(=O)c1cc([nH]c1)C(=O)NCCCn2ccnc2 8R-0305 CCCC(=O)c1cc([nH]c1)C(=O)NCc2ccco2 8R-0306 CC(=C(C#N)C#N)c1cccs1 8R-0307 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SC/C=C/c4ccccc4 8R-0308 CCCC(=O)c1cc([nH]c1)C(=O)NCCCN2CCOCC2 8R-0309 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4ccc(c(c4)Cl)Cl 8R-0310 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN=C(C=C3)C(F)(F)F 8R-0311 c1cc(ccc1S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F)Br 8R-0312 CCOC(=O)CC1COc2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F 8R-0313 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4csc(n4)Cl 8R-0317 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)NCc3ccc(cc3)F 8R-0318 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)OC 8R-0319 CCCCCCCCSC1=Nc2cc(c(cc2C3=NC(=O)C(N31)C(C)C)OC)OC 8R-0320 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)N 8R-0321 CCCC(=O)c1cc([nH]c1)C(=O)NCc2cccnc2 8R-0322 c1ccc(cc1)C2C(c3ccccc3C(=O)O2)C(=O)O 8R-0323 Cc1c(sc(n1)Nc2cccc(c2Cl)Cl)C(=O)C 8R-0327 Cc1c(sc(n1)Nc2ccc(cc2)C(F)(F)F)C(=O)C 8R-0328 c1cc(sc1)c2cc[nH]c(=O)c2C#N 8R-0329 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)OC 8R-0330 CCC(CC)C(=O)c1cc([nH]c1)C(=O)C(Cl)(Cl)Cl 8R-0335 CC(=O)c1cnc(s1)Nc2ccc(cc2)C(F)(F)F 8R-0336 CC(=O)c1cnc(s1)Nc2cccc(c2Cl)Cl 8R-0337 c1ccc2c(c1)ccc3c2cc(o3)C(=O)NNC(=O)c4cccc(c4)Cl 8R-0338 COc1ccc(cc1Cl)CNc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] 8R-0339 COc1ccc(cc1Cl)CNc2ccc(cc2[N+](=O)[O-])Cl 8R-0340 COc1ccc(cc1Cl)CNc2c(cccc2Cl)[N+](=O)[O-] 8R-0341 CN(CCOc1ccc(cc1)c2ccn(n2)c3ncccn3)c4ccccn4 8R-0343 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2cccc(c2)C(F)(F)F 8R-0344 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2ccco2 8R-0345 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2ccccc2 8R-0346 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCCCn2ccnc2 8R-0347 CC(=C(C#N)C#N)c1ccco1 8R-0348 CN(C)/C=N/C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)OC 8R-0350 CCCC(=O)c1cc([nH]c1)C(=O)N2CCOCC2 8R-0352 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2cccnc2 8R-0353 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCCCN2CCOCC2 8R-0354 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCCCN(C)C 8R-0355 CN(C)/C=N/C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)F 8R-0357 CN(C)/C=C/C(=O)c1cnc(s1)N(C)c2ccc(cc2)C(F)(F)F 8R-0358 c1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)c3c(cccc3F)F 8R-0359 c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cc(c[nH]2)C(=O)c3c(cccc3F)F 8R-0362 COc1ccc(cc1Cl)CNc2ccc(cc2[N+](=O)[O-])C(F)(F)F 8R-0363 CC1=C(C(CC(=O)N1)c2ccccc2Cl)C(=O)C 8R-0364 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2ccccc2OC 8R-0365 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2ccc(cc2)F 8R-0366 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5cccc(c5)C(F)(F)F 8R-0367 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccc(cc5Cl)Cl 8R-0368 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccc(cc5)F 8R-0369 c1cc(oc1)c2cc[nH]c(=O)c2C#N 8R-0370 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4ccc(cc4Cl)Cl 8R-0371 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4ccc(cc4)OC 8R-0372 Cc1ccccc1CSC2=Nc3cc(c(cc3C4=NC(=O)C(N42)C(C)C)OC)OC 8R-0373 Cc1ccc(cc1)Cn2ccc(c(c2=O)C#N)c3cccs3 8R-0374 CC(=O)c1cnc(s1)N(C)c2cccc(c2Cl)Cl 8R-0375 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5cc(ccc5Cl)Cl 8R-0376 c1ccc2c(c1)ccc3c2cc(o3)C(=O)NNC(=O)c4ccco4 8R-0377 COc1ccc(cc1)C(=O)Nc2ccc3c(c2)NC4C3CCCC4 8R-0378 COc1ccc(cc1Cl)CNS(=O)(=O)c2ccc(cc2)F 8R-0379 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4ccc(cc4)F 8R-0380 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4ccccc4C(F)(F)F 8R-0381 CC(C)(C)c1cc(=O)[nH]c(n1)SCc2ccccc2 8R-0382 CC(C)C1C(=O)N=C2N1C(=Nc3c2cc(c(c3)OC)OC)SCc4cccc(c4)C(F)(F)F 8R-0383 CC(C)(C)c1cc(=O)[nH]c(n1)SCc2cccc(c2)F 8R-0384 CC(C)(C)c1cc(=O)[nH]c(n1)SCc2cccc(c2)C(F)(F)F 8R-0385 c1cc(cc(c1)[N+](=O)[O-])C(=O)N2CCN=C(C=C2)C(F)(F)F 8R-0387 c1cc(oc1)c2ccn(c(=O)c2C#N)Cc3ccc(cc3)F 8R-0388 CC(C)(C)c1cc(=O)[nH]c(n1)SCc2ccccc2Cl 8R-0392 CC(C)(C)c1ccc(cc1)CSc2[nH]c(=O)cc(n2)C(C)(C)C 8R-0393 c1cc(c(nc1)N2CCOCC2)[N+](=O)[O-] 8R-0394 c1ccc2c(c1)N(C(CO2)CC(=O)O)C(=O)c3ccsc3 8R-0395 CCOC(=O)CC1COc2ccccc2N1C(=O)c3cccc(c3)[N+](=O)[O-] 8R-0396 CCOC(=O)CC1COc2ccccc2N1C(=O)c3ccc(cc3)F 8R-0398 c1cc(cnc1)C2=NOC(C2)C(=O)NNC(=S)Nc3ccc(cc3F)Br 8R-0399 c1cc2c(cc1NS(=O)(=O)c3ccc(c(c3)Cl)Cl)nccn2 8R-0600 COc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)nccn3 8R-0601 COC(=O)CC(c1ccc2c(c1)OCO2)N 8R-0602 CCOc1c(ccc(n1)c2ccc(cc2Cl)Cl)C#N 8R-0603 CCOC(=O)N1CCN(CC1)c2ncc(s2)Cn3cccn3 8R-0604 c1cc(sc1)c2ccnc(n2)N 8R-0605 C/C(=N\O)/C1CC(C1(C)C)CC(=O)O 8R-0610 CCOc1c(ccc(n1)c2ccc(cc2Cl)Cl)C(=O)N 8R-0611 c1ccc(c(c1)C(=O)Nc2nccc(n2)c3cccs3)Cl 8R-0612 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc(c1)OC 8R-0613 Cc1ccc(cc1)C(CC(=O)O)NC(=O)OC(C)(C)C 8R-0614 c1cc(cc(c1)[N+](=O)[O-])C(CC(=O)O)N 8R-0617 c1ccn(c1)c2nccc(n2)c3cccs3 8R-0618 c1ccn(c1)c2ccc3c(c2)nccn3 8R-0620 Cc1cccc(c1)C(CC(=O)O)N2Cc3ccccc3C2=O 8R-0621 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3cccc(c3)F 8R-0622 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(c(c3)Cl)Cl 8R-0623 Cc1cc([nH]c(=O)c1C#N)c2ccccc2 8R-0624 c1cc(ccc1N2CCN(CC2)Cc3cnc(s3)Cl)F 8R-0625 Cc1ccc(n1c2nccc(n2)c3cccs3)C 8R-0627 Cc1c(ccc(n1)N2CCN(CC2)c3ccc(cc3)F)C(=O)C 8R-0628 Cc1cc(nc2c1c3nc(cc(n3n2)C)C)C 8R-0629 c1cc(sc1)c2ccnc(n2)NC(=O)c3cccs3 8R-0631 c1cc(oc1)C(=O)Nc2nccc(n2)c3cccs3 8R-0632 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccco3 8R-0634 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(cc3)F 8R-0635 COc1cccc(c1)C(CC(=O)O)N2Cc3ccccc3C2=O 8R-0636 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccccc3Cl 8R-0638 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3cccc(c3)Cl 8R-0639 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3cccc(c3)[N+](=O)[O-] 8R-0640 Cc1ccccc1C(CC(=O)O)NC(=O)OC(C)(C)C 8R-0641 Cc1cccc(c1)C(CC(=O)O)NC(=O)OC(C)(C)C 8R-0642 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc(c1)[N+](=O)[O-] 8R-0643 c1cc(ccc1C(CC(=O)O)N)O 8R-0644 c1c(sc(n1)N2CCCCC2)CN3CCOCC3 8R-0646 c1cscc1C(CC(=O)O)N 8R-0647 CC(C)(C)c1ccc(cc1)C(CC(=O)O)N 8R-0649 CSc1ccc(cc1)C(CC(=O)O)N 8R-0650 Cc1ccc(cc1)C(=O)Nc2nccc(n2)c3cccs3 8R-0652 CC1CCN(CC1)c2ncc(s2)CN3CCN(CC3)c4ccccc4 8R-0654 CC(C)(C)c1ccc(cc1)/C=C/C(=O)O 8R-0658 CCOC(=O)N1CCN(CC1)c2ncccn2 8R-0659 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3cccc(c3)C(F)(F)F 8R-0660 CCOc1ccc(cc1)C(CC(=O)O)N2Cc3ccccc3C2=O 8R-0661 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccccc3Br 8R-0662 c1cc(cc(c1)O)C(CC(=O)O)N 8R-0664 CCOC(=O)N1CCN(CC1)c2c(cccn2)[N+](=O)[O-] 8R-0665 c1cc(oc1)C2CC(=O)CC(=O)C2n3cncn3 8R-0801 Cc1c(sc(n1)c2ccncc2)c3ccncn3 8R-0802 c1cc(cnc1)c2ncc(s2)c3ccnc(n3)N 8R-0803 Cc1c(nnn1c2ccsc2C(=O)OC)C(=O)c3ccc(cc3Cl)Cl 8R-0804 CC1(CN(C1=O)c2cccc(c2)c3ccnc4n3ncn4)C 8R-0805 CC1=C(/C(=C/c2ccc3c(c2)OCO3)/C(=O)N1CCc4ccc(c(c4)OC)OC)C(=O)OC 8R-0806 c1cc(c(c(c1)Cl)CC2=C(C(C(CC2=O)c3ccc4c(c3)OCO4)n5cncn5)O)Cl 8R-0807 c1cc(ccc1c2c(cnc3n2ncn3)n4cncn4)Cl 8R-0809 c1ccnc(c1)CCNC(=O)Cc2c(cc(cn2)C(F)(F)F)Cl 8R-0810 CC1=C(/C(=C/C=C\c2ccc(cc2)N(C)C)/C(=O)N1CCc3ccccc3)C(=O)OC 8R-0811 c1cc(cnc1)c2ncc(s2)c3ccn[nH]3 8R-0812 CC(=O)c1cnc(s1)c2cccs2 8R-0813 CCCCCCCc1ccc(cc1)C(CC(=O)c2cnc(s2)c3cccnc3)O 8R-0815 Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)C(=O)C 8R-0816 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)C 8R-0817 Cc1c(sc(n1)c2cccc(c2Cl)Cl)C(=O)C 8R-0818 Cc1c(sc(n1)c2cccs2)c3ccn[nH]3 8R-0819 Cc1ccc(cc1)c2nc(c(s2)C(=O)/C=C/N(C)C)C 8R-0820 Cc1c(sc(n1)c2ccc(cc2Cl)Cl)C(=O)/C=C/N(C)C 8R-0821 Cc1c(sc(n1)c2cc[n+](cc2)C)c3ccnc(n3)NC.[I-] 8R-0822 Cc1c(c(n2c(n1)nc(n2)SC)C)Cc3cccc(c3)C(F)(F)F 8R-0823 Cc1c(cnc2n1ncn2)c3ccc(c(c3)OC)OC 8R-0824 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)/C=C/N(C)C 8R-0825 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)/C=C/C=C/c3ccc(cc3)N(C)C 8R-0826 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/c3ccccc3[N+](=O)[O-] 8R-0827 CCCCCCCNC(=O)Cc1c(cc(cn1)C(F)(F)F)Cl 8R-0828 CC(C(=O)c1cn(nn1)c2ccsc2C(=O)OC)Oc3ccccc3 8R-0829 Cc1cc2ncc(c(n2n1)C)c3ccc(c(c3)OC)OC 8R-0831 COc1ccc(cc1)C2CC(=O)C(=C(C2n3cncn3)O)C4c5ccccc5CCN4 8R-0832 c1ccc2c(c1)CCNC2C3C(=O)CC(C(C3=O)n4cncn4)c5ccco5 8R-0833 Cc1c(sc(n1)c2cccc(c2Cl)Cl)C(=O)/C=C/N(C)C 8R-0837 c1cc(cc(c1)NC(=S)N)C(F)(F)F 8R-0839 Cc1ccc(cc1)c2nc(c(s2)c3ccn[nH]3)C 8R-0840 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)c3ccn[nH]3 8R-0842 CC(C)(C)OC(=O)N1CCC2(CC1)CO2 8R-0843 c1c(cnc(c1Cl)CC(=O)NCCN2CCN(CC2)C(=O)Cc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 8R-0845 COc1ccc(cc1)N2CCN(CC2)C(=O)Cc3c(cc(cn3)C(F)(F)F)Cl 8R-0846 CC1=C(C(C(=O)N1CCc2ccc(c(c2)OC)OC)/C=[N+](\C)/[O-])C(=O)OC 8R-0847 c1cc(ccc1N2CCN(CC2)C(=O)Cc3c(cc(cn3)C(F)(F)F)Cl)F 8R-0848 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)F)C#N)N)CSc3ccccc3 8R-0851 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)F)C#N)N)CSc3ccc(cc3)Cl 8R-0852 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)S(=O)(=O)NC(=N)N)F 8R-0854 c1cc(ccc1C(=O)c2cc(cc(c2)C(=O)c3ccc(cc3)F)C(=O)c4ccc(cc4)F)F 8R-0863 CS(=O)(=O)N1CCN(CC1)c2ccc(cc2F)NC(=O)c3cccs3 8R-1000 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)S(=O)(=O)C 8R-1001 CS(=O)(=O)N1CCN(CC1)c2ccc(cc2F)NC(=O)c3ccc(c(c3)Cl)Cl 8R-1002 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3F)NC(=O)C4CC4 8R-1003 CCCCC(=O)Nc1ccc(c(c1)F)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)C 8R-1004 Cc1c(c2ccccc2[nH]1)C(=O)NS(=O)(=O)Nc3ccccc3 8R-1006 CS(=O)(=O)N1CCN(CC1)c2ccccc2[N+](=O)[O-] 8R-1008 CCn1c(nnc1S)COc2ccc(=O)n(n2)c3ccccc3 8R-1012 CCn1c(nnc1SC)COc2ccc(=O)n(n2)c3ccccc3 8R-1014 CCn1c(nnc1SCC(=O)Nc2c(cccc2C)C)COc3ccc(=O)n(n3)c4ccccc4 8R-1015 CCn1c(nnc1SCc2ccc(cc2)OC)COc3ccc(=O)n(n3)c4ccccc4 8R-1017 Cc1cccc(c1)C(=O)Nc2ccc(c(c2)F)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl 8R-1018 CCn1c(nnc1SCC(=O)Nc2ccccc2)COc3ccc(=O)n(n3)c4ccccc4 8R-1020 CS(=O)(=O)N1CCN(CC1)c2ccccc2NC(=O)c3ccc(cc3)F 8R-1024 CS(=O)(=O)N1CCN(CC1)c2ccccc2NC(=O)c3ccc(cc3)Cl 8R-1025 CCn1c(nnc1SCC(=O)NCc2ccccc2)COc3ccc(=O)n(n3)c4ccccc4 8R-1026 Cc1cccc(c1)C(=O)Nc2ccccc2N3CCN(CC3)S(=O)(=O)C 8R-1027 CS(=O)(=O)N1CCN(CC1)c2ccccc2NC(=O)c3cccs3 8R-1028 CCn1c(nnc1SCC(=O)OC)COc2ccc(=O)n(n2)c3ccccc3 8R-1029 CCn1c(nnc1SCc2ccc(cc2)Cl)COc3ccc(=O)n(n3)c4ccccc4 8R-1030 CCn1c(nnc1SCC=C)COc2ccc(=O)n(n2)c3ccccc3 8R-1031 CCn1c(nnc1SCc2ccc(cc2)C)COc3ccc(=O)n(n3)c4ccccc4 8R-1032 Cc1cc(nc(n1)C(C)C)Cl 8R-1033 Cc1cc(nc(n1)C(C)C)N2CCOCC2 8R-1034 c1cc(ccc1SC[C@@H](C(F)(F)F)O)Cl 8R-1060 c1cc(c(c(c1)Cl)SC[C@@H](C(F)(F)F)O)Cl 8R-1061 c1cc(ccc1SC[C@@H](C(F)(F)F)O)Br 8R-1062 C([C@H](C(F)(F)F)O)Sc1nnc(s1)N 8R-1064 c1cc(cc(c1)C(F)(F)F)C(=O)O[C@H](CN2CCC3(CC2)OCCO3)C(F)(F)F 8R-1066 c1cc(sc1)C(=O)O[C@H](CN2CCC3(CC2)OCCO3)C(F)(F)F 8R-1067 c1cc(c(c(c1)F)C(=O)O[C@H](CN2CCC3(CC2)OCCO3)C(F)(F)F)F 8R-1068 C1CN(CCC12OCCO2)/C=C/C(=O)C(F)(F)F 8R-1069 c1ccc(cc1)C[n+]2cccc3c2[nH]cc3.[Br-] 8R-1070 C1CN(CCC12OCCO2)CCC(C(F)(F)F)O 8R-1072 c1ccnc(c1)/C=C\2/C(=O)C3CCN2CC3 8R-1073 c1ccnc(c1)/C=C\2/C(C3CCN2CC3)O 8R-1074 CCn1c(nnc1S)c2cc3cc4ccccc4nc3s2 8R-1122 Cc1ccc(cc1)C(=O)N(Cc2c(nn(c2Cl)C)C(F)(F)F)c3ccc(cc3)OC 8R-1124 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)C(=O)c3ccc(c(c3)Cl)Cl)Cl 8R-1125 CCn1c(nnc1SC)c2cc3cc4ccccc4nc3s2 8R-1127 CCn1c(nnc1SCC=C)c2cc3cc4ccccc4nc3s2 8R-1129 CCn1c(nnc1SCc2ccc(cc2)Cl)c3cc4cc5ccccc5nc4s3 8R-1130 CCn1c(nnc1SCC)c2cc3cc4ccccc4nc3s2 8R-1132 CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)c3cc4cc5ccccc5nc4s3 8R-1133 CCn1c(nnc1SCc2ccc(cc2)C)c3cc4cc5ccccc5nc4s3 8R-1134 CCn1c(nnc1SCCCF)c2cc3cc4ccccc4nc3s2 8R-1135 c1ccc2c(c1)cc3cc(sc3n2)c4nnc(o4)C5CC5 8R-1137 c1ccc2c(c1)cc3cc(sc3n2)c4nnc(o4)S 8R-1141 CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3cc4cc5ccccc5nc4s3 8R-1143 CCn1c(nnc1SCc2ccc(cc2)F)c3cc4cc5ccccc5nc4s3 8R-1144 CCn1c(nnc1SCc2ccccc2)c3cc4cc5ccccc5nc4s3 8R-1146 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)C(=O)c3c(cccc3F)F)Cl 8R-1148 c1cc2c(cc1Br)c(=O)oc(=O)[nH]2 8R-1149 c1ccc2c(c1)cc3cc(sc3n2)C(=O)c4ccccc4Cl 8R-1150 c1ccc2c(c1)cc3cc(sc3n2)C(=O)c4ccc(cc4Cl)Cl 8R-1151 c1ccc(cc1)C(=O)c2cc3cc4ccccc4nc3s2 8R-1152 Cn1c(c(c(n1)C(F)(F)F)/C=N/c2ccc(cc2)Cl)Cl 8R-1153 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)C(=O)c3ccc(cc3)Cl)Cl 8R-1154 Cn1c(c(c(n1)C(F)(F)F)CNc2ccc(cc2)Cl)Cl 8R-1155 c1ccc2c(c1)cc3cc(sc3n2)/C(=N/O)/c4ccccc4Cl 8R-1157 c1ccc2c(c1)cc3cc(sc3n2)/C(=N/O)/c4ccc(cc4Cl)Cl 8R-1158 Cn1c(c(c(n1)C(F)(F)F)/C=N/c2cccc(c2)C(F)(F)F)Cl 8R-1160 Cn1c(c(c(n1)C(F)(F)F)/C=N/c2ccc(c(c2)Cl)Cl)Cl 8R-1161 Cc1cc(cc(c1)/N=C/c2c(nn(c2Cl)C)C(F)(F)F)C 8R-1162 c1ccc2c(c1)cc3cc(sc3n2)c4nnc(o4)SCc5ccc(cc5)Cl 8R-1164 c1ccc2c(c1)cc3cc(sc3n2)c4nnc(o4)SCc5ccc(cc5)F 8R-1170 Cc1ccc(cc1)CSc2nnc(o2)c3cc4cc5ccccc5nc4s3 8R-1171 Cn1c(c(c(n1)C(F)(F)F)CNc2ccc(c(c2)Cl)Cl)Cl 8R-1173 Cn1c(c(c(n1)C(F)(F)F)CNc2cccc(c2)C(F)(F)F)Cl 8R-1174 Cc1cc(cc(c1)NCc2c(nn(c2Cl)C)C(F)(F)F)C 8R-1175 CN1CCN(CC1)c2ccc(cc2F)NC(=O)CSc3ccc(cc3)Cl 8R-1180 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)CSc4ccc(cc4)Cl 8R-1183 Cc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 8R-1184 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)CSc4ccc(cc4)Br 8R-1185 CN1CCN(CC1)c2ccc(cc2F)NC(=O)CSc3ccccc3 8R-1187 Cc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)C 8R-1188 CN1CCN(CC1)c2ccc(cc2F)NC(=O)CSc3ccc(cc3)OC 8R-1189 Cc1ccc(c(c1)C)SCC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)C 8R-1190 c1cc(c(cc1NC(=O)CN2CCOCC2)F)N3CCOCC3 8R-1192 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)CSc4ccccc4 8R-1193 COc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 8R-1194 Cc1ccc(c(c1)C)SCC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 8R-1195 COCC(=O)Nc1ccc(c(c1)F)N2CCN(CC2)c3ccccc3 8R-1196 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)F)N3CCOCC3)Cl 8R-1197 COc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)F)N3CCOCC3 8R-1198 Cc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)F)N3CCOCC3 8R-1199 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)CN4CCOCC4 8R-1200 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3F)NC(=O)CN4CCCCC4 8R-1201 CCN1CCN(CC1)CC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)c4ccccc4 8R-1202 CCN1CCN(CC1)CC(=O)Nc2ccc(c(c2)F)N3CCOCC3 8R-1203 c1ccc(cc1)SCC(=O)Nc2ccc(c(c2)F)N3CCOCC3 8R-1204 Cc1ccc(c(c1)C)SCC(=O)Nc2ccc(c(c2)F)N3CCOCC3 8R-1205 c1ccc(c(c1)SCC(=O)Nc2ccc(c(c2)F)N3CCOCC3)Cl 8R-1206 c1ccc(c(c1)OCC(CS(=O)(=O)Cc2ccc(cc2)Cl)O)Cl 8R-1240 c1ccc(c(c1)CS(=O)(=O)CC(COc2ccccc2Cl)O)Cl 8R-1241 c1csc2c1c(nc(n2)S)O 8R-1301 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)N3CCCC3 8R-1302 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)N3CCCCCC3 8R-1303 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)NC3CCCCC3 8R-1305 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)NC3CC3 8R-1306 c1ccc(cc1)CNC(=O)c2c(ccs2)NC(=O)c3ccccc3 8R-1307 Cc1ccc(cc1)c2nc3ccsc3c(n2)O 8R-1310 c1ccc(cc1)c2nc3ccsc3c(n2)N4CCCC4 8R-1312 c1ccc(cc1)c2nc3ccsc3c(n2)N4CCCCCC4 8R-1313 COc1ccc(cc1)CNC(=O)c2c(ccs2)NC(=O)c3ccccc3 8R-1315 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)NCc3ccc(cc3)Cl 8R-1316 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)NCc3ccncc3 8R-1317 Cc1ccc(cc1)CNC(=O)c2c(ccs2)NC(=O)c3ccccc3 8R-1318 c1ccc(cc1)C(=O)Nc2ccsc2C(=O)NCc3ccc(cc3)F 8R-1319 CSc1nc(c2ccsc2n1)O 8R-1322 Cc1ccc(cc1)c2nc3ccsc3c(n2)Cl 8R-1324 COC(=O)c1c(ccs1)N=C=S 8R-1326 COC(=O)c1ccsc1N=C=S 8R-1327 c1ccc2c(c1)ncc(n2)Oc3cnns3 8R-1422 c1cc2c(ccc(c2nc1)Oc3cnns3)Cl 8R-1423 Cc1c(c(nn1c2ccc(cc2)F)O)c3ccccn3 8R-1503 Cc1ccc(cc1)n2c(c(c(n2)O)c3ccccn3)C 8R-1505 Cc1c(c(nn1c2ccc(c(c2)Cl)Cl)O)c3ccccn3 8R-1506 c1ccc2c(c1)N=C(CC(S2)c3cccc(c3)Cl)c4cccs4 8T-0001 CN(C)/C=C\1/C(=O)N(C(=O)S1)S(=O)(=O)C 8T-0002 c1ccc2c(c1)C(=O)N(C2=O)Cc3cnc(s3)N4CCCCC4 8T-0004 c1ccc2c(c1)C(=O)N(C2=O)Cc3cnc(s3)N4CCOCC4 8T-0005 Cc1cc(nc2c1c(nn2C)NC(=S)N)C 8T-0006 COC(=O)C(c1ccc(cc1)N)C(=O)OC 8T-0010 Cn1c2c(cn1)c(c(cn2)C(=O)Oc3c(c(c(c(c3F)F)F)F)F)NCc4ccc(cc4)OC 8T-0012 CN1C(=O)C(C(=O)N(C1=O)C)Cc2cn(c3c2cccc3)Cc4cnc(s4)Cl 8T-0015 CN1C(=O)/C(=C\Nc2ccc3c(c2)OCO3)/SC1=O 8T-0017 CC(C)CC(CC(=O)O)N 8T-0019 CN1C(=O)/C(=C/c2ccc(cc2)F)/SC1=O 8T-0023 CCOC(=O)c1cnc2c(c1OC(CN)C(F)(F)F)cnn2C 8T-0024 COC(=O)CC(c1ccc2c(c1)OCO2)NS(=O)(=O)C 8T-0028 CNC(=S)NC(CC(=O)OC)c1ccc2c(c1)OCO2 8T-0029 COC(=O)CC(c1ccc2c(c1)OCO2)NC(=O)CCl 8T-0030 c1cc(sc1)/C=C/2\C(=O)NC(=O)S2 8T-0032 Cn1c2c(cn1)c(c(cn2)C(=O)Oc3c(c(c(c(c3F)F)F)F)F)NCc4cccc(c4)C(F)(F)F 8T-0033 CN1CCN(CC1)/C=C/2\C(=O)N(C(=O)S2)C 8T-0038 CCOc1ccc(cc1)/C=C/2\C(=O)N(C(=O)S2)C 8T-0039 CN1C(=O)/C(=C/c2cccc3c2cccc3)/SC1=O 8T-0040 c1cnn(c1)Cc2ccc(cc2)N 8T-0041 c1c2c(cc3c1OCO3)C(=O)NCC2NC(=O)C(F)(F)F 8T-0045 C1CC(CC=C1)C(CC(=O)O)N 8T-0046 CN1C(=O)C(=Cc2ccc(cc2)OCc3cnc(s3)Cl)C(=O)N(C1=O)C 8T-0047 CCC(CC)C(CC(=O)O)N 8T-0051 CCC(C)C(CC(=O)O)N 8T-0052 Cc1ccc(o1)/C=C\2/C(=O)NC(=O)S2 8T-0054 CN1C(=O)/C(=C/c2ccc(cc2)OC)/SC1=O 8T-0055 c1cc(oc1)C(=O)Nc2c(cc(cn2)Cl)Br 8T-0060 CN1CCN(CC1)c2ncc(s2)Cn3ccnc3 8T-0065 CCN1C(=O)/C(=C/c2cccc(c2)Cl)/SC1=O 8T-0070 c1cc(cc(c1)[N+](=O)[O-])/C=C\2/C(=O)NC(=O)S2 8T-0073 c1ccc(cc1)CCCN2C(=O)CSC2=O 8T-0077 CC(c1ccc(cc1)[N+](=O)[O-])C(=O)OC 8T-0081 Cc1cc(nc(c1C#N)OCc2cccc(c2)C(F)(F)F)C 8T-0083 c1ccc(cc1)/C=C/2\C(=O)NC(=O)S2 8T-0084 CCOC(=O)c1nccn1C 8T-0085 CC(c1ccc(cc1)N)C(=O)O 8T-0086 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)C3CCCCC3 8T-0087 CCOC(=O)C1CCN(CC1)c2ncc(s2)Cn3ccnc3 8T-0089 c1ccn(c1)c2c(cc(cn2)Cl)Br 8T-0090 Cc1ccc(n1c2ccc(cc2)C(C(=O)OC)C(=O)OC)C 8T-0093 COC(=O)C(c1ccc(cc1)n2cccc2)C(=O)OC 8T-0095 c1ccc2c(c1)n3c(c(nc3s2)c4ccc(c(c4)Cl)Cl)Cl 8T-0096 COC(=O)C(c1ccc(cc1)NC(=O)c2cccc(c2)Cl)C(=O)OC 8T-0101 COC(=O)C(c1ccc(cc1)NC(=O)c2cccs2)C(=O)OC 8T-0102 COc1cc(ccc1O)/C=C/2\C(=O)N(C(=O)S2)CCCc3ccccc3 8T-0105 CN(C)/C=C\1/C(=O)N(C(=O)S1)CCCc2ccccc2 8T-0106 COc1ccc(c(c1)N)n2cccc2 8T-0200 Cc1cc2nc(c(c(n2n1)Cl)CCCl)C 8T-0201 Cn1c2ccccc2c3c1sc(c3)C(=O)O 8T-0207 CCOC(=O)CNC(=O)c1c(nn(c1Cl)C)C 8T-0209 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)N3CC(OC(C3)C)C 8T-0210 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)NCCCN3CCOCC3 8T-0211 c1ccc2c(c1)nc(o2)c3cc(ccc3F)N 8T-0212 c1cc(c(cc1N)F)C(=O)O 8T-0213 CC(=C)C(=O)NCCCCCCCCCCC(=O)Nc1ccc(cc1)OC 8T-0214 CC(=C)C(=O)NCCCCCCCCCCC(=O)Nc1ccc(cc1)Oc2ccccc2 8T-0215 c1cnc(nc1C2CC2)N 8T-0217 CCOC(=O)c1c[nH]c(=O)c(c1C)C(=O)N 8T-0219 Cc1c(cc(c(=O)[nH]1)C(=O)N)C(=O)C 8T-0220 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)NCCN3CCCC3 8T-0226 CS(=O)(=O)c1cc(ccc1OCc2ccccc2)OCc3ccccc3 8T-0230 Cc1c(c(n(n1)C)Cl)C(=O)NC(c2ccccc2)C(=O)OC 8T-0231 CC(=C)C(=O)NCCCCCCCCCCC(=O)NCCN1CCCCC1 8T-0232 CCCCCC1CCC(CC1)C(=O)Nc2ccc3c(c2)OCO3 8T-0233 c1ccc(cc1)COC(=O)NC(C(=O)O)O 8T-0234 CCCCCC1CCC(CC1)c2ccc(cc2)NC(=O)CCCC(=O)O 8T-0235 Cc1ccc2c(c1)oc3cccc(c3c2=O)NC4CCCCCCC4 8T-0236 CCCCCC1CCC(CC1)C(=O)NCCN2CCOCC2 8T-0238 CC(=C)C(=O)NCCCCCCCCCCC(=O)NCCc1ccccc1 8T-0239 Cn1cc(c(n1)C(F)(F)F)C(=O)NC(c2ccccc2)C(=O)OC 8T-0240 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)n3ccc(n3)C4CC4 8T-0243 c1ccc(cc1)COC(=O)NC(c2ccc3c(c2)OCCO3)C(=O)O 8T-0246 CCCCCC1CCC(CC1)C(=O)Nc2ccccc2OC 8T-0247 CCCCCC1CCC(CC1)C(=O)Nc2cccc(c2C)C 8T-0248 c1cc(c(cc1C(=O)n2ccc(n2)C3CC3)Cl)Cl 8T-0249 c1ccc(cc1)COC(=O)NC(c2ccc3c(c2)OCC3)C(=O)O 8T-0250 c1ccc(cc1)C(C(=O)Nc2nccs2)Br 8T-0252 c1ccc2c(c1)nnn2Cc3ccc(cc3)N 8T-0253 Cc1c(c(n(n1)C)Cl)C(=O)NCCCC(=O)O 8T-0256 c1cc(ccc1N2CCN(CC2)C(=O)Nc3ccc4c(c3)NC(=O)CO4)F 8T-0258 Cc1c(c(=O)n2c([nH]1)ncn2)CCO 8T-0259 COc1ccc(cc1Cl)CNC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 8T-0261 COc1ccc(cc1Cl)CNC(=O)N2CCN(CC2)c3ccc(cc3)F 8T-0262 Cn1cc(c(n1)C(F)(F)F)C(=O)NCCCC(=O)O 8T-0264 c1cc2c(cc1CN3CCN(CC3)C(=O)Nc4ccc5c(c4)NC(=O)CO5)OCO2 8T-0266 c1cc(cc(c1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)NC(=O)CO4)C(F)(F)F 8T-0267 CSc1ccccc1N2CCN(CC2)C(=O)Nc3ccc4c(c3)NC(=O)CO4 8T-0269 CCOC(=O)c1c[nH]c(=S)c(c1C)C(=O)N 8T-0270 c1c2c(c(c(=O)[nH]1)C(=O)N)CCCC2=O 8T-0271 Cc1c(c(n(n1)C)Cl)C(=O)NC(c2ccccc2)C(=O)O 8T-0276 COc1ccc(cc1OC)c2c[nH]nc2N 8T-0279 c1cc(c(cc1Cl)S(=O)(=O)n2ccc(n2)C3CC3)Cl 8T-0280 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)C3CC3 8T-0281 CCCCCC(=O)OCCc1c([nH]c2ncnn2c1=O)C 8T-0282 C/C(=N\c1nc[nH]n1)/C2CCOC2=O 8T-0283 CCOC(=O)C1CCN(CC1)c2ccccc2C#N 8T-0284 c1cc2c(cc1NC(=O)CCCC(=O)O)NC(=O)CO2 8T-0285 CCCCCC(=O)OCCc1c([nH]c2nc3ccccc3n2c1=O)C 8T-0288 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3ccc(cc3)C(F)(F)F 8T-0289 CCC(C(=O)OC)NC(=O)c1cn(nc1C(F)(F)F)C 8T-0290 Cc1ccc(cc1)NC(=O)OCCc2c([nH]c3ncnn3c2=O)C 8T-0291 c1cc(ccc1F)S(=O)(=O)n2ccc(n2)C3CC3 8T-0292 Cc1cccc(c1)C(=O)OCCc2c([nH]c3c(cnn3c2=O)C#N)C 8T-0293 CCNc1nc2ccccc2n1Cc3c(cccc3Cl)F 8T-0295 CCNc1nc2ccccc2n1Cc3cccc(c3)Cl 8T-0296 Cc1c(c2ccccc2[nH]1)C3=CC(=O)c4ccccc4C3=O 8T-0297 COC(=O)c1ccc(cc1O)n2cccc2 8T-0299 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)Nc3ccc4c(c3)NC(=O)CO4 8T-0305 CCNc1nc2ccccc2n1Cc3ccccc3F 8T-0306 C#CCNC(=O)c1ccccc1N 8T-0307 Cn1c(=O)c2c(n(c1=O)C)OC(C2=O)/C=N\OCc3ccc(cc3Cl)Cl 8T-0309 c1ccn(c1)c2ccc3c(c2)NC(=O)CO3 8T-0310 c1cc2c(cc1NC(=O)/C=C/C(=O)O)NC(=O)CO2 8T-0311 c1cc2c(cc1NC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)NC(=O)CO2 8T-0312 c1cc(sc1)c2ccn(c(=N)c2C#N)N 8T-0325 c1cc(oc1)c2ccn(c(=N)c2C#N)N 8T-0329 Cc1c(c(n(n1)C)Cl)C(=O)NC(c2ccccc2)C(=O)Nc3ccc(cc3)OC 8T-0333 Cn1cc(c(n1)C(F)(F)F)C(=O)NCCCC(=O)Nc2ccc(cc2)OC 8T-0334 CC(=O)Nc1ccc(cc1)/C=C/C(=O)O 8T-0336 c1ccc(cc1)C(C(=O)Nc2nccs2)N3CCOCC3 8T-0337 c1cc2c(cc1NC(=O)N3CCOCC3)NC(=O)CO2 8T-0343 Cc1c(c(n(n1)C)Cl)C(=O)NCC(=O)O 8T-0344 c1ccc(cc1)CN(Cc2ccccc2)C(=O)Nc3ccc4c(c3)NC(=O)CO4 8T-0345 CC1(CC2=C(C(C(=C(O2)N)S(=O)(=O)c3ccccc3)c4ccc(cc4)Cl)C(=O)C1)C 8T-0614 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)Cl)/C#N 8T-0622 c1cc(ccc1NC(=O)C2C(C2(C#N)C#N)c3ccc(cc3Cl)Cl)Br 8T-0623 C1CCc2c(c(c(s2)NC(=O)C3CC3)C#N)C1 8T-0631 CCOC(=O)c1c2c(sc1NC(=O)C3CC3)CCCC2 8T-0632 Cc1cc(n(n1)C/C(=N/Nc2ccccc2)/C)C 8T-0800 CSc1ccc(cc1Cl)N 8T-0802 C/C(=N\OCc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)Oc3ccc(cc3)C(C)(C)C 8T-0803 C/C(=N\OCc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)OCC(C(F)F)(F)F 8T-0804 c1c(cnc(c1Cl)C(=O)CC(=O)C(F)(F)F)C(F)(F)F 8T-0805 CCO/C=C(/C(=O)C)\C(=O)c1c(cc(cn1)C(F)(F)F)Cl 8T-0806 COC(=O)c1c(c(cs1)S(=O)(=O)c2ccccc2)N 8T-0813 CCc1ccc2c(cc(=O)oc2c1)C 8T-0815 CCc1ccc2c(cc(=O)oc2c1)C(F)(F)F 8T-0816 Cc1cc(n(n1)/C(=C/N(C)C)/C(=O)c2ccccc2)C 8T-0817 Cc1cc(n(n1)c2cnc3c(cnn3c2c4ccccc4)c5ccccn5)C 8T-0821 Cc1cc(n(n1)CC(=O)c2ccc(cc2)Cl)C 8T-0822 Cc1cc(n(n1)CC(=O)c2ccc(cc2)OC)C 8T-0823 Cc1cc(n(n1)CC(=O)c2cccc(c2)[N+](=O)[O-])C 8T-0824 Cc1cc(n(n1)/C(=C\N(C)C)/C(=O)c2ccc(cc2)Cl)C 8T-0825 Cc1cc(n(n1)c2c([nH]c3c2cccc3)C)C 8T-0826 Cc1cc(n(n1)/C(=C/N(C)C)/C(=O)c2ccc(cc2)OC)C 8T-0828 Cc1cc(n(n1)/C(=C\N(C)C)/C(=O)c2cccc(c2)[N+](=O)[O-])C 8T-0829 Cc1c(c(nn2c1nnc2)C)C/C=C/c3ccccc3 8T-0830 Cc1cc(n(n1)c2cnc3cc(nn3c2c4ccc(cc4)OC)c5cnn(c5C(F)(F)F)C)C 8T-0835 Cc1ccc(n1NC(=O)c2ccncc2)C 8T-0837 c1ccc2c(c1)CC(=O)N(C2=O)CCc3c[nH]c4c3cccc4 8T-0839 Cc1c(c(n(n1)CC(=O)c2ccccc2)C)Br 8T-0844 Cc1cc(n(n1)c2cnc3c(cnn3c2c4cccc(c4)[N+](=O)[O-])c5ccc(cc5)OC)C 8T-0845 Cc1cc(n(n1)c2cnc3cc(nn3c2c4cccc(c4)[N+](=O)[O-])c5cnn(c5C(F)(F)F)C)C 8T-0846 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)c5cccc(c5)[N+](=O)[O-])n6c(cc(n6)C)C)C 8T-0847 Cc1cc(n(n1)c2cnc3cc(nn3c2c4ccccc4)c5cnn(c5C(F)(F)F)C)C 8T-0850 Cc1cc(n(n1)c2cnc3c(cnn3c2c4ccc(cc4)Cl)c5ccccn5)C 8T-0851 CN(C)/C=C\1/c2ccccc2C(=O)N(C1=O)CCc3c[nH]c4c3cccc4 8T-0853 Cc1cc(n(n1)c2cnc3c(cnn3c2c4ccc(cc4)Cl)c5ccc(cc5)Cl)C 8T-0854 Cc1c(c(n(n1)CC(=O)c2ccc(cc2)Cl)C)Br 8T-0856 c1ccc(cc1)CS(=O)(=O)c2cc(ccc2[N+](=O)[O-])C(F)(F)F 8W-0004 Cn1c(c(c(n1)C(F)(F)F)CN)Oc2ccccc2 8W-0010 Cn1c(c(c(n1)C(F)(F)F)CNC(=O)c2ccco2)Oc3ccccc3 8W-0014 c1cc2c(c(c1)Cl)/C(=C/c3ccc(cc3)O)/C(=O)N2 8W-0015 c1ccc2c(c1)cccc2/C=C\3/c4c(cccc4Cl)NC3=O 8W-0016 COc1cccc(c1)/C=C\2/c3c(cccc3Cl)NC2=O 8W-0017 c1cc2c(cc1N)cno2 8W-0024 Cc1c2c(c3cccc(c3n1)Oc4ccccc4)N(CC2)c5ccc(cc5)C(C)C 8W-0200 Cc1c2c(c3cccc(c3n1)Oc4ccccc4)N(CC2)c5ccc(cc5)Oc6ccccc6 8W-0201 c1ccc(cc1)n2cc(c(n2)c3ccc4c(c3)CCC4)/C=C(/C#N)\S(=O)(=O)c5ccccc5 8W-0202 c1cc(ccc1N2CCN(CC2)CCC3C(=O)Nc4ccc(cc4O3)[N+](=O)[O-])[N+](=O)[O-] 8W-0203 COc1ccc(cc1)N2CCN(CC2)CCC3C(=O)Nc4ccc(cc4O3)[N+](=O)[O-] 8W-0204 Cc1ncc(c(n1)C(F)(F)F)C(=O)NCc2ccccc2 8W-0205 COc1ccc(cc1)c2c(n3cc(cc(c3n2)Cl)C(F)(F)F)Br 8W-0206 CCOC(=O)c1cnc([nH]c1=O)n2c(=O)c(c([nH]2)C)Cc3ccccc3 8W-0209 Cc1cc(=O)[nH]c(n1)n2c(=O)c(c([nH]2)C)Cc3ccccc3 8W-0210 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)c(c(n2)C)Cc3ccccc3)Cc4ccccc4 8W-0211 Cc1c2c(c3cccc(c3n1)Oc4ccccc4)N(CC2)c5ccccc5OC 8W-0212 Cc1c2c(c3cccc(c3n1)Oc4ccccc4)N(CC2)c5ccc(cc5)OC(F)(F)F 8W-0213 Cc1c2c(c3cccc(c3n1)Oc4ccccc4)N(CC2)c5ccc(cc5)C(F)(F)F 8W-0214 CSc1nc2ccccc2c(n1)N3CCN(CC3)Cc4ccc5c(c4)OCO5 8W-0216 c1ccc2c(c1)C(=O)N(C2=O)CCC3C(=O)Nc4ccc(cc4O3)[N+](=O)[O-] 8W-0217 Cc1cc2nc(c3ccccc3n2n1)OC(C)(C)C 8W-0218 COC(=O)c1ccc(cc1)c2ccc(cc2)C#N 8W-0219 COc1ccc(cc1)c2cn3cc(ccc3n2)C(=O)NN 8W-0220 C/C(=N\c1ccc(cc1)O)/N(C)CCNS(=O)(=O)c2ccc(cc2)[N+](=O)[O-].I 8W-0221 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)c(cn2)C(=O)O)Cc3ccccc3 8W-0223 CCOC(=O)C1=C(SCC1=O)NC 8W-0225 Cc1cc(=O)[nH]c(n1)n2c(=O)c3c([nH]2)CCCC3 8W-0228 c1cc(ccc1c2c(n3cc(cc(c3n2)Cl)C(F)(F)F)Br)Br 8W-0229 CCOC(=O)c1cnc([nH]c1=O)n2c(=O)c3c([nH]2)CCCC3 8W-0230 c1ccc(cc1)c2cc(=O)[nH]c(n2)n3c(=O)c4c([nH]3)CCCC4 8W-0235 c1cc(c(cc1c2cn3cc(cc(c3n2)Cl)C(F)(F)F)Cl)Cl 8W-0236 CCOC(=O)c1cnc(nc1C(F)(F)F)N 8W-0237 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)cc(n2)c3ccccc3)Cc4ccccc4 8W-0238 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)cc(n2)C(F)(F)F)Cc3ccccc3 8W-0239 Cc1c(ccc2c1oc(=O)cc2CCl)O 8W-0243 c1ccc2c(c1)ccc3c2c(c(s3)C#N)Cl 8W-0244 c1ccc(cc1)CN2CCN(CC2)c3ccc(cn3)C(=O)O 8W-0245 c1c(nc([nH]c1=O)n2c(=O)c3c([nH]2)CCCC3)C(F)(F)F 8W-0249 Cc1c(c(=O)[nH]c(n1)n2c(=O)c3c([nH]2)CCCC3)Cc4ccccc4 8W-0251 COc1ccc(cc1)c2cn3cc(ccc3n2)C(=O)NNS(=O)(=O)c4ccccc4Cl 8W-0252 COc1ccc(cc1)c2cn3cc(ccc3n2)C(=O)N/N=C/c4ccccc4Br 8W-0253 c1c(cnc(c1Br)Cl)C(=O)O 8W-0257 c1cc(ccc1c2cn3cc(ccc3n2)C(=O)NN)Br 8W-0259 c1c(c(nc(n1)N)C(F)(F)F)C(=O)O 8W-0262 c1cc(c(cc1c2c(n3cc(cc(c3n2)Cl)C(F)(F)F)Br)Cl)Cl 8W-0263 CCOC(=O)c1cc(nn1c2c(cccn2)[N+](=O)[O-])C(C)(C)C 8W-0264 CSC1=Nc2ccccc2C3=NCC(N31)CBr 8W-0267 c1cc2c(cc1c3cn4cc(ccc4n3)Cl)OCO2 8W-0268 c1cc(c(cc1[N+](=O)[O-])C(=O)O)N2CCC(CC2)C(=O)O 8W-0274 Cc1ccc(s1)C(=O)c2ccccc2C(=O)O 8W-0276 CCOC(=O)c1cc(nn1CCO)C(C)(C)C 8W-0277 Cc1cc(n(n1)C(C)(C)C)N 8W-0280 COc1ccccc1N2CCN(CC2)c3c4ccccc4nc(n3)SC 8W-0287 COc1ccccc1CNc2c3ccccc3nc(n2)SC 8W-0299 Cc1ccc(cc1)CNc2c3ccccc3nc(n2)SC 8W-0300 Cc1cc(nc(n1)n2c(=O)c(c([nH]2)C)Cc3ccccc3)C(F)(F)Cl 8W-0307 COC(=O)c1ccc2nc(cn2c1)c3cccc(c3)N 8W-0308 CSc1nc2ccccc2c(n1)N3CCN(CC3)c4ccccc4Cl 8W-0310 CSc1nc2ccccc2c(n1)NN 8W-0311 CCCc1cc(=O)[nH]c(n1)n2c(=O)c3c([nH]2)CCCC3 8W-0313 CCOC(=O)Cn1c(c(c(c1N)C#N)C)C 8W-0314 CCCCCCCCNc1c2ccccc2nc(n1)SC 8W-0315 CSc1nc2ccccc2c(n1)NCc3cccc(c3)C(F)(F)F 8W-0316 CSc1nc2ccccc2c(n1)NCc3ccc(cc3)Cl 8W-0317 COc1ccc(cc1)c2cn3cc(ccc3n2)C(=O)NNC(=O)c4cccc(c4)C(F)(F)F 8W-0319 c1cc(ccc1/C=N/NC(=O)c2ccc3nc(cn3c2)c4ccc(cc4)Br)F 8W-0320 c1cnc2nc(cn2c1)c3ccc4c(c3)OCO4 8W-0321 CCOC(=O)C1CCN(CC1)c2ccc(cc2C(=O)OC)N 8W-0322 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)cc(n2)c3ccccc3)CCO 8W-0323 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)cc(n2)C(F)(F)F)CCO 8W-0324 CSc1nc2ccccc2c(n1)NCc3ccco3 8W-0328 CSc1nc2ccccc2c(n1)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 8W-0329 CC(C)(C)c1cc(n(n1)c2ccccc2)C(=O)O 8W-0331 Cc1c(nc(s1)N)C(=O)OC 8W-0333 CCCCCCc1c(nc([nH]c1=O)n2c(=O)c(c([nH]2)C)CCO)C 8W-0335 CN(Cc1ccccc1)c2c3ccccc3nc(n2)SC 8W-0336 Cc1c(c(=O)[nH]c(n1)n2c(=O)c3c([nH]2)CCCC3)CCCN4C(=O)c5ccccc5C4=O 8W-0339 C=CCNc1ncccn1 8W-0340 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)cc(n2)c3ccccc3F)CCO 8W-0342 c1ccc2c(c1)c(nnc2Oc3ccc(cc3)Cl)c4ccc5c(c4)CCC5 8W-0348 Cc1ccc(n1c2ccc(cc2)Br)C 8W-0354 COc1cc(c(c(c1)OC)N)OC.Cl 8W-0406S Cc1ccnc(n1)SCc2ccc(cc2)[N+](=O)[O-] 8W-0808 CCCCCC(=O)N1CCC(=O)Nc2c1cccc2 8W-0811 Cc1ccnc(n1)Sc2c(cccn2)[N+](=O)[O-] 8W-0812 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)SCc4cccc(c4)C(F)(F)F)C(F)(F)F 8W-0813 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)SC)C(F)(F)F 8W-0814 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)SCc4ccc(cc4)C(=O)OC)C(F)(F)F 8W-0815 Cc1c(c(nn2c1nnc2)C)Cc3ccc(nc3)Cl 8W-0816 COc1ccc(cc1)C(=O)NCCc2c[nH]c3c2cc(cc3)OC 8W-0818 CCCCCCc1c(ccn(c1=O)CCc2c[nH]cn2)O 8W-0819 c1c(cnc(c1Cl)CC(=O)NCCN2CCCCC2)C(F)(F)F 8W-0820 Cc1cc2nc(c(c(n2n1)C)Cc3ccc(nc3)Cl)C 8W-0821 c1ccc2c(c1)ccc(c2/C=N/NC(=S)N)OCc3cccc(c3)C(F)(F)F 8W-0822 CN1C(=O)C(=Cc2c3ccccc3ccc2OCc4cccc(c4)C(F)(F)F)C(=O)N(C1=O)C 8W-0823 COc1ccc2c(c1)c(c[nH]2)CCN3C(=O)Cc4ccccc4C3=O 8W-0825 c1ccc2c(c1)ccc-3c2OC(c4c3nc5c(c4)C(=O)CCC5)O 8W-0827 c1ccc(c(c1)Cn2cccc2/C(=N\O)/N)[N+](=O)[O-] 8W-0828 c1ccc(cc1)c2cn3cccnc3n2 8W-0830 c1ccc(c(c1)C(=O)N2CCC(=O)Nc3c2cccc3)F 8W-0831 c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)CN4CCOCC4 8W-0832 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)SCc4ccc(cc4)C(=O)O)C(F)(F)F 8W-0833 COc1ccc2c(c1)c(c[nH]2)CCn3ccc(=O)c4c3CCCC4 8W-0834 Cc1ccnc(n1)S(=O)(=O)Cc2ccc(cc2)[N+](=O)[O-] 8W-0835 c1ccc2c(c1)NC(=O)CCN2S(=O)(=O)c3ccc(cc3)I 8W-0839 c1ccc2c(c1)c3c([nH]2)C(CCC3)O 8W-0840 COc1ccc(cc1)C(=O)N2CCC(=O)Nc3c2ccc(c3)C(F)(F)F 8W-0841 Cn1cc(c2c1cccc2)CCCC(=O)OC 8W-0843 c1ccc2c(c1)ccc(c2/C=C/3\c4ccccc4NC3=O)OCc5cccc(c5)C(F)(F)F 8W-0845 Cc1cc(n(n1)C(=O)c2csc(n2)n3c(cc(n3)C)C(F)(F)F)C 8W-0846 Cc1cc(n(n1)C(=O)c2ccc3c(c2)OCO3)C 8W-0847 c1ccc2c(c1)c(cn2Cc3ccc(cc3)Cl)CCCC(=O)O 8W-0852 c1ccc(cc1)c2csc(n2)Nc3ccc(cc3)F 8W-0855 CC(=O)Nc1ccc(cc1)S(=O)(=O)NNC(=O)c2ccc3c(c2)OCO3 8W-0856 c1cc(ccc1F)S(=O)(=O)NNC(=O)c2ccc3c(c2)OCO3 8W-0857 CC(=O)NNC(=O)c1ccc(cc1)OC 8W-0858 COc1ccc(cc1)/C=N/NC(=O)c2ccc3c(c2)OCO3 8W-0859 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCC(=O)Nc3c2cccc3 8W-0860 Cc1nnc(o1)c2ccc(cc2)OC 8W-0862 c1cc2c(cc1/C=N/NC(=O)c3ccc4c(c3)OCO4)OCO2 8W-0863 c1cc(sc1)/C=N/NC(=O)c2ccc3c(c2)OCO3 8W-0864 CCOc1ccccc1/C=N/NC(=O)c2ccc3c(c2)OCO3 8W-0865 COc1ccc2c(c1)c(c[nH]2)CCNC(=O)Cc3c(cc(cn3)C(F)(F)F)Cl 8W-0866 CCCCCCc1c(ccn(c1=O)CCc2c[nH]c3c2cccc3)Oc4ccc(cn4)C(F)(F)F 8W-0867 c1ccc2c(c1)NCCC(=O)N2Cc3ccc(cc3)Cl 8W-0868 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/c4cccs4)/CC3 8W-0873 c1ccc2c(c1)c3c([nH]2)/C(=N\O)/CCC3 8W-0874 Cn1c(cc(=O)n(c1=O)C)NN 8W-0876 Cc1nnc(o1)c2ccc(cc2)O 8W-0877 CS(=O)(=O)N1CCC(=O)N(c2c1cccc2)Cc3ccc(cc3)Cl 8W-0878 c1cc(sc1)S(=O)(=O)N2CCC(=O)Nc3c2ccc(c3)C(F)(F)F 8W-0880 Cc1ccc(cc1)n2c(nn(c2=O)C(C)C(=O)OC)C 8W-0881 Cc1nn(c(=O)n1c2cccc(c2)OC)CCCC(=O)OC 8W-0882 C1CN(CCC1C(=O)O)C(=O)C(F)(F)F 8W-0884 c1cc([nH]c1)c2ccc3cc(cc(c3n2)Br)Br 8W-0885 COc1cc(c(cc1OC)N)c2ccc3cc(cc(c3n2)Br)Br 8W-0886 Cc1c(sc(n1)C)c2ccc3cc(cc(c3n2)Br)Br 8W-0887 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/c4cccc(c4)F)/CC3 8W-0890 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/c4cccc(c4)[N+](=O)[O-])/CC3 8W-0891 COc1ccccc1/C=C/2\CCc3c4ccccc4[nH]c3C2=O 8W-0892 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/C4CCCCC4)/CC3 8W-0893 c1ccc(c(c1)/C=C/2\CCc3c4ccccc4[nH]c3C2=O)Cl 8W-0894 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/c4cccnc4)/CC3 8W-0895 COc1ccc(cc1)/C=C/2\CCc3c4ccccc4[nH]c3C2=O 8W-0896 COc1ccc(cc1)/C=N/NC(=O)c2csc(n2)c3ccc(cc3)Cl 8W-0897 COc1ccc2c(c1)c(c[nH]2)CCn3ccc(c(c3=O)Cc4ccccc4)O 8W-0900 COc1ccc2c(c1)c(c[nH]2)CCNC(=O)Cc3ccc(cc3)Cl 8W-0901 Cc1c(n(ccc1=O)CCc2c[nH]c3c2cc(cc3)OC)C 8W-0902 COC(=O)c1ccc(cc1)N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4Cl)Cl 8X-0002 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4Cl)Cl 8X-0005 c1cc(c(cc1Cl)Cl)c2cc(n[nH]2)C3CCN(CC3)c4cc(nc(n4)N)Cl 8X-0006 CC(C)(C)c1ccc(cc1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 8X-0023 CC(C)(C)OC(=O)N1CCC(CC1)c2cc([nH]n2)c3ccc(cc3Cl)Cl 8X-0026 c1cc(c(nc1)N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4Cl)Cl)[N+](=O)[O-] 8X-0030 CCOc1ccccc1C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 8X-0046 c1ccc(c(c1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)Br 8X-0047 COc1ccc(c(c1)c2cc(n[nH]2)C3CCNCC3)OC 8X-0048 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4Cl)Cl 8X-0051 c1cc(sc1)c2cc(n[nH]2)C3CCN(CC3)c4cc(nc(n4)N)Cl 8X-0055 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)c3cc([nH]n3)c4cccs4 8X-0056 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4cccs4 8X-0057 CC(C)(C)OC(=O)N1CCC(CC1)c2cc([nH]n2)c3cccs3 8X-0063 c1cc(cc(c1)C(F)(F)F)CN2CCC(CC2)c3cc([nH]n3)c4cccs4 8X-0064 CC(C)c1ccc(cc1)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 8X-0070 c1cc(c(nc1)N2CCC(CC2)c3cc([nH]n3)c4cccs4)[N+](=O)[O-] 8X-0080 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)c3cc([nH]n3)c4cccs4 8X-0081 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)n2c(cc(n2)C3CCNCC3)c4ccc(cc4Cl)Cl.Cl 8X-0088 CC(C)(C)OC(=O)N1CCC(CC1)c2cc(n(n2)C(=O)c3ccc(cc3)OC)c4ccc(cc4Cl)Cl 8X-0090 CC(C)(C)OC(=O)N1CCC(CC1)c2cc(n(n2)C(=O)Nc3ccccc3)c4ccc(cc4Cl)Cl 8X-0091 c1cc(c(cc1Cl)Cl)/C=C\2/C(C3CCN2CC3)O 8X-0092 c1cc(oc1)/C=C\2/C(C3CCN2CC3)O 8X-0093 c1cc(sc1)/C=C\2/C(C3CCN2CC3)O 8X-0103 COc1ccc(c(c1)/C=C\2/C(C3CCN2CC3)O)OC 8X-0114 COc1ccc(cc1)/C=C\2/C(C3CCN2CC3)O 8X-0116 c1cc(ccc1/C=C\2/C(C3CCN2CC3)O)Cl 8X-0119 c1cc(ccc1C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4)[N+](=O)[O-] 8X-0122 COc1cc(ccc1OCC#C)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 8X-0123 COc1ccc(cc1OCC#C)C2c3cc4c(cc3NC5=C2C(=O)OC5)OCO4 8X-0124 Cc1c(n(c(c1S(=O)(=O)C)N)Cc2cccc(c2)OC)C 8X-0200 Cc1c(n(c(c1S(=O)(=O)C)N)CCCN(C)C)C 8X-0201 C/C(=N/NC(=O)Nc1ccc(cc1)Cl)/c2ccc(s2)CC#N 8X-0207 CNC(=S)NNC(=O)C1CCN(CC1)Cc2ccccc2 8X-0209 Cn1c(nnc1S)C2CCN(CC2)Cc3ccccc3 8X-0217 C=CCOc1ccc2cccc(c2c1)/C=N/NC(=O)c3cc4cc(ccc4s3)[N+](=O)[O-] 8X-0227 c1ccc2c(c1)cccc2c3cc(n[nH]3)C4CCN(CC4)C(=O)c5cc6ccccc6s5 8X-0230 c1ccc\2c(c1)CCC/C2=N/Nc3ccc(cc3[N+](=O)[O-])S(=O)(=O)N4CCC(CC4)C(=O)O 8X-0231 CS(=O)(=O)N1CC(Oc2c1cc(cc2)Cl)C(=O)NC3CC3 8X-0232 Cc1ccc(cc1)CNC(=O)C2CN(c3cc(ccc3O2)Cl)S(=O)(=O)C 8X-0233 CCOC(CCNC(=O)C1CN(c2cc(ccc2O1)Cl)S(=O)(=O)C)OCC 8X-0234 CC(=O)c1ccc2cc(ccc2c1)O 8X-0242 C1COCCN1C(=N)NN.I 8X-0245 C/C(=C(\C=C\C(=O)OC)/C(=O)OC)/NCc1ccc(cc1)F 8X-0246 c1cc(ccc1c2c(cnc(n2)NC(=S)N)CCN3CCOCC3)F 8X-0251 COc1ccccc1CNC(=O)C2CN(c3cc(ccc3O2)Cl)S(=O)(=O)C 8X-0254 CS(=O)(=O)N1CC(Oc2c1cc(cc2)Cl)C(=O)NC3CCCC3 8X-0255 COc1cccc(c1)CNC(=O)C2CN(c3cc(ccc3O2)Cl)S(=O)(=O)C 8X-0256 CS(=O)(=O)N1CC(Oc2c1cc(cc2)Cl)C(=O)NCc3ccc(c(c3)Cl)Cl 8X-0257 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)Nc3[nH]c(=O)cc(n3)C(F)(F)F 8X-0264 CC(=O)c1ccc2cc(ccc2c1)N(C)CCO 8X-0270 Cc1cccc(c1N2CCN(CC2)C(=N)N[NH3+])C.[I-] 8X-0273 CCOC(=O)COc1ccc2ccccc2c1C=C3C(=O)N(C(=O)N(C3=O)C)C 8X-0278 COc1cccc(c1)CS/C(=N\c2[nH]c(=O)cc(n2)C(F)(F)F)/N 8X-0287 CCOC(=O)COc1ccc2ccccc2c1C=C(C#N)C#N 8X-0291 CN1C(=O)C(=Cc2ccc(nc2)Oc3cccc(c3)C(F)(F)F)C(=O)N(C1=O)C 8X-0292 CCCc1ccc(cc1)C(=O)/C=C/N(C)C 8X-0295 CC(C)(C)OC(=O)N1CCc2c1ccc(c2)Br 8X-0296 Cc1c(cc(n1Cc2ccc(cc2)F)C(=O)OC)C(=O)OC 8X-0299 CC1(OCCO1)c2cccc(c2)N 8X-0600 c1cc(c(cc1Cl)Cl)Cn2cc(cc(c2=O)C(=O)O)Br 8X-0700 c1ccc(c(c1)C=O)Oc2cc(cc(c2)F)F 8X-0701 c1ccc(c(c1)/C=C/C(=O)O)Oc2cc(cc(c2)F)F 8X-0703 c1ccc(cc1)Oc2ccccc2CCC(=O)O 8X-0704 COc1ccc(cc1)C(=O)N2CCC(CC2)C(=O)O 8X-0705 c1cc(ccc1C(=O)N2CCC(CC2)C(=O)O)Cl 8X-0706 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)O 8X-0707 CCC(=O)c1cc([nH]c1)C(=O)O 8X-0708 c1ccc(c(c1)CCC(=O)O)Oc2ccc(cc2)Cl 8X-0710 c1ccc-2c(c1)CCc3c2sc(c3)C(=O)NN 8X-0712 Cc1ccc(cc1)Oc2ccccc2CCC(=O)O 8X-0713 c1cc(cc(c1)[N+](=O)[O-])C(=O)N2CCC(CC2)C(=O)O 8X-0715 c1ccc(c(c1)CCC(=O)O)Oc2ccc(cc2Cl)Cl 8X-0716 COc1cccc(c1)C(=O)c2cc([nH]c2)C(=O)O 8X-0717 CCCC(=O)c1cc([nH]c1)C(=O)O 8X-0719 COc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)O 8X-0721 Cn1cc(cc1C(=O)O)C(=O)c2ccccc2C(=O)O 8X-0722 COc1ccc(cc1)Oc2ccccc2CCC(=O)O 8X-0723 Cc1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)O 8X-0724 c1ccc(c(c1)C(=O)O)SCC(C(F)(F)F)O 8X-0728 CCOC(=O)c1cc(cn1C)C(=O)c2ccccc2C(=O)O 8X-0729 c1cc(cc(c1)F)COc2ccc(cc2)C(=O)O 8X-0730 c1cc(ccc1C(=O)O)OCc2ccc(c(c2)Cl)Cl 8X-0731 c1cc(cc(c1)F)COc2ccc(cc2)C(=O)NN 8X-0732 CCOC(=O)c1cc2cc(ccc2s1)N 8X-0733 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CCC(=O)O 8X-0734 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CCC(=O)NN 8X-0738 CS(=O)(=O)c1ccc2c(c1)sc3n2cc(n3)C(=O)O 8X-0800 CN(C)Cc1cnc2n1cc(cc2)Cl 8X-0801 Cc1cc(n(n1)c2ccc(cc2)OC)N 8X-0802 c1cc2nccn2cc1[N+](=O)[O-] 8X-0803 CCOC(=O)c1cn2c3ccc(cc3sc2n1)S(=O)(=O)C 8X-0807 Cc1cccn2c1ncc2C(=O)OC 8X-0808 Cc1c2c(cc(nc2n(n1)c3cccc(c3)F)C(F)(F)F)C(F)(F)F 8X-0809 Cc1c2c(cc(nc2n(n1)c3cccc(c3)F)c4ccccc4)C(F)(F)F 8X-0810 c1ccc2cc(ccc2c1)c3ccc(cn3)C(=O)c4ccc5ccccc5c4 8X-0811 Cc1ccc2ncc(n2c1)CN(C)C 8X-0813 Cc1cc(n2c(n1)nc(n2)SCCOc3ccccc3)C 8X-0815 Cc1cc(n2c(n1)nc(n2)SCC(=O)Nc3ccc(cc3)OC)C 8X-0816 COC(=O)c1cnc2n1cc(cc2)Cl 8X-0819 Cc1ccc2c(c1)sc3n2cc(n3)c4ccc(cc4)OC 8X-0820 CCOC(=O)c1cn2c3ccc(cc3sc2n1)F 8X-0821 c1c(cc(c(c1C=O)O)F)Br 8X-0823 c1cc2ncc(n2cc1Cl)C(=O)O 8X-0825 c1cc2ncc(n2cc1Cl)C(=O)NN 8X-0826 Cc1ccc2c(c1)sc3n2cc(n3)c4ccc(cc4)Br 8X-0828 CN(C)Cc1cnc2n1cc(cc2)Br 8X-0831 c1ccc(cc1)CNNC(=S)N 8X-0832 c1cc(cc(c1)[N+](=O)[O-])NNC(=S)N 8X-0833 Cc1cccc(c1C)NNC(=S)N 8X-0834 c1cc(cc(c1)Br)NNC(=S)N 8X-0835 CCOC(=O)c1c(nc(s1)N)C(F)(F)F 8X-0838 CCOC(=O)c1c(nc2n1cc(cc2)Cl)C(F)(F)F 8X-0839 c1cc(c2nccn2c1)O 8X-0841 C1=CC2=NC=C([NH+]2C=C1Cl)C(=O)C(F)(F)Cl.C(=O)(C(F)(F)Cl)[O-] 8X-0842 COC(=O)Cc1c(ccn(c1=O)Cc2cccc3c2cccc3)O 8X-0843 c1ccc2c(c1)cc(cn2)C(=O)C3CC3 8X-0845 c1ccc(cc1)C(CCNC(=O)Cn2cncn2)c3ccccc3 8X-0847 c1ccc(c(c1)CNC(=O)Cn2cncn2)Br 8X-0848 c1cn2cc(cc(c2n1)Cl)C(F)(F)F 8X-0850 Cc1cccc2n1ccn2 8X-0855 Cc1cccc(c1N2CCN(CC2)CC(COc3ccc(cc3)OC)O)C 8X-0856 Cc1ccc(cc1)CNC(=O)Cn2cncn2 8X-0857 c1ccc2c(c1)cccc2CNC(=O)Cn3cncn3 8X-0858 c1cnc(nc1)N2CCN(CC2)C(=O)Cn3cncn3 8X-0859 c1cc(ccc1N2CCN(CC2)C(=O)Cn3cncn3)F 8X-0860 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SCc4ccc(cc4)C(=O)OC)C(F)(F)F 8X-0861 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SCC(=O)N(C)c4ccccc4)C(F)(F)F 8X-0862 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SC(CC(=O)O)C(=O)c4ccccc4)C(F)(F)F 8X-0863 c1cc2ncc(n2cc1C(=O)O)Cl 8X-0864 c1cc2ncc(n2cc1C(=O)O)Br 8X-0865 Cc1cccn2c1ncc2C(=O)O 8X-0866 c1(c(nc(s1)N)C(F)(F)F)C(=O)O 8X-0867 c1cc2nc(c(n2cc1Cl)C(=O)O)C(F)(F)F 8X-0868 Cc1c(nnn1c2ccc(c(c2)Cl)Cl)C(=O)c3c(cc(cn3)C(F)(F)F)c4ccc(cc4)OC 8X-0870 c1ccc(cc1)S(=O)(=O)N/N=C/c2cc(c[nH]2)C(=O)CCl 8X-0925 c1ccc2c(c1)-c3c(c(c(c(n3)/C=C/c4cccc(c4)Br)C#N)c5ccc6c(c5)OCO6)C2=O 8X-0928 c1ccc2c(c1)-c3c(c(c(c(n3)/C=C/c4cccc(c4)Cl)C#N)c5ccc6c(c5)OCO6)C2=O 8X-0929 c1ccc(c(c1)/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccc6c(c5)OCO6)C#N)F 8X-0930 COc1ccc(cc1)/C=C/c2c(c(c3c(n2)-c4ccccc4C3=O)c5ccc6c(c5)OCO6)C#N 8X-0931 c1ccc2c(c1)-c3c(c(c(c(n3)/C=C/c4ccc(c(c4)Cl)Cl)C#N)c5ccc6c(c5)OCO6)C2=O 8X-0932 c1ccc2c(c1)-c3c(c(c(c(n3)/C=C/c4ccc(cc4)[N+](=O)[O-])C#N)c5ccc6c(c5)OCO6)C2=O 8X-0933 Cc1cc(=S)n(c(=S)[nH]1)N 8X-0936 c1cc(ccc1N/N=C/c2cc(c[nH]2)C(=O)CCl)[N+](=O)[O-] 8X-0937 CC(=O)NNC(=O)c1c[nH]c2c1cccc2 8X-0938 COc1cccc(c1)CN(CCO)CCO 8X-0941 Cc1ccc(cc1)CN(CCO)CCO 8X-0945 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N/N=C/c2cc(c[nH]2)C(=O)CCl 8X-0948 COc1cccc(c1)C[NH+](CCCl)CCCl.[Cl-] 8X-0949 Cn1c2ccccc2c(c(c1=O)c3cc(=O)[nH][nH]3)O 8X-0951 Cc1ccc(cc1)C[NH+](CCCl)CCCl.[Cl-] 8X-0952 c1cc2c3c(c1)c4c(c(cc(=O)o4)O)c(=O)n3CC2 8X-0953 Cc1cc(=S)n2c(n1)sc(n2)c3ccc(cc3)C(F)(F)F 8X-0955 CCOC(=O)C1(CCN(CC1)Cc2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)OC 8X-0956 CCOC(=O)C1(CCN(CC1)Cc2ccc(cc2)C)S(=O)(=O)c3ccc(cc3)OC 8X-0957 Cc1c(c(n(n1)C)/C=C/Nc2ccccc2)[N+](=O)[O-] 8X-0958 CN(C)/C=N\c1ncc2c(n1)-c3ccccc3OC2 8X-0963 CC1CN(CC(O1)C)C2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)N2 8X-0964 Cc1ccc(cc1)CO/N=C/Nc2ncc3c(n2)-c4ccccc4OC3 8X-0965 c1ccc2c(c1)-c3c(cnc(n3)N/C=N/OCc4ccc(cc4)F)CO2 8X-0967 Cc1cc(=S)n2c(n1)sc(n2)c3cccc(c3)OC 8X-0968 COc1ccc2c(c1)CC(=O)NC=C2 8X-0973 CCOC(=O)CSc1ccc(cc1)O 8X-0974 CCOC(=O)CSc1ccc(cc1)Cl 8X-0975 CN(C)/C=C/1\CSc2ccc(cc2C1=O)Cl 8X-0976 CCOC(=O)C1CSC2([NH2+]1)CCC(CC2)C.[Cl-] 8X-0977 CC(C)n1c2ccccc2c3c(c1=O)c(cc(=O)o3)O 8X-0978 CCOC(=O)CS(=O)(=O)c1ccc(cc1)Cl 8X-0979 c1ccc(cc1)C(=O)c2ccsc2N 8X-0980 c1ccc(c(c1)N/N=C/c2cc(c[nH]2)C(=O)CCl)Cl 8X-0982 CCCCc1nc2cc(ccc2o1)S(=O)(=O)CC 8X-5012 c1c2c(cc(c1Cl)[N+](=O)[O-])ocn2 8X-5013 CCCCc1nc2cc(ccc2o1)Cl 8X-5014 Cc1nc2cc(c(cc2o1)[N+](=O)[O-])Cl 8X-5015 CCc1nc2cc(c(cc2o1)[N+](=O)[O-])Cl 8X-5016 CC(C)(C)n1c(c(cn1)C(=O)N2CCOCC2)C(F)(F)F 8X-5073 CCCCc1nc2cc(ccc2o1)CC(=O)OC 8X-5074 c1cc(cc(c1)Br)C2C[C@H]2C(=O)O 8X-7015 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CS(=O)(=O)N 8X-7017 c1cc(cc(c1)S(=O)(=O)N2CCOCC2)C(=O)O 8Y-0008 c1cc(c(cc1c2nc3cc(cc(c3o2)Br)O)F)O 8Y-0027 c1cc2c(cc1C(=O)CCl)NC(=O)CO2 8Y-0030 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2ccc(cc2)[N+](=O)[O-] 8Y-0035 C1CC2C1C(=O)OC2=O 8Y-0041 CN1c2ccc(cc2OCC1=O)N 8Y-0701 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCCC(=O)O 8Y-0702 COC(=O)CCNc1ccc(cc1N)C(F)(F)F 8Y-0703 CN1c2cc(ccc2OCC1=O)N 8Y-0704 c1cc(c(cc1[N+](=O)[O-])C(=O)O)N2CCNCC2 8Y-0705 COC(=O)c1cc(c[nH]c1=O)I 8Y-0707 c1c(c(cs1)Br)/C=N/NC(=S)N 8Y-0800 c1cc2c(cc1C/N=C/c3cscc3Br)OCO2 8Y-0801 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc(c1Cl)Cl 8Y-0803 c1cc(cc(c1)N2CCS(=O)(=O)CC2)C(=O)O 8Y-0805 c1cc(ccc1CN2CCS(=O)(=O)CC2)C(=O)O 8Y-0806 COc1ccc(cc1)c2ccc(cc2)C(=O)O 8Y-0809 Cc1cc(n[nH]1)c2ccsc2 8Y-0813 Cc1cc(nc(n1)N)c2ccsc2 8Y-0823 CN1CCCN(CC1)Cc2cnc(s2)Cl 8Y-0824 c1c(sc(n1)Cl)CN2CCCCCC2 8Y-0825 CCCN(Cc1cnc(s1)Cl)CC2CC2 8Y-0826 COC(=O)c1cccc(c1)N2CCS(=O)(=O)CC2 8Y-0827 c1cc2nccn2cc1C#N 8Y-0828 COC(Cn1cccc1)OC 8Y-0829 COc1c(cc(s1)C(=O)CBr)Br 8Y-0830 Cc1nccn1c2ccc(cc2)C(=O)OC 8Y-0831 CC(=O)c1cc(c(s1)OC)Br 8Y-0833 Cc1ccc(cc1[N+](=O)[O-])COc2ccc(cc2Cl)C(=O)C 8Y-0929 CSC1=NCCCN1.I 8Y-5009 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CNC(=O)C 8Y-7010 c1c(cnc(c1Cl)SCCN)C(F)(F)F.Cl 8Z-0031 C1CCC2(C1)CC(=O)NC2 8Z-0036 c1c(cnc(c1Cl)NCCOc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 8Z-0040 c1cc2c(nc1)NC(=O)C(O2)CCCBr 8Z-0204 c1cc2c(nc1)NC(=O)C(O2)CCCCBr 8Z-0205 COc1ccccc1N2CCN(CC2)CCCCC3C(=O)Nc4c(cccn4)O3 8Z-0209 COc1ccccc1N2CCN(CC2)CCCC3C(=O)Nc4c(cccn4)O3 8Z-0210 c1cc(cc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F 8Z-0215 CC(C)C1CNCCN1 8Z-0600 c1cc(c2nccn2c1)[N+](=O)[O-] 8Z-0801 COC(C(=O)N1CCCCC1)OC 8Z-0803 c1cc(c(c(c1)C#N)NCC2CCCO2)C#N 8Z-0804 Cc1ccc(cc1)c2cc[nH]c(=O)c2C#N 8Z-0808 c1cc(c(cc1c2ccn[nH]2)N)N3CCOCC3 8Z-0809 c1cc(cc(c1)I)Oc2ncccn2 8Z-0812 c1cc2c(nc1)NC(=O)C(O2)CCBr 8Z-0814 c1ccc(c(c1)C(=O)N)NC(=O)c2ccc(c(c2)[N+](=O)[O-])N3CCCCCC3 8Z-0820 c1ccc(cc1)COc2cccn3c2ncc3 8Z-0821 c1cc2nc(cn2cc1Cl)C(=O)NCCCO 8Z-0831 COC(CNC(=O)c1cn2cc(ccc2n1)Cl)OC 8Z-0833 Cc1ccc(cc1)c2ccnc(c2C#N)Cl 8Z-0836 CC(C)(C)C(=O)Nc1ccccc1Cl 8Z-0840 Cn1cc(c2c1ccc(c2)OC)C=O 8Z-0841 Cc1ccc(cc1)c2cc(cc3c2cc(c(c3)OC)OC)C(=O)O 8Z-7003 COC(=O)c1ccc(cc1)NC=C2C(=NNC2=O)C(F)(F)F 9B-001 COC(=O)c1c(ccs1)NC=C2C(=NNC2=O)C(F)(F)F 9B-002 Cc1cccc(c1NC=C2C(=NNC2=O)C(F)(F)F)C 9B-003 C(=N/O)\C1C(=NNC1=O)C(F)(F)F 9B-004 Cc1cccc(c1NC=C2C=NNC2=O)C 9B-005 CC(=O)/C(=C/c1ccccc1)/Oc2ccc(cc2)Cl 9B-007 COC(=O)CNC=C1C=NNC1=O 9B-008 c1cc(nc(c1)Cl)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl 9B-010 CC(C)(C)NC(=O)N1CCN(CC1)c2cccc(n2)Cl 9B-011 CS/C(=N/C#N)/N1CCN(CC1)c2cccc(n2)Cl 9B-013 c1cc(nc(c1)Cl)N2CCN(CC2)C(=O)c3ccc(cc3)F 9B-014 c1cc(nc(c1)Cl)N2CCN(CC2)C(=O)c3ccc(cc3)Cl 9B-015 CN(C)/C=C/C(=O)/C(=C/c1ccccc1)/Oc2ccc(cc2)Cl 9B-016 CS(=O)(=O)N1CCN(CC1)c2cccc(n2)Cl 9B-017 c1cc(nc(c1)Cl)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl 9B-018 Cc1c(c(on1)/C=C/N(C)C)[N+](=O)[O-] 9B-022 CCSC(C(=O)N)SCC 9B-026 c1ccc(cc1)C=CC(=O)N2CCN(CC2)c3cccc(n3)Cl 9B-028 c1ccc(cc1)/C=C(\c2ccnc(n2)N)/Oc3ccc(cc3)Cl 9B-031 CN(C)/C=C/1\COC(C1=O)(c2ccccc2)c3ccccc3 9B-033 CN(C)/C=C(\c1ccccn1)/C(=S)N2CCOCC2 9B-037 CN(C)/C=N/C(=O)/C=C/c1ccccc1 9B-038 CCSC(C(=O)NC(=O)C(=O)Nc1ccccc1)SCC 9B-041 CCSC(C(=O)/C=C/N(C)C)SCC 9B-043 CCSC(C1=NC(=O)C(=O)O1)SCC 9B-044 c1ccc2c(c1)c(=O)nc(s2)CC(=O)N 9B-045 c1ccc(cc1)NC(=O)CC#N 9B-046 c1cc(ccc1NC(=O)CC#N)Cl 9B-047 CCSC(C(=O)NC(=O)Nc1ccccc1)SCC 9B-048 CN(C)/C=C(\C(=O)CSc1ccccc1)/Sc2ccccc2 9B-052 CCSC(c1cc[nH]n1)SCC 9B-053 c1ccc(cc1)NC(=O)Cc2nc(=O)c3ccccc3s2 9B-054 c1ccc2c(c1)c(=O)nc(s2)CC(=O)Nc3ccc(cc3)Cl 9B-055 c1ccc(cc1)SCc2cnc(nc2Sc3ccccc3)N 9B-056 c1cc(cc(c1)NC(=O)CC#N)C(F)(F)F 9B-057 CCSC(c1ccnc(n1)N)SCC 9B-058 c1ccc2c(c1)c(=O)nc(s2)CC(=O)Nc3cccc(c3)C(F)(F)F 9B-059 c1ccc(c(c1)C(=O)c2cc(c(nc2O)C(F)(F)F)C(=O)O)O 9B-060 CCSC(c1ccnn1c2ccccc2)SCC 9B-062 c1ccnc(c1)NC(=O)CC#N 9B-063 c1cnccc1NC(=O)CC#N 9B-064 CCSC(c1n[nH]nn1)SCC 9B-070 c1ccc2c(c1)c(=O)nc(s2)CC(=O)Nc3ccccn3 9B-071 COC(=O)c1c[nH]c(=O)c2c1cccc2 9B-073 CN1CCN(CC1)c2ccc(cc2)C(=O)/C=C/N(C)C 9B-075 COC(=O)c1cnc(c2c1cccc2)Cl 9B-078 c1cc(cnc1)NC(=O)CC#N 9B-079 CN(C)/C=C/c1c(cc2c(=O)c3ccccc3oc2n1)C(=O)OC 9B-081 CCSC(c1nc[nH]n1)SCC 9B-083 CN1CCN(CC1)c2ccc(cc2)c3ccn[nH]3 9B-084 c1ccc2c(c1)c(=O)nc(s2)CC(=O)Nc3cccnc3 9B-085 CCSC(c1ccn(n1)C)SCC 9B-086 c1c(cc(cc1Cl)Cl)NC=C2C=NNC2=O 9B-087 CC1=NNC(=O)C1=CNc2cc(cc(c2)Cl)Cl 9B-088 c1c(cc(cc1Cl)Cl)NC=C2C(=NNC2=O)C(F)(F)F 9B-089 CC1=NNC(=O)C1/C=N/O 9B-090 CN(C)C=C1C(=NNC1=O)c2ccccc2 9B-094 CO/N=C/C1C(=NNC1=O)C(F)(F)F 9B-095 CO/N=C/C1C=NNC1=O 9B-096 CC1=NNC(=O)C1/C=N/OC 9B-097 CO/N=C/C1C(=NNC1=O)c2ccccc2 9B-098 COC(=O)CNC=C1C(=NNC1=O)C(F)(F)F 9B-099 CC1=NNC(=O)C1=CNCC(=O)OC 9B-100 COC(=O)CNC=C1C(=NNC1=O)c2ccccc2 9B-101 c1c(cnc(c1Cl)NN)C(F)(F)F 9B-102 c1ccc(cc1)C2=NNC(=O)C2/C=N/O 9B-103 c1ccc(cc1)NNC=C2C(=NNC2=O)C(F)(F)F 9B-104 c1ccc(c(c1)C(=O)NNC=C2C(=NNC2=O)C(F)(F)F)O 9B-105 c1ccc(cc1)S(=O)(=O)NNC=C2C(=NNC2=O)C(F)(F)F 9B-106 c1cc(cc(c1)Cl)C(=O)NNC=C2C(=NNC2=O)C(F)(F)F 9B-107 c1cc(ccc1C(=O)NNC=C2C(=NNC2=O)C(F)(F)F)Cl 9B-108 c1cc(c(c(c1)Cl)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl 9B-109 c1ccc(cc1)C2=NNC(=O)C2=CNc3ccccc3 9B-111 c1ccc(cc1)C2=NNC(=O)C2=CNc3ccccc3Cl 9B-112 c1ccc(cc1)C2=NNC(=O)C2=CNc3cccc(c3)Cl 9B-113 c1ccc(cc1)C2=NNC(=O)C2=CNc3ccc(cc3)Cl 9B-114 c1ccc(cc1)C2=NNC(=O)C2=CNc3cccc(c3)C(F)(F)F 9B-115 Cc1ccc(cc1)NC=C2C(=NNC2=O)c3ccccc3 9B-116 COc1ccc(cc1)NC=C2C(=NNC2=O)c3ccccc3 9B-117 COC(=O)c1ccc(cc1)NC=C2C(=NNC2=O)c3ccccc3 9B-118 COC(=O)c1c(ccs1)NC=C2C(=NNC2=O)c3ccccc3 9B-119 c1ccc(cc1)C2=NNC(=O)C2=CNc3ccc(cc3F)F 9B-120 c1ccc(c(c1)CNC=C2C(=NNC2=O)C(F)(F)F)Cl 9B-122 c1cc(cc(c1)Cl)CNC=C2C(=NNC2=O)C(F)(F)F 9B-123 c1cc(ccc1CNC=C2C(=NNC2=O)C(F)(F)F)Cl 9B-124 COc1ccc(cc1)CNC=C2C(=NNC2=O)C(F)(F)F 9B-125 c1ccc(cc1)C2=NNC(=O)C2=CNCc3cccnc3 9B-126 c1cc(cnc1)CNC=C2C=NNC2=O 9B-127 CC1=NNC(=O)C1=CNCc2cccnc2 9B-128 c1ccc(cc1)C2=NNC(=O)C2=CNCc3ccccn3 9B-129 CC1=NNC(=O)C1=CNCc2ccc(cc2)Cl 9B-130 Cc1ccc(cc1)CNC=C2C(=NNC2=O)C 9B-131 CN1CCN(CC1)c2ccc(cc2)c3ccnc(n3)N 9B-132 CN1CCN(CC1)c2ccc(cc2)c3ccnn3C(=O)Nc4cccc(c4)C(F)(F)F 9B-133 CN1CCN(CC1)c2ccc(cc2)c3ccnn3C(=O)Nc4ccc(cc4Cl)Cl 9B-134 CN1CCN(CC1)c2ccc(cc2)c3ccnn3C(=O)Nc4ccccc4 9B-135 C(C(=N)[NH3+])C(=O)N.[Cl-] 9C-005 CN(C)C(=O)c1c2ccccc2c(=O)n(n1)c3ccccc3 9C-006 COC(=O)c1c2ccccc2c(=O)n(n1)c3ccccc3 9C-009 c1ccc(cc1)NC(=O)c2c3ccccc3c(=O)n(n2)c4ccccc4 9C-011 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)Oc4ccccc4 9C-015 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)Nc4ccc(cc4)Cl 9C-017 Cc1cc(nc(c1C(=O)N)N)C 9C-018 CN(C)C(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)OC 9C-019 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)OC 9C-024 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)Nc4ccccc4 9C-025 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)Nc4ccc(cc4)Cl 9C-026 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)Oc4ccccc4 9C-027 CN(C)C(=O)c1c2ccccc2c(=O)n(n1)c3cccc(c3)C(F)(F)F 9C-031 COC(=O)c1c2ccccc2c(=O)n(n1)c3cccc(c3)C(F)(F)F 9C-032 c1ccc(cc1)NC(=O)c2c3ccccc3c(=O)n(n2)c4cccc(c4)C(F)(F)F 9C-039 CC(C(=O)C)Oc1ccccc1 9C-042 CC(C(=O)C)Oc1ccc(cc1Cl)Cl 9C-043 Cc1cc(nc(c1C(=O)N)NC(=O)Nc2ccccc2Cl)C 9C-050 Cc1cc(nc(c1C(=O)N)NC(=O)Nc2cccc(c2)Cl)C 9C-051 Cc1cc(nc(c1C(=O)N)NC(=O)Nc2ccc(cc2)Cl)C 9C-052 CC(C(=O)C)Oc1cccc(c1)C(F)(F)F 9C-053 Cc1cc(nc(c1C(=O)N)NC(=O)Nc2cccc(c2)C(F)(F)F)C 9C-054 Cc1ccc(cc1)NC(=O)Nc2c(c(cc(n2)C)C)C(=O)N 9C-055 Cc1cc(nc(c1C(=O)N)NC(=O)Nc2ccc(cc2)OC(F)(F)F)C 9C-056 Cc1cc(nc(c1C(=O)N)NC(=O)Nc2ccccc2)C 9C-057 c1ccc(cc1)OC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(cc4)Cl 9C-061 c1ccc(cc1)NC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(cc4)Cl 9C-063 CC(C(=O)C=CN(C)C)Oc1ccccc1 9C-064 CC(C(=O)/C=C/N(C)C)Oc1ccc(cc1Cl)Cl 9C-066 c1ccc(c(c1)c2ccno2)O 9C-067 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)Cl 9C-070 CC(C(=O)C=CN(C)C)Oc1cccc(c1)C(F)(F)F 9C-071 CN(C)c1c(cc(s1)C(=O)c2ccc(cc2)Cl)c3ccccc3 9C-072 CN(C)c1c(cc(s1)C(=O)c2ccc(cc2)F)c3ccccc3 9C-073 c1ccc(cc1)OC(=O)c2c3ccccc3c(=O)n(n2)c4cccc(c4)C(F)(F)F 9C-075 c1ccc2c(c1)c(nn(c2=O)c3cccc(c3)C(F)(F)F)C(=O)Nc4ccc(cc4)Cl 9C-076 CC(c1ccnc(n1)N)Oc2ccccc2 9C-079 CC(c1ccnc(n1)N)Oc2ccc(cc2Cl)Cl 9C-080 CC(c1ccnc(n1)N)Oc2cccc(c2)C(F)(F)F 9C-081 CC(c1ccn[nH]1)Oc2ccccc2 9C-082 CC(c1ccn[nH]1)Oc2ccc(cc2Cl)Cl 9C-083 CC(c1ccno1)Oc2ccc(cc2)Cl 9C-084 CC(c1ccn[nH]1)Oc2cccc(c2)C(F)(F)F 9C-085 CC(=O)c1cc(cc(c1O)Cl)Cl 9C-086 Cc1cc(nc(c1C(=O)O)N)C 9C-087 CC(c1ccno1)Oc2ccc(cc2Cl)Cl 9C-088 CC(c1ccno1)Oc2ccccc2 9C-089 CC(c1ccno1)Oc2cccc(c2)C(F)(F)F 9C-090 c1c(cc(c2c1c(=O)c(co2)C=O)Cl)Cl 9C-091 CC(c1ccnn1C(=O)Nc2ccccc2)Oc3ccccc3 9C-092 CC(c1ccnn1C(=O)c2ccccc2)Oc3ccc(cc3)Cl 9C-093 CC(c1ccnn1C(=O)Nc2ccccc2)Oc3ccc(cc3)Cl 9C-096 CC(c1ccnn1S(=O)(=O)c2ccccc2)Oc3ccccc3 9C-097 CC(c1ccnn1S(=O)(=O)c2ccccc2)Oc3ccc(cc3)Cl 9C-098 CC(C)(C)S(=O)(=O)CC#N 9C-101 CC(c1ccnn1C(=O)c2ccccc2)Oc3ccccc3 9C-104 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)C(F)(F)F)/C#N 9C-111 CC(c1ccnn1C(=O)c2ccccc2)Oc3cccc(c3)C(F)(F)F 9C-113 CC(C)(C)S(=O)(=O)/C(=N/Nc1ccc(cc1)Cl)/C#N 9C-114 Cc1cc(nc(c1C(=O)/N=C/N(C)C)N)C 9C-115 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)C(F)(F)F)/OC2=O 9D-001 COC(=O)c1ccccc1Sc2c(n3ccsc3n2)C=O 9D-003 c1ccc2c(c1)c(n[nH]c2=O)CNc3ccc(cc3)C(F)(F)F 9D-009 COC(=O)c1ccccc1Sc2c(n3ccsc3n2)/C=N\O 9D-010 COC(=O)c1ccccc1Sc2c(n3ccsc3n2)/C=N\OC 9D-011 COC(=O)c1ccccc1Sc2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl 9D-012 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/O 9D-013 Cc1ccc(cc1)SC2=C(/C(=C\N(C)C)/S(=O)(=O)C2)C(=O)C 9D-014 CN(C)c1c(cc(s1)C(=O)c2ccc(cc2)Cl)c3ccc(cc3)Oc4ccccc4 9D-018 CN(C)c1c(cc(s1)C(=O)c2ccc(cc2Cl)Cl)c3ccc(cc3)Oc4ccccc4 9D-019 CN(C)c1c(cc(s1)C(=O)c2ccccc2)c3ccc(cc3)Oc4ccccc4 9D-020 CN(C)c1c(cc(s1)C(=O)c2ccc(cc2)Br)c3ccc(cc3)Oc4ccccc4 9D-022 COc1ccc(cc1)/C=C(/C#N)\C(=O)N/C=N/OCc2ccc(cc2Cl)Cl 9D-023 c1ccc2c(c1)/C(=C/N3CCN(CC3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])/OC2=O 9D-027 c1(c(nc(n(c1=O)N)N)C(F)(F)F)Br 9D-031 c1ccnc(c1)c2nc(c(c(n2)O)C#N)c3ccc(cc3)Cl 9D-033 c1ccnc(c1)c2nc(c(c(n2)Cl)C#N)c3ccc(cc3)Cl 9D-035S c1ccc(cc1)c2nc(c(c(n2)Cl)C#N)c3ccc(cc3)Cl 9D-036S CC(=O)COC(=O)Cc1ccc(cc1)[N+](=O)[O-] 9D-037 c1cc(ccc1C2=C(C(=O)OC2)C#N)Br 9D-038 CC1=C(C(=O)OC1)c2ccc(cc2)[N+](=O)[O-] 9D-039 CC\1=C(C(=O)O/C1=C\N(C)C)c2ccc(cc2)[N+](=O)[O-] 9D-042 c1ccc(cc1)c2ccc(cc2)C3=C(C(=O)OC3)C#N 9D-044 COc1ccc(cc1)C2=C(C(=O)OC2)C#N 9D-045 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)O 9D-046 Cc1ccc(c(c1)C)NCc2c(nc3n2ccs3)Cl 9D-047 CSc1nc(c(c(n1)O)C#N)c2ccccc2 9D-048 c1ccc(cc1)CSc2c(n3ccsc3n2)C=O 9D-055 c1cc(ccc1CSc2c(n3ccsc3n2)/C=N/OCc4ccc(c(c4)Cl)Cl)Cl 9D-056 c1cc(ccc1CSc2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl)Cl 9D-057 c1ccc(cc1)CSc2c(n3ccsc3n2)/C=N/OCc4ccc(c(c4)Cl)Cl 9D-058 c1cc(c(cc1Cl)Cl)Cc2ccc(nn2)NN 9D-060 c1cc(sc1)/C=C(\C#N)/C(=O)N/C=N/OCc2ccc(cc2Cl)Cl 9D-063 c1ccc(cc1)/C=C/C=C(/C#N)\C(=O)N/C=N/OCc2ccc(cc2Cl)Cl 9D-064 c1ccc(cc1)CSc2c(n3ccsc3n2)/C=N/OCc4ccc(cc4Cl)Cl 9D-065 c1ccc(cc1)CSc2c(n3ccsc3n2)/C=N/O 9D-066 Cc1cc(n(n1)c2ccc(nn2)Cc3ccc(cc3Cl)Cl)C 9D-068 c1ccc(cc1)c2ccnn2c3ccc(nn3)Cc4ccc(cc4Cl)Cl 9D-070 c1cc(ccc1C2=C(C(=O)OC2)C#N)F 9D-071 c1ccc(cc1)CSc2c(n3ccsc3n2)/C=N/OCc4c(cccc4Cl)Cl 9D-073 c1csc2n1c(c(n2)Cl)/C=N/O 9D-074 CC(C)Sc1c(n2ccsc2n1)C=O 9D-080 CO/N=C/c1c(nc2n1ccs2)Cl 9D-081 c1cc(c(cc1Cl)Cl)CO/N=C/c2c(nc3n2ccs3)Cl 9D-082 CC(C)Sc1c(n2ccsc2n1)/C=N/O 9D-083 CC(C)Sc1c(n2ccsc2n1)/C=N/OCc3c(cccc3Cl)Cl 9D-084 c1cc(c(cc1CO/N=C/c2c(nc3n2ccs3)Cl)Cl)Cl 9D-085 c1cc(ccc1C(=O)C/C=N/OCc2ccc(cc2Cl)Cl)Br 9D-086 c1cc(c(cc1C(=O)C/C=N/OCc2ccc(cc2Cl)Cl)Cl)Cl 9D-087 c1cc(ccc1/C=C(/C#N)\C(=O)N/C=N/OCc2ccc(cc2Cl)Cl)Cl 9D-088 c1cc(ccc1C(=O)C/C=N/OCc2ccc(cc2Cl)Cl)F 9D-089 c1ccc(cc1)c2ccc(cc2)C(=O)C/C=N/OCc3ccc(cc3Cl)Cl 9D-090 CC\1=C(C(=O)O/C1=C\Nc2ccccc2)c3ccc(cc3)[N+](=O)[O-] 9D-092 c1csc2n1c(c(n2)Cl)C#N 9D-095S c1cc(c(c(c1)Cl)CO/N=C/c2c(nc3n2ccs3)Cl)Cl 9D-096 c1cc(c(cc1Cl)Cl)NC(=O)CC(=O)O 9D-097 CN(C)/C=C/C(=O)Nc1ccc(cc1Cl)Cl 9D-098 Cc1c(c(nc(n1)N)SCC(=O)O)Cl 9D-099 c1cc(c(cc1Cl)Cl)NC(=O)C/C=N/O 9D-100 CO/N=C\CC(=O)Nc1ccc(cc1Cl)Cl 9D-101 c1ccc(cc1)N/C=C/C(=O)Nc2ccc(cc2Cl)Cl 9D-102 COc1ccc(cc1)C(=O)C/C=N/OCc2ccc(cc2Cl)Cl 9D-105 Cc1ccc(cc1)C(=O)C/C=N/OCc2ccc(cc2Cl)Cl 9D-106 c1ccc(cc1)/C=C(/C#N)\C(=O)N/C=N/OCc2ccc(cc2Cl)Cl 9D-107 c1ccc(cc1)/C=C(/C#N)\C(=O)N/C=N/OCc2c(cccc2Cl)Cl 9D-109 c1ccc(cc1)/C=C(/C#N)\C(=O)N/C=N/OCc2ccc(c(c2)Cl)Cl 9D-110 COc1ccc(cc1)/N=C/c2c(nc3n2ccs3)Cl 9D-111 c1cc(c(c(c1)Cl)CO/N=C/CC(=O)c2ccc(cc2)Br)Cl 9D-112 c1cc(c(c(c1)Cl)CO/N=C/CC(=O)c2ccc(cc2)Cl)Cl 9D-113 c1cc(ccc1C(=O)C/C=N/OCc2ccc(c(c2)Cl)Cl)Cl 9D-114 c1cc(ccc1C(=O)C/C=N/OCc2ccc(c(c2)Cl)Cl)Br 9D-115 c1ccc(cc1)C(=O)C/C=N/OCc2c(cccc2Cl)Cl 9D-116 Cc1c(c(ns1)S(=O)(=O)/C(=N\Nc2ccc(cc2)Cl)/C#N)C#N 9D-118 c1ccc(cc1)Nc2ncc(s2)C(=O)CC(=O)Nc3ccccc3 9D-119 c1ccc(cc1)C\2=C(C(=O)O/C2=C/c3ccc(c(c3)Cl)Cl)C#N 9D-120 c1ccc(cc1)C\2=C(C(=O)O/C2=C\c3ccc(cc3)Cl)C#N 9D-121 c1ccc(cc1)/C=C\2/C(=C(C(=O)O2)C#N)c3ccccc3 9D-122 CC(=O)c1ccc(cc1)n2ccc(=O)cc2 9D-124 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)N)Cl 9E-001 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)N)F 9E-002 CN(C)/C=N/C(=O)c1cc(c[nH]1)C(=O)c2ccccc2Cl 9E-003 CN(C)/C=N/C(=O)c1cc(c[nH]1)C(=O)c2ccccc2F 9E-005 c1ccc(cc1)NC(=S)N/C=N\OCc2ccc(cc2Cl)Cl 9E-006 c1ccc(cc1)C(=O)c2cc([nH]c2)C(=O)N 9E-009 c1ccc(cc1)NC(=S)N/C=N\OCc2c(cccc2Cl)Cl 9E-010 CN(C)/C=N/C(=O)c1cc(c[nH]1)C(=O)c2ccccc2 9E-011 CNC(=S)N/C=N\OCc1ccc(cc1Cl)Cl 9E-013 CNC(=S)N/C=N\OCc1c(cccc1Cl)Cl 9E-014 CO/N=C\NC(=S)Nc1ccccc1 9E-015 c1ccc(cc1)N2CCN(CC2)C(=O)N 9E-016 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)N)Cl 9E-017 CN(C)/C=N/C(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2)Cl 9E-018 CN(C)/C=N/C(=S)N 9E-019 CO/C(=C(\C#N)/N=C/c1ccc(cc1)Cl)/N 9E-022 CO/C(=C(\C#N)/N=C/c1ccc(cc1)C#N)/N 9E-023 CN(C)/C=C(\C#N)/C(=O)Nc1ccccc1 9E-024 CO/N=C\NC(=O)c1cc(c[nH]1)C(=O)c2ccccc2 9E-025 CN(C)/C=N/C(=O)N1CCN(CC1)c2ccccc2 9E-026 CC(C)(C)NC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 9E-027 CN(C)CCCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 9E-028 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)NCCO 9E-029 C=CCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 9E-030 CC(C)NC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 9E-031 CC(C)c1ccc(cc1)n2cc3ccsc3c2 9E-032 C#CCNC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 9E-033 Cc1cc(n2c(n1)c(c(n2)CC#N)C#N)C 9E-034 Cc1cc(n2c(n1)c(c(n2)/C(=C/c3ccc(cc3)Cl)/C#N)C#N)C 9E-035 CO/N=C\NC(=O)N1CCN(CC1)c2ccccc2 9E-036 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)NC3CC3 9E-040 CN(C)NC(=O)c1cc(c[nH]1)C(=O)c2ccc(cc2Cl)Cl 9E-041 CO/N=C\NC(=O)c1cc(c[nH]1)C(=O)c2ccccc2F 9E-042 C/C(=N\O)/c1cccc(c1)Oc2c(cc(cn2)C(F)(F)F)Cl 9E-043 CSc1cccc(c1)n2cc3ccsc3c2 9E-044 c1ccc(c(c1)C(=O)c2cc([nH]c2)C(=O)N/C=N\O)F 9E-045 Cc1cc(n2c(n1)c(c(n2)/C(=C/N(C)C)/C#N)C#N)C 9E-046 Cc1cc(n2c(n1)c(c(n2)/C(=C/c3ccc(cc3Cl)Cl)/C#N)C#N)C 9E-047 CO/N=C\NC(=O)c1cc(c[nH]1)C(=O)c2ccccc2Cl 9E-048 c1ccc(cc1)N2CCN(CC2)c3cnc4ccccc4n3 9E-050 c1cc(c(cc1Cl)Cl)C(=O)c2cc([nH]c2)C(=O)NN 9E-051 CN(C)/C=N/c1nc(cs1)c2ccc(cc2)Cl 9E-100 c1cc(ccc1C(=O)Cn2cc(ccc2=O)C(=O)O)Cl 9E-302S c1ccc(cc1)c2cnn(c2N)c3ccccc3 9E-303S c1ccc(cc1)c2cnn(c2N)c3cccc(c3)[N+](=O)[O-] 9E-305S c1ccc(cc1)c2cnn(c2N)c3cccc(c3)Cl 9E-306S c1ccc(cc1)n2c(c(cn2)c3ccc(cc3)Cl)N 9E-307S c1cc(cc(c1)[N+](=O)[O-])n2c(c(cn2)c3ccc(cc3)Cl)N 9E-308S c1cc(ccc1Cn2cc(cc(c2=O)C(=O)N)Cl)Cl 9E-309S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)N 9E-310S COC(=O)c1ccccc1NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)Cl)Cl 9E-312S COc1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)Cl)Cl 9E-313S COC(=O)c1ccccc1NC(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)Cl)Cl 9E-314S c1cc(ccc1Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F)Cl 9E-315S c1cc(c(cc1Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F)Cl)Cl 9E-316S c1cc(c(c(c1)Cl)Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F)Cl 9E-317S COc1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)Cl)Cl 9E-318S c1cc(ccc1Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F)C(F)(F)F 9E-319S COC(=O)c1cc(cn(c1=O)Cc2cccc(c2)Cl)Cl 9E-320S c1cc(cc(c1)Cl)n2c(c(cn2)c3ccc(cc3)Cl)N 9E-321S c1ccc(cc1)n2c(c(cn2)c3cccc(c3)Cl)N 9E-322S c1cc(cc(c1)Cl)c2cnn(c2N)c3cccc(c3)[N+](=O)[O-] 9E-323S c1cc(cc(c1)Cl)c2cnn(c2N)c3cccc(c3)Cl 9E-324S c1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)Cl)Cl 9E-325S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3)Cl 9E-326S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)Nc3ccc(cc3F)F 9E-327S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)Cl)C(=O)Nc3cc(cc(c3)Cl)Cl 9E-328S CC(C)(C)c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 9E-329S COc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 9E-330S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)NCCCl 9E-332S c1cc(c(c(c1)Cl)Cl)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 9E-333S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)Nc3cc(ccc3Cl)Cl 9E-334S Cc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 9E-335S Cc1ccc(cc1C)NC(=O)c2cccn(c2=O)Cc3ccc(cc3)C(F)(F)F 9E-336S c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)C(=O)N 9E-337S CC(C)(C)c1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)Cl)Cl 9E-338S c1ccc(cc1)n2c(c(cn2)c3cccc(c3)C(F)(F)F)N 9E-339S c1cc(cc(c1)C(F)(F)F)c2cnn(c2N)c3cccc(c3)[N+](=O)[O-] 9E-340S c1cc(cc(c1)C(F)(F)F)c2cnn(c2N)c3cccc(c3)Cl 9E-341S COC(=O)c1ccc(cc1)NC(=O)c2cc(c(=O)n(c2)Cc3cccc(c3)Cl)Cl 9E-342S COC(=O)c1cccn(c1=O)Cc2ccc(cc2Cl)Cl 9E-343S c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)C(=O)O 9E-344S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)C(=O)O)Cl 9E-345S c1ccc(c(c1)c2cnn(c2N)c3cccc(c3)[N+](=O)[O-])Cl 9E-346S c1ccc(c(c1)c2cnn(c2N)c3cccc(c3)Cl)Cl 9E-347S c1ccc(cc1)c2cnn(c2N)c3cccc(c3)C(F)(F)F 9E-349S c1cc(cc(c1)n2c(c(cn2)c3ccc(cc3)Cl)N)C(F)(F)F 9E-350S c1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3cccc(c3)C(F)(F)F)Cl 9E-351S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl 9E-352S CN(C)CCNC(=O)c1cc(cn(c1=O)Cc2cccc(c2)C(F)(F)F)Cl 9E-353S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)C(=O)N)Cl 9E-354S CNC(=O)c1cccn(c1=O)Cc2ccc(cc2Cl)Cl 9E-356S c1cc(cc(c1)C(F)(F)F)Cn2cc(cc(c2=O)C(=O)Nc3cccc(c3)C(F)(F)F)Cl 9E-357S CCNC(=O)c1cccn(c1=O)Cc2ccc(cc2Cl)Cl 9E-358S c1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 9E-359S c1cc(c(=O)n(c1)Cc2ccc(cc2Cl)Cl)C(=O)Nc3ccc(cc3)Cl 9E-360S COc1ccc(cc1)NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 9E-361S COC(=O)c1ccccc1NC(=O)c2cccn(c2=O)Cc3ccc(cc3Cl)Cl 9E-362S c1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3cccc(c3)Cl)Cl 9E-364S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)C(=O)Nc3ccc(cc3)C(F)(F)F)Cl 9E-365S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)C(=O)Nc3cccc(c3)C(F)(F)F)Cl 9E-366S COC(=O)c1cc(cn(c1=O)Cc2ccc(cc2)C(F)(F)F)Cl 9E-367S c1cc(ccc1Cn2cc(cc(c2=O)C(=O)O)Cl)C(F)(F)F 9E-368S Cc1ccc(cc1C)NC(=O)c2cc(cn(c2=O)Cc3cccc(c3)Cl)Cl 9E-369S c1cc(cc(c1)C(F)(F)F)Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F 9E-370S c1cc(cc(c1)Cl)Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F 9E-371S c1cc(ccc1Cn2c(ccc(c2=O)C#N)C(F)(F)F)Cl 9E-372S c1cc(c(cc1Cn2c(ccc(c2=O)C#N)C(F)(F)F)Cl)Cl 9E-373S c1cc(cc(c1)C(F)(F)F)Cn2c(ccc(c2=O)C#N)C(F)(F)F 9E-374S c1cc(c(cc1Cn2c(ccc(c2=O)C#N)C(F)(F)F)F)F 9E-378S c1cc(c(cc1Cn2c(ccc(c2=O)C(=O)N)C(F)(F)F)F)F 9E-379S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)C(=O)Nc3ccc(cc3)Cl)Cl 9E-380S Cc1ccccc1c2cnn(c2N)c3ccccc3 9E-381S Cc1ccccc1c2cnn(c2N)c3cccc(c3)[N+](=O)[O-] 9E-382S Cc1ccccc1c2cnn(c2N)c3cccc(c3)Cl 9E-383S c1ccc2c(c1)ncc(n2)Nc3ccc(cc3)C(=O)O 9E-385S CNC(=O)c1cc(cn(c1=O)Cc2ccc(cc2)C(F)(F)F)Cl 9E-386S COC(=O)c1cc(cn(c1=O)Cc2ccc(cc2Cl)Cl)Cl 9E-387S c1cc(cc(c1)Cl)Cn2cc(cc(c2=O)C(=O)Nc3ccc(cc3Cl)Cl)Cl 9E-388S c1cc(c(cc1Cl)Cl)Cn2cc(cc(c2=O)C(=O)O)Cl 9E-389S CN(C)C(=O)c1cc(cn(c1=O)Cc2ccc(cc2)C(F)(F)F)Cl 9E-390S c1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)C(F)(F)F)Cl 9E-391S COc1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)C(F)(F)F)Cl 9E-392S CC(C)(C)c1ccc(cc1)NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)C(F)(F)F)Cl 9E-393S c1cc(ccc1Cn2cc(cc(c2=O)C(=O)Nc3ccc(cc3F)F)Cl)C(F)(F)F 9E-394S c1ccc(c(c1)CSc2cnc3ccccc3n2)Cl 9E-395S c1ccc2c(c1)ncc(n2)SCc3ccc(cc3)Cl 9E-397S c1ccc(cc1)CS(=O)(=O)c2cnc3ccccc3n2 9E-398S Cc1ccccc1CSc2cnc3ccccc3n2 9E-401S c1ccc2c(c1)ncc(n2)SCc3cccc(c3)C(F)(F)F 9E-402S Cc1ccccc1CS(=O)(=O)c2cnc3ccccc3n2 9E-403S c1ccc2c(c1)ncc(n2)S(=O)(=O)Cc3cccc(c3)C(F)(F)F 9E-404S c1cc(c(c(c1)Cl)Cl)NC(=O)c2cc(cn(c2=O)Cc3ccc(cc3)C(F)(F)F)Cl 9E-405S CN(c1ccccc1)C(=O)c2cc(cn(c2=O)Cc3ccc(cc3)C(F)(F)F)Cl 9E-406S c1ccc2c(c1)nc(c3n2cnn3)Cl 9E-902 c1ccc2c(c1)nc(c3n2c(nn3)C(F)(F)F)O 9E-903 c1ccc2c(c1)c3nnc(n3c(n2)N4CCOCC4)c5ccc(cc5Cl)Cl 9E-904 c1ccc2c(c1)c3nnc(n3c(n2)N4CCCCC4)c5ccc(cc5Cl)Cl 9E-905 c1ccc2c(c1)c3nnc(n3c(n2)N4CCCCC4)c5ccccc5F 9E-906 c1ccc2c(c1)c3nnc(n3c(n2)N4CCOCC4)c5ccccc5F 9E-907 c1ccc2c(c1)c3nnc(n3c(n2)N4CCOCC4)c5ccc(c(c5)Cl)Cl 9E-908 c1ccc2c(c1)c3nnc(n3c(n2)N4CCCCC4)c5ccc(c(c5)Cl)Cl 9E-909 COc1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccc(c(c5)Cl)Cl 9E-911 c1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccc(c(c5)Cl)Cl 9E-912 c1ccc(cc1)Nc2nc3ccccc3c4n2c(nn4)c5ccccc5F 9E-913 COc1nc2ccccc2c3n1c(nn3)c4ccccc4F 9E-915 COc1nc2ccccc2c3n1c(nn3)c4ccc(c(c4)Cl)Cl 9E-916 c1cc(c(cc1Cl)Cl)NC(=O)CC(=O)Nc2ccc(cc2Cl)Cl 9E-917 Cc1c(c(no1)c2ccccc2Cl)C(=O)Oc3cccc(c3)Oc4c(cc(cn4)C(F)(F)F)Cl 9F-002 c1cc(cc(c1)C(F)(F)F)C(=O)Oc2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl 9F-003 Cn1cc(cc1C=O)C(=O)c2c(cccc2F)F 9F-004 Cc1nc(c(s1)C(=O)/N=C/N(C)C)C(F)(F)F 9F-005 Cc1nc(c(s1)C(=O)NN)C(F)(F)F 9F-006 Cc1nc(c(s1)c2nc[nH]n2)C(F)(F)F 9F-007 CCOC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)OCC 9F-009 CN(C)/C=C/c1c(cc(cn1)C(F)(F)F)Cl 9F-011 Cn1cc(cc1C=O)C(=O)c2cccc(c2)Cl 9F-013 Cc1nc(c(s1)C(=O)NNC(=N)COc2ccc(cc2Cl)Cl)C(F)(F)F 9F-014 Cc1nc(c(s1)C(=O)N/C=N/OCc2ccc(cc2Cl)Cl)C(F)(F)F 9F-015 c1cc(ccc1N/C=C/c2c(cc(cn2)C(F)(F)F)Cl)Cl 9F-017 c1cc(ccc1[N+](=O)[O-])Oc2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F 9F-018 COc1ccc(cc1)Sc2c3ccccc3c(nn2)Cc4ccccc4 9F-019 c1ccc(cc1)Cc2c3ccccc3c(nn2)Oc4cccc(c4)Cl 9F-021 CCOC(=O)/C=C(/C(F)(F)F)\N 9F-023 Cn1cc(cc1/C=C(\C#N)/c2nnc(o2)N(C)C)C(=O)c3cccc(c3)Cl 9F-027 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)NNc4c(cc(cn4)C(F)(F)F)Cl 9F-028 CN1C(=O)C(=CNNc2c(cc(cn2)C(F)(F)F)Cl)C(=O)N(C1=O)C 9F-029 Cn1cc(cc1/C=C(\C#N)/C(=O)c2ccccc2)C(=O)c3c(cccc3F)F 9F-030 Cn1cc(cc1/C=N\O)C(=O)c2cccc(c2)Cl 9F-031 Cn1cc(cc1C#N)C(=O)c2cccc(c2)Cl 9F-032 CN(C)c1nc(cc(=O)o1)C(F)(F)F 9F-033 CC(=O)c1ccc(cc1)Oc2ccc(cn2)C(F)(F)F 9F-039 CN(C)/C=C(\C(=O)OC)/N=C/c1ccc(cc1)OC 9F-040 Cc1cc(nc(n1)O/N=C(/C)\c2ccccc2)C 9F-041 c1cc(c(cc1Cl)Cl)CO/N=C\Cc2c(cc(cn2)C(F)(F)F)Cl 9F-042 C/C(=N\Oc1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)/c3ccc(cc3)OC 9F-043 C/C(=N\Oc1c(cc(cn1)C(F)(F)F)Cl)/c2ccc(cc2)Cl 9F-044 C/C(=N\Oc1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)/c3ccccc3 9F-045 Cc1cc(nc(n1)O/N=C(/C)\c2ccc(cc2Cl)Cl)C 9F-046 Cc1c(c(ns1)SCc2c(cc(cn2)C(F)(F)F)Cl)C#N 9F-047 C/C(=N\Oc1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F)/c3ccc(cc3Cl)Cl 9F-049 c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl)Cl 9F-050 C/C(=N\Oc1c(cc(cn1)C(F)(F)F)Cl)/c2ccccn2 9F-051 C/C(=N\O)/c1ccc(cc1Cl)Oc2ccc(cc2)Cl 9F-052 Cc1nc(c(s1)c2ncn(n2)c3ccccc3)C(F)(F)F 9F-053 C/C(=N\Oc1c(cc(cn1)C(F)(F)F)Cl)/c2ccc(cc2Cl)Oc3ccc(cc3)Cl 9F-054 CN(C)/C=C(\C(=O)OC)/N=C/c1ccccc1 9F-056 COc1ccc(cc1)/C=C(/C#N)\c2nc(cs2)c3ccc(o3)c4ccc(cc4Cl)Cl 9F-058 Cn1/c(=C\[N+](=O)[O-])/s/c(=C\c2c(cc(cn2)C(F)(F)F)Cl)/c1=O 9F-059 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/c2nc(cs2)c3ccc(o3)c4ccc(cc4Cl)Cl 9F-060 c1cc(ccc1NC(=O)/C(=C/c2c(cc(cn2)C(F)(F)F)Cl)/C#N)Cl 9F-061 CC(/C(=N/O)/C)Oc1ccc(cc1)Cl 9F-063 c1cc(cc(c1)C(F)(F)F)/C=C(\C#N)/c2nc(cs2)c3ccc(o3)c4ccc(cc4Cl)Cl 9F-065 CO/N=C\Cc1c(cc(cn1)C(F)(F)F)Cl 9F-066 c1cc(ccc1N)Oc2ccc(cn2)C(F)(F)F 9F-067 c1c(cnc(c1Cl)Br)C(F)(F)F 9F-069 C/C(=N\O)/c1ccc(cc1)Oc2ccc(cn2)C(F)(F)F 9F-071 Cn1c(c(c(n1)C(F)(F)F)C(=O)O)Oc2cccc(c2)C(F)(F)F 9F-301S c1cc(cc(c1)Cl)n2c(=O)c(c[nH]2)c3ccc(c(c3)Cl)Cl 9F-302S c1cc(c(cc1c2c[nH]n(c2=O)c3ccc(c(c3)Cl)Cl)Cl)Cl 9F-303S COn1c2cccnc2nc1c3ccc(cc3Cl)Cl 9F-306S c1cc2c(nc1)nc(n2OCc3ccc(cc3)Cl)c4ccc(cc4Cl)Cl 9F-307S c1cc(cc(c1)Cl)COn2c3cccnc3nc2c4ccc(cc4Cl)Cl 9F-308S c1ccc(c(c1)COn2c3cccnc3nc2c4ccc(cc4Cl)Cl)Cl 9F-309S c1cc(cc(c1)Cl)C(=N)NCc2ccc(cc2)Cl 9F-310S c1cc(cc(c1)C(F)(F)F)COn2c3cccnc3nc2c4ccc(cc4Cl)Cl 9F-311S Cc1cc(nc(n1)c2ccccn2)O 9F-313S c1cc2c(nc1)nc(n2OCc3ccc(cc3)Br)c4ccc(cc4Cl)Cl 9F-314S Cc1ccc(cc1)COn2c3cccnc3nc2c4ccc(cc4Cl)Cl 9F-315S c1ccc(cc1)COn2c3cccnc3nc2c4ccc(cc4Cl)Cl 9F-316S CC1=CC(SC(=N1)N)(C)C 9F-318S c1cc(cc(c1)Cl)c2cn([nH]c2=O)c3ccc(c(c3)Cl)Cl 9F-319S CC1=CC(SC(=N1)NC)(C)C 9F-321S CCOC(=O)COn1c2cc(ccc2nc1c3ccccc3)Cl 9F-323S c1ccc(cc1)c2nc3ccc(cc3n2OCC(=O)O)Cl 9F-324S c1ccc(cc1)COn2c3cc(ccc3nc2c4ccccc4)Cl 9F-326S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccccc4Cl)Cl 9F-327S c1ccc(cc1)c2nc3ccc(cc3n2OCc4cccc(c4)Cl)Cl 9F-328S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4)Cl)Cl 9F-329S c1ccc(cc1)c2nc3ccc(cc3n2OCc4cccc(c4)C(F)(F)F)Cl 9F-330S CC1=CC(NC(=S)N1)(C)C 9F-334S c1ccc(cc1)c2cnc(c(n2)O)C(=O)N 9F-335S Cc1ccc(cc1)COn2c3cc(ccc3nc2c4ccccc4)Cl 9F-336S c1ccc(cc1)c2nc3ccc(cc3n2OCc4ccc(cc4Cl)Cl)Cl 9F-337S Cc1c(snn1)Sc2ccc(cc2)Br 9F-338S Cc1c(snn1)Sc2ccccc2C(=O)OC 9F-339S Cc1c(snn1)Sc2ccc(c(c2)Cl)Cl 9F-341S Cc1cc(cc(c1)COn2c3cc(ccc3nc2c4ccccc4)Cl)C 9F-342S COn1c2cc(ccc2nc1c3ccccc3)Cl 9F-343S c1ccc(c(c1)c2nc3ccc(cc3n2O)Cl)Cl 9F-345S COn1c2cc(ccc2nc1c3ccccc3Cl)Cl 9F-347S Cc1c(snn1)Sc2ccc(cc2)OC 9F-348S Cc1c(snn1)S(=O)(=O)c2ccc(cc2)Br 9F-350S Cc1c(snn1)S(=O)(=O)c2ccc(c(c2)Cl)Cl 9F-351S Cc1c(snn1)S(=O)(=O)c2ccc(cc2)OC 9F-352S c1cc(ccc1c2nc3ccc(cc3n2O)Cl)Cl 9F-354S Cc1c(snn1)Sc2ccc(cc2)F 9F-356S Cc1c(snn1)Sc2ccc(cc2Cl)Cl 9F-357S Cc1c(snn1)S(=O)(=O)c2ccc(cc2)F 9F-358S Cc1c(snn1)Sc2ccc(cc2)[N+](=O)[O-] 9F-360S c1cc(ccc1COn2c3cc(ccc3nc2c4ccc(cc4)Cl)Cl)Cl 9F-361S c1cc(cc(c1)Cl)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)Cl 9F-362S c1ccc(c(c1)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)Cl)Cl 9F-363S CCOC(=O)COn1c2cc(ccc2nc1c3ccc(cc3)Cl)Cl 9F-364S CCOC(=O)C(C)On1c2cc(ccc2nc1c3ccc(cc3)Cl)Cl 9F-365S COn1c2cc(ccc2nc1c3ccc(cc3)Cl)Cl 9F-366S c1cc(ccc1c2nc3ccc(cc3n2OCC(=O)O)Cl)Cl 9F-367S c1cc(cc(c1)C(F)(F)F)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)Cl 9F-368S COc1ccc(cc1)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)Cl 9F-369S c1cc(ccc1c2nc3ccc(cc3n2OCc4ccc(cc4Cl)Cl)Cl)Cl 9F-370S Cc1ccc(cc1)COn2c3cc(ccc3nc2c4ccc(cc4)Cl)Cl 9F-371S CN(C)C(=O)On1c2cc(ccc2nc1c3ccc(cc3)Cl)Cl 9F-372S Cc1ccc(cc1)Sc2c(nns2)C 9F-374S COc1ccc(cc1)c2nc3ccc(cc3n2O)Cl 9F-376S CCOC(=O)COn1c2cc(ccc2nc1c3ccc(cc3)OC)Cl 9F-377S COc1ccc(cc1)c2nc3ccc(cc3n2OCC(=O)O)Cl 9F-378S COc1ccc(cc1)c2nc3ccc(cc3n2OC)Cl 9F-379S Cc1ccc(cc1)S(=O)(=O)c2c(nns2)C 9F-380S c1ccc(cc1)c2cc\3c(n2c4ccccc4)CCC/C3=N/OCc5ccc(cc5)Cl 9F-900 c1ccc(cc1)c2cc\3c(n2c4ccccc4Cl)CCC/C3=N/OCc5ccc(cc5)Cl 9F-901 c1ccc(cc1)c2cc\3c(n2c4cccc(c4)Cl)CCC/C3=N/OCc5ccc(cc5)Cl 9F-902 c1ccc(cc1)c2cc\3c(n2c4ccc(cc4)Cl)CCC/C3=N/OCc5ccc(cc5)Cl 9F-903 CN(C)c1nc2c(c(nn2c3ccccc3)N)c(=O)o1 9F-904 c1cc(ccc1CON/C=N/C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 9F-905 c1ccc(cc1)c2cc3c(n2c4ccccc4)CCCC3=O 9F-906 c1ccc(cc1)c2cc3c(n2c4ccccc4Cl)CCCC3=O 9F-907 CCOC(=O)NC(=O)/C(=C/N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)/C#N 9F-908 CCOC(=O)CN1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 9F-910 c1cc(ccc1C(=O)CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 9F-911 c1ccc(cc1)C2=N/C(=C/Nc3nccs3)/C(=O)O2 9F-913 c1c(cnc(c1Cl)N2CCN(CC2)CC(=O)NN)C(F)(F)F 9F-914 c1cc(ccc1NC(=O)NNC(=O)CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 9F-915 CN(CCO)C(=O)Cc1ccccc1 9F-916 c1c(cnc(c1Cl)N2CCc3c(cnc(n3)N)C2)C(F)(F)F 9F-918 c1ccc(cc1)NC(=S)NNC(=O)CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9F-919 c1c(cnc(c1Cl)N2CCC(=NO)CC2)C(F)(F)F 9F-920 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)CCl)C(F)(F)F 9F-922 c1ccc(cc1)n2c(nnc2S)CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9F-923 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)CN3CCOCC3)C(F)(F)F 9F-924 c1cc(ccc1SCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 9F-925 c1ccc(cc1)n2c(nnc2SCc3ccc(cc3Cl)Cl)CN4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 9F-926 COc1ccc(cc1)N2CCN(CC2)CC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9F-927 CC(=O)c1ccc(cc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9F-928 c1cc(ccc1C#N)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9F-930 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)CN3CCCCC3)C(F)(F)F 9F-931 c1c(cc(c(c1[N+](=O)[O-])N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-])C(F)(F)F 9F-932 c1c(cnc(c1Cl)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 9F-933 c1ccc2c(c1)C(=O)N(C2=O)Oc3c(cc(cn3)C(F)(F)F)Cl 9F-934 c1cc(c(nc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 9F-935 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9F-936 c1cc(nc(c1)Cl)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9F-937 c1cc(ccc1C(=O)N)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9F-938 c1c(cnc(c1Cl)N2CCN(CC2)CC(=O)O)C(F)(F)F 9F-939 CN(C)/C=N/C(=O)c1ccc(cc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9F-940 c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)CN4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 9F-941 CN(C)/C=N/NC(=O)CN1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 9F-942 c1cc(ccc1CO/N=C\NNC(=O)CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl 9F-943 c1ccc(cc1)n2c(ncn2)c3ccc(cc3)N4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 9F-944 c1cc(ccc1CO/N=C\NC(=O)c2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 9F-945 c1c(cnc(c1Cl)N2CCN(CC2)CC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 9F-946 CCOC(=O)CC(=N)NNC(=O)CN1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl 9F-947 c1c(cnc(c1Cl)N2CCN(CC2)CC(=O)NNC(=N)CC#N)C(F)(F)F 9F-948 c1ccc(cc1)c2cc3c(n2c4ccc(cc4)Cl)CCCC3=O 9F-949 c1ccc(cc1)c2cc3c(n2c4cccc(c4)Cl)CCCC3=O 9F-950 c1c(cnc(c1Cl)N2CCN(CC2)CC#N)C(F)(F)F 9F-951 c1ccc(cc1)c2ncc3c(n2)CCN(C3)c4c(cc(cn4)C(F)(F)F)Cl 9F-953 c1c(cnc(c1Cl)N2CCc3c(c[nH]n3)C2)C(F)(F)F 9F-954 CN(C)/C=C(\C#N)/C(=O)N/C=N/OCc1ccc(cc1)[N+](=O)[O-] 9F-955 COc1ccc(cc1)N/C=C(\C#N)/C(=O)N/C=N/OCc2ccc(cc2)[N+](=O)[O-] 9F-956 CCOC(=O)NC(=O)/C(=C/N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)/C(=O)C 9F-957 c1c(cnc(c1Cl)N2CCN(CC2)C(=N)CC#N)C(F)(F)F 9F-959 C/C(=N\O)/c1ccc(cc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9F-961 c1ccc(cc1)NC(=O)N(/C=N/OCc2c(cccc2Cl)Cl)OCc3c(cccc3Cl)Cl 9G-002 c1cc(c(c(c1)Cl)CO/N=C/N(C(=O)Nc2ccc(cc2)Cl)OCc3c(cccc3Cl)Cl)Cl 9G-003 CC(c1ccc(c(n1)O)C#N)n2cncn2 9G-005 Cc1nnc(n1N)NN.Cl 9G-008 c1cc(c(c(c1)Cl)CON/C(=N\C(=O)Nc2ccc(cc2)Cl)/Cn3cncn3)Cl 9G-009 c1cc(c(c(c1)Cl)CO/N=C/NNc2c(cc(cn2)C(F)(F)F)Cl)Cl 9G-011 c1cscc1C(c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N 9G-013 c1c(cn2c(c1Cl)nnn2)C(F)(F)F 9G-015 Cc1cc(n(n1)c2n[nH+]c(n2N)C)C.[Cl-] 9G-016 c1cc(ccc1C(C#N)c2ccc3c(cc(nc3n2)C(F)(F)F)C(F)(F)F)Cl 9G-017 c1cc(ccc1NC(=O)N/C=C/c2c(cc(cn2)C(F)(F)F)Cl)Cl 9G-019 c1ccc(cc1)C(=O)CN/C=C\C(=O)c2ccccc2 9G-020 CN(/C=N/C(=S)/N=C/N(C)C)C 9G-021 CN(C)/C=N/C(=S)N/C=N\OC 9G-023 Cn1ccc2c1c(c3ccccc3c2c4ccccc4)C#N 9G-024 Cc1cc(no1)/N=C/N(C)C 9G-025 Cc1cc(no1)N/C=N/OCc2c(cccc2Cl)Cl 9G-026 CCOC(=O)/C=C(\C(F)(F)F)/NC(=O)c1ccc(cc1Cl)Cl 9G-031 CCOC(=O)COn1c2ccccc2nc1c3ccccc3 9G-032 c1ccc(cc1)/C=C(\C#N)/c2[nH]c(nn2)Cn3cncn3 9G-033 c1ccc(cc1)C(c2c(cc(cn2)C(F)(F)F)Cl)C(=S)N 9G-034 c1ccc(cc1)C(c2c(cc(cn2)C(F)(F)F)Cl)c3nc(cs3)c4ccc(cc4)Cl 9G-035 c1ccc(cc1)C2c3ccccc3C(=O)NC2=O 9G-036 CN(C)/C=N/C(=S)C(c1ccccc1)c2c(cc(cn2)C(F)(F)F)Cl 9G-037 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(/C=N/OCc2c(cccc2Cl)Cl)OCc3c(cccc3Cl)Cl 9G-038 Cc1cc(c(c(c1OC(=O)C)C)C)OC(=O)C 9G-039 CO/N=C\NC(=S)N/C=N\OC 9G-040 CN(C)/C=N/C(=S)N/C=N\OCc1ccc(cc1)Cl 9G-041 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)Sc3ccc(cc3)Br)F 9G-301S c1cc(ccc1C(=O)Nc2ccc(cc2)Sc3ccc(cc3)Br)F 9G-302S CC(=O)Nc1ccc(cc1)S(=O)(=O)c2ccc(cc2)F 9G-303S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)F 9G-304S Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)NC(=O)C(Cl)Cl 9G-305S Cc1cc(ccc1OC(C(=O)N2CCOCC2)(F)F)Cl 9G-307S c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)Sc3ccc(cc3)Br 9G-309S CC(=O)Nc1ccc(cc1)Sc2ccc(cc2)Br 9G-314S c1cc(ccc1C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)Br)F 9G-315S c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)Br)F 9G-316S c1ccc(cc1)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] 9G-319S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ccc(cn4)[N+](=O)[O-] 9G-320S CC(C)C(=O)Nc1ccc(cc1)Sc2ccc(cc2)Br 9G-322S CC(C)(C)C(=O)Nc1ccc(cc1)Sc2ccc(cc2)Br 9G-323S c1cc(cc(c1)Sc2ccc(cc2)[N+](=O)[O-])C(F)(F)F 9G-324S c1cc(cc(c1)Sc2ccc(cc2)N)C(F)(F)F 9G-325S Cc1cc(ccc1OC(C(=O)Nc2ccc(cc2F)F)(F)F)Cl 9G-326S c1ccc(cc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F 9G-327S c1cc(ccc1N2CCN(CC2)c3ccc(cn3)C(F)(F)F)F 9G-328S c1cc(cc(c1)Cl)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] 9G-329S c1cc(ccc1N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])F 9G-330S c1cc(ccc1NC(=O)C(Cl)(Cl)Cl)Sc2ccc(cc2)Br 9G-331S c1cc(ccc1NC(=O)c2cc(cc(c2)Cl)Cl)Sc3ccc(cc3)Br 9G-332S c1ccc(cc1)N2CCN(CC2)c3c(cccn3)[N+](=O)[O-] 9G-333S c1ccc(c(c1)N2CCN(CC2)c3c(cccn3)[N+](=O)[O-])F 9G-334S c1cc(cc(c1)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])C(F)(F)F 9G-335S c1ccc(cc1)CN2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] 9G-336S c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)S(=O)(=O)c3ccc(cc3)Br 9G-337S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)Sc3cccc(c3)C(F)(F)F 9G-338S CN(C)c1ccc(cc1)Sc2ccc(cc2)Br 9G-339S c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4ccc(cc4)F 9G-340S c1ccc(cc1)CN2CCN(CC2)c3cnc4ccccc4n3 9G-342S c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4cccc(c4)C(F)(F)F 9G-343S c1cc(ccc1NC(=O)c2cc(cc(c2)Cl)Cl)S(=O)(=O)c3ccc(cc3)Br 9G-345S c1cnc(nc1)N2CCN(CC2)c3ccc(cc3)F 9G-346S c1ccc(cc1)N2CCN(CC2)c3ncccn3 9G-347S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ncccn4 9G-348S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)Br 9G-349S c1cc(cc(c1)Sc2ccc(cc2)NC(=O)c3ccc(cc3)F)C(F)(F)F 9G-350S CC(C)C(C(=O)NO)N 9G-351S CC(C)c1c(=O)n(cc(n1)c2ccccc2)O 9G-352S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)Sc3cccc(c3)C(F)(F)F 9G-354S c1cc(c(nc1)N2CCN(CC2)c3ccc(cc3)F)[N+](=O)[O-] 9G-355S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4c(cccn4)[N+](=O)[O-] 9G-356S CC(=O)Nc1ccc(cc1)Sc2cccc(c2)C(F)(F)F 9G-357S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)S(=O)(=O)c3cccc(c3)C(F)(F)F 9G-358S c1cc(cc(c1)S(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)F)C(F)(F)F 9G-359S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F 9G-363S COc1cccc(c1)N2CCN(CC2)c3cnc4ccccc4n3 9G-365S c1cc(cc(c1)Sc2ccc(cc2)NC(=O)C(Cl)(Cl)Cl)C(F)(F)F 9G-366S c1cc(cc(c1)Sc2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl)C(F)(F)F 9G-367S c1cc(ccc1NC(=O)CCl)Sc2ccc(cc2)Br 9G-368S CC(=O)Nc1ccc(cc1)S(=O)(=O)c2cccc(c2)C(F)(F)F 9G-369S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)S(=O)(=O)c3cccc(c3)C(F)(F)F 9G-370S c1ccc(c(c1)Sc2ccc(cc2)[N+](=O)[O-])Cl 9G-371S COc1cccc(c1)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] 9G-372S c1cc(ccc1NC(=O)CCl)Sc2ccc(cc2)F 9G-373S c1cc(ccc1NC(=O)CCl)S(=O)(=O)c2ccc(cc2)Br 9G-374S c1ccc(c(c1)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])F 9G-376S c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4ccccc4F 9G-377S CC(C)C(=O)Nc1ccc(cc1)Sc2ccc(cc2)F 9G-378S CC(C)(C)C(=O)Nc1ccc(cc1)Sc2ccc(cc2)F 9G-379S CC(C)(CCl)C(=O)Nc1ccc(cc1)Sc2ccc(cc2)F 9G-380S c1cc(ccc1NC(=O)CCl)S(=O)(=O)c2ccc(cc2)F 9G-381S CN(C)c1nc(cc(n1)N2CCN(CC2)c3ccc(cc3)F)C(F)(F)F 9G-382S CN(C)c1nc(cc(n1)N2CCN(CC2)C(c3ccccc3)c4ccccc4)C(F)(F)F 9G-383S CN(C)c1nc(cc(n1)N2CCN(CC2)c3ccccc3F)C(F)(F)F 9G-384S CN(C)c1nc(cc(n1)N2CCN(CC2)c3cccc(c3)C(F)(F)F)C(F)(F)F 9G-385S c1ccc(c(c1)Sc2ccc(cc2)N)Cl 9G-386S c1ccc(c(c1)Sc2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl)Cl 9G-388S c1ccc(c(c1)Sc2ccc(cc2)NC(=O)c3c(cccc3F)F)Cl 9G-389S c1ccc(cc1)n2c(nnn2)N3CCN(CC3)c4ccc(cc4)F 9G-390S c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4nnnn4c5ccccc5 9G-391S c1ccc(c(c1)Sc2ccc(cc2)NC(=O)c3ccc(cc3)F)Cl 9G-392S c1ccc(c(c1)S(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl)Cl 9G-393S c1ccc(cc1)CN2CCN(CC2)c3nnnn3c4ccccc4 9G-394S CC(=O)Nc1ccc(cc1)Sc2ccccc2Cl 9G-396S c1ccc(c(c1)S(=O)(=O)c2ccc(cc2)NC(=O)c3c(cccc3F)F)Cl 9G-397S c1ccc(c(c1)S(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)F)Cl 9G-398S c1ccc(c(c1)Sc2ccc(cc2)NC(=O)CCl)Cl 9G-399S c1ccc(c(c1)Sc2ccc(cc2)NC(=O)C(Cl)(Cl)Cl)Cl 9G-400S CN(C)c1nc(cc(n1)N2CCN(CC2)c3ccccc3)C(F)(F)F 9G-401S c1ccc(cc1)n2c(nnn2)N3CCN(CC3)c4ccccc4 9G-402S c1ccc(c(c1)S(=O)(=O)c2ccc(cc2)NC(=O)CCl)Cl 9G-406S Cc1ccc(c(c1)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])C 9G-407S Cc1ccc(c(c1)N2CCN(CC2)c3c(cccn3)[N+](=O)[O-])C 9G-408S c1cc(c(cc1N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl)Cl 9G-409S c1ccc(c(c1)Sc2ccc(cc2)NC(=O)c3cccc(c3)C(F)(F)F)Cl 9G-410S Cc1ccc(c(c1)N2CCN(CC2)c3nnnn3c4ccccc4)C 9G-411S c1ccc(cc1)n2c(nnn2)N3CCN(CC3)c4ccc(c(c4)Cl)Cl 9G-412S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2)Sc3ccccc3Cl 9G-413S c1cnc(nc1)N2CCN(CC2)c3ccc(c(c3)Cl)Cl 9G-414S c1ccc(c(c1)Sc2ccc(cc2)NC(=O)CCCCl)Cl 9G-416S c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4ccccn4 9G-417S Cc1ccc(c(c1)C)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] 9G-418S c1ccnc(c1)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] 9G-419S c1cc(ccc1c2cn(c(=O)cn2)O)C(F)(F)F 9G-420S CCOC(=O)CSc1c(c(nn1C)C(F)(F)F)C#N 9G-421S CCOC(=O)C(C)Sc1c(c(nn1C)C(F)(F)F)C#N 9G-422S Cc1ccc(c(c1)C)N2CCN(CC2)c3c(cccn3)[N+](=O)[O-] 9G-423S Cc1ccc(c(c1)C)N2CCN(CC2)c3nnnn3c4ccccc4 9G-424S c1ccc(c(c1)S(=O)(=O)c2ccc(cc2)NC(=O)C(Cl)(Cl)Cl)Cl 9G-425S c1ccc(c(c1)S(=O)(=O)c2ccc(cc2)NC(=O)c3cccc(c3)C(F)(F)F)Cl 9G-426S Cc1ccc(c(c1)C)N2CCN(CC2)c3cnc4ccccc4n3 9G-427S c1ccc2c(c1)ncc(n2)N3CCN(CC3)c4ccc(c(c4)Cl)Cl 9G-428S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)c3ccc(cc3)F 9G-429S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)c3ccccc3 9G-430S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)c3ccccc3F 9G-431S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)c3cccc(c3)C(F)(F)F 9G-432S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)C 9G-433S c1cc(c(cc1N2CCN(CC2)c3ccc(cn3)C(F)(F)F)Cl)Cl 9G-434S COC(=O)C(c1ccccc1)NS(=O)(=O)c2ccc(cc2)Cl 9G-437S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)c3cccc(c3)OC 9G-438S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)c3ccccn3 9G-439S Cn1c(c(c(n1)C(F)(F)F)C#N)N2CCN(CC2)Cc3ccccc3 9G-440S c1ccc(cc1)c2nnc(n2N)S 9G-441S c1cnccc1c2nnc(n2N)S 9G-443S Cc1c(c(on1)C/C=[N+](\C)/[O-])[N+](=O)[O-] 9G-901 CC1=CCCc2c1cccc2 9G-902 c1ccc2c(c1)C(=O)N(C2=O)OCC(=O)Nc3ccc(cc3)Cl 9G-903 c1c(cnc(c1Cl)NCCNC(=O)CON)C(F)(F)F.Cl 9G-905 C/[N+](=C\CC(=O)c1ccc(cc1)c2ccccc2)/[O-] 9G-906 CN1[C@H]([C@H]2[C@@H](O1)C(=O)N(C2=O)c3ccccc3)CC(=O)c4ccc(cc4)c5ccccc5 9G-907 c1ccc2c(c1)C(=O)N(C2=O)OCC(=O)N3CCOCC3 9G-908 COc1ccccc1NC(=O)CCl 9G-909 c1ccc(c(c1)CON=C2CCN(CC2)c3c4nnc(n4c5cc(ccc5n3)Cl)C(F)(F)F)Cl 9G-910 c1cc(cc(c1)Cl)CON=C2CCN(CC2)c3c4nnc(n4c5cc(ccc5n3)Cl)C(F)(F)F 9G-911 c1ccc(cc1)CON=C2CCN(CC2)c3c4nnc(n4c5cc(ccc5n3)Cl)C(F)(F)F 9G-912 c1cc(ccc1NC(=O)CON)Cl 9G-913 COc1ccccc1NC(=O)CON2C(=O)c3ccccc3C2=O 9G-914 c1cc(ccc1CNC(=O)CCl)Cl 9G-915 c1cc(ccc1CON=C2CCN(CC2)c3c4nnc(n4c5cc(ccc5n3)Cl)C(F)(F)F)Cl 9G-916 c1cc(ccc1C(=O)ON=C2CCN(CC2)c3c4nnc(n4c5cc(ccc5n3)Cl)C(F)(F)F)Cl 9G-917 c1ccc(cc1)C(=O)ON=C2CCN(CC2)c3c4nnc(n4c5cc(ccc5n3)Cl)C(F)(F)F 9G-918 C1COCCN1C(=O)CON.Cl 9G-920 c1cc(ccc1C(=O)NNC(=O)CCl)Cl 9G-921 C/[N+](=C\C1C(=O)CCCC1=O)/[O-] 9G-922 COc1ccccc1NC(=O)CON.Cl 9G-923 c1ccc2c(c1)C(=O)N(C2=O)OCC(=O)NNC(=O)c3ccc(cc3)Cl 9G-924 c1ccc2c(c1)C(=O)N(C2=O)OCC(=O)NCc3ccc(cc3)Cl 9G-926 CN([C@H]1c2cccc(c2OC[C@H]1CO)OC)C(=O)Nc3ccccc3 9G-927 CN([C@H]1c2cccc(c2OC[C@H]1CO)OC)C(=O)Nc3ccc(cc3Cl)Cl 9G-928 CN([C@H]1c2cccc(c2OC[C@H]1CO)OC)C(=O)Nc3cccc(c3)C(F)(F)F 9G-929 Cc1ccc(cc1)S(=O)(=O)N2CC(CC2C(=O)O)O 9G-933 c1ccc(cc1)CCNC(=O)CCl 9G-934 c1cc(ccc1CNC(=O)CON)Cl.Cl 9G-935 c1ccc(cc1)n2c(cc3c2CCCC3=O)c4ccc(cc4)Cl 9G-936 c1c(cnc(c1Cl)NNC(=O)CCl)C(F)(F)F 9G-937 c1ccc(cc1)n2c(cc\3c2CCC/C3=N/OCc4ccc(cc4)Cl)c5ccc(cc5)Cl 9G-939 c1ccc(cc1)c2cc\3c(n2c4ccccc4)CCC/C3=N/OCc5cc(ccc5Cl)Cl 9G-940 c1ccc(cc1)c2cc\3c(n2c4ccccc4)CCC/C3=N/OCc5ccc(c(c5)Cl)Cl 9G-941 c1ccc(cc1)CO/N=C\2/CCCc3c2cc(n3c4ccccc4)c5ccccc5 9G-944 c1ccc(cc1)c2cc\3c(n2c4ccccc4)CCC/C3=N/OCc5ccccc5Cl 9G-945 c1ccc(cc1)c2cc\3c(n2c4ccccc4)CCC/C3=N/OCc5cccc(c5)Cl 9G-946 CN(C1c2cc(ccc2OCC1CO)Br)C(=O)Nc3ccccc3 9G-948 c1ccc(cc1)c2cc\3c(n2c4ccccc4)CCC/C3=N/OCc5ccc(cc5Cl)Cl 9G-949 CN(Cc1cc(ccc1OCC=C)Br)C(=O)Nc2ccc(cc2Cl)Cl 9G-950 CN(C1c2cc(ccc2OCC1CO)Br)C(=O)Nc3cccc(c3)C(F)(F)F 9G-951 c1cc(c(cc1Cl)Cl)C(=O)CC2C(=O)CCCC2=O 9G-952 Cc1ccc(cc1)S(=O)(=O)N2CC(CC2C(=O)OC)O 9G-953 CCOC(=O)C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl 9G-955 CN([C@H]1c2cc(ccc2OC[C@H]1CO)Br)C(=O)Nc3ccc(cc3Cl)Cl 9G-956 c1ccc2c(c1)C(=O)N(C2=O)OCc3ccc(cc3Cl)Cl 9H-002 c1cc(ccc1/C(=N/O)/c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] 9H-004 c1ccc(cc1)C(=O)c2c(cc(cn2)C(F)(F)F)C(C#N)(c3ccccc3)N4CCOCC4 9H-005 CCOc1c(c(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)O)/C=N/OCc3ccc(cc3)C(F)(F)F 9H-006 c1ccc(cc1)S(=O)(=O)C(C2c3ccccc3CCN2C(=O)c4ccc(cc4)F)[N+](=O)[O-] 9H-007 COC(=O)C1CC(=O)N(C1)Nc2c(cc(cn2)C(F)(F)F)Cl 9H-008 c1ccc(cc1)C(=O)c2cc(cnc2C(=O)c3ccccc3)C(F)(F)F 9H-009 c1cc(c(cc1Cl)Cl)C(=O)c2c(cc(cn2)C(F)(F)F)Cl 9H-011 CCOC(=O)C(=O)/C(=C/Nc1ccccc1)/C#N 9H-012 COC(=O)c1cn(c(=O)c2c1cccc2)Nc3c(cc(cn3)C(F)(F)F)Cl 9H-013 c1cc(ccc1c2c3c(cc(cn3)C(F)(F)F)on2)[N+](=O)[O-] 9H-014 c1c(cnc(c1Cl)NN2CC(CC2=O)C(=O)N)C(F)(F)F 9H-015 c1cc(c(cc1Cl)Cl)/C(=N\O)/c2c(cc(cn2)C(F)(F)F)Cl 9H-016 c1ccc(c(c1)N)N/C=C(\C#N)/c2c(=O)[nH]c3ccccc3n2 9H-018 CCOC(=O)C(=O)/C(=C\Nc1ccc(cc1)OC)/C#N 9H-019 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)n2cc(c3ccccc3c2=O)C(=O)OC 9H-020 c1cc(c(cc1Cl)Cl)c2c3c(cc(cn3)C(F)(F)F)no2 9H-021 c1cc(c(cc1Cl)Cl)c2c3c(cc(cn3)C(F)(F)F)on2 9H-022 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NN 9H-024 c1cc(cnc1)/C(=N\O)/c2c(cc(cn2)C(F)(F)F)Cl 9H-025 COC(=O)c1cn(c(=O)c2c1cccc2)Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F 9H-026 c1ccc(cc1)N/C=C(/C#N)\C(=O)CCl 9H-027 c1cc(cnc1)c2c3c(cc(cn3)C(F)(F)F)on2 9H-028 CN(C)/C=C(\C#N)/C(=O)CSc1ccc(cc1)Cl 9H-029 CN(C)/C=C(\C#N)/C(=O)CSc1c(cc(cn1)C(F)(F)F)Cl 9H-031 CN(C)c1nnc2n1cc(cc2Cl)C(F)(F)F 9H-032 CCOC(=O)C(=O)/C(=C/N(C)C)/c1c(cc(cn1)C(F)(F)F)Cl 9H-033 c1ccc(cc1)c2c3cc(cnc3c(nn2)c4ccccc4)C(F)(F)F 9H-036 CCOC1=NN(C(=O)C1/C=N/OCc2ccc(cc2Cl)Cl)c3c(cc(cn3)C(F)(F)F)Cl 9H-038 c1cc(cc(c1)[N+](=O)[O-])C(=O)c2c(cc(cn2)C(F)(F)F)Cl 9H-039 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)n(n2)c4ccccc4 9H-040 c1cc(ccc1CO/N=C/C(=C/c2ccc(cc2)Cl)/C#N)Cl 9H-041 c1cc(ccc1CO/N=C/C(=C/c2ccncc2)/C#N)Cl 9H-042 c1ccc(cc1)/C(=N\Nc2c(cc(cn2)C(F)(F)F)Cl)/c3c(cc(cn3)C(F)(F)F)Cl 9H-043 c1ccnc(c1)c2c3c(cc(cn3)C(F)(F)F)no2 9H-044 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)n(n2)c4c(cc(cn4)C(F)(F)F)Cl 9H-045 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)O 9H-046 COc1ccc(cc1)/C(=N\O)/c2c(cc(cn2)C(F)(F)F)Cl 9H-047 COc1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)on2 9H-048 CN(C)/C=C(/c1c(c(no1)c2ccccc2Cl)C#N)\C(=O)C(F)(F)F 9H-050 CO/N=C/C(=N\Nc1ccc(cc1Cl)Cl)/C#N 9H-051 CCOC(=O)C(=O)/C(=C/Nc1ccc(cc1)C(F)(F)F)/C#N 9H-052 COc1ccc(cc1)NC(=O)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4ccccc4 9H-053 CN(C)S(=O)(=O)c1ccc(cc1)NC(=O)c2c(c3c(s2)cc(cn3)C(F)(F)F)c4ccccc4 9H-054 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)Nc4cccc(c4)C(F)(F)F 9H-055 COC(=O)c1cn(c(=O)c2c1cccc2)c3ccc(cc3)F 9H-056 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)Oc4cccc(c4)C(F)(F)F 9H-057 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c3ccccc3c2=O)C(=O)O 9H-058 c1ccc2c(c1)c(cn(c2=O)c3ccc(cc3)F)C(=O)O 9H-059 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)N4CCOCC4 9H-060 CN(C)/C=C(/c1c(c(no1)c2ccccc2)C#N)\C(=O)C(F)(F)F 9H-062 c1ccc(cc1)c2c3c(cc(cn3)C(F)(F)F)sc2C(=O)N 9H-063 CCOC(=O)C(=O)/C(=C/Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl)/C#N 9H-064 CN(c1c(cc(cn1)C(F)(F)F)Cl)n2cc(c3ccccc3c2=O)C(=O)N 9H-065 CN(C)C(=O)c1cn(c(=O)c2c1cccc2)N(C)c3c(cc(cn3)C(F)(F)F)Cl 9H-066 c1ccc2c(c1)c(cn(c2=O)c3ccc(cc3)F)C(=O)N 9H-068 CN(C)/C=N/C(=O)c1cn(c(=O)c2c1cccc2)c3ccc(cc3)F 9H-069 CN(C)/C=N/C(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)c3ccccc3 9H-071 CN(C)/C=C(/C#N)\C(=O)OC 9H-072 CO/N=C/NC(=O)c1cn(c(=O)c2c1cccc2)c3ccc(cc3)F 9H-073 c1ccc(cc1)/C(=N\N=C(\c2ncc(cc2Cl)C(F)(F)F)/c3ccccc3)/c4ncc(cc4Cl)C(F)(F)F 9H-074 c1ccc2c(c1)c(cn(c2=O)c3ccc(cc3)F)C(=O)N/C=N/O 9H-075 COC(=O)/C(=C\Nc1ccc(cc1Cl)Cl)/C#N 9H-076 c1ccc(c(c1)NC(=O)CS(=O)c2cccc(c2)Cl)Cl 9H-301S c1ccc(c(c1)NC(=O)CS(=O)c2ccc(cc2)F)Cl 9H-302S c1cc(ccc1F)S(=O)CC(=O)N2CCOCC2 9H-303S c1cc(ccc1S(=O)CC(=O)N2CCOCC2)Br 9H-304S c1ccc(c(c1)NC(=O)CS(=O)(=O)c2ccc(cc2)F)Cl 9H-308S COc1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccccc2Cl 9H-309S c1ccc(c(c1)NC(=O)CS(=O)(=O)c2cccc(c2)Cl)Cl 9H-310S c1ccc(c(c1)NC(=O)CS(=O)c2cccc(c2)C(F)(F)F)Cl 9H-311S c1ccc(c(c1)CS(=O)CC(=O)Nc2ccccc2Cl)Cl 9H-312S c1cc(cc(c1)NC(=O)CS(=O)(=O)Cc2ccc(cc2)Cl)C(F)(F)F 9H-313S c1ccc(cc1)S(=O)(=O)c2cnc(nc2c3ccc(cc3)Cl)c4ccccn4 9H-314S c1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2Cl)Cl 9H-315S COc1ccc(cc1)S(=O)(=O)CC(=O)Nc2cccc(c2)C(F)(F)F 9H-316S c1cc(cc(c1)NC(=O)CS(=O)(=O)c2cccc(c2)Cl)C(F)(F)F 9H-317S c1ccc(c(c1)NC(=O)CS(=O)(=O)c2ccc(c(c2)Cl)Cl)Cl 9H-318S c1ccc(c(c1)CS(=O)(=O)CC(=O)Nc2ccccc2Cl)Cl 9H-319S c1ccc(c(c1)NC(=O)CS(=O)(=O)c2cccc(c2)C(F)(F)F)Cl 9H-320S c1ccc(cc1)S(=O)(=O)c2cnc(nc2N)c3ccccn3 9H-321S c1ccc(cc1)c2ncc(c(n2)N)S(=O)(=O)c3ccccc3 9H-322S CN(C)c1ncc(c(n1)N)S(=O)(=O)c2ccccc2 9H-323S CN(C)/C=C(/C(=O)c1ccc(cc1Cl)Cl)\S(=O)(=O)c2ccccc2 9H-324S CN(C)/C=C(/C(=O)c1ccccc1)\S(=O)(=O)c2ccccc2 9H-325S c1ccc(cc1)S(=O)(=O)c2cnc(nc2N)c3cccnc3 9H-326S CCOC(=O)c1c(snn1)Sc2ccc(cc2)Br 9H-327S CN(C)c1ncc(c(n1)c2ccccc2Cl)S(=O)(=O)c3ccccc3 9H-329S c1ccc(cc1)c2ncc(c(n2)c3ccccc3Cl)S(=O)(=O)c4ccccc4 9H-330S c1cc(ccc1F)SCC(=O)Nc2ccc(cc2Cl)Cl 9H-331S c1ccc(c(c1)SCC(=O)Nc2ccc(cc2Cl)Cl)Cl 9H-332S c1cc(cc(c1)Cl)SCC(=O)Nc2ccc(cc2Cl)Cl 9H-333S CN(C)/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)F 9H-334S c1cc(ccc1F)S(=O)CC(=O)Nc2ccc(cc2Cl)Cl 9H-335S c1cc(ccc1F)S(=O)(=O)CC(=O)Nc2ccc(cc2Cl)Cl 9H-336S c1ccc(cc1)S(=O)(=O)c2cnc(nc2c3ccc(c(c3)Cl)Cl)c4ccncc4 9H-337S c1ccc(cc1)S(=O)(=O)c2cnc(nc2c3ccc(c(c3)Cl)Cl)c4cccnc4 9H-338S c1ccc(cc1)S(=O)(=O)c2cnc(nc2c3ccc(c(c3)Cl)Cl)c4ccccn4 9H-339S c1ccc(c(c1)S(=O)(=O)CC(=O)Nc2ccc(cc2Cl)Cl)Cl 9H-340S c1cc(cc(c1)SCC(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F 9H-346S COc1ccc(cc1)SCC(=O)Nc2ccc(cc2Cl)Cl 9H-347S CN(C)c1ncc(c(n1)c2ccc(c(c2)Cl)Cl)S(=O)(=O)c3ccccc3 9H-348S CN(C)c1ncc(c(n1)c2ccccc2)S(=O)(=O)c3ccccc3 9H-349S CN(C)c1ncc(c(n1)c2ccc(cc2Cl)Cl)S(=O)(=O)c3ccccc3 9H-350S CC(C)(C)c1ccc(cc1)CSCC(=O)Nc2ccc(cc2Cl)Cl 9H-351S CNC(=O)c1c(snn1)S(=O)c2ccc(cc2)F 9H-352S CNC(=O)c1c(snn1)S(=O)(=O)c2ccc(cc2)Br 9H-353S c1cc(cc(c1)Cl)S(=O)(=O)CC(=O)Nc2ccc(cc2Cl)Cl 9H-355S c1ccc(c(c1)S(=O)CC(=O)Nc2ccc(cc2Cl)Cl)Cl 9H-356S Cc1ncc(c(n1)c2ccc(cc2Cl)Cl)S(=O)(=O)c3ccccc3 9H-357S Cc1ncc(c(n1)c2ccccc2)S(=O)(=O)c3ccccc3 9H-358S CN(c1ccccc1)C(=O)CSc2cccc(c2)Cl 9H-359S CN(c1ccccc1)C(=O)CSCc2ccccc2Cl 9H-360S c1ccc(cc1)c2ncc(c(n2)O)S(=O)(=O)c3ccccc3 9H-361S CN(C)c1ncc(c(n1)O)S(=O)(=O)c2ccccc2 9H-362S CN(c1ccccc1)C(=O)CSCc2ccc(cc2)Cl 9H-363S COc1ccc(cc1)S(=O)CC(=O)Nc2ccc(cc2Cl)Cl 9H-364S CN(C)/C=C(\C#N)/S(=O)(=O)C 9H-365S CN(C)/C=C(\C(=O)OC)/S(=O)(=O)C 9H-366S c1cc(cc(c1)S(=O)CC(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F 9H-367S CC(C)(C)c1ccc(cc1)CS(=O)CC(=O)Nc2ccc(cc2Cl)Cl 9H-368S COc1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccc(cc2Cl)Cl 9H-369S Cc1ncc(c(n1)O)S(=O)(=O)c2ccccc2 9H-370S c1ccc(cc1)c2c(cnc(n2)c3ccccn3)S(=O)(=O)c4ccccc4 9H-371S c1ccc(cc1)c2c(cnc(n2)c3cccnc3)S(=O)(=O)c4ccccc4 9H-372S c1cc(ccc1SCC(=O)c2ccc(cc2Cl)Cl)Cl 9H-373S c1ccc(cc1)S(=O)(=O)c2cnc(nc2c3ccc(cc3Cl)Cl)c4cccnc4 9H-374S c1ccc(cc1)c2ncc(c(n2)c3ccc(cc3Cl)Cl)S(=O)(=O)c4ccccc4 9H-375S c1cc(cc(c1)S(=O)(=O)CC(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F 9H-380S CN(c1ccccc1)C(=O)CS(=O)c2cccc(c2)Cl 9H-381S CS(=O)(=O)c1cnc(nc1N)c2ccccc2 9H-382S CS(=O)(=O)c1cnc(nc1N)c2cccnc2 9H-383S CN(C)c1ncc(c(n1)N)S(=O)(=O)C 9H-384S CN(c1ccccc1)C(=O)CS(=O)Cc2ccccc2Cl 9H-385S CN(C)/C=C(/C(=O)c1ccccc1)\S(=O)(=O)c2ccc(cc2)Cl 9H-386S Cc1ccc2c(c1)nc(oc2=O)N(C)C 9H-389S CN(C)c1nc2cc(ccc2c(=O)o1)F 9H-391S CS(=O)(=O)CC(=O)c1ccc(cc1)F 9H-392S CN(c1ccccc1)C(=O)CS(=O)Cc2ccc(cc2)Cl 9H-393S CN(c1ccccc1)C(=O)CS(=O)(=O)c2cccc(c2)Cl 9H-394S CS(=O)(=O)c1cnc(nc1O)c2ccccc2 9H-395S c1cc(ccc1S(=O)(=O)CC(=O)c2ccc(cc2Cl)Cl)Cl 9H-396S CN(c1ccccc1)C(=O)CS(=O)(=O)Cc2ccc(cc2)Cl 9H-397S CN(C)c1ncc(c(n1)c2ccccc2)S(=O)(=O)c3ccc(cc3)Cl 9H-398S Cc1ncc(c(n1)c2ccccc2)S(=O)(=O)c3ccc(cc3)Cl 9H-399S CN(C)/C=C(/C(=O)c1ccc(cc1)F)\S(=O)(=O)C 9H-400S CCOC(=O)C1=C(Nc2ccccc2S1=O)C 9H-401S Cc1ccc(cc1C)NC(=O)C(c2ccccc2)SCC(=O)OC 9H-402S Cc1ccc(cc1C)NC(=O)C(c2ccccc2)SCC(=O)O 9H-403S Cc1ccc(cc1C)N2C(=O)CS(=O)C(C2=O)c3ccccc3 9H-404S c1ccc(cc1)C(C(=O)NCc2ccc(cc2Cl)Cl)SCC(=O)O 9H-406S c1ccc(cc1)C2C(=O)N(C(=O)CS2)Cc3ccc(cc3Cl)Cl 9H-407S c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(c(c2)F)F 9H-413S COc1ccc(cc1)NC(=O)c2cccc(c2)C(F)(F)F 9H-414S c1cc(cc(c1)C(F)(F)F)c2nnnn2c3cccc(c3)C(F)(F)F 9H-415S c1cc(cc(c1)C(F)(F)F)c2nnnn2c3ccc(cc3F)F 9H-416S c1cc(cc(c1)C(F)(F)F)c2nnnn2c3ccc(c(c3)F)F 9H-417S COc1ccc(cc1)n2c(nnn2)c3cccc(c3)C(F)(F)F 9H-418S COc1ccc(cc1)C(=O)Nc2cccc(c2)C(F)(F)F 9H-419S COc1ccc(cc1)C(=O)Nc2ccc(cc2F)F 9H-420S COc1ccc(cc1)C(=O)Nc2ccc(c(c2)F)F 9H-421S COc1ccc(cc1)C(=O)Nc2ccc(cc2)OC 9H-422S c1cc(ccc1c2ccc(c(=O)[nH]2)C#N)Cl 9H-424S COc1ccc(cc1)c2nnnn2c3cccc(c3)C(F)(F)F 9H-426S COc1ccc(cc1)c2nnnn2c3ccc(cc3F)F 9H-427S COc1ccc(cc1)c2nnnn2c3ccc(c(c3)F)F 9H-428S COc1ccc(cc1)c2nnnn2c3ccc(cc3)OC 9H-429S CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)Nc2ccc(cc2F)F 9H-431S COc1ccc(cc1)NC(=O)c2ccc(cc2Cl)S(=O)(=O)C 9H-433S c1ccc(cc1)c2ccc(c(=O)[nH]2)C#N 9H-434S c1cc(ccc1c2ccc(c(=O)n2Cc3ccc(c(c3)Cl)Cl)C#N)Cl 9H-435S CS(=O)(=O)c1ccc(c(c1)Cl)c2nnnn2c3cccc(c3)C(F)(F)F 9H-436S CS(=O)(=O)c1ccc(c(c1)Cl)c2nnnn2c3ccc(cc3F)F 9H-437S CS(=O)(=O)c1ccc(c(c1)Cl)c2nnnn2c3ccc(c(c3)F)F 9H-438S COc1ccc(cc1)n2c(nnn2)c3ccc(cc3Cl)S(=O)(=O)C 9H-439S c1ccc(cc1)c2ccc(c(=O)n2Cc3ccc(c(c3)Cl)Cl)C#N 9H-440S Cc1ccc(cc1)Cn2c(ccc(c2=O)C#N)c3ccccc3 9H-448S c1ccc(cc1)c2ccc(c(=O)n2Cc3c(cccc3Cl)Cl)C#N 9H-449S c1ccc(cc1)C(C(=O)Nc2ccc(cc2)C(F)(F)F)SCC(=O)O 9H-450S c1ccc(cc1)c2ccc(c(=O)n2Cc3ccccc3Cl)C#N 9H-451S c1ccc(cc1)c2ccc(c(=O)n2Cc3cccc(c3)Cl)C#N 9H-452S c1ccc(cc1)c2ccc(c(=O)n2Cc3ccc(cc3)Cl)C#N 9H-453S COc1ccc(cc1)Cn2c(ccc(c2=O)C#N)c3ccccc3 9H-454S c1ccc(cc1)c2ccc(c(=O)n2Cc3cccc(c3)C(F)(F)F)C#N 9H-455S CC(C)(C)c1ccc(cc1)Cn2c(ccc(c2=O)C#N)c3ccccc3 9H-456S COc1ccc(cc1)NC(=O)C(c2ccccc2)SCC(=O)O 9H-457S c1ccc(cc1)C(C(=O)Nc2ccc(cc2)C#N)SCC(=O)O 9H-458S c1ccc(cc1)C2C(=O)N(C(=O)CS2)c3ccc(cc3)C(F)(F)F 9H-459S COc1ccc(cc1)N2C(=O)CSC(C2=O)c3ccccc3 9H-460S c1ccc(cc1)C2C(=O)N(C(=O)CS2)c3ccc(cc3)C#N 9H-461S Cn1c(ccc(c1=O)C#N)c2ccccc2 9H-462S CCOC(=O)Cn1c(ccc(c1=O)C#N)c2ccccc2 9H-463S COc1ccc(cc1)N2C(=O)CS(=O)C(C2=O)c3ccccc3 9H-465S c1ccc(cc1)C2C(=O)N(C(=O)CS2=O)c3ccc(cc3)Br 9H-466S C=CCn1c(ccc(c1=O)C#N)c2ccccc2 9H-467S c1ccc(cc1)C(C(=O)Nc2ccc(cc2Cl)Cl)SCC(=O)O 9H-468S c1ccc(cc1)C2C(=O)N(C(=O)CS2)c3ccc(cc3Cl)Cl 9H-469S CCn1c(ccc(c1=O)C#N)c2ccccc2 9H-470S C#CCn1c(ccc(c1=O)C#N)c2ccccc2 9H-471S c1ccc(cc1)C2C(=O)N(C(=O)CS2(=O)=O)c3ccc(cc3)Br 9H-473S c1ccc(cc1)C2C(=O)N(C(=O)CS2(=O)=O)c3ccc(cc3)Cl 9H-474S CC(C)(C)c1ccc(cc1)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl 9H-475S c1cc(cc(c1)Cl)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl 9H-476S c1cc(ccc1Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl)C(F)(F)F 9H-477S c1ccc(c(c1)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl)Cl 9H-478S c1cc(ccc1Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl)Cl 9H-479S COc1ccc(cc1)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl 9H-480S Cn1c(ccc(c1=O)C#N)c2ccc(cc2)Cl 9H-481S C=CCn1c(ccc(c1=O)C#N)c2ccc(cc2)Cl 9H-482S CCn1c(ccc(c1=O)C#N)c2ccc(cc2)Cl 9H-483S c1cc(c(c(c1)Cl)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl)F 9H-484S c1cc(ccc1Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl)F 9H-485S c1cc(cc(c1)F)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl 9H-486S c1cc(c(c(c1)Cl)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl)Cl 9H-487S c1cc(ccc1c2ccc(c(=O)n2Cc3ccc(cc3Cl)Cl)C#N)Cl 9H-488S Cc1ccc(cc1)Cn2c(ccc(c2=O)C#N)c3ccc(cc3)Cl 9H-489S CCOC(=O)Cn1c(ccc(c1=O)C#N)c2ccc(cc2)Cl 9H-490S c1cc(ccc1C(C(=O)Nc2ccc(cc2)Cl)SCC(=O)O)Cl 9H-493S c1cc(ccc1C2C(=O)N(C(=O)CS2)c3ccc(cc3)Cl)Cl 9H-494S CN(c1ccccc1)C(=O)CS(=O)(=O)Cc2ccccc2Cl 9H-501S COc1ccc(cc1)c2c(cnc(n2)c3ccccc3)S(=O)(=O)C 9H-509S COc1ccc(cc1)c2c(cnc(n2)c3ccccn3)S(=O)(=O)C 9H-510S CN(C)c1ncc(c(n1)c2ccc(cc2)F)S(=O)(=O)C 9H-511S CN(C)c1ncc(c(n1)c2ccc(cc2)OC)S(=O)(=O)C 9H-512S CN(C)/C=C(/C(=O)c1ccc(cc1Cl)Cl)\S(=O)(=O)c2ccc(cc2)Cl 9H-513S Cc1ncc(c(n1)c2ccccc2Cl)S(=O)(=O)c3ccccc3 9H-514S c1ccc(cc1)c2c(cnc(n2)c3cccnc3)S(=O)(=O)c4ccc(cc4)Cl 9H-515S CN(C)c1ncc(c(n1)c2ccc(cc2Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl 9H-523S Cc1ncc(c(n1)c2ccc(cc2Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl 9H-524S Cc1c(c(n(n1)C(=O)c2cccc(c2)C(F)(F)F)C)CS(=O)(=O)c3ccccc3 9H-900 COc1ccc(cc1)COc2ccc(cc2OC)C=O 9H-901 c1c(cnc(c1Cl)N2CCC3(CC2)OCC=CCO3)C(F)(F)F 9H-902 COc1cc(ccc1OCc2ccc(cc2)Cl)C=O 9H-903 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)/C=C/C(=O)O 9H-904 C/[N+](=C/c1ccc(c(c1)OC)OCc2ccc(cc2)OC)/[O-] 9H-905 C/[N+](=C/c1ccc(c(c1)OC)OCc2ccc(cc2)Cl)/[O-] 9H-906 Cc1c(c(n(n1)C(=O)C)C)CS(=O)(=O)c2ccccc2 9H-907 CN1C(C(CO1)S(=O)(=O)c2ccccc2)c3ccc(c(c3)OC)OCc4ccc(cc4)Cl 9H-908 CN1C(C(CO1)S(=O)(=O)c2ccccc2)c3ccc(c(c3)OC)OCc4ccc(cc4)OC 9H-909 c1cc(nc(c1)F)N2CCC3(CC2)OCC=CCO3 9H-910 Cc1c(c(n(n1)S(=O)(=O)C(F)(F)F)C)CS(=O)(=O)c2ccccc2 9H-911 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)C=CC2=O 9H-912 c1cc(cc(c1)Br)NC(=O)/C=C\C(=O)O 9H-914 CN(c1c(cc(cn1)C(F)(F)F)Cl)N2C(=O)CC(C2=O)Sc3ccc(cc3)Cl 9H-915 CN1C(C2C(O1)C(=O)N(C2=O)N(C)c3c(cc(cn3)C(F)(F)F)Cl)c4ccccc4 9H-916 Cc1c(c(n(n1)C)C)CS(=O)(=O)c2ccccc2 9H-917 CC1(OCCO1)c2ccc3c(c2)c(on3)c4cccs4 9H-918 Cc1c(c(n(n1)C(=O)c2cccnc2)C)CS(=O)(=O)c3ccccc3 9H-919 c1cc(nc(c1)Cl)N2CCN(CC2)c3c(cc(c(n3)N)C#N)C#N 9H-921 CC(=O)C1=NOC2C1C(=O)N(C2=O)c3ccc(cc3)Cl 9H-922 CN(C)/C=C/C(=O)c1ccncc1 9H-923 CC(C1=NOC(C1)CNc2c(cc(cn2)C(F)(F)F)Cl)O 9H-924 CN(C)/C=N/c1c(cc(c(n1)N2CCN(CC2)c3cccc(n3)Cl)C#N)C#N 9H-925 c1ccc2c(c1)c(c(n2c3c(cc(cn3)C(F)(F)F)Cl)CSc4ccc(cc4)Cl)Br 9H-926 CCOC(=O)C1=NOC2C1COC3(CCN(CC3)c4ccc(cc4)[N+](=O)[O-])OC2 9H-927 Cc1c2c(con2)c(nn1)c3ccccn3 9H-931 c1ccc(c(c1)CC[N+](=O)[O-])NC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9J-001 c1ccc(cc1)N2CCN(CC2)C(=O)Nc3ccccc3CC[N+](=O)[O-] 9J-002 CC(=O)/C(=C\N(C)C)/c1ccccc1 9J-003 c1cnc(nc1)N2CCC(C2=O)/C=N/OCc3ccc(cc3)F 9J-004 c1ccc(c(c1)CC[N+](=O)[O-])NC(=O)N2CCOCC2 9J-006 CN(C)C(=O)Nc1ccccc1CC[N+](=O)[O-] 9J-007 c1ccc(cc1)CO/N=C/C2CCN(C2=O)c3ncccn3 9J-008 c1cnc(nc1)N2CCC(C2=O)/C=N/OCc3ccc(cc3Cl)Cl 9J-009 c1cnc(nc1)N2CC/C(=C/Nc3ccc(cc3)C#N)/C2=O 9J-010 CN1CCN(CC1)C(=O)Nc2ccccc2CC[N+](=O)[O-] 9J-011 c1cc(cc(c1)C(F)(F)F)CO/N=C/C2CCN(C2=O)c3ncccn3 9J-012 c1ccc(c(c1)CC[N+](=O)[O-])NC(=O)Nc2cccc(c2)C(F)(F)F 9J-013 Cc1ccc(cc1)NC(=O)Nc2ccccc2CC[N+](=O)[O-] 9J-014 c1ccc(c(c1)O)OS(=O)(=O)NCc2ccc(cc2Cl)Cl 9J-016 CC(=O)C(/C=N/OC)c1ccccc1 9J-017 c1ccc(cc1)/C=C/c2[nH]c3c(n2)c(ncn3)N 9J-018 c1ccc(cc1)N2CCN(CC2)C(=O)CCc3c(cc(cn3)C(F)(F)F)Cl 9J-020 CN(C)c1nc(n(n1)S(=O)(=O)c2cccc(c2)C(F)(F)F)N(C)C 9J-024 Cc1c(sc(c1c2ccccc2)C#N)C#N 9J-025 Cc1c(c(sc1C(=O)/N=C/N(C)C)C#N)c2ccccc2 9J-026 Cc1c(c(sc1c2nc[nH]n2)C#N)c3ccccc3 9J-027 c1ccc(c(c1)Oc2c(cc(cn2)C(F)(F)F)Cl)OS(=O)(=O)NCc3ccc(cc3Cl)Cl 9J-028 Cc1c(c(sc1c2ncn(n2)C)C#N)c3ccccc3 9J-029 c1cc(ccc1C(=O)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)Cl 9J-034 CN(C)/C=C/c1c(sc(c1c2ccccc2)C#N)C#N 9J-037 Cc1c(c(sc1C#N)C(=O)N)C 9J-039 CCOC(=O)C(=CNc1ccccc1Oc2c(cc(cn2)C(F)(F)F)Cl)C(=O)OCC 9J-041 Cc1c(c(sc1C#N)C#N)C 9J-042 C/C(=N/Nc1c(cc(cn1)C(F)(F)F)Cl)/c2ccncc2 9J-047 CN(C)c1cc(nc(c1C#N)N(C)C)Cl 9J-049 c1ccc2c(c1)nc(c(n2)O)C(F)(F)F 9J-050 Cc1cc(nc(c1S(=O)(=O)c2cccc(c2)Cl)Cl)C 9J-301S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)Cl)C 9J-302S CCOc1c(c(cc(n1)C)C)S(=O)(=O)c2cccc(c2)Cl 9J-303S Cc1ccc(cc1)S(=O)(=O)c2cc(c[nH]c2=O)c3ccc(cc3)Cl 9J-304S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)OC)C 9J-305S Cc1cccc(c1)S(=O)(=O)c2c(cc(nc2Cl)C)C 9J-306S c1ccc2c(c1)[nH]c(n2)c3ccc(nc3)Cl 9J-307S Cc1cc2c(cc1C)nc([nH]2)c3ccc(nc3)Cl 9J-308S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CS(=O)(=O)c2ccc(cc2)Cl 9J-309S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CS(=O)(=O)c2ccc(cc2)F 9J-310S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CS(=O)c2ccc(cc2)Cl 9J-311S Cc1cc(cc(c1OC(=O)N(C)C)C)C(=O)CS(=O)c2ccc(cc2)F 9J-312S CCOc1c(c(cc(n1)C)C)S(=O)(=O)c2ccc(cc2)Cl 9J-313S CCOc1c(c(cc(n1)C)C)S(=O)(=O)c2cccc(c2)C 9J-314S Cc1ccc(cc1)S(=O)(=O)c2cc(cn(c2=O)CC=C)c3ccc(cc3)Cl 9J-315S c1ccc(cc1)S(=O)(=O)c2cc(c[nH]c2=O)c3ccc(cc3)Cl 9J-316S c1ccc(c(c1)Cn2c3ccccc3nc2c4ccc(nc4)Cl)Cl 9J-317S c1ccc2c(c1)nc(s2)c3cccnc3O 9J-319S c1ccc2c(c1)nc(s2)c3cccnc3Cl 9J-320S CCOC(=O)C/C(=N\NC(=O)N)/C(F)(F)F 9J-323S COc1ccc(cc1)Sc2c(cccn2)c3nc4ccccc4s3 9J-324S c1ccc2c(c1)nc(n2Cc3ccc(cc3)Cl)c4ccc(nc4)Cl 9J-325S c1ccc2c(c1)nc(n2Cc3ccc(cc3Cl)Cl)c4ccc(nc4)Cl 9J-326S c1ccc2c(c1)nc(n2Cc3ccc(c(c3)Cl)Cl)c4ccc(nc4)Cl 9J-327S CCOC(=O)Cn1c2ccccc2nc1c3ccc(nc3)Cl 9J-331S Cc1ccccc1Cn2c3ccccc3nc2c4ccc(nc4)Cl 9J-332S COc1c(cccn1)c2nc3ccccc3s2 9J-333S Cc1ccc(cc1)Cn2c3ccccc3nc2c4ccc(nc4)Cl 9J-334S CC(C)Nc1ccc(cc1N)C(F)(F)F 9J-336S CN(C)c1c(cccn1)c2nc3ccccc3s2 9J-341S c1ccc(cc1)Sc2c(cccn2)c3nc4ccccc4s3 9J-342S CC(C)n1c2ccc(cc2nc1c3cccnc3Cl)C(F)(F)F 9J-345S c1ccc2c(c1)nc(s2)c3cccn(c3=O)Cc4ccc(c(c4)Cl)Cl 9J-351S CCOC(=O)CSc1nc(cc(=O)n1CC=C)C(F)(F)F 9J-507S C=CCn1c(=O)cc(nc1SCc2ccc(c(c2)Cl)Cl)C(F)(F)F 9J-508S C=CCn1c(=O)cc(nc1SCc2cccc(c2)C(F)(F)F)C(F)(F)F 9J-509S C=CCn1c(=O)cc(nc1SCc2ccccc2)C(F)(F)F 9J-513S C=CCn1c(=O)cc(nc1SCc2ccccc2Cl)C(F)(F)F 9J-514S C=CCn1c(=O)cc(nc1SCc2ccc(cc2Cl)Cl)C(F)(F)F 9J-519S C=CCn1c(=O)cc(nc1SCc2ccccc2C#N)C(F)(F)F 9J-520S Cc1ccc(cc1)CSc2nc(cc(=O)n2CC=C)C(F)(F)F 9J-522S C=CCn1c(=O)cc(nc1SCc2c(cccc2Cl)F)C(F)(F)F 9J-524S COc1cccc(c1)CSc2nc(cc(=O)n2CC=C)C(F)(F)F 9J-526S CCCn1c(=O)cc(nc1SCC(=O)OCC)C(F)(F)F 9J-530S CCCn1c(=O)cc(nc1SCc2ccc(c(c2)Cl)Cl)C(F)(F)F 9J-532S CCCn1c(=O)cc(nc1SCc2cccc(c2)C(F)(F)F)C(F)(F)F 9J-533S CCCn1c(=O)cc(nc1SCc2ccc(cc2)C(=O)OC)C(F)(F)F 9J-534S CCCn1c(=O)cc(nc1SCc2ccc(cc2)Cl)C(F)(F)F 9J-535S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)F)CSC2 9J-537S Cc1cccc(c1)c2c(c(c3n2CSC3)C(=O)OC)C(=O)OC 9J-539S COC(=O)c1c2n(c(c1C(=O)OC)c3ccccc3)CS(=O)C2 9J-540S COC(=O)c1c2n(c(c1C(=O)OC)c3ccccc3)CS(=O)(=O)C2 9J-541S COc1ccc(cc1OC)C(=O)NCCSc2ccc(cc2)Cl 9J-542S COc1cc(cc(c1OC)OC)C(=O)NCCSc2ccc(cc2)Cl 9J-543S c1cc(cc(c1)F)C(=O)NCCSc2ccc(cc2)Cl 9J-544S CC(=O)Nc1ccc(c(c1)Cl)Cl 9J-545S CC(=O)Nc1cc(c(cc1[N+](=O)[O-])Cl)Cl 9J-546S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(c(c3)Cl)Cl)CSC2 9J-548S COc1ccc(cc1)c2c(c(c3n2CSC3)C(=O)OC)C(=O)OC 9J-551S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)F)CS(=O)C2 9J-552S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)F)CS(=O)(=O)C2 9J-553S Cc1cccc(c1)c2c(c(c3n2CS(=O)C3)C(=O)OC)C(=O)OC 9J-554S Cc1cccc(c1)c2c(c(c3n2CS(=O)(=O)C3)C(=O)OC)C(=O)OC 9J-555S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(cc3)Cl)CCC2 9J-557S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(c(c3)Cl)Cl)CS(=O)C2 9J-559S COC(=O)c1c2n(c(c1C(=O)OC)c3ccc(c(c3)Cl)Cl)CS(=O)(=O)C2 9J-560S COc1ccc(cc1)c2c(c(c3n2CS(=O)C3)C(=O)OC)C(=O)OC 9J-563S COc1ccc(cc1)c2c(c(c3n2CS(=O)(=O)C3)C(=O)OC)C(=O)OC 9J-564S CC(C)(C)c1ccc(cc1)c2c(c(c3n2CSC3)C(=O)OC)C(=O)OC 9J-566S CC(=O)c1c(ccs1)Br 9J-900 c1csc(c1Br)C(=O)CBr 9J-901 c1cc(c(cc1Cl)Cl)/C=C/C(=O)c2c(ccs2)Br 9J-902 c1cnccc1c2nc(cs2)c3c(ccs3)Br 9J-903 c1csc(c1Br)c2csc(n2)N 9J-904 c1cc(ccc1NC(=O)Nc2nc(cs2)c3c(ccs3)Br)Cl 9J-906 c1cc(ccc1CON/C=N\C(=S)Nc2c(cc(cn2)C(F)(F)F)Cl)Cl 9J-908 c1csc(c1Cl)C(=O)CBr 9J-909 c1csc(c1Cl)c2csc(n2)N 9J-910 c1cc(cnc1)c2nc(cs2)c3c(ccs3)Cl 9J-911 CN(C)/C=N/c1nc(cs1)c2c(ccs2)Cl 9J-912 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2nc(cs2)c3c(ccs3)Cl 9J-913 c1cc(c(cc1Cl)S(=O)(=O)Nc2nc(cs2)c3c(ccs3)Cl)Cl 9J-914 c1ccc(cc1)c2nc(cs2)c3c(ccs3)Br 9J-915 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)F)/SC2=O 9K-001 COc1ccc(cc1)N/C=C\2/c3ccccc3C(=O)S2 9K-002 c1ccc2c(c1)/C(=C/Nc3ccc(cc3)Br)/SC2=O 9K-003 Cc1ccc(c(c1)C)N/C=C\2/c3ccccc3C(=O)S2 9K-004 c1cc(ccc1C(C#N)c2ccc(cc2)Cl)C(=O)c3ccc(cc3)F 9K-005 Cc1ccc(cc1)N/C=C\2/c3ccccc3C(=O)S2 9K-006 CCOC(=O)c1cccc(c1)N/C=C\2/c3ccccc3C(=O)S2 9K-007 CO/N=C/C1c2ccccc2C(=O)S1 9K-008 COc1ccc(cc1)C(C#N)c2ccc(cc2)C(=O)c3ccc(cc3)F 9K-009 c1ccc2c(c1)C(SC2=O)/C=N/OCc3cccc(c3)C(F)(F)F 9K-010 c1cc(nc(c1)Cl)C(C#N)c2ccc(cc2)Cl 9K-011 c1ccc2c(c1)/C(=C/Nc3ccc(c(c3)Cl)Cl)/SC2=O 9K-012 c1ccc2c(c1)/C(=C/Nc3cc(ccc3Cl)Cl)/SC2=O 9K-013 c1cc(ccc1C(C#N)c2ccc(cc2Cl)Cl)C(=O)c3ccc(cc3)F 9K-014 c1cc(ccc1C(C#N)c2ccc(cc2)F)C(=O)c3ccc(cc3)F 9K-015 Cc1ccc(cc1)C(C#N)c2ccc(cc2)C(=O)c3ccc(cc3)F 9K-016 c1cc(sc1)CC(C#N)c2c(cc(cn2)C(F)(F)F)Cl 9K-017 COC(=O)CC(C#N)(c1ccccc1)c2cccc(c2C#N)F 9K-018 COc1ccccc1C(C#N)c2cccc(n2)Cl 9K-020 c1ccc(cc1)C(=O)c2ccc(cc2)C(c3ccc(cc3)Br)C(=O)N 9K-021 CN(C)/C=N/C(=O)C(c1ccc(cc1)C(=O)c2ccccc2)c3ccc(cc3)Br 9K-022 CO/N=C\NC(=O)C(c1ccc(cc1)C(=O)c2ccccc2)c3ccc(cc3)Br 9K-024 c1cc(ccc1C(C#N)c2ccc(cc2)Br)C(=O)c3ccc(cc3)F 9K-025 c1ccc(cc1)C(=O)c2ccc(cc2)C(c3ccc(cc3)Br)C(=O)N/C=N\O 9K-026 c1ccc(cc1)C(=O)c2cccc(c2C#N)C(=O)c3ccccc3 9K-027 c1ccc(cc1)C(C#N)(c2cccc(c2C#N)C(C#N)(c3ccccc3)N4CCOCC4)N5CCOCC5 9K-028 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C\Nc4ccccc4)F 9K-029 c1ccc(cc1)C\2c3cccc(c3C(=O)/C2=C\Nc4ccc(cc4)F)F 9K-030 COC(=O)C1=C(c2ccccc2C1(C#N)c3ccccc3)N 9K-031 COc1ccc(cc1)Oc2cccc3c2C(=O)CC3c4ccccc4 9K-033 c1ccc(cc1)C2CC(=O)c3c2cccc3Oc4ccc(cc4)Cl 9K-034 CN(C)/C=C\1/C(c2cccc(c2C1=O)Oc3ccc(cc3)Cl)c4ccccc4 9K-035 CC(=O)C(/C=N/OCc1cccc(c1)C(F)(F)F)c2ccccc2 9K-037 c1ccc(cc1)C2(CC(=O)c3c2cccc3)C(=O)O 9K-038 c1ccc(cc1)C2CC(=O)c3c2cccc3Oc4ccccc4 9K-039 CC(=O)C(/C=N/OCc1c(cccc1Cl)F)c2ccccc2 9K-040 CC(=O)C(/C=N/OCc1ccc(cc1)Cl)c2ccc(c(c2)OC)OC 9K-041 c1ccc(cc1)C2CC(=O)c3c2cccc3 9K-043 c1ccc(cc1)C2CC(=O)c3c2cccc3Oc4cccc(c4)C(F)(F)F 9K-044 CN(C)/C=C\1/C(c2ccccc2C1=O)c3ccccc3 9K-045 c1ccc(cc1)C\2c3ccccc3C(=O)/C2=C\Nc4ccccc4 9K-046 COc1ccc(cc1)N/C=C\2/C(c3ccccc3C2=O)c4ccccc4 9K-047 CNC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(c(c3)Cl)Cl 9K-301S c1ccc(cc1)CNC(=O)c2cnn(c2C(F)(F)F)c3nc(cs3)c4ccc(c(c4)Cl)Cl 9K-302S Cc1ccc(cc1)CNC(=O)c2cnn(c2C(F)(F)F)c3nc(cs3)c4ccc(c(c4)Cl)Cl 9K-303S c1cc(cc(c1)C(F)(F)F)CNC(=O)c2cnn(c2C(F)(F)F)c3nc(cs3)c4ccc(c(c4)Cl)Cl 9K-304S CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)OC 9K-309S COc1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)O)C(F)(F)F 9K-311S CNC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)OC 9K-315S COc1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)NCc4ccccc4)C(F)(F)F 9K-316S Cc1ccc(cc1)CNC(=O)c2cnn(c2C(F)(F)F)c3nc(cs3)c4ccc(cc4)OC 9K-317S COc1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)NCc4cccc(c4)C(F)(F)F)C(F)(F)F 9K-318S COc1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)NCc4ccc(cc4)Cl)C(F)(F)F 9K-319S COc1ccc(cc1)c2csc(n2)n3c(c(cn3)C(=O)NCc4ccc(cc4)F)C(F)(F)F 9K-320S c1ccc(cc1)c2c(nc(nn2)c3cccc(c3)C(F)(F)F)N4CCOCC4 9K-324S Cc1ccc(cc1)c2nc(c(nn2)C)N3CC(OC(C3)C)C 9K-326S Cc1ccc(cc1)c2nc(c(nn2)C)Oc3ccc(cc3Cl)Cl 9K-327S Cc1ccc(cc1)c2nc(c(nn2)C)Sc3ccc(cc3)F 9K-328S c1cc(cnc1)c2nccc(n2)NC(=O)c3ccc(cc3)Cl 9K-332S c1cc(cnc1)c2nccc(n2)NC(=O)c3ccc(c(c3)Cl)Cl 9K-333S c1cc(cnc1)c2nccc(n2)NC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F 9K-334S c1cc(cnc1)c2ncc(cn2)NC(=O)C3CC3 9K-339S CC(=O)Nc1ccnc(n1)c2cccnc2 9K-341S c1cc(cc(c1)Cl)NC(=O)Nc2ccnc(n2)c3cccnc3 9K-342S c1cc(ccc1C(=O)Nc2ccnc(n2)c3ccncc3)Cl 9K-343S Cc1ccc(cc1)C(=O)Nc2ccnc(n2)c3ccncc3 9K-344S Cc1cccc(c1C)S(=O)(=O)c2c(cc([nH]c2=O)C)C 9K-346S CC(C)C(=O)Nc1ccnc(n1)c2cccnc2 9K-347S CCCCC(=O)Nc1ccnc(n1)c2cccnc2 9K-348S CC(C)CC(=O)Nc1ccnc(n1)c2ccncc2 9K-349S c1ccc2c(c1)cc(c(n2)Oc3ccc(cc3)Cl)c4ccc(cc4)Cl 9K-352S c1ccc2c(c1)cc(c(n2)Oc3ccc(cc3Cl)Cl)c4ccc(cc4)Cl 9K-353S COc1ccc(cc1)Oc2c(cc3ccccc3n2)c4ccc(cc4)Cl 9K-354S c1ccc2c(c1)cc(c(n2)Oc3ccccc3[N+](=O)[O-])c4ccc(cc4)Cl 9K-355S Cc1cccc(c1C)S(=O)(=O)c2c(cc(nc2Cl)C)C 9K-356S c1cnccc1c2nccc(n2)NC(=O)C3CC3 9K-358S c1cc(cnc1)c2nccc(n2)NC(=O)c3ccc(cc3)F 9K-359S c1ccc2c(c1)cc(c(n2)Oc3c(cccc3Cl)Cl)c4ccc(cc4)Cl 9K-360S Cc1cc(cc(c1)Oc2c(cc3ccccc3n2)c4ccc(cc4)Cl)C 9K-361S CCOC(=O)CN(c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl 9K-363S Cc1cccc(c1S(=O)(=O)c2c(cc(nc2Cl)C)C)C 9K-365S CCC(=O)Nc1ccnc(n1)c2cccnc2 9K-367S CC(C)(C)C(=O)Nc1ccnc(n1)c2cccnc2 9K-368S CCOC(=O)CN(c1ccccn1)S(=O)(=O)c2ccccc2 9K-372S c1cc(ccc1N(CC(=O)O)S(=O)(=O)c2ccc(cc2)Cl)Cl 9K-373S c1cc(cc(c1)N(CC(=O)O)S(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F 9K-374S Cc1cccc(c1C)S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C 9K-375S Cc1cccc(c1S(=O)(=O)c2c(cc(nc2OCC(C)C)C)C)C 9K-376S CCOC(=O)CN(c1ccccc1Cl)S(=O)(=O)c2cc(ccc2Cl)Cl 9K-377S c1cc(sc1)c2nc(c(nn2)C#N)N3CCOCC3 9K-507S Cc1c(c(on1)C)C(=O)N2CCOCC2 9K-514S Cc1c(c(on1)C)C(=O)N(C)c2ccccc2 9K-515S c1cc(ccc1Sc2ccc(cn2)C(=O)NN)Cl 9K-517S COC(=O)C(CC(=O)c1ccc(cc1)C(F)(F)F)c2ccc(cc2)Cl 9K-520S c1cc(ccc1C2CC(=NNC2=O)c3ccc(cc3)C(F)(F)F)Cl 9K-521S c1cc(cc(c1)F)C2=NNC(=O)C(C2)c3ccc(cc3)Cl 9K-522S COC(=O)C(CC(=O)c1cccc(c1)F)c2ccc(cc2)Cl 9K-523S c1cc(sc1)c2nnc(o2)c3ccc(cc3Cl)Cl 9K-525S Cc1ccccc1c2nnc(o2)c3cccs3 9K-527S c1ccc(c(c1)c2nnc(o2)c3cccs3)Cl 9K-529S Cc1ccccc1c2nnc(o2)c3ccco3 9K-531S c1ccc(c(c1)c2nnc(o2)c3ccco3)Cl 9K-533S C=CCN(CC=C)c1c(cc(cn1)C(F)(F)F)Cl 9K-900 CCOC(=O)/C(=C\Nc1ccc(cc1)OC)/C#N 9L-001 c1cc(c(cc1Cl)Cl)C(=O)c2ccc(s2)CC(=O)N 9L-003 Cc1ccc(cc1)CNS(=O)(=O)Oc2ccccc2O 9L-004 c1ccc(c(c1)O)OS(=O)(=O)NCc2ccc(cc2)Cl 9L-005 c1ccc2c(c1)c(=O)n(c(n2)C(F)(F)F)N 9L-006 c1ccc(c(c1)O)OS(=O)(=O)NCc2cccs2 9L-007 c1ccc(c(c1)O)OS(=O)(=O)NCc2ccccn2 9L-008 CC(=O)c1ccc(s1)/C(=C/c2ccccc2)/C#N 9L-009 CC(=O)c1ccc(s1)/C(=C/c2cccc(c2)OC)/C#N 9L-010 CC(=O)c1ccc(s1)/C(=C/c2cc(ccc2F)F)/C#N 9L-011 Cc1ccc(cc1)CNC(=O)c2ccccc2NC(=O)C(F)(F)F 9L-012 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccc(cc2)C 9L-013 COc1ccccc1CNS(=O)(=O)Oc2ccccc2O 9L-015 CCOC(=O)/C(=C\Nc1ccc(cc1)F)/C#N 9L-016 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccc(cc2)Cl 9L-018 c1ccc(cc1)CNS(=O)(=O)NCc2ccc(cc2)Cl 9L-019 c1cc(ccc1CNS(=O)(=O)NCc2ccc(cc2)Cl)Cl 9L-020 c1ccc2c(c1)c(=O)[nH]c(n2)C(F)(F)F 9L-021 CC(=O)c1ccc(s1)/C(=C/c2ccco2)/C#N 9L-022 CC(=O)c1ccc(s1)/C(=C/c2ccncc2)/C#N 9L-023 CCOC(=O)/C(=C\Nc1ccc(cc1)Cl)/C#N 9L-025 Cc1ccc(cc1)CO/N=C(\C)/c2ccc(s2)CC#N 9L-027 c1ccc(cc1)CNS(=O)(=O)NCc2ccccc2 9L-028 c1ccc(cc1)CNS(=O)(=O)NCc2ccc(cc2Cl)Cl 9L-029 C/C(=N\OCc1ccc(cc1)Cl)/c2ccc(s2)CC#N 9L-030 Cc1ccc(cc1)CNS(=O)(=O)NCc2ccccc2 9L-031 Cc1nc(nn1c2cc(c(cc2Cl)Cl)OC(C)C)C(=O)Nc3ccc(cc3)F 9L-301S c1ccc(cc1)N2c3ccccc3/C(=N/O)/C2=O 9L-302S COc1ccc(cc1)C(=O)O/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-303S CCOC(=O)C(c1ccccc1)Oc2ccccc2n3cccc3 9L-305S Cc1ccc(cc1)C(=O)O/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-307S CC(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-308S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)CCl)/C2=O 9L-309S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)C4CC4)/C2=O 9L-310S CCCC(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-311S c1ccc(cc1)C(C(=O)O)Oc2ccccc2n3cccc3 9L-313S CCCCC(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-315S CC(C)(C)C(=O)O/N=C/1\c2ccccc2N(C1=O)c3ccccc3 9L-316S CC(C)CC(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-317S CC(C)(CNc1ccccc1C(=O)NC)C(=O)NC 9L-319S CCC(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-320S CC(C)C(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-321S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)CCCl)/C2=O 9L-322S CC(C(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3)Cl 9L-323S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)CCCCl)/C2=O 9L-324S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)c4ccc(cc4)Cl)/C2=O 9L-325S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)c4ccccc4Cl)/C2=O 9L-326S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)c4cccc(c4)Cl)/C2=O 9L-327S c1ccc(cc1)N2c3ccccc3/C(=N\OC(=O)c4cccc(c4)C(F)(F)F)/C2=O 9L-328S COc1cccc(c1)C(=O)O/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-329S Cc1ccccc1C(=O)O/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-330S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)c4ccc(c(c4)Cl)Cl)/C2=O 9L-331S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)c4c(cccc4F)F)/C2=O 9L-332S Cc1ccccc1NC(=O)O/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-334S c1ccc(cc1)Cn2c(c(c(c2N)C#N)c3ccccc3)c4ccccc4 9L-336S CNc1nc(c(c(n1)Cl)SC)Cl 9L-337S Cc1cccc(c1NC(=O)O/N=C\2/c3ccccc3N(C2=O)c4ccccc4)C 9L-339S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)Nc4cc(cc(c4)Cl)Cl)/C2=O 9L-340S CCNC(=O)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-341S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)Nc4cccc(c4)C(F)(F)F)/C2=O 9L-342S Cc1ccc(cc1)NC(=O)O/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-344S c1ccc(cc1)N2c3ccccc3/C(=N/OC(=O)NC4CCCCC4)/C2=O 9L-345S c1ccc(cc1)N2c3ccccc3/C(=N/OCc4ccc(cc4)F)/C2=O 9L-346S CO/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-347S c1ccc(cc1)N2c3ccccc3/C(=N/OCc4ccc(cc4Cl)Cl)/C2=O 9L-348S Cc1ccc(cc1)CO/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-349S c1ccc(cc1)Cn2c(c(c3c2ncnc3Cl)c4ccccc4)c5ccccc5 9L-352S CNc1nc(c(c(n1)Cl)SC)N2CCOCC2 9L-355S Cc1cccc(c1)CO/N=C/2\c3ccccc3N(C2=O)c4ccccc4 9L-357S COc1ccc(cc1)CO/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-358S Cc1ccccc1CO/N=C\2/c3ccccc3N(C2=O)c4ccccc4 9L-359S c1ccc(cc1)N2c3ccccc3/C(=N/OCc4cccc(c4)Cl)/C2=O 9L-360S Cc1ccc(cc1)Sc2c3c(c(n(c3ncn2)Cc4ccccc4)c5ccccc5)c6ccccc6 9L-361S CCO/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-362S CC(C)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-363S CCCO/N=C/1\c2ccccc2N(C1=O)c3ccccc3 9L-364S CCC(C)O/N=C\1/c2ccccc2N(C1=O)c3ccccc3 9L-365S c1cc(ccc1c2cc(c(c(=O)[nH]2)C#N)c3ccc(cc3)Cl)F 9L-366S Cc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3ccc(cc3)Cl 9L-367S c1cc(cc(c1)Br)c2cc(c(c(n2)O)C#N)c3ccc(cc3)Cl 9L-368S c1cc(ccc1c2cc([nH]c(=O)c2C#N)c3ccc(cc3)Br)Cl 9L-369S c1cc(ccc1c2cc(nc(c2C#N)O)c3ccc(c(c3)Cl)Cl)Cl 9L-370S c1cc(cc(c1)C(F)(F)F)c2cc(c(c(n2)O)C#N)c3ccc(cc3)Cl 9L-371S c1cc(ccc1c2cc(c(c(n2)O)C#N)c3ccc(cc3)Cl)C(F)(F)F 9L-372S c1ccc(c(c1)c2cc(nc(c2C#N)O)c3ccc(cc3)Cl)C(F)(F)F 9L-373S c1ccc(c(c1)c2cc(nc(c2C#N)O)c3ccc(cc3)F)C(F)(F)F 9L-374S c1ccc(c(c1)c2cc(nc(c2C#N)O)c3ccc(c(c3)Cl)Cl)C(F)(F)F 9L-375S CN(CCSc1ccc(cc1)Br)C(=O)c2ccc(cc2)OC 9L-501S c1c(nns1)C(=O)NO 9L-502S CCOC(=O)C1=C(NC(=O)CC1c2ccccc2[N+](=O)[O-])C 9L-504S CCOC(=O)C1=C(NC(=O)CC1c2ccccc2Cl)C 9L-505S CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2)F)C 9L-506S CCOC(=O)C1=C(NC(=O)CC1c2ccccc2C(F)(F)F)C 9L-507S CCOC(=O)c1c(n(c(=S)s1)c2ccccc2Cl)SC 9L-509S CCOC(=O)c1c(n(c(=S)s1)c2ccc(cc2)C)SC 9L-510S c1ccc(c(c1)C2CC(=O)NC3=C2C(=O)OC3)[N+](=O)[O-] 9L-511S c1ccc(c(c1)C2CC(=O)NC3=C2C(=O)OC3)Cl 9L-512S CCOC(=O)C1=C(NC(=O)CC1c2c(cccc2Cl)Cl)C 9L-515S CC1=C(C(CC(=O)N1)c2ccc(cc2)[N+](=O)[O-])C(=O)OC 9L-516S CC1=C(C(CC(=O)N1)c2cccc(c2)[N+](=O)[O-])C(=O)OC 9L-517S CC1=C(C(CC(=O)N1)c2cccc(c2)Cl)C(=O)OC 9L-518S CC1=C(C(CC(=O)N1)c2ccc(cc2)C(F)(F)F)C(=O)OC 9L-519S CC(C)Oc1cc(c(cc1Cl)Cl)/N=C\2/NCCS2 9L-521S CSc1c(sc(=S)n1c2ccc(cc2)Cl)C#N 9L-522S CSc1c(sc(=S)n1c2cccc(c2)Cl)C#N 9L-523S Cc1ccc(cc1)n2c(c(sc2=S)C#N)SC 9L-525S c1ccc(cc1)C(=O)N2CCCC(=N2)c3ccc(cc3)Cl 9L-526S c1cc(ccc1C2=NN(CCC2)C(=O)C3CC3)Cl 9L-527S COc1cc(nc(n1)Oc2cc(c(cc2Cl)Cl)Cl)OC 9L-528S c1ccc(cc1)C2=NN(CCC2)C(=O)C3CC3 9L-530S COc1cc(c(cc1Cl)Cl)/N=C\2/NCCS2 9L-531S CC1=C(C(CC(=O)N1)c2ccc(cc2)F)C(=O)OC 9L-532S CCOC(=O)C1=C(NC(=O)CC1c2ccc(c(c2)[N+](=O)[O-])Cl)C 9L-533S CCOC(=O)C1=C(NC(=O)CC1c2ccc(c(c2)F)F)C 9L-534S c1cc(ccc1C2=NNC(=O)CC2)F 9L-535S c1cc(ccc1SCc2cc(nc(n2)S)O)Br 9L-540S c1ccc(cc1)SCc2cc(nc(n2)S)O 9L-541S c1cc(ccc1SCc2cc(nc(n2)SCc3ccc(c(c3)Cl)Cl)O)Cl 9L-542S c1cc(c(c(c1)Cl)SCc2cc(nc(n2)S)O)Cl 9L-543S c1c(nns1)C(=O)O 9L-544S C=CCNc1cc(nc(n1)SCc2ccc(cc2)Cl)CSc3ccc(cc3)Cl 9L-552S COc1ccc(cc1)CSc2nc(cc(n2)O)CSc3ccc(cc3)Br 9L-553S c1cc(cc(c1)C(F)(F)F)CSc2nc(cc(n2)O)CSc3c(cccc3Cl)Cl 9L-554S c1cc(cc(c1)C(F)(F)F)CSc2nc(cc(n2)Cl)CSc3c(cccc3Cl)Cl 9L-557S CCOC(=O)/C(=C/c1ccc(cc1Cl)Cl)/C#N 9L-561S c1ccc(cc1)SCc2cc(nc(n2)SCc3c(cccc3Cl)Cl)O 9L-564S CNc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)CSc3ccc(cc3)Cl 9L-565S CNc1cc(nc(n1)SCc2ccc(cc2)OC)CSc3ccc(cc3)Br 9L-566S C=CCNc1cc(nc(n1)SCc2ccc(c(c2)Cl)Cl)CSc3ccc(cc3)Cl 9L-567S CN(C)c1cc(nc(n1)SCc2ccc(cc2)OC)CSc3ccc(cc3)Br 9L-568S c1c(cnc(c1Cl)NC(=O)c2csnn2)Cl 9L-581S c1ccc(cc1)Cn2c3ccccc3nc2NC(=O)c4csnn4 9L-582S c1cc(ncc1Cl)NC(=O)c2csnn2 9L-583S c1cc(c(c(c1NC(=O)c2csnn2)F)Cl)F 9L-584S c1cc(ccc1NC(=O)c2csnn2)Br 9L-585S c1cc(ccc1NC(=O)c2csnn2)Cl 9L-586S c1ccc(cc1)c2c(c(nc(n2)SCc3c(cccc3Cl)Cl)O)C#N 9L-587S c1c(nns1)C(=O)Nc2nncs2 9L-588S COC(=O)c1c(ccs1)NC(=O)c2csnn2 9L-589S c1cc(ccc1c2cc(nc(c2C#N)O)c3ccc(cc3)Cl)Cl 9L-591S c1ccc(c(c1)c2cc(c(c(=O)[nH]2)C#N)c3ccc(cc3)Cl)Cl 9L-592S c1c(cc(cc1Cl)Cl)NC(=O)c2csnn2 9L-593S c1c(nns1)C(=O)N2CCOCC2 9L-594S Cc1cc(nc(c1)NC(=O)c2csnn2)C 9L-595S c1cc(c2ncnn2c1)NC(=O)c3csnn3 9L-596S Cc1cccc(n1)NC(=O)c2csnn2 9L-597S c1cc(cnc1)NC(=O)c2csnn2 9L-599S c1cc(sc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N 9L-702 c1cc(c(cc1Cl)Cl)c2cc(n[nH]2)C3CCN(CC3)CC#N 9L-703 c1ccc2c(c1)/C(=N\Nc3ccc(cc3Br)Br)/C(=O)OC2=O 9L-705 c1ccc2c(c1)c3c(nn2)nn4c(=O)cc(nc4n3)C(F)(F)F 9L-708 CC(C)(CCl)C(=O)Nc1ccc(cc1)[N+](=O)[O-] 9L-709 CC1(CN(C1=O)c2ccc(cc2)[N+](=O)[O-])C 9L-710 c1cc(oc1)c2cc([nH]n2)C3CCNCC3 9L-711 c1ccn(c1)C2=C(C(C3=C(O2)CCCC3=O)c4ccco4)C#N 9L-712 CC(C)(CCl)C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F 9L-714 CC1(CN(C1=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C 9L-715 CC(C)(CCl)C(=O)Nc1ccc(cc1)C#N 9L-716 CC1(CN(C1=O)c2ccc(cc2)C#N)C 9L-717 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)C=O)Sc3ncccn3)C 9L-718 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)C=O)Sc3c(cc(cn3)C(F)(F)F)Cl)C 9L-719 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)/C=N/OCc3ccc(cc3Cl)Cl)Cl)C 9L-720 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)/C=N/OCc3ccc(cc3Cl)F)Cl)C 9L-721 CC(C)(CCl)C(=O)Nc1nccs1 9L-722 CC(C)(CCl)C(=O)Nc1ccc(cc1)S(=O)(=O)N 9L-723 c1cc(oc1)c2cc(n[nH]2)C3CCN(CC3)CC#N 9L-724 c1cc(sc1)/C=C/2\C(=O)C3CCN2CC3 9L-725 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)C=O)Sc3ccccn3)C 9L-726 c1cc(oc1)c2cc(n[nH]2)C3CCN(CC3)Cc4ccc(cc4)[N+](=O)[O-] 9L-727 c1cc(ccc1c2cc([nH]n2)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl 9L-728 CC(C)(CCl)C(=O)Nc1cc(cc(c1)OC)OC 9L-729 CC1(CN(C1=O)c2cc(cc(c2)OC)OC)C 9L-730 c1cc(sc1)c2cc(n[nH]2)C3CCNCC3 9L-731 CCOC(=O)CN1CCC(CC1)c2cc([nH]n2)c3ccc(cc3)Cl 9L-732 CC(C)(CCl)C(=O)Nc1ccc(cc1)OCc2ccccc2 9L-733 CC1(CN(C1=O)c2ccc(cc2)OCc3ccccc3)C 9L-734 CC(C)(CCl)C(=O)Nc1cc(cc(c1)NC(=O)C(C)(C)CCl)C(=O)OC 9L-735 CC1(CN(C1=O)c2cc(cc(c2)N3CC(C3=O)(C)C)C(=O)OC)C 9L-736 c1ccc(cc1)/C=C/C=C/2\C(=O)C3CCN2CC3 9L-738 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4ccco4 9L-739 c1cc(cc(c1)Cl)NC(=O)N2CCC(CC2)c3cc([nH]n3)c4ccco4 9L-740 CC(C)(CCl)C(=O)Nc1cc(cc(c1)Cl)Cl 9L-741 CC1(CN(C1=O)c2cc(cc(c2)Cl)Cl)C 9L-742 C(=O)c1c(nc(s1)Cl)Cl 9L-743 Cc1ccc(cc1)CN2CCC(CC2)c3cc([nH]n3)c4cccs4 9L-744 CC1(CN(C1=O)c2ccc(cc2)S(=O)(=O)N)C 9L-745 CC(=O)Nc1ccc(cc1)NC(=O)C(C)(C)CCl 9L-746 CCOC(=O)c1c(c(c(=O)n2c1nc[nH]2)C#N)c3ccc(cc3)Cl 9L-747 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4cccs4 9L-748 CC(C)(C)OC(=O)N1CC(CC1C(=O)O)O 9L-749 CC(C)(CCl)C(=O)Nc1ccc(cc1)CC#N 9L-753 CC1(CN(C1=O)c2ccc(cc2)CC#N)C 9L-754 CC(C)(CCl)C(=O)Nc1ccc(cc1Br)Br 9L-755 CC1(CN(C1=O)c2ccc(cc2Br)Br)C 9L-756 c1cc(ccc1CN2CCC(CC2)c3cc(n[nH]3)c4ccc(cc4Cl)Cl)Cl 9L-758 c1ccc(cc1)C(=O)/C=C/c2ccc(cc2Cl)Cl 9L-759 CC(=O)Nc1ccc(cc1)N2CC(C2=O)(C)C 9L-760 c1cc(ccc1/C=C\2/C(=O)C3CCN2CC3)[N+](=O)[O-] 9L-761 c1cc(sc1)c2cc(n[nH]2)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-762 CC(C)(CCl)C(=O)Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl 9L-763 c1cc(ncc1I)N 9L-900 CC(=O)Nc1ccc(cn1)I 9L-901 Cc1c(c(nc(c1Br)N)C)Br 9L-902 CN(C)/C=N/C(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 9L-904 c1ccn(c1)c2ccc(cc2CS(=O)(=O)c3ccc(cc3)Cl)C#N 9L-905 CON/C=N/C(=O)c1ccc(c(c1)CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] 9L-907 c1cc(c(c(c1)Cl)Cl)CON/C=N/C(=O)c2ccc(c(c2)CS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] 9L-908 c1ccc(cc1)N2CCN(CC2)C(=O)CON/C=N/C(=O)c3ccc(c(c3)CS(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-] 9L-909 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc(ccc2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 9L-910 COc1cccc(c1)C(=O)Nc2cc(ccc2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F 9L-911 c1cc(c(cc1C(F)(F)F)NC(=O)c2ccc(cc2Cl)Cl)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-912 c1cc(ccc1N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] 9L-913 Cc1ccc(cc1)C(=O)Nc2cccnc2N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-914 c1cc(c(nc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)NC(=O)c4ccc(cc4)F 9L-915 c1cc(c(cc1C(F)(F)F)N)NCCNc2c(cc(cn2)C(F)(F)F)Cl 9L-916 Cc1cc(n2c(c(nc2n1)C(=O)N)C#N)C 9L-917 c1cc(c(nc1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)NC(=O)c4cccs4 9L-918 Cc1cc(n2c(c(nc2n1)C#N)C#N)C 9L-919 Cc1cc(n2cnc(c2n1)C#N)C 9L-920 c1cc(ccc1N)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl.Cl 9L-921 COC(=O)CCCn1c2ccc(cc2nc1S)C(F)(F)F 9L-922 CC1=CC(=Nc2cc(ccc2N1CCNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F)C 9L-923 c1cc(ccc1NC(=O)N)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl 9L-924 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-925 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)F 9L-926 COc1cccc(c1)C(=O)Nc2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-927 c1cc(ccc1NS(=O)(=O)c2ccc(cc2Cl)Cl)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-928 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-929 COc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-930 c1cc2c(cc1C(F)(F)F)ncn2CCNc3c(cc(cn3)C(F)(F)F)Cl 9L-931 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)F 9L-933 c1cc(ccc1C(=O)Nc2cc(ccc2NCCNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F)F 9L-934 Cc1ccc(cc1)C(=O)/C=C\Nc2ccc(cc2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9L-936 c1cc(sc1)C(=O)Nc2cc(ccc2NCCNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F 9L-937 CN(C)C(=C(C#N)C#N)C/C=N/OCc1cccc(c1)F 9M-001 CN(C)C(=C(C#N)C#N)C/C=N/Nc1cccc(n1)Cl 9M-002 COc1ccnc(c1C#N)n2cccc2/C=N/OCc3ccc(cc3)Cl 9M-004 COc1ccnc(c1C#N)n2cccc2/C=N/OCc3c(cccc3Cl)Cl 9M-005 CN(C)C(=C(C#N)C#N)C/C=N/OCCOc1ccccc1 9M-006 Cc1ccc(cc1)CO/N=C/NC(=O)c2c(ccnc2Oc3cccc(c3)C(F)(F)F)OC 9M-008 COc1ccnc(c1C(=O)N/C=N/OCc2cccc(c2)F)Oc3cccc(c3)C(F)(F)F 9M-009 COc1ccnc(c1C(=O)N/C=N/OC)Oc2cccc(c2)C(F)(F)F 9M-010 COc1ccnc(c1C(=O)N/C=N/OCc2ccccc2F)Oc3cccc(c3)C(F)(F)F 9M-011 CN(C)/C=N/C(=O)c1c(ccnc1Oc2ccccc2)OC 9M-012 COc1ccnc(c1C(=O)N/C=N/OCc2ccccc2)Oc3ccccc3 9M-015 COc1ccnc(c1C(=O)N/C=N/OCc2ccccc2F)Oc3ccccc3 9M-016 Cc1c(c(on1)NC(=O)c2ccc(cc2)Cl)Cl 9M-017 Cc1c(c(on1)N(S(=O)(=O)c2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)OC)Cl 9M-018 COc1ccnc(c1c2nc[nH]n2)Oc3ccccc3 9M-019 COc1ccnc(c1C(=O)N/C=N/OC)Oc2ccccc2 9M-020 COc1ccnc(c1C(=O)N/C=N/OCc2ccc(cc2Cl)F)Oc3ccccc3 9M-021 COc1ccnc(c1C(=O)N/C=N/OCc2ccccc2Br)Oc3ccccc3 9M-022 Cc1c(c(on1)N(S(=O)(=O)c2ccc(cc2)Br)S(=O)(=O)c3ccc(cc3)Br)Cl 9M-023 Cc1ccc(cc1)C(=O)N(c2c(c(no2)C)Cl)C(=O)c3ccc(cc3)C 9M-024 CN(C)c1cc[nH]c(=O)c1C#N 9M-025 Cc1c(c(on1)N(S(=O)(=O)c2ccc(c(c2)OC)OC)S(=O)(=O)c3ccc(c(c3)OC)OC)Cl 9M-026 Cc1c(c(on1)NC(=O)c2ccc(c(c2)Cl)Cl)Cl 9M-027 Cc1c(c(on1)NC(=O)c2cccc(c2)C(F)(F)F)Cl 9M-028 Cc1c(c(on1)NC(=O)Nc2ccccc2)Cl 9M-029 CC(=O)C1CC1c2ccc(cc2)OC 9M-030 C/C(=N\OC)/C1CC1c2ccc(cc2)OC 9M-031 Cc1c(c(on1)NC(=O)c2ccc(cc2)F)Cl 9M-032 Cc1c(c(on1)N(S(=O)(=O)c2ccccc2)S(=O)(=O)c3ccccc3)Cl 9M-033 CN(C)c1ccnc(c1C#N)Cl 9M-034 c1ccnc(c1)CNC(=O)N 9M-036 C/C(=N\OCc1ccccc1)/C2CC2c3ccc(cc3)OC 9M-037 c1ccc(cc1)CN2C(=O)C(=O)NC2=O 9M-038 COc1ccccc1CNC(=O)N 9M-039 C/C(=N\O)/C1CC1c2ccc(cc2)OC 9M-041 CCOC(=O)c1c(c2c(ccnc2s1)OC)n3cccc3 9M-042 COc1ccccc1CN2C(=O)C(=O)NC2=O 9M-043 CN(C)c1ccnc(c1C#N)Oc2ccc(cc2)Cl 9M-044 Cc1cccc(c1)Sc2c(c(ccn2)N(C)C)C#N 9M-045 COc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)Cl 9M-046 C/C(=N\OCc1ccc(cc1)F)/C2CC2c3ccc(cc3)OC 9M-047 CCOC(=O)c1c(c2c(ccnc2s1)N(C)C)N 9M-048 C/C(=N\OCc1c(cccc1Cl)Cl)/C2CC2c3ccc(cc3)OC 9M-049 c1cc(cc(c1)Cl)CNC(=O)N 9M-050 Cc1ccc(cc1)CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)Cl 9M-051 COc1ccc(cc1OC)CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)Cl 9M-052 c1cc(cc(c1)C(F)(F)F)CN2C(=O)C(=O)N(C2=O)Cc3ccc(cc3)Cl 9M-053 Cc1cccc(c1)Oc2c3ccc(cc3s(=O)c2c4ccc(cc4)OC)OC 9M-301S Cc1ccc(cc1)Sc2c3ccc(cc3s(=O)c2c4ccc(cc4)OC)OC 9M-302S COc1ccc(cc1)c2c(c3ccc(cc3s2=O)OC)Sc4c(cccc4Cl)Cl 9M-303S COc1ccc(cc1)c2c(c3ccc(cc3s2=O)OC)Sc4ccc(cc4)Br 9M-304S COc1ccc(cc1)c2c(c3ccc(cc3s2=O)OC)Sc4ccc(cc4)F 9M-305S COc1ccc(cc1)c2c(c3ccc(cc3s2=O)OC)Sc4cccc(c4)C(F)(F)F 9M-306S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)Sc3ccc(cc3)Br)C 9M-308S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Br)C 9M-309S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)N3CCOCC3)c4ccccc4 9M-310S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)N3CCN(CC3)C)c4ccccc4 9M-311S CCOC(=O)c1c(nc2n1c(cc(c2)C)C)C 9M-312S COc1ccc(cc1)c2c(c3ccc(cc3s2=O)OC)Oc4ccc(cc4)F 9M-315S COc1ccc(cc1)c2c(c3ccc(cc3s2=O)OC)Oc4ccc(cc4)OC 9M-316S COc1ccc(cc1)c2c(c3ccc(cc3s2=O)OC)Oc4ccc(cc4Cl)Cl 9M-317S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)N3CCN(CC3)Cc4ccccc4)C 9M-322S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)NC)C 9M-323S Cc1cc(nc(c1S(=O)(=O)c2ccc(cc2)Cl)Oc3ccc(cc3)C(C)(C)C)C 9M-324S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2SCc3ccc(cc3)Cl)c4ccccc4)C 9M-326S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Oc3ccc(cc3)C#N)c4ccccc4)C 9M-327S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2N3CCOCC3)c4ccccc4)C 9M-328S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2NC)C)C 9M-335S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2N3CCN(CC3)c4ccccc4F)C)C 9M-336S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2N3CCCCC3)C)C 9M-338S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2N3CCCC3)C)C 9M-339S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Oc3ccc(cc3)C(C)(C)C)C)C 9M-342S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Oc3ccc(cc3)OC)C)C 9M-343S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Oc3cccc(c3C)C)C)C 9M-344S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Oc3cccc(c3)C(F)(F)F)C)C 9M-345S Cc1cc(nc(c1S(=O)(=O)Cc2ccc(cc2)Cl)O)C 9M-346S Cc1c(n2ccccc2n1)C(=O)Nc3ccc(cc3)F 9M-351S Cc1c(n2ccccc2n1)C(=O)Nc3cccc(c3)C(F)(F)F 9M-352S Cc1ccc(cc1C)NC(=O)c2c(nc3n2cccc3)C 9M-353S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2SCc3ccc(cc3)OC)C)C 9M-354S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2S(=O)Cc3ccc(cc3)OC)C)C 9M-355S Cc1ccc(n1c2ccc(cc2)OC)c3ccc(cc3)F 9M-356S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2S(=O)(=O)Cc3ccc(cc3)OC)C)C 9M-358S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2Sc3ccc(cc3)Cl)C)C 9M-359S Cc1ccc(cc1)Sc2c(c(cc(n2)C)C)S(=O)(=O)c3ccc(cc3)C 9M-360S Cc1ccc(cc1)S(=O)c2c(c(cc(n2)C)C)S(=O)(=O)c3ccc(cc3)C 9M-361S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2S(=O)c3ccc(cc3)Cl)C)C 9M-362S CCCNC(=O)c1c(nc2n1cccc2)C 9M-363S CCN(CC)C(=O)c1c(nc2n1cccc2)C 9M-364S Cc1c(n2ccccc2n1)C(=O)N3CCOCC3 9M-365S Cc1ccc(cc1NC(=O)c2c(nc3n2cccc3)C)Cl 9M-367S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2S(=O)(=O)c3ccc(cc3)Cl)C)C 9M-369S Cc1ccc(cc1)S(=O)(=O)c2c(cc(nc2S(=O)(=O)c3ccc(cc3)C)C)C 9M-370S Cc1cc(nc(c1S(=O)(=O)C)Oc2ccccc2OC)c3ccccc3 9M-371S Cc1ccc(n1c2ccc(cc2)Cl)c3ccc(cc3)F 9M-372S Cc1cc(nc(c1S(=O)(=O)C)N2CCN(CC2)C)c3ccccc3 9M-373S Cc1cc(nc(c1S(=O)(=O)C)N(C)C)c2ccccc2 9M-375S Cc1cc(nc(c1S(=O)(=O)C)NC)c2ccccc2 9M-376S Cc1cc(nc(c1S(=O)(=O)C)Oc2ccc(cc2)C(C)(C)C)c3ccccc3 9M-377S Cc1cc(nc(c1S(=O)(=O)C)Oc2cccc(c2)C(F)(F)F)c3ccccc3 9M-378S Cc1c(sc2n1ncn2)/C(=N/OCc3ccccc3)/C 9M-501S CCO/N=C(\C)/c1c(n2c(s1)ncn2)C 9M-502S CCOC(=O)CO/N=C(\C)/c1c(n2c(s1)ncn2)C 9M-504S Cc1c(sc2n1ncn2)/C(=N/OCC=C)/C 9M-505S Cc1cc(n[nH]1)c2ccccc2 9M-508S Cc1c(sc2n1ncn2)/C(=N/OCc3cccc(c3)C(F)(F)F)/C 9M-511S Cc1c(sc2n1ncn2)/C(=N/OCc3ccc(cc3)OC)/C 9M-512S Cc1c(sc2n1ncn2)/C(=N/OCc3ccc(cc3)[N+](=O)[O-])/C 9M-514S CC(=O)Nc1ccc(cc1)OCCF 9M-515S Cc1c(cno1)c2cnc(s2)c3cccc(c3)C(F)(F)F 9M-519S Cc1c(cno1)c2cnc(s2)c3ccccn3 9M-520S CC(=C(C#N)C#N)c1cccc(c1)C(F)(F)F 9M-521S CC(=O)Nc1ccsc1C(=O)O 9M-523S Cc1c(sc2n1ncn2)C(=O)CSc3ccccc3 9M-524S Cc1c(sc2n1ncn2)C(=O)CSCc3cccc(c3)C(F)(F)F 9M-525S Cc1c(sc2n1ncn2)C(=O)CSCc3ccc(cc3)OC 9M-526S Cc1c(sc2n1ncn2)C(=O)CSC3CCCCC3 9M-527S Cc1c(sc2n1ncn2)/C(=N\O)/CSc3ccccc3 9M-529S Cc1c(sc2n1ncn2)/C(=N\O)/CSCc3cccc(c3)C(F)(F)F 9M-530S Cc1c(sc2n1ncn2)/C(=N/OC)/C 9M-536S c1cc(cc(c1)C(F)(F)F)c2ccnc(c2C#N)O 9M-538S CCOc1cnn(c(=O)c1Cl)C 9M-539S c1cc(cc(c1)C(F)(F)F)c2ccnc(c2C#N)Sc3cccc(c3)Cl 9M-542S c1cc(cc(c1)C(F)(F)F)c2ccnc(c2C#N)Sc3ccc(cc3)Br 9M-543S COc1c(c(ccn1)c2cccc(c2)C(F)(F)F)C#N 9M-544S CNc1c(c(ccn1)c2cccc(c2)C(F)(F)F)C#N 9M-545S COC(=O)c1ccccc1Sc2c(c(ccn2)c3cccc(c3)C(F)(F)F)C#N 9M-546S c1cc(ccc1c2cc[nH]c(=O)c2C#N)F 9M-551S CCCNc1c(c(ccn1)c2ccc(cc2)Cl)C#N 9M-552S c1cc(ccc1c2ccnc(c2C#N)NC3CC3)Cl 9M-553S c1ccc(cc1)CNc2c(c(ccn2)c3ccc(cc3)Cl)C#N 9M-554S c1cc(ccc1c2ccnc(c2C#N)Cl)F 9M-555S c1cc(cc(c1)C(F)(F)F)CSc2c(c(ccn2)c3cccc(c3)C(F)(F)F)C#N 9M-558S c1cc(cc(c1)C(F)(F)F)c2ccnc(c2C#N)SCc3ccc(cc3Cl)Cl 9M-559S CCSc1c(c(ccn1)c2ccc(cc2)Cl)C#N 9M-560S COc1c(c(ccn1)c2ccc(cc2)F)C#N 9M-565S CSc1c(c(ccn1)c2ccc(cc2)F)C#N 9M-566S c1cc(ccc1c2ccnc(c2C#N)N3CCOCC3)F 9M-567S c1ccc(cc1)c2ccnc(c2C#N)Oc3ccccc3 9M-568S Cc1c(cno1)c2cn3ccccc3n2 9M-580S Cc1ccn2cc(nc2c1)c3cnoc3C 9M-581S COc1ccc(cc1)Oc2c(c(ccn2)c3ccc(cc3)F)C#N 9M-583S c1ccc(cc1)Oc2c(c(ccn2)c3ccc(cc3)F)C#N 9M-584S COc1cccc(c1)Oc2c(c(ccn2)c3ccccc3)C#N 9M-585S c1cc(ccc1c2ccnc(c2C#N)Sc3ccc(cc3)Br)F 9M-586S c1cc(c(c(c1)Cl)Sc2c(c(ccn2)c3ccc(cc3)F)C#N)Cl 9M-587S Cc1ccc(cc1)Sc2c(c(ccn2)c3ccc(cc3)F)C#N 9M-588S COC(=O)c1ccccc1Sc2c(c(ccn2)c3ccc(cc3)F)C#N 9M-589S CNc1c(c(ccn1)c2ccc(cc2)F)C#N 9M-590S CCCCOc1ccc(cc1)S(=O)(=O)NCC(C)(C)SCc2ccc(cc2)F 9M-702 c1ccc2c(c1)c3c(cco3)c(=O)o2 9M-703 c1cc(ccc1C#Cc2ccc(cc2)N)N 9M-704 c1cc(ccc1CN/C=C/C(=O)c2cc(sc2Cl)Cl)Cl 9M-706 Cc1c(c(=O)ccn1CC(=O)c2ccc(cc2)Cl)Cc3c(cccc3Cl)Cl 9M-707 CC(=O)Nc1ccc(cc1)C#Cc2ccc(cc2)NC(=O)C 9M-708 CC(C)(CNC(=O)c1c(cccc1Cl)Cl)SCc2ccc(cc2)F 9M-709 Cc1c(c(=O)ccn1CCc2ccccc2)Cc3c(cccc3Cl)Cl 9M-710 c1cc(ccc1C#Cc2ccc(cc2)NC(=O)C3CC3)NC(=O)C4CC4 9M-711 CC(C)(CNC(=O)c1cccc(c1)[N+](=O)[O-])SCc2ccc(cc2)F 9M-713 CC(C)C(c1ccoc1)Sc2ccccc2 9M-715 CC(C)(CNC(=O)c1ccc(cc1)F)SCc2ccc(cc2)F 9M-716 CC(C)(CNC(=O)c1ccc(cc1)OC)Sc2c(cc(cn2)C(F)(F)F)Cl 9M-717 Cc1c(c(=O)ccn1CC(C)(C)SCc2ccc(cc2)F)Cc3c(cccc3Cl)Cl 9M-718 CCC(c1ccoc1)Sc2ccccc2 9M-720 Cc1ccc(cc1)n2c(ccn2)c3cc(sc3Cl)Cl 9M-724 Cc1c(c(=O)ccn1Cc2ccccc2Cl)Cc3c(cccc3Cl)Cl 9M-725 Cc1c(c(=O)cc[nH]1)Cc2c(cccc2Cl)Cl 9M-729 c1cc(ccc1N2CC2c3ccncc3)Cl 9M-730 Cc1c(c(=O)ccn1c2ccc(cc2)CC#N)Cc3c(cccc3Cl)Cl 9M-732 CC(=O)C(Cc1ccc(cc1)Cl)C(=O)C 9M-733 Cc1c(c(=O)ccn1C(C)c2ccccc2)Cc3c(cccc3Cl)Cl 9M-734 CC(=O)C(Cc1ccc(cc1)Cl)(Cc2ccc(cc2)Cl)C(=O)C 9M-735 CC(C)C(c1ccoc1)S(=O)c2ccccc2 9M-736 CC(C)C(c1ccoc1)S(=O)(=O)c2ccccc2 9M-738 c1c(cnc(c1Cl)SC(F)F)C(F)(F)F 9M-740 Cc1c(c(=O)ccn1CCCC(=O)O)Cc2c(cccc2Cl)Cl 9M-742 Cc1c(c(=O)ccn1c2cccc(c2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cc4c(cccc4Cl)Cl 9M-743 Cc1c(c(=O)ccn1CCc2ccccn2)Cc3c(cccc3Cl)Cl 9M-745 CC(=O)C(Cc1ccc(cc1)Cl)(Cc2ccc(cc2)Cl)C(=O)/C=C/N(C)C 9M-746 CCC(c1ccoc1)S(=O)c2ccccc2 9M-748 c1ccc(cc1)C(=O)/C=C/c2oc(cc2)/C=C/C(=O)c3ccccc3 9M-900 CC(c1ccoc1)O 9M-902 c1ccc2c(c1)c(=O)n(nn2)c3c(cc(cn3)C(F)(F)F)Cl 9M-903 CC(=O)c1ccoc1 9M-905 c1cc(oc1)/C=C/C(=O)c2ccoc2 9M-906 CN(C)/C=C/c1c(c(=O)n(nc1C(=O)OC)c2ccc(cc2)F)C#N 9M-907 C(C#N)c1c(c(c(c(n1)N)C#N)N)C#N 9M-908 c1ccc2c(c1)c(=O)n(nn2)Cc3ccc(cc3)Br 9M-909 COc1ccc(cc1)N/C=C/c2c(c(=O)n(nc2C(=O)OC)c3ccc(cc3)F)C#N 9M-910 COC(=O)c1c(c(c(=O)n(n1)c2ccc(cc2)F)C#N)/C=C/c3ccco3 9M-913 c1cc(ccc1C(F)(F)F)n2ccc3c(c(=O)n(nc3c2=O)c4ccc(cc4)F)C#N 9M-916 Cc1cc2c(cc1CCc3cc4c(cc3C)OCO4)OCO2 9M-918 COC(=O)c1ccncc1N 9M-919 c1cc(ccc1/C=C/C(=O)c2ccoc2)[N+](=O)[O-] 9M-920 c1ccc2cc(ccc2c1)/C=C/C(=O)c3ccoc3 9M-921 c1ccc(c(c1)/C=C/C(=O)c2ccoc2)F 9M-922 c1cc(cc(c1)C(F)(F)F)/C=C/C(=O)c2ccoc2 9M-923 COc1ccc(cc1)/C=C/C(=O)c2ccoc2 9M-924 c1ccc(cc1)/C=C/C(=O)c2ccoc2 9M-925 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)/C=C/S(=O)(=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl 9N-001 c1c(sc(n1)Cl)CSC2=NCCS2 9N-002 CC(C)c1ccc(cc1)/C=C/S(=O)(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl 9N-003 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3ccc(cc3)F 9N-004 COC(=O)c1c(ccs1)OCc2cnc(s2)Cl 9N-005 c1ccc(cc1)NS(=O)(=O)/C=C/c2ccc3c(c2)OCO3 9N-006 c1cc2cccnc2c(c1)OCc3cnc(s3)Cl 9N-007 Cc1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)OC)Cl 9N-009 COc1ccccc1/C=C/S(=O)(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl 9N-010 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCNCC2 9N-012 c1cncnc1C(=O)O 9N-013 Cc1c(non1)C(=O)C 9N-014 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] 9N-015 c1cc(ccc1Cc2c(cc(cn2)C(F)(F)F)Cl)NC(=O)c3ccc(cc3)I 9N-017 COc1ccc(c(c1)OC)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 9N-018 Cc1ccc(c(c1)C)Oc2ccc(cc2[N+](=O)[O-])C(=O)OC 9N-019 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3ccccn3 9N-020 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Cc3c(cc(cn3)C(F)(F)F)Cl 9N-024 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)c3ccccc3 9N-025 COC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2Cl)Cl 9N-027 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Br 9N-028 COc1ccc(cc1OC)/C=N/NC(=O)c2c(ccs2)OCc3ccc(cc3)F 9N-031 COc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 9N-032 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3ccc(cc3)I 9N-033 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3ccc(cc3)Cl 9N-034 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(c3ccccc3)c4ccccc4 9N-036 c1cc(ccc1N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)O)Cl 9N-037 c1ccc(cc1)/C=N/NC(=O)c2c(ccs2)OCc3ccc(cc3)F 9N-038 Cc1ccc(cc1)/C=N/NC(=O)c2c(ccs2)OCc3ccc(cc3)F 9N-039 c1cc(ccc1COc2ccsc2C(=O)N/N=C/c3ccc(cc3)F)F 9N-040 Cc1ccsc1/C=N/NC(=O)c2c(ccs2)OCc3ccc(cc3)F 9N-041 c1cc(ccc1COc2ccsc2C(=O)N/N=C/c3ccc(cc3)Cl)F 9N-042 c1cc(ccc1COc2ccsc2C(=O)N/N=C/c3ccncc3)F 9N-043 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3c(cccn3)[N+](=O)[O-] 9N-044 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3ccc(c(c3)Cl)Cl 9N-045 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ccc(cc4[N+](=O)[O-])C(=O)O 9N-046 CCOC(=O)C1CCN(CC1)C(=O)OC(C)(C)C 9N-047 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)CC(=O)c3ccc(cc3)c4ccccc4 9N-048 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)C3CC3 9N-049 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 9N-050 Cc1ccc(cc1)COc2ccc(cc2)C(=O)OC 9N-051 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3 9N-052 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)c3ccc(cc3Cl)Cl 9N-053 CC(C)(C)OC(=O)N/N=C/c1ccoc1 9N-054 COC(=O)c1ccc(cc1)OCc2cccc(c2)Cl 9N-055 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC)C 9N-056 Cc1cccc(c1N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC)C 9N-057 c1cc(c(cc1C(=O)O)[N+](=O)[O-])N2CCN(CC2)c3ccc(c(c3)Cl)Cl 9N-058 Cc1ccc(cc1)CN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(=O)OC 9N-060 c1cc2c(cc1CN3CCN(CC3)c4ccc(cc4[N+](=O)[O-])C(=O)O)OCO2 9N-061 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)C(=O)c3cccs3 9N-062 COC(=O)c1ccc(cc1)OCc2ccc(c(c2)Cl)Cl 9N-063 COC(=O)c1ccc(cc1)OCc2cccc(c2)F 9N-064 CCc1ccc(cc1)COc2ccc(cc2)C(=O)OC 9N-065 CC(C)(C)OC(=O)NNCC1CCOC1 9N-066 c1ccc(cc1)C(=O)NC(=S)Nc2ccccc2Oc3ccccc3 9N-068 c1cc[n+](c(c1)SCc2cnc(s2)Cl)[O-] 9N-069 COC(=O)c1ccncn1 9N-070 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)CC(=O)c3ccc(cc3)Br 9N-071 c1cncnc1C(=O)NN 9N-072 Cc1ccc2c(c1)N(C(=O)CCS2)Cc3ccc(cc3)Cl 9N-301S Cc1ccc2c(c1)-c3c(cnc(n3)S)CS2 9N-302S c1ccc(c(c1)CSc2nc3c(c(n2)SCc4ccc(cc4)Cl)CCCC3)Cl 9N-303S CN(C)c1c2c(nc(n1)SCc3ccccc3Cl)CCCC2 9N-304S CN(C)c1c2c(nc(n1)SCc3ccc(cc3)Cl)CCCC2 9N-305S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)Oc4ccc(cc4)F)CCCC3 9N-306S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4ccccc4)CS2 9N-307S Cc1ccc(cc1)CS(=O)(=O)c2nc3c(c(n2)Sc4cccc(c4)OC)CCCC3 9N-308S CC(C)(C)OC(=O)N1CCC(CC1)C2CCNCC2 9N-310S Cc1ccc2c(c1)-c3c(cnc(n3)SC)CS2 9N-311S Cc1ccc2c(c1)-c3c(cnc(n3)SCC=C)CS2 9N-312S Cc1ccc2c(c1)-c3c(cnc(n3)SCC(=O)OC)CS2 9N-313S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4ccc(cc4Cl)Cl)CS2 9N-314S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4ccc(cc4)F)CS2 9N-315S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4ccc(cc4)OC)CS2 9N-316S Cc1ccc2c(c1)-c3c(cnc(n3)SC(C)C)CS2 9N-317S c1cc(ccc1SCCC(=O)O)Cl 9N-320S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4cccc(c4)[N+](=O)[O-])CS2 9N-321S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4cccc(c4)C(F)(F)F)CS2 9N-322S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4ccc(cc4)C(C)(C)C)CS2 9N-323S Cc1cccc(c1)CSc2ncc3c(n2)-c4cc(ccc4SC3)C 9N-324S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4ccc(cc4)Cl)CS2 9N-325S CCSc1ncc2c(n1)-c3cc(ccc3SC2)C 9N-326S CCCSc1ncc2c(n1)-c3cc(ccc3SC2)C 9N-328S Cc1ccc2c(c1)-c3c(cnc(n3)SC(C)C(=O)C)CS2 9N-329S Cc1ccc2c(c1)-c3c(cnc(n3)SCC(=O)C(C)(C)C)CS2 9N-330S Cc1ccc2c(c1)-c3c(cnc(n3)SCCOC)CS2 9N-331S COc1ccc(cc1)/C=C/2\CSc3c(ccs3)C2=O 9N-333S Cc1ccc2c(c1)-c3c(cnc(n3)SCc4c(cccc4Cl)F)CS2 9N-335S c1ccc(cc1)/C=C/2\CSc3c(ccs3)C2=O 9N-348S c1cc(c(cc1Cl)Cl)/C=C/2\CSc3c(ccs3)C2=O 9N-349S c1cc(cc(c1)F)/C=C/2\CSc3c(ccs3)C2=O 9N-350S c1cc(cc(c1)C(F)(F)F)/C=C/2\CSc3c(ccs3)C2=O 9N-351S c1cc(c(cc1/C=C/2\CSc3c(ccs3)C2=O)F)F 9N-354S c1cc(cc(c1)Br)/C=C/2\CSc3c(ccs3)C2=O 9N-355S c1cc(c(cc1Cl)Cl)/C=C/2\CSc3ccc(cc3C2=O)Cl 9N-357S CC(C)(C)c1ccc(cc1)CN2CCSc3c(ccs3)C2=O 9N-358S CO/C=C(\C(=O)OC)/Oc1ccc(cc1Br)Cl 9N-359S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)Cl 9N-360S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)Sc3ccccc3C(=O)OC 9N-361S Cc1ccc(cc1)SC(C)C(=O)NN=C(c2ccccc2)c3ccccc3 9N-362S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)Sc3ccccc3 9N-363S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)Sc3cccc(c3)OC 9N-364S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)Sc3ccc(cc3)Cl 9N-365S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)Sc3c(cccc3Cl)Cl 9N-366S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)Oc3ccc(cc3Cl)Cl 9N-368S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)N3CCOCC3 9N-369S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)N3CCCC3 9N-371S CC(C(=O)NN=C(c1ccccc1)c2ccccc2)NC3CCCCC3 9N-372S c1ccc(c(c1)CN2CCSc3c(ccs3)C2=O)Cl 9N-374S c1cc(c(c(c1)Cl)CN2CCSc3c(ccs3)C2=O)F 9N-375S Cc1cccc(c1)CN2CCSc3c(ccs3)C2=O 9N-376S CCCN1CCSc2c(ccs2)C1=O 9N-377S c1cc2c(cc1Cl)/C(=N/O)/CCS2 9N-378S Cc1ccccc1CN2CCSc3c(ccs3)C2=O 9N-380S c1cc(c(cc1CN2CCSc3c(ccs3)C2=O)Cl)Cl 9N-381S c1cc(c(c(c1)Cl)CN2CCSc3c(ccs3)C2=O)Cl 9N-382S c1cc(cc(c1)Cl)CN2CCSc3c(ccs3)C2=O 9N-383S Cc1ccc(cc1)S(=O)(=O)NN=C(c2ccccc2)c3ccccc3 9N-501S CCOC(=O)CN(N=C(c1ccccc1)c2ccccc2)S(=O)(=O)c3ccc(cc3)C 9N-502S Cc1c2ccccc2nc(c1C(=O)C)N3CCCC3 9N-505S c1ccc(cc1)C(=NNC(=O)CN2CCCCC2)c3ccccc3 9N-507S c1ccc(cc1)C(=NNC(=O)CN2CCCC2)c3ccccc3 9N-508S Cn1c(c(c(n1)C(F)(F)F)C(N2CCOCC2)N3CCOCC3)Cl 9N-511S CN(C)CC(=O)NN=C(c1ccccc1)c2ccccc2 9N-512S CCN(CC)CC(=O)NN=C(c1ccccc1)c2ccccc2 9N-513S CC1CN(CC(O1)C)CC(=O)NN=C(c2ccccc2)c3ccccc3 9N-514S c1ccc(cc1)S(=O)(=O)c2c(nc(s2)N)c3ccc(cc3)Cl 9N-516S c1ccc(cc1)C(=NNC(=O)CN2CCN(CC2)c3ccccc3F)c4ccccc4 9N-517S c1ccc(cc1)C(=NNC(=O)CN2CCN(CC2)c3ncccn3)c4ccccc4 9N-519S CC(=O)Cn1c(=O)c(c(cn1)Cl)Cl 9N-523S CC(=O)Cn1c(=O)c(c(cn1)N2CCOCC2)Cl 9N-524S COc1c(cnc(n1)c2ccccc2)S(=O)(=O)c3ccccc3 9N-566S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2Sc3cccc(c3)C(F)(F)F)c4ccccc4 9N-569S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2Sc3ccc(cc3)F)c4ccccc4 9N-570S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2Sc3ccc(cc3)C(C)(C)C)c4ccccc4 9N-571S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2Oc3ccc(cc3F)F)c4ccccc4 9N-572S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2Oc3ccc(cc3C)Cl)c4ccccc4 9N-573S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2N3CCN(CC3)C)c4ccccc4 9N-574S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2N3CCOCC3)c4ccccc4 9N-575S CCN(CC)c1c(cnc(n1)c2ccccc2)S(=O)(=O)c3ccc(cc3)C 9N-576S Cc1ccc(cc1)S(=O)(=O)c2cnc(nc2Oc3ccc(cc3)NC(=O)C)c4ccccc4 9N-577S CN(C)c1ncc(c(n1)Oc2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)Cl 9N-578S CN(C)c1ncc(c(n1)Sc2ccc(cc2)F)S(=O)(=O)c3ccc(cc3)Cl 9N-579S CCN(CC)c1c(cnc(n1)N(C)C)S(=O)(=O)c2ccc(cc2)Cl 9N-581S COc1ccc(cn1)n2c(=O)cc(c(n2)C(=O)C3CO3)C(F)(F)F 9N-585S CSc1ncc(c(n1)O)S(=O)(=O)c2ccccc2 9N-589S CC(C)Sc1ncc(c(n1)O)S(=O)(=O)c2ccccc2 9N-590S Cc1ccc(cc1)n2c3c(cn2)c(nc(n3)SC)N4CCCC4 9N-643S Cc1ccc(cc1)n2cnn(c2=S)C 9N-645S Cn1c(=S)n(cn1)c2ccc(c(c2)Cl)Cl 9N-646S Cc1ccc(cc1)n2c3c(cn2)c(nc(n3)SC)Oc4ccc5ccccc5c4 9N-647S Cn1c(=S)n(c(n1)C(F)(F)F)c2ccccc2 9N-653S CCSc1nc2c(cnn2c3ccccc3)c(n1)Oc4cccc(c4)C(F)(F)F 9N-656S CCSc1nc2c(cnn2c3ccccc3)c(n1)Oc4ccsc4C(=O)OC 9N-657S c1ccc(cc1)n2c3c(cn2)c(=O)[nH]c(n3)SCC(=O)c4ccc(cc4)Cl 9N-661S c1ccc(cc1)n2c3c(cn2)c(=O)n4c(csc4n3)c5ccc(cc5)Cl 9N-662S COc1ccc(cc1)C(=O)CSc2[nH]c(=O)c3cnn(c3n2)c4ccccc4 9N-663S c1ccc(cc1)C(=O)CSc2[nH]c(=O)c3cnn(c3n2)c4ccccc4 9N-665S c1ccc(cc1)c2csc3n2c(=O)c4cnn(c4n3)c5ccccc5 9N-666S Cc1ccc(cc1)Sc2c3cnn(c3nc(n2)SC)c4ccccc4 9N-673S CSc1nc2c(cnn2c3ccccc3)c(n1)Sc4cccc(c4)C(F)(F)F 9N-675S CSc1nc2c(cnn2c3ccccc3)c(n1)Sc4cc(ccc4Cl)Cl 9N-676S CSc1nc2c(cnn2c3ccccc3)c(n1)Sc4ccc(cc4)F 9N-677S COC(=O)c1ccccc1Sc2c3cnn(c3nc(n2)SC)c4ccccc4 9N-678S CSc1nc2c(cnn2c3ccccc3)c(n1)Sc4ccccc4 9N-679S CSc1nc2c(cnn2c3ccccc3)c(n1)Sc4cccc(c4)Cl 9N-680S CSc1nc2c(cnn2c3ccccc3)c(n1)Sc4ccccc4Cl 9N-682S CSc1nc(c2cnn(c2n1)c3ccccc3)NC4CCCCC4 9N-683S c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)Nc2ccc(cc2)OC(F)(F)F 9N-700 c1ccc(cc1)Cc2c(ccn(c2=O)Cc3ccco3)O 9N-701 COc1ccc(cc1OC)CCNC(=O)c2cccnc2SCCC(=C(F)F)F 9N-702 c1cc(c(nc1)SCCC(=C(F)F)F)C(=O)NN 9N-703 C=CCNc1nc(c(s1)C(=O)c2ccc(cc2)[N+](=O)[O-])N 9N-704 CC(=O)C(Cc1cnc(s1)Cl)(Cc2cnc(s2)Cl)C(=O)C 9N-708 CC(=O)C(Cc1cnc(s1)Cl)C(=O)C 9N-709 COc1ccc(cc1OC)CCn2ccc(c(c2=O)Cc3ccccc3)O 9N-710 C#CCn1ccc(c(c1=O)Cc2ccccc2)O 9N-711 c1ccc(cc1)CCn2ccc(c(c2=O)Cc3ccccc3)O 9N-712 c1ccc(cc1)Cc2c(ccn(c2=O)CCNc3c(cc(cn3)C(F)(F)F)Cl)O 9N-713 CC(=O)Nc1ccc(cc1[N+](=O)[O-])C(=O)O 9N-715 c1ccc2c(c1)nc(o2)c3ccc(cc3)NC(=O)c4ccc(c(c4)Cl)Cl 9N-716 c1ccc(cc1)S(=O)(=O)CCC(C(F)(F)Br)(F)Br 9N-717 c1ccc2c(c1)nc(o2)c3ccc(cc3)NC(=O)c4ccc(cc4Cl)Cl 9N-718 CCOC(=O)C(Cc1ccc(cc1)F)C(=O)C 9N-719 c1ccc2c(c1)nc(o2)c3ccc(cc3)C(F)(F)F 9N-720 c1ccc2c(c1)nc(o2)c3ccc(cc3)NC(=O)c4ccc(cc4)I 9N-721 c1c(c([nH]n1)O)S(=O)(=O)CCC(=C(F)F)F 9N-723 c1ccc(cc1)CNc2c(cccn2)C(=O)O 9N-725 c1ccc2c(c1)nc(o2)c3ccc(cc3)O 9N-726 c1ccc(cc1)C(=O)OCc2cncs2 9N-728 c1ccc2c(c1)nc(o2)c3ccc(cc3)NC(=O)c4cccc(c4Cl)Cl 9N-730 c1ccc(cc1)Cc2c(ccn(c2=O)Cc3ccc4c(c3)OCO4)O 9N-732 c1ccc(cc1)Cc2c(ccn(c2=O)C3CCCCCCC3)O 9N-734 COCCCn1ccc(c(c1=O)Cc2ccc(cc2)F)O 9N-736 c1cc(sc1)C(=O)OCc2cncs2 9N-737 C1CC1(C(=O)O)S(=O)(=O)CCC(=C(F)F)F 9N-738 c1ccc(cc1)CNc2ccc(cc2[N+](=O)[O-])C(F)(F)F 9N-740 COCCNc1ccc(cc1[N+](=O)[O-])C(F)(F)F 9N-741 c1cc(ccc1Cc2c(ccn(c2=O)C3CC3)O)F 9N-742 COc1cccc(c1)Cn2ccc(c(c2=O)Cc3ccc(cc3)F)O 9N-743 Cc1cccc(c1)C(=O)OCc2cncs2 9N-745 c1ccc(c(c1)C(=O)OCc2cncs2)Cl 9N-746 c1cc(ccc1C(=O)OCc2cncs2)C(F)(F)F 9N-747 c1cc(ccc1C(=O)OCc2cncs2)I 9N-750 c1ccc(cc1)/C=C/C(=O)OCc2cncs2 9N-751 c1cc(ccc1Cc2c(ccn(c2=O)Cc3ccc(cc3)F)O)F 9N-752 c1ccnc(c1)CCn2ccc(c(c2=O)Cc3ccc(cc3)F)O 9N-753 c1c(scn1)COC(=O)C2CCCCC2 9N-754 COc1cccc(c1)C(=O)OCc2cncs2 9N-755 c1ccc2c(c1)Nc3c(cccn3)C(=O)N2 9N-757 c1ccc(c(c1)NC(=O)c2cccnc2Cl)O 9N-758 CN1c2ccccc2Nc3c(cccn3)C1=O 9N-759 c1cc(c(nc1)Cl)C(=O)NC2CCCCC2 9N-760 c1ccc(cc1)NC(=O)OCc2cncs2 9N-761 c1cc(ccc1Cc2c(ccn(c2=O)Nc3c(cc(cn3)C(F)(F)F)Cl)O)F 9N-762 c1cc(ccc1Cc2c(ccn(c2=O)Cc3ccc(cc3Cl)Cl)O)F 9N-763 c1cc(ccc1Cc2c(ccn(c2=O)CCc3cnc[nH]3)O)F 9N-764 c1cc(cc(c1)Cl)NC(=O)OCc2cncs2 9N-765 c1cc(ccc1NC(=O)OCc2cncs2)Cl 9N-766 c1ccc(c(c1)NC(=O)OCc2cncs2)Cl 9N-767 Cc1ccc(cc1)NC(=O)OCc2cncs2 9N-769 c1cc(c(cc1NC(=O)OCc2cncs2)Cl)Cl 9N-770 CCOC(=O)C(Cc1ccc(cc1)F)C(=O)C/C=N/OCc2ccc(cc2)C 9N-776 COc1ccc2c(c1)n3ccccc3c2C#N 9N-802 Cc1c(ccc(c1OC)S(=O)Nc2ccc(cc2)OC)OC 9N-803 Cc1c(ccc(c1OC)S(=O)Nc2ccccc2)OC 9N-804 Cc1c(ccc(c1OC)S(=O)NCc2ccccc2)OC 9N-805 Cc1c(ccc(c1OC)S(=O)NC2CCCCC2)OC 9N-806 Cc1c(ccc(c1OC)S(=O)Nc2cccc(c2)C(F)(F)F)OC 9N-807 c1ccn2c(c1)c(c3c2cc(cc3)OCc4cccc(c4)C(F)(F)F)C#N 9N-808 Cc1ccc(cc1)COc2ccc3c(c2)n4ccccc4c3C#N 9N-809 Cc1c(ccc(c1OC)S(=O)N2CCN(CC2)Cc3ccccc3)OC 9N-810 Cc1cc(cc(c1)NS(=O)c2ccc(c(c2OC)C)OC)C 9N-811 CN(C)/C=N\c1c2ccsc2ncn1 9N-812 c1ccc(cc1)CO/N=C/Nc2c3ccsc3ncn2 9N-813 Cc1c(ccc(c1OC)S(=O)N2CCN(CC2)C)OC 9N-814 Cc1c(ccc(c1OC)S(=O)N2CCN(CC2)c3ccccc3F)OC 9N-815 Cc1c(ccc(c1OC)S(=O)Nc2ccc(cc2)Cl)OC 9N-817 Cc1c(ccc(c1OC)S(=O)N2CCN(CC2)c3ccccn3)OC 9N-818 c1ccc(cc1)COc2ccc3c(c2)n4ccccc4c3C#N 9N-819 c1ccn2c(c1)c(c3c2cc(cc3)OCc4cccc(c4)C#N)C#N 9N-820 c1ccn2c(c1)c(c3c2cc(cc3)OCc4ccc(cc4)Br)C#N 9N-821 Cc1c(ccc(c1OC)S(=O)N2CCOCC2)OC 9N-822 Cc1c(ccc(c1OC)S(=O)NCc2ccc(cc2)Cl)OC 9N-823 Cc1c(ccc(c1OC)S(=O)Nc2ccccn2)OC 9N-824 Cc1c(ccc(c1OC)S(=O)NC2CC2)OC 9N-825 Cc1ccc(cc1)Cn2ccnc2/C=C/c3ccc(cc3)Cl 9N-826 Cc1c(ccc(c1OC)S(=O)O)OC 9N-828 Cc1c(ccc(c1OC)S(=O)NCc2ccccc2OC)OC 9N-829 COc1ccc(c(c1)OC)S(=O)N 9N-831 c1ccn2c(c1)c(c3c2cc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)C#N 9N-832 COc1ccc(cc1)NC(=O)COc2ccc3c(c2)n4ccccc4c3C#N 9N-833 c1ccn2c(c1)c(c3c2cc(cc3)OCC(=O)NCc4ccco4)C#N 9N-834 COc1ccc(c(c1)OC)S(=O)Nc2ccc(cc2)Cl 9N-835 COc1ccc(cc1)NS(=O)c2ccc(cc2OC)OC 9N-837 COc1ccc(c(c1)OC)S(=O)NC2CCCCC2 9N-838 COc1ccc(c(c1)OC)S(=O)N2CCOCC2 9N-839 CCOC(=O)/C(=C/c1ccc(cc1)O)/C#N 9N-903 CCOC(=O)/C(=C/c1ccc(cc1)[N+](=O)[O-])/C#N 9N-912 c1cc(ccc1c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N)[N+](=O)[O-] 9N-914 CCOC(=O)/C(=C\c1ccc(c(c1)Cl)Cl)/C#N 9N-915 CCOC(=O)/C(=C/c1ccncc1)/C#N 9N-927 CCOC(=O)/C(=C/c1cccc(c1)C(F)(F)F)/C#N 9N-930 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)/C(=C/C#N)/N 9P-001 c1ccc(c(c1)C#N)Oc2ccccc2F 9P-005 c1cc(cc(c1)Oc2ccc(cc2)c3c(c(c(c(n3)N)C#N)C#N)C#N)C(F)(F)F 9P-006 CC(=O)OCC(C(=O)OC)NC(=O)OCc1ccccc1 9P-008 COC(=O)COc1cccc(c1)C=O 9P-009 CCN(CC)CCOc1ccccc1C=O 9P-011 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)c3c(c(c(c(n3)N)C#N)C#N)C#N 9P-013 c1ccc(cc1)c2cc(c(c(n2)c3ccc(cc3)Oc4ccc(c(c4)F)Cl)C#N)C(F)(F)F 9P-017 CCOC(=O)C(CS)NC(=O)OC(C)(C)C 9P-020 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)C3=C(CCC(=O)N3)C#N 9P-023 c1cc(ccc1C(=O)O)/N=N\c2ccc(c(c2)C=O)O 9P-031 COC(=O)c1cccnc1N 9P-032 Cc1nc2ccccc2c3n1c4ccccc4n3 9P-034 CCc1nc2ccccc2c3n1c4ccccc4n3 9P-039 CCOC(=O)C(CSCCCN1C(=O)c2ccccc2C1=O)NC(=O)OC(C)(C)C 9P-042 c1ccc(cc1)OCc2[nH]c3ccccc3n2 9P-043 c1ccc2c(c1)c3nc4ccccc4n3c(n2)C(F)(F)F 9P-045 Cc1ccc(cc1)S(=O)(=O)N2C=CC3C2CCC(C3=O)Br 9P-046 C/C(=N\NC(=S)N)/c1ccc(cc1)OC 9P-047 C/C(=N\N=C\1/NC(=O)CS1)/c2ccc(cc2)OC 9P-051 C/C(=N\NC(=S)N)/c1ccc(cc1)F 9P-052 C/C(=N/N=C/1\NC(=O)CS1)/c2ccc(cc2)F 9P-060 C/C(=N\NC(=S)N)/c1ccccc1 9P-061 c1cc(ccc1C(=O)N2CCC3(CC2)CO3)Cl 9P-303S Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccccc3 9P-320S Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)Cl 9P-322S Cc1c(c(no1)c2ccccc2)C(=O)Nc3cccc(c3)C(F)(F)F 9P-323S Cc1c(c(no1)c2ccccc2)C(=O)N3CCCCC3 9P-324S CS(=O)(=O)c1c(c(c(s1)C(=O)c2ccccc2)N)C#N 9P-325S Cc1ccc(cc1)SCC2(CCN(CC2)C(=O)c3ccc(cc3)Cl)O 9P-326S Cc1ccc(cc1)Oc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 9P-327S c1ccc(cc1)SCC2(CCN(CC2)C(=O)c3ccc(cc3)Cl)O 9P-332S c1cc(ccc1C(=O)N2CCC(CC2)(CSc3ccc(cc3)Cl)O)Cl 9P-333S c1cc(ccc1C(=O)N2CCC(CC2)(CSc3ccc(cc3Cl)Cl)O)Cl 9P-336S COc1cccc(c1)SCC2(CCN(CC2)C(=O)c3ccc(cc3)Cl)O 9P-337S COc1ccc(cc1)SCC2(CCN(CC2)C(=O)c3ccc(cc3)Cl)O 9P-338S c1cc(ccc1C(=O)N2CCC(CC2)(CSc3ccc(cc3)Br)O)Cl 9P-339S Cc1ccc(cc1)OCC2(CCN(CC2)C(=O)c3ccc(cc3)Cl)O 9P-340S c1cc(c(cc1C(=O)N2CCC(=O)CC2)Cl)Cl 9P-349S c1ccc(cc1)S(=O)(=O)N2CCC(=NO)CC2 9P-354S Cc1cccc(c1)Oc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 9P-358S COC(=O)c1ccc(cc1)COc2ccc(c(c2)O)C=O 9P-359S c1ccc(cc1)C(=O)NN=C2CCN(CC2)S(=O)(=O)c3ccccc3 9P-362S c1ccc(cc1)C(=O)ON=C2CCN(CC2)S(=O)(=O)c3ccccc3 9P-363S CCOC(=O)c1cnc2c(cccc2c1N3CCCC3)C 9P-376S CCOC(=O)c1cnc2c(cccc2c1Nc3ccc(cc3)OC(F)(F)F)C 9P-377S CCOC(=O)c1cnc2c(cccc2c1Nc3ccc(cc3)F)C 9P-378S Cc1cccc2c1ncc3c2[nH]n(c3=O)c4ccccc4 9P-379S c1ccc(cc1)S(=O)(=O)N2CCC(=NNC(=O)c3ccc(cc3)Cl)CC2 9P-381S c1ccc(cc1)S(=O)(=O)N2CCC(=NNC(=O)c3ccc(cc3)F)CC2 9P-382S c1cc(ccc1COc2ccc(c(c2)O)C=O)C(=O)O 9P-383S c1ccc(cc1)S(=O)(=O)N2CCC(=NNC(=O)c3cccc(c3)C(F)(F)F)CC2 9P-384S Cc1ccc(cc1)C(=O)NN=C2CCN(CC2)S(=O)(=O)c3ccccc3 9P-385S c1ccc(cc1)S(=O)(=O)N2CCC(=NNC(=O)c3cccs3)CC2 9P-386S c1ccc(cc1)S(=O)(=O)N2CCC(=NNC(=O)c3ccc(c(c3)Cl)Cl)CC2 9P-388S CCOC(=O)c1cnc2ccc(cc2c1NCc3ccc(cc3)Cl)[N+](=O)[O-] 9P-389S CCOC(=O)c1cnc2ccc(cc2c1NCc3ccc(cc3)C)[N+](=O)[O-] 9P-390S CCOC(=O)c1cnc2ccc(cc2c1NCc3ccc(cc3)OC)[N+](=O)[O-] 9P-391S CCOC(=O)c1cnc2ccc(cc2c1NC(C)C)[N+](=O)[O-] 9P-392S CCOC(=O)c1cnc2ccc(cc2c1NCC=C)[N+](=O)[O-] 9P-393S CCOC(=O)c1cnc2ccc(cc2c1N3CCCC3)[N+](=O)[O-] 9P-394S CCOC(=O)c1cnc2ccc(cc2c1Nc3ccccc3F)[N+](=O)[O-] 9P-395S Cc1cccc(c1C)Oc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 9P-411S c1ccc(cc1)C(=O)c2c(c(c(s2)Oc3ccc4ccccc4c3)C#N)N 9P-412S CC(=O)Nc1ccc(cc1)Oc2c(c(c(s2)C(=O)c3ccccc3)N)C#N 9P-413S c1ccc(cc1)C(=O)c2c(c(c(s2)N3CCOCC3)C#N)N 9P-414S c1cc(c(cc1C(=O)N2CCC(CC2)(CN3CCOCC3)O)Cl)Cl 9P-428S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)CSc4ccc(cc4)Br 9P-504S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)CSc4ccc(cc4)Cl 9P-505S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)CSc4c(cccc4Cl)Cl 9P-506S COC(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 9P-507S COC(=O)c1ccccc1SCC(=O)N2CCC(CC2)c3nc4ccccc4s3 9P-508S c1cc2cc(sc2nc1)C(=O)O 9P-510S c1cc2c(cc1[N+](=O)[O-])cc(s2)C(=O)N3CCOCC3 9P-515S c1cc(ccc1NC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-])Cl 9P-516S CNC(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 9P-517S CN(C)C(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 9P-518S c1cc(ccc1C(F)(F)F)NC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 9P-519S c1ccc2c(c1)nc(s2)C3CCN(CC3)C(=O)CSc4ccc(cc4)F 9P-521S CS(=O)(=O)c1nc2ccsc2c(n1)N3CCOCC3 9P-522S COC(=O)c1cc2cc(ccc2s1)NS(=O)(=O)c3ccc(cc3)F 9P-523S C=CCNC(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 9P-525S CC(C)NC(=O)c1cc2cc(ccc2s1)[N+](=O)[O-] 9P-526S Cc1ccc(cc1Cl)NC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 9P-528S c1cc2c(cc1[N+](=O)[O-])cc(s2)C(=O)Nc3ccc(cc3Cl)Cl 9P-529S COC(=O)c1ccc(cc1)NC(=O)c2cc3cc(ccc3s2)[N+](=O)[O-] 9P-530S Cn1c2c(cc(s2)NC(=O)OCc3ccc(cc3)F)c(n1)C(F)(F)F 9P-571S CC(C)(C)c1ccc(cc1)COC(=O)Nc2cc3c(nn(c3s2)C)C(F)(F)F 9P-572S Cn1c2c(cc(s2)NC(=O)OCc3ccc(cc3)OC)c(n1)C(F)(F)F 9P-573S CC(C)(C)COC(=O)Nc1cc2c(nn(c2s1)C)C(F)(F)F 9P-574S c1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4ccc(cc4)Cl 9P-579S Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)c(=O)c4ccccc4s3 9P-580S c1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4cccs4 9P-581S c1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4cccc(c4)C(F)(F)F 9P-584S c1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4ccc(c(c4)Cl)Cl 9P-585S c1ccc(cc1)C(=O)Nc2ccc3c(c2)c(=O)c4ccccc4s3 9P-588S c1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4ccccc4Cl 9P-589S Cc1cccc(c1)C(=O)Nc2ccc3c(c2)c(=O)c4ccccc4s3 9P-591S c1ccc2c(c1)c(=O)c3cc(ccc3s2)NC(=O)c4cccc(c4)Cl 9P-592S Cc1cccn2c1nc(c2/C=N/OC(=O)c3cccc(c3)C(F)(F)F)c4ccc(cc4)Cl 9P-642S Cc1ccn2c(c1)[nH+]c(c2CN(C)C)c3ccc(cc3)Cl.[Cl-] 9P-643S Cc1cccn2c1nc(c2/C=C(\C#N)/c3ccc(cc3)OC)c4ccc(cc4)Cl 9P-647S Cc1cccn2c1nc(c2/C=C(\C#N)/c3ccc(c(c3)Cl)Cl)c4ccc(cc4)Cl 9P-654S Cc1cccn2c1nc(c2/C=C(\C#N)/c3cccc(c3)OC)c4ccc(cc4)Cl 9P-655S Cc1cccn2c1nc(c2/C=C(\C#N)/c3cccc(c3)Cl)c4ccc(cc4)Cl 9P-656S c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)/C=C(\C#N)/c4cccc(c4)C(F)(F)F 9P-662S COC(=O)c1ccc(nc1)N2CCN(CC2)Cc3ccccc3 9P-667S c1cc(cc(c1)Cl)CSc2nnc(o2)c3cccnc3Sc4ccc(cc4)Cl 9P-668S Cc1ccn2c(c1)nc(c2/C=C(\C#N)/c3cccc(c3)OC)c4ccc(cc4)Cl 9P-674S CC(C)C(C(=O)C)C(=O)c1ccc(cc1)Cl 9P-701 Cc1c(sc(n1)c2ccc(c(c2)OC)OC)C(=O)/C=C/N(C)C 9P-705 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)N 9P-706 Cc1ccccc1NC(=S)NCc2ccccn2 9P-707 Cc1ccccc1NC(=S)NCC=C 9P-708 Cc1ccccc1NC(=S)NCc2ccccc2OC 9P-709 Cc1ccccc1NC(=S)NCc2ccc(cc2)OC 9P-710 Cc1ccc(cc1)CNC(=S)Nc2ccccc2C 9P-711 Cc1ccccc1NC(=S)NCc2cccc(c2)OC 9P-712 c1cc2c(c(c1)I)C(=O)C(=O)N2 9P-718 c1csc2c1c(ncn2)NN 9P-722 c1cnccc1c2[nH]ccn2 9P-723 Cc1c(sc(n1)c2ccc(cc2)Cl)c3cc[nH]n3 9P-724 C/[N+](=C\c1ccc(c(c1O)Cc2ccc(cc2Cl)Cl)O)/[O-] 9P-726 Cc1c(nnn1c2ccc(cc2)OC(F)(F)F)C(=O)c3ccc(cc3)OC 9P-727 Cc1c(c(nc(n1)C)NCc2ccc(cc2)F)I 9P-728 CN(C)/C=C/C(=O)C(Cc1c(cccc1Cl)F)C(=O)c2cn(nn2)c3ccc(cc3)OC(F)(F)F 9P-731 CC(=O)C(Cc1ccc(cc1)Cl)Cc2ncc(s2)Cl 9P-733 c1cc(ccc1/C=N/Nc2c3ccsc3ncn2)F 9P-734 Cc1cc(c(n1c2ccc(cc2)C(=O)O)C)C=O 9P-735 COc1ccc(cc1)n2cc(nn2)C(=O)c3cccc(c3)Oc4c(cc(cn4)C(F)(F)F)Cl 9P-736 CC(C(=O)c1cn(nn1)c2ccc(cc2)OC(F)(F)F)n3cncn3 9P-737 Cc1c(c(nc(n1)C)NN)I 9P-741 Cc1c(sc(n1)c2ccncc2)c3cc[nH]n3 9P-742 Cc1cc(ccc1OC(C)C(=O)c2cn(nn2)c3ccc(cc3)OC(F)(F)F)Cl 9P-743 COc1ccc(cc1)n2cc(nn2)C(=O)c3ccccn3 9P-745 c1ccc2cc(ccc2c1)C(=O)c3cn(nn3)c4c(cc(cn4)C(F)(F)F)Cl 9P-746 CC1(OC(=O)[C-](C(=O)O1)C(c2ccccc2)C(C#N)C(=C(C#N)C#N)N)C.C[NH+]1CCOCC1 9P-748 c1ccc(cc1)SC2CN(N(C2)C=O)C=O 9P-749 CC(C(=O)c1cn(nn1)c2ccc(cc2)OC(F)(F)F)Oc3ccc(cc3F)F 9P-750 COC(=O)Nc1cccc(c1)SC 9P-751 CCOC(=O)c1ccc(cc1)n2cc(nn2)C(=O)c3ccc(cc3Cl)Oc4ccc(cc4)Cl 9P-753 Cc1c(c(nc(n1)C)NCc2cccs2)I 9P-754 CCOC(=O)c1ccc(cc1)n2cc(nn2)C(=O)C(Cc3ccc(cc3Cl)Cl)C(=O)OCC 9P-755 CCOC(=O)c1ccc(cc1)n2cc(nn2)C(=O)c3ccc(cc3)n4ccnc4 9P-756 c1cc(cc(c1)n2ccnc2)C=O 9P-759 CCOC(=O)c1ccc(cc1)n2cc(nn2)C(=O)c3cccnc3 9P-760 c1ccc2c(c1)CCN(C2)Cc3cnc(s3)Cl 9P-900 c1cc(cc(c1)NC(=O)N(Cc2ccc(cc2)Cl)CC(C(F)(F)F)O)C(F)(F)F 9P-904 CC(C)(C)OC(=O)n1cc(c2c1cccc2)C=O 9P-905 CCOC(=O)C1CCN(CC1)C(=O)C(F)(F)Cl 9P-906 c1c(sc(n1)Cl)CN2CCSCC2 9P-909 CC1CN(CC(O1)C)Cc2cnc(s2)Cl 9P-910 Cn1cc2cccc(c2n1)[N+](=O)[O-] 9P-912 COc1cccc2c1oc(c2)C(=O)c3ccccc3 9P-913 CC1CC(=CC(=O)C1C(=O)OC)O 9P-914 c1cc(ccc1C(=O)Nc2ncc(cn2)Cl)Cl 9P-915 C/C(=C\C(=O)C(F)(F)F)/NC(CO)c1ccccc1 9P-916 Cc1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)C=O 9P-917 C/C(=N\O)/c1cc2cccc(c2o1)OC 9P-922 COc1cccc2c1oc(c2)/C(=N/O)/c3ccccc3 9P-923 C/C(=N\NC(=O)c1ccco1)/c2cc3cccc(c3o2)OC 9P-924 c1c(cn2c(c1Cl)nnc2C(F)(F)Cl)C(F)(F)F 9P-926 c1ccc(cc1)N2CCN(CC2)Cc3cnc(s3)Cl 9P-927 CCOC(=O)C(F)(F)Sc1nc2ccccc2s1 9P-928 CC(=O)c1ccc(c2c1cc(o2)C#N)OC 9P-930 c1cc(nn2c1nnc2C(F)(F)Cl)Cl 9P-932 c1cc(nn2c1nnc2C(C(C(F)(F)F)(F)F)(F)F)Cl 9P-933 Cc1c(ccc2c1cn[nH]2)[N+](=O)[O-] 9P-934 Cc1ccc(cc1)C(=O)Nc2ncc(cn2)Cl 9P-939 c1cc(sc1)C(=O)Nc2ncc(cn2)Cl 9P-940 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cn[nH]3)c4ccc(cc4)Cl 9P-942 c1ccc2c(c1)cccc2NNC(=S)N 9P-944 c1ccc2c(c1)c(c[nH]2)CCNC3=C(C(=O)c4ccccc4C3=O)Cl 9P-946 CC(=O)c1ccc(c2c1cc(o2)C(=O)O)OC 9P-947 COc1cc(c(c(c1)Br)O)C=O 9P-948 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnn3C(=O)c4cccc(c4)OC)c5ccc(cc5)Cl 9P-949 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnn3C(=O)c4ccc(cc4)I)c5ccc(cc5)Cl 9P-950 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnn3C(=O)c4ccc(cc4)C)c5ccc(cc5)Cl 9P-951 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnn3C(=O)c4cccc(c4)C(F)(F)F)c5ccc(cc5)Cl 9P-952 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnn3C(=O)c4cccc(c4)Cl)c5ccc(cc5)Cl 9P-953 C/C(=N\NC(=O)c1ccc(cc1)C(F)(F)F)/c2cc3cccc(c3o2)OC 9P-954 c1c(cn2c(c1Cl)nnc2C(F)F)C(F)(F)F 9P-955 c1ccc(cc1)CNC2=C(C(=O)c3ccccc3C2=O)Cl 9P-956 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnc(n3)SCc4ccccc4)c5ccc(cc5)Cl 9P-961 CC(=O)c1cc2cc(cc(c2o1)Br)OC 9P-962 CC(=O)c1cc2cc(cc(c2o1)Br)Br 9P-963 COc1cc(c(c(c1)Br)O)/C=N/NC(=O)c2ccc(cc2)C(F)(F)F 9P-964 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnc(n3)SCc4ccc(cc4)C(F)(F)F)c5ccc(cc5)Cl 9P-965 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnc(n3)SCc4ccc(cc4)[N+](=O)[O-])c5ccc(cc5)Cl 9P-966 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/c2cc3cccc(c3o2)OC 9P-967 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnc(n3)SCc4cccc(c4)C#N)c5ccc(cc5)Cl 9P-969 Cc1cc(c(cc1[N+](=O)[O-])C)N 9P-970 CCCc1ccc(c(c1)F)c2ccc(cc2)c3c(cnc(n3)SCc4cc(cc(c4)C)C)c5ccc(cc5)Cl 9P-971 c1cc(ccc1c2cc(nn2c3nc(c(s3)Br)c4ccc(cc4)Br)Br)F 9R-0003 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3cccs3)Br 9R-0005 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3cccs3)Cl 9R-0006 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccco3)Br 9R-0007 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2Cl)Cl)C(=O)O 9R-0008 CC1=C(C(C(=C(N1)C)C(=O)O)c2ccc(cc2)F)C(=O)C 9R-0009 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccc(o3)Cl)Cl 9R-0010 Cc1c(c2nc(cc(n2n1)c3cccs3)C(F)(F)F)Cl 9R-0011 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)c5ccccc5)C 9R-0012 CC1=C(C(C(=C(N1)C)C(=O)O)c2ccc(cc2)[N+](=O)[O-])C(=O)C 9R-0013 CCOC(=O)c1c(cc(cn1)C(=O)C)C(=O)OC 9R-0014 Cc1c(c2nccc(n2n1)c3ccc(cc3Cl)Cl)Br 9R-0015 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5cnc6n(c5=O)c7ccccc7s6)C 9R-0019 Cc1c(c2nccc(n2n1)c3ccccc3)Br 9R-0020 Cc1c(c2ncc(c(n2n1)C(F)(F)F)C#N)Br 9R-0021 Cc1ccc(cc1)c2ccnc3n2nc(c3Cl)C 9R-0022 Cc1ccc(cc1)c2ccnc3n2nc(c3Br)C 9R-0023 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc(c(c5)CS(=O)(=O)c6ccc(cc6)Cl)[N+](=O)[O-])C 9R-0024 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5ccc(c(c5)[N+](=O)[O-])Cl)C 9R-0025 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5cnc6n(c5=O)ccs6)C 9R-0026 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)O)NC(=O)c5ccccc5)C 9R-0027 CCOC(=O)CN/C=C(\C#N)/c1ccc(cc1)F 9R-0028 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)c5cnc6n(c5=O)CCS6)C 9R-0029 Cc1ccc(n1c2ccsc2c3cc4nccc(n4n3)C(F)(F)F)C 9R-0030 CCOC(=O)/C(=C\Nc1cc(n[nH]1)c2c(ccs2)n3c(ccc3C)C)/C(=O)C(F)(F)F 9R-0032 Cc1ccc(n1c2ccsc2c3cc4nc(ccn4n3)C5=CNC6N(C5=O)CCS6)C 9R-0033 Cc1ccc(n1c2ccsc2c3cc4nc(cc(n4n3)O)CS(=O)(=O)c5ccccc5)C 9R-0034 COC(=O)C(Cc1ccccc1)(Cc2ccccc2)C#N 9R-0037 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccco3)Cl 9R-0038 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CCC(=O)OC 9R-0039 Cc1cc([nH]n1)/N=C/c2c3ccccc3[nH]c2Cl 9R-0040 Cc1cc(n(n1)c2nc(cs2)c3c(ccs3)Br)C 9R-0041 Cc1cc2nccc(n2n1)c3ccc(c(c3)[N+](=O)[O-])Cl 9R-0042 Cc1c(c2nccc(n2n1)c3ccccn3)Cl 9R-0043 Cc1cc2nccc(n2n1)c3ccccn3 9R-0044 Cc1cc2ncc(c(n2n1)N)c3ccc(cc3)F 9R-0045 Cc1cc(n(n1)c2c(c(nc(n2)C)C)I)C 9R-0046 c1cc(c(cc1c2cc([nH]n2)N)Cl)Cl 9R-0047 Cc1ccc(n1c2ccsc2c3cc4ncc(c(n4n3)C)C(=O)Nc5ccsc5C(=O)OC)C 9R-0048 c1ccc(cc1)S(=O)(=O)n2ccc(c2)C(=O)CCC(=O)O 9R-0053 c1cc(c(nc1)N2CCCC2)[N+](=O)[O-] 9R-0201 Cc1ccccc1Cn2ccc(c(c2=O)C#N)c3cccs3 9R-0202 CC1=NCCN1S(=O)(=O)c2ccc(cc2)Cl 9R-0203 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2ccc(cc2)C 9R-0204 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2ccncc2 9R-0205 c1cc(ccc1C(=O)N2CCC(=NC=C2)C(F)(F)F)Cl 9R-0207 c1cc(cc(c1)F)Cn2ccc(c(c2=O)C#N)c3ccco3 9R-0208 CC(C)(C)c1ccc(cc1)Cn2ccc(c(c2=O)C#N)c3ccco3 9R-0209 Cc1c(sc(n1)Nc2cccc(c2)C(F)(F)F)C(=O)C 9R-0210 c1ccc(cc1)/C(=C\c2cccs2)/C(=O)Nc3[nH]nnn3 9R-0211 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5ccc(c(c5)Cl)Cl 9R-0212 COc1cc2c(cc1OC)N=C(N3C2=NC(=O)C3CC4CCCCC4)SCc5cnc(s5)Cl 9R-0213 CC1=[NH+]CCN1S(=O)(=O)c2ccc(cc2)Cl.[I-] 9R-0214 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCCc2ccccn2 9R-0215 CCC(CC)C(=O)c1cc([nH]c1)C(=O)N2CCN(CC2)c3ccc(cc3)OC 9R-0216 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN=C(C=C3)C(F)(F)F 9R-0217 Cc1c(sc(n1)Nc2ccccc2C(F)(F)F)C(=O)C 9R-0218 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCCOC 9R-0219 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCC2CCCO2 9R-0220 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2ccccn2 9R-0221 c1cc(ccc1C(=O)N2CCN=C(C=C2)C(F)(F)F)[N+](=O)[O-] 9R-0222 c1ccc(c(c1)N2CCN(CC2)C(=O)c3cc(ccc3[N+](=O)[O-])Cl)F 9R-0223 C/C(=[NH+]/c1cc(c(c(c1)OC)OC)OC)/N(C)CCNS(=O)(=O)c2ccc(cc2)Cl.[I-] 9R-0225 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCCN(C)C 9R-0226 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)C(CC)CC 9R-0227 CCC(CC)C(=O)c1cc([nH]c1)C(=O)OC 9R-0228 C/C(=[NH+]/c1ccc(cc1)F)/N(C)CCNS(=O)(=O)c2ccc(cc2)Cl.[I-] 9R-0229 Cc1cc(cc(c1)/[NH+]=C(/C)\N(C)CCNS(=O)(=O)c2ccc(cc2)Cl)C.[I-] 9R-0230 CN1CCN(CC1)c2c(cccn2)[N+](=O)[O-] 9R-0231 C/C(=[NH+]/c1ccc(cc1)OC)/N(C)CCNS(=O)(=O)c2ccc(cc2)Cl.[I-] 9R-0233 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cc(ccc3[N+](=O)[O-])Cl 9R-0234 c1cc(ccc1CNC(=O)c2cc(ccc2[N+](=O)[O-])Cl)Cl 9R-0235 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 9R-0236 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCCc3ccccn3 9R-0237 CCC(CC)C(=O)c1cc([nH]c1)C(=O)NCc2cccs2 9R-0238 CCC(CC)C(=O)c1cc([nH]c1)C(=O)N2CCN(CC2)c3ccccc3F 9R-0239 CCC(CC)C(=O)c1cc([nH]c1)C(=O)N2CCN(CC2)c3ccccc3 9R-0240 CCC(CC)C(=O)c1cc([nH]c1)C(=O)O 9R-0241 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCCCN(C)C 9R-0243 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCc3cccc(c3)C(F)(F)F 9R-0244 c1ccc(cc1)/C=C/Cn2ccc(c(c2=O)C#N)c3cccs3 9R-0247 c1cc(c(cc1Cl)C(=O)NCC2CCCO2)[N+](=O)[O-] 9R-0249 C/C(=[NH+]/c1cccc(c1)OC)/N(C)CCNS(=O)(=O)c2ccc(cc2)Cl.[I-] 9R-0250 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCc3ccccc3 9R-0252 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCc3ccco3 9R-0253 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCCOC 9R-0254 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)c2ccccc2C 9R-0255 c1cc(c(cc1Cl)C(=O)NCCCn2ccnc2)[N+](=O)[O-] 9R-0256 CC(=O)N(C)CCNS(=O)(=O)c1ccc(cc1)Cl 9R-0257 CCC(CC)C(=O)c1cc([nH]c1)C(=O)N 9R-0258 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)OC 9R-0259 COc1ccc(cc1Cl)CNC(=S)Nc2ccccc2 9R-0260 c1ccc2c(c1)ccc3c2cc(o3)C(=O)NN 9R-0261 C#CCOc1ccccc1C=O 9R-0262 c1cc(c(cc1N2CCCC2)C(=O)N)[N+](=O)[O-] 9R-0263 CC1=NCCN1S(=O)(=O)c2ccc(cc2)NC(=O)C 9R-0264 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)NCc3ccncc3 9R-0266 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)NCCc3ccccn3 9R-0267 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)NCCCN3CCOCC3 9R-0268 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3 9R-0269 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)NCc3ccco3 9R-0270 c1cc(ccc1N2C(=O)C3C4C=CC(C3C2=O)O4)Cl 9R-0271 COc1ccc(cc1Cl)C/N=C\2/N(C(=O)CS2)c3ccccc3 9R-0272 CC(=O)c1cnc(s1)Nc2ccccc2C(F)(F)F 9R-0273 c1c(cc(c(c1C=O)O)C=O)C=O 9R-0275 COC(=O)c1cc(c[nH]1)C(=O)Cc2ccccc2 9R-0276 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCc3ccccc3OC 9R-0277 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCC3CCCO3 9R-0278 C#CCOc1ccccc1CO 9R-0279 COC(=O)c1ccc(cc1)Oc2c(cccn2)N 9R-0280 Cc1ccc(cc1)S(=O)(=O)c2cn(c(=O)[nH]2)C 9R-0281 c1cc([nH]c1)C(=O)NCCCN2CCOCC2 9R-0283 c1cc(cc(c1)Sc2ccc(cc2N)C#N)C(F)(F)F 9R-0284 c1ccc(cc1)CC(=O)c2cc([nH]c2)C(=O)O 9R-0285 c1ccc(cc1)S(=O)(=O)c2c[nH]c(=O)[nH]2 9R-0286 CC(=O)c1cc([nH]c1)C(=O)C(Cl)(Cl)Cl 9R-0288 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)N3CCN(CC3)c4ccccc4F 9R-0289 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCCCn3ccnc3 9R-0290 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCc3ccc(cc3)F 9R-0291 Cc1ccc(cc1)S(=O)(=O)Cc2c([nH]c(=O)[nH]2)C 9R-0292 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)O 9R-0294 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)N 9R-0295 C/C(=[NH+]/c1ccc(c(c1)Cl)OC)/N(C)CCNS(=O)(=O)c2ccc(cc2)Cl.[I-] 9R-0299 C/C(=[NH+]/c1ccccc1OC)/N(C)CCNS(=O)(=O)c2ccc(cc2)Cl.[I-] 9R-0300 C#CCOc1ccccc1/C=C/C(=O)O 9R-0301 c1ccc(cc1)NC(=O)Nc2cc(ccc2Sc3cccc(c3)C(F)(F)F)C#N 9R-0302 CC(=O)c1cc([nH]c1)C(=O)NCCCN(C)C 9R-0303 CC(=O)c1cc([nH]c1)C(=O)NCCCOC 9R-0304 CC(=O)c1cc([nH]c1)C(=O)NCC2CCCO2 9R-0305 C#CCOc1ccc(cc1C=O)Cl 9R-0306 c1cc(cc(c1)Sc2ccc(cc2[N+](=O)[O-])C#N)C(F)(F)F 9R-0307 CC(=O)c1cc([nH]c1)C(=O)NCc2ccccc2OC 9R-0308 CC(=O)c1cc([nH]c1)C(=O)NCc2ccccc2Cl 9R-0309 CC(=O)c1cc([nH]c1)C(=O)NCc2cccc(c2)C(F)(F)F 9R-0310 CC(=O)c1cc([nH]c1)C(=O)NCc2ccc(cc2)OC 9R-0311 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)/N=C/N(C)C 9R-0312 Cc1ccc(c(c1)C)N2CCN(CC2)C(=O)c3cc(c[nH]3)C(=O)c4ccccc4C 9R-0313 CC1=C(C(CC(=O)N1)c2ccc(cc2)F)C(=O)C 9R-0314 c1ccc(c(c1)NC(=O)Nc2cc(ccc2Sc3cccc(c3)C(F)(F)F)C#N)Cl 9R-0315 C#CCOc1ccccc1/C=N/O 9R-0316 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)N3CCN(CC3)Cc4ccccc4 9R-0318 CCC(C)NC(=O)c1ccc[nH]1 9R-0319 COc1ccc(cc1)CNC(=O)c2ccc[nH]2 9R-0320 c1cc(ncc1[N+](=O)[O-])N2CCOCC2 9R-0322 Cc1ccc(cc1)S(=O)(=O)c2c[nH]c(=O)[nH]2 9R-0323 Cc1ccccc1C(=O)c2cc([nH]c2)C(=O)NCc3cccs3 9R-0324 c1ccc2c(c1)ccc3c2cc(o3)C(=O)O 9R-0325 c1c(cnc(c1Cl)NCCN2C(=O)C3C4C=CC(C3C2=O)O4)C(F)(F)F 9R-0326 COc1ccc(cc1Cl)CNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F 9R-0327 COc1ccc(cc1Cl)CNC(=S)Nc2ccc(cc2F)Br 9R-0328 COc1ccc(cc1Cl)CNC(=S)NCC=C 9R-0330 COc1ccc(cc1Cl)CNC(=O)c2ccc[nH]2 9R-0331 c1cc(cc(c1)N2C(=O)C3C4C=CC(C3C2=O)O4)C(F)(F)F 9R-0332 CCn1cc([nH]c1=O)S(=O)(=O)c2ccc(cc2)C 9R-0333 Cn1cc(n(c1=O)C)S(=O)(=O)c2ccccc2 9R-0334 CC(=O)c1ccc(cc1)OCC#C 9R-0335 c1cc([nH]c1)C(=O)NCC2CCCO2 9R-0337 COc1cc2c(cc1OC)nc(n(c2=N)Cc3cccs3)SCc4ccc(cc4Cl)Cl 9R-0338 CC(=O)c1cc([nH]c1)C(=O)NCc2ccccc2 9R-0339 CCC(C)NC(=O)c1cc(c[nH]1)C(=O)C 9R-0340 c1ccc(cc1)CN2C(=O)C3C4C=CC(C3C2=O)O4 9R-0341 c1cc([nH]c1)C(=O)NCc2ccc(cc2)F 9R-0342 c1cc(cc(c1)C(F)(F)F)CNC(=O)c2ccc[nH]2 9R-0343 c1ccc(c(c1)CNC(=O)c2ccc[nH]2)Cl 9R-0344 Cc1ccc(cc1)CNC(=O)c2ccc[nH]2 9R-0345 Cn1cc(cc1C(=O)O)C(=O)c2cccc(c2Cl)Cl 9R-0349 c1ccc2c(c1)ccc3c2cc(o3)C(=O)N4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl 9R-0350 CCc1c([nH]c(=O)[nH]1)C(C)S(=O)(=O)c2ccc(cc2)C 9R-0351 c1ccc2c(c1)ccc3c2cc(o3)C(=O)NCc4ccccc4Cl 9R-0352 c1ccc2c(c1)ccc3c2cc(o3)C(=O)NCCCn4ccnc4 9R-0353 CCn1cc(n(c1=O)Cc2ccccc2C)S(=O)(=O)c3ccc(cc3)C 9R-0355 c1ccc(cc1)CCCOC(=O)NC2=C(C(=O)c3ccccc3C2=O)Cl 9R-0356 Cc1ccc(cc1)S(=O)(=O)Cc2c(n(c(=O)n2C)C)C 9R-0357 c1ccc2c(c1)ccc3c2cc(o3)C(=O)NCCCN4CCOCC4 9R-0358 CCn1c(c([nH]c1=O)CS(=O)(=O)c2ccccc2)C 9R-0359 CC(C)(C)n1cc([nH]c1=O)S(=O)(=O)c2ccccc2 9R-0360 Cc1ccc(cc1)S(=O)(=O)c2cn(c(=O)[nH]2)C(C)(C)C 9R-0361 c1ccc(c(c1)CO/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])F 9R-0362 c1ccc(cc1)c2c3c(c(c(n2)O)C#N)CCCC3 9R-0364 CC1=[N+](CCN1S(=O)(=O)c2ccc(cc2)F)C.[I-] 9R-0365 c1cc(ccc1CO/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])F 9R-0366 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)CCc3ccccn3 9R-0367 CCc1c([nH]c(=O)n1C(C)(C)C)C(C)S(=O)(=O)c2ccccc2 9R-0369 c1cc(ccc1NC(=O)N)OC(F)(F)F 9R-0371 c1c(c[nH]c1C(=O)C(Cl)(Cl)Cl)C(=O)C2CC2 9R-0372 C/C(=[NH+]\Cc1ccccc1Cl)/N(C)CCNS(=O)(=O)c2ccc(cc2)F.[I-] 9R-0373 c1cc(c(c(c1)Cl)F)CO/N=C\2/CCCCC2c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] 9R-0374 c1cn(cn1)CCCNC(=O)c2cc(c[nH]2)C(=O)C3CC3 9R-0375 COc1ccc(cc1Cl)Cn2c(=N)c3cc(c(cc3[nH]c2=S)OC)OC 9R-0376 COc1cc2c(cc1OC)[nH]c(=S)n(c2=N)Cc3ccco3 9R-0377 c1cnccc1CNC(=O)c2cc(c[nH]2)C(=O)C3CC3 9R-0378 COc1ccc(cc1)CNC(=O)c2cc(c[nH]2)C(=O)C3CC3 9R-0379 CC1=NCCN1S(=O)(=O)c2ccc(cc2)F 9R-0380 c1ccc2c(c1)C(C(OC2=O)c3ccc(cc3Cl)Cl)C(=O)O 9R-0381 c1ccc(c(c1)CNC(=O)c2cc(c[nH]2)C(=O)C3CC3)Cl 9R-0382 c1c(c[nH]c1C(=O)NCCCN2CCOCC2)C(=O)C3CC3 9R-0383 c1cc(ccc1CNC(=O)c2cc(c[nH]2)C(=O)C3CC3)F 9R-0384 Cc1ccc(cc1)CSc2nc3cc(c(cc3c(=N)n2Cc4ccc(c(c4)Cl)OC)OC)OC 9R-0385 COc1ccc(cc1Cl)Cn2c(=N)c3cc(c(cc3nc2SCc4cccc(c4)C(F)(F)F)OC)OC 9R-0386 Cc1ccc(c(c1)CSc2nc3cc(c(cc3c(=N)n2Cc4ccc(c(c4)Cl)OC)OC)OC)C 9R-0387 Cc1ccccc1CSc2nc3cc(c(cc3c(=N)n2Cc4ccc(c(c4)Cl)OC)OC)OC 9R-0388 Cc1ccc(cc1)NC(=O)NC(CC(=O)OC)c2cccc(c2)[N+](=O)[O-] 9R-0603 c1c2cn[nH]c2ncc1NC(=S)N 9R-0605 c1cc(sc1)C(CC(=O)O)NC(=O)C(F)(F)F 9R-0606 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc(c1)Br 9R-0607 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccccc1Br 9R-0608 c1ccc(c(c1)C(=O)N(c2nccc(n2)c3cccs3)C(=O)c4ccccc4Cl)Cl 9R-0609 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccsc1 9R-0610 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc2c(c1)OCO2 9R-0611 c1cc(sc1C(CC(=O)O)NC(=O)C(F)(F)F)Br 9R-0612 Cc1ccc(cc1)C(CC(=O)O)N2Cc3ccccc3C2=O 9R-0613 Cc1ccccc1C(CC(=O)O)N2Cc3ccccc3C2=O 9R-0614 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccc(cc3)O 9R-0615 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)c3ccsc3 9R-0616 CSc1ccc(cc1)C(CC(=O)O)N2Cc3ccccc3C2=O 9R-0617 c1ccc(cc1)N2CCN(CC2)Cc3cnc(s3)N4CCOCC4 9R-0619 c1cc(ccc1C(CC(=O)O)N)[N+](=O)[O-] 9R-0620 COC(=O)CC(c1cccc(c1)F)NC(=O)Nc2cccc(c2)Cl 9R-0621 Cc1ccc(cc1)C(=O)NC(CC(=O)OC)c2ccc3c(c2)OCO3 9R-0622 Cc1ccc(cc1)NC(=O)Nc2nccc(n2)c3cccs3 9R-0624 COC(=O)CC(c1ccc(cc1)O)N2Cc3ccccc3C2=O 9R-0625 c1cc(sc1)C(CC(=O)O)N2CCS(=O)(=O)CC2 9R-0626 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1)SC 9R-0627 COC(=O)CC(c1ccccc1Cl)NS(=O)(=O)c2cccs2 9R-0629 CN1CCN(CC1)Cc2cnc(s2)N3CCOCC3 9R-0630 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1)O 9R-0631 Cc1c(cccc1F)NC(=O)C 9R-0632 CC1CN(CC(O1)C)Cc2cnc(s2)N3CCOCC3 9R-0633 c1cc(ccc1N2CCN(CC2)Cc3cnc(s3)N4CCOCC4)F 9R-0634 c1ccc2c(c1)cccc2C(CC(=O)O)N 9R-0635 Cc1ccc(o1)C(CC(=O)O)N 9R-0637 c1ccc2c(c1)CN(C2=O)C(CC(=O)NN)c3ccc(cc3)O 9R-0638 Cc1c(ccc(c1NC(=O)C)[N+](=O)[O-])F 9R-0639 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1)[N+](=O)[O-] 9R-0640 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc(c1)O 9R-0641 c1ccc(cc1)C(=O)NC(=S)Nc2nccc(n2)c3cccs3 9R-0642 Cc1c(ccc(c1N)[N+](=O)[O-])F 9R-0643 c1cc(c2cn[nH]c2c1[N+](=O)[O-])F 9R-0644 c1cc(c2cn[nH]c2c1NC(=S)N)F 9R-0647 c1ccc(cc1)COc2ccc(c3c2cn[nH]3)[N+](=O)[O-] 9R-0648 c1cc(cc(c1)NC(=O)Nc2nccc(n2)c3cccs3)C(F)(F)F 9R-0652 COC(=O)CC(c1ccc(cc1)OC(=O)c2ccco2)N3Cc4ccccc4C3=O 9R-0654 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(CC(=O)OC)N3Cc4ccccc4C3=O 9R-0655 c1ccc(cc1)COC(=O)NC(CC(=O)O)c2cccs2 9R-0656 CC(C)(C)OC(=O)NC(CC(=O)O)c1ccc(cc1)OC 9R-0657 COc1ccc(cc1OC)C(CC(=O)OC)NC(=O)c2cccs2 9R-0658 CC(C)c1ccc(cc1)C(CC(=O)OC)NC(=O)c2ccco2 9R-0659 Cc1ccc(cc1Cl)NC(=O)C 9R-0661 CC(C)(C)OC(=O)NC(CC(=O)O)c1cccc2c1cccc2 9R-0662 COC(=O)/C=C/c1ccc2c(c1)OCO2 9R-0663 COC(=O)c1ccc(c(c1)N)S(=O)(=O)c2ccccc2 9R-0664 c1ccc(cc1)N2CCN(CC2)Cc3cnc(s3)Oc4ccc(cc4)Br 9R-0665 Cc1ccc(cc1)C(CC(=O)O)NC(=O)OCc2ccccc2 9R-0666 COC(=O)c1ccc(c(c1)N)N2CCN(CC2)c3ccccc3 9R-0667 c1cc(c(c(c1)Cl)C2CC(=O)CC(=O)C2n3cncn3)F 9R-0801 c1ccc2c(c1)CCNC2C3=C(C(C(CC3=O)c4c(cccc4Cl)F)n5cncn5)O 9R-0802 COc1ccc(cc1)C2CC(=O)C(C(=O)C2c3c(cc(cn3)C(F)(F)F)Cl)C4c5ccccc5CCN4 9R-0803 CN(C)/C=C/C(=O)c1cnc(s1)c2ccncc2 9R-0805 CN(C)/C=C/C(=O)c1cnc(s1)c2cccs2 9R-0806 COC(=O)c1c(ccs1)n2cc(nn2)C(=O)c3ccc(cc3)F 9R-0807 c1ccc(cc1)c2cn(nn2)c3ccc(cc3)[N+](=O)[O-] 9R-0809 c1ccc2c(c1)c(c([nH]2)Cl)C=O 9R-0810 c1cc(ccc1C2CC(=O)CC(=O)C2n3cncn3)Cl 9R-0811 CCCCCCCC[n+]1ccc(cc1)c2nc(c(s2)C(=O)/C=C\Nc3ccc(cc3)C)C.[Br-] 9R-0812 CCCCCCCC[n+]1ccc(cc1)c2nc(c(s2)C(=O)/C=C\Nc3ccc(cc3)OC)C.[Br-] 9R-0813 COc1ccc(c(c1OC)OC)c2[nH]c3c(n2)cccn3 9R-0814 Cc1c(sc(n1)c2cccc(c2Cl)Cl)c3ccn[nH]3 9R-0815 c1cnccc1c2ncc(s2)c3ccnc(n3)N 9R-0816 c1cc(sc1)c2ncc(s2)c3ccnc(n3)N 9R-0817 Cc1c(sc(n1)N(c2cccc(c2)C(F)(F)F)C(=O)C)C(=O)C 9R-0818 c1cc(sc1)c2ncc(s2)c3ccn[nH]3 9R-0819 Cc1cc2nc(c(cn2n1)c3ccc(c(c3)OC)OC)C 9R-0831 CCn1c(nnc1SCc2ccc(cc2)C(=O)OC)COc3ccc(=O)n(n3)c4ccccc4 9R-1000 CCn1c(nnc1SCc2ccccc2)COc3ccc(=O)n(n3)c4ccccc4 9R-1001 CCn1c(nnc1SCc2cccc(c2)OC)COc3ccc(=O)n(n3)c4ccccc4 9R-1002 CCn1c(nnc1SCc2ccccc2C)COc3ccc(=O)n(n3)c4ccccc4 9R-1003 CCn1c(nnc1SCc2ccc(cc2)C(C)(C)C)COc3ccc(=O)n(n3)c4ccccc4 9R-1004 c1ccc(cc1)n2c(=O)ccc(n2)OCc3nnc(o3)S 9R-1009 Cc1ccc(n1c2ccccc2C#N)C 9R-1012 Cc1cc(c(n1c2ccccc2C#N)C)C(=O)C(=O)Nc3ccccc3 9R-1013 Cc1cc(c(n1c2ccccc2C#N)C)C(=O)C(=O)Nc3ccc(cc3)C(C)C 9R-1018 Cc1ccc(n1c2ccc(cc2)N3CCOCC3)C 9R-1020 Cc1cc(c(n1c2ccc(cc2)N3CCOCC3)C)C(=O)C(=O)N4CCC5(CC4)OCCO5 9R-1022 Cc1ccc(cc1)C(=O)NCc2ccccc2n3c(ccc3C)C 9R-1023 Cc1ccc(n1c2ccccc2CNC(=O)c3ccc(cc3)C(F)(F)F)C 9R-1024 c1ccc(cc1)C(=O)CSc2nnc(s2)S 9R-1060 C(CF)CSc1nnc(s1)S 9R-1061 CCO/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1064 c1ccc2c(c1)c(c[nH]2)CCNCCC(C(F)(F)Cl)O 9R-1065 C1CN(CCC12OCCO2)/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1066 c1ccc2c(c1)CCN(C2)/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1067 c1ccc(cc1)CN2CCN(CC2)/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1068 c1cc(cnc1)CN/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1069 C1CCCN(CC1)/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1070 CN(Cc1ccccc1)/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1072 C1CCN(CC1)/C=C/C(=O)C(C(F)(F)F)(F)F 9R-1073 c1ccc2c(c1)c(c[nH]2)CCNCCC(C(F)(F)F)O 9R-1074 COc1ccc(cc1)C2c3c(nc[nH]3)CCN2 9R-1075 c1cc(cnc1)CN/C=C(/C(=O)C(F)(F)F)\Br 9R-1078 c1ccc2c(c1)cc3cc(sc3n2)c4nnc(o4)SCCCF 9R-1122 COc1ccc(cc1)C(=O)c2cc3cc4ccccc4nc3s2 9R-1126 CC(C)(C)C(=O)c1cc2cc3ccccc3nc2s1 9R-1127 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)Cl)Cl 9R-1128 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3Cl)Cl)Cl 9R-1133 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)F)Cl 9R-1134 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)S(=O)(=O)c3ccccc3)Cl 9R-1137 Cc1ccc(cc1)S(=O)(=O)N(Cc2c(nn(c2Cl)C)C(F)(F)F)c3ccc(cc3)OC 9R-1138 Cc1ccc2c(c1)C(=O)C(CS2)[NH3+].[Cl-] 9R-1140 Cn1c(c(c(n1)C(F)(F)F)CNc2ccc(cc2)Cl)OC 9R-1141 Cc1ccc(cc1)C(=O)NC2CSc3ccc(cc3C2=O)C 9R-1147 Cc1ccc2c(c1)C(=O)C(CS2)NS(=O)(=O)c3ccc(cc3)Cl 9R-1148 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)OC)Cl 9R-1149 Cn1c(c(c(n1)C(F)(F)F)CN(c2ccc(cc2)OC)S(=O)(=O)c3cc(cc(c3)Cl)Cl)Cl 9R-1150 Cc1ccc2c(c1)C(=O)C(CS2)NC(=O)c3ccc(cc3Cl)Cl 9R-1151 Cc1ccc2c(c1)C(=O)C(CS2)NC(=O)c3cccc(c3)C(F)(F)F 9R-1153 Cc1ccc2c(c1)C(=O)C(CS2)NC(=O)c3ccc(cc3)F 9R-1154 Cc1ccc2c(c1)/C(=N/OS(=O)(=O)c3ccc(cc3)OC)/CCS2 9R-1155 Cc1ccc(cc1)S(=O)(=O)O/N=C/2\CCSc3c2cc(cc3)C 9R-1156 Cc1ccc2c(c1)/C(=N/OS(=O)(=O)c3ccc(cc3)Cl)/CCS2 9R-1157 Cc1ccc2c(c1)/C(=N/OS(=O)(=O)c3ccccc3)/CCS2 9R-1158 Cc1ccc2c(c1)/C(=N/OS(=O)(=O)C)/CCS2 9R-1159 Cc1ccc2c(c1)C(=O)C(CS2)NS(=O)(=O)c3ccc(cc3)OC 9R-1161 c1ccc\2c(c1)CCC/C2=N\OS(=O)(=O)c3ccc(cc3)Cl 9R-1162 Cc1ccc2c(c1)C(=O)C(CS2)NC(=O)c3ccc(c(c3)Cl)Cl 9R-1163 Cc1cccc(c1)C(=O)NC2CSc3ccc(cc3C2=O)C 9R-1164 Cc1ccc(cc1)S(=O)(=O)O/N=C/2\CCCc3c2cccc3 9R-1165 c1ccc(cc1)S(=O)(=O)O/N=C/2\CCCc3c2cccc3 9R-1169 CS(=O)(=O)O/N=C/1\CCCc2c1cccc2 9R-1170 COc1ccc(cc1)S(=O)(=O)O/N=C/2\CCCc3c2cccc3 9R-1171 c1cc(cc(c1)Cl)n2c(=O)c(c(c(n2)C(=O)O)O)I 9R-1173 c1ccc\2c(c1)CCC/C2=N\OC(=O)c3ccc(cc3)F 9R-1174 Cc1ccc(cc1)C(=O)NC2CCc3ccccc3C2=O 9R-1175 c1cc(c(cc1NC(=O)CN2CCCCC2)F)N3CCOCC3 9R-1180 CN1CCN(CC1)c2ccc(cc2F)NC(=O)CN3CCOCC3 9R-1181 CN1CCN(CC1)CC(=O)Nc2ccc(c(c2)F)N3CCOCC3 9R-1182 CN1CCN(CC1)c2ccc(cc2F)NC(=O)CN3CCCCC3 9R-1183 CN1CCN(CC1)c2ccc(cc2F)NC(=O)CN3CCNCC3 9R-1184 CN1CCN(CC1)CC(=O)Nc2ccc(c(c2)F)N3CCN(CC3)C 9R-1185 CN1CCN(CC1)c2ccc(cc2F)NC(=O)CN3CCN(CC3)C(c4ccccc4)c5ccccc5 9R-1186 c1cc(ccc1C(=O)Nc2cc(ccc2N3CCCCC3)Cl)F 9R-1197 Cc1cccc(c1)C(=O)Nc2cc(ccc2N3CCCCC3)Cl 9R-1198 Cc1ccc(cc1)C(=O)Nc2cc(ccc2N3CCCCC3)Cl 9R-1199 c1cc(c(cc1C(=O)Nc2cc(ccc2N3CCCCC3)Cl)Cl)Cl 9R-1200 c1cc(sc1)C(=O)Nc2cc(ccc2N3CCCCC3)Cl 9R-1201 c1cc(c(cc1C(=O)Nc2cc(ccc2N3CCOCC3)Cl)Cl)Cl 9R-1205 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2cc(ccc2N3CCOCC3)Cl 9R-1206 CN1CCN(CC1)c2ccc(cc2NC(=O)c3ccc(c(c3)Cl)Cl)Cl 9R-1208 CN1CCN(CC1)c2ccc(cc2NC(=O)c3cccc(c3)[N+](=O)[O-])Cl 9R-1209 Cc1ccc(cc1)S(=O)OCC(=O)Nc2cc(ccc2N3CCOCC3)Cl 9R-1211 c1ccc(cc1)S(=O)OCC(=O)Nc2cc(ccc2N3CCOCC3)Cl 9R-1212 CN1CCN(CC1)c2ccc(cc2NC(=O)c3ccc(cc3)Cl)Cl 9R-1213 Cc1ccc(cc1)C(=O)Nc2cc(ccc2N3CCN(CC3)C)Cl 9R-1214 c1cc(c(cc1Cl)Cl)C(=O)Nc2cc(ccc2N3CCCCCC3)Cl 9R-1223 CCn1c(nnc1S)COc2cccc(c2)C(F)(F)F 9R-1242 CCn1c(nnc1SCc2ccc(cc2)Cl)COc3cccc(c3)C(F)(F)F 9R-1243 CCn1c(nnc1SCc2ccc(cc2)C)COc3cccc(c3)C(F)(F)F 9R-1244 CCn1c(nnc1S(=O)(=O)Cc2ccc(cc2)Cl)COc3cccc(c3)C(F)(F)F 9R-1245 c1cc(ccc1C(=O)N2CCC(=O)CC2)F 9R-1246 CCn1c(nnc1SCc2ccc(c(c2)Cl)Cl)COc3cccc(c3)C(F)(F)F 9R-1247 CCn1c(nnc1SC)COc2cccc(c2)C(F)(F)F 9R-1248 CCn1c(nnc1SCC(=O)N)COc2cccc(c2)C(F)(F)F 9R-1251 CCn1c(nnc1S(=O)(=O)Cc2ccc(cc2)C)COc3cccc(c3)C(F)(F)F 9R-1252 CCn1c(nnc1S(=O)Cc2ccc(cc2)Cl)COc3cccc(c3)C(F)(F)F 9R-1253 c1ccc(cc1)c2nc3ccsc3c(n2)Sc4ccccc4 9R-1304 CCOC(=O)CSc1nc(c2ccsc2n1)O 9R-1308 COc1cccc(c1)Sc2c3c(ccs3)nc(n2)c4ccccc4 9R-1310 c1ccc(cc1)c2nc3ccsc3c(n2)Sc4ccc(cc4)F 9R-1311 COC(=O)c1ccccc1Sc2c3c(ccs3)nc(n2)c4ccccc4 9R-1312 CCOC(=O)CSc1[nH]c(=O)c2c(n1)ccs2 9R-1314 c1csc2c1c(=O)[nH]c(n2)NN 9R-1316 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2c(ccs2)NC(=O)c3ccccc3 9R-1318 c1cc(ccc1C(=O)Nc2ccsc2C(=O)NC3CCCCC3)F 9R-1320 c1ccc(cc1)CNC(=O)c2c(ccs2)NC(=O)c3ccc(cc3)F 9R-1321 CSc1nc(c2ccsc2n1)N3CCOCC3 9R-1322 CSc1nc(c2ccsc2n1)N3CCCC3 9R-1323 CCN(CC)c1c2ccsc2nc(n1)SC 9R-1324 CSc1nc(c2ccsc2n1)NC3CCCCC3 9R-1325 CSc1nc2c(ccs2)c(n1)Sc3ccccc3 9R-1326 COC(=O)c1ccccc1Sc2c3ccsc3nc(n2)SC 9R-1327 CSc1nc(c2ccsc2n1)Oc3ccccc3 9R-1328 CSc1nc(c2ccsc2n1)Oc3ccc4ccccc4c3 9R-1329 CC(C(=O)NCc1ccc(cc1)Cl)n2c3ccccc3nc2C(F)(F)F 9R-1366 CC(C(=O)NCc1ccccc1Cl)n2c3ccccc3nc2C(F)(F)F 9R-1367 Cc1ccc(cc1)CNC(=O)C(C)n2c3ccccc3nc2C(F)(F)F 9R-1368 CC(C(=O)NCc1ccc(cc1)OC)n2c3ccccc3nc2C(F)(F)F 9R-1369 c1c(cc(cc1C#N)F)C#N 9R-1378 Cc1cc(nc(n1)Nc2ccc(cc2)OC)C 9R-1425 c1cc(ccc1C#N)OCC(CN2CCN(CC2)c3ccc(cc3)F)O 9R-1426 c1cc(ccc1C#N)OCC(CN2CCOCC2)O 9R-1427 c1ccc(c(c1)/C=C/2\C(=O)NC(=O)S2)F 9T-0001 COC(=O)C(c1ccc(cn1)[N+](=O)[O-])C(=O)OC 9T-0002 c1c2c(cc3c1OCO3)C(=O)NCC2[NH3+].[Cl-] 9T-0005 COC(=O)CC(c1ccc2c(c1)OCO2)NS(=O)(=O)c3cccs3 9T-0007 COc1ccc(cc1)S(=O)(=O)NC(CC(=O)OC)c2ccc3c(c2)OCO3 9T-0008 COC(=O)CC(c1ccc2c(c1)OCO2)NS(=O)(=O)c3cc(ccc3Cl)Cl 9T-0009 CCCCCC(=O)NC(CC(=O)OC)c1ccc2c(c1)OCO2 9T-0010 COC(=O)CC(c1ccc2c(c1)OCO2)NC(=O)C3CC3 9T-0011 CCOC(=O)c1cnc2c(c1Oc3cc(nc(n3)C)C)cnn2C 9T-0013 c1ccc(cc1)S(=O)(=O)/C(=C\c2cccc(c2)OCc3cnc(s3)Cl)/C#N 9T-0014 CC(c1ccc(cc1)[N+](=O)[O-])C(=O)NN 9T-0018 c1cc(ccc1/C=C/C(=O)O)OCc2cnc(s2)Cl 9T-0020 CC(c1ccc(cn1)[N+](=O)[O-])(C(=O)OC)C(=O)OC 9T-0021 c1cc(sc1)c2ccn[nH]2 9T-0024 COC(=O)CC(c1ccc2c(c1)OCO2)NC(=S)NCC=C 9T-0027 COC(=O)c1ccccc1N2CCS(=O)(=O)CC2 9T-0028 Cc1ccc(cc1)NC(=S)NC(CC(=O)OC)c2ccc3c(c2)OCO3 9T-0029 CC(C)(C)NC(=O)NC(CC(=O)OC)c1ccc2c(c1)OCO2 9T-0030 COC(=O)CC(c1ccc2c(c1)OCO2)NC(=O)Nc3ccccc3F 9T-0031 COC(=O)CSc1nccc(n1)c2cc3c4ccccc4ccc3o2 9T-0033 c1ccc2c(c1)ccc3c2cc(o3)c4ccnc(n4)SCC#N 9T-0034 Cc1cc(cc(c1N)Cl)[N+](=O)[O-] 9T-0036 Cc1cc(cc(c1N)Br)[N+](=O)[O-] 9T-0037 Cc1cc(cc(c1N)[N+](=O)[O-])Br 9T-0039 CCC(c1ccc(cc1)[N+](=O)[O-])(C(=O)OC)C(=O)OC 9T-0040 CCc1ccc(cn1)[N+](=O)[O-] 9T-0042 CCOC(=O)C(C)(c1ccc(c(c1)F)[N+](=O)[O-])C(=O)OCC 9T-0043 CC(C)C(CC(=O)O)N1Cc2ccccc2C1=O 9T-0044 c1ccc2c(c1)CN(C2=O)C(CC(=O)O)C3CCC=CC3 9T-0046 CCC(CC)C(CC(=O)O)N1Cc2ccccc2C1=O 9T-0047 CCC(C)C(CC(=O)O)N1Cc2ccccc2C1=O 9T-0048 Cc1ccc(cc1)C(=O)/C=C/c2cc(c(c(c2)OC)OC)OC 9T-0049 Cc1ccc(cc1C)NC(=O)c2ccccc2N3CCS(=O)(=O)CC3 9T-0051 COc1cccc(c1O)/C=C/2\C(=O)NC(=O)S2 9T-0055 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)[N+](=O)[O-])C(=O)O 9T-0056 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)[N+](=O)[O-] 9T-0059 c1csc2c1C(CC2=O)N.Cl 9T-0060 c1ccc(cc1)CC2C(=O)NC(=O)S2 9T-0061 CCC(=O)c1ccc(cc1O)Br 9T-0062 CC(c1ccc(cc1)[N+](=O)[O-])C(=O)N/N=C/c2cccn2c3ccc(cc3)OC(F)(F)F 9T-0064 COC(=O)CC(c1cccc(c1)F)NC(=O)CCl 9T-0065 CCOC(=O)c1cnc2c(c1Oc3ccc(cc3)OC)cnn2C 9T-0067 c1cc2c(cc1N3C(=O)C=CC3=O)NC(=O)CO2 9T-0200 c1cc(ccc1S(=O)(=O)n2ccc(n2)C3CC3)Cl 9T-0201 CC(C)(C)c1ccc(cc1)S(=O)(=O)n2ccc(n2)C3CC3 9T-0202 Cc1cc(c(c(c1)C)S(=O)(=O)n2ccc(n2)C3CC3)C 9T-0203 COc1cccc(c1)N2CCN(CC2)C(=O)Nc3ccc4c(c3)NC(=O)CO4 9T-0204 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccc5c(c4)NC(=O)CO5 9T-0205 Cc1c(c(=O)n2c([nH]1)c(cn2)c3ccc(c(c3)OC)OC)CCO 9T-0206 c1c2c(cc(c1Cl)Cl)n3c(n2)SCC3=O 9T-0207 c1ccc(cc1)C(C(=O)Nc2nccs2)N3CCCCC3 9T-0208 Cc1ccc(cc1)CNC(=O)C(c2ccccc2)NC(=O)c3c(nn(c3Cl)C)C 9T-0210 c1cc(sc1)c2ccn3c(c2C#N)nc(n3)c4cccs4 9T-0211 Cc1ccc(cc1)/C(=N/Nc2c(cc(cc2Cl)Cl)Cl)/C 9T-0213 c1ccc2c(c1)[nH]c(=O)o2 9T-0220 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3cccs3 9T-0221 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3c(cccc3F)F 9T-0223 CCC(=O)N1CCN(CC1)Cc2ccccc2 9T-0224 COc1ccc(cc1)S(=O)(=O)n2ccc(n2)C3CC3 9T-0225 c1ccc2cc(ccc2c1)S(=O)(=O)n3ccc(n3)C4CC4 9T-0226 Cc1c(c(=O)n2c([nH]1)ncn2)CCOC(=O)c3ccco3 9T-0228 Cc1ccc(cc1)Cn2ccc(n2)C3CC3 9T-0230 c1cc2c(cc1F)c(=O)c(c[nH]2)C(=O)O 9T-0233 c1ccc(c(c1)CN)N2CCC(CC2)CO 9T-0234 CCCCCC1CCC(CC1)C(=O)NN 9T-0235 c1cc(oc1)c2ccn3c(c2C#N)nc(n3)c4ccc(cc4Cl)Cl 9T-0236 c1ccc(c(c1)C(=O)Nc2ccc3c(c2)NC(=O)CO3)C(=O)O 9T-0238 COc1ccc(cc1)NC(=O)OC 9T-0247 CCOC(=O)C1CCN(CC1)c2ccc(nn2)Cl 9T-0248 Cc1c(c(n2c(n1)ncn2)Cl)CCCl 9T-0249 Cc1c(c(=O)n2c([nH]1)c(cn2)C#N)CCOC(=O)C3CCCCC3 9T-0251 CCc1ccc(cc1)c2[nH]c(=O)c(c(n2)C)CCO 9T-0253 Cc1c(c(=O)n2c([nH]1)c(cn2)C#N)CCOC(=O)c3ccc(cc3Cl)Cl 9T-0256 Cc1c(c(n2c(n1)c(cn2)c3ccc(c(c3)OC)OC)Cl)CCCl 9T-0260 c1ccc2c(c1)C(=O)N(C2=O)c3ccc4c(c3)NC(=O)CO4 9T-0261 c1cc(cc(c1)C(F)(F)F)c2nc3c(c(ccn3n2)c4ccco4)C#N 9T-0263 COc1ccc2c(c1)C=C(CO2)C=O 9T-0266 Cc1ccc(cc1)CN/C(=C(/C=C/C(=O)OC)\C(=O)OC)/C 9T-0267 c1cc(ccc1S(=O)(=O)n2ccc(n2)C3CC3)Br 9T-0268 c1cc(ccc1S(=O)(=O)n2ccc(n2)C3CC3)I 9T-0269 c1ccn(c1)c2ccc3c(c2)N(C(=O)CO3)Cc4ccc(cc4Cl)Cl 9T-0270 Cc1ccc(cc1)Cn2c(c(cc2C(=O)OC)C(=O)OC)C 9T-0272 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)C=O 9T-0276 CCN(CC)C(c1ccccc1)C(=O)Nc2nccs2 9T-0277 COc1ccc(cc1OC)c2cnn3c2nc(cc3)c4ccc(cc4)Cl 9T-0278 Cc1c2c(n3c(n1)c(cn3)c4ccc(c(c4)OC)OC)N(CC2)Cc5ccc(cc5)OC 9T-0279 CC(=O)Nc1ccc(cc1)S(=O)(=O)n2ccc(n2)C3CC3 9T-0282 COc1ccc(cc1OC)c2cnn3c2nc-4c(c3)C(c5c4cc6c(c5)OCO6)NC(=O)C(F)(F)F 9T-0285 Cn1cc(c(n1)C(F)(F)F)C(=O)NCCCC(=O)NCc2ccccc2 9T-0286 Cn1cc(c(n1)C(F)(F)F)C(=O)NCCCC(=O)N2CCCC2 9T-0287 Cc1c(c(n(n1)C)Cl)C(=O)NCC(=O)Nc2ccc(cc2)OC 9T-0288 Cc1c(c(n(n1)C)Cl)C(=O)NCC(=O)NCc2ccccc2 9T-0289 C/C(=N\O)/C(/C(=N/O)/C)Cc1ccc(cc1)O 9T-0292 c1cc(ccc1CN)OCCCCCOc2ccc(cc2)CN 9T-0293 c1cc(ccc1Cn2ccc(n2)C3CC3)Cl 9T-0294 COc1ccc(cc1OC)c2cnn3c2nc(cc3)c4ccccc4O 9T-0295 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)C=C(C#N)C#N 9T-0296 c1ccc(cc1)C(C(=O)Nc2nccs2)N3CCCC3 9T-0298 c1ccc(cc1)c2ccc(cc2)c3c(cn(n3)c4ccccc4)/C=C/C(=O)O 9T-0300 c1ccc(cc1)C(C(=O)Nc2nccs2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl 9T-0301 Cn1c(=O)c2c(n(c1=O)C)OC(C2=O)/C=N/OCCOc3cccc(c3)C(F)(F)F 9T-0303 Cn1c(c(cn1)c2ccc(c(c2)OC)OC)NC(=O)c3ccccc3C(=O)O 9T-0304 Cc1cn2c(c(cn2)c3ccc(c(c3)OC)OC)nc1c4ccc5c(c4)ccc(c5Br)OC 9T-0305 c1ccc(cc1)CN2CCN(CC2)C(c3ccccc3)C(=O)Nc4nccs4 9T-0307 Cc1ccc(cc1)CNC(c2ccccc2)C(=O)Nc3nccs3 9T-0308 COc1ccc(cc1)CNC(c2ccccc2)C(=O)Nc3nccs3 9T-0309 COc1ccc2c(c1)C=C(CO2)C=C3C(=O)c4ccccc4C3=O 9T-0310 Cn1c(c(cn1)c2ccc(c(c2)OC)OC)N3C(=O)c4ccccc4C3=O 9T-0312 COc1ccc(cc1OC)c2cnn3c2nc(cc3)c4ccc(cc4)n5ccc(=O)cc5 9T-0313 COc1ccc(cc1)/C(=C(/c2ccc(cc2)OC)\Cl)/C=O 9T-0314 CC(C)c1ccc(cc1)NC(c2ccccc2)C(=O)Nc3nccs3 9T-0317 Cc1c(c(=O)n2c3ccccc3nc2[nH]1)CCOC(=O)c4ccc(cc4)F 9T-0321 Cc1c(c(n(n1)C)Cl)C(=O)NC(c2ccccc2)C(=O)N3CCOCC3 9T-0322 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)n2ccc(n2)C3CC3 9T-0323 c1cc(c(c(c1)Cl)Cn2ccc(n2)C3CC3)Cl 9T-0326 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccccc3Cl)SCCc4ccccc4 9T-0327 CC(C)(C)c1ccc(cc1)CSc2nc3cc(c(cc3c(=N)n2Cc4ccccc4Cl)OC)OC 9T-0328 COc1cc2c(cc1OC)nc(n(c2=N)Cc3ccccc3Cl)SCc4ccc(cc4Cl)Cl 9T-0329 CCCCCCCCN1CCc2c1n3c(c(cn3)c4ccc(c(c4)OC)OC)nc2C 9T-0330 Cc1c(c(n(n1)C)Cl)C(=O)NCC(=O)N2CCOCC2 9T-0331 Cc1cccc(c1NC(=O)CNC(=O)c2c(nn(c2Cl)C)C)C 9T-0332 Cc1c(c(n(n1)C)Cl)C(=O)NC(c2ccccc2)C(=O)Nc3ccc(cc3)C(C)C 9T-0334 Cc1c(c(c2c(n1)-c3ccccc3C2=O)C4=Cc5cc(ccc5OC4)OC)C#N 9T-0336 Cc1c2c(n3c(n1)c(cn3)C#N)SCC2 9T-0337 Cc1c2c(n3c(n1)c(cn3)C#N)N(NCC2)C 9T-0338 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)S(=O)(=O)c3ccccc3)N)C 9T-0606 C=Cc1ccc(cc1)[N+](=O)[O-] 9T-0616 Cc1c(oc(n1)c2ccc(cc2)F)C(=O)C 9T-0617 Cc1cc(n(n1)CC(=O)c2cccc(c2)N)C 9T-0803 CC(=O)c1c(cc(cn1)C(F)(F)F)N2CCOCC2 9T-0809 C/C(=N\OC)/c1c(cc(cn1)C(F)(F)F)N2CCOCC2 9T-0810 C/C(=N\OCc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)N3CCOCC3 9T-0812 CC(=O)c1c(cc(cn1)C(F)(F)F)N2CCN(CC2)c3ccc(cc3)Cl 9T-0818 C/C(=N\OCc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)N3CCCC3 9T-0819 C/C(=N\OC)/c1c(cc(cn1)C(F)(F)F)N2CCCC2 9T-0820 C/C(=N\O)/c1c(cc(cn1)C(F)(F)F)N2CCCC2 9T-0822 C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/c2c(cc(cn2)C(F)(F)F)N3CCOCC3 9T-0823 Cn1cc(c2c1cccc2)C(=O)N3CCOCC3 9T-1481 Cn1cc(c2c1cccc2)C(=O)NCc3ccccc3 9T-1482 CCn1cc(c2c1cccc2)C(=O)C(F)(F)F 9T-1483 COC(=O)c1cn(c2c1cccc2)S(=O)(=O)c3ccccc3 9T-1484 CCn1cc(c2c1cccc2)C(=O)O 9T-1486 CCn1cc(c2c1cccc2)C(=O)NCc3ccccc3 9T-1488 CCn1cc(c2c1cccc2)C(=O)N3CCCCC3 9T-1489 CCn1cc(c2c1cccc2)C(=O)N3CCOCC3 9T-1490 COCc1cc(nc(n1)c2ccncc2)O 9T-1493 CNC(=O)c1cn(c2c1cccc2)C 9T-1495 Cn1cc(c2c1cccc2)C(=O)N3CCCC3 9T-1496 Cn1cc(c2c1cccc2)C(=O)N3CCCCC3 9T-1497 COc1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)C(=O)OC 9T-1499 COC(=O)c1cn(c2c1cccc2)S(=O)(=O)c3ccc(cc3)F 9T-1500 COC(=O)c1cn(c2c1cccc2)Cc3ccc(cc3)Cl 9T-1501 c1ccc(cc1)Cn2cc(c3c2cccc3)C(=O)C(F)(F)F 9T-1502 c1ccc(cc1)Cn2cc(c3c2cccc3)C(=O)O 9T-1504 c1ccc2c(c1)c(cn2Cc3ccc(cc3)Cl)C(=O)O 9T-1505 CN1Cc2ccccc2NC1=O 9T-1549 CC(C)(C)OC(=O)NC/C(=N/OC(=O)c1cc(ccc1C(F)(F)F)F)/N 9W-0008 CC(C)(C)OC(=O)NC/C(=N/OC(=O)c1ccc(cc1)C#N)/N 9W-0021 CCCOc1ccc(cc1)Oc2c3ccccc3c(nn2)c4ccc5c(c4)CCC5 9W-0202 c1cnc2nc(c(n2c1)Br)c3ccc4c(c3)OCO4 9W-0205 CCCc1ccc(cc1)Oc2c3ccccc3c(nn2)c4ccc5c(c4)CCC5 9W-0209 c1cc2c(cc1c3c(n4cc(ccc4n3)Cl)Cc5c(nc6n5cc(cc6)Cl)c7ccc8c(c7)OCO8)OCO2 9W-0214 c1ccnc(c1)c2ncc(c(n2)C(=O)NCc3ccco3)C(F)(F)F 9W-0215 CCCCCCCCc1c(=O)[nH]c(nc1O)n2c(=O)c(c([nH]2)C)CCO 9W-0218 COC(=O)c1cc(ccc1N2CCOCC2)[N+](=O)[O-] 9W-0222 CC1CN(CC(O1)C)c2ccc(cc2)[N+](=O)[O-] 9W-0224 COC(=O)c1cc(ccc1N2CCOCC2)N 9W-0232 COc1ccc(cc1)c2c(n3cc(ccc3n2)C(=O)O)Br 9W-0234 c1cc2c(cc1/C=C\3/C(=O)NC(=S)N3)OCO2 9W-0235 CSC1=N/C(=C\c2ccc3c(c2)OCO3)/C(=O)N1 9W-0240 CC1CN(CC(O1)C)c2ccc(cc2)N 9W-0242 Cc1ccc(n1c2ccc(cc2)C=O)C 9W-0243 c1ccc(cc1)/C=C/C=C\2/C(=O)NC(=S)N2 9W-0246 Cc1c(c(=O)n([nH]1)c2[nH]c(=O)c(c(n2)O)Cc3ccccc3)CCO 9W-0247 c1cc(ccc1c2c(n3cc(cc(c3n2)Cl)C(F)(F)F)Cl)F 9W-0249 c1ccc2c(c1)c(nnc2Sc3ccccn3)c4ccc5c(c4)CCC5 9W-0250 Cc1ccc(s1)c2c3ccccc3c(=O)[nH]n2 9W-0251 c1c([nH]n(c1=O)C(=N)N)C(F)(F)F 9W-0255 COC(=O)c1ccc2nc(cn2c1)c3ccc4c(c3)OCO4 9W-0257 c1ccc(cc1)CC(C(=O)O)NC2=N/C(=C\c3ccc4c(c3)OCO4)/C(=O)N2 9W-0260 CCOC(=O)c1cnc([nH]c1=O)n2c(=O)cc([nH]2)C(F)(F)F 9W-0262 Cc1c(c(=O)n([nH]1)C(=N)N)CCCN2C(=O)c3ccccc3C2=O 9W-0265 CSC1=N/C(=C\C=C\c2ccccc2)/C(=O)N1 9W-0266 c1c(nc2ncnn2c1O)C(F)(F)F 9W-0268 CC(=O)N1C(C(=O)N2C1=N/C(=C\c3ccc4c(c3)OCO4)/C2=O)Cc5ccccc5 9W-0272 Cc1cc(=O)n([nH]1)c2[nH]c(=O)cc(n2)C 9W-0274 c1cc(ccc1c2c(n3cc(cc(c3n2)Cl)C(F)(F)F)Cl)Br 9W-0279 c1cc2c(cc1c3cn4cc(cc(c4n3)Cl)C(F)(F)F)OCO2 9W-0280 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl 9W-0283 CC(C)(C)OC(=O)N1CCc2c1cc(cc2)N 9W-0285 CCOC(=O)c1cnc([nH]c1=O)n2c(=O)c(c([nH]2)C)CCCN3C(=O)c4ccccc4C3=O 9W-0288 CC(=O)c1ccc(cc1)S(=O)(=O)C 9W-0290 CS(=O)(=O)c1ccc(cc1)C(=O)CBr 9W-0291 c1cc2c(cc1/C=N/n3c(=O)cc(nc3N)C(F)(F)F)OCO2 9W-0292 COC(=O)c1ccc2nc(c(n2c1)Br)c3ccc4c(c3)OCO4 9W-0293 c1ccc(cc1)/C=C/C=N/n2c(=O)cc(nc2N)C(F)(F)F 9W-0297 COc1ccc(c(c1)/C=N/n2c(=O)cc(nc2N)C(F)(F)F)OC 9W-0298 c1ccc(c(c1)/C=N/n2c(=O)cc(nc2N)C(F)(F)F)C(F)(F)F 9W-0299 c1ccc2cc(ccc2c1)/C=N/n3c(=O)cc(nc3N)C(F)(F)F 9W-0300 c1cc2c(cc1c3c(n4cc(cc(c4n3)Cl)C(F)(F)F)Br)OCO2 9W-0304 c1cc2c(cc1c3c(n4cc(cc(c4n3)Cl)C(F)(F)F)Cl)OCO2 9W-0305 c1ccc(cc1)c2cc(=O)[nH]c(n2)n3c(=O)cc([nH]3)C(F)(F)F 9W-0308 C/C(=C\1/CCOC1=O)/Nc2ccc(cc2)Oc3ccccc3 9W-0309 Cc1c(c(=O)n(c(n1)N)N)CCCN2C(=O)c3ccccc3C2=O 9W-0311 c1cc(ccc1F)S(=O)(=O)NCC(=O)O 9W-0322 Cc1ccc(n1c2ccc(c(c2)Cl)O)C 9W-0323 c1ccn(c1)c2ccc(c(c2)Cl)O 9W-0324 Cc1cc2nc-3c(cn2n1)CCc4c3ccc(c4)OC 9W-0325 COc1ccc-2c(c1)CCc3c2nc4c(cnn4c3)C#N 9W-0326 COc1ccc-2c(c1)CCc3c2nc(nc3)N 9W-0327 c1cc(cc(c1)C(F)(F)F)c2n[nH]nn2 9W-0332 COC(=O)c1cc(ccc1N2CCN(CC2)Cc3ccccc3)N 9W-0334 c1cc(ccc1C(=O)CCCN2CCOCC2)F 9W-0337 CN(CC(=O)O)c1ccc(cc1[N+](=O)[O-])S(=O)(=O)N2CCOCC2 9W-0338 Cc1nc2nc(cc(n2n1)O)C(F)(F)F 9W-0340 c1ccc(cc1)COc2ccc(cc2)/C=N/n3c(=O)cc(nc3N)C(F)(F)F 9W-0343 C#CCOc1ccccc1/C=N/n2c(=O)cc(nc2N)C(F)(F)F 9W-0348 C=CCOc1c(ccc2c1cccc2)/C=N/n3c(=O)cc(nc3N)C(F)(F)F 9W-0349 CC(=O)c1ccc(cc1O)OCCCCl 9W-0351 c1cc2c(cc1c3cn4cc(ccc4n3)C(=O)NN)OCO2 9W-0352 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C=N/n3c(=O)cc(nc3N)C(F)(F)F)F 9W-0356 c1ccc(c(c1)/C=N/n2c(=O)cc(nc2N)C(F)(F)F)Oc3ccc(cc3)Cl 9W-0357 C#CCOc1ccc(cc1/C=N/n2c(=O)cc(nc2N)C(F)(F)F)Cl 9W-0358 c1cc(cc(c1)O)/C=N/n2c(=O)cc(nc2N)C(F)(F)F 9W-0359 c1cc(cc(c1)Oc2ncccn2)/C=N/n3c(=O)cc(nc3N)C(F)(F)F 9W-0360 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc3c(c2)NC(=O)C4N3CCC4 9W-0362 COC(=O)c1c(c2ccccc2[nH]1)C=O 9W-0364 COC(=O)C1CC(=O)N(C1)C2CCN(CC2)Cc3ccccc3 9W-0600 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)OC 9W-0607 CC(C)C/C=C/1\CCc2c3ccccc3[nH]c2C1=O 9W-0800 Cn1cc(c2c1cccc2)CCCC(=O)NN 9W-0801 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C/c4ccc(c(c4)Cl)Cl)/CC3 9W-0802 c1ccc(c(c1)/C=C\2/CCc3c4ccccc4[nH]c3C2=O)C(F)(F)F 9W-0803 c1ccc2c(c1)c3c([nH]2)C(=O)/C(=C\c4ccc(cc4)Cl)/CC3 9W-0804 c1ccc(cc1)COc2ccc(cc2)n3cn[nH]c3=O 9W-0805 CCOC(=O)c1cnn2c1nc(c(c2C)Cc3ccc(nc3)Cl)C 9W-0807 Cc1cc(nc(n1)n2cc(nn2)C(=O)OC)C(F)(F)F 9W-0808 Cc1ccc(cc1)/C=C\2/CCc3c4ccccc4[nH]c3C2=O 9W-0810 c1ccc(cc1)/C=C\2/CCc3c4ccccc4[nH]c3C2=O 9W-0811 c1ccc(c(c1)/C=C\2/CCc3c4ccccc4[nH]c3C2=O)F 9W-0812 CCC(CC)/C=C\1/CCc2c3ccccc3[nH]c2C1=O 9W-0813 c1cc(cc(c1)NC(=O)NN)C(F)(F)F 9W-0814 c1ccc2c(c1)cc3c(n2)-c4c(c5ccccc5[nH]4)CC3 9W-0815 CN(c1c(cc(cn1)C(F)(F)F)Cl)N.Cl 9W-0816 Cc1nn(c(=O)n1c2cccc(c2)OC)CCCC(=O)O 9W-0817 CN(C)/C=C/1\CCc2c3ccccc3[nH]c2C1=O 9W-0818 Cc1nn(c(=O)n1c2ccc(cc2)OCc3ccccc3)C(C)C(=O)O 9W-0819 Cc1ccc(cc1)n2c(nn(c2=O)C(C)C(=O)O)C 9W-0820 Cn1cc(c2c1cccc2)CCCC(=O)NNC(=O)NCc3ccc(cc3)Cl 9W-0821 Cn1cc(c2c1cccc2)CCCC(=O)N/N=C\c3c[nH]c4c3cc(cc4)OC 9W-0822 C/C(=N\OC(=O)c1cccc(c1)OC)/c2cnccn2 9W-0825 C/C(=N\OC(=O)c1cccs1)/c2cnccn2 9W-0826 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2cnccn2 9W-0827 COc1ccc(c(c1/C=C/[N+](=O)[O-])[N+](=O)[O-])OC 9W-0829 Cc1ccc2c(c1)c3ccc4c5ccccc5[nH]c4c3[nH]2 9W-0832 C/C(=N\OC(=O)c1ccc(cc1)F)/c2nccs2 9W-0835 C/C(=N/OC(=O)c1cccc(c1)Cl)/c2nccs2 9W-0836 C/C(=N\OC(=O)c1cccc(c1)C(F)(F)F)/c2nccs2 9W-0838 Cc1ccc(cc1)/C=N/NC(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl 9W-0840 CCOc1cc(ccc1O)/C=N/NC(=O)NN(C)c2c(cc(cn2)C(F)(F)F)Cl 9W-0841 Cc1c2c(cc(cn2)C(F)(F)F)sc1C(=O)OC 9W-0845 CCCC/C=C/1\CCc2c3ccccc3[nH]c2C1=O 9W-0846 CC(C)/C=C/1\CCc2c3ccccc3[nH]c2C1=O 9W-0847 CC1(NC(=S)N(N1)c2ccccc2)C 9W-0848 c1ccc(cc1)CO/N=C/2\CCCc3c2[nH]c4c3cccc4 9W-0849 CCOC(=O)Cn1c(=O)n(cn1)c2ccc(cc2)C(C)C 9W-0850 CCOC(=O)Cn1c(=O)n(cn1)c2ccc(cc2)C 9W-0852 COC(=O)c1c(c2ccccc2[nH]1)c3ccc(cc3[N+](=O)[O-])C(F)(F)F 9W-0853 Cc1cccc(c1)CSc2nnc(n2CC=C)c3csc(n3)n4c(cc(n4)C)C(F)(F)F 9W-0854 c1cc(ccc1CN2CCN(C2=O)c3ccc(cc3)F)F 9W-0855 Cc1ccc(cc1)n2cnn(c2=O)CC#N 9W-0858 c1c(cc(cc1C(F)(F)F)n2cn[nH]c2=O)C(F)(F)F 9W-0859 COc1ccc(cc1OC)C(CCO)N 9W-0860 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3CC=C)SC4CCCC4)C(F)(F)F 9W-0861 COc1cccc(c1)CN2CCN(C2=O)c3ccc(cc3)F 9W-0862 C=CCn1c(nnc1Sc2c(cccn2)[N+](=O)[O-])c3ccc4c(c3)OCO4 9W-0863 CCOC(=O)Cn1c(=O)n(cn1)c2ccc(cc2)OC(F)(F)F 9W-0867 c1cc(ccc1n2cnn(c2=O)CC#N)OC(F)(F)F 9W-0868 c1cc(ccc1n2cnn(c2=O)CC#N)Br 9W-0869 c1ccc(cc1)n2cnn(c2=O)CC#N 9W-0870 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(\C)/c3nccs3 9W-0871 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(\C)/c3nccs3 9W-0872 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)O/N=C(\C)/c3nccs3 9W-0873 c1ccc(cc1)c2csc3c2ncc(c3)C(F)(F)F 9W-0875 COc1ccc(cc1OC)C(CCO)NC(=O)c2cccs2 9W-0876 CCOc1ccc(cc1)C(CCO)N 9W-0878 Cc1ccc(cc1)CN2c3cc(ccc3NCCC2=O)C(F)(F)F 9W-0879 c1cc(cc(c1)C(F)(F)F)CN2CCN(C2=O)c3ccc(cc3)F 9W-0880 c1cc2c(cc1[N+](=O)[O-])cc(c(=O)o2)C(=O)O 9W-0881 COc1ccc(cc1)C(=O)O/N=C/2\CCCc3c2[nH]c4c3cccc4 9W-0883 COc1ccc2c(c1)c(c[nH]2)CCn3cc(c4ccccc4c3=O)C(=O)OC 9W-0884 Cc1cccc(c1)CO/N=C/2\CCCc3c2[nH]c4c3cccc4 9W-0886 CC1=C(/C(=C/c2c[nH]c3c2cc(cc3)OC)/C(=O)N1CCc4ccccc4)C(=O)OC 9W-0891 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)c4cc(nc(n4)N)Cl 9X-0007 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)S(=O)(=O)c4ccccc4[N+](=O)[O-] 9X-0008 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)OC 9X-0009 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)c4ccc(cc4[N+](=O)[O-])C(=O)OC 9X-0016 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)c4c(cccn4)[N+](=O)[O-] 9X-0017 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)Cc4cccc(c4)C(F)(F)F 9X-0018 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)Cl 9X-0025 c1cc(ccc1c2cc(n[nH]2)C3CCN(CC3)c4cc(nc(n4)N)Cl)Cl 9X-0026 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)Cl 9X-0027 COc1ccc(c(c1)c2cc(n[nH]2)C3CCN(CC3)c4cc(nc(n4)N)Cl)OC 9X-0035 COc1ccc(c(c1)c2cc(n[nH]2)C3CCN(CC3)c4c(cccn4)[N+](=O)[O-])OC 9X-0036 c1cc(c(nc1)N2CCC(CC2)c3cc([nH]n3)c4ccc(cc4)Cl)[N+](=O)[O-] 9X-0037 CC(C)(C)OC(=O)N1CCC(CC1)c2cc([nH]n2)c3cc(ccc3OC)OC 9X-0045 CC(C)(C)OC(=O)N1CCC(CC1)c2cc([nH]n2)c3ccc(cc3)Cl 9X-0046 CC(C)(C)OC(=O)N1CCC(CC1)c2cc([nH]n2)c3ccc(cc3)OC 9X-0047 c1cc(ccc1c2cc(n[nH]2)C3CCN(CC3)CC(C(F)(F)F)O)Cl 9X-0050 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)CC(C(F)(F)F)O 9X-0058 c1cc(ccc1c2cc(n[nH]2)C3CCN(CC3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl 9X-0070 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCC(CC3)c4cc([nH]n4)c5ccc(cc5)Cl 9X-0076 COc1ccc(cc1)c2cc(n[nH]2)C3CCN(CC3)C4=C(C(=O)c5ccccc5C4=O)Cl 9X-0078 c1cc(c(cc1[N+](=O)[O-])/C=C\2/C(=O)C3CCN2CC3)N4CCOCC4 9X-0083 Cc1cccc(c1N2CCN(CC2)c3ccc(cc3/C=C\4/C(=O)C5CCN4CC5)[N+](=O)[O-])C 9X-0090 c1cc2c(cc1CN3CCN(CC3)c4ccc(cc4/C=C\5/C(=O)C6CCN5CC6)[N+](=O)[O-])OCO2 9X-0091 c1cc(oc1)c2cc(n[nH]2)C3CCN(CC3)c4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] 9X-0097 c1cc(oc1)c2cc(n[nH]2)C3CCN(CC3)CC(C(F)(F)F)O 9X-0098 c1cc(oc1)c2cc(n[nH]2)C3CCN(CC3)c4cc(nc(n4)N)Cl 9X-0099 C#CCOc1ccc2ccccc2c1/C=C(/C#N)\c3ccc(cc3)Cl 9X-0220 Cn1cc(cc1CN2CCOCC2)C(=O)c3ccccc3 9X-0232 c1ccc(cc1)CC2CCN(CC2)Cc3ccccc3OCc4cnc(s4)Cl 9X-0233 c1ccc(c(c1)CN2CCOCC2)OCc3cnc(s3)Cl 9X-0235 Cn1cc(cc1CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])C(=O)c4ccccc4 9X-0239 Cn1cc(cc1CN2CCN(CC2)c3ccc(cc3)OC)C(=O)c4ccccc4 9X-0246 Cn1cc(cc1CN2CCN(CC2)c3ncccn3)C(=O)c4ccccc4 9X-0247 Cn1cc(cc1CN2CCN(CC2)C(c3ccccc3)c4ccccc4)C(=O)c5ccccc5 9X-0248 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)Cc4ccccc4OCc5cnc(s5)Cl 9X-0249 Cn1cc(cc1CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)c4ccccc4 9X-0254 COC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCN(CC2)Cc3c4ccccc4ccc3OCC=C 9X-0261 C#CCOc1ccc2ccccc2c1CN3CCN(CC3)Cc4ccc5c(c4)OCO5 9X-0264 CN(CC(OC)OC)C1=NC(=O)/C(=C\c2cccc3c2cccc3)/S1 9X-0272 CN(CC(OC)OC)C1=NC(=O)/C(=C\c2ccc(cc2)SC)/S1 9X-0281 CN(CCO)C1=NC(=O)/C(=C\c2ccc(cc2)SC)/S1 9X-0282 Cc1c(n(c(c1S(=O)(=O)C)n2cccc2)CCCN(C)C)C 9X-0286 CN1CCN(CC1)C2=NC(=O)/C(=C\c3cccc4c3cccc4)/S2 9X-0289 c1ccc2c(c1)cccc2/C=C/3\C(=O)N=C(S3)N4CCCC(C4)CO 9X-0297 CSc1ccc(cc1)/C=C/2\C(=O)N=C(S2)NCC(=O)O 9X-0298 CSc1ccc(cc1)/C=C/2\C(=O)N=C(S2)N3CCN(CC3)CCO 9X-0299 CSc1ccc(cc1)/C=C/2\C(=O)N=C(S2)N3CCCCC3CCO 9X-0304 c1c2n(nc1CO)CCCNC2 9X-0601 c1cc2c(cc1N)cc(s2)C(=O)O 9X-0700 c1cnc(cc1C#N)N2CCCCC2 9X-0702 COC(=O)c1c(ccs1)O 9X-0703 c1cc(c(cc1[N+](=O)[O-])NC=O)C(=O)O 9X-0800 CN(C)c1ccc(c(c1)O)C(=O)O 9X-0801 CCOC(CNC)OCC 9X-0802 CCSc1ncc(c(n1)N)C#N 9X-0804 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SCc4ccc(cc4)C(F)(F)F)C(F)(F)F 9X-0805 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SC4CCCC4)C(F)(F)F 9X-0806 Cc1cc(n(n1)c2nc(cs2)c3nnc(n3C)SCc4ccc(cc4)C(=O)O)C(F)(F)F 9X-0807 c1cc(sc1)/C=N/c2nncs2 9X-0808 CCOC(=O)c1c(nc2n1cccc2)C(F)(F)F 9X-0811 c1ccc2cc(ccc2c1)C(=O)c3cn(nn3)c4ccc(cc4)C(F)(F)F 9X-0812 Cn1c(c(c(=O)[nH]c1=O)Br)N 9X-0813 CS(=O)(=O)c1ccc(cc1)N 9X-0815 CCOC(=O)c1c(nc2n1cccn2)C(F)(F)F 9X-0816 CCOC(=O)c1c(nc2n1c(ccc2)C)C(F)(F)F 9X-0817 Cc1ccc(c(c1)CSc2nnc(n2C)c3csc(n3)n4c(cc(n4)C)C(F)(F)F)C 9X-0818 c1cc(oc1)C(=O)c2cn(nn2)c3ccc(c(c3)Cl)Cl 9X-0819 CCCCN(C)c1ncc(s1)C=O 9X-0820 CN(c1ncc(s1)C=O)C2CCCCC2 9X-0821 CN(Cc1ccccc1)c2ncc(s2)C=O 9X-0822 c1ccn2c(c1)nc(c2C(=O)O)C(F)(F)F 9X-0823 Cc1cccn2c1nc(c2C(=O)O)C(F)(F)F 9X-0824 c1ccn(c1)c2ccc(nc2)Cl 9X-0825 c1ccn(c1)c2cccnc2Cl 9X-0826 c1ccn(c1)c2c(c(nc(c2Cl)F)F)F 9X-0827 c1ccn(c1)C2=NCCS2 9X-0830 c1cc(c(c(c1)Cl)c2c(c(on2)c3cn(nn3)c4ccc(cc4)C(F)(F)F)C#N)Cl 9X-0831 CC(c1ccc(cn1)C(=O)C(C)Oc2ccc(cc2)F)Oc3ccc(cc3)F 9X-0832 c1cnc2nccn2c1 9X-0834 c1cc(sc1)/C=N/c2ccc(cc2)OC(F)(F)F 9X-0835 c1ccc(cc1)CNc2ccc(cc2C(=O)O)[N+](=O)[O-] 9X-0838 Cc1ccn2ccnc2c1 9X-0841 CN(C)Cc1cnc2n1cc(cc2)C(=O)OC 9X-0843 C1Cc2c(nn(c2N)CCC#N)C1 9X-0844 COC(=O)c1c(c2cc(ccc2[nH]1)I)I 9X-0845 c1c(cc(cc1C(=O)C2CC2)C(=O)C3CC3)C(=O)C4CC4 9X-0846 C1=CC2=NC(=C(C2C=C1I)I)C(=O)O 9X-0848 CC(C)(C)c1ccc(cc1)c2cnco2 9X-0849 Cc1cccc2n1c(c(n2)C(F)(F)F)C(=O)O 9X-0850 c1cc(cc(c1)Br)c2cnco2 9X-0851 Cc1cc(n2ccnc2c1)C 9X-0854 c1ccc2c(c1)c(cc(c2O)C(=O)O)Oc3ccc(cc3)[N+](=O)[O-] 9X-0856 c1cc2c(ccc(n2)C(=O)O)c(c1)[N+](=O)[O-] 9X-0857 COc1cc(ccc1O)/C=C(\C#N)/C(=O)O 9X-0858 Cc1cc(c(s1)C)C(=O)/C=C/N(C)C 9X-0860 c1cc(cc(c1)c2cnco2)C#N 9X-0861 c1cc(cc(c1)[N+](=O)[O-])c2cnco2 9X-0862 CCOC(=O)c1c(nc2n1cc(cc2)I)C(F)(F)F 9X-0863 COC(=O)CC(C(=O)c1cn(nn1)c2ccc(c(c2)Cl)Cl)C(=O)OC 9X-0864 c1ccn(c1)c2cc(cnc2)C(F)(F)F 9X-0865 c1ccc(c(c1)c2cnco2)C(F)(F)F 9X-0866 c1cc(oc1)c2cnco2 9X-0867 CC(C(=O)O)NCc1cnc2n1cc(cc2)Cl 9X-0868 Cc1c(cc2ccccc2n1)OCC(=O)N(C)c3ccccc3 9X-0869 c1ccc2c(c1)CCNC2C3C(=O)CC(C(C3=O)n4cncn4)c5ccccc5Oc6cccc(c6)Cl 9X-0870 Cc1cc(c(s1)C)c2ccnc(n2)N 9X-0872 c1cc(ccc1C#N)c2cnco2 9X-0874 COC(=O)c1c(c2cc(ccc2n1Cc3ccc(c(c3)Cl)Cl)I)I 9X-0875 CC(c1ccccc1)NC(=O)Cn2cncn2 9X-0876 Cc1cccc(c1N2CCN(CC2)C(=O)Cn3cncn3)C 9X-0877 c1cc(c(cc1F)CNC(=O)Cn2cncn2)F 9X-0880 c1cc(c(cc1Br)C(F)(F)F)O 9X-0882 c1ccc(cc1)c2c(nnc(n2)OCc3ccc(cc3)Cl)c4ccccc4 9X-0883 C/C(=N\NC(=S)N)/c1cc(sc1Cl)Cl 9X-0884 Cc1cc(c(s1)C)c2cc[nH]n2 9X-0885 c1ccc(c(c1)c2cnco2)Br 9X-0886 CCOC(=O)c1c(nc2n1cccc2C)C(F)(F)F 9X-0909 CC(C(=O)OC)N(Cc1cnc2n1cc(cc2)Cl)Cc3cnc4n3cc(cc4)Cl 9X-0910 CCCCn1c2ccccc2c3c(c1=O)c(cc(=O)o3)O 9X-0921 Cc1cc(cc(c1/N=C/N(C)C)[N+](=O)[O-])Br 9X-0923 Cc1cc(c(cc1OCc2cccc(c2)Cl)C)CN3CCOCC3 9X-0924 c1ccc2c(c1)c3c(c(cc(=O)o3)O)c(=O)n2C4CCCCC4 9X-0928 c1cc2c3c(c1)c4c(c(cc(=O)o4)O)c(=O)n3CCC2 9X-0929 c1cc(ccc1N/N=C/c2cc(c[nH]2)C(=O)CCl)F 9X-0931 c1cc2c(cc1Cl)-c3c(cnc(n3)N)CS2 9X-0933 Cc1cc(c(cc1OCc2ccc(cc2)Br)C)CN3CCOCC3 9X-0935 c1cc(ccc1C(=O)Nc2ncc3c(n2)-c4cc(ccc4SC3)Cl)Cl 9X-0938 c1ccc(cc1)Cn2c3ccccc3c(c(c2=O)c4cc(=O)[nH][nH]4)O 9X-0940 Cc1cc(c(cc1OC(=O)Nc2ccc(cc2)Cl)C)CN3CCOCC3 9X-0941 Cc1cc(c(cc1OCC(=O)N)C)CN2CCOCC2 9X-0942 Cc1cc(c(c(c1)O)CN2CCOCC2)C 9X-0946 CCOC(=O)C1CCN(CC1)Cc2c(cc(cc2O)C)C 9X-0947 Cc1cc(c(cc1OCCCF)C)CN2CCOCC2.Cl 9X-0948 CCOC(=O)C1(CCN(CC1)Cc2ccccc2)S(=O)(=O)c3ccc(cc3)Cl 9X-0949 CCOC(=O)C1(CCN(CC1)Cc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl 9X-0950 CCOC(=O)C1(CCN(CC1)Cc2ccc(cc2)C)S(=O)(=O)c3ccc(cc3)Cl 9X-0952 Cc1cc(c(c(c1)O)CN2CCN(CC2)c3ccccc3)C 9X-0954 c1cc(ccc1C=O)OCCCCl 9X-0956 CCOC(=O)CS(=O)(=O)c1ccc(cc1)O 9X-0957 CCOC(=O)C1CCN(CC1)Cc2cc(c(c(c2)C(C)C)O)C(C)C 9X-0958 Cc1cc(c(c(c1)CN2CCOCC2)O)C.Cl 9X-0959 Cc1ccc(cc1)C(=O)c2ccsc2N 9X-0960 c1cc(ccc1C(=O)c2ccsc2N)Cl 9X-0961 c1cc(ccc1CN2CCCCC2)OCCCCl 9X-0962 CC(=O)/C=C/c1ccc(cc1)OCCCN2CCCCC2 9X-0963 COc1ccc(cc1)C(=O)c2ccsc2N 9X-0964 c1cc(ccc1/C=C/2\C(=O)NC(=S)N2)n3cncn3.O 9X-0966 CC(=O)/C=C/c1ccc(cc1)OCCCCl 9X-0968 Cc1ccc(cc1)CNC(=O)c2cnn(c2C(F)(F)F)C(C)(C)C 9X-5003 CC(C)(C)n1c(c(cn1)C(=O)NCc2cccc(c2)Cl)C(F)(F)F 9X-5004 CC(=O)NCCc1ccc(c(c1)OC)OC 9X-5048 C=C(c1ccccc1)c2ccc(cc2)N 9X-7013 CCOC(=O)N1CCc2c(c3cc(ccc3[nH]2)F)C1 9Y-0006 COC(=O)c1cc(=O)[nH]c(=O)n1COCC[Si](C)(C)C 9Y-0023 CC1CCCN(C1)c2ccc(cc2[N+](=O)[O-])c3c4ccccc4c(=O)[nH]n3 9Y-0029 COC(=O)c1cc2n(n1)CCCN(C2=O)Cc3ccccc3 9Y-0207 c1cc2c(cc1c3csc(n3)N)NC(=O)CO2.Cl 9Y-0217 COC(=O)c1cc(cnc1Cl)I 9Y-0700 c1cc(ccc1C=O)c2ccc(cn2)C=O 9Y-0701 COC(=O)c1ccc(cc1)c2ccc(cn2)C=O 9Y-0702 c1ccc(cc1)c2ccc(cn2)C=O 9Y-0703 c1cc(ncc1C=O)c2ccsc2 9Y-0705 c1cc(c(nc1)c2ccsc2)C=O 9Y-0708 COC(=O)c1ccc(cc1)c2c(cccn2)C=O 9Y-0709 c1cc(cc(c1)[N+](=O)[O-])c2c(cccn2)C=O 9Y-0712 c1cc(c(nc1)c2ccc(cc2)F)C=O 9Y-0713 c1cc(c(nc1)c2ccc(cc2)Cl)C=O 9Y-0714 COc1cccc2c1c(n[nH]2)N 9Y-0715 c1cc2c(nc1)nc(o2)CCl 9Y-0716 c1cc2c(nc1)NC(=O)CO2 9Y-0717 C/C(=C\C(=O)c1ccccn1)/N(C)C 9Y-0802 c1cc(ccc1N2CCCCCC2)[N+](=O)[O-] 9Y-0803 CCOc1ccc(cc1)C(CC(=O)O)n2cccc2 9Y-0805 COC(=O)c1cc2cc(ccc2oc1=O)[N+](=O)[O-] 9Y-0806 c1cc2ncc(n2cc1C#N)Br 9Y-0808 CC(=O)c1c(c(cs1)Br)Br 9Y-0810 c1ccc(cc1)c2nnc(o2)CCl 9Y-0814 c1cc(ccc1C=C(C#N)C#N)Br 9Y-0818 CC(=O)Nc1cccc(c1)C#CCN2CCN(CC2)c3ccc(cc3)F 9Y-0819 CC(=O)Nc1cccc(c1)C#CCN2CCOCC2 9Y-0820 CC(=O)Nc1cccc(c1)C#CCN2CCCC2 9Y-0823 c1cc(ccc1N)N2CCCCCC2 9Y-0830 CCCC1CCN(CC1)c2ccc(cc2[N+](=O)[O-])c3c4ccccc4c(=O)[nH]n3 9Y-0834 c1cc2nccn2cc1/C(=N/O)/N 9Y-0835 CC(=O)c1cc(c(s1)Br)Br 9Y-0839 c1ccc(cc1)CC2CCN(CC2)c3ccc(cc3[N+](=O)[O-])c4c5ccccc5c(=O)[nH]n4 9Y-0842 c1cc(ccc1C2(CCCCC2)C#N)O 9Y-5009 CC(C)(C)OC(=O)N1CC(CO1)O 9Y-5020 c1cc(c(c(c1)F)C(=O)NCCS(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl)F 9Z-0014 c1ccc(cc1)c2cc(cnc2Oc3ccccc3)C(F)(F)F 9Z-0035 c1cc(c(cc1C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl)Cl)Cl 9Z-0039 c1cc(c(cc1C(=O)NCCS(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl)Cl 9Z-0044 c1cc(c(cc1c2nnnn2CCSc3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl 9Z-0045 COc1ccc(cc1)C(=O)c2c(cc(cn2)C(F)(F)F)c3ccccc3 9Z-0057 c1cc(c(c(c1)F)c2nnnn2CCSc3c(cc(cn3)C(F)(F)F)Cl)F 9Z-0058 COc1cc2c(c(c1)Br)ocn2 9Z-0207 c1cc(cc(c1)NC(=O)c2cccs2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0211 Cn1cccc1C(=O)Nc2cccc(c2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0245 c1ccc2c(c1)cc(s2)C(=O)Nc3cccc(c3)c4cn5cc(cc(c5n4)Cl)C(F)(F)F 9Z-0247 c1ccc(cc1)/C=C/C(=O)c2c(ccs2)Cl 9Z-0260 c1cc(cc(c1)NC(=O)c2cccc(c2)C(F)(F)F)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0261 Cc1ccc(cc1)C(=O)Nc2cccc(c2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0262 c1cc(cc(c1)NC(=O)c2ccc(cc2)F)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0263 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc(c2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0264 c1cc(cc(c1)NC(=O)c2cccc(c2Cl)Cl)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0265 c1cc(cc(c1)NC(=O)c2ccc(cc2)C#N)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0266 CCCCCC(=O)Nc1cccc(c1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 9Z-0267 CCCC(=O)Nc1cccc(c1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 9Z-0268 COc1ccccc1N2CCN(CC2)CC(=O)NN 9Z-0279 c1ccc(cc1)C(=O)Nc2cccc(c2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0802 c1cc(cc(c1)NC(=O)C2CC2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0803 CC(C)(C)c1cc2ccccc2[nH]1 9Z-0804 c1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0805 CCc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0806 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)F)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0807 Cc1cccc2c1[nH]c(c2)C(C)(C)C 9Z-0810 Cc1ccc2c(c1)cc([nH]2)C(C)(C)C 9Z-0814 COc1ccc(cc1)C(=O)Nc2cccc(c2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0815 c1cc(cc(c1)NC(=O)C2CCCCC2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0816 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)[N+](=O)[O-] 9Z-0819 COc1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0823 CCc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0824 c1ccc(cc1)CC2CCN(CC2)c3ncc(s3)C=O 9Z-0825 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)N 9Z-0826 CCCC(=O)Nc1ccc(cc1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 9Z-0827 CCCCCC(=O)Nc1ccc(cc1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 9Z-0828 c1ccc(cc1)C2(CCN(CC2)Cc3cnc4n3cc(cc4)Cl)C#N 9Z-0829 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0830 COCC(=O)Nc1ccc(cc1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F 9Z-0831 c1cc(c(c(c1)Cl)Cl)C(=O)Nc2ccc(cc2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F 9Z-0834 c1cc(ccc1c2cn3cc(cc(c3n2)Cl)C(F)(F)F)NC(=O)CCC(=O)O 9Z-0835 c1cc(c(c(c1)C#N)N2CCCCCC2)C#N 9Z-0837 c1cc(ccc1c2cn3cc(cc(c3n2)Cl)C(F)(F)F)NC(=O)/C=C/C(=O)O 9Z-0839 COc1ccc(cc1)c2c3ccccc3c(=O)[nH]n2 9Z-0844 Cc1ccc(cc1N)C(=O)NN 9Z-0846 c1cc(ccc1c2cn3cc(ccc3n2)[N+](=O)[O-])Br 9Z-0848 c1cc(ccc1c2cn3cc(ccc3n2)[N+](=O)[O-])F 9Z-0849 CCCCCOc1ccc2cc(ccc2c1)Br 9Z-0920 COC(=O)c1cc2c(s1)cccc2Cl 9Z-0922 c1cc(ccc1S(=O)(=O)NC(Cc2c[nH]c3c2ccc(c3)F)C(=O)O)I 9Z-7020 c1ccc2c(c1)c(c[nH]2)CC(C(=O)O)NS(=O)(=O)c3ccc(cc3)I 9Z-7027 CN(C)C1CCN(C1)c2ccc(cc2)Br AA-0268 c1ccc(cc1)C2C/C(=N/O)/c3c2ccs3 AA-0476 CCOC(=O)C1CCN(CC1)S(=O)(=O)C AA-0700 CCOC(=O)c1cccnc1N AA-0701 c1c(cnc(c1CO)N)Br AA-0702 COC(=O)c1ccc(cc1)c2ccc(c(c2)Cl)Cl AA-0703 c1cc(ccc1c2ccc(c(c2)Cl)Cl)C(=O)O AA-0704 COC(=O)c1ccc(cc1)c2ccc(c(c2)F)Cl AA-0705 c1cc(c(nc1)N)CO AA-0706 c1cc(ccc1c2ccc(c(c2)F)Cl)C(=O)O AA-0707 c1ccc(cc1)CN2CCN(CC2)c3ccccc3C=O AA-0710 c1ccc(c(c1)C=O)N2CCOCC2 AA-0711 c1ccc(c(c1)C=O)N2CCCCC2 AA-0712 COC(=O)c1cc(c(cc1F)[N+](=O)[O-])F AA-0713 CCOC(=O)C1CCN(CC1)c2ccc(cc2)C=O AA-0714 CCOC(=O)CC(=O)C(C)Br AA-0715 CCOC(=O)Cc1c(sc(n1)N)C AA-0716 Cc1c(nc(s1)c2ccccc2)CC(=O)O AA-0718 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)Br)c3ccc(cn3)C(F)(F)F AA-0800 c1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3ccc(cn3)C(F)(F)F AA-0801 c1cc(ccc1C(=O)O)Oc2cc(ccn2)C(F)(F)F AA-0802 c1cc(cc(c1)NS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl)c4ccc(cn4)C(F)(F)F AA-0803 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)c4ccc(cn4)C(F)(F)F AA-0804 c1cc(ccc1C(=O)NN)Oc2cc(ccn2)C(F)(F)F AA-0805 c1cc(cc(c1)NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)c4ccc(cn4)C(F)(F)F AA-0806 COc1ccc(c2c1cc(c(n2)c3ccccc3)C#N)OC AA-0808 c1ccc(c(c1)CO/N=C/c2ccc(cc2)c3cc(ccn3)C(F)(F)F)Cl AA-0809 c1ccc(c(c1)CO/N=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)Cl AA-0810 c1cc(ccc1c2cnco2)C(=O)NN AA-0811 c1cc(ccc1C(=O)NNS(=O)(=O)c2ccc(cc2)I)Oc3cc(ccn3)C(F)(F)F AA-0812 c1ccc(cc1)C(=O)NNC(=O)c2ccc(cc2)Oc3cc(ccn3)C(F)(F)F AA-0813 c1ccc(c(c1)CO/N=C/c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl AA-0814 c1cc(ccc1CO/N=C/c2ccc(cc2)c3cc(ccn3)C(F)(F)F)Cl AA-0815 c1cc(ccc1CO/N=C/c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl AA-0816 c1cc(sc1)CNC(=O)c2ccc(cc2)Oc3cc(ccn3)C(F)(F)F AA-0817 CN(C)/C=C(\C#N)/C(=O)c1ccccc1 AA-0821 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)Cl AA-0822 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3cccc(c3)c4ccc(cn4)C(F)(F)F AA-0823 c1cc2c(cn[nH]2)c(c1)NS(=O)(=O)c3ccc(c(c3)[N+](=O)[O-])Cl AA-0828 c1cc(cc(c1)N2CCN(CC2)C(=O)c3c(cccn3)C(F)(F)F)C(F)(F)F AA-0831 COc1cc(c(c(c1)Br)O)[N+](=O)[O-] AA-0832 c1ccc(cc1)N2CCN(CC2)C(=O)c3c(cccn3)C(F)(F)F AA-0834 c1ccc2c(c1)c(c[nH]2)CN3CCC(CC3)C(=O)O AA-0835 c1cc(c(nc1)C(=O)NNS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F AA-0840 c1cc(c(nc1)C(=O)NNS(=O)(=O)c2cccn2c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F AA-0841 c1c(cc(nc1C(F)(F)F)C(F)(F)F)C(=O)NN AA-0843 c1cc(ccc1c2cc(on2)N)Cl AA-0845 CCOC(=O)c1cc2cc(ccc2o1)C=O AA-0847 c1cc(cc(c1)NC(=O)Nc2cccc3c2cn[nH]3)C#N AA-0848 c1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccc3c2cn[nH]3 AA-0849 CCOC(=O)c1cc2cc(cc(c2o1)OC)Br AA-0852 COc1ccc(cc1)C(=O)CC#N AA-0854 CC(=O)NNC(=O)c1cc(nc(c1)C(F)(F)F)C(F)(F)F AA-0857 COc1ccc(cc1)c2cc([nH]n2)N AA-0860 c1ccc(cc1)C(=O)NNC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F AA-0861 c1cc2c(cc1C=O)cc(o2)C(=O)O AA-0864 c1ccc(cc1)c2cc(on2)N AA-0865 c1cc(cc(c1)Cl)C(=O)CC#N AA-0866 c1cc(cc(c1)Cl)c2cc(on2)N AA-0867 COc1ccc(cc1OC)C(=O)CC#N AA-0868 c1cc(cc(c1)Cl)c2cc([nH]n2)N AA-0869 c1ccc(cc1)c2cc([nH]n2)N AA-0871 c1cc(ccc1F)S(=O)(=O)NNC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F AA-0874 c1ccc2c(c1)nc(o2)NN AA-0922 CCC(CC)COc1ccc2cc(ccc2c1)Br AA-0924 c1cc(c(c(c1)Br)F)C=O AA-0926 CCOC(=O)c1c(c2ccccc2[nH]1)Br AB-0012 CCOC(=O)c1c(c2ccccc2[nH]1)C=O AB-0014 c1ccc(cc1)[C@@H](c2c(cc(cn2)C(F)(F)F)Cl)c3n[nH]nn3 AB-0015 c1ccc(cc1)COC(=O)NC(c2ccc3c(c2)OCO3)S(=O)(=O)c4ccccc4 AB-0019 CCOC(=O)c1c(c2ccccc2[nH]1)CO AB-0026 COC(=O)C(Cc1c[nH]c2c1cccc2)N.Cl AB-0201 c1cc(ccc1[N+](=O)[O-])OC(=O)N2CCN(CC2)c3ccc(cc3F)F AB-0203 CC(C)(C)OC(=O)NNC(=O)OCc1ccccc1 AB-0209 CC(C)(C)OC(=O)N1CCCCN1C(=O)OCc2ccccc2 AB-0219 c1cc(cc(c1)OC(F)(F)F)OCC(=S)N AB-0600 c1cc(c(cc1F)F)OCC#N AB-0601 c1cc(c(cc1Br)Br)OCC#N AB-0602 c1cc(c(cc1F)F)OCC(=S)N AB-0603 c1cc(ccc1OCC#N)OC(F)(F)F AB-0604 COc1ccc(cc1)c2c3conc3c(=O)[nH]n2 AB-0700 CC(=O)c1cccc2c1ocn2 AB-0704 Cc1c(c(no1)c2ccccc2)C(=O)C AB-0705 CCCCc1nc2cccc(c2o1)C(=O)C AB-0706 c1ccc2cc(ccc2c1)c3c4conc4c(=O)[nH]n3 AB-0708 c1cc(ccc1C=O)c2ccc3c(c2)OCCCO3 AB-0709 COC(=O)c1ccc(cc1Cl)n2ccnc2 AB-0710 COC(=O)c1ccc(nc1)C=O AB-0711 c1c2c(c(=O)[nH]nc2C3CC3)no1 AB-0712 CCOC(=O)c1c(con1)C(=O)C2CC2 AB-0713 CN(C)/C=C/C(=O)c1cccc2c1ocn2 AB-0716 CCc1nc2cccc(c2o1)C(=O)C AB-0717 Cc1nc2cccc(c2o1)C(=O)C AB-0718 CCOC(=O)c1cnc(cc1O)O AB-0719 C#CCSc1ccc(cn1)[N+](=O)[O-] AB-0720 COc1ccc(cc1)/C=C/C(=O)c2ccccc2O AB-0721 c1cc(ncc1C#N)S AB-0722 COC(=O)c1ccc(cc1)c2ccc3c(c2)OCCCO3 AB-0724 c1ccc(c(c1)C(=O)CSC#N)Cl AB-0725 c1cc(c(cc1N2CCCCC2)Cl)C(=O)NCCO AB-0726 CCOC(=O)c1cnc(cc1Cl)Cl AB-0727 Cc1ccc(cc1)C(=O)COC(=O)C AB-0729 COC(=O)c1ccc(cc1Cl)n2cncn2 AB-0730 c1cc(cc(c1)n2cccn2)/C=N/O AB-0800 Cc1c(c(cc(c1F)Br)[N+](=O)[O-])N AB-0801 c1ccc2c(c1)c(c[nH]2)/C(=N/O)/N AB-0802 c1cc(ccc1C#N)Oc2ncc(cn2)Br AB-0803 C/C(=N\c1ccc2cn[nH]c2c1)/N(C)C AB-0805 c1ccc(c(c1)/C=N/O)n2cccn2 AB-0806 c1cc(c(cc1CC(=O)NN)[N+](=O)[O-])O AB-0808 CCN1CCN(CC1)CC#N AB-0809 Cc1ccc(n1c2cccc(c2)I)C AB-0813 Cc1cc2c(cc1[N+](=O)[O-])cn(n2)C AB-0815 Cc1ccc(n1c2ccc(cc2F)I)C AB-0817 Cc1ccc(n1c2ccc(cc2)I)C AB-0818 c1ccc(cc1)CC2CCN(CC2)CC#N AB-0820 COC(=O)c1ccc(c(c1)[N+](=O)[O-])OCc2ccc(c(c2)Cl)Cl AB-0821 Cc1cc(ccc1NC(=O)C)F AB-0823 Cc1cc(cc(c1NC(=O)C)[N+](=O)[O-])F AB-0824 CN(C)/C=N/c1ccc2c(c1)cn[nH]2 AB-0829 CC(C)C(c1cnccc1Cl)O AB-5006 Cc1cccc(c1)Nc2nc(cs2)c3ccc(cc3)[N+](=O)[O-].Br AB-5041 CCOC(=O)C(C(c1cccc(c1)Cl)NC(=O)OCc2ccccc2)C(=O)OCC AC-0012 Cc1c(c(=O)[nH]c(=O)[nH]1)CN2CCCC2 AC-0031 c1c(cnc(c1I)O)C(=O)O AC-0200 c1c(cnc(c1C(=O)O)O)I AC-0201 COC(=O)c1cc(c(s1)Br)Br AC-0202 c1cc(c(nc1)c2ccc3c(c2)ncnc3O)C(F)(F)F AC-0216 c1c(cnc(c1I)Cl)C(=O)O AC-0218 c1cc(ccc1c2c(c[nH]n2)N)Cl AC-0221 c1cc(ccc1C=O)OCc2ccc(c(c2)F)F AC-0700 c1cc(ccc1/C=C/C(=O)O)OCc2ccc(c(c2)F)F AC-0701 COc1cc(ccc1N)N2CCOCC2 AC-0703 CN(C)c1cc(nc(n1)c2ccccc2)Cl AC-0704 CCOC(=O)C1CCN(CC1)c2ccc(c(c2)OC)N AC-0707 CNc1cc(nc(n1)c2ccccc2)Cl AC-0708 c1ccc(cc1)c2nc(cc(n2)Cl)N3CCCCC3 AC-0709 c1cc(ccc1CO)COc2ccc(c(c2)Cl)Cl AC-0714 CCOC(=O)/C=C/c1ccc(cc1)OCc2ccccc2 AC-0716 CCNc1cc(nc(n1)c2ccccc2)Cl AC-0717 CCOC(=O)COc1cc(c(cc1F)F)[N+](=O)[O-] AC-0718 CNCc1nc2cc(ccc2o1)Cl AC-0720 CNCc1nnc(o1)c2ccc(cc2)Cl AC-0722 COC(=O)c1ccc(cc1)c2cccc(c2)[N+](=O)[O-] AC-0723 CCOC(=O)N1CCN(CC1)C(C)C(=O)c2cccs2 AC-0800 Cn1c(c(c(n1)Br)[N+](=O)[O-])Br AC-0801 CS(=O)(=O)c1ccccc1OCC(=O)O AC-0805 CC(C(=O)c1cccs1)N2CCN(CC2)CCO AC-0808 c1cc([nH]c1)C(=O)CC#N AC-0811 c1ccc2c(c1)c(co2)Br AC-0812 CC(=O)CCc1c[nH]c2c1cc(cc2)Br AC-0815 CS(=O)(=O)CC(=O)c1c[nH]c2c1cccc2 AC-0817 c1cc(c(cc1Br)C=O)OCC(=O)O AC-0818 c1cc(ccc1CO)c2ccc(cc2)[N+](=O)[O-] AC-0825 CS(=O)c1ccccc1c2ccc(cc2)C=O AC-0829 CC(=O)c1c(c2ccccc2o1)Br AC-0830 Cc1c(c2ccccc2[nH]1)C(=O)CC#N AC-0832 c1ccc2c(c1)c(co2)C(=O)O AC-0834 CCOC(=O)C1=NNC2C1C(=O)N(C2=O)C(=O)OC(C)(C)C AC-0839 CC(C)(C)OC(=O)N1CCN(CC1)c2c(c(ncn2)Cl)C=O AC-5003 CC(C)(C)OC(=O)N1CCN(CC1)c2c(c(ncn2)Cl)CO AC-5007 c1cc2c(c(c1)F)c(n[nH]2)N AC-5015 c1cc2c(cc1F)c(n[nH]2)N AC-5024 COCc1nc(no1)c2ccnc(n2)N3CCNCC3.Cl.Cl AD-0023 Cc1ccc(cc1)C(=O)N(C(C)(C)C)NC(=O)[C@@H]2CCCN2c3c(cc(cn3)C(F)(F)F)Cl AD-0044 c1ccc(cc1)COc2ccc(cc2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl AD-0064 CCc1nc(no1)c2ccnc(n2)N3CCNCC3.Cl.Cl AD-0104 c1cc(ccc1C(=O)NNC(=O)CCCl)F AD-0120 CC(C)Cc1nc(no1)c2ccnc(n2)N3CCNCC3.Cl.Cl AD-0122 c1cc(c(c(c1)Cl)c2ncc3n2cc(cc3F)C(F)(F)F)Cl AD-0158 CCc1c(nc(s1)N)CC(=O)OC AD-0159 c1cc(nc(c1[N+](=O)[O-])N)Br AD-0160 c1cnc(nc1c2nc(on2)C3CC3)N4CCNCC4.Cl.Cl AD-0179 c1cc2c(cc1F)OCC(=O)N2 AD-0189 c1cnc(nc1c2nc(on2)C(F)(F)F)N3CCNCC3.Cl.Cl AD-0194 c1cnn(c1)c2ccc(cc2)C(=O)CC#N AD-0212 CCOC(=O)C1CCCN(C1)CCCN AD-0240 CCOC(=O)C1CCCN(C1)CCN AD-0265 c1cc(ccc1C(=O)NN)N2CCOCC2 AD-0295 CC(C)C[C@@]1(CC([C@H](N1)c2nccs2)C(=O)OC(C)(C)C)C(=O)OC AD-0323 CN1CCN(CC1)c2ccc(cc2)C(=O)O.Cl AD-0334 CN1CCN(CC1)c2ccc(cc2)CO AD-0335 CN1CCN(CC1)c2ccc(cc2)C(=O)CC#N AD-0365 CC(C)(C)c1nc(on1)c2ccc(cc2)[N+](=O)[O-] AD-0700 c1cc2ncc(n2cc1F)Br AD-0701 c1cc(nc(c1C(=O)O)N)Cl AD-0702 COc1ccc(c(n1)Cl)C(=O)OC AD-0703 c1cc(c(cc1[N+](=O)[O-])N)N2CCCCC2 AD-0704 c1cc2nc(cn2cc1Cl)CO AD-0705 c1cc(c(cc1[N+](=O)[O-])N)N2CCOCC2 AD-0706 CC(C)(C)c1nc(on1)CCl AD-0709 c1cc2c(cc(s2)C=O)c(c1)Cl AD-0710 c1c(cn2c(cnc2c1I)Br)Cl AD-0711 c1cc(ccc1c2nc(c(s2)C(=O)O)C(F)(F)F)Cl AD-0712 COc1ccc(cc1[N+](=O)[O-])CC(=O)OC AD-0713 CCOC(=O)c1cc(c(cc1N)OC)C AD-0714 c1cc2c(cc1[N+](=O)[O-])cc(o2)/C=C/C(=O)O AD-0716 c1cc2nc(cn2cc1F)C(=O)NN AD-0717 c1cc2nccn2cc1C(F)(F)F AD-0719 Cc1cc(c(cc1OC)NC(=O)CCl)Br AD-0720 c1cc2nc(cn2cc1F)C(=O)O AD-0721 c1ccc(c(c1)c2ccc(cc2)C=O)C3OCCO3 AD-0723 c1cc2ncc(n2cc1C(F)(F)F)Br AD-0724 CCC(=O)c1cc([nH]c1)C(=O)OC AD-0725 CCOC(=O)C1CCN(CC1)c2ccc(cc2N)[N+](=O)[O-] AD-0726 Cc1cc(c(cc1OC)F)Br AD-0727 c1ccc(c(c1)C(=O)O)n2cncn2 AD-0730 c1c(cnc(c1Cl)NC2CC2)C(F)(F)F AD-0733 c1cc(cc2c1cc(s2)CO)C(F)(F)F AD-0734 CN(C(=O)c1cc(cnc1)Br)OC AD-0735 c1cc(ccc1C2OCCO2)Br AD-0736 c1cc(cc2c1cc(s2)C(=O)NN)C(F)(F)F AD-0737 c1ccc(c(c1)CO)n2cncn2 AD-0738 CC(=O)Nc1cc(ccc1F)[N+](=O)[O-] AD-0742 CC(C)(C)c1nc(on1)c2ccc(cc2)C#N AD-0743 c1ccc(cc1)CNc2ccc(cc2N)[N+](=O)[O-] AD-0744 c1cc(c(cc1N2CCCCC2)Cl)CO AD-0745 CS(=O)(=O)Nc1cc(ccc1F)[N+](=O)[O-] AD-0746 Cc1cc(c(cc1OC)N)C(=O)O AD-0747 CS(=O)(=O)N(c1cc(ccc1F)[N+](=O)[O-])S(=O)(=O)C AD-0748 c1cc(ccc1C=O)c2ccc(cc2)C3OCCO3 AD-0750 CC(=O)OCc1ccc2c(c1)nc(o2)CCl AD-0752 c1ccc2c(c1)C(=O)N(C2=O)c3cc(ccc3F)[N+](=O)[O-] AD-0753 c1cc(ncc1/C(=N/O)/N)C(=O)NO AD-0754 Cc1nc(cc(n1)O)NC AD-0756 c1cc(c(cc1[N+](=O)[O-])/C=C/C(=O)O)N2CCOCC2 AD-0758 COc1c(cc(c(n1)Cl)C(=O)O)F AD-0759 COc1c(cc(c(n1)Cl)C(=O)OC)F AD-0760 c1cc(ccc1CO)c2ccc(cc2)C3OCCO3 AD-0761 CCC(=O)c1cc(n(c1)C)C(=O)OC AD-0762 Cc1nc(cc(n1)O)N(C)C AD-0763 COc1cc(ccc1C(F)(F)F)[N+](=O)[O-] AD-0764 c1c(c(nc(c1Br)C2CC2)Cl)C#N AD-0765 CC(C)(C)OC(=O)N1CCCCCN1C(=O)c2ccc(cc2)[N+](=O)[O-] AD-0766 CC(C)(C)OC(=O)N1CCCCCN1C(=O)CCl AD-0767 Cc1nc(c(c(n1)Cl)Br)O AD-0768 COc1cc(ccc1C(F)(F)F)N AD-0769 c1ccc(cc1)Cn2cnc3c2ccc(c3)[N+](=O)[O-] AD-0771 Cc1nc(c(c(n1)Cl)Cl)O AD-0773 c1c(cnc(c1Cl)C(=O)NO)C(F)(F)F AD-0774 c1cc(cc2c1cc(s2)C=O)C(F)(F)F AD-0775 CC(C)(C)OC(=O)N1CCCCCN1C(=O)c2ccc(cc2)N AD-0776 CCC(c1cc([nH]c1)C(=O)C(Cl)(Cl)Cl)O AD-0778 c1c2c(n[nH]c2nc(c1Br)C3CC3)N AD-0779 Cn1c2c(cc(c(n2)C3CC3)Br)c(n1)N AD-0782 COC(=O)c1c(c2cc(c(nc2s1)C3CC3)Br)N AD-0784 Cc1nc2cc(ccc2n1Cc3ccccc3)[N+](=O)[O-] AD-0787 Cc1nc(c(c(n1)Cl)I)O AD-0790 Cc1nc(c(c(n1)O)Cl)NC AD-0791 c1ccc(cc1)Cn2cnc3c2ccc(c3)N AD-0792 C#Cc1ncc(cn1)Br AD-0794 c1cc(ccc1C(=O)N2CCCCCN2)[N+](=O)[O-] AD-0795 COc1cc(ccc1C#C)[N+](=O)[O-] AD-0796 Cc1nc(c(c(n1)O)Cl)N(C)C AD-0797 Cc1nc2cc(ccc2n1Cc3ccccc3)N AD-0799 CCOC(=O)C1CCN(CC1)S(=O)(=O)N(CCCl)C(=O)OC(C)(C)C AD-2002 C[C@@H](c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2c(cccc2Cl)Cl AD-2012 c1cc(c(cc1C(=O)NN)F)F AD-2033 c1c(cc(cc1F)F)C(=O)NN AD-2036 c1cnc(cc1C(F)(F)F)C#N AD-2052 COc1c(cc(cn1)Cl)C(=O)O AD-5000 Cc1nc(c(c(n1)O)Cl)N2CCCC2 AD-5001 Cc1nc(c(c(n1)O)I)NC AD-5002 CCOC(=O)c1c(c2ccccc2n1C)Br AD-5003 c1c(c(nc(c1Cl)C2CC2)Cl)C#N AD-5004 C#Cc1c(cc(cn1)C(F)(F)F)Cl AD-5008 COc1ccc(cc1[N+](=O)[O-])C(=O)CBr AD-5009 Cc1cc2c(cc1[N+](=O)[O-])c(n[nH]2)Br AD-5010 CCOC(=O)c1c(c2ccccc2n1C(=O)OC(C)(C)C)Br AD-5011 Cn1c2c(cc(c(n2)C3CC3)Cl)c(n1)N AD-5012 c1c2c(n[nH]c2nc(c1Cl)C3CC3)N AD-5013 c1ccc(cc1)C(=O)Oc2ccccc2O AE-0005 c1c(c(c(nc1I)Br)O)I AE-0006 c1cc(c(c(c1)O)O)[N+](=O)[O-] AE-0007 c1c(cnc(c1Cl)SCCCSc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F AE-0014 c1cc(c(c(c1)O)O)N AE-0019 Cc1c(c(c2ccccc2n1)Br)O AE-0025 c1cc(ccc1N2CCN(CC2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)Cl AE-0029 c1c(cnc(c1Cl)CNC(=O)N2CCNCC2)C(F)(F)F AE-0030 c1cc(c(c(c1O)C=O)Br)O AE-0031 c1cc(c(cc1NC(=O)C(F)(F)F)C(F)(F)F)Br AE-0032 CN(c1ccc(cc1)Cl)C(c2ccccc2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl AE-0037 c1ccnc(c1)N2CCN(CC2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl AE-0040 COc1cc(cc(c1O)N)C(=O)OC AE-0044 COc1cc(cc(c1OCc2ccccc2)[N+](=O)[O-])C(=O)OC AE-0045 CC(C)(C)[Si](C)(C)Oc1ccc(c(c1Br)C=O)O AE-0054 c1c(c(cc(c1NC(=O)C(F)(F)F)[N+](=O)[O-])Br)C(F)(F)F AE-0056 c1ccc(cc1)C(=O)Oc2cc(cc(c2O)[N+](=O)[O-])Cl AE-0059 c1ccc(cc1)C(=O)Oc2cc(ccc2O)Cl AE-0067 COc1cc(cc2c1OCC(=O)N2)C(=O)OC AE-0068 COc1cc(cc(c1OCc2ccccc2)N)C(=O)OC AE-0069 COc1cc(cc(c1OCc2ccccc2)[N+](=O)[O-])C(=O)O AE-0071 c1ccc(cc1)COc2ccc(nc2Cl)CBr AE-0075 c1c(c(cc(c1NC(=O)C(F)(F)F)N)Br)C(F)(F)F AE-0082 COc1c(cc(nc1Br)I)I AE-0088 COc1c(cc(nc1Cl)I)I AE-0089 c1ccc(cc1)C(=O)Oc2cc(cc(c2O)N)Cl AE-0094 c1cc(ccc1NC(=O)N2CCN(CC2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)Cl AE-0095 c1cc(ccc1S(=O)(=O)N2CCN(CC2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)Cl AE-0096 c1c(cnc(c1Cl)CNC(=O)N2CCN(CC2)S(=O)(=O)C(F)(F)F)C(F)(F)F AE-0097 COc1cc(cc2c1ocn2)C(=O)OC AE-0098 c1ccc(cc1)COc2c(cc(nc2Br)I)I AE-0100 Cc1c(c(=O)c(cn1Cc2ccccc2)I)OCc3ccccc3 AE-0104 Cc1nc2cc(cc(c2o1)OC)C(=O)OC AE-0108 c1cc(ccc1c2cc([nH]n2)NC(=O)CCSc3c(cc(cn3)C(F)(F)F)Cl)Cl AE-0113 c1c(c(c(c(n1)Cl)Cl)C(=O)Cl)Cl AE-0206 c1c(c(c(c(n1)Cl)Cl)C(=O)N)Cl AE-0207 COc1c(c(c(cn1)C(F)(F)F)C(=O)O)Cl AE-0208 c1c(c(c(c(n1)Cl)Cl)C#N)Cl AE-0211 c1c(c(c(c(n1)N)Cl)C#N)C(F)(F)F AE-0214 C=CCN/C(=N\O)/c1c(cc(cn1)C(F)(F)F)Cl AE-0218 COc1c(c(c(cn1)Cl)C#N)Cl AE-0219 CCOC(=O)[C@@H]1CNC[C@@H]1C(=O)OCC.Cl AE-0220 COC(=O)c1c(cnc(c1Cl)Cl)Cl AE-0225 c1cn2cc(c(c(c2n1)Cl)C#N)C(F)(F)F AE-0227 COc1c(c(ccn1)C(F)(F)F)C(=O)O AE-0230 c1cnc(c(c1C(F)(F)F)C(=O)N)Cl AE-0232 CCOC(=O)[C@H]1CN(C[C@@H]1C(F)(F)F)Cc2ccccc2 AE-0236 c1cnc(c(c1C(F)(F)F)C#N)Cl AE-0238 c1cc(c(cc1[N+](=O)[O-])I)Cl AE-0243 COC(=O)c1c(ccnc1N2CCNCC2)C(F)(F)F AE-0246 c1ccc(cc1)CN2C[C@@H]([C@H](C2)C(F)(F)F)C(=O)O AE-0247 Cc1ccc(cc1)S(=O)(=O)N2CCCC(=O)c3c2cccc3 AE-0248 CCOC(=O)/C=C/c1ccncc1 AE-0249 c1cc2c(c[nH]c2nc1)C(=O)CCl AE-0251 CCOC(=O)c1c(ccc(n1)c2ccccc2)C#N AE-0701 c1ccc(cc1)c2ccc(c(n2)C(=O)O)C#N AE-0702 CCOC(=O)c1c(c(c(cn1)C(F)(F)F)C#N)Cl AE-0703 CCOC(=O)c1c(c(ccn1)N(C)C)C#N AE-0706 c1c(c(c(c(n1)C(=O)O)Cl)C#N)C(F)(F)F AE-0707 CCOC(=O)c1cnc2c(c(nn2c1C)C)C#N AE-0708 c1ccc2c(c1)NC3(S2)CCCCC3 AE-0712 C1CCC2(CC1)NC(=O)CS2 AE-0714 CCOC(=O)c1c(cc(cn1)C#N)Cl AE-0716 C1CCC2(CC1)NCCS2.Cl AE-0717 c1cn2cc(cc(c2n1)Cl)C#N AE-0718 C1CCC2(C1)NCCS2.Cl AE-0719 c1c(cnc(c1Cl)C(=O)O)C#N AE-0720 C1CCCC2(CC1)NC(=O)CS2 AE-0721 Cc1c(c2ncc(c(n2n1)C)C(=O)O)C#N AE-0722 Cc1c(c(nc(c1I)C)OC)C#N AE-0723 CC(C)Nc1ccc(cc1C(=O)OC)[N+](=O)[O-] AE-0724 c1cn2cc(cc(c2n1)Br)C#N AE-0725 c1ccc(c(c1)CNc2ccccc2N)N AE-0726 CCOC(=O)C1CSC2(N1)CCCC2.Cl AE-0727 CCOC(=O)c1c(c(cc(n1)C)C)C#N AE-0728 c1cc2c(cc1C(=O)O)NCCS2 AE-0729 C1CCC2(C1)NC(=O)CS2 AE-0730 Cc1cc(nc(c1C#N)C(=O)O)C AE-0731 CCOC(=O)C1CCCCC12NCCS2.Cl AE-0733 c1c(cn2c(cnc2c1Cl)Br)C#N AE-0734 Cc1cc(cc(c1N)I)Cl AE-0735 CCOC(=O)c1cn2cc(cc(c2n1)Cl)C#N AE-0736 CCOC(=O)C1CCCCC12NC(=O)CS2 AE-0738 c1ccc(cc1)CN2CCC3(CC2)NCCS3 AE-0741 CCOC(=O)c1c(c(c(c(n1)C)Br)C)C#N AE-0742 c1cc(c(cc1C(=O)C(F)(F)F)Br)N AE-0743 CC(C)(C)OC(=O)N1CCC2(CC1)NCCS2.Cl AE-0744 c1ccc2c(c1)CCC3(C2)NCCS3.Cl AE-0746 c1cc(nc(c1)Cl)CCl AE-0747 COc1cc(ccc1[N+](=O)[O-])C(=O)CBr AE-0748 CN1CCC2(CC1)NCCS2.Cl AE-0752 CC(C)Nc1ccc(cc1C(=O)O)[N+](=O)[O-] AE-0753 C1CCC2(CC1)NCC(=O)N2 AE-0754 C1CC2(C1)C(=NNC2=O)N AE-0756 c1c(cn2c(cnc2c1Br)Br)C#N AE-0757 c1c(c(cnc1Cl)Cl)C(=O)N AE-0758 COC(=O)c1ccc2c(c1)NCCS2=O AE-0760 c1ccc(cc1)CN2CCC3(CC2)NC(=O)CS3 AE-0761 CCOC(=O)c1cc(ccc1F)[N+](=O)[O-] AE-0763 c1c(cnc(c1C(=O)N)Cl)Cl AE-0764 CN(C(=O)c1ccc(nc1)Cl)OC AE-0765 Cc1c(c(nc(c1Br)C)C(=O)O)C#N AE-0766 c1c(c(cnc1Cl)Cl)C#N AE-0767 c1ccc(cc1)CN2CCC(CC2)(C(=O)N)O AE-0768 c1ccc2c(c1)CCC3(C2)NC(=O)CS3 AE-0770 c1c(cnc(c1C#N)Cl)Cl AE-0771 COc1cc(c(c(c1)Br)O)N AE-0773 c1ccc(cc1)C(c2ccccc2)SCC(=O)O AF-0005 c1ccc(cc1)CC(C(=O)O)NC(=O)C(=O)O AF-0009 c1cc2c(c(c1)F)C(=O)N3[C@@H](C=CC=C3C2=O)N4CC5(CCN(CC5)c6c(cc(cn6)C(F)(F)F)Cl)COC4=O AF-0010 C[C@H]1CCN(C[C@H]1NC)Cc2ccccc2.Cl.Cl AF-0011 CCOC(=O)CSC(c1ccccc1)c2ccccc2 AF-0022 c1ccc(cc1)C(c2ccccc2)S(=O)CC(=O)O AF-0026 c1ccc(cc1)C(c2ccccc2)SCC(=O)NO AF-0032 c1cc(ccc1C(=O)N[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl)Cl AF-0041 c1cc(cc(c1)Cl)C(=O)N[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl AF-0042 c1ccc(c(c1)C(=O)N[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F AF-0043 c1cc(c(c(c1)F)C(=O)N[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl)F AF-0044 c1ccc(cc1)COC(=O)N[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl AF-0045 Cc1nc(c(c(n1)Cl)NC2=NCCN2C(=O)C)Cl AF-0055 c1ccc(cc1)CNc2ccnc(c2)C(F)(F)F AF-0227 CCOC(=O)c1cnc(nc1Cl)c2ccncc2 AF-0701 c1cc(ccc1C(=O)C(C#N)F)Cl AF-0702 CCOC(=O)c1c(c2ccccc2[nH]1)I AF-0703 COc1cc(c(c(c1O)[N+](=O)[O-])C(=O)OC)[N+](=O)[O-] AF-0704 c1cc(ccc1c2c(c([nH]n2)N)F)Cl AF-0706 COc1cc(c(cc1O)C(=O)O)[N+](=O)[O-] AF-0707 Cc1ccc(cc1)C(=O)C(C#N)F AF-0708 c1ccc(cc1)C(=O)C(C#N)F AF-0709 c1cc(cc(c1)C(F)(F)F)C(=O)C(C#N)F AF-0710 CCOC(=O)c1cn2cc(sc2n1)Br AF-0711 COc1cc(c(cc1O)C(=O)OC)[N+](=O)[O-] AF-0712 c1c(c2c([nH]1)ncnc2Cl)F AF-0713 Cc1ccc(cc1)c2c(c([nH]n2)N)F AF-0715 c1c(c2c([nH]1)ncnc2Cl)Br AF-0716 c1cc(c(cc1[N+](=O)[O-])CC#N)Cl AF-0719 c1ccc(cc1)c2c(c([nH]n2)N)F AF-0720 c1c(c(cc(c1F)NN)F)C#N AF-0722 c1cc(nc(c1N)I)Cl AF-0723 Cn1c2ccc(cc2nn1)[N+](=O)[O-] AF-0724 CCOC(=O)Cc1c(sc(n1)c2ccc(cc2)Cl)C AF-0725 c1cc(cc(c1)C(F)(F)F)c2c(c([nH]n2)N)F AF-0726 Cn1c2c(cc(s2)CO)c(n1)c3ccccc3 AF-0727 c1cc(oc1)C(=O)C(C#N)F AF-0728 CCOC(=O)/C(=C(/c1ccccc1)\O)/C#N AF-0730 CNc1cc(nc(n1)c2ccccc2)C(=O)N AF-0731 c1cnc2c(c1Cl)c(c[nH]2)I AF-0733 CCOC(=O)c1c(c2cc(ccc2[nH]1)[N+](=O)[O-])I AF-0734 c1ccc2c(c1)c(cc(n2)N)O AF-0735 COc1cc(c(cc1O)C(=O)OC)N AF-0736 Cc1nc2cc(ccc2n1C)N AF-0737 CCOC(=O)/C(=C(/c1ccc(cc1)C)\O)/C#N AF-0742 c1cc(c(cc1N)CC#N)Cl AF-0743 c1cc(c(cc1N)CC(C#N)c2cc(ccc2Cl)N)Cl AF-0744 Cn1c2c(cc(s2)C=O)c(n1)c3ccccc3 AF-0747 C1COCCN1c2nnc(s2)Br AG-0001 C1CCN(C1)c2nnc(s2)Br AG-0002 c1ccnc(c1)Sc2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl AG-0003 c1cc(sc1)Sc2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl AG-0004 c1cc(ccc1F)Sc2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl AG-0006 c1ccc(c(c1)F)Sc2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl AG-0007 CC(C)(C)OC(=O)N1CCN(CC1)c2nnc(s2)Br AG-0010 c1c(cnc(c1Cl)NC(=O)N2CCCCC2)C(F)(F)F AG-0011 c1ccc(cc1)C(=O)n2cc(c3c2ncc(c3)C(F)(F)F)Cl AG-0013 c1ccc(cc1)CC(=O)n2cc(c3c2ncc(c3)C(F)(F)F)Cl AG-0014 c1ccc(cc1)S(=O)(=O)n2cc(c3c2ncc(c3)C(F)(F)F)Cl AG-0015 CN1CCN(CC1)C(=O)Nc2c(cc(cn2)C(F)(F)F)Cl AG-0016 CCOC(=O)NC(=S)Nc1c(cc(cn1)C(F)(F)F)Cl AG-0018 CC1(CONC1=O)C AG-0019 CC(C)(C)OC(=O)N1CCCN(CC1)c2nnc(s2)Br AG-0020 COc1cccc(c1)Sc2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl AG-0024 Cc1c(cccc1OC)CO AG-0026 c1cc2c(c(c1)[N+](=O)[O-])[nH]c(=O)[nH]2 AG-0030 c1c(cn2c(c1Cl)nc(n2)N)C(F)(F)F AG-0031 C1CN(CCN1)c2nnc(s2)Br AG-0032 c1ccc(cc1)NNC(=O)Cn2cc(c3c2ncc(c3)C(F)(F)F)Cl AG-0039 c1ccc(cc1)COc2cccc3c2c(no3)N AG-0040 CN(C)C(=O)Cn1cc(c2c1ncc(c2)C(F)(F)F)Cl AG-0041 C1CNCCN(C1)c2nnc(s2)Br AG-0044 Cc1c(ccc(c1CO)Br)OC AG-0055 c1ccc(cc1)NNC(=O)CCl AG-0057 CN(c1ccccc1)C(=O)Cn2cc(c3c2ncc(c3)C(F)(F)F)Cl AG-0061 c1cc(ccc1C#N)Oc2nnc(s2)Br AG-0063 c1cc(ccc1NNC(=O)Nc2c(cc(cn2)C(F)(F)F)Cl)F AG-0065 c1cc(cc(c1)Oc2nnc(s2)Br)C#N AG-0066 COc1ccc(cc1)Oc2nnc(s2)Br AG-0067 COc1cc(ccc1F)CNC2CCCC2 AG-0068 CCCCNc1nnc(s1)NCCCC AG-0069 CCCNCc1ccc(c(c1)OC)C AG-0073 COc1cccc(c1)Oc2nnc(s2)Br AG-0079 Cc1c(ccc(c1CO)C#N)OC AG-0085 Cc1ccc(cc1OC)CO AG-0096 Cc1ccc(cc1)C(=O)c2cc(n(c2)C)C=O AG-0201 CCOC(=O)/C=C/c1cc(cn1C)C(=O)c2ccc(cc2)C AG-0203 Cc1ccc(cc1)C(=O)c2cc(n(c2)C)/C=C/C(=O)O AG-0207 CCOC(=O)c1ccc(nc1C)Cl AG-0209 Cc1c2ccccc2oc1C(=O)O AG-0210 Cc1c2cc(ccc2oc1C(=O)OC)OC AG-0214 Cc1c(ccc(n1)Cl)C(=O)O AG-0216 CN1CCc2c(c3ccccc3[nH]2)C1 AG-0220 c1ccc2c(c1)nc(c(n2)Cl)C(=O)O AG-0222 c1cc(ccc1/C=C/CCl)Br AG-0700 Cc1c(nc2ccccc2n1)C(=O)O AG-0701 CCOC(=O)c1c(nc2ccccc2n1)C(F)(F)F AG-0704 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(=O)O AG-0705 c1cnc(cc1C(F)(F)F)C=O AG-0706 c1cnc(cc1C(F)(F)F)CCl AG-0707 CCOC(=O)c1c2cc[nH]c2ncn1 AG-0708 c1c[nH]c2c1c(ncn2)C(=O)O AG-0710 CC(=O)c1ccc(nc1Cl)Cl AG-0712 CCOC(=O)c1c2ccn(c2ncn1)C(=O)OC(C)(C)C AG-0713 c1cc(c(cc1NC(=O)/C=C\C(=O)O)[N+](=O)[O-])Cl AG-0715 c1ccc(cc1)Cc2ccc(nc2)Cl AG-0717 c1cc(c(cc1N2C(=O)C=CC2=O)[N+](=O)[O-])Cl AG-0718 CCOC(=O)c1c(c2c(n1C)cc(cn2)C(F)(F)F)N AG-0721 COC(=O)c1ccc(cc1)Cc2ccc(nc2)Cl AG-0722 COC(=O)c1ccc(cc1)c2ccc(cn2)CO AG-0725 c1cc(c(cc1Br)O)CO AG-0729 COc1ccccc1N2CCN(CC2)CCO.Cl.Cl AH-0024 CC(/C=C\CCCCC(=O)N(C(=O)CCCC/C=C\C(C)C)Cc1cc(c(cc1)O)OC)C AH-0062 c1c(cnc(c1Cl)Nc2c(cc(c(c2[N+](=O)[O-])Cl)[N+](=O)[O-])C(F)(F)F)C(F)(F)F AH-0072 Cc1c(ccc2c1[nH]nc2)[N+](=O)[O-] AH-0082 c1c2c(cc(c1Br)C(F)(F)F)[nH]cc2Cl AH-0701 c1cc(ccc1C(=O)N/N=C/c2cc(ccn2)C(F)(F)F)Cl AH-0704 c1cc\2c(cc1Cl)NC(=O)/C2=C/c3cc(ccn3)C(F)(F)F AH-0705 c1c2c(cc(c1Br)C(F)(F)F)[nH]cc2C=O AH-0711 COc1cc2c(cc1Br)CCC(=O)N2 AH-0713 COC(=O)c1ccc2nc(cn2c1)C(F)(F)F AH-0716 COC(=O)c1cc2ccc(cc2s1)N AH-0717 Cc1c(sc(n1)C(=O)O)C AH-0719 COc1ccc2cc(nc(c2c1)Cl)Cl AH-0722 c1cc(cnc1)C(=O)Nc2ccc(cc2)S(=O)(=O)c3c(cc(cn3)C(F)(F)F)Cl AH-0727 c1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)c3c(cc(cn3)C(F)(F)F)Cl AH-0734 c1ccc(cc1)S(=O)(=O)Cc2cc(ccn2)C(F)(F)F AH-0736 c1cc(ccc1NC(=O)c2ccncc2)S(=O)(=O)c3c(cc(cn3)C(F)(F)F)Cl AH-0741 c1cc(ccc1NCCO)[N+](=O)[O-] AK-0096 CCOC(=O)c1c(c(cc(n1)C)C(F)(F)F)C#N AK-0700 CCOC(=O)c1c(c(ccn1)C(F)(F)F)C#N AK-0703 Cc1cc(cc(c1CC(C(=O)OC)NC(=O)C)C)OC(=O)C AK-0709 CC(C)(C)Oc1ccc(cc1)C[C@@H](C=O)NC(=O)OCC2c3ccccc3-c4c2cccc4 AK-0712 CC(C)(C)OC[C@@H](C(=O)N(C)OC)NC(=O)OCC1c2ccccc2-c3c1cccc3 AK-0715 CC(C)(C)OC[C@@H](C=O)NC(=O)OCC1c2ccccc2-c3c1cccc3 AK-0716 CNc1cc(ncc1C(=O)OC)Cl AK-0717 CN(C(=O)[C@H](Cc1c[nH]c2c1cccc2)NC(=O)OCC3c4ccccc4-c5c3cccc5)OC AK-0718 CCOC(=O)c1cnc2n1cc(cc2I)C AK-0719 CCOC1(CCN(CC1N)C(=O)OC(C)(C)C)OCC AL-0010 c1cc(ncc1C2CC2(F)F)Cl AL-0016 c1ccc(cc1)CN2C(=O)CCC(=N2)c3ccccc3 AL-0202 Cc1cc(c(cc1OCc2ccccc2)N)Br AS-0001 COC(C/N=C/c1ccccc1)OC AS-0002 c1ccc(cc1)P(c2ccccc2)c3ccc(cc3)S(=O)(=O)[O-].[Na+] AS-0003 Cc1ccc(cc1OC)N AS-0004 COc1cc(ccc1CC=O)[N+](=O)[O-] AS-0005 CC(C(=O)c1cccc(c1)Cl)Br AS-0006 CC(C)(C)OC(=O)NCc1ccc(cc1)N AS-0007 Cc1c(cc(cc1C(C)(C)C)C(C)(C)C)CN(C)CCN(C)Cc2cc(cc(c2O)C(C)(C)C)C(C)(C)C AS-0008 C=CCC1C(=NC(=NC1=O)N)O AS-0009 COCOc1ccccc1 AS-0010 CC(C)(C)c1ccc(cc1)C(=O)N AS-0011 CNc1ccc(cc1[N+](=O)[O-])OC AS-0016 c1cc(c(cc1Br)[N+](=O)[O-])N AS-0017 C[n+]1ccc(cc1)CO.[I-] AS-0018 C1[C@H](C2C(O1)[C@@H](CO2)OC(=O)Cl)OC(=O)Cl AS-0019 CCOC(=O)NC(c1cccnc1)NC(=O)OCC AS-0022 CC1=C(CC2C(C1)C(=O)OC2=O)C AS-0028 c1c(cc(c(c1CBr)Cl)Cl)Cl AS-0029 COc1cccc2c1nc(cc2O)C(F)(F)F AS-0032 c1cc2c(cc(nc2c(c1)O)C(F)(F)F)Cl AS-0033 COc1cccc2c1nc(cc2Cl)C(F)(F)F AS-0034 c1ccc(cc1)CN2C(=O)C3CC=CCC3C2=O AS-0035 C[SiH](C)c1ccc(cc1)Cc2ccc(cc2)[SiH](C)C AS-0036 c1cc(ccc1C(c2ccc(cc2)Br)C(Cl)(Cl)Cl)Br AS-0037 CC(=O)c1cc2c(ccc(c2o1)OC)Br AS-0040 CC1(OCCO1)c2cc3c(ccc(c3o2)OC)Br AS-0041 CCOC(=O)CNC(=O)c1ccc(cc1)C(C)(C)C AS-0042 CC1=C(CC2C(C1)C(=O)N(C2=O)Cc3ccccc3)C AS-0043 CCn1c(c(c(=O)n(c1=O)CC)N)N.Cl AS-0045 c1ccc(cc1)/C=C/C(=O)Nc2ccccc2 AS-0046 COc1ccc(cc1OC)c2cc(n3c2c4cc(c(cc4cc3)OC)OC)c5ccccc5 AS-0047 Cc1ccc(cc1Cl)NS(=O)(=O)C AS-0049 c1(c(c(nc(c1F)F)F)F)C(=O)O AS-0050 c1c(c(c(c(n1)F)F)N)F AS-0052 c1c(c(c(cn1)F)N)F AS-0054 CCn1c(cc(=O)n(c1=O)CC)N AS-0055 CCn1c(c(c(=O)n(c1=O)CC)N=O)N AS-0056 c1ccc(cc1)C(=O)NCC(c2ccccc2)(c3ccccc3)O AS-0057 c1ccc(cc1)/C=C/C(=O)N AS-0058 CC1=C(CC(C(C1)C(=O)c2ccccc2)C(=O)O)C AS-0059 COc1cc(cc2c1OC(O2)(c3ccccc3)c4ccccc4)C(=O)Oc5ccc(cc5)[N+](=O)[O-] AS-0060 COc1cc(cc2c1OC(O2)(c3ccccc3)c4ccccc4)C(=O)Oc5cccc(c5)[N+](=O)[O-] AS-0061 COc1cc(cc2c1OC(O2)(c3ccccc3)c4ccccc4)C(=O)OC AS-0062 CCN(CC)C(=O)/C=C/c1ccccc1 AS-0066 CCOC(=O)C(=Cc1ccc(cc1)C)C(=O)OCC AS-0067 c1(c(c(nc(c1F)F)NN)F)N AS-0072 CC(C)(C(C)(C)O[Si](C)(C)C)O[Si](C)(C)C AS-1000 [B-](C#C)(F)(F)F.[K+] AS-1001 [B-](C#Cc1ccccc1)(F)(F)F.[K+] AS-1002 [B-](C#CCCCC)(F)(F)F.[K+] AS-1003 B1(OC(C(O1)(C)C)(C)C)C#C[Si](C)(C)C AS-1004 B1(OC(C(O1)(C)C)(C)C)C#Cc2ccccc2 AS-1005 B1(OC(C(O1)(C)C)(C)C)C#CCCCC AS-1006 B1(OC(C(O1)(C)C)(C)C)C#CCOCc2ccccc2 AS-1007 B1(OC(C(O1)(C)C)(C)C)c2c(nnn2Cc3ccccc3)[Si](C)(C)C AS-1008 Cn1cc([o+]n1)[O-] AS-1009 Cn1c(c([o+]n1)[O-])I AS-1010 Cn1c(c([o+]n1)[O-])C(F)(F)F AS-1011 COc1ccc(cc1)n2cc([o+]n2)[O-] AS-1012 COc1ccc(cc1)n2c(c([o+]n2)[O-])I AS-1013 COc1ccc(cc1)n2c(c([o+]n2)[O-])C(F)(F)F AS-1014 c1cc2c(cc1C(F)(F)F)nc3c(=O)[nH]c(=O)n4c3[n+]2CC4.[Cl-] AS-1015 c1ccc2c(c1)nc3c(=O)[nH]c(=O)n4c3[n+]2CC4.[Cl-] AS-1016 Cn1c(cc(n1)CO)C(F)(F)F AS-1017 Cn1c(cc(n1)CCO)C(F)(F)F AS-1018 Cn1c(cc(n1)CCCO)C(F)(F)F AS-1019 CC(c1cc(n(n1)C)C(F)(F)F)O AS-1020 CC(=O)c1cc(n(n1)C)C(F)(F)F AS-1021 CCOC(=O)c1cc(n(n1)C)C(F)(F)F AS-1022 CC(C)(C)OC(=O)NCc1cc(n(n1)C)C(F)(F)F AS-1023 [B-](c1cc(n[nH]1)c2ccccc2)(F)(F)F.[K+] AS-1024 [B-](c1cc(n[nH]1)c2ccc(cc2)OC)(F)(F)F.[K+] AS-1027 [B-](c1cc(n[nH]1)C(C)(C)C)(F)(F)F.[K+] AS-1028 [B-](c1cc(nn1C)C(C)(C)C)(F)(F)F.[K+] AS-1029 c1ccc(cc1)P(c2ccccc2)c3ccccc3/C=N/C4CCCCC4 AS-2000 CC(C)(C)c1cc(c(c(c1)C(C)(C)C)O)CN2CCN(CC2)Cc3cc(cc(c3O)C(C)(C)C)C(C)(C)C AS-2001 COC(=O)C(=O)[O-].[K+] AS-2003 CCOC(=O)C(=O)[O-].[K+] AS-2004 c1cc(ccc1S(=O)(=O)N2CCOCC2)Br AS-2005 c1c([nH]cn1)C=O AS-2007 CCCCCCCCCCCCCCCCCCOCCO AS-2008 CN1[C@H]2CC3C[C@H]1[C@@H]([C@H]2O)O3 AS-2013 c1csc2c1sc(c2)C=O AS-2014 c1csc2c1scc2 AS-2015 c1c(cn[nH]1)I AS-2016 c1cc2c(cc1Br)non2 AS-2018 CC(C)(C)OC(=O)n1cc(c2c1ncnc2Cl)Br AS-2023 c1ccc(cc1)Cn2cc(c3c2ncnc3Cl)I AS-2025 c1ccc(cc1)Cn2c3ccccc3c4c2ccc(c4)Br AS-2030 Cn1c2ccccc2c3c1ccc(c3)Br AS-2031 c1ccc(cc1)n2c3ccccc3c4c2ccc(c4)Br AS-2032 CCn1c2ccccc2c3c1ccc(c3)Br AS-2033 CC1(c2ccccc2-c3c1cc(cc3)Br)C AS-2034 c1ccc2c(c1)-c3ccc(cc3C2=O)Br AS-2035 CCCCCCc1cc(sc1Br)Br AS-2036 CCCCCCCCCCCCc1ccsc1Br AS-2037 CCCCCCCCCc1ccsc1Br AS-2038 Cc1c(c(n(n1)C)C)I AS-2040 c1c(c2c([nH]1)ncnc2Cl)Cl AS-2041 COC(=O)c1c(ncc(n1)Br)N AS-2042 c1cc2c(cc1Br)nsn2 AS-2043 c1c(c2c([nH]1)ncnc2O)Cl AS-2044 CC(=O)Nc1ccn(c(=O)n1)C2C(C(C(O2)CO)O)O AS-2045 CC(=O)OCC1C(C(C(O1)n2cnc3c2nc(nc3O)N)OC(=O)C)OC(=O)C AS-2047 c1[nH]c2c(n1)c(nc(n2)N)I AS-2048 CC(=O)OC[C@@H]1[C@H]([C@H]([C@@H](O1)n2cnc3c2nc(nc3Cl)Cl)OC(=O)C)OC(=O)C AS-2049 c1nc2c(c(n1)Cl)ncn2[C@H]3[C@@H]([C@@H]([C@H](O3)CO)O)O AS-2050 c1[nH]c2c(n1)c(nc(n2)N)Cl AS-2051 c1ccc(cc1)C(=O)Nc2cc[nH]c(=O)n2 AS-2052 c1c[nH]c2c1c(ncn2)N AS-2057 c1cc(cc(c1)C(=O)O)c2ccc(cc2)Br AS-2061 COc1ccc(cc1)c2cccc(c2)C(=O)O AS-2063 c1cc(cc(c1)C(=O)O)c2ccc(cc2)Cl AS-2064 c1cc(cc(c1)C(=O)O)c2cccc(c2)Br AS-2065 COc1cccc(c1)c2cccc(c2)C(=O)O AS-2066 c1cc(cc(c1)C(=O)O)c2cccc(c2)Cl AS-2067 Cc1ccc(cc1)c2cccc(c2)C(=O)O AS-2068 COC(=O)c1cccc(c1)c2ccc(cc2)Br AS-2073 c1cc(cc(c1)C(=O)O)c2ccc(cc2)C#N AS-2074 COc1ccc(cc1)c2ccc(cc2)Br AS-2078 c1cc(cc(c1)Cl)c2ccc(cc2)C(=O)O AS-2079 c1cc(cc(c1)Br)c2ccc(cc2)C(=O)O AS-2081 c1cc(ccc1c2ccc(s2)C=O)C(=O)O AS-2082 COc1ccccc1c2ccc(cc2)C=O AS-2083 c1cc(cc(c1)C(=O)O)c2ccc(s2)C=O AS-2084 c1cc(ccc1C=O)c2ccc(cc2)Br AS-2085 Cc1ccc(cc1)c2ccc(cc2)C=O AS-2086 COc1cccc(c1)c2ccc(cc2)C=O AS-2089 c1cc(ccc1c2ccc(cc2)F)C(=O)O AS-2091 c1cc(sc1)c2ccc(cc2)C(=O)O AS-2092 COc1ccccc1c2ccc(cc2)C(=O)O AS-2093 C[C@]12CCC3c4ccc(cc4CCC3C1C=C[C@@H]2O)OC AS-2094 c1cc(sc1C=O)c2ccc(s2)Br AS-2096 c1cc(cc(c1)C(=O)O)c2ccc(cc2)F AS-2098 Cc1cccc(c1)c2ccc(cc2)C(=O)O AS-2100 c1ccc2cc(ccc2c1)c3cccc(c3)C(=O)O AS-2101 c1ccc(cc1)c2ccc(cc2)C(=O)O AS-2102 Cc1ccccc1c2ccc(cc2)C(=O)O AS-2104 Cc1cccc(c1)c2cccc(c2)C(=O)O AS-2105 Cc1ccccc1c2cccc(c2)C(=O)O AS-2106 c1cc(cc(c1)C(=O)O)c2ccc(cc2)OC(F)(F)F AS-2107 Cc1ccc(cc1)c2ccc(cc2)C(=O)O AS-2108 c1cc(cc(c1)C(=O)O)c2ccc(cc2)C(F)(F)F AS-2109 c1cc(cc(c1)C(=O)O)c2cccs2 AS-2110 c1cc(ccc1C=O)c2ccc(cc2)F AS-2111 COc1cccc(c1)c2ccc(cc2)C(=O)O AS-2113 c1ccc(c(c1)c2ccc(cc2)C(=O)O)Cl AS-2114 c1cc(cc(c1)F)c2ccc(cc2)C(=O)O AS-2115 c1ccc(c(c1)c2ccc(cc2)C(=O)O)F AS-2118 c1cc(ccc1c2ccc(cc2)C(F)(F)F)C(=O)O AS-2122 c1ccc(cc1)c2ccc(cc2)C=O AS-2124 COc1ccc(cc1)c2cccc(c2)C=O AS-2126 c1cc(cc(c1)F)c2ccc(cc2)C=O AS-2127 Cc1ccccc1c2ccc(cc2)C=O AS-2128 c1cc(cc(c1)Cl)c2ccc(cc2)C=O AS-2129 Cc1cccc(c1)c2ccc(cc2)C=O AS-2130 c1ccc(c(c1)c2ccc(cc2)C=O)Cl AS-2138 c1cc(cc(c1)c2ccc(cc2)Cl)C=O AS-2143 c1cc(cc(c1)Br)c2ccc(cc2)C=O AS-2146 Cc1ccc(cc1c2ccc(cc2)OC)C(=O)O AS-2148 c1cc(ccc1c2ccc(cc2)Br)Cl AS-2149 c1ccc(cc1)c2cccc(c2)CN.Cl AS-2150 Cc1cccc(c1)c2cccc(c2)CO AS-2151 Cc1ccc(cc1)c2cccc(c2)CO AS-2153 c1cc(cc(c1)c2cccc(c2)C(F)(F)F)CO AS-2157 c1cc(cc(c1)c2cccc(c2)Cl)CO AS-2158 CO[Si](C)(C)c1ccccc1 AS-2164 CO[Si](C)(C)c1ccc(cc1)Cl AS-2166 C[Si](C)(C)c1ccccc1 AS-2175 C[Si](C)(C)Cc1ccccc1 AS-2177 C[Si](C)(c1ccccc1)O[Si](C)(C)c2ccccc2 AS-2182 COc1ccc(cc1)[Si](C)(C)O[Si](C)(C)c2ccc(cc2)OC AS-2192 C[Si](C)(c1ccc(cc1)[Si](C)(C)O)O AS-2195 COc1ccccc1[Si](C)(C)[Si](C)(C)c2ccccc2OC AS-2199 C[Si](C)(c1cccs1)[Si](C)(C)c2cccs2 AS-2202 COc1ccc(cc1)[Si](C)(C)c2ccccc2CO AS-2209 C[Si](C)(c1ccccc1CO)c2cccs2 AS-2210 C[Si](C)(c1ccc(cc1)F)c2ccccc2CO AS-2211 C[Si](C)(c1ccc(cc1)Cl)c2ccccc2CO AS-2212 C[Si]1(c2ccccc2CO1)C AS-2213 C[Si](C)(c1ccc(cc1)C#N)c2ccccc2CO AS-2215 C[Si](C)(c1ccc(nc1)Cl)c2ccccc2CO AS-2217 COc1ccccc1[Si](C)(C)c2ccccc2CO AS-2218 COc1cccc(c1)[Si](C)(C)c2ccccc2CO AS-2220 C[Si](C)(c1ccc(cc1)SC)c2ccccc2CO AS-2221 Cc1ccc(cc1)[Si](C)(C)c2ccccc2CO AS-2222 C[Si](C)(c1ccc(cc1)Br)c2ccccc2CO AS-2224 COc1ccc(cc1OC)[Si](C)(C)c2ccccc2CO AS-2225 C[Si](C)(c1ccc2c(c1)OCO2)c3ccccc3CO AS-2226 C[Si](C)(c1ccccc1CO)c2cccc3c2cccc3 AS-2229 C[Si](C)(c1ccc(cc1)c2ccccc2)c3ccccc3CO AS-2230 C[Si](C)(c1ccc(cc1)C(=O)N2CCOCC2)c3ccccc3CO AS-2232 C[Si](C)(c1ccc(cc1)Oc2ccccc2)c3ccccc3CO AS-2234 Cc1cc(c(c(c1)C)[Si](C)(C)c2ccccc2CO)C AS-2236 Cc1ccccc1[Si](C)(C)c2ccccc2CO AS-2237 CN1CCN(CC1)c2ccc(cc2)[Si](C)(C)c3ccccc3CO AS-2239 C[Si](C)(c1ccc-2c(c1)Cc3c2cccc3)c4ccccc4CO AS-2242 C[Si](C)(Cc1ccccc1)c2ccccc2CO AS-2248 C[Si](C)(c1ccc(cc1)Cc2ccccc2)c3ccccc3CO AS-2251 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)non3 AS-2253 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N3CCCCC3 AS-2254 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N3CCOCC3 AS-2255 B1(OC(C(O1)(C)C)(C)C)c2ccccc2 AS-2256 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C AS-2257 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)O AS-2258 B(c1ccccc1)(O)O AS-2259 B(c1ccc(cc1)C)(O)O AS-2260 B(c1ccc(cc1)C(=O)O)(O)O AS-2261 B(c1ccc(cc1)C#N)(O)O AS-2262 B(c1ccc(cc1)C(=O)OC)(O)O AS-2263 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C=O AS-2264 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#N AS-2265 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)OC AS-2266 B(c1ccc(cc1)C=O)(O)O AS-2267 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N3CCCC3 AS-2268 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCc3ccco3 AS-2269 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N3CCCC(C3)C(=O)OCC AS-2270 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N3CCCC3 AS-2271 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N3CCCCC3 AS-2272 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N3CCN(CC3)C AS-2273 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N3CCOCC3 AS-2274 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)NCc3ccco3 AS-2275 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCN(CC3)C AS-2276 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)Cc3ccccc3 AS-2277 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCOCC3 AS-2278 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN3CCN(CC3)C AS-2279 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)Cc3ccccc3 AS-2280 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN3CCOCC3 AS-2281 B(c1cccc(c1)C=O)(O)O AS-2282 B(c1cccc(c1)C(=O)O)(O)O AS-2283 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCCOC AS-2284 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N3CCN(CC3)C(=O)OC(C)(C)C AS-2285 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)O AS-2286 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C=O AS-2287 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N3CCN(CC3)C AS-2288 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)NCCOC AS-2289 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N3CCN(CC3)C(=O)OC(C)(C)C AS-2290 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)NCc3ccccc3 AS-2291 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)NCC3CCCO3 AS-2292 B(c1ccc(s1)C=O)(O)O AS-2293 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCc3ccccc3 AS-2294 B1(OC(C(O1)(C)C)(C)C)c2ccc(s2)C=O AS-2295 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CNc3ccccc3 AS-2296 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCC3CCCO3 AS-2297 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CO AS-2298 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/c3ccccc3 AS-2299 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)c3ccccc3 AS-2300 B1(OC(C(O1)(C)C)(C)C)c2ccc(s2)CN3CCOCC3 AS-2301 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)N AS-2302 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CNc3ccccc3 AS-2303 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(c3ccccc3)C(=O)OC(C)(C)C AS-2304 B1(OC(C(O1)(C)C)(C)C)c2ccccc2C=O AS-2305 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(c3nccs3)O AS-2306 B(c1ccc(cc1)C(=O)OCC)(O)O AS-2307 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)NC(=O)OC(C)(C)C AS-2308 B(c1ccc(cc1)Br)(O)O AS-2310 B(c1ccc(cc1)I)(O)O AS-2311 B(c1cccc(c1)Br)(O)O AS-2312 B(c1cccc(c1)I)(O)O AS-2313 [B-](c1ccc(cc1)Br)(F)(F)F.[K+] AS-2314 [B-](c1ccc(cc1)I)(F)(F)F.[K+] AS-2315 [B-](c1cccc(c1)Br)(F)(F)F.[K+] AS-2316 [B-](c1cccc(c1)I)(F)(F)F.[K+] AS-2317 [B-](c1ccc(cc1)C=O)(F)(F)F.[K+] AS-2318 [B-](c1cccc(c1)C=O)(F)(F)F.[K+] AS-2319 [B-](c1ccccc1C=O)(F)(F)F.[K+] AS-2320 [B-](c1ccc(s1)C=O)(F)(F)F.[K+] AS-2321 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)I AS-2322 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)I AS-2323 [B-](c1ccc2c(c1)non2)(F)(F)F.[K+] AS-2324 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N(C)OC AS-2325 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N(C)OC AS-2326 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/c3ccc(cc3)OC AS-2327 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)Nc3ccccc3 AS-2328 B(c1ccc(cc1)OC)(O)O AS-2329 B(c1cccc(c1)OC)(O)O AS-2330 B(c1ccccc1OC)(O)O AS-2331 B(c1ccc(cc1)F)(O)O AS-2332 B(c1ccc(cc1)Cl)(O)O AS-2333 [B-](c1ccccc1)(F)(F)F.[K+] AS-2334 [B-](c1ccccc1OC)(F)(F)F.[K+] AS-2335 [B-](c1cccc(c1)OC)(F)(F)F.[K+] AS-2336 [B-](c1ccc(cc1)OC)(F)(F)F.[K+] AS-2337 [B-](c1ccc(cc1)C(=O)N2CCOCC2)(F)(F)F.[K+] AS-2338 [B-](c1ccc(cc1)C(=O)OCC)(F)(F)F.[K+] AS-2339 [B-](c1cccc(c1)C(=O)N2CCOCC2)(F)(F)F.[K+] AS-2340 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N(CC)CC AS-2341 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N(CC)CC AS-2342 [B-](c1cccc(c1)C(=O)O)(F)(F)F.[K+] AS-2343 [B-](c1ccc(cc1)C(=O)O)(F)(F)F.[K+] AS-2344 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/Cc3ccco3 AS-2345 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/C(C)(C)C AS-2346 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/C3CCCC3 AS-2347 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/C3CCCCC3 AS-2348 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/C3CCCCCC3 AS-2349 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/Cc3ccccc3 AS-2350 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCCCC3 AS-2351 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCCC3 AS-2352 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCN(CC3)C(=O)OC(C)(C)C AS-2353 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCCCCC3 AS-2354 B1(OC(C(O1)(C)C)(C)C)c2ccc(s2)CN3CCN(CC3)C(=O)OC(C)(C)C AS-2355 B1(OC(C(O1)(C)C)(C)C)c2ccc(s2)CN3CCCCC3 AS-2356 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)/N=C/c3ccc(cc3)OC AS-2358 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CNC(C)(C)C AS-2359 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C=C3C(=O)N(C(=O)N(C3=O)C)C AS-2360 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=C(\C#N)/C(=O)OCC AS-2361 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CC3C(=O)N(C(=O)N(C3=O)C)C AS-2362 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CNCc3ccco3 AS-2363 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CNC3CCCCC3 AS-2365 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CO AS-2366 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCC#C AS-2367 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)NCC#C AS-2368 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(c3nccs3)O AS-2369 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)O AS-2371 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)N3CCN(CC3)C AS-2372 B1(OC(C(O1)(C)C)(C)C)B2OC(C(O2)(C)C)(C)C AS-2373 B1(OC(C(O1)(C)C)(C)C)c2ccoc2 AS-2374 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)Cl AS-2375 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)NC(=O)CCC(=O)O AS-2376 B1(c2ccccc2CO1)O AS-2377 B(c1ccc(cc1)C(=O)OCCC)(O)O AS-2378 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)NC(=O)CNC(=O)OC(C)(C)C AS-2379 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)OC AS-2380 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)OCc3ccccc3 AS-2381 B1(OC(C(O1)(C)C)(C)C)c2ccnn2C3CCCCO3 AS-2382 [B-](c1ccc(cc1)C(=O)N2CCCCC2)(F)(F)F.[K+] AS-2383 [B-](c1ccc(cc1)C(=O)NCc2ccco2)(F)(F)F.[K+] AS-2384 [B-](c1ccc(cc1)C(=O)NCCOC)(F)(F)F.[K+] AS-2385 [B-](c1ccc(cc1)CNc2ccccc2)(F)(F)F.[K+] AS-2386 [B-](c1ccc(cc1)C(=O)Nc2ccccc2)(F)(F)F.[K+] AS-2387 [B-](c1cccc(c1)C(=O)N2CCCCC2)(F)(F)F.[K+] AS-2389 [B-](c1cccc(c1)C(=O)NCc2ccco2)(F)(F)F.[K+] AS-2390 [B-](c1cccc(c1)C(=O)NCCOC)(F)(F)F.[K+] AS-2391 [B-](c1cccc(c1)C(=O)Nc2ccccc2)(F)(F)F.[K+] AS-2392 [B-](c1ccsc1)(F)(F)F.[K+] AS-2393 B1(OC(C(O1)(C)C)(C)C)c2ccc3cc(ccc3c2)OCCCC AS-2395 B1(OC(C(O1)(C)C)(C)C)c2ccc3cc(ccc3c2)OCC(C)C AS-2396 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)B3OC(C(O3)(C)C)(C)C AS-2397 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCc3ccccc3 AS-2398 B1(OC(C(O1)(C)C)(C)C)c2cccc3c2nccc3 AS-2399 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CBr AS-2400 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)OCCOC AS-2401 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)B3OC(C(O3)(C)C)(C)C AS-2402 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)OCc3ccccc3 AS-2403 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C=C3C(=O)N(C(=O)N(C3=O)C)C AS-2404 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CBr AS-2405 B1(OC(C(O1)(C)C)(C)C)c2ccc(c(c2)C=O)OCc3ccccc3 AS-2406 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#Cc3ccccc3 AS-2407 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#C[Si](C)(C)C AS-2408 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C#C[Si](C)(C)C AS-2409 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#Cc3ccc(cc3)B4OC(C(O4)(C)C)(C)C AS-2410 B1(OC(C(O1)(C)C)(C)C)c2ccc(s2)C=C3C(=O)N(C(=O)N(C3=O)C)C AS-2411 B1(OC(C(O1)(C)C)(C)C)c2ccc(s2)/C=N/c3ccccc3 AS-2412 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#C AS-2413 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCCCO AS-2414 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#Cc3ccc(cc3)C(=O)OC AS-2415 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#CCO AS-2416 [B-](c1ccc(cc1)OCc2ccccc2)(F)(F)F.[K+] AS-2417 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C#C AS-2418 [B-](c1ccc(cc1)C(=O)N(CC)CC)(F)(F)F.[K+] AS-2419 [B-](c1ccc(cc1)C(=O)N2CCCC2)(F)(F)F.[K+] AS-2420 [B-](c1ccc(cc1)CN2CCOCC2)(F)(F)F.[K+] AS-2421 [B-](c1ccc(cc1)C(=O)NCc2ccccc2)(F)(F)F.[K+] AS-2422 [B-](c1ccc(cc1)C(=O)N(C)OC)(F)(F)F.[K+] AS-2424 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)N3CCOCC3 AS-2425 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)N3CCCCC3 AS-2426 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#Cc3ccc(cc3)OC AS-2427 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C#Cc3ccc(cc3)Cl AS-2428 [B-](c1ccc(cc1)CO)(F)(F)F.[K+] AS-2430 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CP(c3ccccc3)(c4ccccc4)(c5ccccc5)Br AS-2431 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NN3CCN(CC3)C AS-2432 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NN3CCOCC3 AS-2433 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CP(c3ccccc3)(c4ccccc4)(c5ccccc5)Br AS-2435 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)c3ccc(cc3)OC AS-2436 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)c3ccc(cc3)Cl AS-2437 B1(OC(C(O1)(C)C)(C)C)c2c3ccccc3c(c4c2cccc4)B5OC(C(O5)(C)C)(C)C AS-2438 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCc4ccccc4C3 AS-2439 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3C(=O)CCC3=O AS-2440 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)Nc3ccc(cc3)Cl AS-2441 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN3CCN(CC3)C(=O)OC(C)(C)C AS-2442 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN3CCN(CC3)c4ccccc4 AS-2443 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(CCOC)CCOC AS-2444 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCN(CC3)c4ccccc4 AS-2445 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)c4ccccc4n3Cc5ccccc5 AS-2446 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)ccn3Cc4ccccc4 AS-2447 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)N(c3ccccc3)c4ccccc4 AS-2448 B1(OC(C(O1)(C)C)(C)C)c2ccc-3c(c2)Cc4c3cccc4 AS-2449 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)n3c4ccccc4c5c3cccc5 AS-2450 B1(OC(C(O1)(C)C)(C)C)c2cn(c3c2cccn3)Cc4ccccc4 AS-2451 B1(OC(C(O1)(C)C)(C)C)c2ccc-3c(c2)C(c4c3cccc4)(C)C AS-2452 B1(OC(C(O1)(C)C)(C)C)c2ccc-3c(c2)C(=O)c4c3cccc4 AS-2453 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)c4ccccc4n3C AS-2454 B1(OC(C(O1)(C)C)(C)C)c2ccc-3c(c2)C(c4c3cccc4)(CCCCCCCC)CCCCCCCC AS-2455 B1(OC(C(O1)(C)C)(C)C)c2ccc-3c(c2)C(c4c3ccc(c4)B5OC(C(O5)(C)C)(C)C)(C)C AS-2456 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)c3ccc(cc3)B4OC(C(O4)(C)C)(C)C AS-2457 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)c4ccccc4n3c5ccccc5 AS-2459 B1(OC(C(O1)(C)C)(C)C)c2ccc-3c(c2)C(c4c3ccc(c4)B5OC(C(O5)(C)C)(C)C)(CCCCCCCC)CCCCCCCC AS-2460 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3C(=O)c4ccccc4C3=O AS-2462 B(c1ccc(cc1)C(=O)N2CCOCC2)(O)O AS-2463 B(c1ccc(cc1)OCc2ccccc2)(O)O AS-2468 B(c1cccc(c1)OCc2ccccc2)(O)O AS-2469 B(c1ccc(cc1)N(c2ccccc2)c3ccccc3)(O)O AS-2471 B(c1ccc-2c(c1)C(c3c2cccc3)(C)C)(O)O AS-2472 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)nsn3 AS-2473 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NC3CCCC3 AS-2474 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NC3CC3 AS-2475 B1(OC(C(O1)(C)C)(C)C)c2ccccc2CBr AS-2478 B1(OC(C(O1)(C)C)(C)C)c2ccccc2CN3C(=O)c4ccccc4C3=O AS-2480 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)Cn3cccn3 AS-2481 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(Cc3ccccc3)Cc4ccccc4 AS-2482 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NOCc3ccccc3 AS-2483 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)COc3ccccc3 AS-2484 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)Cn3c4ccccc4c5c3cccc5 AS-2486 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)c4ccccc4n3CC AS-2487 B(c1cccc(c1)O)(O)O AS-2488 B(c1ccc(cc1)CCCC)(O)O AS-2489 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)O AS-2490 [B-](c1ccc(cc1)CCCC)(F)(F)F.[K+] AS-2494 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2C)C AS-2495 B(c1cccc(c1C)C)(O)O AS-2496 B(c1ccc(cc1)C=C)(O)O AS-2498 [B-](c1ccc-2c(c1)C(c3c2cccc3)(C)C)(F)(F)F.[K+] AS-2500 [B-](c1cccc(c1)CO)(F)(F)F.[K+] AS-2503 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)COCCOC AS-2504 B(c1cccc(c1)N)(O)O AS-2507 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C AS-2508 B(c1ccc(cc1)C(F)(F)F)(O)O AS-2509 B(c1ccc(cc1)OC(F)(F)F)(O)O AS-2510 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)Cl AS-2511 B(c1cccc(c1)C)(O)O AS-2512 B(c1cccc(c1)Cl)(O)O AS-2513 B(c1ccccc1C)(O)O AS-2514 B(c1ccccc1C=O)(O)O AS-2515 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)Br AS-2516 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OC(F)(F)F AS-2517 B1(OC(C(O1)(C)C)(C)C)c2ccccc2C AS-2518 [B-](c1cccs1)(F)(F)F.[K+] AS-2519 B(c1ccc-2c(c1)C(c3c2ccc(c3)B(O)O)(C)C)(O)O AS-2520 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CC3CCCCC3 AS-2521 B1(OC(C(O1)(C)C)(C)C)c2ccc3cc(ccc3c2)C(C)(C)C AS-2523 B(c1ccc(cc1)S(=O)(=O)C)(O)O AS-2524 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN3C(=O)c4ccccc4C3=O AS-2525 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN3C(=O)CCC3=O AS-2526 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)Cn3cccn3 AS-2527 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)COC AS-2528 B1(OC(C(O1)(C)C)(C)C)c2c(ccs2)CCCCCC AS-2529 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)N3C(=O)C=CC3=O AS-2530 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)I AS-2531 B1(Nc2cccc3c2c(ccc3)N1)c4cccs4 AS-2532 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)Br AS-2533 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)C#C AS-2535 B1(OC(C(O1)(C)C)(C)C)c2c(ccs2)CCCCCCCCC AS-2536 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(nc4)Cl AS-2538 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)C#C[Si](C)(C)C AS-2539 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/O AS-2540 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)C(=O)O AS-2541 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN=[N+]=[N-] AS-2542 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C3Nc4cccc5c4c(ccc5)N3 AS-2543 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C#Cc3cccc(c3)B4OC(C(O4)(C)C)(C)C AS-2546 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN=[N+]=[N-] AS-2547 [B-](c1ccc(cc1)CN=[N+]=[N-])(F)(F)F.[K+] AS-2548 B1(OC(C(O1)(C)C)(C)C)c2ccccc2CN=[N+]=[N-] AS-2549 B1(OC(C(O1)(C)C)(C)C)c2cc(ccc2C)C(=O)OC AS-2552 [B-](c1cccc(c1)CN=[N+]=[N-])(F)(F)F.[K+] AS-2555 B1(OC(C(O1)(C)C)(C)C)c2cccs2 AS-2556 [B-](c1ccccc1CN=[N+]=[N-])(F)(F)F.[K+] AS-2559 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCSCC3 AS-2562 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN.Cl AS-2563 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCOCC3.Cl AS-2564 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN3CCCC3.Cl AS-2566 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(C)C.Cl AS-2567 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN.Cl AS-2568 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)B3OC(C(O3)(C)C)(C)C)B4OC(C(O4)(C)C)(C)C AS-2569 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)OC)OC AS-2570 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)Br)Br AS-2571 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)Br)OC AS-2572 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OC AS-2574 B1(OC(C(O1)(C)C)(C)C)c2ccccc2OC AS-2576 [B-](c1cccc2c1cccc2)(F)(F)F.[K+] AS-2577 [B-](c1ccc(cc1)C)(F)(F)F.[K+] AS-2578 [B-](c1ccc(cc1)O)(F)(F)F.[K+] AS-2579 [B-](c1cccc(c1)C)(F)(F)F.[K+] AS-2580 [B-](c1ccc(cc1)F)(F)(F)F.[K+] AS-2582 [B-](c1cccc(c1)F)(F)(F)F.[K+] AS-2583 [B-](c1ccc(cc1)C#N)(F)(F)F.[K+] AS-2584 [B-](c1ccc(cc1)C(F)(F)F)(F)(F)F.[K+] AS-2585 [B-](c1ccccc1C)(F)(F)F.[K+] AS-2586 [B-](c1ccc2ccccc2c1)(F)(F)F.[K+] AS-2587 [B-](c1cccnc1)(F)(F)F.[K+] AS-2588 [B-](c1ccc(nc1)Cl)(F)(F)F.[K+] AS-2589 [B-](c1ccc(s1)Br)(F)(F)F.[K+] AS-2590 B(c1cccc(c1)C#N)(O)O AS-2591 B(c1cccc(c1)F)(O)O AS-2592 B(c1cccnc1)(O)O AS-2593 B(c1ccccc1Cl)(O)O AS-2594 B(c1ccccc1F)(O)O AS-2595 [B-](c1ccc(cc1)Cl)(F)(F)F.[K+] AS-2597 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)N3C(=O)C4C5CC(C4C3=O)C=C5 AS-2598 B1(OC(C(O1)(C)C)(C)C)c2ccccc2Cl AS-2599 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)c3ccccc3OC AS-2600 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)COC AS-2601 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C[NH+]3CCCCC3.[Cl-] AS-2602 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCCOC AS-2603 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)NC(=O)C AS-2604 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)N AS-2605 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)O AS-2606 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)NC=O AS-2608 B(c1cc(cc(c1)Br)Br)(O)O AS-2609 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)NC(=O)OC(C)(C)C AS-2611 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CN3CCOCC3.Cl AS-2612 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C[NH+]3CCCCCC3.[Cl-] AS-2613 B1(OC(C(O1)(C)C)(C)C)c2ccccc2CN.Cl AS-2615 B(c1ccccc1OCc2ccccc2)(O)O AS-2616 B1(OC(C(O1)(C)C)(C)C)c2ccccc2OCc3ccccc3 AS-2617 B(c1ccc2ccccc2c1)(O)O AS-2618 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)F AS-2619 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)Cl AS-2620 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)Br AS-2621 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(CC)CC.Cl AS-2622 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(CCC)CCC.Cl AS-2623 B(c1ccc(cc1)SC)(O)O AS-2624 B(c1cc(ccc1OC)F)(O)O AS-2625 B(c1ccc(c(c1)C)F)(O)O AS-2626 B(c1cc2ccccc2o1)(O)O AS-2627 B(c1ccc(cc1)CC)(O)O AS-2628 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)SC AS-2629 B1(OC(C(O1)(C)C)(C)C)c2cc(ccc2OC)F AS-2630 B1(OC(C(O1)(C)C)(C)C)c2ccc(c(c2)C)F AS-2631 B1(OC(C(O1)(C)C)(C)C)c2cc3ccccc3o2 AS-2632 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)c3ccc(cc3)C=O AS-2633 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(C)Cc3ccccc3.Cl AS-2634 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CC AS-2635 B1(OCC(CO1)(C)C)B2OCC(CO2)(C)C AS-2636 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)c3ccc(cc3)C=O AS-2637 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(C)Br AS-2638 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(C)[NH+]3CCOCC3.[Cl-] AS-2639 B1(c2cc(ccc2CO1)C(=O)O)O AS-2640 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)c3cccc(c3)C(=O)OC AS-2641 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(C)N3CCOCC3 AS-2642 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CN(C)c3ccccc3 AS-2643 B(c1c2ccccc2cc3c1cccc3)(O)O AS-2644 B1(OC(C(O1)(C)C)(C)C)c2ccc3ccccc3c2 AS-2646 B1(OC(C(O1)(C)C)(C)C)c2cccc3c2cccc3 AS-2647 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)F AS-2648 B(c1cccc2c1cccc2)(O)O AS-2649 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CCCC AS-2650 B(c1cccc(c1)C(F)(F)F)(O)O AS-2651 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(F)(F)F AS-2653 B1(OC(C(O1)(C)C)(C)C)c2ccsc2 AS-2654 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)C AS-2655 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(C)N=[N+]=[N-] AS-2656 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CNCCOC AS-2657 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(C)O AS-2658 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)N(CC)C(C)C AS-2659 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)COCC=C AS-2660 B(c1ccc(cc1)O)(O)O AS-2661 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)C AS-2662 B1(OC(C(O1)(C)C)(C)C)c2cccnc2 AS-2663 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)NC3CCCC3 AS-2664 B1(OC(C(O1)(C)C)(C)C)c2c3ccccc3cc4c2cccc4 AS-2666 [B-](c1ccc(cc1)Cn2cnc3c2ncnc3Cl)(F)(F)F.[K+] AS-2672 [B-](c1cccc(c1)NC(=O)C)(F)(F)F.[K+] AS-2674 [B-](c1cc(ccc1OC)F)(F)(F)F.[K+] AS-2676 [B-](c1cccc(c1C)C)(F)(F)F.[K+] AS-2677 [B-](c1cccc(c1)C#N)(F)(F)F.[K+] AS-2678 [B-](c1cccc(c1)Cl)(F)(F)F.[K+] AS-2679 [B-](c1cccc(c1)OCc2ccccc2)(F)(F)F.[K+] AS-2680 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)Cn3ccnc3 AS-2682 [B-](c1ccc(cc1)C(C)(C)C)(F)(F)F.[K+] AS-2683 [B-](c1ccccc1OCc2ccccc2)(F)(F)F.[K+] AS-2685 [B-](c1ccc(c(c1)C=O)OC)(F)(F)F.[K+] AS-2686 [B-](c1ccccc1Cl)(F)(F)F.[K+] AS-2687 [B-](c1cc(cc(c1)Br)Br)(F)(F)F.[K+] AS-2688 [B-](c1ccc(cc1)OC(F)(F)F)(F)(F)F.[K+] AS-2689 [B-](c1cccc(c1)C(F)(F)F)(F)(F)F.[K+] AS-2690 B(c1ccccc1C#N)(O)O AS-2691 [B-](c1ccc(cc1)S(=O)(=O)C)(F)(F)F.[K+] AS-2692 [B-](c1cc(cc(c1)Cl)Cl)(F)(F)F.[K+] AS-2693 [B-](c1cc(cc(c1)C(F)(F)F)C(F)(F)F)(F)(F)F.[K+] AS-2694 [B-](c1ccc(cc1)SC)(F)(F)F.[K+] AS-2695 [B-](c1ccc(c(c1)Cl)F)(F)(F)F.[K+] AS-2696 [B-](c1ccc2c(c1)OCO2)(F)(F)F.[K+] AS-2697 [B-](c1ccccc1C#N)(F)(F)F.[K+] AS-2698 [B-](c1ccc(cc1Cl)Cl)(F)(F)F.[K+] AS-2699 CCCCCCCCc1ccc(cc1)c2ccc(cc2)C#N AS-2700 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)OC AS-2706 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)Cl AS-2707 B1(Nc2cccc3c2c(ccc3)N1)c4cccc(c4)I AS-2708 B1(Nc2cccc3c2c(ccc3)N1)c4cccc(c4)C AS-2709 B1(Nc2cccc3c2c(ccc3)N1)c4cccc(c4)OC AS-2710 B1(Nc2cccc3c2c(ccc3)N1)c4cccc(c4)Cl AS-2711 B1(Nc2cccc3c2c(ccc3)N1)c4cc(cc(c4)Br)Br AS-2712 [B-](c1cccc(c1)[N+](=O)[O-])(F)(F)F.[K+] AS-2713 B1(Nc2cccc3c2c(ccc3)N1)c4ccc(cc4)C5Nc6cccc7c6c(ccc7)N5 AS-2714 B(c1cccc(c1)[N+](=O)[O-])(O)O AS-2715 [B-](c1ccncc1)(F)(F)F.[K+] AS-2716 c1cc(sc1C=O)c2ccc(s2)c3ccc(s3)Br AS-2717 CC(C)(C)OC(=O)NNC(C)(C)C[N+](=O)[O-] AS-2718 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)N3CCN(CC3)C AS-2719 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)NC3CCCCC3 AS-2720 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)N3CCOCC3 AS-2721 [B-](CC)(F)(F)F.[K+] AS-2722 B1(OC(C(O1)(C)C)(C)C)c2ccccc2C#N AS-2723 [B-](c1cc(cc(c1)Br)OC)(F)(F)F.[K+] AS-2724 c1cc(ccc1c2ccc(cc2)N)C(=O)O AS-2725 [B-](c1ccc(cc1)C(=O)NCC#C)(F)(F)F.[K+] AS-2726 [B-](c1cc2ccccc2o1)(F)(F)F.[K+] AS-2727 B(c1cc(ccc1I)OC)(O)O AS-2728 [B-](c1ccc(cc1)c2ccc(cc2)OC)(F)(F)F.[K+] AS-2729 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C#N AS-2730 [B-](c1ccc(cc1)C(=O)C)(F)(F)F.[K+] AS-2731 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)/C=C(\C#N)/C(=O)OCC AS-2732 [B-](c1c(cccc1F)F)(F)(F)F.[K+] AS-2733 [B-](c1cccc(c1)N)(F)(F)F.[K+] AS-2734 CC(=O)Nc1ccc(cc1[N+](=O)[O-])C=O AS-2735 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)NCc3ccccc3 AS-2736 c1cc2c(cc1Br)CCCO2 AS-2737 COCCNCc1ccc(cc1)OC AS-2738 CN1CCN(CC1)S(=O)(=O)c2ccc(cc2)Br AS-2764 c1cc(ccc1C(=O)c2ccc(cc2)F)N AS-2765 c1cc(ccc1C(=O)c2ccc(cc2)Br)[N+](=O)[O-] AS-2766 COC(=O)COc1ccc(cc1)I AS-2768 CCOC(=O)N1CCN(CC1)c2ccc(c(c2)N)[N+](=O)[O-] AS-2769 CN(C)CCNc1ccc(c(c1)N)[N+](=O)[O-] AS-2770 c1cc(c(cc1N2CCN(CC2)CCO)N)[N+](=O)[O-] AS-2771 c1cc(sc1)c2ccc(s2)c3ccc(s3)C=O AS-2779 Cc1ccc(cc1)c2ccc(c(c2)C(=O)O)O AS-2780 CCN(CC)S(=O)(=O)c1ccc(cc1)Br AS-2782 CCCCC(CC)COc1ccc(cc1)Br AS-2783 CC(C)(C)OC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(cc2)Br AS-2784 CC(C)(C)OC(=O)n1ccc2c1cc(cc2)Br AS-2785 c1cc(c(cc1N2CCSCC2)N)[N+](=O)[O-] AS-2787 CC(=O)OCCOc1ccc(cc1)Br AS-2789 CCOC(=O)c1coc(n1)C AS-2805 c1cc(ccc1S(=O)(=O)N2CCCCC2)Br AS-2817 [B-](c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)C)(F)(F)F.[B-](c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)C)(F)(F)F.O.[K+].[K+] AS-2840 [B-](c1ccc(cc1)Cc2ccccc2)(F)(F)F.[K+] AS-2841 [B-](c1cccc(c1)CN2CCN(CC2)C)(F)(F)F.CCCC[N+](CCCC)(CCCC)CCCC AS-2846 CCCCC(CC)COc1ccccc1 AS-2847 COCCNc1ccc(c(c1)N)[N+](=O)[O-] AS-2873 c1ccc(cc1)c2ccc(cc2)CC(=O)O AS-2883 CC(=O)OCCCOc1ccc(cc1)Br AS-2903 COCCOc1cc(ccc1C#N)Br AS-2908 COCCOc1ccc(cc1[N+](=O)[O-])Br AS-2910 c1cc(c(cc1Br)OCc2ccoc2)C#N AS-2911 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCC AS-2944 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N(CCC)CCC AS-2946 c1cc(cc(c1)[N+](=O)[O-])C#CCO AS-2950 CCCOc1cc(ccc1C#N)Br AS-2965 CC(C)CCOc1cc(ccc1C#N)Br AS-2967 CCCCOc1cc(ccc1C#N)Br AS-2969 c1cc(c(cc1Br)NCCCCO)C#N AS-2977 [B-](c1cccc(c1)CN2C(=O)c3ccccc3C2=O)(F)(F)F.[K+] AS-3003 c1cc(c(cc1Br)N2CCOCC2)C#N AS-3005 c1cc2c(cc1Br)c(=O)nc[nH]2 AS-3007 COCCOC(=O)NC(=O)Nc1ccc(cc1)I AS-3038 c1c(c2c(ncnc2[nH]1)N)I AS-3045 c1ccc-2c(c1)-c3cccc4c3c2ccc4Br AS-3074 CC(=O)Oc1cc(ccc1OC)Br AS-3075 COc1ccccc1c2cccc(c2)C(=O)OC AS-3076 c1cc(ncc1Br)I AS-3077 c1cc(=O)oc2c1cc(cc2)Br AS-3079 CC1(CC(c2ccccc2O1)(C)c3ccc(cc3)O)C AS-3083 c1cc(=O)oc2c1cc(cc2)[N+](=O)[O-] AS-3090 CC(=O)c1ccc(cc1)c2ccc(cc2)C(F)(F)F AS-3101 COc1cc2cc([nH]c2c(c1OC)OC)C(=O)O AS-3102 B1(OC(C(O1)(C)C)(C)C)CC(C)C AS-3112 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)NC(C)COC AS-3113 B1(OC(C(O1)(C)C)(C)C)c2cccnc2Cl AS-3114 B1(OC(C(O1)(C)C)(C)C)c2cccnc2N3CCCC3 AS-3115 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)NC(CC)CC AS-3116 c1ccc(cc1)Cn2cc(ccc2=O)Br AS-3117 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)NCC=C AS-3118 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(C)(C)C(=O)OC AS-3119 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)NCCCC AS-3120 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)NCC(C)C AS-3121 B(c1ccc(cc1)c2ccc(cc2)OC)(O)O AS-3122 B1(OC(C(O1)(C)C)(C)C)c2ccccc2CC(C)C AS-3123 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCCC AS-3124 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)Cc3ccc(cc3)Cl AS-3125 B1(OC(C(O1)(C)C)(C)C)c2ccc(nc2)NC AS-3126 [B-](c1ccc(cc1)N(c2ccccc2)c3ccccc3)(F)(F)F.[K+] AS-3127 B1(OC(C(O1)(C)C)(C)C)c2ccc3cc(ccc3c2)OCc4ccccc4 AS-3128 B1(OC(C(O1)(C)C)(C)C)c2ccc(c(c2)C(=O)OC)O AS-3129 B1(OC(C(O1)(C)C)(C)C)c2ccc3cc(ccc3c2)OC(=O)C AS-3130 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)S(=O)(=O)N AS-3131 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)S(=O)(=O)N3CCN(CC3)C AS-3132 B(c1ccc-2c3c1cccc3-c4c2cccc4)(O)O AS-3133 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)OCC AS-3134 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)OCCCC AS-3135 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCCCCCC AS-3136 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)OCCCCCC AS-3137 B1(OC(C(O1)(C)C)(C)C)c2ccc(=O)n(c2)Cc3ccccc3 AS-3138 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)c4cc(ccc4o3)B5OC(C(O5)(C)C)(C)C AS-3139 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)N3CCN(CC3)CC AS-3140 B1(OC(C(O1)(C)C)(C)C)c2ccc3cc(ccc3c2)O AS-3141 c1c(cc(c(c1O)[N+](=O)[O-])F)F AS-3142 c1cc(=O)oc2c1c(c(c(c2)Br)N)Br AS-3143 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)C(=O)N3CCN(CC3)CC AS-3144 B(c1ccc2c(c1)c3ccccc3n2c4ccccc4)(O)O AS-3145 Cc1cccc(c1)c2ccccc2C=O AS-3146 Cc1ccc(cc1)c2ccccc2C=O AS-3147 B1(OC(C(O1)(C)C)(C)C)c2cc(cs2)CCCCCC AS-3148 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=C\3/C(=O)N(CC(=O)N3)C(=O)C AS-3150 B(c1cc(cc(c1)C)C)(O)O AS-3151 Cc1ccc(cc1O)NC(=O)OC(C)(C)C AS-3152 Cc1ccc(cc1)c2ccc(cc2)CO AS-3153 Cc1cccc(c1)c2ccc(cc2)CO AS-3154 Cc1cccc(c1)c2ccccc2C(=O)O AS-3155 Cc1cccc(c1)c2ccc(c(c2)C)C AS-3157 Cc1ccc(cc1)c2ccccc2C(=O)OC AS-3158 Cc1cccc(c1)c2ccccc2C(=O)OC AS-3159 Cc1ccc(cc1)c2ccccc2CO AS-3160 B(c1ccc(c(c1)C)C)(O)O AS-3161 Cc1ccc(cc1C)c2ccc(c(c2)C)C AS-3162 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)C)C AS-3163 Cc1ccc(cc1)c2ccc(c(c2)C)C AS-3164 [B-](c1cccc(c1)OCC)(F)(F)F.[K+] AS-3165 Cc1ccc(cc1)Cc2ccccc2 AS-3166 Cc1cccc(c1)Cc2ccccc2 AS-3167 Cc1ccccc1Cc2ccccc2 AS-3168 B1(OC(C(O1)(C)C)(C)C)c2ccc(c(c2)C)C AS-3183 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCCCO AS-3196 CCCCC(CC)CN1C(=O)C2C3CC(C2C1=O)C=C3 AS-3197 Cc1cccc(c1)c2cccc(c2)C(=O)OC AS-3198 CCCCCCCCCCCCCCCCCCOCCOCCOCCO AS-3199 Cc1ccc-2c(c1)C(=O)c3c2cccc3 AS-3200 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)F)F AS-3201 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)CC(=O)N3CCOCC3 AS-3202 C1C2C=CC1C3C2C(=O)N(C3=O)CCO AS-3203 [B-](c1ccc(cc1)C(=O)C)(F)(F)F.CCCC[N+](CCCC)(CCCC)CCCC AS-3204 Cn1cc(c2c1ncnc2Cl)I AS-3205 CC(C)(C)OC(=O)n1ccc2c1ncnc2Cl AS-3206 CC(C)CN1C(=O)C2C3CC(C2C1=O)C=C3 AS-3207 c1ccc(cc1)CN2C(=O)C3C4CC(C3C2=O)C=C4 AS-3208 C=CCN1C(=O)C2C3CC(C2C1=O)C=C3 AS-3209 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCCCl AS-3211 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)OCCCCl AS-3212 B1(OC(C(O1)(C)C)(C)C)c2cccc(c2)NC(=O)[C@H](C(C)C)NC(=O)OCc3ccccc3 AS-3213 CC(C)[C@H]1C(=O)OC(=O)N1C(=O)OCc2ccccc2 AS-3214 Cc1ccc-2c(c1)C(=O)c3c2ccc(c3)C AS-3215 c1cc(cc(c1)c2ccc(cc2)C(=O)O)CO AS-3216 Cc1cc(cc(c1)c2ccc(cc2)C(=O)O)C AS-3217 COC(=O)c1ccc(cc1)c2cccc(c2)CBr AS-3218 Cc1ccc(cc1)c2cccc(c2)O AS-3219 Cc1ccc(c(c1)c2ccccc2)C(=O)O AS-3220 Cc1ccc(cc1)c2ccc(cc2)COC(=O)C AS-3221 Cc1ccc(cc1C)c2ccc(cc2)C(=O)O AS-3222 Cc1ccc-2c(c1)Cc3c2cccc3 AS-3223 Cc1cccc(c1)c2cc(cc(c2)C)C AS-3224 Cc1cccc(c1C(=O)OC)c2ccccc2 AS-3225 c1c(cc(c(c1[N+](=O)[O-])N)[N+](=O)[O-])Br AS-3227 c1ccc(cc1)COc2cc(ccc2[N+](=O)[O-])N3CCOCC3 AS-3228 Cc1cccc(c1COc2cc(ccc2[N+](=O)[O-])F)C AS-3229 CC(C)(C)OC(=O)N(c1c(cc(cc1[N+](=O)[O-])Br)[N+](=O)[O-])C(=O)OC(C)(C)C AS-3230 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)/C=N/CCCC AS-3231 c1ccc2c(c1)CCCO2 AS-3232 Cc1cccn2c1nc(cc2=O)O AS-3233 B1(OC(C(O1)(C)C)(C)C)c2cnn(c2)c3ccc(cc3)C#N AS-3234 [B-](c1ccc(cc1)CC(=O)OC)(F)(F)F.[K+] AS-3236 Cc1ccc(cc1)c2ccc(c(c2)C(=O)O)C AS-3237 B1(OC(C(O1)(C)C)(C)C)c2cnn(c2)Cc3ccc(cc3)OC AS-3238 CCCC[Sn](CCCC)(CCCC)c1cccc(n1)C AS-3239 CC(C)(C)OC(=O)NCCOCCOCCOCCN=[N+]=[N-] AS-3240 B1(OC(C(O1)(C)C)(C)C)c2cnn(c2)Cc3cccc(c3F)Cl AS-3241 B1(OC(C(O1)(C)C)(C)C)c2cnn(c2)CC(=O)OC AS-3242 CCCCCCCCC1(c2ccccc2-c3c1cc(cc3)Br)CCCCCCCC AS-3248 c1ccnc(c1)c2[nH]c3cc(ccc3n2)C(=O)O AS-3249 c1ccnc(c1)c2[nH]c3ccc(cc3n2)C#N AS-3250 B1(OC(C(O1)(C)C)(C)C)c2cc(c(c(c2)F)C(=O)OC)F AS-3251 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CCOC(=O)C AS-3252 Cc1cccc(c1)c2ccc(cc2)C(=O)OC AS-3254 CCOC(=O)N(c1c(cc(cn1)N)I)C(=O)OCC AS-3255 CCOC(=O)N(c1c(cc(cn1)[N+](=O)[O-])I)C(=O)OCC AS-3256 B1(OC(C(O1)(C)C)(C)C)c2ccccc2C(=O)OC AS-3257 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)F)OC(=O)C AS-3258 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CCc3ccc(cc3)B4OC(C(O4)(C)C)(C)C AS-3259 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)c3ccccc3OCc4ccccc4 AS-3260 c1cc2ccc3ccc(c4c3c2c(c1)cc4)CBr AS-3261 CC(=O)Oc1cc(cc(c1)Br)F AS-3262 Cc1cc(cc(c1)Br)C(=O)OC AS-3263 c1cc(ccc1C(=O)c2ccc(cc2)F)[N+](=O)[O-] AS-3264 COC(=O)c1ccc(cc1)c2cccc(c2)Br AS-3265 B1(OC(C(O1)(C)C)(C)C)c2cc(cc(c2)C(=O)OC)C AS-3266 B1(O[C@H]2[C@H]3C[C@H](C3(C)C)C[C@]2(O1)C)c4cccc5c4nccc5 AS-3267 B1(OC(C(O1)(C)C)(C)C)c2cc(c(c(c2)F)N(C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)F AS-3268 c1cc(cc2c1ccc(=O)o2)OCC(=O)O AS-3269 CC(C)(C)OC(=O)N/N=C(/c1cccc(c1)C(F)(F)F)\N AS-5000 CC(C)(C)OC(=O)N/N=C(/COc1ccccc1)\N AS-5001 CC(C)(C)OC(=O)N/N=C(/Cc1ccccc1)\N AS-5002 Cc1ccc(cc1)C/C(=N/NC(=O)OC(C)(C)C)/N AS-5003 Cc1cccc(c1)/C(=N/NC(=O)OC(C)(C)C)/N AS-5004 CC(C)(C)OC(=O)N/N=C(/c1ccc(cc1)OC(F)(F)F)\N AS-5005 CC(C)(C)OC(=O)N/N=C(/Cc1ccc(cc1)Cl)\N AS-5006 CC(C)(C)OC(=O)N/N=C(/c1ccc(cc1)OC)\N AS-5007 Cc1ccc(cc1)/C(=N/NC(=O)OC(C)(C)C)/N AS-5008 CC(C)(C)OC(=O)N/N=C(/COc1ccc(cc1)OC)\N AS-5009 CC(C)(C)OC(=O)N/N=C(/Cc1ccc(cc1)OC)\N AS-5010 CC(C)(C)OC(=O)N/N=C(/COc1ccc(cc1)Cl)\N AS-5011 CC(C)(C)OC(=O)N/N=C(/COc1cccc(c1)Cl)\N AS-5012 CC(C)(C)OC(=O)N/N=C(/c1ccccc1Cl)\N AS-5013 CC(C)(C)OC(=O)N/N=C(/COc1cccc(c1)C(F)(F)F)\N AS-5014 CC(C)(C)OC(=O)N/N=C(/COc1ccccc1Cl)\N AS-5015 CC(C)(C)OC(=O)N/N=C(/c1ccc(c(c1)Cl)F)\N AS-5016 CC(C)(C)OC(=O)N/N=C(/c1cc(cc(c1)C(F)(F)F)C(F)(F)F)\N AS-5017 Cc1ccc(cc1F)/C(=N/NC(=O)OC(C)(C)C)/N AS-5018 CC(C)(C)OC(=O)N/N=C(/c1ccc2ccccc2c1)\N AS-5019 CC(C)(C)OC(=O)N/N=C(/Cc1c(cccc1Cl)Cl)\N AS-5020 CC(C)(C)OC(=O)N/N=C(/Cc1ccccc1Cl)\N AS-5021 CC(C)(C)OC(=O)N/N=C(/COc1cc(cc(c1)Cl)Cl)\N AS-5022 CC(C)(C)OC(=O)N/N=C(/c1ccc(cc1)Cl)\N AS-5023 CC(C)(C)OC(=O)N/N=C(/Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)\N AS-5024 CCOC(=O)c1c(c(on1)C)C(=O)C AS-5025 CC(C)(C)OC(=O)N1CCN(CC1)CCCN AS-5026 CCOC(=O)c1cc(on1)C AS-5027 Cc1cc(no1)C(=O)O AS-5028 CCOC(=O)c1cc(c(nc1C)O)C#N AS-5029 CCOC(=O)c1cc(c(nc1C)Cl)C#N AS-5030 CCOC(=O)c1cc(c(nc1C(F)(F)F)O)C#N AS-5031 CCOC(=O)c1cc(c(nc1C(F)(F)F)Cl)C#N AS-5032 Cc1cc(nc(c1C(=O)O)O)C AS-5033 CCOC(=O)c1nc(on1)C AS-5034 CCOC(=O)c1nc(on1)CCNC(=O)OC(C)(C)C AS-5035 CCOC(=O)c1nc(on1)c2ccccc2 AS-5036 CCOC(=O)c1nc(on1)c2ccc(cc2)OC AS-5037 CCOC(=O)c1nc(on1)c2cccc(c2)Cl AS-5038 CCOC(=O)c1nc(on1)c2cccs2 AS-5039 CCOC(=O)c1nc(on1)c2ccc(cc2)Br AS-5040 CCOC(=O)c1nc(on1)c2cccc(c2)C(F)(F)F AS-5041 CCOC(=O)c1nc(no1)C AS-5042 CCOC(=O)c1nc(no1)c2ccccc2 AS-5043 CCOC(=O)c1nc(no1)c2ccc(cc2)OC AS-5044 CCOC(=O)c1nc(no1)c2cccnc2 AS-5045 CCOC(=O)c1nc(no1)c2ccc(cc2)F AS-5046 CCOC(=O)c1nnc(o1)CNC(=O)OC(C)(C)C AS-5047 c1cnc(cn1)/C(=N/C#N)/N AS-5048 c1ccc(cc1)c2ccnc(n2)Nc3ccc(cc3)Cl AS-5049 CC/C(=N\NC(=O)OC(C)(C)C)/NC1CCCC1 AS-5050 CC(C)(C)OC(=O)N/N=C(/NCc1ccccc1)\NCC(F)(F)F AS-5051 CC(C)(C)OC(=O)N/N=C(/COc1ccccc1)\NC2CCC2 AS-5052 CC/C(=N\NC(=O)OC(C)(C)C)/NC1CC1 AS-5053 CC(C)(C)OC(=O)N/N=C(\Cc1ccccc1)/NCc2ccco2 AS-5054 CC(C)(C)OC(=O)N/N=C(\Cc1ccccc1)/NC2CC2 AS-5055 CC(C)(C)OC(=O)N/N=C(/COc1ccccc1)\NC2CC2 AS-5056 CC(C)(C)OC(=O)N/N=C(\Cc1ccc(cc1)Cl)/NC2CC2 AS-5057 CC(C)(C)OC(=O)N/N=C(\Cc1ccc(cc1)Cl)/NC2CCC2 AS-5058 CC(C)(C)OC(=O)N/N=C(/Cc1ccc(cc1)Cl)\NCCOC AS-5059 CC(C)(C)OC(=O)N/N=C(/c1ccccc1)\N AS-5060 CC(C)(C)OC(=O)N/N=C(\Cc1ccc(cc1)OC)/NC2CCCC2 AS-5061 CC(C)(C)OC(=O)N/N=C(\Cc1ccc(cc1)OC)/NCC(F)(F)F AS-5062 CC(C)(C)OC(=O)N/N=C(\Cc1ccccc1)/NC2CCCC2 AS-5063 CC(C)(C)OC(=O)N/N=C(\Cc1ccccc1)/NC2CCC2 AS-5064 CC/C(=N\NC(=O)OC(C)(C)C)/NC1CCC1 AS-5065 CC(C)(C)OC(=O)N/N=C(\Cc1ccc(cc1)Cl)/NCc2ccco2 AS-5066 CC(C)(C)OC(=O)N/N=C(/COc1ccccc1)\NCC(F)(F)F AS-5067 CC(C)(C)OC(=O)N/N=C(/COc1ccccc1)\NC2CCCC2 AS-5068 CC(C)(C)OC(=O)N/N=C(/COc1ccccc1)\NCCOC AS-5069 CC(C)(C)OC(=O)N/N=C(/Cc1ccc(cc1)Cl)\NCC(F)(F)F AS-5070 CCOC(=O)C1CCN(CC1)CCC#N AS-5071 CC(C(=O)O)Sc1c(cc(cn1)C(F)(F)F)Cl AS-5072 c1cc(ccc1Sc2c(cc(cn2)C(F)(F)F)Cl)Br AS-5073 COC(=O)CNc1c(cc(cn1)C(F)(F)F)Cl AS-5074 CCOC(=O)C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl AS-5075 c1c(cnc(c1Cl)OCC(=O)O)C(F)(F)F AS-5076 c1c(c(c(nc1N2CCOCC2)Cl)Br)C(F)(F)F AS-5077 c1c(cc(nc1NCCN)N2CCOCC2)C(F)(F)F AS-5078 c1c(c(c(nc1N2CCOCC2)Cl)[N+](=O)[O-])C(F)(F)F AS-5079 CN(c1cc(cc(n1)Cl)C(F)(F)F)N AS-5080 c1c(cc(nc1SCC(=O)O)SCC(=O)O)C(F)(F)F AS-5081 c1ccc(cc1)c2cc(nc(c2C#N)Cl)c3ccccc3 AS-5082 CCOC(=O)CNc1c(c(cc(n1)C)C)C#N AS-5083 Cc1c(c(nc(c1[N+](=O)[O-])C)Cl)C#N AS-5084 COC(=O)CSc1c(cccn1)C(F)(F)F AS-5085 COC(=O)CSc1nc(cc(n1)O)O AS-5086 COC(=O)CSc1nccc(n1)O AS-5087 COc1ccc(cc1OC)/C(=N/O)/N AS-5088 CC(C)(C)OC(=O)N1CCCC(C1)/C(=N/O)/N AS-5089 CC(C)(C)OC(=O)N1CCCCC1/C(=N/O)/N AS-5090 CC(C)(C)OC(=O)N1CCC(CC1)/C(=N/O)/N AS-5091 c1cc(cc(c1)OC(F)(F)F)/C(=N/O)/N AS-5092 CC(C)(C)OC(=O)N1CCN(CC1)C/C(=N/O)/N AS-5093 CCOC(=O)CNC(=O)C1CCN(CC1)C(=O)OCc2ccccc2 AS-5094 CCOC(=O)c1cc(on1)C=O AS-5095 c1cc2c(cc1/C(=N/O)/N)OCO2 AS-5096 COc1ccc(c(c1)C2N[C@@H](CS2)C(=O)O)OC AS-5097 COc1ccc(cc1)C2N[C@@H](CS2)C(=O)O AS-5098 C1COCCN1C/C(=N/O)/N AS-5099 c1ccc(cc1)COC(=O)N2CCC2C(=O)O AS-5100 COc1cccc(c1)Cc2nc(cs2)C(=O)O AS-5101 c1cc(ccc1Cc2nc(cs2)C(=O)O)Br AS-5102 CC(C)(C)OC(=O)c1cccc(c1)CN AS-5103 CC(C)(C)OC(=O)c1ccccc1C=O AS-5104 CC(C)(C)OC(=O)c1cccc(c1)C=O AS-5105 CCOC(=O)c1csc(n1)Cc2ccccc2Br AS-5106 c1ccc(c(c1)Cc2nc(cs2)C(=O)O)Br AS-5107 CCOC(=O)c1cc(n(n1)C(C)(C)C)C AS-5108 CCOC(=O)C1CCN(CC1)CC#N AS-5109 c1c(cc(nc1N2CCNCC2)N3CCOCC3)C(F)(F)F AS-5110 CCCCNC(=O)c1nc(on1)c2ccccc2 AS-5111 COC(=O)CSc1cc(cc(n1)Cl)C(F)(F)F AS-5112 CC(C(=O)O)Sc1cc(cc(n1)Cl)C(F)(F)F AS-5113 c1c(c(c(nc1N2CCOCC2)NCCN)Br)C(F)(F)F AS-5114 c1ccc(cc1)c2nc(no2)C(=O)NN AS-5115 CC(C)(C)c1cc(n[nH]1)C(F)(F)F AS-5117 CCOC(=O)CN1CCC(CC1)C(=O)OCC AS-5120 CCOC(=O)c1cn(nc1C(F)(F)F)c2ccccc2 AS-5121 CC(C)(C)OC(=O)NCc1nc(no1)c2ccccc2 AS-5122 CC(C)(C)OC(=O)NCc1nc(no1)c2ccc(cc2)F AS-5123 CC(C)(C)OC(=O)NCc1nc(no1)c2cccnc2 AS-5124 c1ccc(c(c1)Cc2nc(cs2)CC(=O)O)Br AS-5125 c1cc(ccc1Cc2nc(cs2)CC(=O)O)Br AS-5126 Cn1c(cc(n1)CO)C(=O)OC AS-5127 Cn1c(cc(n1)C(=O)OC)CO AS-5128 CCOC(=O)c1c(sc(n1)C)C(=O)C AS-5129 CCOC(=O)c1c(sc(n1)c2ccccc2)C(=O)C AS-5130 CCOC(=O)C(C(=O)C)Oc1ccc(cc1)Cl AS-5131 CCOC(=O)C(C(=O)C)Oc1ccc(cc1)OC AS-5132 CCOC(=O)C(C(=O)C)Oc1ccc(cc1)C(F)(F)F AS-5133 CCOC(=O)c1c(noc1C(=O)C)C AS-5134 CCOC(=O)c1c(noc1C(C)O)C AS-5135 CCOC(=O)c1c(noc1C(C)O)c2ccccc2 AS-5136 CCOC(=O)c1c(noc1CO)C AS-5137 CCOC(=O)c1c(noc1C=O)C AS-5138 c1ccc(c(c1)C2N[C@@H](CS2)C(=O)O)O AS-5139 CCOC(=O)c1cnc(nc1)Cl AS-5140 CC(C)(C)OC(=O)NCc1nc(no1)c2ccc(cn2)C(F)(F)F AS-5141 c1c(cc(nc1N2CCCC2)Cl)C(F)(F)F AS-5142 c1c(cc(nc1NCCN)N2CCCC2)C(F)(F)F AS-5143 COc1c(cc(cn1)[N+](=O)[O-])C(=O)O AS-5144 c1cc(cc(c1)C(F)(F)F)c2ncnc(n2)Cl AS-5145 c1cc(cc(c1)Cl)c2ncnc(n2)Cl AS-5146 c1cc(cc(c1)[N+](=O)[O-])c2ncnc(n2)Cl AS-5147 c1c(cnc(c1C(=O)O)O)Cl AS-5148 CCOC(=O)C1C(=O)CCN1C(=O)OC(C)(C)C AS-5149 c1cc(ccc1c2nc(sn2)Cl)Br AS-5150 c1cc(ccc1c2nc(sn2)Cl)F AS-5151 CCCCNc1cc(cc(n1)Cl)C(F)(F)F AS-5152 c1ccc(cc1)C(/C(=N/O)/N)N2CCOCC2 AS-5153 CCOC(=O)c1c(c(nc(n1)C)Cl)C AS-5154 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)O AS-5155 COC(c1c(cnn1c2ccccc2)C(=O)OC)OC AS-5156 COC(=O)c1cnn(c1C=O)c2ccccc2 AS-5157 CCOC(=O)C1CN(CC1=O)C(=O)OC(C)(C)C AS-5158 CCOC(=O)C1CCN(CC1)CC(=O)N AS-5159 c1cc2c(cc1[N+](=O)[O-])C(=O)OC2 AS-5160 CCOC(=O)c1cc(nc(c1C#N)S)C AS-5161 CCOC(=O)c1cc(nc(c1C#N)O)C AS-5162 CCOC(=O)CNc1cc(cc(n1)Cl)C(F)(F)F AS-5163 c1ccc(c(c1)N2CC(CC2=O)C(=O)O)OC(F)(F)F AS-5164 c1(c([nH]nc1C(=O)O)C(=O)O)[N+](=O)[O-] AS-5165 CCOC(=O)c1cc(nn1Cc2ccccc2)C(C)(C)C AS-5166 CCOC(=O)c1cnc(nc1Cl)C(F)(F)F AS-5167 CCOC(=O)c1cc(n[nH]1)C(C)(C)C AS-5168 c1cc(nc(c1C(=O)O)Cl)O AS-5169 Cc1cc(c(nc1)C#N)[N+](=O)[O-] AS-5170 c1ccc(cc1)Oc2c(cccn2)C(=O)O AS-5171 c1c(cnc(c1Cl)O)I AS-5172 c1c(c(cnc1O)Br)C(F)(F)F AS-5173 CCOC(=O)c1ccc(cc1)c2ccc(cn2)C(F)(F)F AS-5174 COC(=O)c1ccc(c(c1)O)C(=O)OC AS-5175 CCOC(=O)/C(=C(\C)/NC(C)c1ccccc1)/C AS-5176 CCOC(=O)C/C(=N/O)/N AS-5177 Cc1cc(on1)C(=O)O AS-5178 CCOC(=O)c1c(nccn1)Cl AS-5179 CCOC(=O)c1c(oc(n1)c2ccccc2)C AS-5180 CCOC(=O)C1CN(CCN1C)C AS-5181 c1cc(cnc1)c2nc(cs2)C(=O)O AS-5182 CC(=O)Oc1cscc1C(=O)OC AS-5183 c1ccc(cc1)c2nc(sn2)Cl AS-5184 CN(C)c1cc(cc(n1)c2ccc(cc2)C(=O)O)C(F)(F)F AS-5185 c1c(cc(nc1N2CCC(CC2)C(=O)O)Cl)C(F)(F)F AS-5186 c1cc(c(nc1)c2ccc(cc2)C(=O)O)C=O AS-5187 Cc1cc(cc(c1I)C)O AS-5188 c1c(csc1[N+](=O)[O-])C(=O)O AS-5189 CCOC(=O)/C(=C(\C)/c1ccccc1)/C#N AS-5190 c1cc(cc(c1)Br)n2cccn2 AS-5191 Cc1cccc(c1)n2cccn2 AS-5192 c1cnn(c1)c2ccc(cc2)Br AS-5193 c1cnn(c1)c2ccc(cc2)Cl AS-5194 Cc1c(c(n(n1)c2cccc(c2)Cl)C)C=O AS-5195 Cc1c(c(n(n1)c2cccc(c2)Cl)C)C(=O)O AS-5196 Cc1c(c(n(n1)c2ccc(cc2)Cl)C)C=O AS-5197 Cc1c(c(n(n1)c2ccc(cc2)Cl)C)C(=O)O AS-5198 Cc1cc(n(n1)c2ccccc2)C AS-5199 Cc1c(c([nH]n1)C(=O)O)[N+](=O)[O-] AS-5200 CCOC(=O)c1c(c(n[nH]1)C)[N+](=O)[O-] AS-5201 CCOC(=O)c1cnn(c1C)c2ccccc2 AS-5202 COc1ccc(cc1OC)CN2CC(CC2=O)C(=O)O AS-5203 CCSc1cc(cc(n1)Cl)C(F)(F)F AS-5204 c1ccc(c(c1)C#N)Oc2ccc(cc2)F AS-5205 CCOC(=O)c1nc(no1)c2ccccn2 AS-5206 CC(C)(C)OC(=O)N1CCN(CC1)Cc2c(cc(cn2)C(F)(F)F)Cl AS-5207 c1cc(ccc1NC(=S)N2CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl AS-5208 c1c(cc(c2c1COCO2)C(=O)O)F AS-5209 CSc1nc(cc(n1)O)O AS-5210 Cn1c(cc(n1)C(=O)OC)C(=O)OC AS-5211 CN(C)c1c(cc(cn1)C(F)(F)F)Br AS-5212 COC(=O)c1c(nsc1SC)O AS-5213 CCOC(=O)c1ccc(nc1)CO AS-5214 COC(=O)c1cc(cnc1O)I AS-5215 c1ccc(cc1)c2cc(nc(n2)O)O AS-5216 c1ccc(cc1)c2cc(nc(n2)S)O AS-5217 c1c(nc(nc1O)C(F)(F)F)O AS-5218 CCOC(=O)c1cn(nc1O)C AS-5219 CCOC(=O)c1c[nH]nc1O AS-5220 CCOC(=O)c1cc(n(n1)C)O AS-5221 Cn1c(cc(n1)C(=O)OC)O AS-5222 COc1cc(c(cc1O)[N+](=O)[O-])C(=O)OC AS-5223 c1cc(ccc1C(=O)Nc2cc(cc(n2)Cl)C(F)(F)F)Cl AS-5224 CN(C)c1cc(cc(n1)c2ccc(cc2)O)C(F)(F)F AS-5225 CN(C)c1cc(cc(n1)c2cccc(c2)C=O)C(F)(F)F AS-5226 CN/N=C/c1ccc(cc1)c2cc(cc(n2)N(C)C)C(F)(F)F AS-5227 CN(C)c1cc(cc(n1)c2cccc(c2)O)C(F)(F)F AS-5228 CCOC(=O)CCN(CC(=O)OCC)C(=O)OC(C)(C)C AS-5229 Cc1cc(c(c(c1)C)n2c(c(c(c2NC(=O)C)C#N)C)C)C AS-5230 COC(=O)c1ccc(c(c1)OCC#C)F AS-5231 Cc1c(c(on1)c2ccccc2)C(=O)OC AS-5232 Cc1c(cc(cn1)C(F)(F)F)Cl AS-5233 CCOC(=O)CN(C)c1c2ccccc2nc(n1)C(F)(F)F AS-5234 CN(CC(=O)O)c1c2ccccc2nc(n1)C(F)(F)F AS-5235 CCOC(=O)C(=O)CC(=O)c1cccs1 AS-5237 CC(C)(C)OC(=O)N1CCN(CC1)CCCN2C(=O)c3ccccc3C2=O AS-5238 CCOC(=O)c1nc(on1)C(C)(C)C AS-5239 CCc1nc(on1)C(=O)OCC AS-5240 CCOC(=O)c1nc(no1)C2CC2 AS-5241 c1cc(sc1)c2cc(no2)C(=O)O AS-5242 CC(C)(C)OC(=O)N1CCN(CC1)CCCCN AS-5243 CN(C)c1c(cc(cn1)C(F)(F)F)c2cccc(c2)O AS-5244 CN(C)c1c(cc(cn1)C(F)(F)F)c2cccc(c2)C=O AS-5245 CC(=O)Nc1cccc(c1)c2cc(cnc2N(C)C)C(F)(F)F AS-5246 CCOC(=O)c1c(nc(s1)NC(=O)C2(CCCC2)c3ccccc3)C AS-5247 CN(C)CC/N=C/c1ccc(cc1)Br AS-5248 CN(C)c1c(cc(cn1)C(F)(F)F)c2ccc(cc2)N AS-5249 CCOC(=O)Cc1nc(on1)c2ccccc2 AS-5250 c1cc2c(cc1Br)[nH]c(n2)C(F)(F)F AS-5251 CCOC(=O)c1ccc(cc1)c2c(cccn2)C#N AS-5252 CCOC(=O)Cc1nc(on1)c2ccc(cc2)F AS-5253 CC(C)C(C#N)c1ccc(c(c1)OC)OC AS-5254 CCOC(=O)c1c[nH]c(=O)nc1 AS-5255 c1ccc(cc1)c2nc(co2)C(=O)O AS-5256 Cc1ccnc(c1C(=O)O)O AS-5257 c1cc(cnc1)c2nc(no2)N AS-5258 CCOC(=O)C1=C(C(=O)N(C1)Cc2ccccc2)O AS-5259 CCOC(=O)C1CN(C(=O)C1=O)Cc2ccccc2 AS-5260 Cc1ccc(cc1)c2c(c(no2)C)C(=O)OC AS-5261 Cc1ccc(cc1)c2c(c(no2)C)C(=O)O AS-5262 c1ccc(cc1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl AS-5263 Cc1cc(cc(n1)c2cccc(c2)C(=O)OC)C(F)(F)F AS-5264 c1ccc(cc1)c2cc(no2)C(=O)O AS-5265 CC(=O)c1ccc(cc1)c2cc(cc(n2)N(C)C)C(F)(F)F AS-5266 Cn1cnc(c1C(=O)O)C(=O)O AS-5267 c1c(n[nH]c1O)C(=O)O AS-5268 CCOC(=O)c1cc([nH]n1)O AS-5269 Cc1c(c(on1)c2ccc(cc2)Br)C(=O)O AS-5270 COC(=O)c1c(nns1)C2CC2 AS-5271 C1CC1c2c(snn2)C(=O)O AS-5272 Cc1c(c(ncn1)C)C(=O)OC AS-5273 Cc1c(oc(n1)NC(=O)OC(C)(C)C)C(=O)OC AS-5274 COc1ccc(nc1Br)[N+](=O)[O-] AS-5275 c1ccc(cc1)c2nc(on2)O AS-5276 CCOC(=O)c1c(snc1c2ccccc2)C AS-5277 CC(=O)/C=C/Nc1ccccc1 AS-5278 CC(C)(C)OC(=O)CNCc1ccccc1 AS-5279 c1cc(c(c(c1)Cl)C2CC(=O)CC(=O)C2)F AS-5280 CC(C)(C)OC(=O)Nc1cnc(cc1C(=O)O)Cl AS-5281 c1cc(ccc1c2cc(ccn2)C(F)(F)F)C(=O)O AS-5282 COC(=O)c1ccc(cc1)c2cc(ccn2)C(F)(F)F AS-5283 COC(=O)c1cccc(c1)c2cc(ccn2)C(F)(F)F AS-5284 c1cc(cc(c1)C(=O)O)c2cc(ccn2)C(F)(F)F AS-5285 c1ccc(cc1)c2ccnc(c2C(=O)O)Br AS-5286 CCOC(=O)c1cc(nn1Cc2c(cc(cn2)C(F)(F)F)Cl)C AS-5287 CCOC(=O)c1cc(on1)C(=O)C AS-5288 CCOC(=O)CCN(CC(=O)OCC)C(=O)OCc1ccccc1 AS-5289 CCOC(=O)c1c(ccnc1Br)c2ccccc2 AS-5290 CCOC(=O)c1c(ccnc1c2ccc(cc2)C=O)C AS-5291 Cc1c(c(on1)c2ccc(cn2)Br)C(=O)O AS-5292 c1ccc(c(c1)C(CC(=O)O)N)[N+](=O)[O-] AS-5293 Cc1c(c(on1)c2ccc(cc2)Br)C(=O)OC AS-5294 c1ccc2c(c1)ncc(n2)C(=O)O AS-5295 Cc1nnc(o1)c2cccc(c2)[N+](=O)[O-] AS-5296 c1cc2c(cc1[N+](=O)[O-])CC(=O)O2 AS-5297 CN(C)c1cc(cc(n1)c2ccc(cc2)C(=O)OC)C(F)(F)F AS-5298 c1cc(ccc1C=O)c2cc(cc(n2)Cl)C(F)(F)F AS-5299 CCOC(=O)COc1c(cc(cn1)C(F)(F)F)Cl AS-5300 CCOC(=O)C1COc2ccccc2O1 AS-5301 Cc1cc(cc(n1)Cl)C(F)(F)F AS-5302 Cc1c(c(nc(c1Br)C)O)C(=O)O AS-5303 c1ccc2c(c1)ncc(n2)C(C(C(CO)O)O)O AS-5304 COC(=O)/C(=C\C=C\c1ccccc1)/C#N AS-5305 COC(=O)c1cnc2ccccc2n1 AS-5306 CCOC(=O)c1c(c(=O)[nH]c(n1)C)C AS-5307 c1ccc(c(c1)c2cnco2)[N+](=O)[O-] AS-5308 c1cc(ccc1CN2CCOCC2)C(=O)O AS-5309 COC(=O)c1ccc(cn1)C(=O)O AS-5310 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)O AS-5311 c1cc2c(nc1)nc(o2)O AS-5312 CCOC(=O)c1c(snn1)C AS-5313 c1ccc(cc1)n2cc(c(n2)C(F)(F)F)C(=O)O AS-5314 COC(=O)c1ccc(cn1)O AS-5315 CN(C)CCOc1ccccc1C(=O)O AS-5316 CCOC(=O)c1cnc(nc1C(F)(F)F)C(F)(F)F AS-5317 c1ccc(cc1)Oc2ccc(cn2)/C=C/C(=O)O AS-5318 c1cc(ccc1C#N)SC(F)(F)F AS-5319 c1cc2c(cc1Cl)sc(n2)Cl AS-5320 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)c2ccc(cc2)F AS-5321 COC(=O)c1ccc(c(c1)O)CO AS-5322 CC(C)(C)OC(=O)N1CCN(CC1)CCCCN2C(=O)c3ccccc3C2=O AS-5323 CC(C)(C)OC(=O)N1CCN(CC1)CCC#N AS-5324 c1cc2c(cc1C(=O)NN)nccn2 AS-5325 CCOC(=O)c1cc(cc(c1)[N+](=O)[O-])C(F)(F)F AS-5326 CCOC(=O)c1nc(no1)C(C)C AS-5327 Cc1c(c(n(n1)c2ccccc2)C)Br AS-5328 c1c(c(c(nc1Cl)N2CCOCC2)[N+](=O)[O-])C(F)(F)F AS-5329 Cn1nc(nn1)c2cccc(c2)S(=O)(=O)N AS-5330 CC(C)S(=O)(=O)c1csc(c1N)C(=O)OC AS-5331 c1cc(ccc1c2ccnc(n2)S)[N+](=O)[O-] AS-5332 CC(C)S(=O)(=O)c1csc(c1Cl)C(=O)OC AS-5333 CC(C)S(=O)(=O)c1csc(c1Cl)C(=O)O AS-5334 CC(C)(C)OC(=O)Cn1ccc(n1)c2ccc(cc2)[N+](=O)[O-] AS-5335 CC(C)(C)OC(=O)NCC(=O)O/N=C(\c1ccccc1)/N AS-5336 COC(=O)C1CC(=O)N(C1)Cc2ccc(cc2)F AS-5337 CC(C)Sc1c(cccc1Cl)[N+](=O)[O-] AS-5338 Cn1nc(nn1)c2cccc(c2)[N+](=O)[O-] AS-5339 CCOC(=O)CNS(=O)(=O)c1ccc(cn1)C(F)(F)F AS-5340 COc1ccc(c(c1OC)Cl)/C=C/C(=O)O AS-5341 c1ccc(cc1)c2cn(cc2CO)c3ccccc3 AS-5342 CCOC(=O)c1cnc(nc1C(F)(F)F)O AS-5343 COC(=O)c1ccc(nc1)C(=O)OC AS-5344 CCOC(=O)c1cc(no1)C AS-5345 CC(C)(C)c1ccc(cc1)/C(=N/O)/N AS-5346 CCOC(=O)CNc1ccccc1 AS-5347 Cc1nc(no1)c2ccc(cc2)C(=O)OC AS-5348 CCOC(=O)N1CCN(CC1)c2c(cc(cn2)Br)C(F)(F)F AS-5349 c1cc(ccc1c2nnc(o2)C(F)(F)F)[N+](=O)[O-] AS-5350 CCOC(=O)c1nnc(o1)c2cccc(c2)[N+](=O)[O-] AS-5351 Cc1nnc(o1)c2ccc(cc2)[N+](=O)[O-] AS-5352 CC(C)(C)OC(=O)c1ccccc1C(=O)O AS-5353 c1(c(nc(nn1)O)O)C(=O)O AS-5354 c1cc(cc(c1)[N+](=O)[O-])c2n[nH]nn2 AS-5355 CCOC(=O)CCNCc1ccccc1 AS-5356 CCOC(=O)c1cc(nn1Cc2ccc(cc2)F)C(C)(C)C AS-5357 c1cc(sc1)c2ccc(cc2)Br AS-5358 CCSc1nnc(o1)CNC(=O)OC(C)(C)C AS-5359 CCOC(=O)CS(=O)(=O)Cc1cc(nc(c1)Cl)Cl AS-5360 CCOC(=O)c1c(c(nn1C)C)[N+](=O)[O-] AS-5361 CCOC(c1cc(nc(n1)SCc2ccccc2)O)OCC AS-5362 CCOC(=O)CSCc1cc(nc(c1)Cl)Cl AS-5363 CCOC(=O)c1cc(oc1)S(=O)(=O)N AS-5364 Cc1c(nc(nc1Cl)C(F)(F)F)C AS-5365 c1ccc(cc1)c2ccc(nn2)S AS-5366 CCOC(=O)c1cnn(c1)Cc2cccc(c2)C(F)(F)F AS-5367 CCOC(=O)c1cnn(c1)Cc2ccccc2 AS-5368 CCOC(=O)c1cc2c(s1)nccn2 AS-5369 c1c(cc(c2c1CCO2)Br)Br AS-5370 CCOC(=O)c1c(nc(s1)c2ccc(cc2)OC)C AS-5371 CC(C)(C)c1cc(no1)C(=O)CC#N AS-5372 CCOC(=O)c1cc(on1)C(C)(C)C AS-5373 c1ccc(cc1)c2cc(c(nn2)O)C(=O)O AS-5374 CCCCN1CCC(CC1)CO AS-5375 CCCCN1CCC(CC1)C(=O)OCC AS-5376 c1c(cnc(c1Cl)C(=C(S)S)C#N)C(F)(F)F AS-5377 COc1ccc(c(c1)/C=N/Nc2cc(cc(n2)Cl)C(F)(F)F)OC AS-5378 CN(c1cc(cc(n1)Cl)C(F)(F)F)NC(=O)c2ccccc2 AS-5379 CCNC(=O)CSc1cc(cc(n1)Cl)C(F)(F)F AS-5380 CCOC(=O)NNC(=O)CSc1cc(cc(n1)Cl)C(F)(F)F AS-5381 c1c(c(c(nc1N2CCOCC2)N3CCCC3)[N+](=O)[O-])C(F)(F)F AS-5382 c1cc(ccc1N)Oc2cc(cc(n2)Cl)C(F)(F)F AS-5383 Cc1cc(n(n1)C(C)(C)C)C(=O)O AS-5384 CCOC(=O)c1cc(nn1C)C AS-5385 Cc1cc(n(n1)C)C(=O)O AS-5386 CCOC(=O)c1csc(n1)C AS-5387 CSc1c(ccc(n1)C=O)C#N AS-5388 c1cc(ncc1C(F)(F)F)/C(=N\O)/N AS-5389 c1c(cc(c2c1CC(=O)N2)Br)Br AS-5390 c1ccc(cc1)c2ncnc(n2)S AS-5391 Cc1cc([nH]n1)C(=O)O AS-5392 c1c(cnc(c1Cl)OCCO)C(F)(F)F AS-5393 c1cncc(c1Cl)C(=O)O AS-5394 COC(=O)c1cnccc1Cl AS-5395 c1c(cn(c(=O)c1Cl)CCC(=O)O)C(F)(F)F AS-5396 c1c(cnc(c1Cl)SCCO)C(F)(F)F AS-5397 Cc1cc(nc(c1C#N)N2CCNCC2)C AS-5398 c1c(cc(nc1N2CCOCC2)Cl)C(F)(F)F AS-5399 c1c(cc(nc1N2CCNCC2)Cl)C(F)(F)F AS-5400 CNc1cc(cc(n1)Cl)C(F)(F)F AS-5401 Cc1ccc(c(n1)O)C#N AS-5402 Cc1cc(nc(c1C(=O)N)O)C AS-5403 Cc1cc(nc(c1C(=O)N)Cl)C AS-5404 CCOC(=O)c1c(c2c(cc(nc2s1)C)C)N AS-5405 Cc1cc(nc(c1C#N)N2CCCC2)C AS-5407 c1ccc(c(c1)CC(=S)N)Br AS-5408 c1cc(ccc1CC(=S)N)Br AS-5409 c1cc(ncc1/C(=N/O)/N)Cl AS-5410 c1cscc1/C(=N\O)/N AS-5411 c1cc(ncc1C(F)(F)F)C(=S)N AS-5412 c1cc(ccc1/C(=N/O)/N)F AS-5413 c1cc(cc(c1)F)/C(=N/O)/N AS-5414 c1ccc(c(c1)/C(=N/O)/N)C(F)(F)F AS-5415 c1ccc(c(c1)C(=S)N)C(F)(F)F AS-5416 c1cc(cc(c1)C(F)(F)F)C(=S)N AS-5417 COc1ccccc1/C(=N/O)/N AS-5418 COc1ccc(cc1)/C(=N/O)/N AS-5419 CC(C)(C)OC(=O)C1CCNC1 AS-5420 c1cc2c(cc1C#N)sc(n2)N AS-5421 c1c(nc(s1)C(F)(F)F)C(=O)O AS-5422 Cc1ccc(nc1)C#N AS-5423 CCOC(=O)c1csc(n1)C(F)(F)F AS-5424 C1COCCN1CC#N AS-5425 c1cc(c(cc1C2N[C@@H](CS2)C(=O)O)Cl)Cl AS-5426 c1cc(ccc1C2N[C@@H](CS2)C(=O)O)Cl AS-5427 Cc1ccc(cc1)C2N[C@@H](CS2)C(=O)O AS-5428 Cc1c(cnc(n1)N)C(=O)C AS-5429 c1ccc(cc1)c2ccnc(n2)N AS-5430 c1c(cc(nc1SCC(=O)O)Cl)C(F)(F)F AS-5431 c1c(cc(nc1O)Cl)C(F)(F)F AS-5432 COc1cccc(c1)CC(=S)N AS-5433 C=C1CC(C1)C(=O)O AS-5434 c1c(c(nc(c1F)Cl)Cl)C#N AS-5435 c1ccc(c(c1)C(=O)NC=O)O AS-5436 Cc1c(c(nc(c1Br)C)O)C#N AS-5437 c1ccc(cc1)C/C(=N/O)/N AS-5438 Cc1c(sc(n1)c2ccc(cc2)F)C(=O)O AS-5439 CC(C)(C)OC(=O)c1cccc(n1)F AS-5440 Cc1c(sc(n1)Cc2ccccc2)C(=O)O AS-5441 c1cc(ccc1c2[nH]c(cn2)CO)C(F)(F)F AS-5442 c1cc(ccc1c2[nH]c(cn2)CO)Cl AS-5443 c1ccnc(c1)c2[nH]c(cn2)CO AS-5444 c1ccc(cc1)c2nc(c(s2)C=O)Cl AS-5445 c1cc(ccc1c2nc(c(s2)C=O)Cl)F AS-5446 c1cc(sc1)C2N[C@@H](CS2)C(=O)O AS-5447 c1c(cnc(c1C(=O)O)N)I AS-5448 C=C1CC(C1)C#N AS-5449 c1ccc(c(c1)c2nc(nc(n2)N)N)F AS-5450 Cc1cc(c2c(c(sc2n1)C#N)N)C(F)(F)F AS-5451 c1c(cc(nc1SCCO)Cl)C(F)(F)F AS-5452 Cn1ccc(n1)c2ccc(cc2)N AS-5453 c1cc(ccc1c2ncnc(n2)Cl)F AS-5455 c1ccc(c(c1)c2cnco2)N AS-5457 Cn1ccc(n1)c2cccc(c2)N AS-5458 Cn1ccc(n1)c2ccccc2N AS-5459 Cc1nc(cs1)c2cccc(c2)N AS-5460 COc1ccc2cc([nH]c2c1)C(=O)OC AS-5462 COc1ccc2cc([nH]c2c1)C(=O)O AS-5463 Cc1cccc2c1cc([nH]2)C(=O)OC AS-5464 Cc1cccc2c1cc([nH]2)C(=O)O AS-5465 COC(=O)c1cc2ccoc2[nH]1 AS-5466 COC(=O)c1cc2c([nH]1)cco2 AS-5467 c1coc2c1[nH]c(c2)C(=O)O AS-5468 c1c(nc(nc1Cl)C(F)(F)F)Cl AS-5469 c1cc(cc(c1)C(=N)N)C#N AS-5470 c1cc(cc(c1)/C(=N\O)/N)C#N AS-5471 Cc1cc(c(nc1)S)C#N AS-5472 c1cc(ncc1C#N)N2CCNCC2 AS-5473 CCn1c(c(c(n1)C)Br)C(=O)O AS-5474 Cc1ncc(s1)c2ccccc2N AS-5475 c1cc(ncc1C(F)(F)F)C#N AS-5476 c1cc(nc(c1)O)C(F)(F)F AS-5477 CC(C)(C)OC(=O)C1CCN(C1)C AS-5478 CN1CC(CC1=O)C(=O)OC AS-5479 c1ccc(cc1)CN2CC(CC2=O)C(=O)O AS-5480 Cc1ccc(cc1)N2CC(CC2=O)C(=O)O AS-5481 c1ccnc(c1)/C(=N/C#N)/N AS-5482 Cn1cncc1C(=O)O AS-5483 c1ccc(cc1)N2CC(CC2=O)C(=O)O AS-5484 c1cc(c(cc1F)F)N2CC(CC2=O)C(=O)O AS-5485 c1cc(nc(c1)N2CCC(CC2)C(=O)O)C(F)(F)F AS-5486 c1cc(cc(c1)N2CCOCC2)N AS-5487 c1cc(ncc1C(F)(F)F)N2CCC(CC2)C(=O)O AS-5488 c1ccc(cc1)c2nc(nc(n2)N)N AS-5489 c1cnc(cc1C(=O)O)Cl AS-5490 c1cc(ccc1C2=NCCS2)O AS-5491 c1ccc(cc1)c2c(snn2)N AS-5492 COc1cscc1C(=O)O AS-5493 Cc1cc(nn1C(C)(C)C)C(=O)O AS-5494 Cc1c(c(nc(n1)C2CC2)O)Cl AS-5495 c1cc(sc1)c2nc(sn2)Cl AS-5496 CC(=O)c1ccc(c(n1)S)C#N AS-5497 CCOC(=O)c1cc(n[nH]1)C AS-5498 Cc1cc(c(nc1)N)C#N AS-5499 c1c(cnc(c1S(=O)(=O)N)N)Cl AS-5500 Cc1cc(c(nc1)Br)[N+](=O)[O-] AS-5501 CC(=O)c1cc(ccn1)Cl AS-5502 CC(=O)c1cc(ccn1)OC AS-5503 c1cc(c(nc1)Cl)S(=O)(=O)N AS-5504 Cc1cc(c(nc1)Cl)[N+](=O)[O-] AS-5505 COc1ccnc(c1)C#N AS-5506 COC(=O)c1ccc(nc1F)F AS-5507 CCOC(=O)c1cc(cnc1)N AS-5508 c1cc2c(cc1N)ncs2 AS-5509 Cc1c(c(sn1)N)C#N AS-5510 Cc1c(c(sn1)N)Cl AS-5511 Cc1cc(sn1)Br AS-5512 Cc1cc(sn1)C(=O)O AS-5513 Cc1ccsn1 AS-5514 Cc1c(c(no1)N)Cl AS-5515 Cc1coc(n1)N AS-5516 c1cn[nH]c1O AS-5517 CCOC(=O)c1c(nn(c1Cl)C)C(F)(F)F AS-5518 c1ccc2c(c1)OCC(O2)C#N AS-5519 Cc1c(sc(n1)N)C(=O)O AS-5520 CN1CCC(C1)C#N AS-5521 c1ccc(cc1)c2nc(sn2)N3CCNCC3 AS-5522 Cc1c(snn1)CO AS-5523 Cc1c(snn1)C=O AS-5524 C1C(=COC1=O)O AS-5525 c1cc(c2c(c1)scn2)N AS-5526 c1cc2c(cc1[N+](=O)[O-])ncs2 AS-5527 CC(C)(C)c1cccc(c1)CN AS-5528 C1COCCC1O AS-5529 Cn1c(ccn1)c2ccccc2N AS-5530 Cn1c(ccn1)c2ccc(cc2)N AS-5531 c1cc(cc(c1)[N+](=O)[O-])n2ccnc2 AS-5532 Cc1cc2c(cc1C)nc([nH]2)S AS-5533 c1c(cc(nc1N)Cl)C(F)(F)F AS-5534 c1c(scn1)CO AS-5535 CCOC(=O)c1c(c2c(cccc2s1)C)N AS-5536 COC(=O)c1c(c2ccc(cc2s1)Br)O AS-5537 c1cc(cc(c1)n2ccnc2)N AS-5538 c1c(cc(cc1C(F)(F)F)N2CCOCC2)C(=O)O AS-5539 c1c(cc(cc1C(F)(F)F)N2CCOCC2)C#N AS-5540 Cc1c(c(n(n1)c2ccccc2)C)C=O AS-5541 Cc1cc(n[nH]1)C AS-5542 c1c(cn[nH]1)Br AS-5543 C1C=CC(=C1)Cl AS-5544 c1cc(ccc1CN2CC(CC2=O)CO)F AS-5545 c1cc(ccc1CN2CC(CC2=O)C(=O)O)F AS-5546 CN1CC(CC1=O)C(=O)O AS-5547 C1C(CNC1=O)CO AS-5548 CN(C)c1cc(cc(n1)Cl)C(F)(F)F AS-5549 COc1cc(cc(n1)Cl)C(F)(F)F AS-5550 Cn1c(ccn1)C=O AS-5551 CC(=O)/C=C/c1cccc(c1)Br AS-5552 CC(C)(C)c1ccc(cn1)C#N AS-5553 c1c(cnc(c1Br)Cl)C=O AS-5554 Cc1ccc(c(n1)Cl)C(=O)OC AS-5555 Cc1cc(nnc1Cl)Cl AS-5556 c1cc(c(nc1)N2CCNCC2)C(F)(F)F AS-5557 c1cc2c(cc1N)nn[nH]2 AS-5558 CN1CCN(CC1)C2CCNCC2 AS-5559 CN(C)c1ccc(cn1)C(F)(F)F AS-5560 c1ccc2c(c1)cc(o2)C=O AS-5561 C/C(=N/O)/N AS-5562 c1ccnc(c1)c2nc(sn2)Cl AS-5563 c1(nnc(s1)Br)C(F)(F)F AS-5564 c1(nnc(s1)Cl)C(F)(F)F AS-5565 C1COCCN1c2nc(sn2)Cl AS-5566 c1ccc2c(c1)CC(=S)N2 AS-5567 Cc1c(csn1)C(=O)O AS-5568 c1cnoc1N AS-5569 CCOC(=O)c1c(nc(s1)C(F)(F)F)C(F)(F)F AS-5570 c1cc(ncc1F)C#N AS-5571 c1cnc(cc1Cl)C#N AS-5572 c1cnc(nc1C(F)(F)F)O AS-5573 Cc1c(c(nc(n1)O)C)Cl AS-5574 c1c(c(nc(n1)N)C(F)(F)F)Br AS-5575 c1cc(ccc1c2c[nH]nc2)F AS-5576 c1cc(cc2c1cc(s2)C=O)Br AS-5577 c1cc2c(cc1Br)cc(s2)CO AS-5578 c1cc2c(cc1Br)cc(s2)C=O AS-5579 c1ccc2c(c1)c(nc(n2)C(F)(F)F)O AS-5580 Cc1c2cc(ccc2sc1C(=O)C)Cl AS-5581 Cc1c(c(on1)c2ccccc2)C=O AS-5582 c1cc(sc1)c2cc(no2)C=O AS-5583 CC1Cc2ccccc2C1=O AS-5584 CC1(Nc2ccccc2CO1)C AS-5585 CC(=O)/C=C/c1ccccc1C(F)(F)F AS-5586 COc1cccc(c1)/C=N/O AS-5587 c1ccnc(c1)c2cccs2 AS-5588 CC(=O)C1Cc2ccccc2C1 AS-5589 Cc1ccnc(c1S(=O)(=O)N)Cl AS-5590 Cc1c(c(on1)c2ccccc2)CO AS-5591 Cc1ccc(cc1F)C(=S)N AS-5592 Cc1cc(c(nc1)C(=O)N)N AS-5593 COC(=O)c1cnc(s1)c2ccccc2 AS-5594 c1ccc(cc1)c2ncc(s2)C(=O)O AS-5595 CC(=O)/C=C/c1ccc(cc1)Br AS-5596 c1c(c(c(cn1)Br)O)Br AS-5597 c1cc(cnc1)c2cnco2 AS-5598 c1ccc(cc1)c2c(nccn2)C#N AS-5599 c1cc2c(cc1[N+](=O)[O-])nc([nH]2)C(F)(F)F AS-5600 CC(C)(C)OC(=O)N1CCN(CC1)C(=N)N AS-5601 c1ccc(cc1)n2cccc2C=O AS-5602 CCOC(=O)c1ccc(nc1C)C(F)(F)F AS-5603 CCOC(=O)c1cccnc1C(F)(F)F AS-5604 COc1ccc(nc1Br)N AS-5605 Cc1cccnc1NN AS-5606 c1cc(ncc1Cl)N2CCNCC2 AS-5607 c1ccc(cc1)c2nc(on2)Cl AS-5608 Cc1c(c(sn1)N)C(=O)N AS-5609 c1cc2c(cc1Cl)sc(n2)S AS-5610 c1cnc(cc1C(F)(F)F)OCCO AS-5611 C(=O)(C(F)(F)F)NN AS-5612 c1cc(c(cc1I)[N+](=O)[O-])N AS-5613 c1cc(c(cc1I)N)N AS-5614 c1ccc(cc1)C2CC(=CC(=O)C2)Cl AS-5615 c1ccc(cc1)C2CC(=CC(=O)C2)O AS-5616 c1c(c(cnc1Cl)N)C(=O)O AS-5617 CC(C)/C(=N/O)/N AS-5618 CCOC(=O)c1c(ccnc1Br)C AS-5619 Cc1ccnc(c1C(=O)O)Br AS-5620 CCOC(=O)c1ccn[nH]1 AS-5621 c1ccc(cc1)c2cc[nH]n2 AS-5622 Cc1csc2c1cc(cc2)F AS-5623 c1cc(c(cc1F)Cl)C/C(=N\O)/N AS-5624 COC(=O)c1cc(cnc1)F AS-5625 CC1CC(=O)c2c1cccc2 AS-5626 Cc1c(c(n[nH]1)C(F)(F)F)Br AS-5627 CC(C)(C)OC(=O)Nc1ccc(nc1)Cl AS-5628 C1C(CNC1=O)C(=O)N AS-5629 c1c(c(c(nc1Cl)Cl)C(=O)N)C(F)(F)F AS-5630 C1CCN(CC1)CCC#N AS-5631 Cc1ccnc(c1C#N)Cl AS-5632 c1csc2c1[nH]c(c2)C(=O)NN AS-5633 Cc1nnc(o1)c2cccc(c2)N AS-5634 c1c(cc(nc1Cl)Cl)C(=O)NN AS-5635 c1c(c(cc(c1F)F)N)N AS-5636 Cc1cccc(n1)CCCO AS-5637 COC(=O)C1CC(=O)NC1 AS-5638 c1ccc(cc1)CNc2ccc(cn2)N AS-5639 c1ccc(c(c1)c2cc[nH]n2)[N+](=O)[O-] AS-5640 c1cc(cc(c1)C(=O)N)C(=O)N AS-5641 Cc1c(sc(n1)c2ccccc2)CO AS-5642 CC(=O)/C=C/c1cccc(c1)Cl AS-5643 CCOC(=O)c1cc(nc(c1)Cl)Cl AS-5644 c1ccn2c(c1)nnc2S AS-5645 CC(C)(C)OC(=O)N1CCC(CC1)C#N AS-5646 c1ccc2c(c1)c(cs2)C(=O)O AS-5647 COC(=O)c1ccc(cc1F)Br AS-5648 c1cc2c(cc1N)C(=O)OC2 AS-5649 c1cc(nc(c1)Br)C=O AS-5650 c1cscc1C2CC(=O)CC(=O)C2 AS-5651 c1ccc(cc1)CNc2ccc(cn2)[N+](=O)[O-] AS-5652 Cn1c(c(cn1)C(=O)O)N AS-5653 Cc1nc(cs1)c2cccc(c2)[N+](=O)[O-] AS-5654 c1cc(nc(c1)Br)N2CCOCC2 AS-5655 c1ccn2c(c1)c(cn2)C(=O)O AS-5656 c1ccc(cc1)NC2(CCCCC2)C#N AS-5657 CN1CC(CC1=O)CO AS-5658 c1cc(ccc1C(=O)NN)OC(F)(F)F AS-5659 c1c(cc(cc1N)N2CCOCC2)C(F)(F)F AS-5660 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N AS-5661 c1c(cc(cc1Cl)Cl)CC#N AS-5662 CNCc1ccc(cc1)OC AS-5663 Cn1ccc(n1)c2ccc(cc2)[N+](=O)[O-] AS-5664 CC(=O)/C=C/c1ccsc1 AS-5665 c1cnc(nc1O)C(F)(F)F AS-5666 c1ccc(c(c1)C(F)(F)F)N2CCC(CC2)C(=O)O AS-5667 Cn1ccc(n1)c2cccc(c2)[N+](=O)[O-] AS-5668 Cc1c(cnn1c2ccc(cc2)F)C(=O)O AS-5669 c1ccc2c(c1)ncc(n2)C=O AS-5670 CC(C)(C)c1cccc(c1)N AS-5671 COC(=O)c1ccc(cc1)C=O AS-5672 c1cc2c(c(c1)Cl)snn2 AS-5673 Cc1cc(sn1)S(=O)(=O)N AS-5674 c1cnn(c1)c2ccc(cc2)CN AS-5675 c1cnn(c1)c2ccc(cc2)C#N AS-5676 c1cc(cc(c1)C(F)(F)F)c2nc(no2)N AS-5677 c1cc(ccc1c2ccnc(n2)S)N AS-5678 Cc1cc(nc(c1C#N)N(C)C)C AS-5679 CSc1nccc(n1)c2ccc(cc2)N AS-5680 Cc1c(c(nc(n1)S)N)C#N AS-5681 Cc1ccc(cn1)[N+](=O)[O-] AS-5682 c1cc(ccc1N2CC(CC2=O)C(=O)O)F AS-5683 CC(C)(C)c1ccc(c(c1)C#N)N AS-5684 CC(C)Sc1c(cccc1Cl)N AS-5685 C1CN(CCC1C(=O)O)C(=N)N AS-5686 CCOC(=O)c1ccc(nc1)N AS-5687 c1cc(cc(c1)N)c2nnc(o2)C(F)(F)F AS-5688 c1ccc(cc1)c2ccc(nn2)O AS-5689 COc1cscc1C(=O)OC AS-5690 Cc1cc(sn1)I AS-5691 Cc1c(c(sn1)C(=O)O)Br AS-5692 Cc1c(c(sn1)N)Br AS-5693 Cc1cc(sn1)c2ccc(cc2)C(=O)OC AS-5694 Cc1cc(sn1)c2cccc(c2)C=O AS-5695 Cc1cc(sn1)c2cccc(c2)NC(=O)C AS-5696 Cc1cc(sn1)c2cccc(c2)N AS-5697 CC(C)(C)OC(=O)Nc1cccs1 AS-5698 Cn1cc(nc1)C=O AS-5699 c1cc2c(cc1N)sc(n2)Cl AS-5700 c1csc2n1cc(n2)CO AS-5701 Cn1c(ccn1)c2ccccc2[N+](=O)[O-] AS-5702 c1cc([nH]c1)c2[nH]nnn2 AS-5703 CCOC(=O)c1cn2ccsc2n1 AS-5704 c1ccc(c(c1)/C=C/C(=O)O)C#N AS-5705 C1CC1/C(=N/O)/N AS-5706 c1cc(cc(c1)N)c2csc(n2)C(F)(F)F AS-5707 c1ccc2c(c1)C(NC2=O)CC(=O)O AS-5708 C1CSCc2c1nc(nc2O)S AS-5709 c1c(nc(nn1)S)S AS-5710 COC(=O)CC1c2ccccc2C(=O)N1 AS-5711 CC(=O)Nc1ccc(cc1)C(C)(C)C AS-5712 CN1CCN(CC1)c2c(cccn2)C(F)(F)F AS-5713 Cn1ccc(n1)c2ccccc2[N+](=O)[O-] AS-5714 COC(=O)c1c(cc(cn1)C(F)(F)F)Cl AS-5715 CN1CCc2c1cccc2 AS-5716 Cc1ccc(cn1)C#N AS-5717 c1cc(ccc1/C(=N\C#N)/N)F AS-5718 c1c(cnc(c1[N+](=O)[O-])F)Cl AS-5719 C=C(CN1CCCCC1)C#N AS-5720 Cc1c(nc(nc1O)C(F)(F)F)C AS-5721 CC(C)(C)OC(=O)N(C)c1ccc(cc1)N AS-5723 c1ccc(cc1)Cn2cc(cn2)C(=O)O AS-5724 c1c2n(nc1C(=O)O)CCCC2 AS-5725 Cc1c2cc(ccc2sc1S(=O)(=O)N)F AS-5726 Cc1c(c(sn1)Br)[N+](=O)[O-] AS-5727 c1cc(c(cc1N)O)C(F)(F)F AS-5728 c1cc(c(cc1[N+](=O)[O-])O)C(F)(F)F AS-5729 CC(C)(C)OC(=O)Nc1ccc(c(c1)O)Cl AS-5730 CN(C)c1cc(cc(n1)C#N)C(F)(F)F AS-5731 c1ccc(cc1)c2cc3c(n[nH]c3nn2)N AS-5732 c1ccc(cc1)c2cc(c(nn2)Cl)C(=O)N AS-5733 c1ccc(cc1)CN2[C@@H](CCC2=O)CC#N AS-7001 c1ccc(cc1)CN2[C@H](CCC2=O)CC#N AS-7002 c1ccc(cc1)CN2[C@@H](CCC2=O)CCl AS-7003 c1ccc(cc1)CN2[C@H](CCC2=O)CCl AS-7004 c1ccc(cc1)CN2[C@@H](CCC2=O)CO AS-7005 c1ccc(cc1)CN2[C@@H](CCC2=O)C(=O)O AS-7007 CNS(=O)(=O)Cc1ccc(cc1)[N+](=O)[O-] AS-7011 CNS(=O)(=O)Cc1ccc(cc1)N.Cl AS-7012 CCCS(=O)c1ccc2c(c1)nc([nH]2)NC(=O)OC AS-7013 CCCS(=O)(=O)c1ccc2c(c1)nc([nH]2)NC(=O)OC AS-7014 COC(=O)c1c2ccccc2ccc1O AS-7015 CCOC(=O)[C@@H]1CCC(=O)N1Cc2ccccc2 AS-7019 CC(C(=O)c1cnccn1)C(=O)OC AS-7021 COC(=O)[C@H]1CCC(=O)N1 AS-7023 C1COCCN1CCC(=O)O.Br AS-7031 Cc1c(ssc1=S)c2cnccn2 AS-7036 C1COCCN1CC2CN(C(=O)O2)N AS-7038 c1cc(oc1/C=N/NC(=O)c2cc(cc(c2O)[N+](=O)[O-])[N+](=O)[O-])[N+](=O)[O-] AS-7049 CC(C)(C)OC(=O)c1ccc(cc1)C=O AS-7050 CC(C)(C)OC(=O)c1ccc(cc1)CN AS-7052 c1nc2c(nc(nc2[n@]1C3[C@@H]([C@@H]([C@H](O3)CO)O)O)I)N AS-7057 CC(=O)OC[C@@H]1[C@H]([C@H]([C@@H](O1)n2cnc3c2nc(nc3Cl)N)OC(=O)C)OC(=O)C AS-7059 CC(=O)OC[C@@H]1[C@H]([C@H]([C@@H](O1)n2cnc3c2nc(nc3Cl)I)OC(=O)C)OC(=O)C AS-7060 c1ccc(cc1)Cn2c(c(cn2)C#N)N AS-7067 c1c(c(n(n1)CC(F)(F)F)N)C#N AS-7068 Cc1c(c(n(n1)CC(F)(F)F)N)C#N AS-7070 Cc1c(c(n(n1)Cc2ccccc2)N)C#N AS-7071 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)CCN3CCOCC3 AS-7078 Cc1c(nc2ccccc2n1)C(=O)[O-].[Na+] AS-7080 c1ccc(cc1)OC(=O)NC(=O)Oc2ccccc2 AS-7082 c1cc(ccc1/C=N/NC(=O)N)[N+](=O)[O-] AS-7083 CC(=O)OC1CCC2C1(CCC3C2CCc4c3ccc(c4)C(=O)O)C AS-7084 c1cn2cc(cc(c2n1)Br)F AS-8000 Cc1ccc(cc1)Oc2cccc3c2c(n[nH]3)N AS-8001 CC(=O)c1ccc(c(c1)N)O AS-8002 CCOC(=O)Cc1ccc(cc1)I AS-8003 Cc1c(cc(c2c1cn[nH]2)[N+](=O)[O-])Br AS-8004 CCOC(=O)c1ccc2c(c1)OCC(=O)N2 AS-8005 CCOc1ccc(cc1N)N AS-8006 COC(=O)Cc1ccccc1[N+](=O)[O-] AS-8007 c1cc(c(nc1)Oc2ccc(cc2)Cl)C#N AS-8008 Cc1c(sc(n1)C)C(=O)/C=C/N(C)C AS-8009 Cc1c(sc(n1)C)c2cc[nH]n2 AS-8010 CCOC(=O)Cc1ccc(c(c1)[N+](=O)[O-])O AS-8011 CC(c1ccc(c(c1)OC)OC)O AS-8012 CCOC(=O)Cc1ccc(c(c1)N)O AS-8013 c1ccc(c(c1)C(=O)O)Oc2c(cc(cn2)C(F)(F)F)Cl AS-8014 COC(=O)c1ccccc1Oc2c(cc(cn2)C(F)(F)F)Cl AS-8015 CCOC(=O)c1ccc(nc1)O AS-8016 CN(C)/C=C/C(=O)c1cccc(c1)OC(F)(F)F AS-8017 c1cc(cc(c1)OC(F)(F)F)c2cc[nH]n2 AS-8018 CCOc1ccc(c(c1)N)[N+](=O)[O-] AS-8019 CC(C)(C)c1cc(c(c(c1)[N+](=O)[O-])O)C(C)(C)C AS-8020 Cc1cc(nn1C)C(=O)NN AS-8021 Cc1cc(n(n1)C)C(=O)NN AS-8022 Cc1cc([nH]n1)C(=O)NN AS-8023 CCOC(=O)c1c(c(n(n1)C)C)Br AS-8024 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)OC AS-8025 CCOC(=O)c1cc(c(nc1)O)Br AS-8026 CCOC(=O)c1c(c([nH]n1)C)Br AS-8027 Cn1ccc2c1cccc2/C(=N\O)/N AS-8028 CCOC(=O)c1cc(c(nc1)O)Cl AS-8029 COC(=O)c1ccn2c(c1)ncc2[N+](=O)[O-] AS-8030 c1c(cn2c(cnc2c1Cl)[N+](=O)[O-])C(F)(F)F AS-8031 c1c(c(c(c(c1F)O)F)F)C(=O)O AS-8032 c1c(c(c(c(c1F)NN)F)F)C(=O)NN AS-8033 c1cc(ncc1Br)c2cnco2 AS-8034 Cc1cn2cc(ccc2n1)[N+](=O)[O-] AS-8035 c1cc(c(cc1C(F)(F)F)N)N2CCCCC2 AS-8037 CC(=O)N(C)Cc1cccnc1 AS-8038 COC(=O)c1cc(c(c(c1F)F)O)F AS-8039 COC(=O)c1ccc(nc1)NC(=O)CCCCl AS-8040 CCOC(=O)c1ccc(cc1)NC(=O)CCCCl AS-8041 Cc1c(cccc1[N+](=O)[O-])NC(=O)CCCCl AS-8042 CC(C)(C)OC(=O)Cn1ccc2c1ccc(c2)[N+](=O)[O-] AS-8043 CCOC(=O)c1cc(c(c(c1F)F)O)F AS-8044 c1cc(ccc1/C(=N/O)/N)[N+](=O)[O-] AS-8045 Cc1nc(no1)c2ccc(cc2)[N+](=O)[O-] AS-8046 COc1c(cc(c(c1F)F)C(=O)OC)F AS-8047 c1cnc(nc1n2ccnc2)Cl AS-8048 c1cnc(nc1Cl)n2ccnc2 AS-8049 CC(=O)N/C(=N\O)/c1ccc(cc1)[N+](=O)[O-] AS-8050 COC(=O)c1cc(c(c(c1F)F)N2CCOCC2)F AS-8051 CCOC(=O)c1cc(c2nccn2c1)Cl AS-8052 COC(=O)c1cc(c(c(c1F)F)N2CCCCC2)F AS-8053 COC(=O)c1cc(c(c(c1F)F)N2CCCC2)F AS-8054 c1cc2ncc(n2cc1C(F)(F)F)N AS-8055 CN1CCN(CC1)c2c(cc(c(c2F)F)C(=O)OC)F AS-8056 c1c(cc(c(c1Br)O)Br)CCC(=O)O AS-8057 CN(OC)S(=O)(=O)c1ccccc1N AS-8058 CCOC(=O)c1cc2cc(cc(c2o1)Br)Cl AS-8059 COc1c(cc(c(c1F)F)C(=O)Cl)F AS-8060 COc1c(cc(c(c1F)F)C(=O)N)F AS-8061 COc1c(cc(c(c1F)F)C#N)F AS-8062 CC1CN(CC(O1)C)c2c(cc(c(c2F)F)C(=O)OC)F AS-8063 c1c(c(c(c(c1F)N2CCCC2)F)F)C(=O)O AS-8064 COC(=O)c1cc(c(c(c1F)F)n2cccn2)F AS-8065 Cn1ccc2c1c(ccc2)C#N AS-8066 CCOC(=O)c1cc2c([nH]1)cccc2Cl AS-8067 Cn1ccc2c1c(ccc2)CN AS-8068 CC(C)Sc1ccc(cc1)Br AS-8069 c1cc(ncc1[N+](=O)[O-])OCC2CCOCC2 AS-8070 c1cc(c(cc1c2csc(n2)N)[N+](=O)[O-])Cl AS-8071 COc1cc(c(cc1F)C(=O)OC)F AS-8072 COC(=O)c1cc(c(cc1F)N2CCOCC2)F AS-8073 c1ccc2c(c1)cc(s2)C(=O)NN AS-8074 c1cc2cc(sc2nc1)CO AS-8075 CCOC(=O)c1cc(c(cc1F)F)F AS-8076 c1cc(c(cc1CC(=O)N)Cl)Cl AS-8077 c1cnc(nc1)N2CCC(CC2)C(=O)NN AS-8078 c1cc2cc(sc2nc1)C#N AS-8079 Cc1ccnc(c1[N+](=O)[O-])n2ccnc2 AS-8080 CN1CCN(CC1)c2cc(c(cc2F)C(=O)OC)F AS-8081 CN1CCN(CC1)c2cc(c(cc2F)C(=O)O)F AS-8082 CC1CN(CC(O1)C)c2cc(c(cc2F)C(=O)OC)F AS-8083 COC(=O)c1cc(c(cc1F)N2CCCCC2)F AS-8084 Cn1c2ccccc2cc1C#N AS-8085 CCOc1cc(c(cc1F)C(=O)OCC)F AS-8086 c1cc(cc(c1)C#N)CN2CCCCC2 AS-8087 c1cc2nccn2cc1[N+](=O)[O-].Cl AS-8088 CC1CN(CC(O1)C)Cc2cccc(c2)C#N AS-8089 c1cc(cc(c1)C#N)CN2CCOCC2 AS-8090 COc1cc(c(cc1F)C(=O)O)F AS-8091 c1cc(cc(c1)OC(F)F)NC(=O)CCl AS-8092 c1cc(ccc1NC(=O)Nc2ccc(cc2)Cl)F AS-8093 c1cc(ccc1NC(=O)Nc2ccc(cc2)Cl)OC(F)(F)F AS-8094 CC1CN(CC(O1)C)C(=O)Nc2ccc(cc2)Cl AS-8095 c1cc(cc(c1)OC(F)F)NC(=O)Nc2ccc(cc2)Cl AS-8096 CC1C(=O)Nc2cc(ccc2O1)Cl AS-8097 CCC1CCCCN1c2nnc(s2)N AS-8098 CC(C)c1ccc(c(c1)Br)NC(=S)N AS-8099 c1c(cc(c(c1F)NC(=S)N)Br)Br AS-8100 CCOC(=O)c1cc(sc1Cl)Cl AS-8101 CC(C)c1ccc(c(c1)Br)NC(=S)Nc2cccc(c2)OC(F)F AS-8102 c1cc(cc(c1)OC(F)F)n2cn[nH]c2=O AS-8103 COC(=O)c1ccccc1N2CCOCC2 AS-8104 COC(=O)C12CC3CC(C1)CC(C3)(C2)O AS-8105 c1c(nc(nc1Cl)N)NCCO AS-8106 COc1cc(c(cc1Cl)OC)NC(=S)N AS-8107 Cn1c2ccccc2c(n1)NC(=S)Nc3cc(c(cc3OC)Cl)OC AS-8108 Cc1cc(cc(c1NC(=S)Nc2c3ccccc3n(n2)C)Cl)Cl AS-8109 CNS(=O)(=O)c1ccc(cc1)I AS-8110 c1cc(ccc1NC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl)Cl AS-8111 Cc1cc(cc(c1NC(=S)N2CCOCC2)Cl)Cl AS-8112 c1cc(c(cc1NC(=O)N2CCOCC2)[N+](=O)[O-])Cl AS-8113 COC(=O)c1ccc(nc1)NC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl AS-8114 c1cc(c(cc1NC(=O)N2CCCC2)[N+](=O)[O-])Cl AS-8115 CN1CCN(CC1)C(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl AS-8116 c1cc(c(cc1NC(=O)N2CCCCC2)[N+](=O)[O-])Cl AS-8117 c1cnn(c1)C(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl AS-8118 c1cc(cc(c1)Br)N2CC(CC2=O)C(=O)O AS-8119 c1cc(c(cc1NC(=O)n2ccnc2)[N+](=O)[O-])Cl AS-8120 Cc1cccc(c1NC(=S)Nc2cccc(c2)OC(F)F)C(C)C AS-8121 C(CO)Nc1nnc(s1)N AS-8122 CCc1ccccc1NNC(=S)N AS-8123 CCOC(=O)c1c(nn(c1C)c2cc(cc(c2)Cl)Cl)C AS-8124 c1cc(c(cc1S(=O)(=O)NN)Cl)Cl AS-8125 COC(=O)c1cc2c(s1)cccn2 AS-8126 c1ccn(c1)c2c(cc(cn2)Br)C(F)(F)F AS-8127 c1cc(c(nc1)N2CCCCC2)/C(=N/O)/N AS-8128 c1cc(c(nc1)N2CCCC2)C#N AS-8129 Cc1c(n2ccccc2n1)Br AS-8130 Cc1nc2c(cccc2o1)C(=O)O AS-8131 COC(=O)c1cc2c(s1)nc(nc2Cl)N AS-8132 c1cc(c2c(c1)ocn2)C(=O)O AS-8133 Cn1cc(c(n1)CO)Br AS-8134 Cc1c2cccnc2n(n1)C AS-8135 CN(C)C(=O)c1ccc(cc1)[N+](=O)[O-] AS-8136 CCOC(=O)c1ccc2cn(nc2c1)C(=O)C AS-8137 c1cc(ccc1C(=O)N2CCCCC2)[N+](=O)[O-] AS-8138 CC1(CCCC(N1C(=O)c2ccc(cc2)[N+](=O)[O-])(C)C)C AS-8139 CCOC(=O)c1ccc2cn[nH]c2c1 AS-8140 CC(C)N(C(C)C)C(=O)c1ccc(cc1)[N+](=O)[O-] AS-8141 CN(C(=O)c1ccc(cc1)[N+](=O)[O-])OC AS-8142 Cn1c2c(cccn2)c(n1)C(=O)OC AS-8143 c1ccn2cc(nc2c1)c3ccc(cc3)C#N AS-8144 c1ccn2cc(nc2c1)c3ccc(cc3)C(=O)O.O.Cl AS-8145 CCOC(=O)c1ccc(cc1)c2cn3ccccc3n2 AS-8146 COC(=O)c1ccc(cc1)c2cn3ccccc3n2 AS-8147 c1cc(ccc1C#N)c2cn3cc(ccc3n2)Br AS-8148 c1cc(c2nc(cn2c1)c3ccc(cc3)C#N)C(F)(F)F AS-8149 c1cc(ccc1C#N)c2cn3cc(ccc3n2)C(F)(F)F AS-8150 c1cc(ccc1C#N)c2cn3cc(ccc3n2)Cl AS-8151 c1cc(ccc1C#N)c2cn3ccc(cc3n2)Br AS-8152 c1cnc2nc(cn2c1)c3ccc(cc3)C#N AS-8153 c1ccn2c(c1)nc(c2Br)c3ccc(cc3)C#N AS-8154 c1cc(ccc1C#N)c2cn3ccc(cc3n2)Cl AS-8155 c1cc(ccc1C#N)c2cn3cc(ccc3n2)F AS-8156 c1cc(ccc1C#N)c2cn3cc(cc(c3n2)Cl)C(F)(F)F AS-8157 c1cc(c2nccn2c1)C#N AS-8158 c1ccn2cc(nc2c1)c3ccc(cc3)/C(=N/O)/N AS-8159 CC(C)N(C(C)C)S(=O)(=O)c1ccc(cc1Cl)Cl AS-8160 CC(C)N(C(C)C)C(=O)Nc1ccc(c(c1)[N+](=O)[O-])Cl AS-8161 CC(C)c1ccc(c(c1)Br)NC(=S)N(C(C)C)C(C)C AS-8162 CC(C)N(C(C)C)C(=S)Nc1c(cc(cc1Br)Br)F AS-8163 c1cc(c(cc1NC(=O)NCCCl)C(F)(F)F)C#N AS-8164 Cc1c(c(c(nc1C)O)C#N)C AS-8165 C1CCN(C1)CC(C(F)(F)F)O AS-8166 c1cnn(c1)CC(C(F)(F)F)O AS-8167 CC(C)N(C(C)C)S(=O)(=O)c1ccc(cc1)OC(F)(F)F AS-8168 CNC(=O)c1c[nH]c2c1cccc2 AS-8169 CC(C)N(C(C)C)C(=O)c1c[nH]c2c1cccc2 AS-8170 CC(C)N(C(C)C)C(=O)c1ccc(cc1Cl)Cl AS-8171 CNC(=O)c1cc2cccc(c2s1)Br AS-8172 c1cc2cc(sc2c(c1)Br)C(=O)N AS-8173 CC(C)(C)OC(=O)N1CCN(CC1)CC(C(F)(F)F)O AS-8174 c1cc2cc(sc2c(c1)Br)C=O AS-8175 CC(C)N(C(C)C)C(=O)c1cccc(c1)Br AS-8176 Cn1cccc1C(=O)N AS-8177 Cn1cccc1C#N AS-8178 CCCCCc1ccc(cc1)C(=O)N(C(C)C)C(C)C AS-8179 CC(C)N(C(C)C)C(=O)c1ccc(nc1)C(F)(F)F AS-8180 Cc1cc(cc(c1NC(=S)N(C(C)C)C(C)C)Cl)Cl AS-8181 Cn1ccc2c1cc(cc2)C#N AS-8182 C=CCOc1cccc(c1)C=O AS-8183 CC(C)(C)OC(=O)N1CCN(CC1)Cc2cccc(c2)C#N AS-8184 Cc1nc(cn1C)S(=O)(=O)N(C)C AS-8185 CN1CCOc2c1ccc(c2)C=O AS-8186 C(CO)N(CCO)CCS(=O)(=O)[O-].[Na+] AS-8187 c1cc(c(cc1C(=O)O)[N+](=O)[O-])N AS-8188 c1cc(c(c(c1C(=O)O)O)O)O AS-8189 c1c(cc(c(c1F)N)F)Br AS-8191 c1cnc(cc1F)Cl AS-8192 c1cc(ccc1C(F)(F)F)O AS-8193 Cc1c(cccc1OC(=O)C)C(=O)O AS-8194 c1cc(c(cc1C#N)[N+](=O)[O-])O AS-8195 COC(=O)c1cccc(c1)C=O AS-8196 c1cn2cc(cc(c2n1)[N+](=O)[O-])Br AS-8197 COC(=O)c1cc(c(c(c1)Cl)N)[N+](=O)[O-] AS-8198 c1ccn2c(c1)nc(c2Cl)C(=O)O AS-8199 CCOC(=O)c1c(n2ccccc2n1)Cl AS-8200 c1cc2nc(cn2c(c1)Cl)C(=O)NN AS-8201 c1c(cn2cc(nc2c1Br)C(=O)NN)Cl AS-8202 c1cc2c(cc1I)cn[nH]2 AS-8203 c1ccn2cc(nc2c1)C(=O)NCCO AS-8204 CN(C)Cc1cnc2n1cc(cc2)Cl.Cl AS-8205 COc1ccc2c(c1)nc(o2)CCl AS-8206 c1c(c(c(c(c1Cl)Cl)[N+](=O)[O-])O)[N+](=O)[O-] AS-8207 COc1ccc2c(c1)C(CC2=O)N.Cl AS-8208 CC(=O)n1cc2c(n1)cccc2Cl AS-8209 CC(=O)n1cc2cc(ccc2n1)I AS-8210 c1cc2ncc(n2cc1/C(=N/O)/N)Br AS-8211 CC(=O)Oc1cc2cn[nH]c2c(c1)[N+](=O)[O-] AS-8212 c1cc2c(cc1C#N)nc(o2)CCl AS-8213 CCOC(=O)c1cccc(c1)NC(=O)NCCCl AS-8214 c1ccn2c(c1)nc(c2Cl)C(=O)NN AS-8215 c1cc2c(cc1NC(=O)NCCCl)OCO2 AS-8216 CCOC(=O)c1c(n2c(n1)cccc2Cl)Cl AS-8217 CCOC(=O)c1c(n2c(n1)cccc2Cl)Br AS-8218 Cn1c2ccc(cc2c(n1)N)[N+](=O)[O-] AS-8219 c1cc(ccc1c2nnco2)[N+](=O)[O-] AS-8220 c1ccn(c1)c2cccc(c2)CO AS-8221 Cn1c2cccc(c2c(n1)N)I AS-8222 c1cc2c(cc1Cl)nc([nH]2)CCl AS-8223 Cn1c2cc(ccc2c(n1)N)Cl AS-8224 Cn1c2cc(ccc2c(n1)N)OC AS-8225 Cc1coc(n1)c2ccccc2 AS-8226 COC(=O)c1ccn2c(c1)ncc2Br AS-8227 c1cn2c(cc1C(=O)O)ncc2Br AS-8228 c1cn2c(cc1C(=O)NN)ncc2Br AS-8229 CCOC(=O)c1cn2ccc(cc2n1)C(=O)OC.Br AS-8230 c1cc(c2c(c1)nco2)C(=O)O AS-8231 COC(=O)c1cc(c2nccn2c1)Br AS-8232 c1cc2c(c(c1)C(F)(F)F)[nH]nc2N AS-8233 Cn1c2c(cccc2C(F)(F)F)c(n1)N AS-8234 COC(=O)c1ccn2c(c1)ncc2Cl AS-8235 CCOC(=O)c1c(c2cccc(c2s1)C(F)(F)F)N AS-8236 CCOC(=O)CSc1ccnc2c1ccc(c2)Cl AS-8237 c1c(cnc(c1Cl)n2cc(cn2)Br)C(F)(F)F AS-8238 c1cc2c(ccnc2cc1Cl)SCC(=O)O AS-8239 c1cc(ccc1C(=O)NN)Oc2c(cc(cn2)C(F)(F)F)Cl AS-8240 c1cc(ccc1C(=O)O)Oc2c(cc(cn2)C(F)(F)F)Cl AS-8241 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N AS-8242 CC1(COc2ccccc2NC1=O)C AS-8243 COC(=O)c1cccc2c1c(n[nH]2)Br AS-8244 CCOc1ccc(cc1[N+](=O)[O-])N AS-8245 COC(=O)c1cc(c(c(c1)Br)N)N AS-8246 Cc1cc(c(c(c1)Br)N)N AS-8247 COC(=O)CSc1ccc(cc1[N+](=O)[O-])N AS-8248 c1cc2nccn2cc1C(=O)N AS-8249 CCOC(=O)c1cccc(c1)c2cnco2 AS-8250 c1cc(ccc1NC(=O)CCl)Br AS-8251 c1c(c2c(cn[nH]2)c(c1Br)[N+](=O)[O-])Br AS-8252 Cn1c2ccccc2c(n1)n3cccc3 AS-8253 Cn1c2ccccc2c(n1)N3CCCC3=O AS-8254 COC(=O)c1cc2c(c(c1)Br)nc[nH]2 AS-8255 COc1cccc(c1)n2cn[nH]c2=O AS-8256 c1cc(cc(c1)Br)/C=C/C(=O)O AS-8257 CCOC(=O)c1c(n2c(cccc2n1)C)Br AS-8258 Cc1cccc2n1cc(n2)C(=O)NN AS-8259 COC(=O)c1cc2cn[nH]c2c(c1)Br AS-8260 CCOC(=O)c1cn2c(c(cc(c2n1)Br)Br)C AS-8261 CCOC(=O)c1cccc(c1)N2CCNC2=O AS-8262 c1cc(cc(c1)N2CCNC2=O)C(=O)O AS-8263 Cc1cc(cc2c1nn(c2)C(=O)C)Br AS-8264 CCOC(=O)c1cnc2n1cc(cc2)Cl AS-8265 CCCCCCCn1c2cc(ccc2cn1)N AS-8266 Cc1cc(c(cc1C)O)[N+](=O)[O-] AS-8267 Cc1cc(cc(c1O)Cl)[N+](=O)[O-] AS-8268 c1cc(ccc1n2cn[nH]c2=O)F AS-8269 Cn1c2ccccc2cc1C(=O)NN AS-8270 Cc1c(c(n(n1)CO)C)Br AS-8271 Cn1c2ccc(cc2cn1)NC(=O)CCl AS-8272 c1cc2c(cc1C(F)(F)F)[nH]nc2Br AS-8273 CCOc1c(cccn1)C(=O)OCC AS-8274 CCOc1c(cc(cn1)Br)C(=O)OCC AS-8275 c1cn2cc(cc(c2n1)C(F)(F)F)Br AS-8276 c1cn2cc(cc(c2n1)Br)C(F)(F)F AS-8277 c1cc(c2nccn2c1)C(F)(F)F AS-8278 c1cc(c2ncc(n2c1)Br)C(F)(F)F AS-8279 Cc1ccc(c2c1c(n[nH]2)Br)[N+](=O)[O-] AS-8280 c1cc(c2c(c1)[nH]nc2Cl)C(F)(F)F AS-8281 CCOC(=O)c1c(n2cc(ccc2n1)F)Br AS-8282 CCOC(=O)c1cc(c2nccn2c1)Br AS-8283 c1cn2cc(cc(c2n1)Br)C(=O)O AS-8284 Cc1ccc(c(c1C)n2cccc2)[N+](=O)[O-] AS-8285 c1c(c(c2cn[nH]c2c1Br)N)Br AS-8286 Cc1cc(ccc1Br)NC(=O)CCCCl AS-8287 CC(=O)n1cc2cc(c(c(c2n1)Br)C(=O)OC)Br AS-8288 Cc1cc(ccc1Br)N2CC(CC2=O)C(=O)O AS-8289 Cc1cc(ccc1Br)n2cn[nH]c2=O AS-8290 Cn1c2ccccc2c(n1)n3cn[nH]c3=O AS-8291 COC(=O)c1ccc2c(c1)[nH]nc2Br AS-8292 COC(=O)c1cc2cn[nH]c2c(c1)Cl AS-8293 c1ccn(c1)c2cccc3c2[nH]nc3 AS-8294 CCOC(=O)c1c(n2ccc(cc2n1)Cl)Br AS-8295 c1cc(ccc1CO)NC(=O)/C=C\C(=O)O AS-8296 Cn1c2ccccc2c(n1)NC(=O)/C=C\C(=O)O AS-8297 Cn1c2ccccc2c(n1)NC(=O)CCC(=O)O AS-8298 Cn1c2ccccc2c(n1)N3C(=O)C=CC3=O AS-8299 COC(=O)c1ccsc1NC(=O)/C=C\C(=O)O AS-8301 Cc1cc(cc(c1NC(=S)N)Cl)Cl AS-8302 c1cc(c(cc1NC(=O)/C=C\C(=O)O)[N+](=O)[O-])F AS-8303 Cc1cc(cc(c1NC(=S)NC)Cl)Cl AS-8304 Cc1ccc2cn[nH]c2c1 AS-8305 CN(c1ccc(cn1)Cl)N AS-8306 COC(=O)c1cnc2n1cc(cc2)Br AS-8307 c1cc2ncc(n2cc1Br)C(=O)NN AS-8308 c1csc(n1)c2cnco2 AS-8309 Cn1c2ccc(cc2cc1C(=O)NN)Br AS-8310 C[C@@H](C(C(=O)O)[N@@]1Cc2ccccc2C1=O)O AS-8311 c1cc2c(cc1C#N)[nH]c(=S)o2 AS-8312 CC(C)(C)C(C(=O)O)[N@@]1Cc2ccccc2C1=O AS-8313 CC(C(C(=O)OC)N1Cc2ccccc2C1=O)O AS-8314 CCC(C(=O)O)N1Cc2ccccc2C1=O AS-8315 Cc1nc2cc(ccc2o1)OC AS-8316 c1cc2c(cc1C#N)nco2 AS-8317 CC(C(=O)OC)N1Cc2ccccc2C1=O AS-8318 c1ccc2c(c1)CN(C2=O)c3cccc(c3)C(=O)O AS-8319 CC(C)C(C(=O)OC)N1Cc2ccccc2C1=O AS-8320 COC(=O)CCN1Cc2ccccc2C1=O AS-8321 c1cc(sc1c2cnco2)S(=O)(=O)N AS-8322 c1c(c(cc2c1OCO2)[N+](=O)[O-])[N+](=O)[O-] AS-8323 CCOC(=O)c1ccc2c(c1)c(n[nH]2)Br AS-8324 CCOC(=O)c1ccn2c(c1)ncc2Br AS-8325 c1cc(c(cc1c2cnco2)I)F AS-8326 Cn1c2ccccc2c(n1)NC(=O)CCCCl AS-8327 Cn1c2ccccc2c(n1)NS(=O)(=O)c3ccc(cc3)I AS-8328 CN1CCOc2c1cccc2 AS-8329 CCOC(=O)c1cc2cc(cc(c2o1)Br)[N+](=O)[O-] AS-8330 CCc1nc2c(o1)cccn2 AS-8331 c1cc(cc(c1)[N+](=O)[O-])c2ccsc2 AS-8332 CC1(CC(c2c1cc3c(c2[N+](=O)[O-])cn[nH]3)(C)C)C AS-8333 Cc1c(c(c2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)Br)N AS-8334 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NC(=O)NCCCl AS-8335 CC1(CC(c2c1cc3c(c2N)cn[nH]3)(C)C)C AS-8336 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)n3cccc3 AS-8337 c1cc2cnc(nc2cc1Br)N AS-8338 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCCCC4 AS-8339 c1cc2ncc(n2cc1C(=O)NN)Cl AS-8340 c1cc2cc(sc2c(c1)C(F)(F)F)C(=O)NN AS-8341 COC(=O)CCSc1cccc(c1C=O)Cl AS-8342 c1cc2ncc(n2cc1C#N)Cl AS-8343 c1c(cnc(c1Cl)SCCC(=O)NN)C(F)(F)F AS-8344 Cn1c(c(cn1)Br)C=O AS-8345 COC(=O)CCSc1ccc(cn1)[N+](=O)[O-] AS-8346 CCOc1c(cc(cn1)Cl)C(=O)O AS-8347 c1cc2c(cc1I)c(n[nH]2)N AS-8348 CN(C)/C=C/c1ccncc1[N+](=O)[O-] AS-8350 COc1ccc(nn1)I AS-8351 Cc1ccc(c(c1)C)C(=O)/C=C/N(C)C AS-8352 CCOC(=O)c1c(c2ccc(cc2s1)Br)N AS-8353 c1cc2ncc(n2cc1C#N)I AS-8354 CCOC(=O)c1c(c2c(s1)cccc2Br)N AS-8355 c1ccc2c(c1)c(c([nH]2)C(=O)NN)I AS-8356 c1ccc2c(c1)c(c([nH]2)C(=O)O)I AS-8357 CCOC(=O)c1c(c2cc(ccc2s1)I)N AS-8358 CCOC(=O)c1c(c2ccc(cc2s1)Br)n3cccc3 AS-8359 Cn1c2ccc(cc2c(n1)N)I AS-8360 CCOC(=O)c1c(c2cc(ccc2[nH]1)OC(F)(F)F)Br AS-8361 CCOC(=O)Cc1csc(n1)C AS-8362 CCc1nc2cccc(c2o1)C(=O)OC AS-8363 Cc1c(c(no1)c2ccccc2)C(=O)/C=C/N(C)C AS-8364 c1cc2c(c(c1)Cl)c(c([nH]2)Cl)C=O AS-8365 CCn1c2ccccc2c(c1Cl)C=O AS-8366 c1cn2cc(nc2cc1Cl)C(=O)NN AS-8367 CCc1[nH]c2cc(c(cc2n1)Cl)Cl AS-8368 C1COCCN1c2nnc(s2)N AS-8369 C1CCN(CC1)c2nnc(s2)N AS-8370 C1CCN(C1)c2nnc(s2)N AS-8371 CN1CCN(CC1)c2nnc(s2)N.Br AS-8372 Cc1cc(cn2c1nc(c2)C(=O)O)I AS-8373 COC(=O)c1cccc2c1OCC(=O)N2 AS-8374 CCCCc1[nH]c2ccccc2n1 AS-8375 CCCc1nnc(o1)c2ccc(cc2)[N+](=O)[O-] AS-8376 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)Br)C AS-8377 CCN(CC)c1nnc(s1)N AS-8378 CC1(CC(c2c1c(c3cn[nH]c3c2Br)[N+](=O)[O-])(C)C)C AS-8379 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NC(=O)C AS-8380 CN1c2c(cccc2OCC1=O)[N+](=O)[O-] AS-8381 COc1ccc2c(c1)NC(=O)CO2 AS-8382 CCCc1nnc(o1)c2ccc(cc2)N AS-8383 CC(=O)Nc1c(cccc1F)[N+](=O)[O-] AS-8386 c1cc(c2cnc(nc2c1)N)C(F)(F)F AS-8387 c1cc2c(cc1C(F)(F)F)cnc(n2)N AS-8388 COC(=O)c1cc(nc(c1)Cl)N2CCOCC2 AS-8389 COC(=O)c1cc(nc(c1)Cl)N2CCCCC2 AS-8390 COC(=O)c1cc(nc(c1)Cl)N2CCNCC2 AS-8391 CN1CCN(CC1)c2cc(cc(n2)Cl)C(=O)OC AS-8392 c1cc(c(c(c1)F)N)[N+](=O)[O-] AS-8393 CC(=O)Nc1ccc(cc1F)[N+](=O)[O-] AS-8394 c1c(cc(c(c1[N+](=O)[O-])N)F)I AS-8395 c1cc(c(cc1[N+](=O)[O-])I)N AS-8396 CCOC(=O)c1cn2cccc(c2n1)[N+](=O)[O-] AS-8397 CCOC(=O)c1cc2cc(ccc2s1)Br AS-8398 c1cc(c(c(c1)Cl)N2CCNCC2)[N+](=O)[O-] AS-8399 CCOC(=O)c1cc([nH]c1C)C AS-8400 Cc1c(c(cc(c1[N+](=O)[O-])Br)Br)N AS-8401 CC(=O)N1CCCN(CC1)c2ccc(cc2)[N+](=O)[O-] AS-8402 COC(=O)c1cc(c(nc1)N)Cl AS-8403 CCOC(=O)c1cccn1C AS-8404 CCCCCCCCc1ccc(cc1)C(=O)OCC AS-8405 c1cc(ccc1c2cnco2)C(F)(F)F AS-8406 CCCCc1nc2cc(ccc2o1)C(=O)OC AS-8407 COc1cccc2c1c(c(s2)C(=O)OC)N AS-8408 Cn1c2cccc(c2c(n1)N)Br AS-8409 Cn1c2cccc(c2c(n1)N)OC AS-8410 CCOC(=O)c1c(c2c(cccc2s1)OC)N AS-8411 c1cc2ncc(n2cc1Cl)Br AS-8412 c1cc2c(cc1c3cnco3)OCCO2 AS-8413 c1cc2ncc(n2cc1CO)Br AS-8414 CNC(=O)c1ccc(nc1)Cl AS-8415 CCOc1c(cc(cn1)I)C(=O)OC AS-8416 Cc1c(cc2c(c1N)C(CC2(C)C)(C)C)NC(=O)C AS-8417 c1c(c(cc(c1Br)F)O)[N+](=O)[O-] AS-8418 CCOC(=O)c1c(ocn1)c2ccccc2 AS-8419 c1cc2ncc(n2cc1C=O)Br AS-8420 CC(=O)n1cc2ccc(cc2n1)I AS-8421 CC(=O)n1cc2c(cccc2n1)C(=O)OC AS-8422 CCc1ccc(cc1)S(=O)(=O)NC AS-8423 CC(=O)Nc1cc(ccc1O)C(=O)O AS-8424 CCc1nc2ccc(cc2o1)C(=O)OC AS-8425 CNS(=O)(=O)c1cccs1 AS-8426 COC(=O)c1ccc2c(c1)ocn2 AS-8427 CNS(=O)(=O)c1ccccc1C(F)(F)F AS-8428 COc1ccc(cc1)c2csc(=O)[nH]2 AS-8429 c1ccc2c(c1)nc(o2)NCCO AS-8430 c1cc(c(nc1)O)C#N AS-8431 Cc1cccc(c1)S(=O)(=O)NC AS-8432 CCNS(=O)(=O)c1ccc(cc1)Cl AS-8433 c1cc(c2cn[nH]c2c1)C(=O)NN AS-8434 CCOC(=O)c1ccc(c(c1)O)[N+](=O)[O-] AS-8435 CNc1c(cc(cn1)C(F)(F)F)Cl AS-8436 CC(=O)n1cc2cc(ccc2n1)C(=O)OC AS-8437 CCNc1c(cc(cn1)C(F)(F)F)Cl AS-8438 c1cc(cc(c1)[N+](=O)[O-])C(=O)NN AS-8439 CCOC(=O)c1c(c2cc(ccc2s1)Br)N AS-8440 Cn1c2cc(ccc2c(n1)N)C(F)(F)F AS-8441 CCOC(=O)c1c(nc(s1)C)O AS-8442 c1cc(ncc1C#N)NN AS-8443 CC(C)(C)OC(=O)n1c2ccc(cc2c(n1)N)[N+](=O)[O-] AS-8444 CCOC(=O)c1ccc(cc1)OCCCN2C(=O)c3ccccc3C2=O AS-8445 c1ccc(cc1)c2ncc(s2)CO AS-8446 CNS(=O)(=O)c1cccc(c1)[N+](=O)[O-] AS-8447 c1cc(c(cc1Cl)Cl)c2csc(=O)[nH]2 AS-8448 Cc1c(cnc(c1C#N)N)Br AS-8449 CCNc1ccc(cn1)C(F)(F)F AS-8450 c1cc2c(c(c1)[N+](=O)[O-])c(n[nH]2)Cl AS-8451 c1cnc(nc1c2nccs2)N AS-8452 Cc1cc(nc(n1)N)c2nccs2 AS-8453 CCOC(=O)c1ccc2c(c1)ocn2 AS-8454 CCOC(=O)c1ccc2c(c1)oc(n2)C AS-8455 CCc1nc2ccc(cc2o1)C(=O)OCC AS-8456 CCCc1nc2ccc(cc2o1)C(=O)OCC AS-8457 CCCCc1nc2ccc(cc2o1)C(=O)OCC AS-8458 CCCc1nc2ccc(cc2o1)C(=O)OC AS-8459 c1cc(cc(c1)[N+](=O)[O-])c2nnco2 AS-8460 c1cc(cc(c1)N)c2nnco2 AS-8461 CCCNc1c(cc(cn1)C(F)(F)F)Cl AS-8462 CC(=O)n1cc2ccc(cc2n1)F AS-8463 c1cc2cn[nH]c2cc1F AS-8464 COc1cccc(c1)c2cnco2 AS-8465 CCCCNc1c(cc(cn1)C(F)(F)F)Cl AS-8466 c1cc(nc(c1)NN)C(F)(F)F AS-8467 CN(c1ccc(cn1)[N+](=O)[O-])N AS-8468 c1ccn2c(c1)nc(c2Br)C(=O)NN AS-8469 CN(c1cccc(n1)C(F)(F)F)N AS-8470 CC1C(=O)Nc2c(cccn2)O1 AS-8471 CCc1nnc(o1)c2ccc(cc2)[N+](=O)[O-] AS-8472 CNC(=O)CC#N AS-8473 CCCCc1nc2ccccc2s1 AS-8474 CCCc1nc2ccccc2s1 AS-8475 CCc1nc2ccccc2s1 AS-8476 c1c(nc(c(n1)N)Cl)Br AS-8477 CCNc1c(cccn1)C#N AS-8478 Cc1nc(cs1)CC(=O)NN AS-8479 CCNS(=O)(=O)c1ccccc1Cl AS-8480 CNc1c(cc(cn1)Cl)C#N AS-8481 CNc1c(cc(cn1)Br)C#N AS-8482 c1(c([nH]c(n1)Br)Br)N AS-8483 CCCCc1nc2c(o1)cccn2 AS-8484 CCOC(=O)Cc1cn2cc(ccc2n1)Cl AS-8485 CCNc1c(cc(cn1)Br)C#N AS-8486 CNc1c(cc(cn1)C(F)(F)F)Br AS-8487 Cc1nc(cs1)CC(=O)O AS-8488 CCOC(=O)c1cccc(c1[N+](=O)[O-])C AS-8489 CCOC(=O)c1cccc(c1N)C AS-8490 CC1CNc2ccccc2O1 AS-8491 Cc1nc2cc(ccc2o1)CC(=O)OC AS-8492 CCc1nc2cc(ccc2o1)CC(=O)OC AS-8493 Cc1c(c(=O)n(c(c1Br)C)C)C#N AS-8494 CC(=O)n1cc2cc(ccc2n1)Cl AS-8495 COC(=O)c1cccc2c1[nH]nc2Br AS-8496 c1cc2c(c(c1)N)[nH]nc2Br AS-8497 c1cc2cn[nH]c2c(c1)C(=O)NN AS-8498 CC(=O)n1cc2cc(cc(c2n1)Br)Cl AS-8499 CCOC(=O)c1cn2cccc(c2n1)C(F)(F)F AS-8500 CCOC(=O)c1ccc(c(c1)C)[N+](=O)[O-] AS-8501 CCOC(=O)c1ccc(c(c1)C)N AS-8502 c1cc2cn[nH]c2cc1N AS-8503 Cc1ccc(cc1[N+](=O)[O-])C(=O)OC AS-8504 CC(=O)n1cc2ccc(cc2n1)C(=O)OC AS-8505 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])C AS-8506 CCOC(=O)c1cc(c(c(c1)Br)N)C AS-8507 c1c(cnc(c1C(=O)NN)N)Cl AS-8508 CCOC(=O)c1cc2cc(ccc2s1)C(F)(F)F AS-8509 CC1C(=O)Nc2cccc(c2O1)C(=O)OC AS-8510 CCOC(=O)c1ccc(c(c1)N)C AS-8511 CC1C(=O)Nc2ccc(cc2O1)[N+](=O)[O-] AS-8512 CC1C(=O)Nc2cccc(c2O1)C(=O)O AS-8513 CC1C(=O)Nc2ccc(cc2O1)N AS-8514 Cn1c2c(ccc(c2F)OC)c(n1)N AS-8515 CNC(=O)c1ccc2c(c1)nccn2 AS-8516 c1cc2cn[nH]c2cc1C(=O)NN AS-8517 c1c(cnc(c1Cl)O)C=O AS-8518 Cn1cc2c(n1)cccc2[N+](=O)[O-] AS-8519 CCOC(=O)c1cc2cccc(c2s1)Br AS-8520 c1cc2cc(sc2c(c1)Br)C(=O)NN AS-8521 c1c2c(cc(c1Cl)Cl)nc([nH]2)CCl AS-8522 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])O AS-8523 c1cc(c(c(c1)Br)CO)F AS-8524 Cc1cc(cc(c1N)Br)OC(F)(F)F AS-8525 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])N AS-8526 CC1C(=O)Nc2c(cccc2O1)[N+](=O)[O-] AS-8527 CCOC(=O)c1cc(c(nc1)N)Cl AS-8529 COC(=O)c1cc(c(nc1)O)Cl AS-8530 CC1C(=O)Nc2c(cccc2O1)N AS-8531 COc1ccc2c(c1)c(n[nH]2)Br AS-8532 c1cc(c2nc(cn2c1)C(=O)O)C(F)(F)F AS-8533 CCOC(=O)c1c(n2cccc(c2n1)C(F)(F)F)Br AS-8534 c1cc(c2nc(c(n2c1)Br)C(=O)O)C(F)(F)F AS-8535 CCOC(=O)c1c(n2cccc(c2n1)C(F)(F)F)Cl AS-8536 c1cc(c2nc(c(n2c1)Cl)C(=O)O)C(F)(F)F AS-8537 CCOc1c(cc(cn1)C(F)(F)F)Cl AS-8538 CSc1c(cc(cn1)C(F)(F)F)Cl AS-8539 CN(C)/C=C/1\Cc2ccccc2C1=O AS-8540 CCOC(=O)c1c(n2cc(cc(c2n1)Cl)C(F)(F)F)Br AS-8541 CCOC(=O)c1c(n2cc(cc(c2n1)Cl)C(F)(F)F)Cl AS-8542 CCC(C)Nc1c(cc(cn1)C(F)(F)F)Cl AS-8543 COC(=O)c1cc(c(nc1)O)I AS-8544 CCOC(=O)c1cnccn1 AS-8545 c1ccn2c(c1)ncc2Cl AS-8546 Cc1c(c(n(n1)C)C)C(=O)N AS-8547 c1cc(cc(c1)Cl)n2cn[nH]c2=O AS-8548 Cn1c(=O)n(cn1)c2cccc(c2)Cl AS-8549 COc1cccc2c1[nH]nc2 AS-8550 c1cc(ccc1C(=O)NN)Br AS-8551 Cc1nnc(o1)c2ccc(cc2)Br AS-8552 c1cc(ccc1c2nnco2)Br AS-8553 c1cc(ccc1C(=O)NN)C(=O)O AS-8554 COC(=O)c1ccc(cc1)CO AS-8555 CCOC(=O)c1cccc(c1C)[N+](=O)[O-] AS-8556 CC(C)(C)[Si](C)(C)OCc1ccc(cc1)C(=O)NN AS-8557 COC(=O)c1ccc(c(c1)Cl)F AS-8558 c1cc(c(cc1C(=O)NN)Cl)F AS-8559 Cc1nnc(o1)c2ccc(cc2)CO AS-8560 CCOC(=O)c1cccc(c1C)N AS-8561 Cc1c(nc2cc(ccc2n1)Br)C AS-8562 c1cc(ccc1/C(=N/O)/N)OC(F)(F)F AS-8563 c1cc(c(cc1c2cnco2)N)N3CCOCC3 AS-8564 COC(=O)c1cccc2c1oc(n2)CCl AS-8565 c1cc2nc(cn2cc1Br)C(=O)NN AS-8566 CCOC(=O)c1c(nc2n1cc(cc2)Br)C(F)(F)F AS-8567 c1cc2nc(c(n2cc1Br)C(=O)O)C(F)(F)F AS-8568 c1cc2nc(c(n2cc1Br)C(=O)NN)C(F)(F)F AS-8569 c1cc(ccc1CO)c2nnco2 AS-8570 c1cc2c(cc1Cl)cc(s2)C(=O)NN AS-8571 c1ccc(c(c1)C(=O)NN)F AS-8572 c1cc(ncc1C(=O)N)Cl AS-8573 c1cc(cc(c1)Br)C(=O)NN AS-8574 CC1(CCC(c2c1cc3c(c2)C(CCC3(C)C)(C)C)(C)C)C AS-8575 c1ccc2c(c1)N(CCO2)C(=O)NCCCl AS-8576 c1cc(cc(c1)OC(F)F)NC(=O)NCCCl AS-8577 c1c(cc(c(c1F)NC(=O)NCCCl)F)Br AS-8578 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])O AS-8579 Cc1ccc(c(c1)C)NC(=O)C AS-8580 c1cc2c(cc1C(=O)NN)nc[nH]2 AS-8581 c1cc(ccc1c2cnco2)I AS-8582 c1cc2c(cc1C(F)(F)F)cc(s2)C(=O)NN AS-8583 c1cc(c2ncc(n2c1)Br)N AS-8584 c1cc(cc(c1)N2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F AS-8585 CCOC(=O)c1ccc(c(c1)F)[N+](=O)[O-] AS-8586 CN(C)/C=C/C(=O)c1ccccc1[N+](=O)[O-] AS-8587 Cn1ccc2c1ccc(c2)C#N AS-8588 Cn1ccc2c1cccc2C#N AS-8589 CCOC(=O)c1cc2cccc(c2s1)Cl AS-8590 c1cc2cnc(nc2c(c1)Cl)N AS-8591 COc1ccc2c(c1)c(c[nH]2)CO AS-8592 Cn1ccc2c1cccc2C(=O)O AS-8593 COC(=O)Cc1ccc(c(c1)F)O AS-8594 c1cc(cc(c1)OC(F)F)N2CCNC2=O AS-8595 COC(=O)c1cc(nc(c1)Cl)N2CCCNCC2 AS-8596 Cc1cc(cc(c1N)Cl)C(=O)OC AS-8597 CC1C(=O)Nc2ccccc2S1 AS-8598 Cn1ccc2c1cccc2C(=O)OC AS-8599 CCOC(=O)c1cccc2c1ccn2C AS-8600 c1c(cc(c2c1cn[nH]2)C(=O)O)Br AS-8601 c1cc(nc(c1)Br)N2CCCCC2 AS-8602 c1cnc(cc1C(=O)N)N2CCCC2 AS-8603 CCCCCc1ccc(cc1)C(=O)N AS-8604 CCCCCc1ccc(cc1)C(=O)NC AS-8605 CCCCCc1ccc(cc1)C(=O)NCC AS-8606 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)N)N4CCCCCC4 AS-8607 Cc1ccc(cc1C)c2cnco2 AS-8608 CN(C)/C=C/1\Cc2ccc(cc2C1=O)F AS-8609 c1c(cc(c(c1C(F)(F)F)F)F)C(=O)O AS-8610 COC(=O)c1cc(c(c(c1)F)F)C(F)(F)F AS-8611 CNS(=O)(=O)c1ccc(cc1)OC(F)(F)F AS-8612 Cn1cc(c2c1ccc(c2)OC)CO AS-8613 c1ccc2c(c1)C(=O)N(C2=O)Cc3ccc4nccn4c3 AS-8614 COc1ccc2c(c1)nco2 AS-8615 CNS(=O)(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl AS-8616 CCNS(=O)(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl AS-8617 COC(=O)c1ccc2nc(cn2c1)c3ccnc(c3)Cl AS-8618 c1cc2c(cc1C=C(C#N)C#N)OCCO2 AS-8619 COc1cc(ccc1O)/C=C\2/c3ccccc3NC2=O AS-8620 COc1cccc(c1)/C=C\2/c3ccccc3NC2=O AS-8621 CNC(=O)Cc1ccc2ccccc2c1 AS-8622 CCOC(=O)c1cnc(nc1c2ccccc2)SC AS-8623 CSc1ncc(c(n1)c2ccccc2)C(=O)O AS-8624 c1cc2c(cc1Br)CCC2O AS-8625 c1cc2c(cc1C=O)OCCCO2 AS-8626 CCOC(=O)c1cnc(nc1c2ccccc2)c3ccncc3 AS-8627 c1ccc(cc1)c2c(cnc(n2)c3ccncc3)C(=O)O AS-8628 CN(C(=O)c1ccc(o1)Br)OC AS-8629 c1cc(nc(c1)Oc2ccc(cc2)Br)C(F)(F)F AS-8630 CCOC(COc1ccccc1Br)OCC AS-8631 CCOC(COc1cc(ccc1F)Br)OCC AS-8632 CCOC(COc1ccc(cc1F)Br)OCC AS-8633 c1cc(c2ccoc2c1F)Br AS-8634 CC(C)(C(=O)OC)Oc1ccc(cc1)Cl AS-8635 CC(C)(CO)Oc1ccc(cc1)Cl AS-8636 Cc1cccc(c1)Oc2ccc(cc2)O AS-8637 CC(=O)c1cc2cc(ccc2o1)Br AS-8638 CN(C)/C=C/C(=O)c1cc2cc(ccc2o1)Br AS-8639 c1cc2c(cc1Br)cc(o2)c3cc[nH]n3 AS-8640 CCOC(=O)c1cncnc1C(F)(F)F AS-8641 c1c(c(ncn1)C(F)(F)F)C(=O)O AS-8642 CN(C)/C=C/C(=O)c1ccc(cc1)C(=O)OC AS-8643 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)CNC AS-8644 CC(C)(C)c1ccc(cc1)Oc2ccccc2CNC AS-8645 Cc1ccccc1CNC AS-8646 CNCc1ccc(cc1)Oc2ccc(cc2)Br AS-8647 CNCc1c(cccc1Cl)Cl AS-8648 Cc1ccc(cc1)Oc2ccccc2CNC AS-8649 CNCc1ccc(cc1)Oc2cccc(c2)F AS-8650 CCOC(=O)c1cc(cs1)C AS-8651 CN(C)/C=C/C(=O)c1ccc2cc(ccc2c1)OC AS-8652 COc1ccc2cc(ccc2c1)c3cc[nH]n3 AS-8653 Cc1ccc(c(c1)C(=O)C)OCc2ccccc2 AS-8654 CCOC(=O)COc1ccc(cc1C(=O)C)C AS-8655 Cc1ccc(c(c1)C(=O)C)OCC(=O)O AS-8656 CNCc1ccccc1Oc2ccccc2F AS-8657 c1ccc(c(c1)c2ccc(cc2)CO)Cl AS-8658 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)N)Cl AS-8659 c1ccc(cc1)Oc2ccc(cc2C(F)(F)F)[N+](=O)[O-] AS-8660 c1ccc(cc1)Oc2ccc(cc2C(F)(F)F)N AS-8661 CNS(=O)(=O)c1ccc(cc1)Oc2ccc(cc2C(F)(F)F)[N+](=O)[O-] AS-8662 CN(C)S(=O)(=O)c1ccc(cc1)Oc2ccc(cc2C(F)(F)F)[N+](=O)[O-] AS-8663 CN(C)S(=O)(=O)c1ccc(cc1)Oc2ccc(cc2C(F)(F)F)N AS-8664 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)[N+](=O)[O-])S(=O)(=O)N AS-8665 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)N)S(=O)(=O)N AS-8666 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)[N+](=O)[O-])S(=O)(=O)N3CCCCC3 AS-8667 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)N)S(=O)(=O)N3CCCCC3 AS-8668 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)[N+](=O)[O-])S(=O)(=O)N3CCOCC3 AS-8669 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)N)S(=O)(=O)N3CCOCC3 AS-8670 c1ccc(cc1)C(c2c(c(c(c(c2F)F)F)F)F)O AS-8671 CC(=O)c1ccc(cc1)c2cccs2 AS-8672 c1ccn(c1)c2c(cc(cc2Cl)C(F)(F)F)Cl AS-8673 CCOC(=O)c1c(c(on1)C)I AS-8674 c1coc2c1cc(cc2Br)F AS-8675 c1cc(ccc1C=O)Oc2ccc(cn2)C(F)(F)F AS-8676 CC(=O)CCc1ccc(cc1)Oc2ccc(cc2)C#N AS-8677 c1cc(c(nc1)Oc2ccc(cc2)C=O)C(F)(F)F AS-8678 c1cc(c2c(c1F)cco2)Br AS-8679 CC(=O)CCc1ccc(cc1)OCC(=O)OC AS-8680 Cc1cc2ccoc2c(c1)Br AS-8681 c1cc(nc(c1)Oc2ccc(cc2)C=O)C(F)(F)F AS-8682 CCOC(=O)c1ccc(cc1)Oc2cccc(n2)C(F)(F)F AS-8683 c1ccc(cc1)Oc2ccc(cn2)C(F)(F)F AS-8684 c1ccc(cc1)Oc2ccc(cc2)CO AS-8685 c1ccc(cc1)Oc2ccc(cc2)CBr AS-8686 c1ccc(cc1)Oc2ccccc2CBr AS-8687 c1cc(nc(c1)N2CCCNCC2)C(F)(F)F AS-8688 c1cc(nc(c1)NCCN)C(F)(F)F AS-8689 c1c(cc(c(c1CO)O)Br)Cl AS-8690 c1cc(c(cc1/C=C/C(=O)O)[N+](=O)[O-])N2CCOCC2 AS-8691 CCOC(=O)c1ccc(cc1)OCC#N AS-8692 Cc1ccc(c(c1)Br)OCC#N AS-8693 c1ccc(cc1)COc2ccc(cc2)OCC#N AS-8694 c1cc(c(nc1)Sc2ccc(cc2)Cl)N AS-8695 CCOC(=O)c1cc[nH]n1 AS-8696 CCCCCCCCc1ccc(cc1)C(=O)OC AS-8697 CCCCCCCCc1ccc(cc1)CO AS-8698 c1cc(c(nc1)Oc2ccc(cc2)C=O)C#N AS-8699 c1cc(ccc1C=O)Oc2ccc(cc2)C#N AS-8700 Cc1c(ccc(n1)C(F)(F)F)CBr AS-8701 COc1cc(c(cc1OCc2ccccc2)[N+](=O)[O-])C=O AS-8702 Cc1cc(ccc1[N+](=O)[O-])Oc2ccccc2 AS-8703 Cc1cc(ccc1[N+](=O)[O-])N2CCOCC2 AS-8704 Cc1cc(ccc1[N+](=O)[O-])N2CCCC2 AS-8705 CCCOc1cccc(c1)C=O AS-8706 CCOC(=O)C1CCCN(C1)c2ccc(c(c2)C)[N+](=O)[O-] AS-8707 Cc1cc(ccc1[N+](=O)[O-])N2CCN(CC2)C AS-8708 Cc1cc(ccc1[N+](=O)[O-])n2ccnc2 AS-8709 c1cc(c(nc1)Oc2ccc(cc2)CO)C#N AS-8710 CCOC(=O)C1CCCN(C1)Cc2ccc(nc2C)C(F)(F)F AS-8711 c1c(c(cc(c1Br)Cl)Cl)C(=O)O AS-8712 COC(=O)c1cc(c(cc1Cl)Cl)Br AS-8713 c1c(c(cc(c1Br)Cl)Cl)C(=O)N AS-8714 c1ccc(c(c1)C=O)Oc2ccccc2F AS-8715 c1ccc(c(c1)C=O)Oc2ccc(cc2)Br AS-8716 c1cc(ccc1C=O)Oc2ccc(cc2)Br AS-8717 c1ccc(c(c1)CO)Oc2ccccc2F AS-8718 c1ccc(c(c1)CO)Oc2ccc(cc2)Br AS-8719 c1cc(ccc1CO)Oc2ccc(cc2)Br AS-8720 c1ccc(c(c1)CBr)Oc2ccc(cc2)F AS-8721 c1ccc(c(c1)CBr)Oc2ccccc2F AS-8722 c1cc(ccc1C=O)Oc2ccc(cc2)F AS-8723 c1cc(ccc1CO)Oc2ccc(cc2)F AS-8724 c1cc(ccc1CBr)Oc2ccc(cc2)F AS-8725 c1ccc(c(c1)Oc2ccc(cc2)C=O)F AS-8726 c1ccc(c(c1)Oc2ccc(cc2)CO)F AS-8727 Cc1ccc(cc1C)Oc2ccccc2C=O AS-8728 CC(C)(C)c1cccc(c1)Oc2ccccc2C=O AS-8729 Cc1ccc(cc1C)Oc2ccccc2CO AS-8730 CC(C)(C)c1cccc(c1)Oc2ccccc2CO AS-8731 CC(C)(C)c1ccc(cc1)Oc2ccccc2CBr AS-8732 Cc1ccc(cc1)Oc2ccccc2CBr AS-8733 Cc1ccc(cc1C)Oc2ccccc2CBr AS-8734 CC(C)(C)c1cccc(c1)Oc2ccccc2CBr AS-8735 c1cc(cc(c1)F)Oc2ccc(cc2)C=O AS-8736 Cc1ccc(cc1)Oc2ccc(cc2)C=O AS-8737 Cc1cccc(c1)Oc2ccc(cc2)C=O AS-8738 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)C=O AS-8739 c1cc(cc(c1)F)Oc2ccc(cc2)CO AS-8740 Cc1ccc(cc1)Oc2ccc(cc2)CO AS-8741 Cc1cccc(c1)Oc2ccc(cc2)CO AS-8742 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)CO AS-8743 c1cc(cc(c1)F)Oc2ccc(cc2)CBr AS-8744 Cc1ccc(cc1)Oc2ccc(cc2)CBr AS-8745 Cc1cccc(c1)Oc2ccc(cc2)CBr AS-8746 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2)CBr AS-8747 c1cc(ccc1CO)c2ccc(cc2)Cl AS-8748 COC(=O)c1ccc(cc1)c2ccccc2Cl AS-8749 c1ccc(c(c1)c2ccc(cc2)CBr)Cl AS-8750 COC(=O)c1ccc(cc1)c2ccc(cc2)F AS-8751 c1cc(ccc1CO)c2ccc(cc2)F AS-8752 COC(=O)c1ccc(cc1)c2ccccc2F AS-8753 c1ccc(c(c1)c2ccc(cc2)CO)F AS-8754 c1ccc(c(c1)c2ccc(cc2)CBr)F AS-8755 Cc1cc(ccc1[N+](=O)[O-])Oc2ccc(cc2)Br AS-8756 Cc1cc(ccc1N)Oc2ccc(cc2)Br AS-8757 Cc1cc(ccc1N)Oc2ccccc2 AS-8758 Cc1cc(ccc1N)N2CCOCC2 AS-8759 c1cc(ccc1Oc2ccc(cc2C(F)(F)F)N)Br AS-8760 c1cscc1c2csc(n2)N AS-8761 CCOC(=O)c1cscn1 AS-8762 Cc1nc(on1)c2ccsc2Br AS-8763 CCc1nc(on1)c2ccc(cc2)C(=O)OC AS-8764 CCc1nc(on1)c2ccc(cc2)C(=O)O AS-8765 CCc1nc(on1)c2ccc(cc2)C(=O)N AS-8766 Cc1cc(n(n1)c2ccccc2)NC(=O)CCl AS-8767 c1cc(cc(c1)C(F)(F)F)C(=O)NN AS-8768 COC(=O)c1cc(c(c(c1F)F)F)F AS-8769 c1c(c(c(c(c1F)F)F)F)C(=O)N AS-8770 c1ccc(cc1)OC(=O)CCl AS-8771 Cc1ccc(cc1)Oc2ccc(cn2)Br AS-8772 c1cc(cc(c1)Oc2ccc(cn2)Br)C=O AS-8773 c1cc(cc(c1)Oc2c(cccn2)C(F)(F)F)CO AS-8774 COc1cc(cc(c1[N+](=O)[O-])F)F AS-8775 CC(=O)c1cccc(c1)Oc2c(cccn2)C(F)(F)F AS-8776 CCOC(COc1ccc(cc1Br)C)OCC AS-8777 COc1cccc(c1C(=O)OC)OC AS-8778 COCOc1ccc(cc1Br)C=O AS-8779 COc1ccc(c(c1C(=O)O)OC)Cl AS-8780 CCOC(COc1ccc(cc1Br)F)OCC AS-8781 CNS(=O)(=O)c1ccc(n1c2c(cc(cc2Cl)C(F)(F)F)Cl)S(=O)(=O)NC AS-8782 CC(=O)Nc1ccc(cc1C(F)(F)F)Oc2ccccc2 AS-8783 Cn1cccc1C(=O)C(F)(F)F AS-8784 c1cnc2nccn2c1C(F)(F)F AS-8785 CC(=O)Nc1ccc(cc1)C(=O)CBr AS-8786 CC(C)(C)OC(=O)N1CCN(CC1)C(c2ccc(cc2)OC)C(=O)O AS-8787 c1ccc2c(c1)C(=O)N(C2=O)CCc3cnc(s3)N.Br AS-8788 Cn1c(ccc1C(=O)CCl)CC(=O)OC AS-8789 Cc1ccc(cc1C(=O)O)S(=O)(=O)N AS-8790 CCCCCCOc1ccc(cc1OC)C=O AS-8791 c1cc(ccc1N2CCCC2=O)S(=O)(=O)N AS-8792 Cc1c2c(cc(nc2n(n1)C)Oc3ccc(cc3)C=O)C(F)(F)F AS-8793 c1cc(ncc1C(F)(F)F)N2CCN(CC2)CCC(=O)O AS-8794 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2ccc(cc2)C=O AS-8795 c1cc(ccc1C#N)c2csc(n2)n3c(ccn3)C(F)(F)F AS-8796 c1cnc(nc1C(F)(F)F)N2CCCN(CC2)CCC(=O)O AS-8797 Cc1c(ccc(n1)C(F)(F)F)C=O AS-8798 CC(C)Oc1ccc(cc1F)Br AS-8799 c1cc(c(nc1)Cl)Oc2ccc(cn2)[N+](=O)[O-] AS-8800 CCOC(=O)c1ccc(cc1)OCCN2CCN(CC2)OC(=O)C(C)(C)C AS-8801 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2ccc(cc2)C(=O)O AS-8802 c1cc(c(cc1Br)OC(F)(F)F)NC(=S)N AS-8804 COC(=O)CCn1cc(c2c1cccc2)C=O AS-8805 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2cccnc2Cl AS-8806 Cn1cc(c(n1)C#N)Br AS-8807 c1cc2c(cc1S(=O)(=O)N)CCC2 AS-8808 c1cnn(c1)c2nccc(n2)C(F)(F)F AS-8809 Cn1cc(c(n1)/C=N/O)Br AS-8810 COc1ccc(cc1F)S(=O)(=O)C AS-8811 c1cc(ccc1C#N)C2(OCCO2)CBr AS-8812 Cc1c2ccccc2nc(c1C#N)Cl AS-8813 CC(=O)c1ccc(cc1)N2CC(CC2=O)C(=O)O AS-8814 CC(C)(C)OC(=O)N1CCN(CC1)CCn2cc(cn2)Br AS-8815 Cc1c(ccc(n1)C(F)(F)F)N AS-8816 Cn1c(ccc1c2csc(n2)N)CC(=O)OC AS-8817 CS(=O)(=O)OC1CCOCC1 AS-8818 CCOC(=O)c1cc(c(nc1C(F)(F)F)C)C#N AS-8819 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2ccccc2C=O AS-8820 Cc1nc(cs1)c2ccc(n2C)CC(=O)OC AS-8821 Cc1nc(cs1)c2ccc(n2C)CC(=O)O AS-8822 Cc1c(ccc(n1)C(F)(F)F)C=C(C#N)C#N AS-8823 c1cc(c(c(c1)Cl)CN2CCN(CC2)CCO)F AS-8824 c1cc(ccc1Cn2cc(cn2)Br)F AS-8825 Cc1c(ccc(n1)C(F)(F)F)/C=N/O AS-8826 CC(=O)N1CCN(CC1)c2ccc(cc2C(F)(F)F)N AS-8827 C1CC(=O)N(C1=O)CC#N AS-8828 Cc1c(ccc(n1)C(F)(F)F)NC(=O)NCc2ccccc2 AS-8829 Cc1c(ccc(n1)C(F)(F)F)C(=O)NN AS-8830 c1cc(c(cc1N2CCOCC2)C(F)(F)F)N AS-8831 c1cc(c(cc1N2CCCCC2)C(F)(F)F)N AS-8832 c1cc(c(cc1N2CCCC2)C(F)(F)F)N AS-8833 CN1CCN(CC1)c2ccc(c(c2)C(F)(F)F)N AS-8834 c1cc(ccc1N)n2cc(cn2)Br AS-8835 c1cc(ccc1C=O)n2cc(cn2)Br AS-8836 c1cc(ccc1CO)n2cc(cn2)Br AS-8837 CC(=O)c1ccc(cc1)n2cc(cn2)Br AS-8838 c1cc(ccc1C(=O)CBr)n2cc(cn2)Br AS-8839 CC(C)(C)OC(=O)N1CCCN(CC1)CCC(=O)O AS-8840 CCOC(=O)C1CCN(CC1)c2cc(c3c(nn(c3n2)C)C)C(F)(F)F AS-8841 CC(C)(C)OC(=O)N1CCCN(CC1)CCC(=O)OC AS-8842 c1cc(ccc1/C=C/C(=O)O)n2cc(cn2)Br AS-8843 Cc1ccc(cc1C(=O)O)S(=O)(=O)N(C)C AS-8844 CC(C)(C)OC(=O)N1CCc2c(sc(c2C(=O)O)n3cccc3)C1 AS-8845 COC(=O)c1cc2c(s1)CCCC2 AS-8846 Cc1c(ccc(n1)C(F)(F)F)C(=O)NC AS-8847 Cc1cccc(c1)c2nc(on2)C(C)(C)CCl AS-8848 CNc1nccc(n1)C(F)(F)F AS-8849 c1ccn(c1)c2ccsc2C=O AS-8850 Cn1c2c(c(cc(=O)[nH]2)C(F)(F)F)c(=O)n(c1=O)C AS-8851 c1c2c(sc1C=O)CCCC2 AS-8852 Cc1c(sc(n1)C)S(=O)(=O)N AS-8853 c1c(c(nc(n1)N2CCOCC2)C(F)(F)F)C(=O)O AS-8854 Cc1c(ccc(n1)C(F)(F)F)NC(=O)CCl AS-8855 CC(C)(C)c1cc(c(s1)C(=O)O)n2cccc2 AS-8856 CC(C)(C)OC(=O)N1CCC(CC1)(CNC)O AS-8857 CCN(CC)c1ccc2cc(c(=O)oc2c1)C(=O)O AS-8858 COC(=O)c1c2c(sc1N)CN(CC2)c3nccc(n3)C(F)(F)F AS-8859 CCOC(=O)c1ccc(cc1)Oc2nccc(n2)C(F)(F)F AS-8860 C1COCCN1/C=C/C(=O)C(F)(F)F AS-8861 CN1CCN(CC1)/C=C/C(=O)C(F)(F)F AS-8862 c1csc2c1c(ncn2)N3CCC(=O)CC3 AS-8863 Cc1c(c(no1)c2ccccc2)C(=O)CBr AS-8864 c1cc(ccc1N2CCN(CC2)CC(COc3ccc(cc3)F)O)[N+](=O)[O-] AS-8865 c1csc(c1Br)C(=O)NN AS-8866 c1cnc(nc1C(F)(F)F)N2CCN(CC2)CCO AS-8867 CCOC(=O)C1CCN(CC1)c2nccc(n2)C(F)(F)F AS-8868 c1c2c(sc1C(=O)NN)CCCC2 AS-8869 CC(C)(C)OC(=O)N1CCc2c(sc3c2c(=O)[nH]cn3)C1 AS-8870 c1cc(ccc1C(=O)C(Br)Br)N2CCOCC2 AS-8871 c1cc(ccc1c2csc(n2)N)N3CCOCC3 AS-8872 Cc1c(c2c(cc1Br)nsn2)C AS-8873 CCOC(=O)Cc1c(c(sc1C(=O)OCC)N)C(=O)OCC AS-8874 c1ccc(cc1)COC(=O)N2CCc3c(c[nH]n3)C2 AS-8875 c1cc(sc1)c2csc3c2c(ncn3)O AS-8876 c1cc(sc1)c2csc3c2c(ncn3)Cl AS-8877 c1cc(ccc1C=C(C#N)C#N)F AS-8878 c1cc(c(cc1Br)OC(F)(F)F)NC(=S)NCCO AS-8879 c1cc(c(cc1Br)OC(F)(F)F)NC2=NCCS2 AS-8880 c1c2c(sc1C=O)CCC2 AS-8881 CCOC(=O)c1c(csc1N)c2ccc(cc2)F AS-8882 CCc1c(c([nH]c1COC(=O)C)C(=O)OCC)C AS-8883 Cc1c(ccc(n1)C(F)(F)F)NC(=O)/C=C/C(=O)O AS-8884 Cc1ccc(s1)S(=O)(=O)N AS-8885 c1cc(sc1)c2csc3c2c(ncn3)NN AS-8886 Cn1cc(cn1)N AS-8887 CCc1c(c([nH]c1COC(=O)C)C(=O)O)C AS-8888 CC(=O)N1CCc2c1ccc(c2)S(=O)(=O)NCCNC(=O)OC(C)(C)C AS-8889 CC(C)(C)OC(=O)NCCNC(=O)c1cccc(c1)Br AS-8890 CC(C)(C)OC(=O)NCCNC(=O)c1ccccc1Br AS-8891 CC(C)(C)OC(=O)NCCNC(=O)c1ccc(cc1)Br AS-8892 c1ccc(cc1)COC(=O)N2CCC(CC2)NC(=O)N AS-8893 CNC(=O)c1ccc2c(c1)nnn2C AS-8894 c1cc2c(cc1N)nc([nH]2)C(F)(F)F AS-8895 COC(=O)CCn1cc(c2c1cccc2)CN3CCOCC3 AS-8896 CC(C)(C)OC(=O)NCCNc1ccc(cc1[N+](=O)[O-])C(=O)OC AS-8897 c1ccc2c(c1)c(cn2CCC(=O)O)CN3CCOCC3 AS-8898 c1csc2c1CCCC2 AS-8899 CC(C)(C)OC(=O)NCCNc1ccc(cc1N)C(=O)OC AS-8900 c1ccc2c(c1)C(=O)N(C2=O)CCCn3cc(cn3)[N+](=O)[O-] AS-8901 c1c(cc(c(c1F)C#N)F)N2CCOCC2 AS-8902 CC(C)(C)OC(=O)NCCn1cnc2c1ccc(c2)C(=O)OC AS-8903 CC(C)(C)OC(=O)NCCn1cnc2c1ccc(c2)C(=O)O AS-8904 CN1CCN(CC1)S(=O)(=O)c2ccc(c(c2)C(F)(F)F)Br AS-8905 COC(=O)c1cc2cc(cc(c2oc1=O)Br)Cl AS-8906 Cc1c(ccc(n1)C(F)(F)F)/C=C/C(=O)O AS-8907 CN(c1nccc(n1)C(F)(F)F)N AS-8908 C1CCC(C1)(CC(=O)O)C(=O)O AS-8909 CC(C)(C)c1cc(cc(c1O)Br)Br AS-8910 c1ccc(cc1)N2C(=O)CC3(C2=O)CCCC3 AS-8911 CCN(CC)C(=S)Nc1ccc(cc1)N2CCOCC2 AS-8912 c1c2c(sc1Br)CCCC2 AS-8913 c1csc(c1Br)c2nnco2 AS-8914 c1cc(ccc1N2C(=O)CC3(C2=O)CCCC3)Br AS-8915 c1csc2c1c3nncn3cn2 AS-8916 CCOC(=O)CNC(=O)OC(C)(C)C AS-8917 CC(C)(C)OC(=O)N1CCC(CC1)OS(=O)(=O)C AS-8918 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NN AS-8919 c1c(c(n[nH]1)C=O)Br AS-8920 c1cc(ccc1c2cnco2)F AS-8921 Cc1cccc2c1nc(cc2Cl)C(F)(F)F AS-8922 CCOC(=O)C1CCN(CC1)Cc2c(cn(n2)C)Br AS-8923 c1cc(c(cc1CN2CCC(=O)CC2)Cl)Cl AS-8924 Cc1c(sc(n1)C2CCN(CC2)C(=O)OC(C)(C)C)C(=O)O AS-8925 Cc1cc(nc(c1C#N)c2cccs2)C AS-8926 CCOC(=O)c1csc(n1)c2cccnc2 AS-8927 COc1ccccc1c2nc(no2)CCl AS-8928 c1c(c(sc1S(=O)(=O)N)Br)Br AS-8929 Cc1c(ccc(n1)C(F)(F)F)S(=O)(=O)N AS-8930 c1ccc2c(c1)C(=O)N(C2=O)CC3CCCCO3 AS-8931 C1CCOC(C1)CN AS-8932 C1CCOC(C1)CN.Cl AS-8933 c1cc(ccc1OCC(CN2CCOCC2)O)F AS-8934 Cc1c(c(nc(n1)c2ccncc2)Cl)Cl AS-8935 Cc1csc2c1ncnc2O AS-8936 c1ccn2cc(nc2c1)c3cccs3 AS-8937 c1cc(c(cc1S(=O)(=O)N2CCOCC2)C(=O)O)N3CCOCC3 AS-8938 Cc1nc2ccc(cc2s1)S(=O)(=O)N AS-8939 Cn1c(nnc1SCC(COc2ccc(cc2)F)O)C(F)(F)F AS-8940 CC(C)(C)OC(=O)N1CCC(CC1)(CSc2nnc(n2C)C(F)(F)F)O AS-8941 c1cc2c(cc1C(=O)NN)non2 AS-8942 c1ccc(c(c1)CSCCN2CC(CC2=O)C(=O)O)Cl AS-8943 CC(C)(C)OC(=O)N1CCC(CC1)(CNCC2CCCO2)O AS-8944 CCOC(=O)c1c2c(sc1N)COCC2 AS-8945 c1[nH]c(=O)c2c3c(sc2n1)COCC3 AS-8946 c1nc2c(c3c(s2)COCC3)c(n1)Cl AS-8947 CN(C)/C=C/1\COCCC1=O AS-8948 CCOC(=O)c1c(c2cc(ccc2o1)Cl)N AS-8949 CCOC(=O)C1CCN(CC1)C2CCN(C2)C(=O)OC(C)(C)C AS-8950 c1cc2c(cc1Cl)c3c(o2)c(=O)[nH]cn3 AS-8951 c1cc2c(cc1Cl)c3c(o2)c(ncn3)Cl AS-8952 CC(=O)c1c(ccs1)OC AS-8953 CC(C)(C)OC(=O)N1CCN(CC1)CC(COc2ccc(cc2)F)O AS-8954 CC(C)(C)OC(=O)N1CCC(C1)N2CCC(CC2)C(=O)O AS-8955 C1CN(CCN1CCO)c2nnc(s2)C(F)(F)F AS-8956 COc1ccsc1/C=N/O AS-8957 CS(=O)(=O)c1ccc(c(c1)F)NN AS-8958 COc1ccsc1C#N AS-8959 c1c2c(sc1c3nnc(s3)N)CCCC2 AS-8960 CC(C)(C)Nc1c2cnn(c2ncn1)C AS-8961 c1c2c(sc1S(=O)(=O)N)CCCC2 AS-8962 Cc1ccc(s1)NC(=O)OC(C)(C)C AS-8963 COc1ccsc1c2cnco2 AS-8964 CC(C)(C)c1ccc(cc1)c2nc(=S)[nH]n2c3ccccc3 AS-8965 Cc1nc(cs1)c2ccc(cc2)N3CC(CC3=O)C(=O)O AS-8966 Cc1c(scn1)S(=O)(=O)N2CCC(CC2)C(=O)O AS-8967 CC(C)(C)c1csc(n1)C=O AS-8968 c1c(nc(nc1Cl)I)Cl AS-8969 c1cc2c3c(c(=O)[nH]cn3)sc2nc1 AS-8970 c1ccn(c1)c2ccc3c(c2)ccs3 AS-8971 c1cc(c(cc1Br)OC(F)(F)F)NC(=S)Nc2cnn(c2)C3CCOCC3 AS-8972 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)C(=O)NN AS-8973 Cc1c(scn1)S(=O)(=O)NC AS-8974 c1c2c(sc1C(=O)O)CCOC2 AS-8975 CC(C)(C)c1cc2c(s1)c(=O)[nH]cn2 AS-8976 CC(C)(C)c1cn2cc(ccc2n1)Br AS-8977 c1c2c([nH]n1)CCOC2 AS-8978 CCOC(=O)Cn1cc(cn1)[N+](=O)[O-] AS-8979 CCOC(=O)c1c(nc2ccccc2n1)N3CCOCC3 AS-8980 c1ccc2cc(ccc2c1)Cn3cc(cn3)N AS-8981 c1cc(sc1)c2cc(c(c(n2)Cl)C#N)C(F)(F)F AS-8982 c1ccc2c(c1)C(=O)N(C2=O)CCc3cn4cc(ccc4n3)F.Br AS-8983 Cc1c(ccc(n1)C(F)(F)F)c2ccn[nH]2 AS-8984 c1c(cc(c2c1COCO2)c3cnco3)F AS-8985 CCOC(=O)c1c(nc2ccccc2n1)N3CCCN(CC3)C(=O)OC(C)(C)C AS-8986 Cc1cc(n2c(n1)cc(n2)c3cccs3)C AS-8987 Cc1c(ccc(n1)C(F)(F)F)c2ccnc(n2)S AS-8988 Cc1c(ccc(n1)C(F)(F)F)C(=O)CBr.Br AS-8989 Cc1c(ccc(n1)C(F)(F)F)c2csc(n2)N AS-8990 CCOC(=O)c1ccc(nc1c2ccccc2)C(F)(F)F AS-8991 COC(=O)c1c[nH]cc1c2ccccc2 AS-8992 CC(C)(C)c1cn2cc(ccc2n1)C(=O)OC AS-8993 CC(C)(C)c1cn2cc(ccc2n1)C(=O)O AS-8994 c1c(cn(n1)CCN2CCNCC2)[N+](=O)[O-] AS-8995 c1c(cn(n1)C2=C(CCCC2)C=O)[N+](=O)[O-] AS-8996 C1COCCC1C(=O)NN AS-8997 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cnn(c2)C3CCOCC3 AS-8998 Cc1cc(n(c(=O)c1C#N)Cc2ccccc2)C AS-8999 c1cc(oc1)C(=O)Nc2ccc3c(c2)CCO3 AS-9000 c1ccc2c(c1)c(=O)n(c(n2)S)c3cccnc3 AS-9001 c1cc(cnc1)n2ccnc2S AS-9002 Cc1cc(cc(c1NC(=S)NN)Cl)Cl AS-9003 c1cc(ccc1N)S(=O)(=O)Nc2cnn(c2)C3CCOCC3 AS-9004 c1cc(cnc1)NC(=S)NNC(=O)C2CCOCC2 AS-9005 c1cc(cnc1)n2c(nnc2S)C3CCOCC3 AS-9006 CC(C)c1ccc(cc1)NC(=S)NNC(=O)C2CCOCC2 AS-9007 COC(=O)c1c(nc(s1)Nc2cccnc2)N AS-9008 CC(C)c1ccc(cc1)n2c(nnc2S)C3CCOCC3 AS-9009 CCOC(=O)C1CCN(CC1)c2c3c(c(sc3ncn2)c4ccccc4)C AS-9010 CC(C)(C)C(=O)c1c(nc(s1)Nc2cccnc2)N AS-9011 Cc1c(c(no1)c2ccccc2)NC(=O)NCC3CCCO3 AS-9012 c1nnc(o1)C2CCOCC2 AS-9013 c1c(cn(n1)CC2CCCO2)N AS-9014 Cc1c(ccc(n1)C(F)(F)F)c2nnco2 AS-9015 Cc1cccc(c1Nc2nc(c(s2)C(=O)OC)N)C(C)C AS-9016 c1ccc(cc1)c2cc(c3c(csc3n2)N)C(F)(F)F AS-9017 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)n4cc(cn4)Br AS-9018 c1cc(c(nc1)N2CCNCC2)[N+](=O)[O-] AS-9019 c1cc(ccc1Oc2ccc(cn2)N)Cl AS-9020 Cc1ccc(s1)S(=O)(=O)NC AS-9021 Cc1c2c(ncnc2sc1c3ccccc3)N4CCC(CC4)C(=O)O AS-9022 c1cc(c(nc1)N2CCN(CC2)CC(COc3ccc(cc3)F)O)[N+](=O)[O-] AS-9023 c1ccc(cc1)C2CC(=NN2c3ccc(cc3)Cl)C(=O)O AS-9024 c1ccc(cc1)C2CC(=NN2c3ccc(cc3)Cl)C(=O)NN AS-9025 c1cc(c(nc1)N2CCN(CC2)C3CCOCC3)N AS-9026 c1cc2c(cc1C(=O)CBr)CCO2 AS-9027 Cc1c(c(n(n1)C)N2CCOCC2)[N+](=O)[O-] AS-9028 Cc1c(c(n(n1)C)NN)[N+](=O)[O-] AS-9029 c1c(c2c(c(c1Br)Cl)c(ncn2)O)Br AS-9030 C1C=NN(C1(C(F)(F)F)O)C(=S)N AS-9031 c1ccc2c(c1)C(=O)N(C2=O)CCc3cn4cc(ccc4n3)F AS-9032 c1cc2nc(cn2cc1F)CCN AS-9033 Cc1c(c(n(n1)C)N2CCOCC2)N AS-9034 Cc1nc(cs1)c2ccc(cc2)S(=O)(=O)N AS-9035 c1csc(c1Cl)C(=O)NN AS-9036 CC1CC1C(=O)NN AS-9037 Cc1c(ccc(n1)C(F)(F)F)NC(=O)Nc2cccc(c2)Cl AS-9038 c1c(cnc(c1S(=O)(=O)N2CCOCC2)N)Cl AS-9039 COC(=O)CCN1CCN(CC1)c2c(cccn2)[N+](=O)[O-] AS-9040 Cc1c(ccc(n1)C(F)(F)F)C(=O)N(C(C)C)C(C)C AS-9041 c1cc2c(cc1C=O)non2 AS-9042 c1c2c(sc1C(=O)N)CCCC2 AS-9043 CC(C)N(C(C)C)C(=O)c1c(ccs1)Cl AS-9044 CCOC(=O)c1c(c2cc(ccc2o1)Cl)n3cccc3 AS-9045 Cc1c(ccc(n1)C(F)(F)F)NC(=O)Nc2cccc(c2)N3CCCC3 AS-9046 Cc1c(ccc(n1)C(F)(F)F)NC(=O)NCc2ccc(c(c2)F)OC AS-9047 c1c2c(sc1C(=O)CC#N)CCCC2 AS-9048 CC(C)N(C(C)C)C(=O)c1cc2c(s1)CCCC2 AS-9049 c1cc(ccc1CI)[N+](=O)[O-] AS-9050 c1cc(c(cc1CI)Cl)Cl AS-9051 c1cc2c(cc1S(=O)(=O)NCC3CCCO3)scn2 AS-9052 c1cc(c(cc1S(=O)(=O)NCC2CCCO2)F)Br AS-9053 Cc1ccc(s1)S(=O)(=O)NCC2CCCO2 AS-9054 c1c2c(sc1S(=O)(=O)N3CCOCC3)CCCC2 AS-9055 Cc1c(scn1)S(=O)(=O)N2CCOCC2 AS-9056 CC(=O)N1CCc2c1ccc(c2)S(=O)(=O)N3CCOCC3 AS-9057 COc1ccc(cc1)n2cn[nH]c2=O AS-9058 CC(=O)CCc1cccc(c1)Br AS-9059 c1cc(c(cc1Cl)CC#N)[N+](=O)[O-] AS-9060 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)N AS-9061 c1c(c(c(c(c1Br)Cl)C(=O)O)N)Br AS-9062 c1cc(ccc1C23CC4CC(C2)CC(C4)C3)OCC(CN5CCCCC5)O.Cl AS-9063 c1cc(c2c(c1)OCCCO2)CO AS-9064 c1c(cc(cc1C(F)(F)F)NCCC2CCCCN2)C(F)(F)F AS-9065 Cc1nc(cs1)c2cccc(c2)C#N AS-9066 c1ccnc(c1)Oc2cccc(c2)[N+](=O)[O-] AS-9067 c1cc(oc1CO)c2cc(cc(c2)C(F)(F)F)C(F)(F)F AS-9068 c1cc(oc1)c2cc(c(c(n2)O)C#N)c3cccs3 AS-9069 CCOC(=O)C1=C(N2CCN=C2S1)C.Cl AS-9070 CCO/C=C(\C#N)/S(=O)(=O)c1ccc2ccccc2c1 AS-9071 Cc1c(c(n(n1)Cc2nnc(o2)S)C)Br AS-9072 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)CC(=S)N AS-9073 CC(C)(C)OC(=O)NCc1nnc(n1C2CC2)S AS-9074 CCOC(=O)c1cnc(s1)NCc2ccccc2 AS-9075 CCC12CC3CC(C1)CC(C3)(C2)Br AS-9076 CC(=O)c1c(cc(s1)c2ccc(cc2)C(C)(C)C)N AS-9077 CC1(Cc2c(c(sc2Cl)SC)C(=O)C1)C AS-9078 CC(C)(C)OC(=O)N1CCCC(C1)Oc2ccc(cc2)[N+](=O)[O-] AS-9080 CC(C(=O)O)Sc1c(ccc(n1)OC)[N+](=O)[O-] AS-9081 Cc1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)/C=C/C(=O)O AS-9082 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=C/C(=O)O AS-9083 CCOC(=O)c1c(n(c(c1C=O)C)C2CC2)C AS-9084 CCCOc1ccc(cc1)/C(=N/O)/N AS-9085 Cc1c(cc(n1c2ccc(cc2)SC)c3ccccc3)C(=O)O AS-9086 C/C(=C(\C(=O)c1cc(nc(c1)Cl)Cl)/C(=O)OC)/NC AS-9087 CSc1nn(c(=S)s1)CO AS-9088 COc1ccc(cc1)n2c(nnc2S)c3ccc(cc3)OC(F)(F)F AS-9089 CC(=O)c1cc(no1)c2ccc(c(c2)Cl)Cl AS-9090 c1cc(oc1)Cn2c(nnc2S)c3ccc(cc3Cl)Cl AS-9091 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)S AS-9092 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3S)c4ccco4 AS-9093 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(o3)S AS-9094 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)c3nnc(n3C)S AS-9095 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2C=O)[N+](=O)[O-] AS-9096 c1cc(ccc1Sc2ccc(cc2/C=C\C(=O)O)[N+](=O)[O-])Cl AS-9097 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])/C=C/C(=O)O AS-9098 c1cc(c(nc1)Sc2ccc(cc2)Cl)[N+](=O)[O-] AS-9099 Cc1cc(c2ccccc2n1)Sc3nnc(s3)N AS-9100 c1cc(ccc1Sc2ccc(cc2C#N)[N+](=O)[O-])Cl AS-9101 CCOC(=O)c1c(c(c(=N)n(n1)c2ccc(cc2)C)C#N)C AS-9102 c1ccc(cc1)COc2cccc(c2OCc3ccccc3)CCC#N AS-9103 CC(C)(C)OC(=O)N1CCN(CC1)Cc2cccc(c2)[N+](=O)[O-] AS-9104 c1cc(c(c(c1[N+](=O)[O-])O)C#N)O AS-9105 CCSc1c(cccn1)C(=O)NC(CCSC)C(=O)O AS-9106 Cc1cc(cc(c1Cl)C)Oc2c(cccn2)[N+](=O)[O-] AS-9107 Cc1c(c(c(c(c1C)C)C(=O)Cc2ccccc2)C)C AS-9108 C#CCOc1c(cccc1Cl)Cl AS-9109 CSCCC(C(=O)O)NC(=O)c1cccnc1SC AS-9110 c1cc(cc(c1)OCC2CO2)C=O AS-9111 c1cc(c(nc1)Oc2cc(cnc2)Cl)[N+](=O)[O-] AS-9112 Cc1ccc(cc1)Sc2c(cccn2)C(=O)N AS-9113 CCOC(=O)/C=C/c1ccc(c(c1Cl)OC)OC AS-9114 CCCCCCCCCCc1ccc(cc1)N.Cl AS-9115 CCOC(=O)c1cnc2cc(nn2c1C)c3cccs3 AS-9116 CCOC(=O)c1c-2c(c(s1)SC)S(=O)(=O)N(c3c2cccc3)C AS-9117 CCOC(=O)c1c2c(c(s1)SCC=C)C(=O)CCC2 AS-9118 c1cc(ccc1Sc2ccc(s2)S(=O)(=O)N)Cl AS-9119 c1cc(sc1)Sc2ccc(s2)S(=O)(=O)N AS-9120 CSc1c(cn(n1)c2ccccc2)C#N AS-9121 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)C(=S)N AS-9122 CC(C)(C)OC(=O)NCc1nnc(n1CC=C)S AS-9123 CCOC(=O)c1c([nH]c(=O)[nH]c1=S)C AS-9124 c1cc(ccc1OCC2CO2)F AS-9125 CC(C)c1nc(nc(n1)SC)N AS-9126 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C=O AS-9127 Cc1nc(cn1CC(=O)c2ccc(cc2)OC)[N+](=O)[O-] AS-9128 COC(=O)CC12CC3CC(C1)CC(C3)C2 AS-9129 c1ccnc(c1)c2nc(nc(n2)NN)N AS-9130 Cc1ccc(cc1)COc2ccc(cc2)CC#N AS-9131 C#CCc1ccc(cc1)OCc2ccc(c(c2)Cl)Cl AS-9132 Cc1nc(c(n1CCC#N)Br)[N+](=O)[O-] AS-9133 CN1CCN(CC1)Cc2cccc(c2)[N+](=O)[O-] AS-9134 c1cc2c(cc1Cl)C(=C(CS2)C=O)Cl AS-9135 c1cc(n(c1)c2ccc(cc2)I)C=O AS-9136 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)S AS-9137 c1ccc(cc1)c2c(ssc2=S)S AS-9138 c1cc(c(cc1C(F)(F)F)NC(=S)N)Cl AS-9139 CCOC(=O)C(=O)c1ccc(cc1)C AS-9140 c1ccc(cc1)CN2CCN(CC2)c3c(cccn3)[N+](=O)[O-] AS-9141 CC(=O)c1ccc2c(c1)OCCCO2 AS-9142 CCCCCCCCc1ccc(cc1)C(=O)O AS-9143 CCCCCCCCc1ccc(cc1)C(=O)CCC(=O)O AS-9144 COc1ccc(c(c1OC)Cl)CO AS-9145 CCOC(=O)c1cnc(nc1N)S AS-9146 c1cc2cccc(c2c(c1)SCC(=O)O)Cl AS-9147 CCOc1cc(c(cc1Cl)OCC)[N+](=O)[O-] AS-9148 Cc1cc(no1)n2cnc(n2)CC(=O)C AS-9150 c1ccc-2c(c1)Cc3c2ccc(c3)c4csc(n4)N AS-9151 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)N AS-9152 CCSc1c2c(c(s1)C(=O)OC)CC(CC2=O)(C)C AS-9153 CCOC(=O)c1c2c(c(s1)SC(C)C)C(=O)CC(C2)(C)C AS-9154 CCCCSc1c2c(c(s1)C(=O)OCC)CCCC2=O AS-9155 c1c(cc(c2c1nc(cc2O)C(F)(F)F)Cl)Cl AS-9156 c1c(cc(c2c1nc(cc2Cl)C(F)(F)F)Cl)Cl AS-9157 COC(=O)CSc1cc(nc2c1cccc2)C(F)(F)F AS-9158 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)C#N AS-9159 Cc1ccc2c(c1[N+](=O)[O-])c(cc(n2)C(F)(F)F)Cl AS-9160 Cc1cccc2c1nc(cc2O)C(F)(F)F AS-9161 Cc1[nH]c(c(n1)I)I AS-9162 CCOc1cccc(c1C#N)OCC(F)(F)F AS-9163 CCOC(=O)c1cc(c(c(c1)I)N)I AS-9164 C1CCC(CC1)c2c(c(=O)[nH]c(=S)[nH]2)C#N AS-9165 CSc1ccc(s1)C#N AS-9166 c1cc(c(c(c1[N+](=O)[O-])C#N)Cl)Cl AS-9167 c1cc(ccc1c2csc(n2)CC#N)[N+](=O)[O-] AS-9168 c1cc(ccc1C2SCCS2)O AS-9169 c1c(cc(cc1Cl)Cl)OCC#N AS-9170 c1cc(sc1)/C=N/NC(=S)N AS-9171 CCOC(=O)c1cc(nn1Cc2c(cc(cc2C)C)C)C(C)(C)C AS-9172 CCCCc1ccc(c(c1)C)I AS-9173 c1cc(c(cc1/C=C/C(=O)O)[N+](=O)[O-])N2CCCC2 AS-9174 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=C/C(=O)O AS-9175 COc1ccc(c(c1C(=O)N)OC)Cl AS-9176 CC(=O)C12CC3CC(C1)CC(C3)C2 AS-9177 C1C(C1(Cl)Cl)C(=O)N AS-9178 C1C=C(CS1(=O)=O)Cl AS-9179 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)O)C)C AS-9180 CC1N=C(N2N1C(=NC2C)S)S AS-9181 CCOC(=O)C(=CNc1cc(nn1C)C)C(=O)OCC AS-9182 c1ccc(cc1)CN2CCC(CC2)OCCC(=O)N AS-9183 CCOC(=O)c1cc(ccc1Cl)[N+](=O)[O-] AS-9184 c1cc(c(cc1Br)OC(F)(F)F)N=C=S AS-9185 CCCCOC1=CC(=O)CCC1 AS-9186 CC(=O)Nc1ccc(cc1)C=O AS-9187 c1ccc2c(c1)nc(c(=O)n2c3ccc(cc3)Cl)O AS-9188 c1ccc2c(c1)[nH]c(n2)CO AS-9189 COC(=O)CSCCC(=S)N AS-9190 CC(C)c1ccc(c(c1)Br)N=C=S AS-9191 CC(=O)Nc1ccc(cc1F)Br AS-9192 CCCCC#Cc1ccc(cc1)C=O AS-9193 Cc1ccc(n1c2cc(c(cc2Cl)[N+](=O)[O-])Cl)C AS-9194 CCOC(=O)CC(=O)c1cc(c(nc1Cl)Cl)F AS-9195 Cc1ccc(cc1I)F AS-9196 Cc1ccc(cc1Cl)I AS-9197 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)O AS-9198 c1cc2c(cc1[N+](=O)[O-])c(ns2)N AS-9199 c1ccc(cc1)c2nc(cs2)CO AS-9200 Cc1c2c(ncnc2sc1c3ccccc3)O AS-9201 CC(=O)c1cc2cc(cc(c2oc1=O)Cl)Cl AS-9202 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCCC2 AS-9203 Cc1c(nn(n1)c2ccccc2)C(=O)NN AS-9204 c1c(cc(c(c1Br)N)Br)C2CCCCC2 AS-9205 CCCCCSc1c(cccn1)C(=O)O AS-9206 CSc1c(cccn1)C(=O)N AS-9207 c1c(cc(c(c1[N+](=O)[O-])N)Cl)C(F)(F)F AS-9208 c1ccc2c(c1)c(c(s2)C(=O)N)Cl AS-9209 Cc1cc(c(c2c1CCC2)OC)C#N AS-9211 Cc1ccc(c2c1CCC2)OC(=O)C AS-9212 C1CN2CCC1/C(=N/O)/C2.Cl AS-9213 CCOC(=O)Cc1c(c([nH]c1C(=O)OCC)C)C(=O)OCc2ccccc2 AS-9214 CCN(CC)CCc1ccccn1 AS-9215 C1CC(=O)C2CCC(=O)C1C2 AS-9216 CCC12CC3CC(C1)CC(C3)(C2)C(=O)O AS-9217 c1cc2c(cc1C(=S)N)OCO2 AS-9218 c1ccc2c(c1)OCC(O2)CCl AS-9219 CCOC(=O)c1c2ccccc2n(n1)C AS-9220 CNCc1ccc(cc1)c2cccs2 AS-9221 Cc1c(cnn1c2ccccc2)CNC AS-9222 Cc1c2cc(sc2n(n1)C)CO AS-9223 c1ccc2c(c1)C=C(CO2)C(=S)N AS-9224 CC(C)(C)OC(=O)N1CCN(CC1)Cc2ccc(cc2)C(=O)OC AS-9225 CC(C)(C)OC(=O)N1CCN(CC1)Cc2cccc(c2)CO AS-9226 CC(C)NCc1ccc(cc1)N2CCCCC2 AS-9227 CNCc1ccc(cc1)c2ccco2 AS-9228 CCOC(=O)c1ccc(cc1)c2nc(on2)C AS-9229 CCOC(=O)c1cccc(c1)c2nccs2 AS-9230 c1cc(c(nc1)C#N)N2CCCCC2 AS-9231 CNCc1ccc(cc1)c2ccccn2 AS-9232 CNCc1cccc(c1)OCCN2CCOCC2 AS-9233 Cc1nc(c(s1)CO)c2ccccc2 AS-9234 CNCc1cccc(c1)c2cccs2 AS-9235 CNCc1cccc(c1)CN2CCCCC2 AS-9236 c1cc(ccc1c2nc(cs2)C=O)C(F)(F)F AS-9237 Cn1c(cc(n1)CO)c2cccs2 AS-9238 Cn1c(cc(n1)c2cccs2)CO AS-9239 CN1CCN(CC1)Cc2ccccc2N AS-9240 CNCc1c2c(cs1)OCCO2 AS-9241 Cc1c(c(n(n1)c2ccccc2)C)CO AS-9242 CNCc1cccc(c1)c2ccsc2 AS-9243 c1ccc(c(c1)CN2CCOCC2)CO AS-9244 Cc1nc(on1)c2cccc(c2)Br AS-9245 c1ccnc(c1)Oc2cccc(c2)CO AS-9246 c1cnc(cc1CO)N2CCCCC2 AS-9247 c1cnc(cc1CO)N2CCSCC2 AS-9248 CN(C)CCOc1ccccc1CO AS-9249 CN(C)CCOc1ccc(cc1)CO AS-9250 CNCc1ccccc1OC2CCOCC2 AS-9251 CNCc1ccc(cc1)c2ccc(cn2)C(F)(F)F AS-9252 c1cc(sc1CO)N2CCOCC2 AS-9253 c1cc(ccc1CN2CCCC2)CO AS-9254 CN1CCCN(CC1)Cc2ccc(cc2)CN AS-9255 c1cc(cc(c1)C=O)Cn2cccn2 AS-9256 c1cc(cc(c1)CO)Cn2cccn2 AS-9257 c1cc(c(cc1C(F)(F)F)CO)N2CCOCC2 AS-9258 CNCc1cc(ccc1N2CCOCC2)C(F)(F)F AS-9259 CN(C)CCCOc1cccc(c1)CO AS-9260 CN1CCCN(CC1)c2ccc(cc2)CO AS-9261 CN1CCCN(CC1)c2ccccc2CO AS-9262 CN1CCCN(CC1)c2ccccc2CN AS-9263 CN1CCCN(CC1)c2ccccc2C#N AS-9264 CNCC1CCSCC1 AS-9265 c1cc(sc1)C2(CCOCC2)CO AS-9266 Cn1c(ccn1)C(=O)Oc2c(c(c(c(c2F)F)F)F)F AS-9267 c1ccc(cc1)OCc2cccc(c2)N AS-9268 Cc1cc(n(n1)c2ccc(cc2)CO)C AS-9269 Cc1cc(n(n1)c2ccc(cc2)CN)C AS-9270 Cc1nc(cs1)c2ccccc2N AS-9271 CNCC1CCN(CC1)Cc2ccco2 AS-9272 CNCC1CCN(CC1)Cc2cccnc2 AS-9273 c1cc(sc1)Cc2ccc(cc2)CBr AS-9274 Cc1cc(n(n1)C2=NCCN2)C.Br AS-9275 Cc1c(sc(n1)C)C(=O)C AS-9276 C1CC/C(=N\O)/NCC1 AS-9277 COc1cc(c(cc1I)OC)Cl AS-9278 c1cc(ccc1CC(=S)N)Cl AS-9279 Cc1csc(c1N=C=S)C(=O)OC AS-9280 COC(=O)c1c(c(cs1)C#N)n2cccc2 AS-9281 CS(=O)(=O)c1csc(c1Cl)C(=O)O AS-9282 CC(C)S(=O)(=O)c1csc(c1N)C(=O)O AS-9283 COc1ccc(cc1)c2c(c(sc2C(=O)O)SC)C#N AS-9284 CCOC(=O)c1c2c(c(s1)SCc3ccccc3)C(=O)CCC2 AS-9285 CCCSc1c2c(c(s1)C(=O)OCC)CCCC2=O AS-9286 c1ccc(cc1)S(=O)(=O)c2ccsc2 AS-9287 COC(=O)C1NCCS1.Cl AS-9288 c1cc2c(cc1C#N)non2 AS-9289 CSc1nc2ccc(cc2s1)[N+](=O)[O-] AS-9290 CC(C)n1cc(c(=O)[nH]c1=O)C#N AS-9291 c1c(c(sc1S(=O)(=O)N)N2CCNCC2)[N+](=O)[O-] AS-9292 c1cc2c(cc(nc2c(c1)F)C(F)(F)F)Cl AS-9293 Cc1c(c(c(n1C2CC2)C)C(=O)O)C(=O)C AS-9294 CC1CCN(CC1)C(=O)C2CCCNC2.Cl AS-9295 CC1CCN(CC1)C(=O)C2CCNCC2.Cl AS-9296 C1CCN(CC1)C(=O)C2CCCCN2.Cl AS-9297 CC1CCN(CC1)C(=O)C2CCCCN2.Cl AS-9298 C1CCNC(C1)C(=O)N2CCOCC2.Cl AS-9299 c1ccc(c(c1)c2cccc(c2)C=O)C(=O)O AS-9300 CC(C)(C)OC(=O)n1cc(c2c1cc(cc2)C(=O)OC)C=O AS-9301 C1CCN(CC1)C2CCN(CC2)C(=N)N.I AS-9302 C1CCC(CC1)N2CCN(CC2)C(=N)N.I AS-9303 Cn1c(c(cn1)Br)c2cccc(c2)N AS-9304 B(c1cc(ncc1Br)Br)(O)O AS-9305 Cc1c2cc(ccc2sc1C(=O)CCl)Cl AS-9306 C1C2CC3(CC1CC(C2)(C3)Cl)C(=O)O AS-9307 CSc1nc(nc(n1)N)C2CC2 AS-9308 c1ccc(cc1)C(=O)Oc2cccc3c2CCC3=O AS-9309 COc1cc(c(cc1Cl)OC)N=C=S AS-9310 Cc1cc(cc(c1N=C=S)Cl)Cl AS-9311 c1c(cc(c(c1F)N=C=S)Br)Br AS-9312 c1cc(c(cc1N=C=O)[N+](=O)[O-])Cl AS-9313 Cc1cccc(c1N=C=S)C(C)C AS-9314 c1ccc(cc1)c2cc(c3c(c(sc3n2)C(=O)O)N)C(F)(F)F AS-9315 Cc1ccc(cc1)c2csnn2 AS-9316 c1c(cc(c(c1Cl)N)Cl)C(F)(F)F AS-9317 COC(=O)c1cc2c(s1)-c3cc(ccc3SC2)Cl AS-9318 CCOC(=O)CC1C(=O)N(CCN1C)C AS-9319 c1cc(oc1C=O)c2c(cc(cc2Cl)C(F)(F)F)Cl AS-9320 CCOC(=O)c1cnn(c1C)c2ccc(cc2)N AS-9321 c1cc(c(cc1c2ccc(o2)C=O)C(F)(F)F)F AS-9322 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)O)Br AS-9323 C1CCC(CC1)n2c(nnc2S)O AS-9324 CCOC(=O)c1csc(n1)c2cccc(c2Cl)Cl AS-9325 CCOC(=O)c1cc(on1)c2cccs2 AS-9326 c1cc(c(cc1F)N)n2ccnc2 AS-9327 CCOC(COc1ccc(cc1)Br)OCC AS-9328 c1cc(ccc1OCCCBr)Br AS-9329 CCOC(=N)c1cccs1.Cl AS-9330 COc1ccc2c(cc(=O)oc2c1)CCl AS-9331 c1cc2c(cc1N)nco2.Cl AS-9332 CCOC(=O)C1CC1C AS-9333 CC1CNc2ccccc2S1 AS-9334 COc1ccc(c(c1)O)N AS-9335 c1cc(ccc1C(=O)O)N2CCNC2=O AS-9336 CC(C)N(c1nnc(s1)N)C(C)C AS-9337 CC1CN(CC(O1)C)c2nnc(s2)N AS-9338 CCNc1nnc(s1)N AS-9339 CCOC(=O)c1ccc(c(c1)N)OC AS-9340 CNc1cc(nc(n1)N)Cl AS-9341 CC1CN(CC(O1)C)c2cc(nc(n2)N)Cl AS-9342 CCOc1cc(nc(n1)N)Cl AS-9343 CCOC(=O)c1cc(ccc1N2CC(OC(C2)C)C)[N+](=O)[O-] AS-9344 CC1CN(CC(O1)C)c2ccc(cc2C(=O)O)[N+](=O)[O-] AS-9345 COC(=O)c1cc(c(cc1F)F)F AS-9346 c1cc(c(cc1F)C(=O)NN)F AS-9347 c1ccc(c(c1)c2nnco2)OC(F)(F)F AS-9348 Cc1nnc(o1)c2ccccc2OC(F)(F)F AS-9349 c1cc(cc(c1)OC(F)F)NC(=O)/C=C\C(=O)O AS-9350 Cc1ccc(cc1F)n2cccc2 AS-9352 CCOC(=O)c1ccc2nccn2c1 AS-9353 CCOC(=O)c1ccc2ncc(n2c1)Cl AS-9354 c1cn2cc(cc(c2n1)Br)Cl AS-9355 CCOC(=O)C(c1ccc(cc1)F)Br AS-9356 c1cc(c2cc(sc2c1)C(=O)NN)C(F)(F)F AS-9357 c1cc(cc2c1cc(s2)C(=O)NN)Br AS-9358 CCOC(=O)c1c(c2ccccc2s1)n3cccc3 AS-9359 c1cc2nc(c(n2c(c1)Cl)Cl)C(=O)O AS-9360 c1cc(c2c(c1)[nH]nc2Br)C(F)(F)F AS-9361 c1cc2c(c(c1)C(F)(F)F)[nH]nc2Br AS-9362 c1cc(ccc1c2cnco2)OC(F)(F)F AS-9363 COc1ccc2c(c1)NCCO2 AS-9364 COC(=O)/C=C/c1ccc(c(c1)Cl)O AS-9365 CC1(CC(=O)c2cc(ccc2O1)O)C AS-9366 CN(CCO)C(=O)Nc1cc(ccc1OC)OC AS-9367 COc1ccc(c(c1)OC)CNC(=O)CCl AS-9368 COC(=O)c1cc(n[nH]c1=O)c2ccccc2 AS-9369 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)N AS-9370 c1cc(c(cc1F)F)C(=O)NN AS-9371 c1cc(c(cc1F)F)c2nnc(o2)CCl AS-9372 COC(=O)c1cc(cc(c1O)NO)Br AS-9373 c1cc2ncc(n2cc1Cl)C(=O)C(Cl)(Cl)Cl AS-9374 c1cn2c(cc1Cl)ncc2Br AS-9375 c1cc2c(cc1C(=O)O)[nH]nc2Br AS-9376 Cc1cccc2n1c(cn2)Br AS-9377 Cc1cccc2n1c(cn2)Cl AS-9378 c1cc2c(cc1C#N)nc(o2)Cl AS-9379 c1ccn2c(c1)nc(c2Br)C(=O)O AS-9380 c1cc(c2c(c1)NC(=O)CO2)C(=O)O AS-9381 CN1c2cccc(c2OCC1=O)C(=O)OC AS-9382 CN1c2cccc(c2OCC1=O)C(=O)O AS-9383 c1cc(ccc1c2ccnc(n2)N)Br AS-9384 c1c(cc(c2c1cn[nH]2)Br)N AS-9385 Cc1ccc2c(c1N)nn[nH]2 AS-9386 COC(=O)c1c(nc(s1)N2CCCC2)N AS-9387 COC(=O)c1ccc(cc1[N+](=O)[O-])C(F)(F)F AS-9388 CCOC(=O)c1ccc(cc1[N+](=O)[O-])C(F)(F)F AS-9389 CCOC(=O)c1ccc(cc1N)C(F)(F)F AS-9391 COC(=O)/C=C/c1ccc(c(c1)Cl)Cl AS-9392 COC(=O)c1cc(ccc1F)Cl AS-9393 CCOC(=O)c1cc(ccc1F)Cl AS-9394 c1cc(c(cc1Cl)C(=O)NN)F AS-9395 c1cc(cc(c1)Br)c2nnc(o2)CCl AS-9396 c1ccc(c(c1)c2nnc(o2)CCl)F AS-9397 COC(=O)c1ccc(c(c1O)O)O AS-9398 Cn1cc(c2c1cccc2)C(=O)N AS-9399 Cn1cc(c2c1cccc2)C#N AS-9400 c1cc2cnccc2c(c1)[N+](=O)[O-] AS-9401 c1c(cc(cc1Cl)Cl)NN.Cl AS-9402 c1cc2c3c(ccc(c3c1)Br)CC2 AS-9403 c1cc2c(cc1[N+](=O)[O-])C(=O)NC2=O AS-9405 Cc1cc(c(c(c1Cl)C)Cl)O AS-9406 CC(=O)c1cc(cc(c1)OC(=O)C)OC(=O)C AS-9407 Cn1c(n[nH]c1=S)C(F)(F)F AS-9408 c1c(c(=O)[nH]c(=O)[nH]1)Br AS-9409 c1c(c(cc(c1F)F)F)C(=O)O AS-9410 Cc1cc(n(n1)CO)C AS-9411 c1cc(c(cc1C(=O)O)N)N AS-9412 c1cnccc1CCl.Cl AS-9413 CCOC(=O)c1cc2c(s1)cccc2Br AS-9414 c1cc2c(cc(s2)C(=O)NN)c(c1)Br AS-9415 Cn1ccc2c1ccc(c2)OC AS-9416 c1c2c(cc(c1Cl)Cl)nc([nH]2)C(F)(F)F AS-9417 CCC1CCCCN1c2cc(nc(n2)N)Cl AS-9418 c1c(c(cc(c1F)F)F)C(=O)NN AS-9419 Cc1ccc(cc1F)NC(=O)CCl AS-9421 Cc1ccc(cc1F)NC(=O)/C=C\C(=O)O AS-9422 CCOC(=O)c1cc(c(c(c1F)F)F)F AS-9424 Cc1c(c(nn1C)C(=O)OC)Br AS-9425 c1ccc2c(c1)C(=O)N(C2=O)CCC3CCCCC3 AS-9426 COC(=O)c1ccc2c(c1)nc(o2)S AS-9427 COc1ccc2c(c1)nc(o2)S AS-9428 Cc1c2cc(sc2n(n1)C)C=O AS-9429 CC(C)(C)OC(=O)N1CCN(CC1)c2nnc(s2)N AS-9430 CC(C)(C)OC(=O)COc1ccccc1C#N BA-0038 c1ccc(cc1)NC(=O)NC(=O)Cn2cncn2 BA-0080 c1ccc(cc1)Cc2ccc3c(c2)[nH]c(=O)n3c4ccc(cc4)Br BA-0286 COC(=O)Cc1ccc(cc1)Br BA-0600 COC(=O)C(CC(=O)c1ccc(cc1)S(=O)(=O)C)(C(=O)c2cc(cc(c2)F)F)C(=O)OC BA-0606 c1nc(c(c(n1)Cl)C=O)N2CCCCC2 BA-0608 COc1cc(cc(c1)OC)C(=O)CC#N BA-0800 c1c(cc(nc1C(=O)O)C(F)(F)F)C(F)(F)F BA-0802 Cc1cc2nccc(n2n1)c3c(cc(cn3)C(F)(F)F)Cl BA-0803 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNC(=O)c3cc(nc(c3)C(F)(F)F)C(F)(F)F BA-0804 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNC(=O)c3cc(nc(c3)C(F)(F)F)C(F)(F)F BA-0805 COc1ccc(cc1OC)c2cc([nH]n2)N BA-0806 COc1ccc(cc1OC)c2cc(on2)N BA-0807 COc1cccc(c1)C(=O)CC#N BA-0809 c1ccc(cc1)N2CCN(CC2)C(=O)c3cc(nc(c3)C(F)(F)F)C(F)(F)F BA-0810 COc1cc(cc(c1)OC)c2cc([nH]n2)N BA-0811 COc1cc(cc(c1)OC)c2cc(on2)N BA-0812 c1cc(cc(c1)Br)c2cc(on2)N BA-0814 c1cc(cc(c1)Br)c2cc([nH]n2)N BA-0815 CN1CCN(CC1)C(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F BA-0817 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cc(nc(c3)C(F)(F)F)C(F)(F)F BA-0818 c1cc(cc(c1)N2CCN(CC2)C(=O)c3cc(nc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F BA-0819 c1ccc(cc1)NC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F BA-0822 COc1cccc(c1)c2cc(on2)N BA-0825 c1ccc(c(c1)NC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F)Cl BA-0826 c1cc(cc(c1)NC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F BA-0827 CCc1ccc(c(c1)C=O)O BA-0829 c1cc(ccc1NC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F)Cl BA-0830 COc1cccc(c1)NC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F BA-0831 c1c(cc(nc1C(F)(F)F)C(F)(F)F)C(=O)NC2CC2 BA-0832 c1cc(c(cc1/N=C\2/c3cc(ccc3NC2=O)Br)Cl)Cl BA-0833 Cc1ccc(c(c1)C(=O)/C=C/N(C)C)O BA-0834 c1cc(cnc1)CNC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F BA-0835 c1ccnc(c1)CNC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F BA-0836 Cc1ccc(c(c1)F)/N=C\2/c3cc(ccc3NC2=O)Br BA-0837 Cc1ccc(cc1Cl)/N=C\2/c3cc(ccc3NC2=O)Br BA-0838 c1cc(ccc1/N=C\2/c3cc(ccc3NC2=O)Br)O BA-0839 CCCCCCCCc1ccc(c(c1)C=O)O BA-0840 CNC(=O)c1cc(nc(c1)C(F)(F)F)C(F)(F)F BA-0841 Cc1ccc(c(c1)c2cc[nH]n2)O BA-0843 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)OC)C BA-0846 CCc1cc(c(c(c1)CN(C)C)O)CN(C)C BA-0847 CCC(C)c1ccc(c(c1)CN(C)C)O BA-0848 c1cc(cc(c1)Br)NC(=O)NCCCl BA-0850 c1ccc(cc1)CN2CCN(CC2)c3ncc(s3)/C=C/4\c5ccccc5NC4=O BA-0852 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)C(C)C)C BA-0853 c1cc(ccc1N2C(=O)C(SC23c4cc(ccc4NC3=O)Br)CC(=O)O)O BA-0857 Cc1cc(c(c(c1)OC)O)CN(C)C BA-0858 CCCCOc1ccc(cc1)/N=C\2/c3cc(ccc3NC2=O)Br BA-0859 CCC(C)Cc1ccc(c(c1)CN(C)C)O BA-0860 CNC(=O)c1cc(cc(n1)C(=O)NC)C(F)(F)F BA-0861 c1c(cc(nc1C(=O)NC2CC2)C(=O)NC3CC3)C(F)(F)F BA-0862 c1ccc(cc1)c2nccc(n2)c3c(cc(cn3)C(F)(F)F)Cl BA-0866 c1cc(c(c(c1)Br)C=O)F BA-0930 c1cc2c(cc1[N+](=O)[O-])sc(n2)Cl BA-0932 COC(=O)c1ccc(cc1)C(=S)N BA-0935 c1cc2c(cc1C(=O)O)sc(n2)N BA-0937 CCCOc1cnn(c(=O)c1Cl)C BA-7011 C[C@@H](c1cccc(n1)COc2c3ccccc3c4nnc(n4n2)C(F)(F)F)NCCc5ccccc5 BA-7035 CC(C)C(NC(=O)OCc1ccccc1)S(=O)(=O)c2ccccc2 BB-0004 c1c(c(=O)[nH]c(=S)[nH]1)CN2CCOCC2 BB-0036 c1c(c(=O)[nH]c(=S)[nH]1)CN2CCCCC2 BB-0052 CN1CCN(CC1)Cc2c[nH]c(=S)[nH]c2=O BB-0053 C[C@@H](C(=O)O)Nc1c(cc(cn1)C(F)(F)F)Cl BB-0056 CC(C)(C)OC(=O)N1CCCCN1 BB-0202 CC(C)(C)OC(=O)N1CCCN1 BB-0207 CCOC(=O)CN1CCCCN1C(=O)OC(C)(C)C BB-0210 CC(C)(C)OC(=O)N1CCCCCN1C(=O)OCc2ccccc2 BB-0218 CCOC(=O)c1c(cccn1)C#N BB-0600 CCOC(=O)c1ccc(cn1)C(=O)O BB-0601 CCOC(=O)c1cc(ccn1)C#N BB-0602 c1cc(c(cc1F)Cl)OCC#N BB-0603 c1cc(ccc1OCC(=S)N)OC(F)(F)F BB-0604 CCOC(=O)c1ccc(cn1)C#N BB-0605 CCOC(=O)c1ccc(cn1)Cl BB-0606 c1cc(ncc1Cl)C(=O)O BB-0607 c1cnc(cc1C#N)C(=O)O BB-0608 c1cc(c(cc1F)Cl)OCC(=S)N BB-0609 c1cc(c(cc1Br)Cl)OCC#N BB-0610 c1cc(ncc1C#N)C(=O)O BB-0611 c1cc(c(nc1)S)C#N BB-0700 CC(=O)OCC(=O)c1ccc(cc1)OC BB-0701 CC(=O)OCC(=O)c1ccc(cc1)[N+](=O)[O-] BB-0702 c1ccc(cc1)COc2ccc3ccc(cc3c2)OCc4ccccc4 BB-0704 CC(=O)OCC(=O)c1ccc(cc1)Cl BB-0705 CC(=O)OCC(=O)c1ccc(cc1)F BB-0706 CCOC(=O)c1c(con1)C(=O)c2ccc(cc2)Oc3ccccc3 BB-0707 c1cc(c(cc1n2ccnc2)Cl)C(=O)NCCO BB-0708 c1cc(c(cc1N2CCCCC2)Cl)C(=O)O BB-0710 Cc1ccc(cc1)C(C=O)C=O BB-0711 c1cc(cc(c1)Cl)C(C=O)C=O BB-0712 CCOC(=O)C(C)(C)Sc1ccc(cn1)[N+](=O)[O-] BB-0713 CC(C)(C(=O)O)Sc1ccc(cn1)[N+](=O)[O-] BB-0714 c1cc(ccc1c2ccc3c(c2)OCCCO3)C(=O)O BB-0716 c1cc(ccc1c2ccc3c(c2)OCCCO3)C(=O)NN BB-0717 c1cc(c(nc1)S)[N+](=O)[O-] BB-0720 c1cc(c(cc1n2cncn2)Cl)C(=O)O BB-0721 c1cc(c(nc1)S)Cl BB-0722 c1cc(c(cc1n2cncn2)Cl)C(=O)NCCO BB-0725 c1cc(c(cc1n2cncn2)Cl)C(=O)NN BB-0728 COC(=O)c1c(cnc(n1)SC)Br BB-0729 COC(=O)C(c1ccc(cc1)F)N.Cl BB-0800 Cc1cc(cc(c1N)[N+](=O)[O-])F BB-0801 c1ccc(c(c1)Oc2cc(cc(n2)C(F)(F)F)Cl)OC(=O)O BB-0802 Cc1ccc(cc1)C(C(=O)OC)N.Cl BB-0803 COc1ccc(cc1)C(C(=O)OC)N.Cl BB-0808 COC(=O)C(c1cccc(c1)F)N.Cl BB-0809 CCCCn1cc(c(=O)[nH]c1=O)C#N BB-0810 c1ccc2c(c1)C(=O)N(C2=O)OCc3nc4ccccc4o3 BB-0811 c1c(c(=O)[nH]c(=O)n1CC(=O)O)C#N BB-0812 CCOC(=O)c1cc2cc(ccc2o1)[N+](=O)[O-] BB-0814 c1cc2c(cc1NC(=S)N)cn[nH]2 BB-0815 CC(=O)Nc1ccc(cc1)c2csc(n2)N BB-0818 CCO/C(=C(/C#N)\C(=O)NC(=O)OCC)/C BB-0819 c1cc(ccc1C=O)I BB-0825 c1c2c(sc1CO)CCC2 BB-0827 c1cnc(nc1C(F)(F)F)NCCN BB-0828 CCOC(=O)c1cn2cc(cc(c2n1)C)I BB-0834 c1cc(ccc1C=O)c2cc(ccn2)C(=O)O BB-0835 Cn1c2cc(ccc2cn1)[N+](=O)[O-] BB-0836 Cn1cc2ccc(cc2n1)[N+](=O)[O-] BB-0837 Cc1c(c(=O)[nH]c(=O)n1CC(=O)O)C#N BB-0841 c1cc(ccc1c2cn3ccsc3n2)N BB-0842 c1ccc(c(c1)C(C#N)c2c(cc(cn2)C(F)(F)F)Cl)Cl BB-5010 c1ccc(c(c1)[C@@H](c2c(cc(cn2)C(F)(F)F)Cl)c3[nH]nnn3)Cl BB-5020 c1cc(cc(c1)C(F)(F)F)C(C#N)C2=NC=CCC2C(F)(F)F BB-5023 c1cc(cc(c1)C(F)(F)F)[C@@H](c2c(cc(cn2)C(F)(F)F)Cl)c3[nH]nnn3 BB-5024 c1ccc(cc1)[C@@H](c2ccccn2)c3[nH]nnn3 BB-5026 c1ccnc(c1)[C@H](c2ccc(cc2)Cl)c3[nH]nnn3 BB-5027 c1cc(cc(c1)Cl)[C@@H](c2c(cc(cn2)C(F)(F)F)Cl)c3[nH]nnn3 BB-5030 c1ccc(cc1)[C@@H](c2c(cccn2)C(F)(F)F)c3[nH]nnn3 BB-5031 c1cc(c(c(c1)Cl)[C@@H](c2c(cccn2)C(F)(F)F)c3[nH]nnn3)Cl BB-5032 c1cc(cc(c1)C(F)(F)F)[C@@H](c2c(cccn2)C(F)(F)F)c3[nH]nnn3 BB-5033 c1cc(ccc1[C@@H](c2c(cc(cn2)C(F)(F)F)Cl)c3[nH]nnn3)Cl BB-5034 c1cc(ccc1[C@@H](c2c(cc(cn2)C(F)(F)F)Cl)c3[nH]nnn3)[N+](=O)[O-] BB-5035 c1cc(c(nc1)[C@H](c2ccc(cc2)Cl)c3[nH]nnn3)C(F)(F)F BB-5036 Cc1cccc(c1)[C@@H](c2c(cc(cn2)C(F)(F)F)Cl)c3[nH]nnn3 BB-5038 c1ccc(cc1)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl BB-5046 CNc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl BB-5050 c1cc(ccc1Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl BB-5051 c1ccc(c(c1)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl BB-5057 c1cc(cc(c1)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F BB-5058 COC(=O)c1c(ccs1)NC(=O)c2ccc(cc2)Br BC-0028 c1cc(c(nc1)c2ccc3c(c2)ncnc3Nc4ccc(cc4)C(F)(F)F)C(F)(F)F BC-0200 c1ccnc(c1)C2CCNC2 BC-0203 c1cc2c(cc1Br)c(cc(n2)N)O BC-0204 COC(=O)c1cc(c(s1)C=O)Br BC-0205 CCOC(=O)C1CN(c2ccccc2O1)C BC-0602 c1cc(ccc1c2csc(n2)N3CCC(CC3)C(=O)NCCO)Cl BC-0700 c1c(cnc(c1Br)OCC2CC2)C(=O)O BC-0702 CC(=O)Nc1cc(c(cc1Cl)Cl)OCc2ccc(cc2)[N+](=O)[O-] BC-0703 c1c(cnc(c1C(=O)O)OCC2CC2)Br BC-0705 c1cc(cc(c1)[N+](=O)[O-])c2ccc(cc2)C(=O)O BC-0710 c1cc(ccc1C(=S)N2CCCCC2)Oc3c(cc(cn3)C(F)(F)F)Cl BC-0711 c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)Cl)C=O)F BC-0713 c1cc(ccc1Cn2cc(cc(c2=O)Cl)C=O)Cl BC-0714 c1cc(ccc1Cn2cc(cc(c2=O)Cl)C=O)F BC-0715 CCOC(=O)c1c(n2ccccc2n1)I BC-0718 c1ccc2c(c1)nc(o2)N(CCC#N)N BC-0721 CCOC(=O)c1cn2cc(cc(c2n1)Cl)Cl BC-0729 c1cc2c(cc1Br)nco2 BC-0732 COC(=O)Cn1c(c(c(n1)Br)[N+](=O)[O-])Br BC-0801 c1cc(ncc1[N+](=O)[O-])N2CCC(CC2)C(F)(F)F BC-0802 c1cnc(c(c1Cl)C(=O)O)Cl BC-0803 COC(=O)C1(CCCC1)C#N BC-0805 C(C(=O)O)n1c(c(c(n1)Br)[N+](=O)[O-])Br BC-0807 COC(=O)c1cc(c[nH]1)C=O BC-0808 c1ccc2c(c1)c(c[nH]2)C(=O)CC#N BC-0809 COC(=O)C1(CCC1)C#N BC-0812 c1cnc(c(c1Cl)C=O)Cl BC-0813 c1cc(c(nc1)c2ccc(cc2)C=O)C(F)(F)F BC-0814 c1c(c[nH]c1C(=O)C(Cl)(Cl)Cl)I BC-0815 COC(=O)c1cc(c[nH]1)I BC-0819 C1CCC(C1)(C#N)C(=O)O BC-0820 CCOC(=O)C(C(=O)OCC)N(C)C BC-0821 COC(=O)c1ccc(nc1)N2CCC(CC2)C(F)(F)F BC-0822 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)C(=O)OC BC-0823 c1cc2c(c[nH]c2nc1)[N+](=O)[O-] BC-0824 c1cc2c(c[nH]c2nc1)C=O BC-0825 c1cc2c(cc1[N+](=O)[O-])cc(o2)CO BC-5019 CC(C)(C)OC(=O)N1CCc2c(cnc(n2)N)C1 BC-5021 c1ccc(cc1)OC(=O)NN BD-0001 c1cc(c(c(c1)Cl)C(=O)NCc2ccc(cn2)C(F)(F)F)Cl BD-0007 c1cc(c(c(c1)Cl)c2ncc3n2cc(cc3)C(F)(F)F)Cl BD-0023 Cc1c2ccccc2sc1N.Cl BD-0037 Cc1c2ccccc2sc1NS(=O)(=O)c3ccc(cc3)C(=O)OC BD-0060 c1cc(c(c(c1)Cl)C(=O)NCc2cc(ccn2)C(F)(F)F)Cl BD-0063 CC(C(=O)OC)Oc1ccc(cc1)c2ncc3n2cc(cc3Cl)C(F)(F)F BD-0064 c1cc(c(c(c1)Cl)c2ncc3n2ccc(c3)C(F)(F)F)Cl BD-0065 Cc1c2ccccc2sc1N(Cc3ccc(c(c3)C(F)(F)F)F)S(=O)(=O)c4ccc(cc4)C(=O)OC BD-0067 CCOC(=O)c1c[nH]cc(c1=O)C(=O)OCC BD-0078 Cc1c(c(=O)[nH]c(n1)N)Cc2cccc(c2)Oc3ccccc3 BD-0084 CC(C(=O)/C=C/N(C)C)n1cc(ccc1=O)C(F)(F)F BD-0102 CCOC(=O)C1=C(NC(=O)NC1C(C)C)C BD-0109 CCOC(=O)c1cncc(c1Cl)C(=O)OCC BD-0110 CCOC(=O)c1c(nc[nH]1)C(F)(F)F BD-0119 c1cc(ccc1C(=O)CC#N)N2CCOCC2 BD-0200 c1cc(ccc1C(=O)O)N2CCCC2 BD-0212 c1cc(ccc1C(=O)O)N2CCCCC2 BD-0213 c1cc(ccc1C(=O)CC#N)N2CCCC2 BD-0221 c1cc(ccc1C(=O)CC#N)N2CCCCC2 BD-0225 c1cc2c(cc1Br)cc(o2)C(=O)CC#N BD-0227 c1ccc2c(c1)cc(o2)C(=O)CC#N BD-0229 CCCCO/C=C/C(=O)C(F)(F)F BD-0230 CCOC(=O)c1cn(cc1C(F)(F)F)C BD-0247 COC(=O)/C(=C/C=C(/C(F)(F)F)\[O-])/C#N.[K+] BD-0268 COC(=O)c1ccc(nc1Br)C(F)(F)F BD-0273 CCOC(=O)c1c(c2cc(ccc2o1)Br)N BD-0274 Cn1cc(c(c1)C(F)(F)F)C(=O)O BD-0278 CCOC(=O)c1c[nH]cc1C(F)(F)F BD-0280 c1c(cn[nH]1)C(F)(F)F BD-0296 COC(=O)c1c(c2cc(c(nc2s1)C3CC3)Cl)N BD-0700 Cn1c2ccccc2c(c1C(=O)O)Br BD-0701 CCC(c1cc(n(c1)C)C(=O)OC)O BD-0702 Cc1nc(c(c(n1)O)Br)NC BD-0706 COC(=O)c1cc(ccc1[N+](=O)[O-])N2CCCCC2 BD-0708 Cc1nc(c(c(n1)O)Br)N(C)C BD-0711 c1cc2c(cc1Br)c(=O)n(cn2)CC(F)(F)F BD-0713 COc1ccc(cc1N)CC(=O)OC BD-0715 c1cc(c(cc1N2CCCCC2)C(=O)O)[N+](=O)[O-] BD-0716 CCC(=O)c1cc(n(c1)C(=O)OC(C)(C)C)C(=O)OC BD-0717 c1cc(c(cc1N2CCCCC2)C(=O)NN)[N+](=O)[O-] BD-0719 c1cc2nc(cn2cc1C(F)(F)F)CCl BD-0721 CC(C)c1ccc(cc1)C(=S)N BD-0724 COC(=O)c1cc(ccc1F)N BD-0725 c1cc(ccc1CSc2ccc(cc2)Br)N BD-0727 c1ccc2c(c1)CCC(=C2Cl)CO BD-0728 c1c(c(c(c(n1)Cl)Cl)C(=O)O)C(F)(F)F BD-0730 Cc1cc(nc(n1)N)N BD-0732 COc1cc(ccc1[N+](=O)[O-])C#N BD-0733 c1c(cnc(n1)C(F)(F)F)Br BD-0736 Cc1cc(c2c(c1)nco2)C(=O)OC BE-0007 c1c(cc(c(c1C#N)N)I)C(F)(F)F BE-0009 c1cc(ccc1c2cc([nH]n2)NC(=O)CSc3c(cc(cn3)C(F)(F)F)Cl)Cl BE-0013 Cc1nc2cc(cc(c2o1)C(=O)OC)Br BE-0015 COC(=O)c1cc(cc2c1ocn2)Br BE-0016 CC(C)NC(=O)N1CCN(CC1)C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl BE-0026 c1cc(c(cc1Cl)Cl)c2cc([nH]n2)NC(=O)CCSc3c(cc(cn3)C(F)(F)F)Cl BE-0028 Cc1c(c(c(cn1)Br)O)OCc2ccccc2 BE-0031 COC(=O)c1cc(cc2c1oc(=O)[nH]2)Br BE-0036 Cc1cc(c2c(c1)nc(o2)C)C(=O)OC BE-0038 C[Si](C)(C)C#Cc1cc(cc(c1N)C#N)C(F)(F)F BE-0039 COc1cc(c(c(c1)[N+](=O)[O-])O)C(=O)OC BE-0042 Cc1cc(c2c(c1)nc(o2)CCl)C(=O)OC BE-0043 COc1c(cc(cc1OC(=O)c2ccccc2)Cl)[N+](=O)[O-] BE-0044 c1ccc(cc1)COc2c(cc(cc2OC(=O)c3ccccc3)Cl)[N+](=O)[O-] BE-0045 CC(C)(C)OC(=O)N1CCC2(CC1)CC(C2)C#N BE-0046 COc1cc(c(c(c1)N)O)C(=O)OC BE-0047 COc1cc(c2c(c1)nc(o2)CCl)C(=O)OC BE-0048 COC(=O)c1cc(cc2c1oc(n2)CCl)Br BE-0049 COc1cc(cc2c1OC(CN2)C#N)C(=O)OC BE-0051 C#Cc1cc(cc(c1N)C#N)C(F)(F)F BE-0058 c1c(cnc(c1Cl)CNC(=O)N2CCN(CC2)c3cc(ncn3)Cl)C(F)(F)F BE-0060 c1c[nH]c2c1cc(cc2C#N)C(F)(F)F BE-0067 c1ccc(cc1)COc2c(cc(cc2OC(=O)c3ccccc3)Cl)N BE-0069 CNC(=O)c1cc(ccc1NC(=O)c2ccccc2Cl)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl BE-0070 c1cc(ccc1c2cn[nH]c2NC(=O)CSc3c(cc(cn3)C(F)(F)F)Cl)Cl BE-0075 c1cc(ccc1c2cn[nH]c2NC(=O)CCSc3c(cc(cn3)C(F)(F)F)Cl)Cl BE-0081 c1c(cnc(c1Cl)CNC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F BE-0082 COc1cc(cc2c1oc(n2)CCl)C(=O)OC BE-0089 COc1c(cc(cc1OC(=O)c2ccccc2)Cl)N BE-0097 c1c(cc2c(c[nH]c2c1C#N)Br)C(F)(F)F BE-0098 CCOC(=O)/C=C/c1ccccn1 BE-0204 COC(=O)Cc1cn2cc(ccc2n1)C(F)(F)F BE-0207 c1c[nH]nc1C2CNCCN2 BE-0212 c1cc2nc(cn2cc1C(F)(F)F)CC(=O)NN BE-0213 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cc(cn2)Br)[N+](=O)[O-] BE-0214 c1cc2nc(cn2cc1C(F)(F)F)CC(=O)O BE-0215 Cc1cn(cn1)C(c2ccccc2)(c3ccccc3)c4ccccc4 BE-0216 c1cnc(nc1C#N)N BE-0222 c1c(cnc(c1[N+](=O)[O-])N2CCNCC2)Br BE-0225 CCOC(=O)c1c(ccnc1Cl)C(F)(F)F BE-0226 Cc1c(c(c(s1)I)Br)I BE-0228 CCOC(=O)[C@H]1CNC[C@@H]1C(F)(F)F BE-0230 CCN(CC)c1nccc(n1)C#N BE-0234 CCOC(=O)[C@H]1CNC[C@@H]1C(=O)OCC BE-0236 c1ccc2c(c1)CCC3(C2)Nc4ccccc4S3 BE-0701 C1CCC2(C(C1)C(=O)O)NC(=O)CS2 BE-0702 C1CCCC2(CC1)NCCS2.Cl BE-0705 CC(=O)c1cccnc1C(=O)O BE-0707 c1ccc(cc1)CN2CCC3(CC2)Nc4ccccc4S3 BE-0708 c1ccc2c(c1)NC3(S2)CCCC3 BE-0710 Cc1cc(=O)[nH]c2c1CCC2 BE-0711 C1COCCC12NCCS2.Cl BE-0712 CC(C)(C)OC(=O)NC1CCCN(C1)c2ccc(cc2C(=O)OC)[N+](=O)[O-] BE-0715 c1c(cnc(c1Cl)C2CC(C2)C(=O)O)C(F)(F)F BE-0716 c1c(cn2cc(nc2c1Cl)C(=O)O)C#N BE-0717 Cc1cc(=O)[nH]c2c1CCCC2 BE-0718 c1ccc2c(c1)NC3(S2)CCOCC3 BE-0721 CCOC(=O)c1ccc(cn1)C(=O)C BE-0722 Cc1cc(cc(c1N)[N+](=O)[O-])I BE-0723 CC(C)(C)OC(=O)N1CCC2(CC1)NCC(=O)N2 BE-0724 CC(C)(C)OC(=O)N1CCC2(CC1)Nc3ccccc3S2 BE-0725 CCOC(=O)c1ccc(cn1)CC#N BE-0726 CC(=O)c1ccc(nc1)C(=O)O BE-0727 C1COCCC12NC(=O)CS2 BE-0728 Cc1cc(nc2c1CCC2)Cl BE-0729 C1CCC2CC3(CCC2C1)NCCS3 BE-0731 COC(=O)c1cc(ccc1N2CC(C2)C(=O)O)[N+](=O)[O-] BE-0732 CC1(OC(=O)C(C(=O)O1)Br)C BE-0733 CC(c1ccc(c(c1)OC)N)O BE-0736 C1CCC2(C(C1)O)NCCS2.Cl BE-0738 C1Cc2c([nH]c(=O)[nH]c2=O)C1 BE-0739 CC(C)(C)OC(=O)N1CCC2(CC1)N(CCS2)C(=O)NCCCl BE-0741 C1CSC(=O)N1 BE-0742 c1ccc2c(c1)NC3(S2)CCC4CCCCC4C3 BE-0743 CC1CCC2(CC1)NCCS2 BE-0745 c1ccc(cc1)C2CCC3(CC2)Nc4ccccc4S3 BE-0746 CCOC(=O)c1cc(c(nc1C2CC2)C(=O)OCC)C#N BE-0747 COC(=O)c1cc(ccc1N2CC3CC3C2C(=O)O)[N+](=O)[O-] BE-0748 Cc1cc([nH]c(=O)c1)c2ccc(cc2)Cl BE-0749 c1ccc(cc1)C2CCC3(CC2)NC(CS3)C(=O)O BE-0750 c1cc(ccc1Sc2ccc(cn2)[N+](=O)[O-])Cl BE-0751 c1cc(ccc1Sc2ccc(cn2)[N+](=O)[O-])Br BE-0753 CC(C)(C)OC(=O)N1CCCC(C1)C(=O)NN BE-0754 c1ccc(cc1)C2CCC3(CC2)NCCS3.Cl BE-0756 c1ccc(cc1)C2CCC3(CC2)NC(=O)CS3 BE-0757 Cc1c(cnc(n1)S(=O)(=O)C)C(=O)OC BE-0759 c1cc(ccc1Sc2ccc(cn2)N)Cl BE-0760 CC1CCC2(CC1)NC(CS2)C(=O)O BE-0761 c1ccc(cc1)Sc2ccc(cn2)N BE-0762 c1cc(ncc1CC#N)C(=O)O BE-0765 c1cc(ccc1S(=O)(=O)c2ccc(cn2)[N+](=O)[O-])Cl BE-0766 COc1cc(c(cc1C(=O)OC)I)N BE-0768 Cc1c(cnn1C(C)(C)C)C(=O)OC BE-0771 CC(=O)c1cc(cnc1Cl)Cl BE-0773 COc1ccc(cc1)Sc2ccc(cn2)N BE-0775 Cc1c(cnn1C(C)(C)C)C(=O)O BE-0777 c1c([nH]c(=O)[nH]1)C(=O)O BF-0007 Cn1c(c[nH]c1=O)C(=O)O BF-0008 CC(C)(C)OC(=O)NCCNC1CCN(CC1)C(=O)OCc2ccccc2 BF-0015 CC(C)(C)OC(=O)NCCCNC1CCN(CC1)C(=O)OCc2ccccc2 BF-0016 c1ccc(cc1)COC(=O)N2CCC(CC2)NCCN.Cl.Cl BF-0023 c1ccc(cc1)COC(=O)N2CCC(CC2)NCCCN.Cl.Cl BF-0024 c1c(cnc(c1Cl)CN2CCC(=O)CC2)C(F)(F)F BF-0041 COc1ccc(cc1)Cn2c3ccnc(c3c(n2)I)Cl BF-0054 c1ccc(cc1)Nc2ccnc(c2)C(F)(F)F BF-0206 c1c(cc(cc1[N+](=O)[O-])I)C(=O)O BF-0220 c1cc(c2c(c1)[nH]c(=O)[nH]2)N BF-0246 c1cc(c(cc1[N+](=O)[O-])C(C#N)c2cc(ccc2Cl)[N+](=O)[O-])Cl.O BF-0700 c1cc(oc1)c2c(c([nH]n2)N)F BF-0702 CC/C(=C(\C#N)/C(=O)OCC)/O BF-0703 C1Cc2c(nc(nc2Cl)Cl)C1 BF-0704 Cn1c2ccc(cc2nn1)N BF-0707 COc1c2c(nc(n1)Cl)CCC2 BF-0710 COC(=O)c1ccc(c(c1)N2CCCCC2)[N+](=O)[O-] BF-0711 CCOC(=O)c1cc(cnc1O)[N+](=O)[O-] BF-0712 c1c[nH]c2c(c1=O)cc(cc2C(=O)O)Br BF-0713 CCOC(=O)c1c(c2cc(ccc2[nH]1)[N+](=O)[O-])Br BF-0714 C1Cc2c(nc(nc2N)Cl)C1 BF-0715 COC(=O)c1ccc(c(c1)N2CCOCC2)[N+](=O)[O-] BF-0717 Cn1c2ccc(cc2[nH]c1=O)N BF-0719 CNc1cc(nc(n1)c2ccccc2)C#N BF-0720 CCOC(=O)c1c(nc(o1)N)C BF-0722 Cc1c(nc([nH]1)NC(=O)C)C BF-0723 Cc1c(sc(n1)NC(=N)N)C.Br BF-0725 CCOC(=O)c1csc(n1)NC(=N)N.Br BF-0728 CCOC(=O)c1c(nc(s1)NC(=N)N)C.Cl BF-0729 CCc1cc(=O)[nH]c(=O)[nH]1 BF-0730 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2ccccc2N BF-0731 CCOC(=O)C1CCCN(C1)C(=O)c2ccccc2N BF-0732 CCOC(=O)C1CCN(CC1)C(=O)c2ccccc2N BF-0733 c1cc(c(cc1CO)C#N)F BF-0734 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2C#N)C=O BF-0737 CCOC(=O)C1CCN(CC1)c2ccc(cc2C#N)C=O BF-0738 c1cc(c(cc1C=O)C#N)N2CCCCC2 BF-0739 c1cc2cc(sc2c(c1)Br)C(=O)O BF-0740 CCOC(=O)Cc1csc(n1)NC(=N)N.Cl BF-0741 c1cc2c(cc(s2)C(=O)Cl)c(c1)Br BF-0742 c1cc(c(nc1)Cl)c2ccnc(n2)c3ccncc3 BF-0743 c1cc(cnc1)c2nccc(n2)c3cccnc3Cl BF-0744 c1cc(c(cc1C=O)C#N)N2CCOCC2 BF-0745 c1ccnc(c1)c2nccc(n2)c3cccnc3Cl BF-0747 CN(C)c1ccc(cc1C#N)C=O BF-0748 CCOC(=O)c1cnc(nc1Cl)c2ccccn2 BF-0750 COC(=O)c1ccc(c(c1)N2CCCCC2)N BF-0751 CCOC(=O)c1c(nc(s1)NC)C.Cl BF-0752 COC(=O)c1cc(c(c(c1)Br)N)F BF-0753 CCOC(c1ccc(c(c1)C#N)F)OCC BF-0754 c1cc(ccc1CSc2cc(nc(n2)N)Cl)Cl BF-0755 COc1cc(cc(c1OC)OC)NC(=O)c2ccccc2N BF-0757 c1ccc(c(c1)C(=O)Nc2ccc3c(c2)OCO3)N BF-0758 CC(C)(C)OC(=O)N1CCC(CC1)NC(=O)c2ccccc2N BF-0759 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3C#N)C=O BF-0760 Cc1ccc(cc1)Sc2cc(ccc2[N+](=O)[O-])C(=O)OC BF-0761 c1cc(c(c(c1)O)[N+](=O)[O-])C(F)(F)F BF-0762 COC(=O)c1cc(c(c(c1)I)N)F BF-0763 CCOC(=O)c1cnc(nc1O)c2cccnc2 BF-0764 Cc1c(sc(n1)NC)C.Br BF-0765 COC(=O)c1ccc(c(c1)N)[N+](=O)[O-] BF-0766 c1ccc(cc1)NNC(=O)c2ccccc2N BF-0768 COc1ccc(cc1Cl)NC(=O)c2ccccc2N BF-0769 CCOC(=O)c1cnc(nc1Cl)c2cccnc2 BF-0770 CN(C)C(=O)c1ccccc1N BF-0772 CC(C(=O)O)Nc1cc(ccc1[N+](=O)[O-])C(=O)OC BF-0773 CC(C)(C)OC(=O)NC1CCCN(C1)c2ccc(cc2C(=O)OC)N BF-0774 CCOC(=O)c1c(nns1)C(C)C BF-0775 c1cc2c(cc(s2)C(=O)N)c(c1)Br BF-0776 CCOC(=O)C(=Cc1ccccc1[N+](=O)[O-])C(=O)OCC BF-0777 COc1ccc(cc1)C(=O)C(C#N)F BF-0779 c1cc(ccc1[N+](=O)[O-])Oc2nnc(s2)Br BG-0002 Cc1cc(c(cc1OC)CO)Br BG-0004 CC(C)NCC(COc1ccc(cc1)CCOC)O BG-0006 c1cc(cc(c1)Oc2nnc(s2)Br)[N+](=O)[O-] BG-0007 c1cnn2c1[nH]c(=O)cc2 BG-0010 c1cc(ccc1O)Oc2nnc(s2)Br BG-0012 c1c(c(cnc1Cl)[N+](=O)[O-])C(=O)O BG-0014 CC(C)(C#N)NCc1ccccc1 BG-0016 CCOC(=O)c1cc(ncc1N(=O)=O)Cl BG-0018 CC(C)(C#N)NCc1ccc(cc1)OC BG-0021 c1cc(ccc1N)Oc2nncs2 BG-0029 c1cc(cc(c1)Oc2nncs2)N BG-0038 CC(C)(C)OC(=O)N1CCC(CC1)Nc2cccnc2N BG-0046 CC(C)NC(C)(C)C#N BG-0047 CCOC(=O)c1cc(ncc1N)Cl BG-0053 CCOC(=O)CCCN1C(=O)c2cccc3c2c(ccc3)C1=O BG-0061 CCOC(=O)CCCCCN1C(=O)c2cccc3c2c(ccc3)C1=O BG-0062 COc1cc(ccc1CBr)C(=O)OC BG-0064 CCCNC(C)(C)C#N BG-0065 CC(C)(C)OC(=O)N1CCC(CC1)n2c3cccnc3[nH]c2=O BG-0067 CC(C)CNC(C)(C)C#N BG-0074 c1cc2c([nH]c(=O)n2C3CCNCC3)nc1.Cl.Cl BG-0075 CN1CCN(CC1)C(=S)SC BG-0081 COc1cc(ccc1CN2CCCC2)C(=O)OC BG-0084 c1cc(c(nc1)N)N BG-0085 c1cc2c(c(c1)F)N(C(=O)CC2)CCN3CCCCC3 BG-0086 CC(C)(C)OC(=O)N1CCC(CC1)n2cnc3c2cccn3 BG-0087 c1cn2ccnc2cc1C#N BG-0205 CC(=O)c1ccc2c(c1)oc(=O)n2C(=O)Oc3ccc(cc3)OC BG-0210 COC(=O)c1ccn2c(c1)ncc2I BG-0211 c1cc2c(cc1S(=O)(=O)Cl)c(=O)oc(=O)[nH]2 BG-0213 CC(=O)c1ccc2c(c1)oc(=O)[nH]2 BG-0216 CN(C)Cc1c[nH]c2c1cccn2 BG-0217 CC(C)(C)OC(=O)N1CCCCC1C=C BG-0500 c1cc(c(cc1Br)O)C=O BG-0702 c1ccc(cc1)COc2cccn3c2ncc3I BG-0703 CC1Cc2ccccc2N1C(=O)C BG-0704 CC(C)(C)OC(=O)N1CCC2(CCCCN2Cc3ccccc3)CC1 BG-0705 COc1cc(ccc1N)C(=O)N BG-0706 c1ccc(cc1)CN2CCCCC23CCNCC3 BG-0708 Cn1cc(cc1N)C#N BG-0709 Cc1c(n2ccccc2n1)CO BG-0710 c1ccc(cc1)COc2cccn3c2ncc3Br BG-0711 CCOC(=O)c1cnc2cc(nn2c1N)C BG-0713 Cn1cc(c2c1ncc(c2)C(=O)OC)C#N BG-0715 CCOC(=O)c1cc(c(nc1)C(=O)O)Cl BG-0716 CCOC(=O)c1ccc(cn1)C BG-0720 c1cc(c(nc1)C=O)F BG-0721 Cn1cc(c2c1ncc(c2)C(=O)O)C#N BG-0722 COC(=O)c1cnc(nc1)N2CCNCC2 BG-0723 COC(=O)c1ccc(cc1)CNC(=N)N BH-0007 COC(=O)c1ccc(cc1)CNc2nccc(n2)c3cccnc3 BH-0020 c1cc(cnc1)c2ccnc(n2)NCc3ccc(cc3)C(=O)O BH-0037 c1ccc2c(c1)cccc2C(=O)N3CCc4c(c5cc(ccc5[nH]4)F)C3 BH-0039 c1ccc(c(c1)N2CCNCC2)F BH-0401 CS(=O)(=O)c1ccc(c(c1)F)N BH-0405 Cn1c2ccccc2nc1c3ccc(cc3)F BH-0407 c1cc(ccc1CC(=O)O)F BH-0409 c1cc(ccc1OCC(=O)O)F BH-0410 c1cc(c(cc1F)Cl)SCC(=O)O BH-0411 c1cc(c(cc1O)F)C#N BH-0414 c1cc(c(c(c1)F)C#N)N BH-0415 c1cc(ccc1C(=O)CC#N)OC(F)(F)F BH-0416 c1ccc(cc1)COc2cccc(c2C#N)F BH-0417 c1cc2c(cc1F)nc([nH]2)C(=O)O BH-0418 c1cc(cc(c1)C(F)(F)F)c2ccc(o2)C(=O)O BH-0425 COc1ccc(c(c1)C(=O)N)F BH-0429 c1cc(c(cc1F)Cl)CC#N BH-0430 c1c(cc(c(c1Cl)CC(=O)O)Cl)C(F)(F)F BH-0431 c1cc(c(nc1)C(F)(F)F)C(=O)O BH-0434 c1cc(ccc1CN2CCOC(C2)CN)F BH-0435 c1cc2c(cc1F)C(=O)C(=O)N2 BH-0436 c1cc2c(cc1F)CC(=O)N2 BH-0437 c1cc(cc2c1cc[nH]2)F BH-0438 c1cc2c(cc1F)[nH]cc2CC#N BH-0439 c1cc(cc2c1cc([nH]2)C(=O)O)F BH-0440 Cc1ccc(cc1F)C(=O)O BH-0441 CC(C)(C)OC(=O)N1CCN(CC1)c2c(c(nc(n2)Cl)C(=O)OC)Cl BH-0700 c1cc2ncc(n2cc1F)[N+](=O)[O-] BH-0703 c1cc2ncc(n2cc1F)I BH-0704 CC(C)(C)OC(=O)NNc1c(c(nc(n1)Cl)C(=O)OC)Cl BH-0707 CC(C)(C)OC(=O)N/N=C/c1c(ncnc1Cl)N BH-0708 c1cc2cc(nc(c2nc1)Br)N BH-0712 COC(=O)c1cc(ccc1Oc2ccccc2C=O)[N+](=O)[O-] BH-0713 COC(=O)c1cc(ccc1NC2CCCCC2)[N+](=O)[O-] BH-0714 COC(=O)c1cc(ccc1SC)[N+](=O)[O-] BH-0715 c1cc2c(cc1C(=O)O)NCCO2 BH-0716 c1cc2c(cc1Cl)CCC(=O)N2 BH-0717 CC1(C=Cc2cc(c(cc2O1)[N+](=O)[O-])NC(=O)Cc3ccc(cc3)OC)C BK-0237 Cc1cc(c(c(n1)C(=O)O)C#N)C(F)(F)F BK-0700 c1cnc(c(c1C(F)F)Cl)Cl BK-0701 Cc1cc(cc(c1CC(C(=O)O)N)C)O.Cl BK-0702 c1ccc(cc1)Oc2ccc(cc2Br)C=O BK-0704 c1ccc2c(c1)c(c[nH]2)C[C@@H](C=O)NC(=O)OCC3c4ccccc4-c5c3cccc5 BK-0705 Cc1cc(c(c(c1)[N+](=O)[O-])N)C BK-0709 c1cnc(c(c1C(F)(F)F)CCl)Cl BK-0711 c1cc(ncc1OC(F)(F)F)Cl BK-0714 c1cc(nc(c1)Cl)OC(F)(F)F BK-0715 c1cc(nc(c1C(=O)O)OC(F)(F)F)Cl BK-0716 C[C@H]([C@@H](C=O)NC(=O)OCC1c2ccccc2-c3c1cccc3)OC(C)(C)C BK-0719 c1c(c(cnc1Cl)C(F)F)Cl BK-0726 CC(C)(C)OC(=O)NCCCC[C@@H](C(=O)N(C)OC)NC(=O)OCC1c2ccccc2-c3c1cccc3 BK-0728 CC(C)(C)c1cc(c(c(c1)Br)O)C=O BK-0729 c1c(ncc(n1)N2CCCCC2)C(=O)O BL-0025 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC#N BL-0037 c1ccc(cc1)c2c(n3c(n2)SCC3)C=O BL-0038 CC(C)N(c1ccc(cc1)F)C(=O)CCl BL-0050 c1cc2c(cc1C(F)(F)F)ncc3c2NCCNC3=O BL-0778 c1cc2c(c(c1)Cl)ncc3c2NCCNC3=O BL-0779 c1cc(c(c(c1)F)CBr)C(F)(F)F BM-0758 COc1ccc(c(n1)C(=O)O)F BM-0774 c1c(cnc(c1C(F)(F)F)Cl)C(=O)O BS-0001 CCOC(=O)[C@H](Cc1c[nH]c2c1cc(cc2)OCc3ccccc3)NC(=O)OC(C)(C)C BS-0004 Cc1cc(nn1c2ccccc2C(=O)O)C(=O)OC BS-0009 Cc1cc(nn1c2ccccc2C(=O)OC(C)(C)C)C(=O)O BS-0010 Cc1cc(nn1c2ccccc2C=O)C(=O)OC BS-0011 Cc1cc(nn1c2ccccc2C(=O)OC(C)(C)C)C=O BS-0012 Cc1cc(nn1c2ccccc2C(=O)OC(C)(C)C)NC(=O)OCc3ccccc3 BS-0016 Cc1cc(nn1c2ccccc2CO)C(=O)OC BS-0018 Cc1cc(nn1c2ccccc2N)C(=O)OC BS-0019 Cc1cc(nn1c2ccc(cc2)N)C(=O)OC BS-0022 Cc1cc(nn1c2ccccc2C(=O)OC(C)(C)C)CO BS-0023 Cc1cc(nn1c2ccccc2[N+](=O)[O-])C(=O)O BS-0024 CC1(Oc2cc(cc(c2C(=O)O1)OS(=O)(=O)C(F)(F)F)OS(=O)(=O)C(F)(F)F)C BS-0026 CCOC(=O)c1cn(c2ccccc2c1=O)Cc3ccc(cc3)OC BS-0027 Cc1cc(nn1c2ccccc2C#N)C(=O)OC BS-0028 B(c1ccc(cc1)NS(=O)(=O)C)(O)O BS-2000 B(c1ccc(nc1)c2ccccc2)(O)O BS-2016 Cc1c2ccccc2ccc1Br BS-2034 Cc1cc(c(nc1)N)I BS-2036 c1ccc(cc1)COc2cc(ncn2)Cl BS-2064 B(c1ccc2ccccc2c1C)(O)O BS-2088 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCCN(C)C BS-2119 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)C(=O)NCCCN(C)C BS-2130 c1cc(c(=O)[nH]c1)S(=O)(=O)N2CCCC2 BS-3000 c1ccc(cc1)c2nc(on2)C3(CCCCC3)N.Cl BS-3001 Cc1ccc(cc1)Cn2cc(c3c2cccc3)C(=O)O BS-3002 COC(=O)c1c(cc(=O)n2c1CCCC2)O BS-3003 c1cc(ccc1c2nc(on2)CC3CCNCC3)F.Cl BS-3004 c1cscc1c2nc(on2)C3(CCCCC3)N.Cl BS-3005 c1cnc(cn1)c2nc(on2)C3(CCCCC3)N.Cl.Cl BS-3006 c1cnccc1c2nc(on2)C3(CCCCC3)N.Cl.Cl BS-3007 c1cc(cnc1)c2nc(on2)C3CCCCN3.Cl.Cl BS-3008 c1cnccc1c2nc(on2)C3CCCCN3.Cl.Cl BS-3009 COc1ccc(cc1)c2nc(on2)C3CCCN3.Cl BS-3010 c1cc(ccc1c2nc(on2)C3CCCN3)F.Cl BS-3011 CN(C(=O)C1CC(=O)N(C1)c2ccc(cc2)OC)OC BS-3012 COc1ccc(cc1)CN2CC(CC2=O)C#N BS-3013 c1cc(c(cc1F)Cl)CN2CC(CC2=O)C(=O)O BS-3014 CCc1ccc(cc1)CN2CC(CC2=O)C(=O)O BS-3015 Cc1ccc(c(c1)N2CC(CC2=O)C(=O)O)F BS-3016 c1cc2c(c(c1)N3CC(CC3=O)C(=O)O)CCCC2 BS-3017 c1cc(sc1)C(=O)N2CCC(CC2)C(=O)NN BS-3019 CCN1CCn2c(n[nH]c2=O)C1=O BS-3020 Cc1cccc(c1)CN2CCn3c(n[nH]c3=O)C2=O BS-3021 c1ccc(c(c1)CN2CCn3c(n[nH]c3=O)C2=O)F BS-3022 c1cc(cc(c1)N)C(=O)N/N=C/2\CCCN2 BS-3023 CN(C(=O)c1cc(n[nH]1)c2ccccc2)OC BS-3024 c1ccc(c(c1)n2c(cnn2)CN3CCC(CC3)C(=O)O)F BS-3025 COc1ccccc1c2c3[nH]c(=O)c4ccccc4n3nn2 BS-3027 c1ccc2c(c1)N(C(=O)CNS2(=O)=O)Cc3ccc(cc3)F BS-3028 CCOc1ccc(cc1Cl)C2C(=C(NC(=O)N2)CCl)C(=O)OCC BS-3029 c1cc(cc(c1)Cl)COc2cccc3c2cc([nH]3)C(=O)O BS-3030 Cc1ccc2c(c1)c(c(n2C)C(=O)OC)N BS-3031 CCOC(=O)c1c(c2cc(c(cc2[nH]1)OC)OC)N BS-3032 c1cc(cc(c1)F)c2nc(on2)c3cccnc3N4CCC(CC4)C(=O)O BS-3033 c1cc(cc(c1)F)Cn2cc(nn2)/C(=N/O)/N BS-3035 Cc1c(nnn1Cc2cccc(c2)F)/C(=N/O)/N BS-3036 CCN1c2ccccc2C(=O)CS1(=O)=O BS-3037 C1CCc2c(c(=O)[nH]c(=S)[nH]2)C1 BS-3038 c1c([nH]c(=S)[nH]c1=O)C(F)(F)F BS-3039 c1ccc(cc1)c2nc(on2)CN3CCC(CC3)C(=O)O BS-3040 COc1ccc(cc1NC(=O)N)C(=O)O BS-3041 COc1cc(nc2c1cc(cc2F)F)C(=O)O BS-3042 c1cc(ccc1C2=NC3(CCCCC3)NC2=S)Cl BS-3043 c1cc(ccc1C2=NC3(CCCC3)NC2=S)Cl BS-3045 CCOCc1cnc(nc1N)C BS-3046 Cc1cc(cc2c1nc(cc2OC)C(=O)O)F BS-3047 COc1cc(nc2c1cccc2F)C(=O)O BS-3048 c1cc2c(cc1F)c(=O)c3c([nH]2)CCNC3 BS-3049 c1ccc(c(c1)CNC(=O)c2c(c(sn2)C(=O)O)N)Cl BS-3050 Cc1cccc(c1)C2=NC3(CCCCC3)NC2=S BS-3051 COCCc1nc(on1)c2ccc(nc2)Cl BS-3052 CN1CCC2(CC1)NC(=S)C(=N2)c3ccccc3 BS-3053 c1cc2c(cc1c3cc4c(=O)[nH]ccn4n3)OCO2 BS-3055 Cn1ccc2c1c(=O)[nH]cc2 BS-3056 c1ccc2c(c1)c(c(cn2)C#N)N3CCC(CC3)C(=O)O BS-3057 CC(C)(C)c1nc(on1)c2ccnc(c2)Cl BS-3058 CCN1c2ccc(cc2C(=O)NC13CCNCC3)C BS-3060 c1ccc(cc1)C2=NNS(=O)(=O)c3c2cccc3 BS-3061 c1ccc(cc1)c2cc([nH]n2)C(=O)N3CCC(CC3)N BS-3063 Cc1ccc(cc1C)n2c(=O)c3c(ccs3)[nH]c2=S BS-3064 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=S)C(=N2)c3ccccc3 BS-3065 CCn1ccc2c1c(=O)[nH]cc2 BS-3066 Cc1nc(on1)c2ccn3c(c2)nnc3CC(=O)O BS-3067 COCCn1ccc2c1c(=O)[nH]cc2 BS-3068 CCc1nc(on1)c2ccn3c(c2)nnc3CC(=O)O BS-3069 C=CCn1ccc2c1c(=O)[nH]cc2 BS-3070 c1c[nH]c(=O)c2c1ccn2CC3CC3 BS-3071 Cc1ccc(cc1)C2=NC3(CCNCC3)NC2=O BS-3072 Cc1cc(ccc1Br)n2c(c(nn2)C(=O)O)C BS-3073 c1cc(cc(c1)F)n2cc(nn2)c3nc(on3)C(=O)NN BS-3074 c1ccc(cc1)c2cc3c(=S)[nH]ccn3n2 BS-3075 c1cc(c2n[nH]c(=O)n2c1)c3nc(no3)c4ccc(cc4)Cl BS-3076 COC(=O)c1c(n(nn1)c2ccc(cc2)F)N BS-3077 c1cc(ccc1c2cc3c(=O)[nH]ccn3n2)F BS-3078 CC(C)c1ccc(cc1)c2cc3c(=O)[nH]ccn3n2 BS-3079 c1cc(cc(c1)F)c2cc3c(=O)[nH]ccn3n2 BS-3080 c1cc2c(cc1Br)c(cc(=O)[nH]2)C(=O)O BS-3081 COc1ccccc1n2c(cc(=O)[nH]c2=O)N BS-3082 CCOC(=O)c1c[nH]nc1S(=O)(=O)N2CCN(CC2)c3ccc(cc3)Cl BS-3084 CCN1CCN(CC1)S(=O)(=O)c2c(c[nH]n2)C(=O)OCC BS-3085 CCOC(=O)c1c[nH]nc1S(=O)(=O)N2CCN(CC2)C(C)C BS-3086 CCOC(=O)c1c[nH]nc1S(=O)(=O)N2CCN(CC2)C BS-3087 c1cc(c(cc1N2CC(CC2=O)C(=O)O)Cl)F BS-3088 CNC(=O)Nc1cccc(c1)F BS-3089 c1ccc(cc1)C2=NC3(CCNCC3)NC2=O BS-3090 c1c(c(cc(c1F)Cl)F)C(=O)N2CCC(CC2)C(=O)NN BS-3091 c1([nH]c(nn1)N)C(=O)O BS-3092 COc1cccc(c1)c2[nH]c(c(n2)c3ccc(cc3)F)S BS-3093 Cc1ccc(cc1)c2nc(on2)Cn3c(=O)c4ccccc4[nH]c3=O BS-3094 CC(C)(C)OC(=O)N1CCN(CC1)c2cc(n[nH]2)c3ccccc3 BS-3095 CCOC(=O)c1c(n(c(=S)s1)CCc2ccccc2)N BS-3097 Cc1c(nnn1c2ccc(cc2)F)C(=O)O BS-3099 CCOc1ccc(cc1)c2cc3c(=O)[nH]ccn3n2 BS-3100 c1cc(sc1)c2cc3c(=O)[nH]ccn3n2 BS-3101 c1ccc(cc1)c2c(c3c(=O)[nH]ccn3n2)C=O BS-3102 COc1ccc(cc1)c2c(c3c(=O)[nH]ccn3n2)C=O BS-3103 c1cc(cc(c1)F)c2cc3c(nccn3n2)Cl BS-3104 Cc1ccc(cc1)c2c(c3c(nccn3n2)Cl)C=O BS-3105 c1cn2c(c3c(n2)CCCC3)c(n1)N4CCCC(C4)C(=O)O BS-3106 c1cn2c(c3c(n2)CCCC3)c(n1)N4CCNCC4.Cl BS-3107 c1ccc(cc1)C2=NC3(CCCC3)NC2=S BS-3108 CC1(NC(=O)C(=N1)c2ccc(cc2)F)C BS-3110 c1ccc2c(c1)-c3c(c([nH]n3)C(=O)O)CO2 BS-3111 c1ccc-2c(c1)CCc3c2n[nH]c3C(=O)O BS-3112 Cc1nc(on1)c2cccnc2n3cc(nc3)C(=O)O BS-3113 c1cc(cc(c1)N2C(=O)CC(=N2)C(=O)O)N BS-3115 CC(=O)c1c(c2ccccc2o1)N BS-3116 CC(=O)Cn1c(c(nn1)C(=O)OC)C(=O)OC BS-3117 COc1cccc(c1)Cn2c(=O)c3c(c4ccccc4o3)[nH]c2=S BS-3118 Cc1ccc(cc1)NCc2ccccc2O BS-3119 c1ccc2c(c1)C(=NC3(N2)CCCCCC3)S BS-3120 c1ccc2c(c1)C(=NC3(N2)CCCC3)S BS-3121 CN1CCN(CC1)C(=O)c2cnc3ccc(cc3c2O)F BS-3122 c1ccc2c(c1)C(=NC3(N2)CCCCC3)S BS-3123 COC(=O)c1c(n(nn1)CC(=O)c2ccccc2)C(=O)OC BS-3124 CCOC(=O)c1c(n(c(=S)s1)c2ccccc2)N BS-3127 Cc1ccc(n1C)/C(=N/O)/N BS-3128 c1cc(cc(c1)F)c2cc([nH]n2)C(=O)O BS-3129 Cc1nc(on1)C2=NNC(=O)CC2 BS-3130 COc1ccc(cc1OC)c2c(c3c(nccn3n2)Cl)C=O BS-3131 CCCCCn1cc(c2c1cccc2)C(=O)O BS-3132 c1c2c(cc3c1OCO3)[nH]c(=O)n(c2=O)CCCC(=O)O BS-3133 c1c2c(cc3c1OCO3)[nH]c(=O)n(c2=O)CCC(=O)O BS-3134 c1cc(ccc1c2nc(on2)CN3CCNCC3)F BS-3135 CCOC(=O)c1c(n[nH]c1N)c2cccc(c2)Cl BS-3136 Cc1cc(cc(c1)n2c(=O)c3ccc(cc3[nH]c2=O)C(=O)O)C BS-3137 c1csc2c1[nH]c(=O)n(c2=O)CCCC(=O)O BS-3138 COc1ccc(cc1OC)c2c(c[nH]n2)C(=O)O BS-3139 Cc1cc([nH]n1)CCl.Cl BS-3140 c1c([nH]cn1)CCN.Cl.Cl BS-3141 COC(=O)c1c(c2cc(ccc2[nH]1)Br)N BS-3142 COc1ccc(cc1F)n2c(cnn2)CN3CCNCC3.Cl.Cl BS-3143 c1ccc(c(c1)n2c(cnn2)CN3CCNCC3)Cl.Cl.Cl BS-3144 Cc1nc(on1)c2cccnc2N3CCC(CC3)N.Cl.Cl BS-3145 Cc1ccc(cc1)c2nc(on2)C3CCNCC3.Cl BS-3146 COc1ccc(cc1)c2nc(on2)C3CCNCC3.Cl BS-3147 COc1ccccc1c2nc(on2)C3CCNCC3.Cl BS-3148 COC(=O)c1c(n(nn1)CCN2C(=O)c3ccccc3C2=O)C(=O)OC BS-3149 Cc1ccccc1n2c(cnn2)CN3CCNCC3.Cl.Cl BS-3151 COc1ccccc1n2c(cnn2)CN3CCNCC3.Cl.Cl BS-3152 c1cc(c(=O)[nH]c1)c2nc(no2)c3ccncc3 BS-3153 c1ccc(c(c1)n2c(cnn2)CN3CCNCC3)F.Cl.Cl BS-3154 c1cc(c(=O)[nH]c1)c2nc(no2)c3ccsc3 BS-3155 c1ccc(cc1)n2c(cnn2)CN3CCNCC3.Cl.Cl BS-3156 c1c(nnn1CCN)C(=O)O.Cl BS-3158 c1ccc(cc1)c2cn3c(cc(n3)C(=O)O)c(=O)[nH]2 BS-3160 CCOC(=O)c1c(n(nn1)CC(=O)c2ccc(cc2)F)C(=O)OCC BS-3161 COC(=O)c1c(n(nn1)CC(=O)c2ccc(cc2)F)C(=O)OC BS-3162 c1cc(ccc1c2nc(on2)CCN)Br.Cl BS-3163 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc(cc2)Cl)C(=O)OCC BS-3164 c1cc(ccc1c2ccc3n[nH]c(=O)n3n2)Cl BS-3165 c1ccc(c(c1)c2ccc(nn2)N3CCC(C3)N)F BS-3166 c1ccc(c(c1)c2ccc(=O)[nH]n2)F BS-3167 c1cc(cc(c1)F)c2ccc(nn2)N3CCC(CC3)N BS-3168 c1ccc(c(c1)c2ccc(=O)[nH]n2)Cl BS-3169 Cc1c(nnn1Cc2cccc(c2)F)C(=O)O BS-3170 CC(C)(C)OC(=O)N1CCN(CC1)CC(=O)NN BS-3171 c1cc2nc(cn2cc1F)CCl BS-3173 CCOC(=O)[C@H](C(C)C)N BS-3175 CC(C)(C)OC(=O)N1CCC(CC1)c2nnc3n2CCCCC3 BS-3177 CC(C)(C)OC(=O)N1CCCC1c2nnc3n2CCCCC3 BS-3178 C1CCc2nnc(n2CC1)C3CCCNC3.Cl.Cl BS-3179 c1cc(=O)n2c(c1C(=O)O)CCCCC2 BS-3180 c1cc(ccc1C(=N)N)N.Cl BS-3189 c1cc(cc(c1)Br)c2nc(on2)CCl BS-3194 c1cscc1c2nc(on2)CCl BS-3195 c1cc(ccc1Cn2ccn3c(c2=O)c4c(n3)CCCC4)C(=O)O BS-3200 C1CCc2c(n[nH]c2C(=O)O)CC1 BS-3201 C=CCn1c(=O)c2ccccc2[nH]c1=O BS-3202 Cc1c(c(=O)[nH]c(n1)c2ccc(cc2)Cl)CCO BS-3206 Cc1c(c(=O)[nH]c(n1)c2cccc(c2)Cl)CCO BS-3208 c1cc(c(cc1Cl)NC(=O)CCCl)O BS-3209 Cc1ccc2c(c1)c(=O)n3cccc(c3n2)C(=O)O BS-3210 COc1ccc2c(c1)cc(c(=O)[nH]2)C=O BS-3212 Cc1ccc2cc(c(=O)[nH]c2c1)CNc3ccccc3 BS-3213 COc1cc2cc(c(=O)[nH]c2cc1OC)C=O BS-3214 c1c2cc3c(cc2[nH]c(=O)c1C=O)OCCO3 BS-3215 c1c2cc3c(cc2[nH]c(=O)c1C=O)OCO3 BS-3216 COc1ccc(cc1)NCc2cc3ccc(cc3[nH]c2=O)OC BS-3217 COc1ccc2cc(c(=O)[nH]c2c1)CNc3ccccc3 BS-3218 c1cc(c(nc1)NN)S(=O)(=O)N2CCCC2 BS-3222 c1cc(c2n[nH]c(=O)n2c1)S(=O)(=O)N3CCCC3 BS-3223 c1cc(c2n[nH]c(=O)n2c1)S(=O)(=O)N3CCN(CC3)c4ccc(cc4)F BS-3224 c1cc(c2n[nH]c(=O)n2c1)S(=O)(=O)N3CCOCC3 BS-3225 c1cc(c2n[nH]c(=O)n2c1)S(=O)(=O)N3CCCCCC3 BS-3226 Cc1ccc(cc1C)c2nc(on2)c3c4ccccc4c(=O)[nH]n3 BS-3227 c1c(cnc(n1)NN)C(=O)N2CCCC2 BS-3228 COc1ncc(cn1)C(=O)O BS-3229 c1cc(ccc1NS(=O)(=O)c2ccc(nc2)NN)F BS-3230 c1cn2c(c(n1)N3CCC(CC3)N)n[nH]c2=O BS-3233 c1cc(=O)[nH]cc1S(=O)(=O)N2CCOCC2 BS-3237 CCc1c(sc(n1)n2cccc2)C(=O)O BS-3239 CCCc1c(sc(n1)n2cccc2)C(=O)O BS-3240 CNS(=O)(=O)c1c2ccccc2sc1C(=O)OC BS-3241 c1ccn(c1)c2c3cccnc3sc2C(=O)O BS-3242 COc1ccc2c(c1)c(cc(n2)C(=O)O)OC BS-3247 CCOc1ccc2c(c1)c(cc(n2)C(=O)O)OC BS-3248 Cc1ccc2c(c1)c(cc(n2)C(=O)O)OC BS-3249 CCOc1cc(nc2c1cc(cc2)OC)C(=O)O BS-3250 CCOc1cc(nc2c1cc(cc2)C)C(=O)O BS-3251 CCOc1cc(nc2c1cc(cc2)F)C(=O)O BS-3252 CCOc1cc(nc2c1cccc2)C(=O)O BS-3253 CCOc1cc(nc2c1cc(cc2F)F)C(=O)O BS-3254 COc1cc(nc2c1cc(cc2)F)C(=O)O BS-3255 c1ccc(cc1)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F BS-3256 CCn1cc(c(=O)c2c1cccc2)C(=O)O BS-3257 CCCn1cc(c(=O)c2c1cccc2)C(=O)O BS-3258 CCCn1cc(c(=O)c2c1ccc(c2)F)C(=O)O BS-3260 c1cc2c(nc1)N(N=C(S2(=O)=O)C(=O)O)c3ccc(cc3)F BS-3262 Cc1ccc(cc1)c2nc(on2)c3c[nH]c4c3cccc4 BS-3263 CCOC(=O)c1c(c(cs1)c2ccccc2)N BS-3264 CCOC(=O)c1c(c2c(cccc2s1)F)N BS-3265 COC(=O)c1c(c(cs1)c2ccccc2F)N BS-3266 COC(=O)c1c(c(cs1)c2ccccc2Cl)N BS-3267 c1cc2n[nH]c(=O)n2cc1S(=O)(=O)N3CCSCC3 BS-3269 c1cc2c(nc1)NN=C(S2(=O)=O)C(=O)N3CCCC3 BS-3272 c1cc2c(cc1Cl)NN=C(S2(=O)=O)C(=O)N3CCOCC3 BS-3273 c1ccc2c(c1)NN=C(S2(=O)=O)C(=O)N3CCCCCC3 BS-3274 CNS(=O)(=O)c1cccnc1Cl BS-3275 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cccnc2Cl BS-3276 CCNS(=O)(=O)c1cccnc1Cl BS-3277 c1ccc2c(c1)C(=O)N(C2=O)c3cc([nH]n3)C(=O)O BS-3279 Cc1c(cnc(n1)OC)C(=O)O BS-3280 c1cc(sc1)c2nc(on2)CN3CCCC(C3)N.Cl BS-3282 Cc1nc(nn1c2ccccc2)C(=O)O BS-3283 CCCc1c(sc(n1)n2cccc2)CO BS-3285 CC(=O)Cc1nc(no1)c2ccccc2 BS-3291 COc1ccc(cc1)COc2ccc(cc2)C=O BS-3292 COC(=O)c1c2n(nc1C(=O)OC)CCCC2 BS-3293 COC(=O)c1c2n(nc1CO)CCCC2 BS-3294 COC(=O)c1c2n(nc1CO)CCC2 BS-3295 COC(=O)c1c2n(nc1C(=O)OC)CCC2 BS-3296 Cc1ccc(cc1)S(=O)(=O)Cc2c(c3n(n2)CCCC3)C(=O)OC BS-3297 c1cnccc1c2nc(on2)CC3CCNCC3 BS-3298 c1cc(cc(c1)F)c2nc(on2)C3CCCCN3 BS-3299 c1cc(c2nncn2c1)S(=O)(=O)Nc3ccc(c(c3)F)F BS-3300 Cc1nnc2n1cccc2S(=O)(=O)Nc3ccc(cc3)F BS-3301 COc1ccc(cc1)c2nc(on2)CC3CCNCC3.Cl BS-3303 COc1cc2c(cc1OC)[nH]cc(c2=O)C(=O)c3ccccc3 BS-3304 c1ccc(c(c1)N2CCN(CC2)C(=O)CN)F.Cl BS-3305 C1CC/C(=C(\C#N)/C(=O)N)/NCC1 BS-3306 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)OC)CCl BS-3308 CCOC(=O)C1=C(NC(=O)NC1c2ccccc2Cl)CCl BS-3309 Cc1ccc(cc1)c2nc(on2)c3cccnc3N4CCC(CC4)C(=O)O BS-3310 c1cc(cc(c1)Cl)c2nc(on2)c3cccnc3N4CCC(CC4)C(=O)O BS-3311 COC(=O)c1c(n(nn1)c2ccccc2)N BS-3312 c1ccc(cc1)COc2ccccc2c3nc(on3)CCl BS-3313 c1ccc(cc1)COc2ccc(cc2)c3nc(on3)CCl BS-3314 c1cc(ncc1Br)NC(=S)N BS-3315 c1cc(ccc1c2cc3c(=O)n(ccn3n2)C/C(=N/O)/N)F BS-3316 c1cc(sc1)c2cc3c(=O)n(ccn3n2)C/C(=N/O)/N BS-3317 CSc1cccc(c1)NC(=O)N BS-3319 COc1ccc(cc1OC)c2cc3c(nccn3n2)N4CCC(CC4)C(=O)O BS-3322 CCOC(=O)c1ccc(cc1)NC(=O)N BS-3323 CC(C)(C)c1ccc(cc1)C2=NC3(CCN(CC3)C(=O)OC(C)(C)C)NC2=O BS-3325 COc1cccc(c1)CNC(=O)CC#N BS-3326 c1cc(ccc1C2=NC3(CCCCC3)NC2=S)F BS-3327 COc1ccc(cc1)C2=NC3(CCCCC3)NC2=S BS-3328 COC(=O)c1cc(=O)c2ccccc2[nH]1 BS-3329 c1ccc(cc1)C2=NC3(CCCCC3)NC2=S BS-3330 Cc1ccc(c(c1)C)n2c(=O)c3c(ccs3)[nH]c2=S BS-3332 c1ccc(cc1)NC(=O)c2cccc(c2)n3cc[nH]c3=S BS-3333 Cc1ccc(o1)CNC(=O)c2cccc(c2)n3cc[nH]c3=S BS-3334 c1cc(cc(c1)n2cc[nH]c2=S)C(=O)NCc3ccco3 BS-3335 CCCCNC(=O)c1cccc(c1)n2cc[nH]c2=S BS-3336 CCOc1ccc(cc1OC)/C(=N/O)/N BS-3337 COc1ccc(cc1)S(=O)(=O)CC#N BS-3338 c1c(c(nc(n1)S)N)C(=O)N BS-3339 c1ccc(cc1)CN2CC(CC2=O)NC(=O)NC3CC(=O)N(C3)Cc4ccccc4 BS-3340 CCOC(=O)c1cn(nc1S(=O)(=O)N2CCCCC2)C BS-3341 CCOC(=O)c1c[nH]nc1S(=O)(=O)N2CCOCC2 BS-3342 c1c(n[nH]c1C(=O)N2CCCCC2)C3CC3 BS-3343 Cc1ccc(cc1C)n2c(c(cn2)C(=O)O)n3cccc3 BS-3344 COc1ccc(cc1)c2[nH]c(c(n2)c3ccccc3)S BS-3345 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=O)C(=N2)c3ccc(cc3)Cl BS-3346 Cc1c(nnn1c2ccc(cc2)Cl)C(=O)NN BS-3347 c1cc(cc(c1)Cl)c2nc(on2)c3cccnc3NN BS-3348 Cc1c(c([nH]c1C(=O)NCC(OC)OC)C)C(=O)C BS-3349 c1ccc(cc1)c2nc(on2)Cn3c(=O)c4ccccc4[nH]c3=O BS-3350 c1ccc(cc1)CC(=S)N2CCOCC2 BS-3351 Cc1cc([nH]c(=O)c1c2nc(no2)c3ccccc3)C BS-3352 c1cc(oc1C(=O)N2CCCCC2)[N+](=O)[O-] BS-3353 c1ccc(cc1)c2nc(on2)c3cccnc3NN4C(=O)CCC4=O BS-3354 CCc1ccc(cc1)n2c(cc(c(c2=O)C#N)C)C BS-3355 CCCC(=O)c1cc2cccc(c2oc1=O)OC BS-3359 CCOC(=O)c1c(n(c(=S)s1)c2cccc(c2)C(F)(F)F)N BS-3360 COc1ccc(cc1)c2c(cn[nH]2)C(=O)O BS-3361 c1ccc2c(c1)[nH]c(n2)C(Cc3ccc(cc3)Cl)C(=S)N BS-3362 CN(C)c1ccc(cc1)CC(c2[nH]c3ccccc3n2)C(=S)N BS-3363 COc1ccc(cc1)CC(c2[nH]c3ccccc3n2)C(=S)N BS-3364 COc1cccc(c1)c2cc3n(n2)C(CNC3=O)O BS-3365 Cc1ccccc1c2cc3c(=O)[nH]ccn3n2 BS-3366 CC1(NC(=S)C(=N1)c2ccccc2)C BS-3368 CCOC(=O)c1c(c(sc1N)C(=O)N2CCOCC2)C BS-3369 c1ccc(cc1)C2CC2C(=O)NN BS-3370 c1cc(ccc1C2=NC3(CCCCC3)NC2=O)Cl BS-3371 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc[nH]c3=O BS-3372 c1cc(=O)[nH]cc1S(=O)(=O)N2CCCCCC2 BS-3373 CC1CCN(CC1)S(=O)(=O)c2ccc[nH]c2=O BS-3374 CN(c1ccccc1)S(=O)(=O)c2cccnc2Cl BS-3375 CCc1nnc2n1cccc2S(=O)(=O)Nc3ccccc3 BS-3376 CC(C)c1ccc(cc1)NS(=O)(=O)c2cccn3c2nnc3 BS-3377 CCc1nnc2n1cccc2S(=O)(=O)Nc3cccc(c3)F BS-3378 Cc1cccc(c1)NS(=O)(=O)c2cccn3c2nnc3C BS-3379 COc1ccc(c(c1)OC)C(=O)ON2C(=O)CCC2=O BS-3380 COc1ccc(cc1)N2CC(CC2=O)C(=O)Nc3ccc(cc3)C(=O)O BS-3381 COc1ccc(cc1)N2CC(CC2=O)C(=O)Nc3cccc(c3)C(=O)O BS-3382 C1CCNC(C1)C(=O)N.Cl BS-3383 CCOc1ccc(cc1)C2C(=C(NC(=O)N2)CCl)C(=O)OCC BS-3384 CCOC(=O)C1=C(NC(=O)NC1c2ccccc2OC)CCl BS-3385 c1ccc(cc1)Cn2c(c(nn2)C(=O)NN)c3cccnc3 BS-3386 CCCCOc1ccccc1c2cc([nH]n2)C(=O)O BS-3387 CCCNC(=S)Nc1ccc(cc1)OCC BS-3388 CCCc1c([nH]c(=S)[nH]c1=O)C BS-3389 c1cc(ccc1C2=NC3(CCNCC3)NC2=O)Cl BS-3390 Cc1ccc(cc1)c2c(c[nH]n2)C(=O)O BS-3391 COc1ccc(cc1)c2nc(on2)c3ccc(nc3)SCC(=O)O BS-3392 COc1ccc(cc1)c2cc([nH]n2)C(=O)N3CCC(CC3)N BS-3393 c1c[nH]c2c1cc[nH]c2=O BS-3394 Cc1ccc(cc1C)C2=NC3(CCN(CC3)C(=O)OC(C)(C)C)NC2=S BS-3395 c1cc2c(cc1Cl)NC3(CCNCC3)NC2=O BS-3396 CCOc1ccc(cc1)S(=O)(=O)c2c(c3ccc(cc3[nH]c2=O)C(=O)O)O BS-3397 CN1c2cc(ccc2C(=O)NC13CCNCC3)F BS-3398 Cc1ccc(cc1)S(=O)(=O)c2c(c3ccc(cc3[nH]c2=O)C(=O)O)O BS-3399 CCN1c2cc(ccc2C(=O)NC13CCNCC3)F BS-3400 c1ccc2c(c1)cccc2c3cc4c(=O)[nH]ccn4n3 BS-3401 CC(C)(C)c1ccc(cc1)C2=NC3(CCN(CC3)C(=O)OC(C)(C)C)NC2=S BS-3402 c1cc(c(nc1)S)c2nc(no2)c3ccc(cc3)F BS-3403 Cc1c(cnn1c2ccc(cn2)c3nc(no3)c4ccc(cc4)F)C(=O)O BS-3404 COc1ccc(cc1OC)c2nc(on2)c3cn(cn3)Cc4ccc(cc4)N BS-3405 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=S)C(=N2)c3ccc(cc3)F BS-3406 c1ccc(cc1)c2nc(on2)c3ccc(nc3)SCC(=O)O BS-3407 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=S)C(=N2)c3ccc(cc3)OC BS-3408 Cc1cccc(c1)C2=NC3(CCN(CC3)C(=O)OC(C)(C)C)NC2=S BS-3409 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=O)C(=N2)c3ccc(cc3)OC BS-3410 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=S)C(=N2)c3cccc(c3)F BS-3411 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2)Cl)CCl BS-3412 c1cc(ccc1Cn2cnc3c(c2=O)cn[nH]3)Cl BS-3413 c1ccc(c(c1)Cn2c(=O)c3c(ccs3)[nH]c2=S)F BS-3414 c1ccc2c(c1)cccc2c3cc4c(=O)[nH]ncn4n3 BS-3415 c1ccc(cc1)CNC(=O)c2cccc(c2)n3cc[nH]c3=S BS-3416 c1cc(cc(c1)Cl)c2nc(on2)c3cccn4c3n[nH]c4=O BS-3417 Cc1cccc(c1)c2nc(on2)c3cccn4c3n[nH]c4=O BS-3418 Cc1cc(ccc1n2c(=O)c3c(ccs3)[nH]c2=O)F BS-3419 CC(C)(C)c1ccc(cc1)C(=O)N2CCNCC2.Cl BS-3420 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)CN.Cl BS-3421 CCOc1ccccc1C(=O)NC2CCCNC2.Cl BS-3422 CCOc1ccccc1C(=O)NCC2CCNCC2.Cl BS-3423 CC(C)(C)c1ccc(cc1)C(=O)NCC2CCCNC2.Cl BS-3424 CC(C)(C)c1ccc(cc1)C(=O)NCCN.Cl BS-3425 CC(C)(C)c1ccc(cc1)C(=O)N2CCCC(C2)N.Cl BS-3426 Cc1ccccc1c2nc(on2)Cn3cccc3C(=O)O BS-3427 CCOC(=O)c1ncn(n1)CC(=O)c2ccc(cc2)Cl BS-3428 CC(C)(C)OC(=O)NCC(=O)NNC(=O)c1ccc(cc1)Cl BS-3429 CCOC(=O)c1ccc(cc1)NC(=O)C2CC(=O)N(C2)c3ccc(cc3)Cl BS-3430 CCOC(=O)c1cccc(c1)NC(=O)C2CC(=O)N(C2)c3ccc(cc3)Cl BS-3431 CC(C)(C)c1ccc(cc1)C(=O)NC2CCNCC2.Cl BS-3432 CC(C)(C)c1ccc(cc1)C(=O)NCC2CCNCC2.Cl BS-3433 COc1ccc(cc1)N2CCN(CC2)C(=O)CN.Cl BS-3434 CCOc1ccccc1N2CCN(CC2)C(=O)CN.Cl BS-3435 COc1ccccc1N2CCN(CC2)C(=O)CN.Cl BS-3436 COc1ccccc1CN2CC(CC2=O)C(=O)N BS-3437 COC(=O)c1c(c2c(cccc2s1)F)S(=O)(=O)N3CCOCC3 BS-3438 CCOC(=O)C(CCc1ccccc1)(C(=O)OCC)NC(=O)C BS-3439 Cc1cccc(c1)CN2CC(CC2=O)C(=O)O BS-3440 c1cc(cc(c1)Cl)n2cc(nn2)/C(=N/O)/N BS-3441 c1cc(sc1)CCn2c(=O)c3c(ccs3)[nH]c2=S BS-3442 Cc1ccc(c(c1)c2cc3c(=O)n(ncn3n2)CC(=O)O)C BS-3443 Cc1cc(cc(c1)n2c(=O)c3c(ccs3)[nH]c2=O)C BS-3444 Cc1cccc(c1)c2c3[nH]c(=O)c4ccccc4n3nn2 BS-3445 Cc1ccccc1c2c3[nH]c(=O)c4ccccc4n3nn2 BS-3446 CCCCOc1ccc(cc1)c2cc3c4n[nH]c(=S)n4ccn3n2 BS-3447 c1cc(ccc1Cn2c(=O)c3c(ccs3)[nH]c2=O)F BS-3448 CSc1ncc(c(n1)N)c2ccc(cc2)Cl BS-3450 COc1ccc(cc1)c2cc3n(n2)C(CNC3=O)O BS-3452 c1cc(cc(c1)F)c2c(c3c(=O)[nH]ccn3n2)C=O BS-3453 Cc1ccc(cc1)c2c(c3c(=O)[nH]ccn3n2)C=O BS-3454 c1cn2c(c3c(n2)CCCC3)c(n1)N4CCC(CC4)C(=O)O BS-3455 c1ccc(cc1)C2=NC3(CCCC3)NC2=O BS-3456 CCOC(=O)c1c(c(sc1N)C(=O)N2CCCC2)C BS-3457 COC(=O)c1ccc(cc1)NCc2ccccc2O BS-3458 CCOC(=O)c1cccc(c1)NCc2ccccc2O BS-3459 CCOC(=O)c1c(n(c(=S)s1)c2ccc(cc2)[N+](=O)[O-])N BS-3460 CSc1ncc(c(n1)N)C(=O)NCc2ccccc2 BS-3461 CC12CC(c3cccc(c3O1)OC)NC(=S)N2c4ccc(cc4)Cl BS-3462 c1cc(c(=O)[nH]c1)c2nc(no2)c3cnccn3 BS-3463 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc(c(c2)OC)OC)C(=O)OCC BS-3464 COC(=O)c1c(n(cn1)CC(=O)c2ccc(cc2)F)C(=O)OC BS-3465 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc(cc2)C)C(=O)OCC BS-3466 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc(cc2)OC)C(=O)OCC BS-3467 CCc1c(c(n(n1)CC(c2ccccc2)O)N)C(=O)OCC BS-3468 CC(C)(C)OC(=O)NC1CCN(CC1)c2ccc(nn2)c3cccc(c3)F BS-3469 CC(C)(C)OC(=O)NC1CCN(C1)c2ccc(nn2)c3ccccc3F BS-3470 CC(C)(C)OC(=O)NC1CCCN(C1)c2ccc(nn2)c3ccccc3Cl BS-3471 Cc1cccc(c1)c2ccc(=O)[nH]n2 BS-3472 CCCCCn1c(=O)c2ccc(cc2[nH]c1=S)C(=O)O BS-3473 c1ccc(cc1)CSCC(C(=O)O)N BS-3474 c1ccc(cc1)CN2CCc3c(c(=O)[nH]c(n3)c4cccc(c4)Cl)C2 BS-3475 CCCNC(=O)c1ccc2c(c1)[nH]c(=O)cn2 BS-3476 COc1cccc(c1)NC(=S)N BS-3477 c1cnccc1c2cc([nH]n2)C(=O)NN BS-3478 CC1CCN(CC1)C(=N)N.CC1CCN(CC1)C(=N)N.OS(=O)(=O)O BS-3479 C1CSCCN1C(=N)N.I BS-3480 Cc1ccc(o1)CNC(=N)N.Cc1ccc(o1)CNC(=N)N.OS(=O)(=O)O BS-3481 COc1ccc(cc1)c2nc(on2)CC#N BS-3482 c1ccc(c(c1)N2CCN(CC2)C(=N)N)F.c1ccc(c(c1)N2CCN(CC2)C(=N)N)F.OS(=O)(=O)O BS-3483 C1CCC(C1)NC(=N)N.C1CCC(C1)NC(=N)N.OS(=O)(=O)O BS-3484 c1ccc(cc1)CCNC(=N)N.c1ccc(cc1)CCNC(=N)N.OS(=O)(=O)O BS-3485 c1ccc(c(c1)CNC(=N)N)F.c1ccc(c(c1)CNC(=N)N)F.OS(=O)(=O)O BS-3486 CCCn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cccc(c3)C BS-3488 Cc1ccc(cc1)NCc2cc3cc4c(cc3[nH]c2=O)OCCO4 BS-3489 COc1cc2cc(c(=O)[nH]c2cc1OC)CNc3ccccc3 BS-3490 COc1ccc(cc1)NCc2cc3cc4c(cc3[nH]c2=O)OCO4 BS-3491 COc1ccc(cc1)NCc2cc3cc(c(cc3[nH]c2=O)OC)OC BS-3492 CCc1ccc(cc1)CNS(=O)(=O)c2c(cn[nH]2)C(=O)OC BS-3493 c1cc(ccc1S(=O)(=O)c2c[nH]c3ccc(cc3c2=O)F)Cl BS-3494 c1cc(c(nc1)NN)S(=O)(=O)N2CCOCC2 BS-3495 c1cc(c2n[nH]c(=O)n2c1)S(=O)(=O)N3CCCCC3 BS-3496 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3cccn4c3n[nH]c4=O BS-3497 c1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-3498 c1nc([nH]n1)C(=O)N BS-3499 Cc1ccc(cc1)n2c(nc(n2)C(=O)OC)C BS-3500 c1cc(ccc1S(=O)(=O)Nc2ccsc2C(=O)O)Cl BS-3501 c1ccc(cc1)NS(=O)(=O)c2ccc[nH]c2=S BS-3502 Cc1cc(cc2c1nc(cc2OC)C(=O)O)OC BS-3503 CCOc1cc(nc2c1cc(cc2C)OC)C(=O)O BS-3504 Cc1cccc2c1nc(cc2OC)C(=O)O BS-3505 CCOc1cc(nc2c1cccc2F)C(=O)O BS-3506 Cn1cc(c(=O)c2c1ccc(c2)F)C(=O)O BS-3507 CCOC(=O)C1=C(c2ccccc2S1(=O)=O)N BS-3508 Cc1ccc(cc1)n2ccc(=O)c(n2)C(=O)NN BS-3509 CCOc1ccccc1c2nc(c(o2)C)C/C(=N/O)/N BS-3510 CCOc1ccc(cc1)c2nc(c(o2)C)C/C(=N/O)/N BS-3511 CC1CCN(CC1)S(=O)(=O)c2ccc3n[nH]c(=O)n3c2 BS-3512 CCOc1cc(=O)n(nc1C(=O)O)c2ccc(c(c2)F)F BS-3513 COc1cc(=O)n(nc1C(=O)O)c2ccc(cc2)F BS-3514 COc1cc(=O)n(nc1C(=O)O)c2cccc(c2)F BS-3515 c1ccc2c(c1)NN=C(S2(=O)=O)C(=O)N3CCCCC3 BS-3516 Cc1nnc2n1cccc2S(=O)(=O)Nc3ccc(cc3)Cl BS-3517 Cc1ccc(cc1)N2C=C(S(=O)(=O)c3c2cccc3)C#N BS-3518 CN(c1ccsc1C(=O)O)S(=O)(=O)c2ccc(cc2)Cl BS-3519 CCN1C=C(C(=NS1(=O)=O)C)C(=O)OCC BS-3520 Cc1ccc(cc1C)c2cc(n[nH]2)C(=O)NN BS-3521 COc1cc2c(cc1OC)nc(nc2N)SC BS-3522 c1ccc2c(c1)c(n[nH]2)C(=O)n3ccnc3 BS-3523 c1cc2c(cc1C(=O)n3ccnc3)OCO2 BS-3524 c1cc(ccc1C(=O)n2ccnc2)F BS-3525 c1cnc2nc(nn2c1)C(=O)n3ccnc3 BS-3526 Cn1c2ccccc2c(n1)C(=O)n3ccnc3 BS-3527 CCOC(=O)c1nc(no1)c2ccc3c(c2)OCO3 BS-3529 CCOC(=O)c1nc(no1)c2ccc(c(c2)OC)OC BS-3530 CCOC(=O)c1nc(no1)c2ccccc2F BS-3531 CCOC(=O)c1ncn(n1)CC(=O)c2cccc(c2)Cl BS-3532 Cc1c(ccc2c1[nH]c3c(c2=O)CNCC3)Cl BS-3533 c1cc(c(nc1)S)c2nc(no2)c3cccs3 BS-3535 Cc1ccc(cc1)c2nc(on2)c3cccnc3S BS-3536 COc1ccccc1Cn2c(=O)c3c(ccs3)[nH]c2=S BS-3537 CN1c2ccccc2C(=O)NC13CCNCC3 BS-3539 CCOC(=O)c1c(n(c(=S)s1)c2cc(ccc2OC)OC)N BS-3540 COc1ccc(cc1)C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-3541 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)N BS-3542 c1ccc(c(c1)/C=N/c2[nH]ncn2)O BS-3543 CCOC(=O)c1c(n(c(=S)s1)c2c(cccc2C)C)N BS-3544 Cc1c(c(n[nH]1)C)CCC(=O)NN BS-3545 c1ccc2c(c1)c(=O)n(c(=O)[nH]2)CCCCC(=O)O BS-3546 CCOC(=O)c1c(c2ccccc2[nH]1)NC(=O)C BS-3547 c1cnc2nc(cn2c1)C(F)(F)F BS-3549 c1ccc(c(c1)c2ccc(nn2)Cl)Cl BS-3550 c1ccc(c(c1)c2ccc(nn2)Cl)F BS-3551 Cc1ccccc1c2ccc(nn2)Cl BS-3552 c1cc(cc(c1)F)c2ccc(nn2)Cl BS-3553 C1CCN(CC1)C(=N)N.C1CCN(CC1)C(=N)N.OS(=O)(=O)O BS-3554 c1cc(ccc1C/C(=N/O)/N)F BS-3555 CCOc1ccccc1/C(=N/O)/N BS-3556 COc1ccc2cc(c(=O)[nH]c2c1)C=O BS-3557 CC(C)(C)c1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)O BS-3558 CCc1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)O BS-3559 c1cc(ccc1F)S(=O)(=O)Nc2ccsc2C(=O)O BS-3560 Cc1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)O BS-3561 Cc1ccc(cc1Cl)S(=O)(=O)Nc2ccsc2C(=O)O BS-3562 CCCc1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)O BS-3563 CN(c1ccsc1C(=O)O)S(=O)(=O)c2ccc(cc2)Br BS-3564 c1cc(ccc1S(=O)(=O)Nc2ccsc2C(=O)O)Br BS-3565 CC(C)c1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)O BS-3566 Cc1ccccc1c2csc3c2nc[nH]c3=O BS-3567 c1cc(cc(c1)F)c2csc3c2nc[nH]c3=O BS-3568 COc1ccc(cc1)NS(=O)(=O)c2ccsc2C(=O)O BS-3569 c1ccn(c1)c2c3cccnc3sc2C(=O)n4ccnc4 BS-3570 Cn1cc(c(=O)c2c1cccc2)C(=O)O BS-3571 Cn1cc(c(=O)c2c1cc(c(c2)F)N3CCCCC3)C(=O)O BS-3572 CCn1cc(c(=O)c2c1cc(c(c2)F)N3CCOCC3)C(=O)O BS-3573 Cc1nc(nn1c2ccc(cc2)F)C(=O)O BS-3574 CCOC(=O)c1c(nc(s1)N)C(C)C BS-3575 c1ccc(cc1)/C(=C/2\CCCCN2)/C#N BS-3576 Cc1cc2c([nH]1)c(=O)n(c(=S)[nH]2)C(C)C BS-3579 COc1ccc(cc1F)c2nc(on2)CN.Cl BS-3580 c1cc(ccc1c2nc(on2)CN)Cl.Cl BS-3581 c1c[nH]c(=O)c2c1cco2 BS-3582 CCOc1ccc(cc1)c2cc3c(=O)n(ccn3n2)CCN BS-3583 COc1cccc(c1)c2cc3c(=O)n(ccn3n2)CCN BS-3584 c1cc2c(cc1C(Cn3cc(nn3)C(=O)O)O)OCO2 BS-3585 c1cc2nc(cn2cc1Cl)CN3CCNCC3.Cl BS-3586 CCc1nc(on1)c2cccnc2O BS-3587 c1cc(ccc1c2cc3c(=O)n(ccn3n2)CC(=O)O)F BS-3588 c1cc(ccc1c2cc3c(=O)n(ccn3n2)CCC(=O)O)F BS-3589 CCOC(=O)c1cn(c(n1)C(=O)OCC)CC(=O)c2ccccc2 BS-3590 CCOC(=O)c1cn(c(n1)C(=O)OCC)CC(=O)c2ccc(cc2)OC BS-3591 c1cc(cnc1)c2nc(on2)C3CCN(CC3)c4cc(ncn4)Cl BS-3592 c1cc2c(cc1c3nc(on3)CN)OCO2.Cl BS-3593 COc1cc(=O)n2c(c1C(=O)OC)CCCC2 BS-3594 CNCc1nc(no1)c2ccc3c(c2)OCO3.Cl BS-3595 CNCc1nc(no1)c2ccc(cc2)Cl.Cl BS-3596 Cc1ccc(cc1)c2nc(on2)CNC.Cl BS-3597 CNCc1nc(no1)c2ccc(cc2)OC.Cl BS-3598 CNCc1nc(no1)c2ccc(cc2)F.Cl BS-3599 CNCc1nc(no1)c2ccc(c(c2)F)OC.Cl BS-3600 c1cc(cnc1)c2nc(on2)C3CCNCC3.Cl.Cl BS-3601 Cc1cc2c([nH]1)c(=O)[nH]cn2 BS-3602 Cc1cc(=O)[nH]c(n1)N2CCCCC2 BS-3603 c1cc(sc1)c2c(c[nH]n2)CO BS-3604 c1ccc(cc1)c2c(c[nH]n2)CO BS-3605 CC(C)(C)OC(=O)N1CCN(CC1)c2nc([nH]n2)N BS-3606 COCc1cc(=O)n2c([nH]1)nc(n2)N3CCNCC3.Cl BS-3607 c1c([nH]c2nc(nn2c1=O)N3CCNCC3)C4CC4.Cl BS-3608 c1ccc(cc1)n2c(c(nn2)C(=O)O)c3ccncc3 BS-3609 Cc1cn2c(cc(n2)C(=O)N3CCC(C3)N)c(=O)[nH]1.Cl BS-3610 c1c([nH]c2nc(nn2c1=O)N3CCNCC3)C(F)(F)F.Cl.Cl BS-3611 c1cc(ccc1c2c([nH]nn2)C(=O)O)F BS-3612 CCOC(=O)c1c(n(nn1)CC(=O)C)C(=O)OCC BS-3613 C1CCN(CC1)c2nc([nH]n2)N BS-3614 COc1ccccc1n2c(c(nn2)C(=O)O)c3ccncc3 BS-3615 COC(=O)c1c(n(nn1)Cc2ccccc2)N BS-3616 COc1ccc(cc1)n2c3c(cn2)c(=O)[nH]cn3 BS-3617 c1ccc(c(c1)n2c3c(cn2)c(=O)[nH]cn3)Cl BS-3618 c1cc([nH]c1)c2cc([nH]n2)C(=O)NN BS-3619 c1c[nH]cc1c2cc([nH]n2)C(=O)NN BS-3620 CC(C)(C)OC(=O)N1CCc2c(c3cc(ccc3[nH]2)OC)C1 BS-3621 Cn1cccc1c2nc(on2)C3CCNCC3.Cl BS-3622 Cn1cccc1c2nc(on2)C3CCNC3.Cl BS-3623 c1ccc2c(c1)c(nc(=O)[nH]2)NCc3cccs3 BS-3626 c1cnc(c(=O)[nH]1)N2CCCC(C2)N.Cl BS-3627 c1c(nc[nH]1)C(=O)NN BS-3628 CNCc1nc(no1)C2CC2.Cl BS-3629 Cn1ccnc(c1=O)N2CCCC(C2)N.Cl BS-3630 Cn1ccnc(c1=O)N2CCC(CC2)N.Cl BS-3631 Cc1nc(on1)c2ccc(cc2)CN.Cl BS-3632 Cc1nnc2n1ccnc2Cl BS-3633 Cc1nc(on1)C2CCCNC2.Cl BS-3634 Cc1nc(on1)C2CCNCC2.Cl BS-3635 c1ccc(cc1)Cn2cc(nc2)C(=O)O BS-3636 COC(=O)c1ccc2c(c1)[nH]c(=S)[nH]c2=O BS-3637 c1cnc(nc1)N2CCNCC2.Cl.Cl BS-3638 CC(C)(C)OC(=O)N1CCC(CC1)n2c(=O)c3ccccc3[nH]c2=O BS-3639 c1ccc(cc1)c2ccc(nn2)NN BS-3640 c1cc(sc1)c2ccc(nn2)NN BS-3641 c1ccc(c(c1)c2ccc(nn2)NN)F BS-3642 c1ccc2c(c1)c(=O)n(c(=O)[nH]2)C3CCNCC3.Cl BS-3643 c1cc2c(cc1F)c(=O)n(c(=O)[nH]2)C3CCNCC3.Cl BS-3644 c1ccn2c(c1)nc3c(c2=O)CNCC3 BS-3645 c1ccc(cc1)Cn2c(c(nn2)C(=O)O)c3ccncc3 BS-3646 c1ccnc(c1)c2c(cno2)C(=O)O BS-3647 c1ccc(cc1)C2Cn3c(c(cn3)C(=O)O)N2 BS-3648 C1CSCCN1C/C(=N/O)/N BS-3649 CNCc1nc(no1)c2ccncc2.Cl BS-3650 c1cc(cnc1)c2nc(on2)C3CCNC3.Cl BS-3651 COc1ccc(cc1)Cn2cnc3c(c2=O)cn[nH]3 BS-3652 c1ccc(c(c1)C2=NNS(=O)(=O)c3c2cc(cc3)Cl)F BS-3653 Cc1ccc(cc1)C2=NC3(CCN(CC3)C(=O)OC(C)(C)C)NC2=S BS-3654 C(CNC(=O)CC#N)CNC(=O)CC#N BS-3655 Cc1cccc(c1)Cn2c(=O)c3c(csn3)[nH]c2=O BS-3656 CCCOc1ccc(cc1OC)/C(=N/O)/N BS-3657 CCOC(=O)c1nc(no1)c2cn(nn2)c3ccc(cc3)F BS-3659 CCc1c(nnn1c2ccccc2)/C(=N/O)/N BS-3660 Cc1c(ccc2c1[nH]c3c(c2=O)CN(CC3)C(=O)C(F)(F)F)Cl BS-3661 c1cc2c(cc1Cl)c(=O)c3c([nH]2)CCN(C3)C(=O)C(F)(F)F BS-3662 COC(=O)c1c(n(nn1)CC(=O)c2cccs2)C(=O)OC BS-3663 c1cc(c(nc1)NN)c2nc(no2)C3CC3 BS-3664 CCCc1nc(on1)c2cccnc2NN BS-3665 C(C(=O)N)Sc1nc(c(s1)C(=O)N)N BS-3666 COc1cc(cc(c1)OC)NC(=O)CC#N BS-3668 c1ccc2c(c1)c3c(o2)c(=O)n(c(=S)[nH]3)Cc4ccc5c(c4)OCO5 BS-3670 COC(=O)c1c(n(nn1)CC(=O)c2ccc3c(c2)OCO3)C(=O)OC BS-3671 COc1ccc2c(c1)c3c([nH]2)c(=O)n(c(=S)[nH]3)CCC(=O)O BS-3672 Cc1c(sc2c1c(=O)n(c(=O)[nH]2)c3ccc(cc3)C(=O)O)C BS-3673 CCc1ccc(cc1)n2c(=O)c3ccc(cc3[nH]c2=O)C(=O)O BS-3674 CN(C)c1nc2cc(sc2n1c3ccc(cc3)OC)C(=O)O BS-3675 CCOC(=O)C(C)N1CCN(CC1)c2ccc(cc2)OC BS-3676 CCOC(=O)C(C)N1CCN(CC1)c2ccccc2F BS-3677 CCOC(=O)/C=C/1\NCCN1Cc2ccccc2F BS-3678 c1cc(ccc1C(=N)N)Cl BS-3680 Cc1ccc(cc1)NCc2cc3cc(c(cc3[nH]c2=O)OC)OC BS-3690 COc1ccc(cc1)S(=O)(=O)c2c[nH]c3ccc(cc3c2=O)Cl BS-3691 COc1ccc2cc(c(=O)[nH]c2c1)CNc3ccc(c(c3)OC)OC BS-3692 Cc1ccc(cc1)NCc2cc3ccc(cc3[nH]c2=O)OC BS-3693 CN(c1ccsc1C(=O)O)S(=O)(=O)c2ccc(cc2)F BS-3694 COc1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)O BS-3695 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)O BS-3696 Cc1cc(c(c(c1)C)S(=O)(=O)Nc2ccsc2C(=O)O)C BS-3697 Cc1cc(cc(c1)n2ccc(=O)c(n2)C(=O)O)C BS-3698 CSc1cccc(c1)n2ccc(=O)c(n2)C(=O)O BS-3699 c1cc(cc(c1)F)n2ccc(=O)c(n2)C(=O)O BS-3700 c1cc(c(cc1n2ccc(=O)c(n2)C(=O)O)F)F BS-3701 c1cc(ccc1c2csc3c2nc[nH]c3=O)F BS-3702 c1cc(ccc1c2csc3c2nc[nH]c3=O)Br BS-3703 COc1ccc(cc1)c2csc3c2nc[nH]c3=O BS-3704 COc1ccc(cc1OC)c2csc3c2nc[nH]c3=O BS-3705 c1cc(cc(c1)Cl)c2csc3c2nc[nH]c3=O BS-3706 Cc1cccc(c1)c2csc3c2nc[nH]c3=O BS-3707 c1cc(ccc1c2csc3c2nc[nH]c3=O)Cl BS-3708 Cc1ccc(cc1)c2csc3c2nc[nH]c3=O BS-3709 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCC(CC4)C(=O)O)F BS-3710 Cc1ccc(cc1)N2CNS(=O)(=O)c3c2nccc3 BS-3711 c1cc(ccc1S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F)Cl BS-3712 Cc1cc(cc(c1)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F)C BS-3713 Cc1ccc(c(c1)C)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F BS-3714 c1cc(cc(c1)Cl)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F BS-3715 CCn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cccc(c3)Cl BS-3716 Cn1cc(c(=O)c2c1cc(c(c2)F)N3CCCC3)C(=O)O BS-3717 CCn1cc(c(=O)c2c1cc(c(c2)F)N3CCC(CC3)C)C(=O)O BS-3718 CC1CCN(CC1)c2cc3c(cc2F)c(=O)c(cn3C)C(=O)O BS-3719 CCn1cc(c(=O)c2c1cc(c(c2)F)N3CCCCC3)C(=O)O BS-3720 Cn1cc(c(=O)c2c1cc(c(c2)F)N3CCOCC3)C(=O)O BS-3721 CCN1CCN(CC1)c2cc3c(cc2F)c(=O)c(cn3C)C(=O)O BS-3722 c1cc(c(nc1)Cl)S(=O)(=O)CC(=O)N2CCCC2 BS-3723 Cc1ccc2c(c1)NN=C(S2(=O)=O)C(=O)N3CCOCC3 BS-3724 CC1CCN(CC1)C(=O)C2=NNc3cc(ccc3S2(=O)=O)Cl BS-3725 CCc1ccc(cc1)NS(=O)(=O)c2cccn3c2nnc3 BS-3726 c1cc(c(nc1)Cl)S(=O)(=O)N2CCSCC2 BS-3727 COc1cc2c(cc1OC)nc(nc2N3CCNCC3)Cl BS-3728 c1cnccc1N BS-3729 c1cnccc1O BS-3730 c1cc(cnc1)O BS-3731 c1cncnc1N BS-3732 C1CC(=S)NC1 BS-3733 CC(=O)c1ccc[nH]1 BS-3734 Cc1ccnc(n1)N BS-3735 c1cc([nH]c1)C(=O)N BS-3736 Cc1cc(=O)[nH]cn1 BS-3737 c1c(=O)[nH]c(=O)[nH]n1 BS-3739 c1c(nn[nH]1)C(=O)O BS-3740 C1CCN(C1)C(=N)N BS-3741 C1CC1CNC(=N)N BS-3742 Cn1ccnc1S BS-3743 C1COCCC1=NO BS-3744 C1CCNC(=S)C1 BS-3746 c1(nc([nH]n1)S)N BS-3747 CN1CCNC1=S BS-3748 C1CN(C(=S)N1)N BS-3749 c1ccc(cc1)C(=N)N BS-3750 c1cnccc1C(=N)N BS-3751 c1ccc(cc1)C(=O)O BS-3752 c1cnc(cn1)C(=N)N BS-3753 c1cnccc1C(=O)O BS-3754 Cc1cc(nc(n1)N)C BS-3755 c1ccc(c(c1)CO)O BS-3756 COC(=O)c1cnc[nH]1 BS-3757 Cc1c(cnn1C)CO BS-3758 Cc1c(c(on1)C)CN BS-3759 COC(=O)c1c[nH]nn1 BS-3760 c1c(nc(nc1O)N)O BS-3761 Cc1c(scn1)C=O BS-3762 C1C(=O)NC(=O)NC1=O BS-3763 c1cc(sc1)C(=O)O BS-3764 Cc1ccc(s1)CO BS-3765 Cc1ccsc1CO BS-3766 C1COCCN1C(=N)N BS-3767 CCc1nnc(s1)N BS-3768 COCC1CCNCC1 BS-3769 C1CCC(=S)NCC1 BS-3770 c1cc2c(cc1N)CCC2 BS-3771 Cc1nnc2n1ccnc2 BS-3772 COc1ncc(cn1)C#N BS-3773 c1cc2c(=O)[nH]ncn2c1 BS-3774 c1cnn2c1c(=O)[nH]cc2 BS-3775 Cc1ccc(cc1)C(=O)N BS-3776 Cc1ccc(cc1)C(=O)O BS-3777 c1cc(cnc1)C(=O)NN BS-3780 c1cc(oc1)/C=C/C(=O)O BS-3783 c1cnc(cn1)C(=O)NN BS-3784 c1cc(ccc1C(=N)N)F BS-3785 CCCc1cc(=O)[nH]cn1 BS-3786 Cc1cc(nc(n1)NN)C BS-3787 c1cc(=O)[nH]cc1C(=O)O BS-3788 Cn1cccc1/C(=N/O)/N BS-3789 c1cc(oc1)CNC(=N)N BS-3790 c1c(c(=O)[nH]cn1)C(=O)O BS-3792 c1c(cnc(n1)O)C(=O)O BS-3793 c1ccc(c(c1)C(=O)O)F BS-3794 c1cc(cc(c1)F)C(=O)O BS-3795 COC(=O)Cn1ccnc1 BS-3796 CCn1ccc(n1)C(=O)O BS-3797 c1cn(cn1)C/C(=N/O)/N BS-3798 Cn1c(cc(=O)[nH]c1=O)N BS-3799 CCOC(=O)c1[nH]ncn1 BS-3800 CC(C)n1cnnc1CO BS-3801 CC1CCCN(C1)C(=N)N BS-3802 c1ccc2c(c1)c(c[nH]2)C#N BS-3804 Cc1ccc(s1)C(=O)O BS-3805 C1CCC(CC1)(C(=O)N)N BS-3807 C1CCC(CC1)NC(=O)N BS-3808 CN1CCN(CC1)C(=N)N BS-3809 C1CSCCN1CC#N BS-3810 COC(=O)c1c(non1)N BS-3811 C1CC(=O)N(C1)CC(=O)O BS-3812 C1CCC(CC1)(C(=O)O)N BS-3813 C1CC(OC1)CNC(=N)N BS-3814 c1cc(c(cc1F)F)NN BS-3815 C1C(=O)NC(=S)NC1=O BS-3816 c1cc(c2cc[nH]c2c1)C=O BS-3817 CCc1c[nH]c2c1cccc2 BS-3818 c1ccc2c(c1)[nH]c(n2)C=O BS-3819 c1cc(cc2c1cc[nH]2)CO BS-3820 c1c(c(c2n1CCC2)C#N)N BS-3821 c1ccc2c(c1)C(=O)CCO2 BS-3822 C1C(=O)N(C(=S)S1)N BS-3823 Cc1cc2c(=O)[nH]ccn2n1 BS-3824 CCc1ccc(cc1)C(=O)N BS-3825 Cc1ccc(cc1)/C(=N/O)/C BS-3826 Cc1ccc(cc1)NC(=O)C BS-3827 Cc1nnc2n1cc[nH]c2=O BS-3828 c1ccc(cc1)CCC(=O)O BS-3829 Cc1ccccc1/C(=N/O)/N BS-3830 Cc1ccc(cc1)NC(=O)N BS-3831 c1ccnc(c1)CNC(=N)N BS-3832 c1cc(ccc1CC(=O)O)N BS-3833 Cc1c(cccc1N)C(=O)O BS-3834 C1C/C(=C(\C#N)/C(=O)N)/NC1 BS-3835 COc1cccc(c1)C(=O)O BS-3836 c1ccc(cc1)OCC(=O)O BS-3837 Cc1ccc(o1)/C=C/C(=O)O BS-3838 c1cc(ccc1C(=O)NN)O BS-3839 c1cc(cc(c1)O)C(=O)NN BS-3840 c1c(n[nH]c1C(=O)O)C2CC2 BS-3841 c1nc([nH]n1)C(=O)NC2CC2 BS-3842 Cc1c(sc(c1C#N)N)C BS-3843 c1cc(c(cc1C(=O)O)N)O BS-3844 COC(=O)c1cnc(nc1)N BS-3845 C1CCc2n[nH]c(=O)n2CC1 BS-3846 c1ccnc(c1)NC(=S)N BS-3847 COC(=O)c1cnc[nH]c1=O BS-3848 c1ccc(c(c1)CC(=O)O)F BS-3849 c1cc(cc(c1)F)CC(=O)O BS-3850 Cc1cc(c([nH]1)C(=O)OC)N BS-3851 CCc1[nH]c(c(n1)C)C(=O)O BS-3852 CCOC(=O)c1c(nc[nH]1)C BS-3853 CC(C)c1cc([nH]n1)C(=O)O BS-3854 c1c(cc(nc1O)O)C(=O)O BS-3855 c1cc(c(c(c1)F)C(=O)O)N BS-3856 Cc1c(c(on1)C)CC(=O)O BS-3857 c1c(c(nc(n1)O)O)C(=O)O BS-3858 C1CC(=NC1)NCCC(=O)O BS-3859 c1cc(oc1)CNC(=S)N BS-3860 Cc1c([nH]c(=S)[nH]c1=O)C BS-3861 Cc1ccc(s1)C(=O)NN BS-3862 C[C@@H]1CC[C@H]([C@@H](C1)O)C(C)C BS-3863 Cc1c(cccc1Cl)NN BS-3864 c1ccc(cc1)C(=N)N.Cl BS-3865 COC(=O)N/N=C/1\CCCN1 BS-3866 C1[C@@H](CC[C@H](C1)C(=O)O)CN BS-3867 c1cc(c(cc1F)C(=O)O)F BS-3868 c1cc(c(c(c1)F)C(=O)O)F BS-3869 c1cc(c(cc1C(=O)O)F)F BS-3870 C1COCCN1CCC(=O)O BS-3871 c1ccc(cc1)C2=NNC(=O)C2 BS-3872 Cc1[nH]c(=O)c2ccccc2n1 BS-3873 C1CC(OC1)CNC(=S)N BS-3874 c1nc2[nH]nc(c(=O)n2n1)C#N BS-3875 c1ccc2c(c1)c(=O)[nH][nH]c2=O BS-3876 C/C(=C\c1ccccc1)/C(=O)O BS-3877 c1ccc(cc1)C2(CC2)C(=O)O BS-3878 c1cc2cn[nH]c2cc1[N+](=O)[O-] BS-3879 c1ccc2c(c1)C(CN2)C(=O)O BS-3880 CN(Cc1ccccc1)C(=N)N BS-3881 Cc1cccc(c1)CNC(=N)N BS-3882 c1c(nc[nH]c1=O)C(F)(F)F BS-3883 c1cc(oc1)CNC(=O)CC#N BS-3884 CCc1ccc(cc1)CC(=O)O BS-3885 CC(C)c1ccc(cc1)C(=O)O BS-3886 CCC(c1ccccc1)C(=O)O BS-3887 Cc1ccc(c(c1)C)C(=O)NN BS-3888 Cc1ccccc1C/C(=N\O)/N BS-3889 Cc1ccc(c(c1)NC(=O)N)C BS-3890 Cc1cccc(c1C)NC(=O)N BS-3891 CCc1cccc(c1)NC(=O)N BS-3892 Cc1ccc(cc1C)NC(=O)N BS-3893 CCc1ccccc1NC(=O)N BS-3894 Cc1cc(cc(c1)NC(=O)N)C BS-3895 c1ccnc(c1)CCNC(=N)N BS-3896 C1CCN(CC1)S(=O)(=O)N BS-3897 C1CCN/C(=C(/C#N)\C(=O)N)/C1 BS-3898 c1cc2c(cc1C(=O)O)OCO2 BS-3899 Cc1c(ccc(c1O)C(=O)C)O BS-3900 Cc1ccc(cc1)OCC(=O)O BS-3901 Cc1cc(ccc1C(=O)O)OC BS-3902 CC(C(=O)O)Oc1ccccc1 BS-3903 Cc1ccccc1OCC(=O)O BS-3904 COC(=O)c1cc(n[nH]1)C2CC2 BS-3905 C1CCc2c(c([nH]n2)C(=O)O)C1 BS-3906 c1nc([nH]n1)C(=O)N2CCCC2 BS-3907 Cc1cccc(c1)NC(=S)N BS-3908 COc1ccc(cc1N)C(=O)O BS-3909 Cc1nc(on1)C2CCCCN2 BS-3910 c1ccc(cc1)NC(=S)NN BS-3911 C1CCC(=CC1)CCNC(=N)N BS-3912 CC(=O)c1ccc(c(c1O)O)O BS-3913 c1cc(cc(c1)F)C/C(=N/O)/N BS-3914 Cc1cc(ccc1NC(=O)N)F BS-3915 Cc1cc(n(n1)CC(=O)OC)C BS-3916 C1CC(OC1)CNC(=O)CC#N BS-3917 C=CCN1CCN(CC1)C(=N)N BS-3918 c1c(c2c(s1)CCCC2)CO BS-3919 Cc1nc(cc2n1cnn2)Cl BS-3920 COC(=O)/C=C\1/CCCCCN1 BS-3921 c1cc(sc1)CCNC(=N)N BS-3922 COC(=O)c1cnc(nc1O)O BS-3923 C1COCCC12C(=O)NC(=O)N2 BS-3924 CCOC(=O)/C=C/1\NCCN1C BS-3925 C1CN(CCC1C(=O)N)C(=N)N BS-3926 CCc1c([nH]c(=S)[nH]c1=O)C BS-3927 CCCc1cc(=O)[nH]c(=S)[nH]1 BS-3928 c1cc(ccc1CC(=O)O)Cl BS-3929 c1ccc(c(c1)CC(=O)O)Cl BS-3930 c1ccc(c(c1)NC(=O)N)Cl BS-3931 c1(c([nH]c(=O)[nH]c1=O)C(=O)O)N BS-3932 CCn1c(cc(=O)[nH]c1=S)N BS-3934 CCc1nnc(s1)NC(=O)C BS-3935 c1cc(c(cc1/C(=N/O)/N)F)F BS-3936 c1cc(c(cc1NC(=O)N)F)F BS-3937 c1cc(c(cc1F)NC(=O)N)F BS-3938 CN1CCN(CC1)CCC(=O)O BS-3939 c1cc(c(cc1[N+](=O)[O-])Cl)N BS-3940 CCc1[nH]c(=O)c(c(n1)C)Cl BS-3941 c1c(c(cc(c1F)F)N)C(=O)O BS-3943 Cc1ccccc1NC(=O)CC#N BS-3944 c1ccc(cc1)C2CCC(=O)CC2 BS-3945 c1cc(c(c(c1)Cl)C(=O)O)F BS-3946 c1cc(c(cc1F)C(=O)O)Cl BS-3947 c1cc(c(cc1C(=O)O)Cl)F BS-3948 c1cc(c(cc1Cl)C(=O)O)F BS-3949 c1cc(c(cc1F)Cl)C(=O)O BS-3950 c1ccc2c(c1)CCC2NC(=N)N BS-3951 c1ccc2c(c1)CCN(C2)C(=N)N BS-3952 CC(C)(C)c1cn2cccnc2n1 BS-3953 Cc1c(c([nH]n1)N)Br BS-3954 C1Cc2c(c(=O)[nH]c(=O)n2C1)C#N BS-3955 Cc1nc(on1)c2ccc[nH]c2=O BS-3956 Cc1ccc(cc1C)CNC(=N)N BS-3957 CCc1ccc(cc1)CNC(=N)N BS-3958 c1ccc(cc1)CCCNC(=N)N BS-3959 c1cc2c(cc1F)c(ncn2)NN BS-3962 COc1ccccc1/C=C/C(=O)O BS-3963 c1cc(sc1)c2c(c[nH]n2)C=O BS-3964 c1cc(sc1)c2ccc(=O)[nH]n2 BS-3965 CC(C)(C)c1ccc(cc1)C(=O)O BS-3966 CC(=O)Nc1cccc(c1)C(=O)O BS-3967 c1ccc(cc1)C(=O)NCC(=O)O BS-3968 CN(C)c1ccc(cc1)C(=O)NN BS-3969 CN(C)c1cccc(c1)C(=O)NN BS-3970 COc1ccccc1CNC(=N)N BS-3971 c1cc(=O)n2c(c1C(=O)O)NCC2 BS-3972 CC(=O)c1c(cccc1OC)OC BS-3973 COc1cccc(c1)CCC(=O)O BS-3974 COc1ccccc1CCC(=O)O BS-3975 CCOc1ccc(cc1)C(=O)NN BS-3976 Cc1cc(ccc1C(=O)NN)OC BS-3977 COc1ccc(cc1)C/C(=N/O)/N BS-3978 COc1ccc(cc1)OCC(=N)N BS-3979 CCOc1ccccc1NC(=O)N BS-3980 c1cc(sc1)CNC(=O)CC#N BS-3981 Cc1cc([nH]n1)CN2CCNCC2 BS-3982 Cc1cccc(c1C)NC(=S)N BS-3983 Cc1c(c([nH]c1C(=O)O)C)C(=O)C BS-3984 c1cn(cn1)C(=O)N2CCOCC2 BS-3985 CCc1nc(on1)C2CCCCN2 BS-3986 Cc1nc(on1)C2(CCCCC2)N BS-3987 COc1cc(cc(c1)OC)C(=O)O BS-3988 COc1ccc(cc1OC)C(=O)O BS-3989 COc1ccc(c(c1)OC)C(=O)O BS-3990 COc1ccc(cc1)OCC(=O)O BS-3991 COc1cccc(c1OC)C(=O)O BS-3992 Cc1cc(c([nH]1)C(=O)OC)NC=O BS-3993 Cc1c(c(n(n1)C)C)CCC(=O)O BS-3994 CC1CCC2(CC1)C(=O)NC(=O)N2 BS-3995 CCNc1cc(ccc1C(=O)O)F BS-3997 CCn1cnc(c1C(=O)O)C(=O)O BS-3998 COc1ncc(c(n1)O)C(=O)OC BS-3999 COC(=O)c1c(nc[nH]1)C(=O)OC.Cl BS-4000 CC(C)CN1CCN(CC1)C(=N)N BS-4001 Cc1ccc(c(c1)Cl)NC(=O)N BS-4002 Cc1ccc(cc1NC(=O)N)Cl BS-4003 Cc1c(cccc1Cl)NC(=O)N BS-4004 Cc1ccc(cc1Cl)NC(=O)N BS-4005 c1c(cc(cc1F)F)CNC(=N)N BS-4006 c1cc(c(cc1F)F)CNC(=N)N BS-4007 Cc1ccc(cc1)S(=O)(=O)NC BS-4008 COc1ccc2ccccc2c1C=O BS-4009 Cc1ccc(cc1)/C=C(\C#N)/C(=O)N BS-4010 Cc1[nH]c(=O)cc(n1)c2ccccc2 BS-4011 Cc1cc(=O)[nH]c(n1)c2ccccc2 BS-4012 Cc1ccccc1c2ccc(=O)[nH]n2 BS-4013 c1cc(cc(c1)Cl)NC(=S)N BS-4014 COCCN1CC(CC1=O)C(=O)O BS-4015 Cc1ccc2cc(c(=O)[nH]c2c1)C=O BS-4016 c1cc2cc(ccc2nc1)C(=O)NN BS-4017 c1cc(ccc1NN)S(=O)(=O)N BS-4018 Cc1ccc(c2c1nccc2)[N+](=O)[O-] BS-4020 c1ccc(cc1)c2c(c[nH]n2)C(=O)O BS-4021 Cc1cccc(c1NC(=O)CC#N)C BS-4022 CCc1ccc(cc1)NC(=O)CC#N BS-4023 CC1(NC(=O)C(=N1)c2ccccc2)C BS-4024 c1cnc(nc1)N2CCC(CC2)C#N BS-4025 c1cc(c(c(c1)Cl)CC(=O)O)F BS-4026 c1cc(c(cc1/C(=N/O)/N)Cl)F BS-4027 c1ccc2c(c1)c(=O)c(c[nH]2)C(=O)O BS-4028 c1ccc(cc1)c2c([nH]nn2)C(=O)O BS-4029 c1ccnc(c1)n2cc(cn2)C(=O)O BS-4030 Cn1cc(c2c1cccc2)C(=O)OC BS-4031 Cn1c2ccccc2cc1C(=O)OC BS-4032 Cc1ccc(cc1N)c2nc(no2)C BS-4033 Cc1cc2c([nH]1)c(=O)n3c(n2)CCC3 BS-4034 c1cn2c(c3c(n2)CCCC3)c(=O)[nH]1 BS-4035 c1c2c(=N)n3c(nc2[nH]n1)CCCC3 BS-4036 c1ccc(cc1)CN2CCCC(=O)C2 BS-4037 c1cc(ccc1C(=O)O)C(F)(F)F BS-4038 c1ccc(c(c1)C(=O)O)C(F)(F)F BS-4039 c1cn(cn1)c2ncc(cn2)C(=O)O BS-4040 c1cc(ccc1c2[nH]nnn2)C(=O)O BS-4041 CN1C=C(C=NS1(=O)=O)C(=O)O BS-4043 COc1ccccc1NC(=O)CC#N BS-4044 COC(=O)Cc1cn2ccccc2n1 BS-4045 Cc1ccc(cc1)n2cc[nH]c2=S BS-4046 c1ccc(cc1)c2ccc(nn2)Cl BS-4047 c1cc(c(cc1Cl)C(=O)O)Cl BS-4048 C1CCn2c(c(c(=O)[nH]c2=O)C#N)C1 BS-4049 COC(=O)c1cc(n[nH]1)c2ccc[nH]2 BS-4050 c1cscc1c2nc(on2)CC#N BS-4051 Cc1ccccc1NC(=O)CC(=O)C BS-4052 C1C(=O)N(C(=S)S1)CC(=O)O BS-4053 c1ccc(cc1)C(C2CCNCC2)O BS-4054 CC(CCc1ccccc1)NC(=N)N BS-4055 CCOC(=O)c1cc([nH]n1)N.Cl BS-4056 c1cc(ccc1NN)OC(F)(F)F BS-4057 c1cc(ccc1CNC(=O)CC#N)F BS-4058 Cc1ccc(cc1)C(=O)CCC(=O)O BS-4059 Cc1c(sc(n1)n2cccc2)C=O BS-4060 CC1(Nc2ccccc2C(=N1)S)C BS-4061 CC(=O)Nc1ccc2c(c1)OCCO2 BS-4062 C1CCNC(C1)c2nc(no2)C3CC3 BS-4063 c1cc(cc(c1)Cl)c2cn[nH]c2N BS-4064 Cc1cn2c(c(nn2)C(=O)O)c(=O)[nH]1 BS-4065 COC(=O)c1cc2n(n1)CCCC2=O BS-4067 c1cc(sc1)c2c(c[nH]n2)C(=O)O BS-4068 COC(=O)/C(=C\1/CCCCCN1)/C#N BS-4069 COc1cccc(c1)CCC(=O)NN BS-4070 COc1ccc(cc1)CCC(=O)NN BS-4071 Cc1c(sc(n1)n2cccc2)CO BS-4072 c1ccn(c1)c2nc(cs2)CCO BS-4073 c1cc(cc(c1)Cl)NC(=O)CC#N BS-4074 Cc1cc(=O)[nH]c(n1)N2CCOCC2 BS-4075 CC(C)c1nc(on1)C2CCCCN2 BS-4076 Cc1ccc(cc1C)NC(=S)NN BS-4077 c1cc(ncc1Cl)NC(=O)CC#N BS-4078 Cc1nc(on1)c2cccnc2Cl BS-4079 Cc1nc(on1)c2ccnc(c2)Cl BS-4080 Cc1nc(on1)c2ccc(nc2)Cl BS-4081 C1Cc2c(c(nn2C1)C(=O)O)C(=O)O BS-4082 COC(=O)c1c2n(nn1)CCNC2=O BS-4083 c1cc(ccc1C(=O)CCC(=O)O)F BS-4084 COc1ccc(cc1OC)CC(=O)O BS-4085 COc1cc(cc(c1)OC)NC(=O)N BS-4086 COC(=O)c1cc2n(n1)CCCC2O BS-4087 c1ccc(c(c1)N)S(=O)(=O)CC#N BS-4088 Cc1c(c(n(n1)C)C)CCCC(=O)O BS-4089 C1CCc2c(c(c(s2)N)C(=O)N)C1 BS-4090 c1cc(c(nc1)Cl)CN2CCCC2 BS-4092 COc1cc(c(cc1OC)N)C(=O)O BS-4093 C1CCC(C1)N2CC(CC2=O)C(=O)O BS-4094 COCc1nc(on1)C2CCCCN2 BS-4095 CCOC(=O)c1cc([nH]n1)C(=O)OC BS-4096 Cc1ccc(cc1)n2c(c(nn2)C#N)C BS-4097 Cn1c(=O)c2c(ccs2)[nH]c1=S BS-4098 CSc1[nH]c(=O)c2c(n1)ccs2 BS-4099 CCOc1ccc(cc1Cl)C(=O)C BS-4100 c1ccc(c(c1)F)S(=O)(=O)CC#N BS-4101 Cc1nc(on1)c2cc3ccccc3[nH]2 BS-4102 Cc1ccc2c(c1)c3c([nH]2)c(=O)[nH]cn3 BS-4103 CC(C)(C)OC(=O)CN1CCCC1=O BS-4104 c1csc2c1c(=O)n(c(=S)[nH]2)N BS-4105 c1cc(ccc1NC(=O)C(=O)O)Cl BS-4106 c1[nH]c(=O)c2c(n1)c(c3n2CCC3)C#N BS-4107 COCCNC(=O)CN1CCCC1=O BS-4108 Cc1ccc(cc1C)c2ccc(=O)[nH]n2 BS-4109 Cc1ccc(cc1)N2CC(CC2=O)C#N BS-4110 CCc1c(sc(n1)N)C(=O)OCC BS-4111 CCOCC(=O)N1CCC(CC1)CN BS-4112 CC(C(=O)O)Oc1cccc(c1)Cl BS-4113 COC(=O)c1c(c(n[nH]1)C2CC2)Cl BS-4114 c1ccc(cc1)C(=O)NCCN.Cl BS-4115 Cc1cc(=O)[nH]c(n1)Nc2ccccc2 BS-4116 c1ccc2c(c1)c3c([nH]2)c(=S)[nH]cn3 BS-4117 c1cc(c(cc1C(=O)O)[N+](=O)[O-])Cl BS-4118 c1cc(c(cc1F)Cl)CNC(=N)N BS-4119 COc1ccc(cc1)c2cc([nH]n2)C=O BS-4120 COc1ccccc1c2ccc(=O)[nH]n2 BS-4121 Cc1ccc(cc1)c2cc([nH]n2)C(=O)O BS-4122 Cc1c(nnn1c2ccccc2)C(=O)N BS-4123 CNS(=O)(=O)c1cccnc1NN BS-4124 CC(CNC(=O)CC#N)c1ccccc1 BS-4125 c1cc2c(cc1F)c3c([nH]2)c(=O)[nH]cn3 BS-4126 Cc1ccc2c(c1)c(=O)c(c[nH]2)C(=O)O BS-4127 COc1cc(nc2c1cccc2)C(=O)O BS-4128 c1cc(ccc1C(=O)N)NC(=O)CC#N BS-4129 Cc1ccc(cc1)n2cc(nn2)C(=O)O BS-4130 c1cc(c(nc1)O)c2nc(no2)C3CC3 BS-4131 c1cc(=O)[nH]cc1c2nc(no2)C3CC3 BS-4132 c1cc(c(=O)[nH]c1)c2nc(no2)C3CC3 BS-4133 c1cc([nH]c(=O)c1)c2nc(no2)C3CC3 BS-4134 c1ccc(cc1)n2c(c(nn2)C(=O)N)N BS-4135 CCn1cc(c2c1ccc(c2)OC)C=O BS-4136 Cc1cc2c([nH]1)c(=O)n3c(n2)CCCC3 BS-4137 c1cc(ccc1C(=O)NN)C(F)(F)F BS-4138 c1ccc(c(c1)C(F)(F)F)NC(=O)N BS-4139 COC(=O)c1cnc(nc1)n2ccnc2 BS-4140 c1cc(ccc1N2CC(CC2=O)C#N)F BS-4141 CC1=NS(=O)(=O)N(C=C1C(=O)O)C BS-4142 CCOC(=O)C1=CNS(=O)(=O)N=C1 BS-4143 COc1ccc(cc1)CC(C#N)C(=O)N BS-4144 COc1ccccc1CNC(=O)CC#N BS-4145 c1ccc2c(c1)cc([nH]2)C(CC(=O)O)N BS-4146 CCc1nc2c(c3n1c(=O)[nH]n3)CCC2 BS-4147 CCc1nc(on1)c2cc(n[nH]2)C3CC3 BS-4148 c1ccc(cc1)c2cc(=O)[nH]c(=S)[nH]2 BS-4149 c1cc(ccc1NC(=O)CN)F.Cl BS-4151 c1cc(c(cc1NC(=S)N)Cl)F BS-4152 c1cc(c(cc1NC(=O)N)Cl)Cl BS-4153 c1c(cc(cc1Cl)Cl)NC(=O)N BS-4154 c1cc(c(cc1Cl)Cl)NC(=O)N BS-4155 CCOC(=O)c1c(c2ccccc2o1)N BS-4156 C1CCc2c(c(=O)[nH]c(=O)n2CC1)C#N BS-4157 CCc1nc(on1)c2cccnc2NN BS-4158 Cc1ccc(c(c1)C)NC(=O)CC(=O)C BS-4159 c1ccnc(c1)N2CCN(CC2)C(=N)N BS-4161 c1cc(ccc1C(=O)O)OC(F)(F)F BS-4163 c1cc(cc(c1)OC(F)(F)F)C(=O)O BS-4164 c1cc(ccc1c2c(c[nH]n2)C(=O)O)F BS-4165 c1cc(ccc1c2cc(n[nH]2)C(=O)O)F BS-4166 Cc1c(c([nH]n1)S(=O)(=O)O)C(=O)O BS-4167 c1cnc(cn1)N2CCC(CC2)C(=O)N BS-4168 Cc1c2c(=O)cc([nH]c2n(n1)C)C(=O)O BS-4169 Cc1nc(nn1c2cccc(c2)F)CO BS-4170 CCOC(=O)C(=O)Nc1cccc(c1)C BS-4171 CCOC(=O)C(=O)Nc1ccc(cc1)C BS-4172 Cc1cc2c([nH]1)c(=O)n(c(=O)[nH]2)C(C)C BS-4173 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)N BS-4174 Cc1cc(=O)[nH]c(n1)N2CCC(CC2)C BS-4175 Cc1cc(=O)[nH]c(n1)N2CCCC(C2)C BS-4176 C1CCC(CC1)(c2nc(no2)C3CC3)N BS-4177 CC1(CCCNC1)c2nc(no2)C3CC3 BS-4178 c1cn2c(c3c(n2)CCCC3)c(n1)Cl BS-4179 Cc1cn2c(c(nn2)C(=O)OC)c(=O)[nH]1 BS-4180 CCOC(=O)c1ccc(=O)n2c1NCC2 BS-4181 c1cc(ccc1C(=O)NCCC(=O)O)N BS-4182 COC(=O)CSc1c(cccn1)C#N BS-4183 Cc1c(sc(n1)n2cccc2)C(=O)O BS-4184 Cc1ccc(cc1NC(=O)CC#N)Cl BS-4185 Cc1c(cccc1Cl)NC(=O)CC#N BS-4186 COc1ccc(cc1OC)CNC(=N)N BS-4187 CC(C)c1nc(on1)CC2CCNCC2 BS-4188 C1CCn2c(c(c(n2)C(=O)O)C(=O)O)C1 BS-4189 C1Cc2c(c(=O)[nH]c(=O)n2C1)/C(=N/O)/N BS-4190 CCOc1ccc(cc1OCC)C(=O)O BS-4191 CCn1c2ccccc2c3c1ccc(c3)N BS-4192 CC(C)c1nc(on1)CN2CCNCC2 BS-4193 COc1ccc(cc1Cl)c2ncon2 BS-4194 CCOC(=O)C(=O)Nc1cccc(c1)F BS-4195 c1cc2c(cc[nH]2)cc1C(=O)n3ccnc3 BS-4196 c1ccc2c(c1)c(c[nH]2)C(=O)n3ccnc3 BS-4197 c1ccc(cc1)c2cc3c(=O)[nH]ccn3n2 BS-4198 CC1=NS(=O)(=O)c2cccnc2N1C BS-4199 C1CCC(CC1)N2CC(CC2=O)C(=O)O BS-4200 c1cc(cc(c1)NC(=O)CN)C#N.Cl BS-4201 CCOC(=O)c1cc(n[nH]1)C(=O)OCC BS-4202 c1ccc(cc1)c2cn3c(cnn3)c(=O)[nH]2 BS-4203 c1ccc(cc1)C2(CC2)C(=O)n3ccnc3 BS-4204 c1cc(c(cc1NC(=O)CC#N)Cl)F BS-4205 c1cnc2c(cnn2c1)C(=O)n3ccnc3 BS-4206 c1cc(c(nc1)Nc2ccc(cc2)F)C#N BS-4207 Cc1ccc(c(c1)F)S(=O)(=O)CC#N BS-4208 c1ccc2c(c1)cc3n(c2=O)CCCCC3 BS-4209 CCc1ccc(cc1)Nc2c(cccn2)N BS-4210 c1ccc-2c(c1)CCc3c2[nH]nc3C(=O)O BS-4211 CC(C)c1ccc(cc1)c2ccc(=O)[nH]n2 BS-4212 CCc1ccc(cc1)N2CC(CC2=O)C#N BS-4213 Cc1ccc2c(c1)c(=O)c3c([nH]2)CCNC3 BS-4214 Cc1cc(cc(c1)NC(=O)CN)C.Cl BS-4215 Cc1ccc(cc1C)NC(=O)CN.Cl BS-4216 CCc1ccccc1NC(=O)CN.Cl BS-4217 c1ccc(c(c1)NC(=O)N)Br BS-4218 c1cc(ccc1NC(=O)N)Br BS-4219 c1cc(cc(c1)Br)/C(=N/O)/N BS-4220 CC(C)(C)OC(=O)N1CCCC1C(=O)O BS-4221 c1ccc(cc1)c2nc(on2)C3CCCN3 BS-4222 CCCNc1c(cccn1)S(=O)(=O)N BS-4223 c1cc2c(cc1c3ccc(=O)[nH]n3)OCO2 BS-4224 c1ccc2c(c1)-c3c(c(n[nH]3)C(=O)O)CO2 BS-4225 CC1(Cc2c(cc(c(=O)[nH]2)C#N)C(=O)C1)C BS-4226 COC(=O)c1cn(cn1)Cc2ccccc2 BS-4227 COC(=O)c1cncn1Cc2ccccc2 BS-4228 COc1cccc(c1)CC(=O)n2ccnc2 BS-4229 Cc1c(c(=O)[nH]c(=O)[nH]1)Cc2ccccc2 BS-4230 CCc1ccc(cc1)c2cc([nH]n2)C(=O)O BS-4231 Cc1ccc(c(c1)c2cc([nH]n2)C(=O)O)C BS-4232 COc1ccc(cc1)N2CC(CC2=O)C#N BS-4233 CC(C)(C)OC(=O)N1CCNC(=S)C1 BS-4234 Cc1nc(on1)c2ccn3c(c2)n[nH]c3=O BS-4235 c1ccc(c(c1)CNC(=N)N)C(F)(F)F BS-4237 c1cc(c(cc1F)F)S(=O)(=O)CC#N BS-4238 c1cc(c(cc1F)S(=O)(=O)CC#N)F BS-4239 c1ccc(c(c1)F)S(=O)(=O)CC(=O)N BS-4240 Cc1ccc2c(c1)c(=O)c(cn2C)C(=O)O BS-4241 Cc1ccc(cc1)n2c(nc(n2)C(=O)O)C BS-4242 Cc1ccc(cc1)n2cc(nn2)C(=O)OC BS-4243 Cc1cccc(c1)n2c(c(nn2)C(=O)O)C BS-4244 CCc1c(nnn1c2ccccc2)C(=O)O BS-4245 Cc1ccc(cc1)n2c(c(nn2)C(=O)O)C BS-4246 Cc1c(nnn1c2ccccc2)/C(=N/O)/N BS-4247 Cc1ccccc1n2c(c(nn2)C(=O)N)N BS-4248 c1ccc(cc1)Cn2cc(nn2)/C(=N/O)/N BS-4249 Cc1cccc(c1)n2c(c(nn2)C(=O)N)N BS-4250 c1c(cn2cnnc2n1)C(=O)N3CCCC3 BS-4251 c1ccc(cc1)C(=O)C(=O)N2CCCCC2 BS-4252 Cc1cc2c([nH]1)c(=O)n3c(n2)CCCCC3 BS-4253 CCc1nc(on1)C2CCCCN2.Cl BS-4254 COC(=O)c1ccc(cc1)NC(=O)CC#N BS-4256 COc1ccccc1c2cc([nH]n2)C(=O)O BS-4257 COc1ccccc1c2c(c[nH]n2)C(=O)O BS-4258 COc1cccc(c1)c2c(c[nH]n2)C(=O)O BS-4259 COc1ccc(cc1)c2cc([nH]n2)C(=O)O BS-4260 Cc1ccc(cc1)c2nc(on2)C(=O)NN BS-4261 c1cc(ccc1CN2CC(CC2=O)C#N)F BS-4262 c1cc2c(c(c1)F)[nH]c3c(c2=O)CNCC3 BS-4263 CCOC(=O)C1=CN(S(=O)(=O)N=C1)C BS-4264 CCN1C=C(C(=NS1(=O)=O)C)C(=O)O BS-4265 c1ccc2c(c1)c3c(o2)c(=O)[nH]c(=S)[nH]3 BS-4266 Cc1cccc(c1)CN2CCNC(=O)C2=O BS-4267 Cc1ccc(cc1)N2CC(CC2=O)C(=O)N BS-4268 Cc1ccccc1N2CC(CC2=O)C(=O)N BS-4269 CCc1nc2c(c3n1c(=O)[nH]n3)CCCC2 BS-4270 CCOC(=O)c1c(nc(s1)SC)N BS-4271 Cc1cccc(c1)N2CCN(CC2)C(=N)N BS-4272 CCOC(=O)c1nc(no1)c2ccncc2 BS-4273 Cc1cc(=O)[nH]c(n1)Nc2ccc(cc2)F BS-4274 Cc1ccccc1N2CC(CC2=O)C(=O)O BS-4275 c1ccc(cc1)N2CC(CC2=O)/C(=N/O)/N BS-4276 Cc1ccc(cc1)CN2CCCC2C(=O)O BS-4277 COc1ccc(c(c1)OC)NC(=O)CC#N BS-4278 c1csc2c1nc3n(c2=O)CCCCC3 BS-4279 C1CCc2nnc(n2CC1)C3CCNCC3 BS-4280 c1ccc(c(c1)O)Oc2ccccc2Cl BS-4281 Cc1cc(=O)[nH]c(n1)c2ccc(cc2)Cl BS-4282 Cc1cc(=O)[nH]c(n1)c2cccc(c2)Cl BS-4283 COc1ccccc1c2ccc(nn2)Cl BS-4284 c1cc(ccc1N2CC(CC2=O)C#N)Cl BS-4285 c1cc(c(cc1Cl)Cl)OCC(=O)O BS-4286 c1cc(ccc1NC(=O)CN)Cl.Cl BS-4287 c1cc(ccc1n2c(cc(=O)[nH]c2=O)N)F BS-4288 c1cc(ccc1n2cc(nn2)/C(=N/O)/N)F BS-4289 CCOC(=O)c1cn2cc([nH]c(=O)c2n1)C BS-4290 c1cc(cc2c1cc(c(=O)o2)C(=S)N)O BS-4291 CCOC(=O)C(=O)Nc1ccc(cc1C)C BS-4292 CCOC(=O)C(=O)Nc1ccc(c(c1)C)C BS-4293 COC(=O)c1c(ccs1)S(=O)(=O)N BS-4294 c1c(cnc(n1)NN)C(=O)N2CCCCC2 BS-4295 c1cnc(cn1)N2CCC(CC2)/C(=N/O)/N BS-4297 Cc1ccc(cc1)S(=O)(=O)n2cccc2 BS-4298 CCOC(=O)c1c(c2ccccc2s1)N BS-4299 CC1=C(Sc2ccccc2N1)C(=O)NN BS-4300 COc1cc2c(cc1OC)[nH]c(=O)[nH]c2=O BS-4302 c1cc(cc(c1)F)CN2CCNC(=O)C2=O BS-4303 c1cc(ccc1N2CC(CC2=O)C(=O)N)F BS-4304 c1ccc(cc1)c2c3ccccc3[nH]c(=O)n2 BS-4306 c1cc(oc1)C(=O)N2CCN(CC2)C(=N)N BS-4307 c1cc(c(cc1F)F)NC(=O)CN.Cl BS-4308 c1cc(ccc1c2c(c[nH]n2)C(=O)O)Cl BS-4309 c1cc(ccc1CCNC(=O)CC#N)Cl BS-4310 CC1(NC(=O)C(=N1)c2ccc(cc2)Cl)C BS-4311 c1cc(cc(c1)F)N2CC(CC2=O)C(=O)O BS-4312 c1ccc(c(c1)N2CC(CC2=O)C(=O)O)F BS-4313 CCOC(=O)C(=O)Nc1ccccc1OC BS-4314 CCOC(=O)C(=O)Nc1cccc(c1)OC BS-4315 COc1cc(=O)n2c(c1C(=O)O)CCCC2 BS-4316 CCOC(=O)c1cc2n(n1)CCCNC2=O BS-4317 c1cc2cc(ccc2c(c1)S(=O)(=O)O)N BS-4318 CCOC(=O)CC(c1ccc(cc1)OC)N BS-4319 CCCn1c(=O)c2c(cc([nH]2)C)[nH]c1=S BS-4320 Cc1c(nnn1c2ccc(cc2)Cl)CO BS-4321 CCOc1ccc(cc1OCC)CC(=O)O BS-4322 CC(C)(C)C1CCC2(CC1)C(=O)NC(=O)N2 BS-4323 COCCCNC(=S)Nc1ccccc1 BS-4324 c1cc2c(cc1Cl)cc(c(=O)o2)C(=O)O BS-4325 c1cc(c(cc1S(=O)(=O)NN)Cl)F BS-4326 c1nc2c(c3c(s2)CCCC3)c(n1)Cl BS-4327 CCOC(=O)C(=O)Nc1ccc(c(c1)F)C BS-4328 COc1cccc(c1OC)C(CC(=O)O)N BS-4329 Cc1ccc(cc1)c2cc3c(=O)[nH]ccn3n2 BS-4330 C1CCC(CC1)CN2CC(CC2=O)C(=O)O BS-4331 Cc1ccc(cc1)c2nc(on2)CN.Cl BS-4333 CNCc1nc(no1)c2ccccc2.Cl BS-4334 C1CCC2(CC1)C(=O)N(C(=O)N2)CC(=O)O BS-4335 CCCn1c(=O)c2c(ccs2)[nH]c1=S BS-4336 c1cc(ncc1C(=O)N2CCOCC2)Cl BS-4337 c1ccc(cc1)C(=O)N2CCNCC2.Cl BS-4338 CC(=O)CS(=O)(=O)c1ccc(cc1)OC BS-4339 c1cc(=O)[nH]cc1S(=O)(=O)N2CCCC2 BS-4340 CC(C)Cc1ccc(cc1)c2ccc(=O)[nH]n2 BS-4341 CCc1ccc2c(c1)c(=O)c3c([nH]2)CCNC3 BS-4342 Cc1ccc(c2c1c(=O)c3c([nH]2)CCNC3)C BS-4343 Cc1cc(ccc1Br)NC(=O)N BS-4344 Cc1ccc(c(c1)Br)NC(=O)N BS-4345 CCOC(=O)C(=O)Nc1ccc(c(c1)F)F BS-4346 c1ccc(cc1)NNc2c(cccn2)C(=O)O BS-4347 c1ccc(cc1)c2cc3n(n2)C(CNC3=O)O BS-4348 Cc1c(c(sc1C(=O)OC)N)C(=O)OC BS-4349 CC(C)(C)OC(=O)N1CCCC1C(=O)NN BS-4350 CC(C)(C)OC(=O)N1CCCC1/C(=N/O)/N BS-4351 Cc1cc(=O)[nH]c(n1)N(C)Cc2ccccc2 BS-4352 Cc1ccc(cc1)c2nc(on2)C3CCCN3 BS-4353 CCCCNc1c(cccn1)S(=O)(=O)N BS-4354 C1CC1c2nc(on2)C3CCNCC3.Cl BS-4355 c1ccc(cc1)c2c3n(nn2)C(CNC3=O)O BS-4356 Cc1nc(cc(n1)NN)c2ccc(cc2)OC BS-4357 Cc1ccc(cc1C)n2c(c(nn2)C(=O)N)C BS-4358 COc1cc(c(cc1NC(=O)N)Cl)OC BS-4359 COc1ccccc1C(=O)NCCN.Cl BS-4360 CCOc1ccccc1NC(=O)CN.Cl BS-4361 CCOC(=O)/C(=N/Nc1ccc(cc1)C)/C#N BS-4362 CCc1ccccc1n2c(c(nn2)C(=O)O)C BS-4364 CCc1c(nnn1c2ccc(cc2)C)C(=O)O BS-4365 Cc1cc(cc(c1)n2c(c(nn2)C(=O)O)C)C BS-4366 Cc1ccc(cc1C)n2c(c(nn2)C(=O)O)C BS-4367 COc1ccc(cc1)C2Cn3c(cnn3)CO2 BS-4368 Cc1ccc(cc1)n2c(c(nn2)C(=O)NN)C BS-4369 Cc1cccc(c1C)n2c(c(nn2)C(=O)N)N BS-4370 Cc1ccc(cc1)n2c(c(nn2)/C(=N/O)/N)C BS-4371 CCc1ccc(cc1)n2c(c(nn2)C(=O)N)N BS-4372 c1cnc(cn1)c2nc(on2)C3CCCCN3 BS-4373 c1ccc2c(c1)CN(C(=O)CO2)C3CCCC3 BS-4374 Cc1ccc(cc1)C2=NOC3(N2)CCNCC3 BS-4375 CC(C)c1nc(on1)C2CCCCN2.Cl BS-4376 c1ccc(c(c1)F)S(=O)(=O)CC(=O)NN BS-4377 CCOC(=O)c1nc(no1)c2ccc(cc2)C BS-4378 COc1ccccc1c2cc([nH]n2)C(=O)OC BS-4379 Cc1ccccc1c2nc(on2)CCC(=O)O BS-4380 Cc1cc(n(n1)C(=O)c2cnc(nc2)OC)C BS-4381 c1cc(ccc1C2=NC3(CCCC3)NC2=O)F BS-4382 Cc1cc(cc2c1[nH]c3c(c2=O)CNCC3)F BS-4383 COc1ccc(cc1OC)S(=O)(=O)NN BS-4384 COc1ccc(c(c1)S(=O)(=O)NN)OC BS-4385 c1cc2c(cc1c3ccc(=S)[nH]n3)OCO2 BS-4386 CCc1ccc(cc1)N2CC(CC2=O)C(=O)N BS-4387 Cn1cccc1c2nc(on2)C3CCNCC3 BS-4388 CCOC(=O)c1c(nc(s1)SCC)N BS-4389 c1ccc(cc1)CN2CCC(CC2)NC(=N)N BS-4390 c1cc(ccc1/C(=C\2/CCCCN2)/C#N)Cl BS-4391 c1cc(c(cc1Br)F)NC(=O)N BS-4392 c1cc(ccc1c2c(c[nH]n2)C(=O)O)[N+](=O)[O-] BS-4393 Cc1c(nnn1c2ccc(cc2)OC)C(=O)O BS-4394 Cc1c(nnn1c2cccc(c2)OC)C(=O)O BS-4395 COc1ccccc1n2c(c(nn2)C(=O)N)N BS-4396 COc1ccc(cc1)n2c(c(nn2)C(=O)N)N BS-4397 Cc1cccc(c1N2CC(CC2=O)C(=O)O)C BS-4400 Cc1ccc(c(c1)N2CC(CC2=O)C(=O)O)C BS-4401 Cc1ccc(cc1C)N2CC(CC2=O)C(=O)O BS-4402 Cc1cc(cc(c1)N2CC(CC2=O)C(=O)O)C BS-4403 Cc1ccc(c(c1)C)N2CC(CC2=O)C(=O)O BS-4404 CCc1ccc(cc1)N2CC(CC2=O)C(=O)O BS-4405 Cc1ccc(cc1)CN2CC(CC2=O)C(=O)O BS-4406 Cc1ccccc1CN2CC(CC2=O)C(=O)O BS-4407 Cc1cccc(c1)N2CC(CC2=O)/C(=N/O)/N BS-4408 c1ccc(cc1)CN2CC(CC2=O)/C(=N/O)/N BS-4409 Cc1ccc(cc1)N2CC(CC2=O)/C(=N/O)/N BS-4410 c1ccc2c(c1)C(=NC3(N2)CCNCC3)S BS-4411 c1cc(c(cc1Cl)F)S(=O)(=O)CC#N BS-4412 c1cc(c(cc1Cl)S(=O)(=O)CC#N)F BS-4413 c1nc(no1)c2c3n(c(=O)[nH]c2=O)CCCC3 BS-4414 Cc1c(nnn1Cc2cccc(c2)F)C(=O)N BS-4415 CCOC(=O)c1c(c2cc(ccc2[nH]1)OC)N BS-4416 COc1ccc(cc1)N2CC(CC2=O)C(=O)N BS-4417 c1cn2c(c(n1)N3CCCC(C3)N)n[nH]c2=O BS-4418 COc1cccc(c1)c2cc(=O)[nH]c(=S)[nH]2 BS-4419 COc1ccc(cc1)c2cc(=O)[nH]c(=S)[nH]2 BS-4420 COC(=O)c1c(c(cs1)c2ccccn2)N BS-4421 COc1ccc(cc1)N2CCN(CC2)C(=N)N BS-4422 CC(C)(C)C1CCc2c(sc(c2C#N)N)C1 BS-4423 c1ccc(c(c1)O)OCc2ccc(cc2)Cl BS-4424 Cc1cc(n(n1)C(=O)c2cccc(c2)Cl)C BS-4425 Cc1c(cccc1Cl)NC(=O)CN.Cl BS-4426 CCn1cc(c(=O)c2c1ccc(c2)F)C(=O)O BS-4427 Cc1nc(nn1c2cccc(c2)F)C(=O)OC BS-4428 Cc1ccc(cc1F)n2c(c(nn2)C(=O)O)C BS-4429 CCc1c(nnn1c2ccc(cc2)F)C(=O)O BS-4430 CCc1c(nnn1c2cccc(c2)F)C(=O)O BS-4431 Cc1cc(ccc1F)n2c(c(nn2)C(=O)O)C BS-4432 Cc1cc(ccc1n2c(c(nn2)C(=O)O)C)F BS-4433 Cc1ccc(c(c1)F)n2c(c(nn2)C(=O)O)C BS-4434 Cc1c(nnn1c2ccc(cc2)F)/C(=N/O)/N BS-4435 c1cc(cc(c1)F)Cn2c(c(nn2)C(=O)N)N BS-4436 CCC(C(=O)O)N1c2ccccc2OCC1=O BS-4437 COc1ccccc1N2CC(CC2=O)C(=O)O BS-4438 c1cc(sc1)c2cc3n(n2)C(CNC3=O)O BS-4439 c1c2cc3c(cc2nc(c1C=O)Cl)OCO3 BS-4440 CCOC(=O)c1nc(on1)c2ccc(cc2)F BS-4441 COC(=O)c1c(n(nn1)c2cccc(c2)F)N BS-4442 Cc1c(nnn1c2cccc(c2)F)C(=S)N BS-4443 c1[nH]c(=O)c2c(n1)nc(s2)N3CCCCC3 BS-4444 CCN(CC)CCOC(=O)c1ccc(cc1)N.Cl BS-4445 c1ccc(cc1)NC(=S)NCC2CCCO2 BS-4446 CCOC(=O)C(=O)N1CCCC(C1)N.Cl BS-4447 c1ccc(cc1)c2cc3[nH]nc(c(=O)n3n2)C#N BS-4448 Cc1ccc(cc1F)N2CC(CC2=O)C(=O)O BS-4449 Cc1cc(ccc1N2CC(CC2=O)C(=O)O)F BS-4450 c1ccc(c(c1)CN2CC(CC2=O)C(=O)O)F BS-4451 c1cc(ccc1N2CC(CC2=O)/C(=N/O)/N)F BS-4452 c1cc(cc(c1)F)N2CC(CC2=O)/C(=N/O)/N BS-4453 CCOC(=O)C(=O)Nc1cc(ccc1OC)C BS-4454 CCOc1ccc(cc1)NC(=O)C(=O)OCC BS-4455 CCOc1ccccc1NC(=O)C(=O)OCC BS-4456 CCOC(=O)c1c(cc(=O)n2c1CCCC2)O BS-4457 Cc1c(sc(n1)C)c2cc([nH]n2)C(=O)OC BS-4459 COC(=O)c1cc(=O)c2cc(ccc2[nH]1)Cl BS-4461 c1cc(cc(c1)Cl)n2c(c(nn2)C(=O)N)N BS-4462 C=CCN1Cc2cc(ccc2OCC1=O)Cl BS-4463 c1cc2c(cc1Cl)CN(C(=O)CO2)C3CC3 BS-4464 COc1cc(cc(c1OC)OC)/C=C/C(=O)O BS-4465 CCCCNc1ccc(cc1[N+](=O)[O-])C(=O)O BS-4466 CC(C)Cn1c(=O)c2c(cn(n2)C)[nH]c1=S BS-4467 C1CCc2c(c3c(=O)[nH]c(=S)[nH]c3s2)C1 BS-4468 COC(=O)c1cc2cc(ccc2oc1=O)Cl BS-4469 c1cc(c(cc1N2CC(CC2=O)C#N)Cl)F BS-4470 c1cc(ccc1N2CC(CC2=O)C(=O)N)Cl BS-4471 c1cc(cc(c1)Cl)N2CC(CC2=O)C(=O)N BS-4472 COC(=O)c1cc(=O)c2cc(c(cc2[nH]1)F)F BS-4473 COC(=O)c1cc(=O)c2cc(cc(c2[nH]1)F)F BS-4474 Cc1c(nnn1c2cc(cc(c2)F)F)C(=O)O BS-4475 c1ccc(cc1)c2nc(on2)c3ccc[nH]c3=O BS-4476 COC(=O)C1=C(c2ccccc2S1(=O)=O)N BS-4477 CC1(OC(=O)C(=C2CCCCCN2)C(=O)O1)C BS-4478 CCOc1cc(cc(c1OCC)N)C(=O)OC BS-4479 CCc1ccc(cc1)c2cc3c(=O)[nH]ccn3n2 BS-4480 Cc1ccc(cc1C)c2cc3c(=O)[nH]ccn3n2 BS-4481 Cc1ccc(c(c1)C)c2cc3c(=O)[nH]ccn3n2 BS-4482 c1cc(sc1)CCN2CC(CC2=O)C(=O)O BS-4483 c1cc(sc1)CN2CC(CC2=O)/C(=N/O)/N BS-4484 c1cc(ccc1N2CC(CC2=O)C(=O)O)Cl BS-4485 c1cc(cc(c1)Cl)N2CC(CC2=O)C(=O)O BS-4486 c1ccc(cc1)c2[nH]c(=O)cc(n2)C(F)(F)F BS-4487 COc1cc(c(cc1OC)NC(=O)N)C(=O)O BS-4488 c1ccc(cc1)c2nc(on2)c3cnc[nH]c3=O BS-4489 c1cc(=O)[nH]cc1c2nc(no2)c3ccncc3 BS-4490 COC(=O)CN1C(=O)C2(CCCCC2)NC1=O BS-4491 c1ccc(cc1)CNc2nc3ccccc3s2 BS-4492 c1ccc(cc1)C(=O)NC2CCCNC2.Cl BS-4493 c1ccc(cc1)C(=O)NC2CCNCC2.Cl BS-4494 c1ccc(cc1)C(=O)N2CCC(CC2)N.Cl BS-4495 c1ccc(cc1)C(=O)N2CCCC(C2)N.Cl BS-4496 Cc1ccc2c(c1)CCCN2C(=O)CN.Cl BS-4497 c1cc(c(cc1N2CC(CC2=O)C(=O)O)F)F BS-4498 c1c(cc(cc1F)F)N2CC(CC2=O)C(=O)O BS-4499 c1cc(=O)[nH]cc1c2nc(no2)c3cnccn3 BS-4500 CCOC(=O)c1ccn(n1)c2ccc(cc2)C#N BS-4501 COc1cccc(c1)c2cc3c(=O)[nH]ccn3n2 BS-4502 COc1ccccc1c2cc3c(=O)[nH]ccn3n2 BS-4503 COc1ccc(cc1)c2cc3c(=O)[nH]ccn3n2 BS-4504 CCOC(=O)CSc1ccccc1[N+](=O)[O-] BS-4505 CC(=O)c1ccc2c(c1)Nc3ccccc3S2 BS-4506 c1cc(c(nc1)N2CCCCC2)S(=O)(=O)N BS-4507 c1c(c(c2n(c1=O)CCCCC2)C(=O)O)Cl BS-4508 CCOC(=O)C(=O)Nc1cccc(c1C)Cl BS-4509 COc1ccc(cc1)c2nc(on2)CN.Cl BS-4510 COC(=O)c1c(n(nn1)CC(=O)N)C(=O)OC BS-4511 c1cc(=O)[nH]nc1c2nc(no2)c3cnccn3 BS-4512 CCOC(=O)CSc1c(cccn1)[N+](=O)[O-] BS-4513 COc1ccc(cc1)COc2ccccc2C=O BS-4514 CCOC(=O)C(=O)NNC(=O)C1CCCCC1 BS-4515 CCc1ccc(cc1)Nc2c(cccn2)C(=O)O BS-4516 c1ccc(cc1)C2=N/C(=C\3/CCCCN3)/C(=O)O2 BS-4517 c1cc(c(=O)[nH]c1)S(=O)(=O)N2CCCCC2 BS-4518 CC(C)(C)OC(=O)NC1(CCCCC1)C(=O)N BS-4519 c1ccc(cc1)C2=NC3(CCCCCC3)NC2=O BS-4520 c1ccc(cc1)CNC(=S)Nc2ccccc2 BS-4521 CC(C)c1ccc(cc1)c2csc(n2)CC#N BS-4522 c1cc(c(cc1Cl)Cl)CNC(=O)CC#N BS-4523 c1cc(ccc1c2nc(on2)CN)C(F)(F)F BS-4524 COc1ccc(cc1)n2c3c(c(=O)[nH]cn3)nn2 BS-4525 c1cc(ccc1CN2CCCC2=O)C(F)(F)F BS-4526 c1ccc(c(c1)CNc2ccc(cc2)C(=O)O)O BS-4527 Cc1ccc(cc1)c2cc3n(n2)C(CNC3=O)O BS-4528 Cc1c(nnn1c2ccc3c(c2)CCC3)C(=O)O BS-4529 CC(C)(C)OC(=O)N1CCCC(C1)CC(=O)O BS-4530 CC1(CCCN(C1)C(=O)OC(C)(C)C)C(=O)O BS-4531 CC(C)(C)OC(=O)NC1(CCCCC1)C(=O)O BS-4532 c1ccc(cc1)c2nc(on2)C3(CCCCC3)N BS-4533 CC(=O)Nc1ccc(cc1)NC(=O)CN.Cl BS-4534 Cc1ccc(cc1)c2cc3c(nccn3n2)Cl BS-4535 c1ccc(cc1)c2ccc(=O)n(n2)CCC(=O)O BS-4536 COc1ccc(cc1)S(=O)(=O)CC(=O)OC BS-4537 c1cc(c(=O)[nH]c1)S(=O)(=O)N2CCOCC2 BS-4538 c1ccc(cc1)n2c(=O)c3c(ccs3)[nH]c2=O BS-4539 c1cc(cnc1)c2nc(on2)C3(CCCCC3)N BS-4540 COC(=O)c1ccc(cc1)NC(=O)CN.Cl BS-4541 COC(=O)c1c(c(n[nH]1)C2CC2)Br BS-4542 Cc1ccc(c(c1)Br)NC(=S)N BS-4543 COC(=O)CN1CCCC(C1)N.Cl.Cl BS-4544 c1ccc(cc1)C2Cn3c(c(nn3)C(=O)O)CO2 BS-4545 c1cc(cc(c1)C(F)(F)F)C2(CCNCC2)O BS-4546 c1cc(sc1)c2nc(on2)c3ccc(=O)[nH]c3 BS-4547 c1cc(=O)[nH]cc1c2nc(no2)c3ccsc3 BS-4548 CCCn1cc(c(=O)c2c1ccc(c2)C)C(=O)O BS-4549 c1ccc2c(c1)CCC2N3CC(CC3=O)C(=O)O BS-4550 c1cc2c(c(c1)C(=O)O)C(=O)N(C2)C3CCCC3 BS-4551 c1cc2c(cc1N3CC(CC3=O)C(=O)O)CCC2 BS-4552 CCOC(=O)c1c([nH]nc1N)c2ccc(cc2)C BS-4553 Cc1ccc(cc1)c2nc(c(o2)C)C/C(=N/O)/N BS-4554 CCc1ccc(cc1)n2c(c(nn2)C(=O)O)CC BS-4555 CCc1ccccc1n2c(c(nn2)C(=O)O)CC BS-4556 CCc1c(nnn1c2cc(cc(c2)C)C)C(=O)O BS-4557 Cc1ccc(cc1)Cn2c(c(nn2)/C(=N/O)/N)C BS-4559 c1cnc(cn1)c2nc(on2)CC3CCNCC3 BS-4560 CC1CCc2c(c3c(n2C(=O)C)CCC(C3)C)C1 BS-4562 c1cc(cc(c1)Cl)c2nc(on2)c3ccc[nH]3 BS-4563 c1cc(ccc1c2cc3c(=O)[nH]ccn3n2)Cl BS-4564 c1cc(cc(c1)Cl)c2cc3c(=O)[nH]ccn3n2 BS-4565 c1c(ncnc1N2CCC(CC2)N)C(F)(F)F BS-4566 Cc1nc(cc(n1)N2CCNCC2)C(F)(F)F BS-4567 c1cc(sc1)c2nc(on2)c3cnc[nH]c3=O BS-4568 c1cscc1c2nc(on2)c3cnc[nH]c3=O BS-4569 CCn1cc(c(=O)c2c1nc(cc2)C)C(=O)OC BS-4570 COc1ccc(cc1)c2c[nH]c(c2N)C(=O)OC BS-4571 COc1ccc(cc1OC)N2CC(CC2=O)C#N BS-4572 CCOc1ccc(cc1)c2cc([nH]n2)C(=O)NN BS-4573 Cc1ccc2c(c1)c3c([nH]2)c(=O)n(c(=S)[nH]3)N BS-4574 c1cc(cc(c1)N)C(=O)N/N=C/2\CCCCCN2 BS-4575 CC(C)CC1(NC(=S)C(=N1)c2ccccc2)C BS-4576 CN(c1ccccc1)C(=O)c2ccc(nc2)Cl BS-4577 Cc1c(nnn1c2ccc3c(c2)OCO3)C(=O)O BS-4578 c1cc(cc(c1)F)c2cc3n(n2)C(CNC3=O)O BS-4579 c1cc(ccc1c2cc3n(n2)C(CNC3=O)O)F BS-4580 CCc1c(nnn1c2ccc(cc2)OC)C(=O)O BS-4581 CCOc1ccccc1n2c(c(nn2)C(=O)O)C BS-4582 CCOc1ccc(cc1)n2c(c(nn2)C(=O)O)C BS-4583 c1ccc(cc1)C(Cn2cc(nn2)C(=O)NN)O BS-4584 COc1cccc(c1)Cn2c(c(nn2)C(=O)N)N BS-4585 CCOc1ccc(cc1)n2c(c(nn2)C(=O)N)N BS-4586 c1cc(ccc1c2nc(on2)C3CCCNC3)F BS-4587 c1ccc(cc1)C(=O)NC2(CCCCC2)C(=O)O BS-4588 Cc1cc(c(c(c1)C)N2CC(CC2=O)C(=O)O)C BS-4589 COc1ccc2c(c1)OC3(CCNCC3)CC2=O BS-4590 CCc1ccc(cc1)N2CC(CC2=O)/C(=N/O)/N BS-4591 Cc1cccc(c1)CN2CC(CC2=O)/C(=N/O)/N BS-4592 Cc1ccc(cc1)CN2CC(CC2=O)/C(=N/O)/N BS-4593 c1ccc(cc1)CCN2CC(CC2=O)/C(=N/O)/N BS-4594 c1ccc(cc1)CC(C#N)c2[nH]c3ccccc3n2 BS-4595 c1cc(ccc1c2cc3c(nccn3n2)Cl)F BS-4596 c1cc(c(nc1)N)C(=O)Nc2ccc(cc2)Cl BS-4597 c1ccc(c(c1)C(=O)O)I BS-4598 c1cc(cc(c1)F)c2ccc(=O)n(n2)CC(=O)O BS-4599 COc1ccc(c(c1)OC)c2cc([nH]n2)C(=O)O BS-4600 COc1ccccc1n2c(c(nn2)C(=O)OC)N BS-4601 COc1ccc(cc1)C(=O)NCC2CCCNC2 BS-4602 Cc1ccc(cc1)N2CCN(CC2)CCC(=O)O BS-4603 c1ccc(c(c1)N)SSc2ccccc2N BS-4604 COC(=O)CS(=O)(=O)c1ccccc1Cl BS-4605 CCc1c(nnn1c2ccc(c(c2)F)C)C(=O)O BS-4606 CCc1c(nnn1c2ccc(cc2C)F)C(=O)O BS-4607 CCc1c(nnn1Cc2ccccc2F)C(=O)O BS-4608 CCc1c(nnn1c2ccc(cc2F)C)C(=O)O BS-4609 CCc1c(nnn1c2cc(ccc2F)C)C(=O)O BS-4610 CCc1c(nnn1c2ccc(c(c2)C)F)C(=O)O BS-4611 CCOc1ccc(cc1)N2CC(CC2=O)C(=O)O BS-4612 Cc1ccc(c(c1)N2CC(CC2=O)C(=O)O)OC BS-4613 COc1cccc(c1)CN2CC(CC2=O)C(=O)O BS-4614 COc1ccccc1CN2CC(CC2=O)C(=O)O BS-4615 COc1ccc(cc1)CN2CC(CC2=O)C(=O)O BS-4616 CCc1ccc(cc1)C(=O)O/N=C(\CC(=O)N)/N BS-4617 COc1cccc(c1)N2CC(CC2=O)/C(=N/O)/N BS-4618 c1ccc(cc1)C(Cn2c(c(nn2)CO)CO)O BS-4619 c1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccccn2 BS-4620 Cc1c(nnn1c2ccc(cc2)SC)C(=O)O BS-4621 C1CCC(CC1)c2nc(no2)CN3CCCC3=O BS-4623 C1CCC(CC1)c2nc(on2)CN3CCCC3=O BS-4624 CN(C)CCn1c(=O)c2ccccc2[nH]c1=S BS-4625 Cc1cc2c([nH]1)c(=O)n(c(=S)[nH]2)C3CCCC3 BS-4626 Cc1cc(=O)[nH]c(n1)NCc2ccc(cc2)Cl BS-4627 c1cc(cc(c1)F)n2c(=O)cc(c(n2)C(=O)O)O BS-4628 c1cc(c(nc1)Nc2ccc(c(c2)F)F)C(=O)O BS-4629 c1ccc(cc1)C(=O)NCCCCC(C(=O)O)N BS-4630 CC(C)(C)OC(=O)NCC(=O)Nc1ccccc1 BS-4631 Cc1c(nnn1Cc2cccc(c2)F)C(=S)N BS-4632 COCCCn1c(=O)c2ccccc2[nH]c1=S BS-4633 CC(C)(C)c1c(sc(n1)n2cccc2)C(=O)O BS-4634 C1CCC(=CC1)CCNC(=O)CN2CCCC2=O BS-4635 c1cc(ccc1C(Cn2cc(nn2)C(=O)O)O)F BS-4636 COCc1c(nnn1c2ccc(cc2)F)C(=O)O BS-4637 COCc1c(nnn1c2cccc(c2)F)C(=O)O BS-4638 COCc1c(nnn1c2ccccc2F)C(=O)O BS-4639 CCOC(=O)C(=O)Nc1ccc2c(c1)OCCO2 BS-4640 CCOC(=O)c1cc(n(n1)CCC#N)C(=O)OC BS-4641 COC(=O)c1ccc2c(c1)[nH]c(=S)n(c2=O)N BS-4642 c1ccc(c(c1)F)S(=O)(=O)Cc2cccnc2 BS-4643 COC(=O)c1c(c(cs1)c2cccc(c2)F)N BS-4644 CC(C)(C)OC(=O)NCc1ccc(cc1)C(=O)O BS-4645 Cc1ccc(cc1NC(=O)OC(C)(C)C)C(=O)O BS-4646 CCOc1cc(=O)n2c(c1C(=O)OC)CCCC2 BS-4647 CCOc1cc(=O)n2c(c1C(=O)O)CCCCC2 BS-4648 CC(C)(C)OC(=O)Nc1ccc(cc1)/C(=N/O)/N BS-4649 c1ccc(cc1)NC(=O)C(Cc2cccnc2)C#N BS-4650 c1cc(ccc1CNC2(CCCCC2)C(=O)O)F BS-4651 CSc1cccc(c1)N2CC(CC2=O)C(=O)O BS-4652 Cc1ccc(cc1)Cn2cc(c3c2cccc3)CO BS-4653 Cc1nc(nn1c2ccc(cc2)Cl)C(=O)OC BS-4654 Cc1nc(nn1c2ccc(cc2)Cl)C(=O)NN BS-4655 c1cc(cc(c1)Cl)Cn2c(c(nn2)C(=O)N)N BS-4656 c1ccc(cc1)c2nc(on2)C3CCC[NH2+]3.[Cl-] BS-4657 COc1ccc(cc1)NC(=O)C(=O)NCC(=O)O BS-4658 COC(=O)c1cc2n(n1)CCC(C2=O)C(=O)OC BS-4659 COc1ccc(cc1)n2c(=O)c3ccccc3cn2 BS-4660 c1cc(ccc1N2CCN(CC2)CCC(=O)O)F BS-4661 COc1cc2c(cc1OC)nc([nH]c2=O)SC BS-4662 CC(C)(C)OC(=O)NCc1nnc2n1CCCC2 BS-4663 CC(C)CCn1c(=O)c2c(cn(n2)C)[nH]c1=S BS-4664 CCOC(=O)c1nc(no1)c2ccc(cc2)Cl BS-4665 c1cc(c(c2c1c(=O)c3c([nH]2)CCNC3)F)Cl BS-4666 c1cnccc1c2nc(on2)C3CCCN3.Cl BS-4667 CCOC(=O)c1c[nH]c2cc(c(cc2c1=O)F)F BS-4670 CCn1cc(c(=O)c2c1cc(c(c2)F)F)C(=O)O BS-4671 Cn1c2c(c(=O)n(c1=O)C)C(=O)CC(N2)C(=O)O BS-4672 CCOC(=O)C(=O)Nc1cc(cc(c1)OC)OC BS-4673 Cc1ccc(cc1)c2nc(on2)c3ccc[nH]c3=O BS-4674 c1cc(sc1)C(Cn2cc(nn2)C(=O)NN)O BS-4675 Cc1ccc(c(c1)Cl)N2CC(CC2=O)C(=O)O BS-4676 c1cc(ccc1CN2C(CCC2=O)C(=O)O)Cl BS-4678 c1cc(ccc1CN2CC(CC2=O)C(=O)O)Cl BS-4679 Cc1ccc(cc1Cl)N2CC(CC2=O)C(=O)O BS-4680 c1ccc(c(c1)CN2CC(CC2=O)C(=O)O)Cl BS-4681 c1cc(cc(c1)Cl)N2CC(CC2=O)/C(=N/O)/N BS-4682 Cc1ccc2cc(c(nc2c1)Cl)C=C(C#N)C#N BS-4683 CCC(C)N1Cc2cc(ccc2OCC1=O)Cl BS-4684 c1ccc(cc1)n2c(c(nn2)C(=O)O)n3cccc3 BS-4685 COC(=O)Cc1c(c(sc1C(=O)OC)N)C#N BS-4686 CCOc1cc(cc(c1OCC)OCC)C(=O)O BS-4687 CC(=O)N1CCc2c(sc(c2C(=O)OC)N)C1 BS-4688 CC(=O)CS(=O)(=O)c1ccc(cc1)C(C)(C)C BS-4689 Cc1ccc(cc1)CNc2nc3ccccc3s2 BS-4690 COc1cc(c(cc1NC(=O)CC#N)Cl)OC BS-4691 c1ccc(cc1)C(=O)N2CCC(CC2)CN.Cl BS-4692 c1cc(ccc1C(CN2CCC(CC2)N)O)Cl BS-4693 c1cc(c(cc1F)F)CN2CC(CC2=O)C(=O)O BS-4694 c1c(cc(cc1F)F)CN2CC(CC2=O)C(=O)O BS-4695 c1ccc(cc1)c2nc(on2)c3cccnc3S BS-4696 c1ccc(cc1)c2csc(c2n3cccc3)CO BS-4697 C[n+]1ccccc1Cl.[I-] BS-4698 Cc1c(nnn1c2ccc(c(c2)Cl)F)C(=O)O BS-4699 c1cc(c(cc1n2c(c(nn2)C(=O)N)N)Cl)F BS-4700 CC1C(=O)N(c2cc(ccc2O1)Cl)CC(=O)O BS-4701 COC(=O)c1c(cc(=O)n2c1CCCCC2)Cl BS-4702 C1CC1c2c(c([nH]n2)C(=O)N3CCOCC3)Cl BS-4703 c1cc(oc1)c2nc(no2)C3CCCNC3.Cl BS-4704 CCOC(=O)c1c(c2c(s1)cccc2Cl)N BS-4705 Cc1ccc2c(c1)c(=O)c3c([nH]2)CCN(C3)C(=O)C BS-4706 c1ccc(cc1)C2=N/C(=C\3/CCCCCN3)/C(=O)O2 BS-4707 c1ccc(cc1)c2nc(c3n2CCCCC3)C(=O)O BS-4708 COC(=O)c1c2n(c(n1)c3ccccc3)CCCC2 BS-4709 CC(=O)Nc1cccc(c1)c2nnc3n2CCCC3 BS-4710 c1cc(c(=O)[nH]c1)S(=O)(=O)N2CCCCCC2 BS-4711 COc1c(cccn1)S(=O)(=O)N2CCCCC2 BS-4712 COc1ccc(cn1)S(=O)(=O)N2CCCCC2 BS-4713 Cc1ccc(c(c1)c2csc3c2nc[nH]c3=O)C BS-4714 Cc1ccc(cc1)c2csc3c2ncn(c3=O)C BS-4715 c1cc(c(nc1)NN)S(=O)(=O)N2CCCCC2 BS-4716 Cc1ccc(cc1)C2=NC3(CCCCCC3)NC2=O BS-4717 c1cc(c(cc1N2CC(CC2=O)C(=O)N)Cl)F BS-4718 c1ccc2c(c1)cnn(c2=O)c3cccc(c3)Cl BS-4719 c1ccc(cc1)c2nc(on2)c3ccc(o3)[N+](=O)[O-] BS-4720 CC(c1nc(no1)c2ccc(cc2)C(F)(F)F)N BS-4721 c1ccc(c(c1)c2nc(on2)c3ccc(=O)[nH]c3)F BS-4722 c1ccc(cc1)/C(=N/OC(=O)c2ccc[nH]c2=O)/N BS-4723 Cc1ccc2c(c1)c3c([nH]2)c(=O)n(cn3)CC(=O)O BS-4724 c1ccc(c(c1)CNCc2ccc(cc2)C(=O)O)O BS-4725 Cc1c(c(c(cn1)CO)/C=N/Nc2ccccc2)O BS-4726 CCOC(=O)c1ccc(cc1)Nc2c(cccn2)N BS-4727 Cc1cccc(c1)N2CC(CC2=O)c3nc(no3)C BS-4729 Cc1ccc(c(c1)C)c2cc3n(n2)C(CNC3=O)O BS-4731 c1cc2c(cc1c3nnc4n3CCCCC4)OCO2 BS-4732 CC(C)(C)OC(=O)NCC1CCC(CC1)C(=O)O BS-4733 Cc1ccc(cc1)n2c(cnn2)CN3CCNCC3 BS-4734 c1cc(c(cc1F)N2CC(CC2=O)C(=O)O)Cl BS-4735 c1cc(c(cc1Cl)F)N2CC(CC2=O)C(=O)O BS-4736 CCOC(=O)C(=O)Nc1cc(ccc1OC)Cl BS-4737 c1ccc(cc1)c2c(c3c(nccn3n2)Cl)C=O BS-4738 Cc1ccc(cc1C)c2cc3c(nccn3n2)Cl BS-4739 c1cc(ccc1c2[nH]c(=O)cc(n2)C(F)(F)F)F BS-4740 CCc1cc2n[nH]c(=O)n2c(n1)c3ccc(cc3)F BS-4741 Cc1ccc(cc1)COC(=O)c2cnc(nc2)OC BS-4742 COC(=O)c1c2n(cn1)CC(OC2)c3ccccc3 BS-4743 CCOc1ccc(cc1)S(=O)(=O)CC(=O)OC BS-4744 CCOC(=O)CS(=O)(=O)/C(=C/1\CCCN1)/C#N BS-4745 Cc1ccccc1n2c(=O)c3c(ccs3)[nH]c2=O BS-4746 Cc1ccc(cc1)c2csc3c2NCN(C3=O)C BS-4747 CC1CCC2(CC1)NC(=S)C(=N2)c3ccccc3 BS-4748 c1ccc(cc1)c2nc(cc(n2)Cl)C(F)(F)F BS-4749 c1ccc(cc1)c2nc(on2)c3cncnc3Cl BS-4750 COc1cc2c(cc1OC)nc(nc2Cl)Cl BS-4751 COC(=O)/C(=C/N)/S(=O)(=O)c1ccccc1F BS-4753 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)N BS-4754 c1ccc2c(c1)CCC2N3CC(CC3=O)/C(=N/O)/N BS-4755 Cc1cccc(c1)CN2C(=O)C3(CCNC3)NC2=O BS-4756 Cc1ccc(cc1)CN2C(=O)C3(CCNC3)NC2=O BS-4757 c1ccc2c(c1)CN(C(=O)CO2)C3CCCCCC3 BS-4758 CC1CCC(CC1)N2Cc3ccccc3OCC2=O BS-4759 COc1cccc(c1)c2cc3c(nccn3n2)Cl BS-4760 COc1ccc(cc1)c2cc3c(nccn3n2)Cl BS-4761 COc1ccccc1c2cc3c(nccn3n2)Cl BS-4762 CCOc1cc(=O)n(nc1C(=O)O)c2ccccc2 BS-4763 Cc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)NN)O BS-4764 Cc1nc(cc(n1)N2CCC(CC2)N)C(F)(F)F BS-4765 CCCCOc1ccc(cc1)c2c(c[nH]n2)C(=O)O BS-4766 CCCCOc1ccc(cc1)c2cc([nH]n2)C(=O)O BS-4767 CN(C)/C=N/c1c(c2n(c1C(=O)OC)CCC2)C#N BS-4768 CCOC(=O)c1c[nH]c(=S)nc1c2ccccc2 BS-4769 COc1ccc(c(c1)c2csc(n2)CC#N)OC BS-4770 COc1ccc(cc1OC)c2csc(n2)CC#N BS-4771 c1cnc(cn1)c2nc(on2)c3cncnc3Cl BS-4772 CCc1ccc(cc1)NC(=O)c2ccc(nc2)Cl BS-4773 C1CCC(C1)CC(=O)N2CCC(CC2)CN.Cl BS-4774 Cc1c(nnn1c2ccc3c(c2)OCCO3)C(=O)O BS-4775 CCc1c(nnn1c2ccc3c(c2)OCO3)C(=O)O BS-4776 Cc1nc(on1)C2CC(=O)N(C2)c3ccc(cc3)F BS-4777 CCOC(=O)c1cnn(c1N)c2ccc(cc2)OC BS-4778 Cc1c(nc(o1)c2ccccc2OC)C/C(=N/O)/N BS-4779 COc1ccc(cc1)c2cc([nH]n2)C(=O)NCCO BS-4780 Cc1c(nc(o1)c2ccc(cc2)OC)C/C(=N/O)/N BS-4781 CCc1c(nnn1c2ccc(cc2)OCC)C(=O)O BS-4782 CCc1ccc(cc1)n2c(c(nn2)C(=O)O)COC BS-4783 c1cn2c(c3c(n2)CCCC3)c(=O)n1CCC(=O)O BS-4784 CC(=O)Cc1nc(sn1)NC(=O)c2ccccc2 BS-4787 CCOC(=O)C1CN(CCC1=O)Cc2ccccc2 BS-4788 CCOC(=O)c1c(c(cs1)c2ccc(cc2)C)N BS-4790 c1ccc(c(c1)Cn2c3c(c(=O)[nH]cn3)nn2)Cl BS-4791 c1nc(nn1CCO)C(=O)N2CCNCC2.Cl BS-4792 c1cc(cc(c1)F)CN2CCn3c(n[nH]c3=O)C2=O BS-4793 c1cc(sc1)c2cn3c(c(nn3)C(=O)O)c(=O)[nH]2 BS-4794 COc1ccc(cc1OC)c2cc([nH]n2)C(=O)NN BS-4795 Cc1nc(no1)c2c3n(c(=O)[nH]c2=O)CCCCC3 BS-4796 c1cc(ccc1C#N)NC(=O)Nc2ccc(cc2)C#N BS-4797 c1ccc(cc1)c2c3[nH]c(=O)c4ccccc4n3nn2 BS-4798 CC(C)(C)C(=O)c1c(n(nn1)c2ccccc2F)N BS-4799 C=CCn1c(=O)c2ccc(cc2nc1S)C(=O)O BS-4800 COC(=O)c1ccc2c(c1)nc3n(c2=O)CCS3 BS-4801 CC(=O)/C(=C/N(C)C)/C(=O)Nc1ccccc1OC BS-4802 COc1ccccc1CNC(=O)CN2CCCC2=O BS-4803 c1cc(c(cc1C(F)(F)F)NC(=O)CC#N)Cl BS-4805 c1cc(c(cc1NC(=O)CC#N)C(F)(F)F)Cl BS-4806 c1cc(c(cc1NC(=O)CC#N)Cl)C(F)(F)F BS-4807 COc1cc2c(cc1OC)nc(cc2OC)C(=O)O BS-4808 c1cc2c(cc1N3CC(CC3=O)C(=O)O)OCCO2 BS-4809 COCc1c(nnn1c2ccc(cc2)OC)C(=O)O BS-4810 c1cc(ccc1CN2C(=O)C3(CCNC3)NC2=O)F BS-4811 COc1ccccc1CN2CC(CC2=O)/C(=N/O)/N BS-4812 Cc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccccn2 BS-4813 Cc1ccc(cc1)S(=O)(=O)n2ccc(c2)C(=O)C BS-4814 Cc1ccc(cc1)S(=O)(=O)n2cccc2C(=O)C BS-4815 COc1ccc(cc1)c2csc(c2N)C(=O)OC BS-4816 COc1cccc(c1)c2csc(c2N)C(=O)OC BS-4817 c1ccc(cc1)CNc2c(cccn2)S(=O)(=O)N BS-4818 Cc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-4819 CC(=O)Cc1nc(sn1)Nc2ccc(cc2)OC BS-4820 c1ccc2c(c1)nc(s2)/C(=C/c3ccncc3)/C#N BS-4821 c1cc(cc(c1)Cl)c2cc3c(nccn3n2)Cl BS-4822 c1cc(ccc1c2cc3c(nccn3n2)Cl)Cl BS-4823 COCCn1c(=O)c2ccc(cc2[nH]c1=O)C(=O)O BS-4824 CCOC(=O)C(=CNc1ccccn1)C(=O)OCC BS-4825 COc1ccc(cc1OC)N2CC(CC2=O)C(=O)N BS-4826 c1cc(cc(c1)F)NC(=O)c2cnc(nc2N)S BS-4827 c1ccc(cc1)NS(=O)(=O)c2cccnc2NN BS-4828 Cc1ccc(cc1)CS(=O)(=O)c2ccccc2F BS-4829 Cc1cccc(c1)NC(=O)CNC(=O)OC(C)(C)C BS-4830 Cc1ccccc1NC(=O)CNC(=O)OC(C)(C)C BS-4831 CCc1ccc(cc1)S(=O)(=O)/C(=C/N(C)C)/C#N BS-4832 CCCc1c(sc(n1)n2cccc2)C(=O)OCC BS-4833 c1cc(cc(c1)Cl)c2ccc(=O)n(n2)CC(=O)O BS-4834 Cc1cc(ccc1F)n2c(c(nn2)C(=O)O)COC BS-4835 Cc1ccc(c(c1)F)n2c(c(nn2)C(=O)O)COC BS-4836 Cc1ccc(c(c1)n2c(c(nn2)C(=O)O)COC)F BS-4837 c1ccc(c(c1)C(Cn2cc(nn2)C(=O)NN)O)F BS-4838 COCCN1Cc2cc(ccc2OCC1=O)C(=O)O BS-4839 COc1ccc(cc1OC)N2CC(CC2=O)C(=O)O BS-4840 COc1ccc(c(c1)OC)N2CC(CC2=O)C(=O)O BS-4841 COc1ccc(cc1F)C2=NOC3(N2)CCNCC3 BS-4842 CCOC(=O)c1cn(nn1)CC(=O)c2ccsc2 BS-4843 CC(C)(C)OC(=O)N1CCCC1C(=O)n2ccnc2 BS-4844 Cc1cccc(c1)NC(=O)C(Cc2ccncc2)C#N BS-4845 Cc1ccccc1NC(=O)C(Cc2ccncc2)C#N BS-4846 Cc1cccc(c1)NC(=O)C(Cc2cccnc2)C#N BS-4847 Cc1ccccc1NC(=O)C(Cc2cccnc2)C#N BS-4848 Cc1ccc(cc1)NC(=O)C(Cc2cccnc2)C#N BS-4849 CCOC(=O)c1cc(c2cc(ccc2n1)Cl)OC BS-4850 CCc1c(nnn1c2ccc(c(c2)C)Cl)C(=O)O BS-4851 c1cc2c(cc1Cl)CN(C(=O)CO2)C3CCCC3 BS-4852 Cc1ccccc1c2nc(on2)C3CCCN3.Cl BS-4853 c1ccc(cc1)c2nc(on2)C3CCNCC3.Cl BS-4855 c1ccc(cc1)n2c(c(nn2)C(=O)O)c3ccccn3 BS-4856 c1ccc2c(c1)NC(=O)C3CCCCN3S2(=O)=O BS-4857 CC(C)(C)OC(=O)NCc1nnc2n1CCCCC2 BS-4858 COC(=O)CS(=O)(=O)c1ccc(c(c1)Cl)F BS-4859 CCOc1ccc(cc1Cl)c2c(c[nH]n2)C(=O)O BS-4860 CCOc1ccc(cc1Cl)c2cc([nH]n2)C(=O)O BS-4861 c1cc(cnc1)c2nc(on2)C3CCNCC3.Cl BS-4862 c1cc(cc(c1)Br)c2c(c[nH]n2)C(=O)O BS-4863 c1cc(ccc1c2cc([nH]n2)C(=O)O)Br BS-4864 CCc1c(nnn1Cc2ccc(cc2F)F)C(=O)O BS-4865 CCOC(=O)/C(=N/NC(=O)Cc1ccc(cc1)F)/N BS-4866 c1ccc(c(c1)Nc2c(cccn2)S(=O)(=O)N)F BS-4867 Cc1ccc(cc1)c2nc(on2)c3cccnc3NN BS-4868 CCOC(=O)c1cn(nn1)CC(c2cccs2)O BS-4869 CCCCn1cnc2c(c[nH]c2c1=O)c3ccccc3 BS-4871 CCOC(=O)c1c2c(sc1NC(=O)C)CCCC2 BS-4872 CCSc1nc2c(s1)c(=O)n3c(n2)CCCC3 BS-4873 c1cc(cc(c1)Cl)C(Cn2cnc(n2)C(=O)O)O BS-4874 c1cc(cc(c1)Cl)C(Cn2cc(nn2)C(=O)O)O BS-4875 Cc1c(nnn1c2ccc(c(c2)Cl)OC)C(=O)O BS-4876 c1cc(ccc1CCN2CC(CC2=O)C(=O)O)Cl BS-4877 COC(=O)c1c(c(cs1)c2cccc(c2)Cl)N BS-4878 COC(=O)c1c(c(cs1)c2ccc(cc2)Cl)N BS-4879 CCOC(=O)c1cn(c(n1)C(=O)OCC)CC(=O)C BS-4880 CCOC(=O)c1cc(n(n1)CC(=O)C)C(=O)OCC BS-4881 CC(C)(C)OC(=O)NCC(=O)Nc1cccc(c1)F BS-4882 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1)F BS-4883 CC(C)(C)OC(=O)NCC(=O)Nc1ccccc1F BS-4884 CCN.COc1cc(=O)n2c(c1C(=O)O)CCCC2 BS-4885 Cc1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S BS-4887 CSc1nc2ccccc2c(=O)n1c3ccccc3 BS-4888 c1ccc(cc1)NC2=NC3CS(=O)(=O)CC3S2 BS-4889 c1ccc2c(c1)nc(s2)/C(=C/c3cccs3)/C#N BS-4890 c1ccc(cc1)N2C(=O)NC3(N2)CCNCC3.Cl BS-4891 c1ccc(cc1)c2cn3c(cc(n3)C(=O)NN)c(=O)[nH]2 BS-4892 c1ccc(c(c1)NC(=O)C(Cc2ccncc2)C#N)F BS-4893 c1cc(ccc1NC(=O)C(Cc2ccncc2)C#N)F BS-4894 c1cc(cnc1)CC(C#N)C(=O)Nc2ccc(cc2)F BS-4895 Cc1ccc(cc1)NC(=O)c2cc3n(n2)CCCC3=O BS-4896 CN(C)/C=C(\C(=O)OC)/S(=O)(=O)c1ccccc1 BS-4898 Cc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2nccs2 BS-4899 CCc1c(nnn1c2ccc(c(c2)Cl)F)C(=O)O BS-4900 COc1ccc(cc1Cl)N2CC(CC2=O)C(=O)O BS-4901 COc1ccc(cc1N2CC(CC2=O)C(=O)O)Cl BS-4902 c1cc(cc(c1)F)c2nc(on2)C3CCCN3.Cl BS-4903 c1cc(ccc1c2nc(on2)C3CCC[NH2+]3)F.[Cl-] BS-4904 COC(=O)CCn1c(cc(n1)C(=O)OC)C(=O)OC BS-4906 COC(=O)c1ccn(n1)c2ccc(cc2)c3ncon3 BS-4907 COC(=O)c1c2c(=O)[nH]c(cn2nn1)c3ccccc3 BS-4908 Cc1ccc(cc1)N/N=C(\C(=O)OC)/S(=O)(=O)C BS-4910 c1ccc(cc1)c2c([nH]c(n2)c3cccc(c3)F)S BS-4911 CCC(=O)Nc1cccc(c1)c2nnc3n2CCCC3 BS-4912 CC(C)(C)c1ccc(cc1)S(=O)(=O)CC(=O)OC BS-4914 Cc1ccc(cc1)NC(=O)C(Cc2cccs2)C#N BS-4915 Cc1c(nnn1c2cccc(c2)C(F)(F)F)C(=O)O BS-4917 Cc1c(nnn1c2ccccc2C(F)(F)F)C(=O)O BS-4918 Cc1c(nnn1c2ccc(cc2)C(F)(F)F)C(=O)O BS-4919 Cc1nc(on1)c2ccnc(c2)n3cc(nc3)C(=O)O BS-4920 c1cc(cc(c1)F)c2nc(on2)c3cccnc3NN BS-4921 c1cc(c(nc1)NN)c2nc(no2)c3ccc(cc3)F BS-4922 COc1ccc(cc1OC)c2cc3c(=O)[nH]ccn3n2 BS-4923 c1ccc2c(c1)CN(C(=O)CO2)Cc3ccccc3F BS-4924 Cc1ccc(cc1F)N2Cc3ccccc3OCC2=O BS-4925 CCOC(=O)C1CN(CCC1=O)C(=O)OC(C)(C)C BS-4926 Cc1ccc(cc1)NCc2c(c3n(n2)CCC3)C(=O)O BS-4929 Cc1ccc(cc1)NC(=O)c2cc3n(n2)CCCC3O BS-4930 Cc1ccc(cc1)NC2CCCn3c2cc(n3)C(=O)O BS-4931 Cc1c2c([nH]c(=S)n(c2=O)N)sc1C(=O)OC BS-4932 Cc1cc2c([nH]1)c(=O)n(c(=S)[nH]2)Cc3ccccc3 BS-4933 Cc1ccc(cc1)c2nc(on2)c3cccnc3Cl BS-4934 Cc1ccc(cc1)c2nc(on2)c3ccnc(c3)Cl BS-4935 CCOC(=O)C(=O)Nc1cccc(c1)Br BS-4936 CCN1CCN=C1SC.I BS-4937 c1cc(cc(c1)C(Cn2cc(nn2)C(=O)NN)O)C#N BS-4938 Cc1ccc(cc1C)c2ccc(=O)n(n2)CCC(=O)O BS-4939 CCc1ccc(cc1)c2ccc(=O)n(n2)CCC(=O)O BS-4940 Cc1ccc(cc1)C2Cn3cnc(c3CO2)C(=O)OC BS-4941 Cc1ccc(c(c1)C)n2c(=O)c3c(ccs3)[nH]c2=O BS-4944 Cc1ccc(cc1)Cn2c(=O)c3c(ccs3)[nH]c2=O BS-4945 Cc1ccc(c(c1)n2c(=O)c3c(ccs3)[nH]c2=O)C BS-4946 CC(C)(C)OC(=O)N1CCCC(C1)C(=O)N(C)OC BS-4947 Cc1cccc(c1)C2=NC3(CCCCCC3)NC2=S BS-4949 Cc1cc(n(n1)S(=O)(=O)c2cccnc2Cl)N BS-4950 COC(=O)c1cc2cc(cc(c2oc1=O)Cl)Cl BS-4951 c1cc(ccc1c2cn3cc(nc3c(=O)[nH]2)C(=O)O)F BS-4952 c1cc(ccc1c2cn3c(cc(n3)C(=O)O)c(=O)[nH]2)F BS-4953 Cc1ccc(cc1)C2Cn3c(c(nn3)C(=O)OC)CO2 BS-4955 CCO/C=N/c1c(nnn1Cc2ccccc2)C(=O)N BS-4956 Cc1ccc(cc1)C2Cn3c(c(nn3)/C(=N/O)/N)CO2 BS-4957 COC(=O)c1cn[nH]c1S(=O)(=O)N2CCCCC2 BS-4958 Cc1ccc(cc1)Cn2c(=O)c3c(csn3)[nH]c2=O BS-4959 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)N BS-4960 COc1cccc(c1)c2nc(on2)CC3CCNCC3 BS-4962 Cc1ccc(c(c1)CN2C(=O)C3(CCNC3)NC2=O)C BS-4963 c1ccc(cc1)CN2CCc3c(c(=O)[nH]c(=S)[nH]3)C2 BS-4964 c1ccc(c(c1)c2nc(on2)c3ccc(=O)[nH]c3)Cl BS-4965 c1ccc(c(c1)c2nc(on2)c3ccc[nH]c3=O)Cl BS-4966 CCOC(=O)CS(=O)(=O)c1c(cccn1)[N+](=O)[O-] BS-4967 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)n3ccnc3 BS-4968 c1cc(ccc1C(=O)NCc2nnc3n2CCCC3)F BS-4969 c1cc(ccc1N2CCN(CC2)C(=O)n3ccnc3)F BS-4970 c1cc(cc(c1)Nc2c(cccn2)S(=O)(=O)N)C#N BS-4971 CCOC(=O)c1cc2c(nc(cn2n1)C)N3CCCC3 BS-4972 Cc1ccc(cc1)c2csc3c2[nH]c(=S)[nH]c3=O BS-4973 Cc1cccc(c1)n2c(=O)c3c(ccs3)[nH]c2=S BS-4974 Cc1ccccc1n2c(=O)c3c(ccs3)[nH]c2=S BS-4975 c1cc(cc(c1)Cl)c2[nH]c(=O)cc(n2)C(F)(F)F BS-4976 c1cc(ccc1c2nc(on2)CCn3ccnc3)Cl BS-4977 CC1CCN(CC1)S(=O)(=O)c2cccnc2Cl BS-4978 c1c(ncnc1N2CCC(CC2)C(=O)O)C(F)(F)F BS-4979 c1cc2c(cc1C(=O)O)nc([nH]c2=O)N3CCOCC3 BS-4980 CCc1c(nnn1c2ccc3c(c2)OCCO3)C(=O)O BS-4981 CC(C)(C)OC(=O)NCC(=O)Nc1cccc(c1)C#N BS-4983 CCOC(=O)c1cnn(c1N)CC(c2ccccc2)O BS-4984 CC(C)c1ccc(cc1)n2c(c(nn2)C(=O)O)COC BS-4985 c1cc(ccc1c2c(c3c(nccn3n2)Cl)C=O)F BS-4987 COc1ncc(cn1)COC(=O)c2cnc(nc2)OC BS-4988 c1ccc2c(c1)c3c(o2)c(=O)n(c(=S)[nH]3)CC(=O)O BS-4989 COC(=O)c1c2c(=O)[nH]c(cn2nn1)c3ccsc3 BS-4990 COC(=O)c1c2c(=O)[nH]c(cn2nn1)c3cccs3 BS-4991 c1ccc(c(c1)Cn2c(=O)c3c(ccs3)[nH]c2=O)F BS-4992 Cc1cc(ccc1F)n2c(=O)c3c(ccs3)[nH]c2=O BS-4993 COC(=O)c1c(n(cn1)CC(c2ccccc2)O)CO BS-4994 CCc1nc(no1)c2c3n(c(=O)[nH]c2=O)CCCCC3 BS-4995 COC(=O)c1ccc2c(c1)nc(n(c2=O)CC=C)S BS-4996 c1ccc(cc1)C(=O)NS(=O)(=O)c2ccc(cc2)N BS-4997 CCOC(=O)N1CCc2c(cc(nn2)N3CCCC3)C1 BS-4998 c1cc(ccc1C2=NC3(CCCCCC3)NC2=S)F BS-4999 CCOc1ccc(cc1)CC(=O)N2CCC(CC2)CN BS-5000 C1CCC2(CC1)Nc3c(c4c(s3)CCCC4)C(=O)N2 BS-5001 c1cc(ccc1c2nc(cc(n2)Cl)C(F)(F)F)F BS-5002 COc1ccc(cc1)COc2ccc(cc2C=O)Cl BS-5003 CN(C)/C=C(\C#N)/S(=O)(=O)c1ccc(s1)Cl BS-5004 COCc1c(nnn1c2ccc3c(c2)OCO3)C(=O)O BS-5005 CCOC(=O)c1cn(nn1)CC(=O)c2ccccc2F BS-5006 CCOc1cc(nc2c1cc(c(c2)OC)OC)C(=O)O BS-5007 COC(=O)c1c(n(nn1)CC(c2ccccc2)O)CO BS-5008 CCOc1ccccc1n2c(c(nn2)C(=O)O)COC BS-5009 CCOc1ccc(cc1)n2c(c(nn2)C(=O)O)COC BS-5010 c1cc2c(cc1CN3CC(CC3=O)/C(=N/O)/N)OCO2 BS-5011 COc1ccccc1C(Cn2cc(nn2)C(=O)NN)O BS-5012 COc1ccccc1C(Cn2cnc(n2)C(=O)NN)O BS-5013 CCc1cccc(c1)Nc2c(cccn2)S(=O)(=O)N BS-5014 CCc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5015 Cc1ccc(cc1C)Nc2c(cccn2)S(=O)(=O)N BS-5016 Cc1cc(cc(c1)Nc2c(cccn2)S(=O)(=O)N)C BS-5017 COc1ncc(cn1)C(=O)NCc2ccc(cc2)Cl BS-5018 c1cc(cc(c1)Cl)c2nc(no2)CN3CCCC3=O BS-5019 c1cc(ccc1OCC(=O)O)I BS-5021 c1cc(c(cc1Br)F)S(=O)(=O)CC#N BS-5022 CCOc1cc(=O)n(nc1C(=O)O)c2ccc(cc2)F BS-5023 c1ccc(cc1)C(=O)CS(=O)(=O)c2ccccc2F BS-5024 c1cc(ccc1CNC(=O)c2cnc(nc2N)S)F BS-5025 c1ccc(c(c1)n2c(=O)c3c(ccs3)[nH]c2=S)F BS-5027 CC(C)Cn1c(=O)c2cc3c(cc2[nH]c1=S)OCO3 BS-5028 Cc1cn2c(cc(n2)C(=O)O)c(n1)N3CCSCC3 BS-5029 CCc1ccc(cc1)NC(=O)CNC(=O)OC(C)(C)C BS-5030 Cc1ccc(cc1C)NC(=O)CNC(=O)OC(C)(C)C BS-5031 CCc1ccccc1NC(=O)CNC(=O)OC(C)(C)C BS-5032 Cc1cc(cc(c1)NC(=O)CNC(=O)OC(C)(C)C)C BS-5033 Cc1ccc(c(c1)NC(=O)CNC(=O)OC(C)(C)C)C BS-5034 Cc1cccc(c1C)NC(=O)CNC(=O)OC(C)(C)C BS-5035 Cc1ccc(cc1)NCc2cc3ccc(cc3[nH]c2=O)C BS-5036 CC(CC(C#N)(c1ccccc1)c2ccccc2)N(C)C BS-5037 CC(CN(C)C)C(C#N)(c1ccccc1)c2ccccc2 BS-5038 c1cc(cc(c1)Cl)c2ccc(=O)n(n2)CCC(=O)O BS-5039 c1cc(ccc1c2ccc(=O)n(n2)CCC(=O)O)Cl BS-5040 c1ccc(c(c1)C2Cn3c(c(nn3)C(=O)N)CO2)Cl BS-5041 c1cc(ccc1n2c(=O)c3c(ccs3)[nH]c2=O)Cl BS-5042 COc1ccc(cc1)COc2ccc(cc2CO)Cl BS-5043 c1ccc(cc1)c2nc(on2)CC3CCNCC3.Cl BS-5044 c1cc(ccc1c2csc(n2)CC#N)Br BS-5045 c1ccc(cc1)c2nc(on2)c3cccn4c3n[nH]c4=O BS-5046 CCOC(=O)c1cn(nn1)CC(c2ccccc2F)O BS-5047 COc1ccc(cc1OC)N2CC(CC2=O)/C(=N/O)/N BS-5048 COc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccccn2 BS-5049 COc1ccccc1/C=C(\C#N)/C(=O)Nc2ccccn2 BS-5050 COc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5051 Cc1ccc(cc1)Cn2cc(c3c2cccc3)C(=O)OC BS-5052 COC(=O)c1c2n(nc1CN3CCOCC3)CCCC2 BS-5054 CCc1ccc(cc1)NC(=O)C(Cc2ccncc2)C#N BS-5055 Cc1cc(cc(c1)NC(=O)C(Cc2ccncc2)C#N)C BS-5056 CCc1ccc(cc1)NC(=O)C(Cc2cccnc2)C#N BS-5057 CCc1ccccc1NC(=O)C(Cc2cccnc2)C#N BS-5058 Cc1cccc(c1C)NC(=O)C(Cc2cccnc2)C#N BS-5059 Cc1cc(cc(c1)NC(=O)C(Cc2cccnc2)C#N)C BS-5060 Cc1ccc(c(c1)C)NC(=O)C(Cc2cccnc2)C#N BS-5061 Cc1ccc(c(c1)NC(=O)C(Cc2cccnc2)C#N)C BS-5062 Cc1ccc(cc1)N2CCN(CC2)c3ncc(cn3)C#N BS-5063 c1ccc(cc1)c2cc3c(nccn3n2)N4CCC(C4)N BS-5064 c1csc2c1nc(n(c2=O)CCN3CCCC3)NN BS-5065 c1cc(ccc1c2cc([nH]n2)C(=O)NCC(=O)O)Cl BS-5066 c1cc(ccc1C2Cn3c(c(nn3)C(=O)O)CO2)Cl BS-5067 c1cc(ccc1CN2C(=O)C3(CCNC3)NC2=O)Cl BS-5068 Cc1ccc(cc1)c2nc(no2)C3CCCNC3.Cl BS-5070 Cc1ccc(cc1)c2nc(no2)C3CCNCC3.Cl BS-5071 CCN1c2cc(ccc2C(=O)NC13CCNCC3)Cl BS-5072 CC1(CCCNC1)c2nc(no2)c3ccccc3.Cl BS-5073 c1csc2c1[nH]c(=O)n(c2=O)c3cc(cc(c3)F)F BS-5074 COc1ccc2cc(c(=O)oc2c1)C(=O)c3ccccc3 BS-5075 Cc1ccc(cc1)N/N=C\2/c3ccccc3C(=O)OC2=O BS-5076 c1ccc(cc1)c2c3ccccc3n(c(=O)n2)CC(=O)O BS-5077 Cc1cn2c(cc(n2)C(=O)NCC(OC)OC)c(=O)[nH]1 BS-5078 Cc1ccccc1n2c(c(nn2)C(=O)O)c3ccncc3 BS-5079 Cc1cccc(c1)n2c(c(nn2)C(=O)O)c3cccnc3 BS-5080 Cc1cccc(c1)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5081 c1ccc(cc1)n2c(c(nn2)/C(=N/O)/N)c3ccncc3 BS-5082 CC1=NS(=O)(=O)N(C=C1C(=O)O)Cc2ccccc2 BS-5083 CCOC(=O)C1=CNS(=O)(=O)N=C1c2ccccc2 BS-5084 c1ccc(c(c1)F)S(=O)(=O)/C(=C/2\CCCCN2)/C#N BS-5085 c1ccc(c(c1)NCc2cccc(c2)F)S(=O)(=O)N BS-5086 COc1ccccc1NC(=O)C(Cc2ccccc2)C#N BS-5087 COc1ccccc1CC(C#N)C(=O)Nc2ccccc2 BS-5088 COc1cccc(c1)CC(C#N)C(=O)Nc2ccccc2 BS-5089 COc1ccc(cc1)CC(C#N)C(=O)Nc2ccccc2 BS-5090 Cc1ccc(cc1)NS(=O)(=O)c2ccc[nH]c2=S BS-5093 COc1ccc(cc1)c2cc3c4n[nH]c(=O)n4ccn3n2 BS-5095 Cc1cc(ccc1F)Nc2c(cccn2)S(=O)(=O)N BS-5096 Cc1ccc(cc1F)Nc2c(cccn2)S(=O)(=O)N BS-5097 Cc1ccc(c(c1)Nc2c(cccn2)S(=O)(=O)N)F BS-5098 Cc1ccc(c(c1)F)Nc2c(cccn2)S(=O)(=O)N BS-5099 Cc1ccc(cc1)Cn2c(=O)c(c3n(c2=O)CCC3)C#N BS-5100 COc1ccccc1NC(=O)C(Cc2ccncc2)C#N BS-5101 COc1cccc(c1)NC(=O)C(Cc2ccncc2)C#N BS-5102 COc1ccc(cc1)NC(=O)C(Cc2ccncc2)C#N BS-5103 COc1ccccc1NC(=O)C(Cc2cccnc2)C#N BS-5104 COc1cccc(c1)NC(=O)C(Cc2cccnc2)C#N BS-5105 COc1ccc(cc1)NC(=O)C(Cc2cccnc2)C#N BS-5106 CCc1ccc(cc1)n2c(c(cn2)C(=O)O)n3cccc3 BS-5107 Cc1ccc(cc1)c2nc(on2)c3c(cc([nH]c3=O)C)C BS-5108 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2[nH]ncn2 BS-5109 Cc1nc(on1)C2(CCCCC2)NC(=O)OC(C)(C)C BS-5112 c1ccc2c(c1)CCN(C2)c3[nH]c(=O)c4c(n3)CCCC4 BS-5113 CCc1c(nnn1c2ccc(c(c2)Cl)OC)C(=O)O BS-5114 Cc1ccc(cc1Cl)n2c(c(nn2)C(=O)O)COC BS-5115 Cc1cc(c(cc1Cl)OC)n2c(c(nn2)C(=O)O)C BS-5116 c1cc(cc(c1)Cl)C(Cn2cnc(n2)C(=O)NN)O BS-5117 c1cc(ccc1C(Cn2cnc(n2)C(=O)NN)O)Cl BS-5118 COc1ccc(cc1)c2nc(on2)C3CCC[NH2+]3.[Cl-] BS-5119 Cc1c(nnn1c2cccc(c2)Br)C(=O)O BS-5120 c1ccc(cc1)c2nc(on2)c3c4n(nn3)CCNC4=O BS-5121 c1cc(c(nc1)NN)S(=O)(=O)Nc2ccc(cc2)F BS-5122 Cc1cc(ccc1NC(=O)CNC(=O)OC(C)(C)C)F BS-5123 Cc1ccc(cc1NC(=O)CNC(=O)OC(C)(C)C)F BS-5124 Cc1ccc(c(c1)F)NC(=O)CNC(=O)OC(C)(C)C BS-5125 c1cc2n[nH]c(=O)n2cc1S(=O)(=O)N3CCCCC3 BS-5126 c1cc(cc(c1)NC(=O)C2CC2)c3nnc4n3CCCC4 BS-5127 CCc1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S BS-5129 CCN1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)N)C1 BS-5130 CC1(NC(=S)C(=N1)c2ccc(cc2)Br)C BS-5131 c1csc2c1[nH]c(=O)n(c2=O)CC(=O)NCC(=O)O BS-5132 COC(=O)c1cccn1Cc2nc(on2)c3ccccc3 BS-5133 CCOC(=O)c1cc2c(=O)[nH]c(cn2n1)c3ccccc3 BS-5134 COC(=O)c1cccn1Cc2nc(no2)c3ccccc3 BS-5135 CCOc1ccc(cc1)N2Cc3ccccc3OCC2=O BS-5136 Cc1cccc(c1)N2CC(CC2=O)c3nc(no3)C4CC4 BS-5138 COC(=O)c1c(c(cs1)c2ccccc2)n3cccc3 BS-5139 c1ccc(cc1)c2csc(c2n3cccc3)C(=O)NN BS-5140 CN(C)c1ccc(cc1)C(=O)NC2CCNCC2.Cl BS-5142 c1ccc(c(c1)n2c(c(nn2)C(=O)O)c3ccccn3)F BS-5143 c1ccnc(c1)c2c(nnn2c3cccc(c3)F)C(=O)O BS-5144 c1cc(cc(c1)F)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5145 CCOC(=O)c1cn(nn1)CC(=O)c2cccc(c2)C#N BS-5146 Cc1nc(no1)c2ccc(cc2)n3ccc(n3)C(=O)OC BS-5147 c1cc(c(cc1F)S(=O)(=O)/C(=C/2\CCCN2)/C#N)F BS-5148 c1cc(c(cc1F)F)S(=O)(=O)/C(=C/2\CCCN2)/C#N BS-5149 COc1ccccc1c2ccc(nn2)N3CCC(CC3)N BS-5153 Cc1ccc(cc1)c2cc([nH]n2)C(=O)N3CCC(CC3)N BS-5154 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1)Cl BS-5156 CCc1c(nnn1c2ccc(cc2)C(F)(F)F)C(=O)O BS-5157 CCc1c(nnn1c2cccc(c2)C(F)(F)F)C(=O)O BS-5158 CCc1c(nnn1c2ccccc2C(F)(F)F)C(=O)O BS-5159 CCc1nc(on1)c2ccc(nc2)n3cc(nc3)C(=O)O BS-5160 c1cc(c(nc1)Nc2cc(cc(c2)F)F)S(=O)(=O)N BS-5161 c1cc(c(nc1)Nc2ccc(c(c2)F)F)S(=O)(=O)N BS-5162 COc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2nccs2 BS-5164 COc1ccccc1/C=C(\C#N)/C(=O)Nc2nccs2 BS-5165 COc1cccc(c1)/C=C(\C#N)/C(=O)Nc2nccs2 BS-5166 Cc1cccc(c1)N2CC(CC2=O)c3nc(no3)C(C)C BS-5167 CCc1c(c2n(n1)CC(N2)c3ccccc3)C(=O)OCC BS-5169 CCOC(=O)Cn1c2c(c(=O)[nH]c(n2)C)sc1=S BS-5170 Cc1ccc(cc1)n2cc(nn2)C(=O)N3CCC(CC3)N BS-5171 CSc1cccc(c1)N2Cc3ccccc3OCC2=O BS-5172 c1cc(cnc1)CC(C#N)C(=O)Nc2ccc(cc2)Cl BS-5173 c1ccc(c(c1)NC(=O)C(Cc2cccnc2)C#N)Cl BS-5174 c1cc(cc(c1)Cl)NC(=O)C(Cc2cccnc2)C#N BS-5175 c1ccc2c(c1)C(=O)N(C2=O)CCn3cc(nn3)C(=O)O BS-5176 COc1ccccc1c2cn3c(c(nn3)C(=O)O)c(=O)[nH]2 BS-5177 c1cc2c(cc1c3nc(on3)C4=NNC(=O)CC4)OCO2 BS-5178 c1ccn(c1)c2c(nnn2c3ccc(cc3)F)C(=O)NN BS-5179 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1F)F BS-5180 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(c(c1)F)F BS-5181 Cc1ccc(cc1)n2ccc(=O)c(n2)C(=O)NNC(=O)C BS-5182 CCOC(=O)c1cn(nn1)CC(c2cccc(c2)C#N)O BS-5183 c1ccc(cc1)S(=O)(=O)c2cc3ccccc3oc2=O BS-5184 CC(C)c1ccc(cc1)c2ccc(=O)n(n2)CCC(=O)O BS-5186 CCOC(=O)CS(=O)(=O)/C(=C\1/CCCCCN1)/C#N BS-5188 c1ccc2c(c1)c3c(o2)c(=O)n(c(=S)[nH]3)C4CCCC4 BS-5189 COc1ccccc1NC(=O)C(Cc2cccs2)C#N BS-5190 CCc1ccc(cc1)NS(=O)(=O)c2ccccc2C#N BS-5191 Cc1cccc(c1)n2c(=O)c3c(c(sc3[nH]c2=O)C)C BS-5192 Cc1ccc(cc1C)Cn2c(=O)c3c(ccs3)[nH]c2=O BS-5193 CCOC(=O)C1CCN(CC1)C(C#N)c2ccc(cc2)C BS-5194 Cc1ccc(cc1)CSc2[nH]c(=O)c3c(n2)CCCC3 BS-5195 Cc1c(nnn1c2cccc(c2)OC(F)(F)F)C(=O)O BS-5196 c1cc(ccc1CN2CC(CC2=O)C(=O)O)C(F)(F)F BS-5197 COc1ccc(cc1F)c2nc(on2)c3ccc(=O)[nH]c3 BS-5198 CCCc1nc(on1)c2ccn3c(c2)nnc3CC(=O)O BS-5199 CC(C)c1nc(on1)c2ccn3c(c2)nnc3CC(=O)O BS-5200 CN(C)/C=C(/C(=O)OC)\S(=O)(=O)c1ccccc1F BS-5203 CCOC(=O)c1c[nH]nc1S(=O)(=O)N2CCCCC2 BS-5204 CCOc1ccc(cc1OCC)c2nnc3n2CCCC3 BS-5205 COc1ccc(cc1)c2c(c3c(nccn3n2)Cl)C=O BS-5206 c1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5207 c1ccc2c(c1)CN(C(=O)CO2)Cc3ccccc3Cl BS-5208 COc1ccc(cc1F)c2nc(on2)c3ccc(=O)[nH]n3 BS-5209 c1cscc1c2nc(on2)c3c4n(nn3)CCNC4=O BS-5212 COc1ccc(cc1)C2Cn3cnc(c3CO2)C(=O)OC BS-5213 Cc1nc(on1)c2ccc(nc2)N3CCCC(C3)C(=O)O BS-5214 Cc1c(c(on1)C)S(=O)(=O)N2CCC(CC2)C(=O)O BS-5215 COc1cccc(c1)Cn2c(=O)c3c(ccs3)[nH]c2=O BS-5217 CCOc1ccc(cc1)n2c(=O)c3cn[nH]c3[nH]c2=S BS-5218 CN(C)/C=N/c1c(csc1C(=O)OC)c2ccccc2 BS-5220 CCCCNC(=O)C1CC(=O)N(C1)c2ccc(cc2)CC BS-5221 Cc1cc(cc(c1)n2c(=O)c3c(ccs3)[nH]c2=S)C BS-5222 Cc1ccccc1c2csc3c2nc([nH]c3=O)SC BS-5223 CCCCN1CCCCC1C(=O)Nc2c(cccc2C)C BS-5224 c1ccc2c(c1)c3c(s2)NC4(CCCCC4)NC3=S BS-5225 c1ccc(c(c1)c2ccc(nn2)N3CCC(CC3)N)Cl BS-5226 c1cc(ccc1C(=O)N2CCC(CC2)CN)Cl.Cl BS-5227 c1cc(ccc1n2cc(nn2)c3nc(on3)C(=O)NN)F BS-5228 Cc1nc(cc(n1)N2CCC(CC2)C(=O)O)C(F)(F)F BS-5229 c1ccc2c(c1)CN(C(=O)CO2)Cc3ccc(cc3F)F BS-5230 CCOC(=O)NC(=O)CS(=O)(=O)c1ccccc1F BS-5231 Cc1cc(cc(c1)n2c(c(nn2)C(=O)OC)C(=O)OC)C BS-5232 CCOC(=O)c1cn(nn1)CC(=O)c2ccccc2OC BS-5233 COC(=O)CN1C(=O)CCC(=N1)C(=O)Nc2ccccc2 BS-5234 CC(C)c1nc(on1)C2CC(=O)N(C2)c3ccccc3F BS-5236 c1ccc2c(c1)N(c3ccccc3S2(=O)=O)CC(=O)O BS-5237 c1cc(cc(c1)F)n2cc(nn2)C(=O)N3CCC(CC3)N BS-5238 c1ccc2c(c1)C3=NC(C(=O)N3C(=S)N2)CCC(=O)O BS-5239 c1ccc2c(c1)c3c([nH]2)c(=O)n(c(=S)[nH]3)CCC(=O)O BS-5240 Cc1ccc(cc1)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5241 Cc1nc(on1)c2ccc(cc2)CNC(=O)OC(C)(C)C BS-5242 Cc1nc(on1)C(c2ccccc2)NC(=O)OC(C)(C)C BS-5243 Cc1ccc(cc1)c2nc(on2)CNC(=O)OC(C)(C)C BS-5244 Cc1ccc(cc1NC(=O)OC(C)(C)C)c2nc(no2)C BS-5245 c1cc(c(nc1)Nc2ccc3c(c2)CCC3)S(=O)(=O)N BS-5247 c1cc(ccc1c2cn3c(c(nn3)C(=O)N)c(=O)[nH]2)Cl BS-5248 COc1ccc(cc1OC)c2cc3c(nccn3n2)Cl BS-5249 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2nccs2)Cl BS-5250 c1cc(ccc1c2cc3c(=O)[nH]ccn3n2)Br BS-5251 c1cc(cc(c1)Br)c2cc3c(=O)[nH]ccn3n2 BS-5252 Cc1ccc(cc1)C(Cn2cnc(c2CO)C(=O)OC)O BS-5253 CCn1c2c(c(n1)C)[nH]c(=S)n(c2=O)Cc3ccco3 BS-5254 CC(C)(C)OC(=O)NCC(=O)Nc1ccc2c(c1)CCC2 BS-5255 Cc1ccc(cc1)CN2CCN(CC2)C(=O)OC(C)(C)C BS-5256 c1ccc(c(c1)NC(=O)C(Cc2cccs2)C#N)Cl BS-5257 CC12CC(c3cccc(c3O1)OC)C(C(=O)N2)C(=O)OC BS-5258 Cc1ccc(cc1)C(Cn2c(c(nn2)C(=O)OC)CO)O BS-5259 CCOC(=O)c1cn(nn1)CC(c2ccccc2OC)O BS-5260 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3ccc(cc3)F BS-5261 c1cc(ccc1CN2CCc3c(c(=O)[nH]c(=S)[nH]3)C2)F BS-5262 CC(C)c1cccc(c1)Nc2c(cccn2)S(=O)(=O)N BS-5263 CC(C)c1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5264 CC(C)Cn1c(=O)c2c(c3cccnc3s2)[nH]c1=S BS-5267 CC(C)(C)OC(=O)CS(=O)(=O)c1cccnc1Cl BS-5269 c1cc(c2nncn2c1)S(=O)(=O)Nc3ccc(cc3)F BS-5270 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccccc2F BS-5271 Cc1ccc(cc1)C(=O)CS(=O)(=O)c2ccccc2F BS-5272 COC(=O)c1c2[nH]c(=O)c3ccccc3n2c(=S)s1 BS-5273 Cc1cc(ccc1n2c(=O)c3c(ccs3)[nH]c2=S)F BS-5274 Cc1cc(ccc1F)n2c(=O)c3c(ccs3)[nH]c2=S BS-5275 CSc1[nH]c(=O)c2c(n1)c(cs2)c3ccccc3F BS-5276 CSc1[nH]c(=O)c2c(n1)c(cs2)c3ccc(cc3)F BS-5277 CSc1[nH]c(=O)c2c(n1)c(cs2)c3cccc(c3)F BS-5278 CCc1ccc(cc1)NS(=O)(=O)c2ccc(nc2)NN BS-5279 CCc1ccc(cc1)NS(=O)(=O)c2cccnc2NN BS-5280 CC(C)c1ccc(cc1)NC(=O)CNC(=O)OC(C)(C)C BS-5281 CC(C)c1cccc(c1)NC(=O)CNC(=O)OC(C)(C)C BS-5282 c1cc(cc(c1)Cl)c2nc(cc(n2)Cl)C(F)(F)F BS-5283 COC(=O)CS(=O)(=O)c1ccc(cc1)Br BS-5284 c1cc(cc(c1)F)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5285 Cc1ccc(cc1)c2nc(on2)c3cccn4c3n[nH]c4=O BS-5286 COc1ccc(cc1OC)CCN2CC(CC2=O)C(=O)O BS-5287 CCOc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccccn2 BS-5288 Cc1ccc(cc1)/C(=N/OC(=O)c2c[nH]c3c2cccc3)/N BS-5289 COc1ccc(cc1OC)c2csc(c2N)C(=O)OC BS-5290 CCOc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5291 CC(=O)Cc1nc(sn1)Nc2ccc(c(c2)OC)OC BS-5292 Cc1ccc2c(c1)NN=C(S2(=O)=O)C(=O)N3CCCC3 BS-5293 CC(C)(C)OC(=O)N1CCCC(C1)c2nc(no2)C3CC3 BS-5294 CCOC(=O)c1cn(nn1)CC(=O)c2cccc(c2)Cl BS-5295 c1ccc(c(c1)C2Cn3c(c(nn3)/C(=N/O)/N)CO2)Cl BS-5296 c1cc(cnc1)c2nc(on2)c3cn(nn3)CCN.Cl BS-5297 c1cc(sc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5298 CC1CCC(CC1)N2Cc3cc(ccc3OCC2=O)Cl BS-5299 COC(=O)c1ccccc1NN=C(C(=O)OC)C(=O)OC BS-5300 c1ccc2c(c1)c(nc3n2nnc3c4ccc(cc4)F)NN BS-5301 COc1cccc2c1o/c(=N\c3ccccc3)/c(c2)C(=O)N BS-5302 CCc1cccc(c1)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5303 Cc1ccc(cc1C)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5304 CCc1ccccc1n2c(c(nn2)C(=O)O)c3ccccn3 BS-5305 c1ccc(cc1)Cn2c(c(nn2)C(=O)NN)c3ccncc3 BS-5306 CC1=NS(=O)(=O)N(C=C1C(=O)O)CCc2ccccc2 BS-5307 Cc1cccc(c1)CN2C=C(C(=NS2(=O)=O)C)C(=O)O BS-5308 CCOC(=O)C1=CN(S(=O)(=O)N=C1c2ccccc2)C BS-5309 c1ccc(c(c1)F)S(=O)(=O)/C(=C/2\CCCCCN2)/C#N BS-5310 CCOc1ccc(cc1)NC(=O)CNC(=O)OC(C)(C)C BS-5311 CCOc1ccccc1NC(=O)CNC(=O)OC(C)(C)C BS-5312 Cc1ccc(c(c1)NC(=O)CNC(=O)OC(C)(C)C)OC BS-5313 CCOC(=O)c1c2n(c(c1N)C(=O)OC(C)(C)C)CCC2 BS-5314 Cc1ccc(cc1)CC(C#N)C(=O)Nc2ccccc2OC BS-5315 Cc1ccccc1NC(=O)C(Cc2ccccc2OC)C#N BS-5316 Cc1cccc(c1)NC(=O)C(Cc2ccccc2OC)C#N BS-5317 Cc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)C#N BS-5318 Cc1cccc(c1)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5319 Cc1ccccc1NC(=O)C(Cc2cccc(c2)OC)C#N BS-5320 Cc1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5321 Cc1ccc(cc1)NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5322 Cc1ccccc1NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5323 Cc1cccc(c1)NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5324 CC(C)(C)OC(=O)NC1CCCN(C1)c2c(=O)[nH]ccn2 BS-5325 CCOC(=O)c1c(n(c(=S)s1)Cc2ccccc2)N BS-5326 c1cc(cc(c1)Cl)n2c(=O)c3c(ccs3)[nH]c2=S BS-5327 c1cc(ccc1n2c(=O)c3c(ccs3)[nH]c2=S)Cl BS-5328 c1ccc(c(c1)n2c(=O)c3c(ccs3)[nH]c2=S)Cl BS-5329 c1cc([nH]c1)c2nc(no2)c3ccc(cc3)OC(F)(F)F BS-5330 Cc1ccc(cc1)N/N=C(/C#N)\S(=O)(=O)CC(=O)OC BS-5331 CCOc1ccc(cc1)NC(=O)C(Cc2cccnc2)C#N BS-5332 Cc1ccc(cc1)n2c(c(nn2)C(=O)n3c(cc(n3)C)C)C BS-5333 CC(=O)N1CCC2(CC1)Nc3ccccc3S(=O)(=O)N2 BS-5334 Cc1nc(on1)C2CCC(CC2)CNC(=O)OC(C)(C)C BS-5335 CSc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5336 CSc1cccc(c1)Nc2c(cccn2)S(=O)(=O)N BS-5337 c1cc(ncc1S(=O)(=O)N2CCCC2)N3CCCCC3 BS-5338 Cc1ccc(cc1)CC(c2[nH]c3ccccc3n2)C(=S)N BS-5339 CCOC(=O)c1cn(nn1)CC(c2cccc(c2)Cl)O BS-5340 CCc1c(nnn1c2cc(c(cc2OC)Cl)C)C(=O)O BS-5341 CC(=O)Cc1nc(sn1)NC(=O)c2cccc(c2)Cl BS-5342 COc1cccc(c1)c2nc(no2)C3CCCNC3.Cl BS-5343 COc1cc(=O)n(nc1C(=O)OC)c2ccc(c(c2)F)F BS-5344 COc1ccccc1n2c(c(nn2)C(=O)O)c3ccccn3 BS-5345 COc1ccc(cc1)n2c(c(nn2)C(=O)O)c3cccnc3 BS-5346 c1csc2c1[nH]c(=S)n(c2=O)c3cc(cc(c3)F)F BS-5348 COc1cccc2c1OC(=C(C2)C(=O)N)Nc3ccccc3 BS-5349 COc1cc(ccc1O)CC(C#N)C(=O)Nc2ccccc2 BS-5350 CC(C)(C)OC(=O)C1=NN(c2ccccc2S1(=O)=O)C BS-5351 CC(C)(C)OC(=O)NCC(=O)Nc1cccc(c1)SC BS-5354 c1cc(ccc1c2nc(on2)CC3CCNCC3)F.[Cl-] BS-5355 c1cc(cc(c1)F)c2nc(on2)CC3CCNCC3.Cl BS-5356 Cc1ccc(cc1)NCc2cc3ccc(cc3nc2Cl)C BS-5357 c1cc(c2n[nH]c(=O)n2c1)c3nc(no3)c4ccc(cc4)F BS-5358 c1cc(cc(c1)F)c2nc(on2)c3cccn4c3n[nH]c4=O BS-5359 c1cc(ncc1c2nc(no2)C3CC3)n4cc(nc4)C(=O)O BS-5360 c1cc(c(nc1)n2cc(nc2)C(=O)O)c3nc(no3)C4CC4 BS-5361 COc1ccc(cc1F)Nc2c(cccn2)S(=O)(=O)N BS-5362 Cc1ccccc1c2nc(on2)Cn3cccc3C(=O)OC BS-5363 CCOc1cccc(c1)CN2Cc3ccccc3OCC2=O BS-5364 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccccc2 BS-5365 Cc1ccc(cc1C)S(=O)(=O)N2CCC(CC2)C(=O)O BS-5368 CNS(=O)(=O)c1cccnc1NN=C2CCN(CC2)C BS-5369 Cc1c(nnn1c2cc(c(cc2OC)OC)Cl)C(=O)O BS-5370 COCc1c(nnn1c2cc(ccc2OC)Cl)C(=O)O BS-5371 Cc1ccc(cc1Cl)Nc2c(cccn2)S(=O)(=O)N BS-5373 Cc1cc(ccc1Cl)Nc2c(cccn2)S(=O)(=O)N BS-5374 CN(C)c1cccc(c1)C(=O)N2CCC(CC2)CN.Cl BS-5375 c1ccc(c(c1)Cn2c(c(nn2)C(=O)O)c3ccncc3)F BS-5376 Cc1ccc(cc1F)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5377 Cc1ccc(c(c1)n2c(c(nn2)C(=O)O)c3ccncc3)F BS-5378 Cc1ccc(c(c1)n2c(c(nn2)C(=O)O)c3ccccn3)F BS-5379 Cc1ccc(c(c1)F)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5380 Cc1cc(ccc1n2c(c(nn2)C(=O)O)c3ccccn3)F BS-5381 Cc1ccc(cc1F)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5382 Cc1ccc(c(c1)n2c(c(nn2)C(=O)O)c3cccnc3)F BS-5383 Cc1cc(ccc1n2c(c(nn2)C(=O)O)c3ccncc3)F BS-5384 Cc1ccc(c(c1)F)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5385 CC1=NS(=O)(=O)N(C=C1C(=O)O)Cc2ccccc2F BS-5386 CC1=NS(=O)(=O)N(C=C1C(=O)O)Cc2ccc(cc2)F BS-5387 CCc1nc(no1)c2ccc(cc2)n3ccc(n3)C(=O)OC BS-5388 COc1ccccc1CC(C#N)C(=O)Nc2ccccc2F BS-5389 COc1ccccc1CC(C#N)C(=O)Nc2ccc(cc2)F BS-5390 COc1cccc(c1)CC(C#N)C(=O)Nc2ccc(cc2)F BS-5391 COc1cccc(c1)CC(C#N)C(=O)Nc2ccccc2F BS-5392 COc1ccc(cc1)CC(C#N)C(=O)Nc2ccc(cc2)F BS-5393 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)CC(=O)N2CCCC2 BS-5394 COC(=O)C1CCCCN1S(=O)(=O)c2ccccc2N BS-5395 c1ccc2c(c1)cc(/c(=N/c3ccc(cc3)Cl)/o2)C(=O)N BS-5396 Cc1cn2c(c(nn2)C(=O)N3CCC(C3)N)c(=O)[nH]1.Cl BS-5397 c1cc(ccc1NS(=O)(=O)c2ccc(nc2)NN)Cl BS-5398 c1cc(c(nc1)NN)S(=O)(=O)Nc2ccc(cc2)Cl BS-5399 c1cscc1c2nc(on2)c3cn(nn3)CCN.Cl BS-5400 Cc1ccc(cc1Cl)NC(=O)CNC(=O)OC(C)(C)C BS-5401 CCc1c(nnn1Cc2cccc(c2)C(F)(F)F)C(=O)O BS-5402 C=CCNC(=O)Cn1c(=O)c2c(c3ccccc3o2)[nH]c1=O BS-5403 CC(C)c1nc(on1)c2ccc(nc2)n3cc(nc3)C(=O)O BS-5404 CC(C)c1nc(on1)c2cccnc2n3cc(nc3)C(=O)O BS-5405 CCCc1nc(on1)c2cccnc2n3cc(nc3)C(=O)O BS-5406 CCc1nc(on1)c2ccnc(c2)n3c(c(cn3)C(=O)O)C BS-5407 CCOC(=O)c1nc(no1)c2cn(nn2)c3ccc(cc3)C BS-5408 CN(C)/C=C(\C(=O)OC)/S(=O)(=O)c1ccc(cc1)OC BS-5409 CCOc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2nccs2 BS-5410 Cc1nc(on1)C2(CCCCC2)NC(=O)Cc3ccccc3 BS-5411 CCOc1ccc(cc1)c2cc([nH]n2)C(=O)N3CCCCC3 BS-5412 CCc1cccc(c1)n2cc(nn2)C(=O)N3CCC(CC3)N BS-5413 CCc1ccc(cc1)n2cc(nn2)C(=O)N3CCC(CC3)N BS-5414 Cc1cc(cc(c1)n2cc(nn2)C(=O)N3CCC(CC3)N)C BS-5415 COCc1c(nnn1Cc2c(cccc2Cl)F)C(=O)O BS-5416 Cc1ccc(cc1)C(=O)c2cnc3ccc(cc3c2Cl)F BS-5417 C1CC1c2c(c([nH]n2)C(=O)N3CCOCC3)Br BS-5418 COC(=O)c1cn(nn1)CCN2C(=O)c3ccccc3C2=O BS-5419 COc1ccccc1c2cn3c(c(nn3)C(=O)OC)c(=O)[nH]2 BS-5420 c1cc(c(nc1)NN)S(=O)(=O)Nc2cc(cc(c2)F)F BS-5421 c1cc(c2n[nH]c(=S)n2c1)S(=O)(=O)N3CCOCC3 BS-5424 CCOc1ccccc1NC(=O)C(Cc2cccs2)C#N BS-5425 c1csc2c1nc3n(c2=O)C4CS(=O)(=O)CC4S3 BS-5426 CCc1c(nc(s1)n2cccc2)C(=O)n3c(cc(n3)C)C BS-5427 CCOc1ccc(cc1)NC(=S)NCCc2ccccc2 BS-5428 c1ccc(c(c1)n2c(c(nn2)C(=O)O)c3ccccn3)Cl BS-5429 c1ccc(c(c1)n2c(c(nn2)C(=O)O)c3ccncc3)Cl BS-5430 c1ccc(c(c1)n2c(c(nn2)C(=O)O)c3cccnc3)Cl BS-5431 c1cc(cnc1)c2c(nnn2c3ccc(cc3)Cl)C(=O)O BS-5432 c1cc(cc(c1)Cl)n2c(c(nn2)C(=O)O)c3cccnc3 BS-5433 c1cc(c(cc1Cl)S(=O)(=O)/C(=C/2\CCCN2)/C#N)F BS-5434 c1cc(c(cc1Cl)F)S(=O)(=O)/C(=C/2\CCCN2)/C#N BS-5435 c1ccc2c(c1)CC(=C(O2)Nc3ccc(cc3)Cl)C(=O)N BS-5436 c1ccc2c(c1)cnn(c2=O)c3cccc(c3)Br BS-5438 CCc1c(nnn1c2ccc(cc2)OC(F)(F)F)C(=O)O BS-5439 COCc1c(nnn1c2cccc(c2)C(F)(F)F)C(=O)O BS-5440 COCc1c(nnn1c2ccccc2C(F)(F)F)C(=O)O BS-5441 COCc1c(nnn1c2ccc(cc2)C(F)(F)F)C(=O)O BS-5442 CCOC(=O)c1cn2cc([nH]c(=O)c2n1)c3ccc(cc3)F BS-5443 c1ccn2c(c1)ncc(c2=O)C(=O)N3CCCC(C3)C(=O)O BS-5444 Cc1ccc(cc1)CN2c3ccccc3C(=O)CS2(=O)=O BS-5447 CCn1cc(c(n1)S(=O)(=O)N2CCCC2)C(=O)OCC BS-5448 Cc1ccc(cc1)n2c3c(cc(s3)C(=O)O)nc2N(C)C BS-5449 c1ccc(cc1)CN2CCN(CC2)C(=O)CN3CCCC3=O BS-5450 c1cc(c(nc1)Nc2ccc(c(c2)Cl)F)S(=O)(=O)N BS-5451 c1cc(c(nc1)Nc2ccc(c(c2)F)Cl)S(=O)(=O)N BS-5452 Cc1ccc(cc1Cl)n2c(c(cn2)C(=O)O)n3cccc3 BS-5453 COC(=O)c1c(c(cs1)c2ccc(c(c2)Cl)Cl)N BS-5455 c1ccnc(c1)c2c(nnn2c3cc(cc(c3)F)F)C(=O)O BS-5456 c1cnccc1c2c(nnn2c3cc(cc(c3)F)F)C(=O)O BS-5457 COC(=O)c1ccc2c(c1)[nH]c(=O)n(c2=O)NC(=O)CC#N BS-5458 COC(=O)c1c(n(cn1)CC(=O)c2ccccc2)C(=O)OC BS-5459 c1cc(sc1)Cn2c(=O)c3ccc(cc3[nH]c2=O)C(=O)O BS-5460 COc1ccccc1Cn\2c(=O)c3c(ccs3)[nH]/c2=N\N BS-5461 CC(C)(C)OC(=O)c1c(c(c2n1CCC2)C#N)/N=C/N(C)C BS-5462 Cc1ccc(cc1)c2csc(c2/N=C/N(C)C)C(=O)OC BS-5463 Cc1ccccc1c2csc3c2nc(n(c3=O)C)SC BS-5464 CCCCOc1ccc(cc1)C2=NC3(CCCC3)NC2=S BS-5465 c1cc(cc(c1)Cl)c2ccc3nnc(n3n2)CCC(=O)O BS-5466 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(c(c1)Cl)F BS-5467 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(c(c1)F)Cl BS-5468 c1ccc(c(c1)CN2CCN(CC2)c3ccc(cc3)Cl)O BS-5469 COc1cc2c(cc1OC)[nH]c3c2ncn(c3=O)CC(=O)O BS-5470 COc1ccc(cc1)C(=O)Cn2c(c(nn2)C(=O)N)C(=O)N BS-5471 CCOC(=O)c1cn2c(n1)C(=O)NC(C2)c3ccc(cc3)F BS-5472 CCOC(=O)c1cn(c(n1)C(=O)N)CC(c2ccccc2)O BS-5473 CCOC(=O)c1c2n(nn1)CC(OC2)c3ccc(cc3)OC BS-5474 Cc1cc(ccc1F)n2cc(nn2)C(=O)N3CCC(CC3)N BS-5475 COc1cccc2c1OC(=C(C2)C(=O)Nc3nccs3)N BS-5476 COc1ccc(cc1)N2CCN(CC2)C(=O)C3CCC(=O)N3 BS-5478 Cc1ccc(cc1C)c2nc(on2)c3cn(c4c3cccc4)C BS-5479 COc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=S)N BS-5480 COc1ccccc1CN2CCc3c(c(=O)[nH]c(=S)[nH]3)C2 BS-5481 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3ccc(cc3)NN BS-5482 CN(C)/C=C(\C(=O)OC)/S(=O)(=O)c1ccc(cc1)Cl BS-5484 c1cc(c(nc1)Cl)S(=O)(=O)N2CCC(CC2)C(=O)N BS-5485 COc1ccc(c(c1)c2ccc(=O)n(n2)CCC(=O)O)OC BS-5486 c1cc(ccc1CN2C(=O)C3(CCOCC3)NC2=O)C(=O)O BS-5487 Cc1cn2c(cc(n2)C(=O)N3CCC(CC3)C(=O)O)c(=O)[nH]1 BS-5488 c1ccc2c(c1)CCCN2S(=O)(=O)c3ccc(nc3)NN BS-5489 CC(C)(C)OC(=O)NCC(=O)Nc1cccc2c1CCCC2 BS-5490 COc1ccc(cc1)C2CCC(=O)N2CCN3CCOCC3 BS-5491 COc1ccc(cc1)c2csc3c2nc([nH]c3=O)SC BS-5492 COc1cccc(c1)c2csc3c2nc([nH]c3=O)SC BS-5493 CN(C)/C=C(\C(=O)OC)/S(=O)(=O)c1cccnc1Cl BS-5494 Cc1cc(=O)[nH]c(n1)N2CCN(CC2)c3cccc(c3)Cl BS-5495 COc1ccc(cc1)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-5496 Cc1cn2c(c(nn2)C(=O)N3CCC(CC3)C(=O)O)c(=O)[nH]1 BS-5497 Cc1ccc(cc1)c2nc(on2)c3nc(no3)c4cccnc4 BS-5498 COc1cccc(c1)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5499 CC(C)(C)OC(=O)NCc1nc(no1)c2ccc(cc2)OC BS-5500 CC(C)OC(=O)c1ncn(n1)CC(c2ccccc2OC)O BS-5501 Cn1cc(c2c1cccc2)c3nc(no3)c4ccc(cc4)OC BS-5503 CCN(CC)CC.CCOC(=O)C1=CNS(=O)(=O)N=C1 BS-5504 CCCCc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5505 CC(C)CCn1c(=O)c2c(c3cccnc3s2)[nH]c1=S BS-5507 Cc1c(nnn1c2cc(ccc2Cl)C(F)(F)F)C(=O)O BS-5508 Cc1c(nnn1c2ccc(c(c2)C(F)(F)F)Cl)C(=O)O BS-5509 c1cc(ccc1CN2Cc3cc(ccc3OCC2=O)Cl)F BS-5510 c1cc(cc(c1)Cl)n2cc(nn2)C(=O)N3CCC(CC3)N BS-5511 c1cc(ccc1n2cc(nn2)C(=O)N3CCC(CC3)N)Cl BS-5512 c1cc2c(cc1Cl)CN(C(=O)CO2)CCC3=CCCCC3 BS-5513 Cc1ccc(cc1)NCC(c2ccc(cc2)Br)O BS-5514 c1ccc(cc1)c2c3[nH]c(=O)c4ccc(cc4n3nn2)C(=O)O BS-5515 c1cscc1/C(=N/OC(=O)c2c3n(nn2)CCNC3=O)/N BS-5516 COc1ccc(cc1)C(Cn2cnc(c2CO)C(=O)OC)O BS-5517 CCOC(=O)c1c(c2cc(c(cc2[nH]1)OC)OC)NC(=O)C BS-5518 CCOc1cccc2c1oc(=O)c(c2)c3[nH]c4ccccc4n3 BS-5519 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3)C#N BS-5520 CN(C)/C=N/c1c(csc1C(=O)OC)c2ccc(cc2)F BS-5521 CN(C)/C=N/c1c(csc1C(=O)OC)c2cccc(c2)F BS-5522 Cc1ccc(cc1)S(=O)(=O)c2cnc3n(c2=O)ccs3 BS-5523 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3ccccc3)C BS-5524 Cc1cccc(c1)NC(=O)c2cn(cn2)Cc3ccc(cc3)N BS-5525 CCCCc1ccc(cc1)NC(=O)CNC(=O)OC(C)(C)C BS-5526 c1cc(cc(c1)Cl)N2CC(CC2=O)C(=O)N3CCCCC3 BS-5527 Cc1cc(ccc1F)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5528 Cc1ccc(cc1F)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5529 COc1ccc(cc1)C(Cn2c(c(nn2)C(=O)OC)CO)O BS-5530 COc1cccc(c1)C(Cn2c(c(nn2)C(=O)OC)CO)O BS-5531 CC(C)(C)OC(=O)N(C)Cc1nc(no1)c2ccc(cc2)F BS-5532 COC(=O)c1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5533 COC(=O)c1cccc(c1)Nc2c(cccn2)S(=O)(=O)N BS-5534 c1cc(c(nc1)Nc2ccc3c(c2)OCCO3)S(=O)(=O)N BS-5535 CCOc1ccc(cc1OCC)CN2CC(CC2=O)C(=O)O BS-5536 CC(=O)Nc1ccc(cc1)NC(=O)CNC(=O)OC(C)(C)C BS-5537 CC1CCN(CC1)C(=O)C2=NNc3ccccc3S2(=O)=O BS-5539 CC(C)(C)OC(=O)NC1(CCCCC1)c2nc(no2)C3CC3 BS-5540 c1cc(sc1)CCN2Cc3cc(ccc3OCC2=O)Cl BS-5541 COc1ccc(cc1)C(=O)C[n+]2ccccc2.[Br-] BS-5542 c1ccc(cc1)c2nc(cc(n2)N3CCNCC3)C(F)(F)F BS-5543 COc1ccc(cc1)C(=O)CS(=O)(=O)c2ccccc2F BS-5544 CC(C)(C)OC(=O)NCC(=O)Nc1ccc2c(c1)OCCO2 BS-5545 COc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccc(cc2)OC BS-5546 c1ccc(cc1)NCc2cc3cc4c(cc3[nH]c2=O)OCCO4 BS-5547 Cc1c(nnn1c2ccccc2)C(=O)Nc3ccc(cc3)OC BS-5548 CCOCCCn1c(=O)c2cc3c(cc2[nH]c1=S)OCO3 BS-5554 Cc1ccc(c(c1)F)S(=O)(=O)/C(=C/2\CCCCCN2)/C#N BS-5555 Cc1cc(cc(c1)NC(=O)C(Cc2ccccc2OC)C#N)C BS-5556 Cc1ccc(c(c1)C)NC(=O)C(Cc2ccccc2OC)C#N BS-5557 Cc1ccc(cc1C)NC(=O)C(Cc2ccccc2OC)C#N BS-5558 CCc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)C#N BS-5559 Cc1cccc(c1C)NC(=O)C(Cc2ccccc2OC)C#N BS-5560 CCc1ccccc1NC(=O)C(Cc2ccccc2OC)C#N BS-5561 Cc1ccc(c(c1)NC(=O)C(Cc2ccccc2OC)C#N)C BS-5562 Cc1cccc(c1C)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5563 CCc1ccccc1NC(=O)C(Cc2cccc(c2)OC)C#N BS-5564 Cc1ccc(cc1C)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5565 CCc1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5566 Cc1cc(cc(c1)NC(=O)C(Cc2cccc(c2)OC)C#N)C BS-5567 Cc1ccc(c(c1)NC(=O)C(Cc2cccc(c2)OC)C#N)C BS-5568 Cc1ccc(c(c1)C)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5569 CCc1ccccc1NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5570 Cc1cccc(c1C)NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5571 Cc1ccc(c(c1)NC(=O)C(Cc2ccc(cc2)OC)C#N)C BS-5572 CCc1ccc(cc1)NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5573 Cc1ccc(cc1C)NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5574 Cc1cc(cc(c1)NC(=O)C(Cc2ccc(cc2)OC)C#N)C BS-5575 CCc1ccc(cc1)NCc2cc3ccc(cc3[nH]c2=O)OC BS-5576 CC(C)(C)OC(=O)NC1CCCN(C1)c2c(=O)n(ccn2)C BS-5577 CC(C)(C)OC(=O)NC1CCN(CC1)c2c(=O)n(ccn2)C BS-5578 COc1ccc(cc1)c2nc(on2)CC3CCNCC3.[Cl-] BS-5579 CSc1[nH]c(=O)c2c(n1)c(cs2)c3cccc(c3)Cl BS-5580 CSc1[nH]c(=O)c2c(n1)c(cs2)c3ccccc3Cl BS-5581 CSc1[nH]c(=O)c2c(n1)c(cs2)c3ccc(cc3)Cl BS-5582 COC(=O)c1c(n(nn1)CC(=O)c2ccsc2)C(=O)OC BS-5583 COc1ccc(c(c1)OC)/C=C(\C#N)/C(=O)Nc2ccccn2 BS-5584 COc1ccc(c(c1)/C=C(\C#N)/C(=O)Nc2ccccn2)OC BS-5585 COc1cc(cc(c1)OC)Nc2c(cccn2)S(=O)(=O)N BS-5586 COc1ccc(cc1OC)Nc2c(cccn2)S(=O)(=O)N BS-5587 CCc1ccc(cc1)NS(=O)(=O)c2c(cn[nH]2)C(=O)OC BS-5588 Cc1ccc(cc1)N(C)S(=O)(=O)c2c(cn[nH]2)C(=O)OC BS-5589 CC(C)(C)OC(=O)N1CCCC(C1)c2cc([nH]n2)C(=O)OC BS-5590 c1csc2c1[nH]c(=S)n(c2=O)CCCN3CCCCC3 BS-5592 c1cc(cc(c1)Cl)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5593 c1cc2c(nc1)N(C(=O)NS2(=O)=O)c3ccc(cc3)Cl BS-5594 CC(C)(C)OC(=O)NCc1nc(no1)c2ccc(cc2)Cl BS-5595 c1cc2c(cc1c3nc(on3)C4CCNCC4)OCO2.Cl BS-5596 CCc1c(nnn1Cc2ccc(cc2)Br)C(=O)O BS-5597 c1cc2c(cc1n3c(c(nn3)C(=O)O)c4ccncc4)OCO2 BS-5598 Cc1ccc2c(c1)c(=O)c3c([nH]2)CCN(C3)C(=O)C(F)(F)F BS-5599 c1cc(c2nncn2c1)S(=O)(=O)Nc3cc(cc(c3)F)F BS-5600 COc1ccccc1C(=O)c2cc3cccc(c3oc2=O)OC BS-5601 CCOc1ccccc1n2c(c(nn2)C(=O)O)c3ccccn3 BS-5602 CCOc1ccc(cc1)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5603 CCOc1ccccc1n2c(c(nn2)C(=O)O)c3ccncc3 BS-5604 CCOc1ccc(cc1)n2c(c(nn2)C(=O)O)c3cccnc3 BS-5605 COc1cccc(c1)c2nc(on2)c3cc4n(n3)CCCC4=O BS-5606 COc1ccc(cc1)c2nc(on2)c3cc4n(n3)CCCC4=O BS-5607 CC1=NS(=O)(=O)N(C=C1C(=O)O)Cc2ccc(cc2)OC BS-5608 CN(C)S(=O)(=O)c1ccc(nc1)n2cc(nc2)C(=O)OC BS-5609 CC(C)(C)OC(=O)NCC(=O)Nc1cc(ccc1OC)OC BS-5610 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1OC)OC BS-5611 Cc1cccc(c1)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-5612 Cc1ccc(cc1)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-5613 COc1cccc(c1)NC(=O)C(Cc2ccccc2OC)C#N BS-5614 COc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)C#N BS-5615 COc1ccccc1CC(C#N)C(=O)Nc2ccccc2OC BS-5616 COc1ccc(c(c1)CC(C#N)C(=O)Nc2ccccc2)OC BS-5617 COc1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5618 COc1cccc(c1)CC(C#N)C(=O)Nc2ccccc2OC BS-5619 COc1ccc(cc1)CC(C#N)C(=O)Nc2ccccc2OC BS-5620 COc1ccc(cc1)CC(C#N)C(=O)Nc2cccc(c2)OC BS-5621 CC(C)(C)OC(=O)N1CCCC(C1)C(=O)N/N=C\2/CCCN2 BS-5622 COC(=O)c1c(n(cn1)CC(c2ccc(cc2)Cl)O)CO BS-5624 Cc1c(c([nH]n1)S(=O)(=O)N2CCNCC2)C(=O)O.Cl BS-5625 Cc1c(cnn1c2ccc(cn2)c3nc(no3)C4CC4)C(=O)O BS-5626 Cc1c(cnn1c2cc(ccn2)c3nc(no3)C4CC4)C(=O)O BS-5627 CCOc1ccc(cc1)NS(=O)(=O)c2c(cn[nH]2)C(=O)O BS-5628 COCCCNC(=O)NNC(=O)COc1ccc(cc1)OC BS-5629 Cc1ccc(c(c1)C)c2cc3c(=O)n(ccn3n2)C/C(=N/O)/N BS-5630 Cc1ccc2cc(c(nc2c1)S(=O)(=O)c3ccccc3)C=O BS-5631 CCCOc1ccc(cc1)CN2Cc3ccccc3OCC2=O BS-5632 CN(c1ccccc1)S(=O)(=O)c2ccsc2C(=O)OC BS-5633 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)C4CC4 BS-5634 CN(c1ccsc1C(=O)NN)S(=O)(=O)c2ccccc2 BS-5636 Cc1ccc2cc(c(=O)[nH]c2c1)CCS(=O)c3ccccc3 BS-5637 c1cc(c(nc1)N2CCOCC2)S(=O)(=O)N3CCCCC3 BS-5638 COC(=O)c1c(n(nn1)CC(c2ccc(cc2)Cl)O)CO BS-5639 COc1ccc(cc1OC)c2nc(on2)C3CCCN3.Cl BS-5640 COC(=O)c1c(c(cs1)c2ccc(cc2)Br)N BS-5641 COc1ccc(c(c1)NC(=O)c2cc(n[nH]2)c3ccc[nH]3)OC BS-5643 CCCc1nc(no1)c2ccc(cc2)n3ccc(n3)C(=O)OC BS-5644 COc1ccc(cc1OC)c2[nH]c(c(n2)c3ccccc3)S BS-5645 c1ccc(c(c1)F)S(=O)(=O)CC(=O)c2ccc(cc2)Cl BS-5646 CCOc1ccc(cc1)NS(=O)(=O)c2cccnc2Cl BS-5647 CCOc1ccc(cc1)CC(=O)N2CCC(CC2)CN.Cl BS-5648 c1cc(c(cc1Cl)Cl)C2=NC3(CCCCC3)NC2=S BS-5649 Cc1c(cnn1c2cc(ccn2)c3nc(no3)C(C)C)C(=O)O BS-5650 COc1ccc(cc1)c2cc3c(=O)n(ccn3n2)C/C(=N/O)/N BS-5651 COc1ccc(cc1OC)CN2Cc3ccccc3OCC2=O BS-5652 COC(=O)c1c(ccs1)N(S(=O)(=O)C)S(=O)(=O)C BS-5653 COc1ccc(cc1Cl)Nc2c(cccn2)S(=O)(=O)N BS-5654 c1cc2c(cc1F)c(=O)c3c([nH]2)CCN(C3)C(=O)C(F)(F)F BS-5655 Cc1ccc(cc1)c2nc(on2)C3=NN(C(=O)CC3)CC(=O)O BS-5656 Cc1ccc(cc1)Cn2c(=O)c(c3n(c2=O)CCC3)/C(=N/O)/N BS-5657 Cc1cc(cc(c1)NC(=O)Cn2c(=O)n3c(n2)CCCCC3)C BS-5660 Cc1cc(n(n1)C(=O)c2c(sc(n2)n3cccc3)C(C)C)C BS-5661 CCCc1c(nc(s1)n2cccc2)C(=O)n3c(cc(n3)C)C BS-5662 Cc1ccc(cc1)C2=NC3(CCC(CC3)C(C)(C)C)NC2=S BS-5663 Cc1ccc(cc1Cl)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5664 Cc1ccc(cc1Cl)n2c(c(nn2)C(=O)O)c3cccnc3 BS-5665 Cc1ccc(cc1Cl)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5666 Cc1cc(ccc1Cl)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5667 CC1=NS(=O)(=O)N(C=C1C(=O)O)Cc2cccc(c2)Cl BS-5668 CC1=NS(=O)(=O)N(C=C1C(=O)O)Cc2ccc(cc2)Cl BS-5669 c1cc(c(cc1Cl)F)S(=O)(=O)/C(=C/2\CCCCN2)/C#N BS-5670 c1cc(c(cc1Cl)S(=O)(=O)/C(=C/2\CCCCN2)/C#N)F BS-5671 CC(C)(C)OC(=O)NCC(=O)Nc1cc(ccc1OC)Cl BS-5672 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(c(c1)Cl)OC BS-5673 COc1cccc(c1)CC(C#N)C(=O)Nc2ccccc2Cl BS-5674 CCOC(=O)c1cn2c(n1)C(=O)NC(C2)c3ccc(cc3)OC BS-5675 CC(C)CNC(=O)Cn1c(=O)c2c(c3ccccc3o2)[nH]c1=O BS-5676 c1ccc(cc1)c2nc(on2)C(=O)NNC(=O)NC3CCCC3 BS-5677 COC(=O)c1c(c(cs1)S(=O)(=O)c2ccccc2F)N BS-5678 COC(=O)c1c(ccs1)S(=O)(=O)Nc2ccc(cc2)F BS-5679 CN(c1ccc(cc1)F)S(=O)(=O)c2ccsc2C(=O)O BS-5680 COc1ccc(c(c1)/C=C(\C#N)/C(=O)Nc2nccs2)OC BS-5681 COc1ccc(c(c1)OC)/C=C(\C#N)/C(=O)Nc2nccs2 BS-5682 COc1ccc(cc1OC)/C=C(\C#N)/C(=O)Nc2nccs2 BS-5683 CC(C)(C)OC(=O)N1CCCC1c2nc(on2)c3ccccc3 BS-5685 CC(C)(C)OC(=O)N1CCCC1c2nc(no2)c3ccccc3 BS-5686 CCc1ccc(cc1)N2CC(CC2=O)C(=O)NC3CCNCC3 BS-5687 c1cc(sc1)CNC(=O)c2ccc(cc2)n3cc[nH]c3=S BS-5688 c1ccc(cc1)CCCN2Cc3cc(ccc3OCC2=O)Cl BS-5689 CCc1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5690 CC1=NS(=O)(=O)N(C=C1C(=O)O)Cc2ccc(cc2F)F BS-5691 c1cc(ccc1n2c(=O)c3ccc(cc3[nH]c2=S)C(=O)O)F BS-5692 Cc1ccc(cc1)C(=O)Cn2cnc(c2C(=O)OC)C(=O)OC BS-5693 Cc1ccc(cc1)S(=O)(=O)c2cc3ccc(cc3oc2=O)O BS-5694 COc1ccc(cc1)S(=O)(=O)c2cnc3ccccn3c2=O BS-5695 CC(C)(C)OC(=O)N1CCCC1c2nc(no2)c3ccncc3 BS-5697 Cc1cc(cc(c1)NS(=O)(=O)c2cccn3c2nnc3C)C BS-5698 CCOc1ccc(cc1)NC(=S)NCc2ccc(cc2)OC BS-5699 CN(C)c1ccc(cc1)N2Cc3cc(ccc3OCC2=O)Cl BS-5700 Cc1ccc(cc1Cl)S(=O)(=O)c2c[nH]c(=S)[nH]c2=O BS-5701 Cc1ccc(cc1)C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-5702 Cc1ccc(cc1)N2c3c(cccn3)S(=O)(=O)C(=N2)C(=O)O BS-5703 Cc1cc(cc(c1)NC(=O)C2=NN(C(=O)CC2)CC(=O)OC)C BS-5704 c1ccc(cc1)c2nc(on2)c3cn(cn3)Cc4ccc(cc4)N BS-5705 COC(=O)/C(=C/Nc1ccccc1)/S(=O)(=O)c2ccccc2 BS-5706 Cc1cc(n(n1)C(=O)c2cn(nn2)CC(c3cccs3)O)C BS-5707 CC(=O)Cc1nc(sn1)NC(=O)c2ccc(cc2)C(C)(C)C BS-5708 CC1CCN(CC1)CCCn2c(=O)c3ccccc3[nH]c2=S BS-5710 COc1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5711 COc1cccc(c1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5712 c1cc(c(=O)[nH]c1)c2nc(no2)c3ccc(cc3)Br BS-5713 c1cc(cc(c1)F)c2nc(on2)C3=NN(C(=O)CC3)CC(=O)O BS-5714 Cc1ccc(cc1)S(=O)(=O)Oc2cc(ncn2)C(F)(F)F BS-5715 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1)C(F)(F)F BS-5716 CCOC(=O)c1cn(c2cc(c(cc2c1=O)F)N3CCCC3)C BS-5718 c1cc(ccc1CNC(=O)Cn2c(=O)n3c(n2)CCCCC3)F BS-5720 Cc1cc(=O)n2c([nH]1)c(c(n2)NC)S(=O)(=O)c3ccccc3 BS-5721 c1cc(ccc1Cn2c(=O)c3c(ccs3)[nH]c2=S)C(=O)O BS-5722 c1cc2c(cc1Cn3c(=O)c4c(ccs4)[nH]c3=S)OCO2 BS-5723 CN(C)/C=N/c1c(csc1C(=O)OC)c2ccc(cc2)OC BS-5725 Cc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)/N=C/N(C)C BS-5726 CC1CCC2(CC1)NC(=S)C(=N2)c3cc(cc(c3)OC)OC BS-5727 CCOC(=O)c1cn(c(n1)C(=O)N)CC(=O)c2ccc(cc2)F BS-5729 CC(C)(C)OC(=O)NCc1nc(no1)c2ccc3c(c2)OCO3 BS-5730 c1ccc(cc1)C(=O)c2ccccc2S(=O)(=O)NCC(=O)O BS-5731 COc1ccc(cc1)CN2c3c(cccn3)S(=O)(=O)NC2=O BS-5732 CC(C)(C)OC(=O)N(C)Cc1nc(no1)c2ccc(cc2)OC BS-5733 CC(C)(C)OC(=O)N1CCCC(C1)c2nc(on2)c3ccco3 BS-5734 c1ccc2c(c1)cc(c(=O)o2)c3csc(n3)SCC(=O)O BS-5735 CC(C)(C)OC(=O)N1CCC(CC1)c2nc(on2)c3cc[nH]n3 BS-5739 CCc1c(nnn1c2ccc(c(c2)C(F)(F)F)Cl)C(=O)O BS-5742 c1cc(cnc1)CC(C#N)C(=O)Nc2ccc(c(c2)Cl)Cl BS-5743 c1cc(cnc1)CC(C#N)C(=O)Nc2cc(ccc2Cl)Cl BS-5744 COC(=O)c1c(n(cn1)CC(=O)c2ccccc2F)C(=O)OC BS-5745 COC(=O)c1c(n(cn1)CC(=O)c2cccc(c2)F)C(=O)OC BS-5746 CCc1c(nc2n1cccc2)c3cc4cccc(c4oc3=O)OC BS-5747 COc1ccc(cc1)Cn2cc(nn2)C(=O)NCC(OC)OC BS-5748 CC(C)(C)OC(=O)NC1CCN(C1)c2c3n[nH]c(=O)n3ccn2 BS-5751 Cc1ccc(cc1)NC(=O)c2c(n(nn2)c3ccc(c(c3)C)C)C BS-5753 CCc1ccc(cc1)NC(=O)c2cn(cn2)Cc3ccc(cc3)N BS-5754 Cc1ccc(c(c1)C)NC(=O)c2cn(cn2)Cc3ccc(cc3)N BS-5755 Cc1cc(cc(c1)NC(=O)c2cn(cn2)Cc3ccc(cc3)N)C BS-5756 CN(C)/C=C(\C#N)/S(=O)(=O)c1ccc(s1)Br BS-5758 COC(=O)c1c(n(nn1)CC(=O)c2cccc(c2)F)C(=O)OC BS-5759 COC(=O)c1c(n(nn1)CC(=O)c2ccccc2F)C(=O)OC BS-5760 CCOC(=O)c1cn(c(n1)C(=O)N)CC(c2ccc(cc2)F)O BS-5761 CCOC(=O)c1c(n(nn1)CC(c2ccc(cc2)OC)O)CO BS-5762 CCOC(=O)c1ccc(cc1)Nc2c(cccn2)S(=O)(=O)N BS-5764 CCOC(=O)c1cccc(c1)Nc2c(cccn2)S(=O)(=O)N BS-5765 Cc1ccc(cc1)C(=O)Nc2c3cc(ccc3[nH]c2C(=O)NC)C BS-5766 CSc1cccc(c1)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5767 CSc1ccc(cc1)N2c3c(cccn3)S(=O)(=O)NC2=O BS-5768 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3C BS-5769 Cc1ccc(cc1)NC(=O)C(Cc2cccc(c2)C)c3n[nH]nn3 BS-5770 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3cccc(c3)C BS-5771 Cc1ccc2c(c1)NN=C(S2(=O)=O)C(=O)N3CCCCCC3 BS-5772 Cc1ccc2c(c1)NN=C(S2(=O)=O)C(=O)N3CCC(CC3)C BS-5773 CN(C)/C=C(\C(=O)OC)/S(=O)(=O)c1ccc(c(c1)Cl)F BS-5774 c1ccc(cc1)CN2c3ccc(cc3C(=O)CS2(=O)=O)Cl BS-5775 c1cc(ccc1CN2Cc3cc(ccc3OCC2=O)Cl)Cl BS-5776 c1ccc(cc1)c2nc(on2)c3nc(no3)Cc4ccc(cc4)F BS-5777 c1ccc(cc1)NC(=O)c2cn(cn2)Cc3ccc(cc3)[N+](=O)[O-] BS-5778 Cc1c(nnn1Cc2cccc(c2)F)C(=O)NCC(OC)OC BS-5779 c1ccc(cc1)c2nnc3n2CCN(C3=O)Cc4ccccc4F BS-5780 CCOC(=O)c1ccc(cc1)NC(=O)CNC(=O)OC(C)(C)C BS-5781 CCOC(=O)c1cccc(c1)NC(=O)CNC(=O)OC(C)(C)C BS-5782 CCc1ccc(cc1)NCc2cc3cc4c(cc3[nH]c2=O)OCO4 BS-5783 CCOc1ccc(cc1)NC(=O)c2c(n(nn2)c3ccccc3)C BS-5784 COc1ccc(cc1)NC(=O)c2cn(cn2)Cc3ccc(cc3)N BS-5785 COc1cccc(c1)NC(=O)c2cn(cn2)Cc3ccc(cc3)N BS-5786 CC(C)(C)OC(=O)N1CCC(CC1)NC(=O)c2cccc(c2)F BS-5788 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3Cl)Cl BS-5789 c1cc(ccc1C2=NC3(CCCCC3)NC2=S)Br BS-5790 CN(C)/C=C(/C(=O)OC)\S(=O)(=O)c1cc(c(cc1F)F)F BS-5791 CC(C)(C)OC(=O)NCc1nc(no1)c2ccc(c(c2)F)OC BS-5792 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3 BS-5795 COc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3 BS-5796 COc1ccccc1CC(c2n[nH]nn2)C(=O)Nc3ccccc3 BS-5797 Cc1ccc(cc1)c2cn3c(c(nn3)C(=O)N4CCCC4)c(=O)[nH]2 BS-5798 Cc1ccc2c(c1)c3c([nH]2)c(=O)n(cn3)Cc4nc(no4)C(C)C BS-5799 c1cc(c(cc1Cl)Cl)C(=O)N2CCC(CC2)CN.Cl BS-5800 CCOc1ccc(cc1Cl)C2Cn3c(c(nn3)C(=O)O)CO2 BS-5801 CC(C)(C)OC(=O)N(C)Cc1nc(no1)c2ccc(cc2)Cl BS-5802 c1cc2c(cc1n3c(c(nn3)C(=O)O)c4ccncc4)OCCO2 BS-5803 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3ccc(cc3)F)C BS-5804 Cc1cc(ccc1NC(=O)c2cn(cn2)Cc3ccc(cc3)N)F BS-5805 CCc1ccc(cc1)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-5806 CCc1ccccc1NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-5807 Cc1ccc(c(c1)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N)C BS-5808 Cc1cccc(c1C)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-5809 Cc1ccc(cc1C)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-5810 Cc1cc(cc(c1)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N)C BS-5811 CCOc1ccccc1NC(=O)C(Cc2ccccc2OC)C#N BS-5812 CCOc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)C#N BS-5813 Cc1ccc(cc1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-5814 Cc1ccccc1NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-5815 Cc1cccc(c1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-5816 Cc1ccccc1NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-5817 Cc1cccc(c1)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-5818 Cc1ccc(cc1)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-5819 CCOc1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)C#N BS-5820 CCOc1ccc(cc1)NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5821 CCOc1ccccc1NC(=O)C(Cc2ccc(cc2)OC)C#N BS-5822 Cc1ccc2cc(c(=O)[nH]c2c1)CNc3ccc(c(c3)OC)OC BS-5823 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2ccc(cc2)Cl BS-5828 CCOc1ccc(cc1)NS(=O)(=O)c2c(cn[nH]2)C(=O)OC BS-5829 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3F BS-5830 CCc1ccc(cc1)S(=O)(=O)c2csc(c2N)C(=O)OC BS-5834 Cc1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)OC BS-5835 Cc1ccc(cc1C)S(=O)(=O)Nc2ccsc2C(=O)OC BS-5836 CC(C)c1ccc(cc1)S(=O)(=O)N(C)c2ccsc2CO BS-5837 c1cc(ccc1c2nc(cc(n2)N3CCNCC3)C(F)(F)F)F BS-5838 Cc1cn2c(cc(n2)C(=O)Nc3ccc(cc3)C(=O)OC)c(=O)[nH]1 BS-5839 COc1cccc(c1)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-5840 Cc1ccc(cc1)n2c(=O)c3ccc(cc3[nH]c2=S)C(=O)OC BS-5841 c1ccc(cc1)CCn2c(=O)c3c4c(sc3[nH]c2=O)CCCC4 BS-5842 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCNCC4 BS-5843 c1cc(cc(c1)Cl)NC(=O)c2cn(cn2)Cc3ccc(cc3)N BS-5845 c1cc(c(cc1Cl)Cl)C2=NC3(CCCCCC3)NC2=S BS-5846 CC1CCC2(CC1)NC(=S)C(=N2)c3ccc(cc3Cl)Cl BS-5847 c1ccc2c(c1)c3c(o2)c(=O)n(c(=O)[nH]3)CC(=O)NC4CCCC4 BS-5848 Cc1c(cnn1c2ccc(cn2)c3nc(no3)C(C)(C)C)C(=O)O BS-5850 Cc1c(cnn1c2cc(ccn2)c3nc(no3)C(C)(C)C)C(=O)O BS-5851 CCOC(=O)C(=CNc1ccsc1C(=O)OC)C(=O)OCC BS-5852 CCOc1ccc(cc1)NS(=O)(=O)c2ccsc2C(=O)O BS-5853 Cc1ccc(cc1)C2Cn3c(c(nn3)C(=O)N4CCNCC4)CO2 BS-5854 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NC4CCCC4 BS-5855 c1ccc(c(c1)Cn2cnc3c4cc(ccc4[nH]c3c2=O)F)Cl BS-5856 Cc1ccc(cc1NC(=O)c2c(n(nn2)c3ccccc3)N)Cl BS-5857 c1cc(c(nc1)Nc2ccc(cc2)Br)S(=O)(=O)N BS-5858 c1cc(cc(c1)Br)Nc2c(cccn2)S(=O)(=O)N BS-5859 c1cc(ccc1Cn2cc(nc2)C(=O)Nc3ccc(cc3F)F)N BS-5860 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)C3CC3)C(F)(F)F BS-5861 COc1ccc(c(c1)CC(C#N)C(=O)Nc2ccc(cc2)F)OC BS-5862 COc1ccc(c(c1)OC)CC(C#N)C(=O)Nc2ccc(cc2)F BS-5863 COc1ccc(c(c1)OC)CC(C#N)C(=O)Nc2ccccc2F BS-5864 Cc1cc(cc2c1oc(=O)c(c2)S(=O)(=O)c3ccccc3)C=O BS-5865 COC(=O)C1CCCCN1S(=O)(=O)c2ccccc2[N+](=O)[O-] BS-5866 CCc1cccc(c1)C(=O)NNC(=O)COc2ccc(cc2)OC BS-5867 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1)S(=O)(=O)C BS-5869 CCc1ccc(cc1)n2c(c(nn2)c3nc(c(s3)C(=O)O)C)C BS-5871 Cc1ccc(cc1C)NC(=O)NC2(CCCCC2)c3nc(no3)C BS-5873 CC(C)(C)OC(=O)NCC(=O)Nc1cccc(c1)Br BS-5874 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1)Br BS-5875 CCOC(=O)C1CCN(CC1)C(=O)c2cnc3ccccn3c2=O BS-5876 CN(c1ccc(cc1)F)S(=O)(=O)c2ccsc2C(=O)OC BS-5877 c1cc(ccc1c2nc(on2)CC3CCN(CC3)C(=O)C4CC4)F BS-5878 Cc1ccc(cc1)N2C=C(S(=O)(=O)c3c2cccc3)C(=O)OC BS-5879 Cc1nc(on1)C2(CCCCC2)NC(=O)C(C)Oc3ccccc3 BS-5880 Cc1ccc(cc1)c2nc(on2)C3CCCN3C(=O)OC(C)(C)C BS-5881 Cc1cc(n(n1)C(=O)CN2CCCCC2c3nc(no3)C4CC4)C BS-5882 CC(C)c1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5884 COc1ccc(cc1)CCc2ncc(s2)c3ccc(cc3)Cl BS-5885 c1cc(ccc1NC(=O)C(Cc2ccncc2)C#N)Br BS-5886 c1ccc(c(c1)NC(=O)C(Cc2cccnc2)C#N)Br BS-5887 c1cc(cnc1)CC(C#N)C(=O)Nc2ccc(cc2)Br BS-5888 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3ccc4n[nH]c(=O)n4c3 BS-5889 COc1ccc(cc1)CC(C#N)C(=O)Nc2cccc3c2cccc3 BS-5890 CCn1c2c(c(n1)C)[nH]c(=S)n(c2=O)Cc3ccc(cc3)OC BS-5892 COc1ccc(cc1Cl)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5893 COc1ccc(cc1Cl)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5894 COc1ccc(cc1n2c(c(nn2)C(=O)O)c3ccccn3)Cl BS-5895 CN(C)c1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5896 Cc1ccc(c(c1)C)C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-5897 Cc1ccc(cc1)N2c3c(cccn3)S(=O)(=O)C(=N2)C(=O)OC BS-5898 Cc1ccc(cc1C)S(=O)(=O)c2c[nH]c3c(c2=O)cccc3F BS-5899 Cc1ccc(cc1)N/N=C(\C#N)/S(=O)(=O)c2cc(ccc2F)C BS-5900 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2)/C(=O)OC BS-5902 Cc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccccc2 BS-5903 COc1ccccc1C(=O)Nc2c(c3c(s2)CCCC3)C(=O)O BS-5904 CCCn1cc(c(n1)S(=O)(=O)N2CCOCC2)C(=O)OCC BS-5905 c1ccc2c(c1)c(=O)[nH]c3n2c(=S)sc3C(=O)N4CCCC4 BS-5906 c1cc(sc1)CC(=O)NC2(CCCCC2)c3nc(no3)C4CC4 BS-5909 c1cc2c(cc1CN3Cc4cc(ccc4OCC3=O)Cl)OCO2 BS-5912 CCOc1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5913 CCOc1cccc(c1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5914 c1ccn(c1)c2c(cnn2c3ccc(cc3)Br)C(=O)O BS-5916 COc1ccc(cc1)C(=O)c2cnc3ccc(cc3c2Cl)Cl BS-5917 COc1ccc(cc1)C(=O)Cn2cnc(c2C(=O)OC)C(=O)OC BS-5918 COCCc1nc(on1)c2nc(no2)c3ccc(c(c3)OC)OC BS-5919 CC(C)(C)OC(=O)N1CCN(CC1)c2cc(ncn2)C(F)(F)F BS-5920 CCOC(=O)Cn1cnc2c(csc2c1=O)c3ccc(cc3)F BS-5922 CCOC(=O)C1CCN(CC1)C(=O)c2cc3c(=O)[nH]c(cn3n2)C BS-5923 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccn2)/C(=O)OC BS-5925 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=O)N(N2)c3ccccc3 BS-5926 c1cc(c(cc1F)Cl)Cn2c(c(nn2)C(=O)O)c3ccncc3 BS-5932 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)CC(=O)N2CCCC2 BS-5933 COc1cccc(c1)C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-5934 COc1ccccc1C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-5935 CCOC(=O)c1cn(c(n1)C(=O)N)CC(c2ccc(cc2)OC)O BS-5936 CC(C)(C)OC(=O)N(C)Cc1nc(no1)c2ccc3c(c2)OCO3 BS-5937 CCOC(=O)C1CCN(CC1)C(=O)c2c3c(=O)[nH]c(cn3nn2)C BS-5938 Cc1cc(n(n1)C(=O)c2cc3c(=O)[nH]c(cn3n2)c4ccccc4)C BS-5939 CC(C)(C)OC(=O)N1CCCC1c2nc(no2)c3ccc(cc3)F BS-5940 Cc1ccc(cc1)c2cc3c(=O)n(ccn3n2)Cc4ccccc4F BS-5941 Cc1ccc(cc1)N/C=C(/C(=O)C)\S(=O)(=O)c2ccccc2F BS-5942 c1ccc(cc1)CNC(=O)c2c(c3cccnc3s2)n4cccc4 BS-5946 Cc1cccc(c1)N2CCN(CC2)C(=O)CNC(=O)OC(C)(C)C BS-5947 Cc1ccccc1N2CCN(CC2)C(=O)CNC(=O)OC(C)(C)C BS-5948 Cc1ccc(cc1)N2CCN(CC2)C(=O)CNC(=O)OC(C)(C)C BS-5949 c1cc(ccc1c2cc3c(nccn3n2)N4CCNCC4)F.Cl BS-5950 CSc1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-5951 c1ccc(c(c1)C(F)(F)F)n2c(c(nn2)C(=O)O)c3cccnc3 BS-5952 c1cc(ccc1C(F)(F)F)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5953 c1ccc(c(c1)C(F)(F)F)n2c(c(nn2)C(=O)O)c3ccccn3 BS-5954 c1ccnc(c1)c2c(nnn2c3cccc(c3)C(F)(F)F)C(=O)O BS-5955 c1ccc(c(c1)C(F)(F)F)n2c(c(nn2)C(=O)O)c3ccncc3 BS-5956 CC(C)(C)OC(=O)NCC(=O)Nc1cccc(c1)OC(F)(F)F BS-5957 COc1ccc2c(c1)cc(c(=O)o2)S(=O)(=O)c3ccc(cc3)F BS-5958 Cc1ccc(cc1)N2c3ccc(cc3S(=O)(=O)C(=N2)C(=O)O)F BS-5959 Cc1ccc(cc1)S(=O)(=O)Cc2c(c3n(n2)CCCC3)C(=O)O BS-5961 Cc1ccc(cc1)S(=O)(=O)Cc2c(c3n(n2)CCC3)C(=O)OC BS-5962 CCOc1ccc(cc1)C(=O)N2CCN(CC2)C(=O)OC(C)(C)C BS-5963 COc1ccc(cc1OC)c2csc3c2nc([nH]c3=O)SC BS-5964 CCc1ccc(cc1)NC(=O)c2c(n(nn2)c3ccc(c(c3)C)C)C BS-5965 Cc1ccc(cc1C)NC(=O)c2c(n(nn2)c3ccc(c(c3)C)C)C BS-5966 Cc1ccc(c(c1)C)NC(=O)c2c(n(nn2)c3ccc(c(c3)C)C)C BS-5967 Cc1nc(on1)C2(CCCCC2)NC(=O)Nc3ccccc3Cl BS-5969 Cc1cccc(c1)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F BS-5970 Cc1ccc(cc1)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F BS-5971 COC(=O)/C(=C\Nc1ccccc1)/S(=O)(=O)c2ccc(cc2)F BS-5972 COC(=O)/C(=C/Nc1ccc(cc1)F)/S(=O)(=O)c2ccccc2 BS-5973 CCOc1ccc(cc1)NS(=O)(=O)c2ccccc2C(=O)OC BS-5978 Cc1ccc(cc1)Nc2c(cncn2)c3nc(no3)c4ccsc4 BS-5979 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3cc(ccc3C)C BS-5980 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccc(cc3C)C BS-5981 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3cc(cc(c3)C)C BS-5982 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccc(c(c3)C)C BS-5983 CCc1ccccc1NC(=O)C(Cc2cccc(c2)C)c3n[nH]nn3 BS-5984 COCc1c(nnn1c2ccc(c(c2)C(F)(F)F)Cl)C(=O)O BS-5985 CNC(=O)c1c(n(nn1)CC(=O)c2ccc(cc2)Cl)C(=O)NC BS-5986 c1cc(ccc1CCN2Cc3cc(ccc3OCC2=O)Cl)Cl BS-5987 c1cc2c(cc1c3nc(on3)c4nc(no4)c5cnccn5)OCO2 BS-5988 Cc1ccccc1Cc2nc(on2)c3nc(no3)c4ccccc4F BS-5991 COc1cccc(c1OC)/C=C/C(=O)c2cc3ccccc3oc2=O BS-5992 c1cc(ncc1S(=O)(=O)N2CCCC2)n3cc(nc3)C(=O)NN BS-5997 CCc1ccc(cc1)NCc2cc3cc4c(cc3[nH]c2=O)OCCO4 BS-6002 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3ccc(cc3)OC)C BS-6003 CC1=NS(=O)(=O)N(C=C1C(=O)OC(C)(C)C)Cc2ccccc2 BS-6007 Cc1ccc(cc1)c2csc3c2nc([nH]c3=O)n4c(cc(n4)C)C BS-6008 c1ccc(cc1)CN2CCC(CC2)N3Cc4ccccc4OCC3=O BS-6009 COC(=O)c1c(n(cn1)CC(=O)c2ccc(cc2)Cl)C(=O)OC BS-6010 c1cc(ccc1S(=O)(=O)c2cc3ccc(cc3oc2=O)O)Cl BS-6011 CCc1nnc2n1cccc2S(=O)(=O)Nc3ccc(cc3)Cl BS-6012 CC(C)(C)OC(=O)N(C)Cc1nc(no1)c2ccc(c(c2)F)OC BS-6013 c1ccnc(c1)Cn2cnc3c(csc3c2=O)c4cccc(c4)F BS-6018 COC(=O)c1ccc(cc1)Cn2ccn3c(c2=O)c4c(n3)CCCC4 BS-6020 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3OC BS-6021 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccc(cc3)OC BS-6022 Cc1ccccc1NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6023 Cc1ccc(cc1)NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6024 Cc1ccccc1NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6025 Cc1cccc(c1)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6026 Cc1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6027 Cc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6028 Cc1ccccc1NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6029 Cc1cccc(c1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6030 CC(C)(C)OC(=O)NCC(=O)N1CCN(CC1)c2ccccc2F BS-6031 CC(C)(C)OC(=O)NCC(=O)N1CCN(CC1)c2ccc(cc2)F BS-6032 c1cc2c(nc1)N(N=C(S2(=O)=O)C(=O)O)c3ccc(cc3)Cl BS-6034 c1cc(ccc1F)S(=O)(=O)c2c[nH]c3ccc(cc3c2=O)Cl BS-6035 c1cc(cc(c1)Cl)S(=O)(=O)c2c[nH]c3c(c2=O)cccc3F BS-6036 COc1ccc(cc1OC)C(=O)CS(=O)(=O)c2ccccc2F BS-6037 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4)CCCC3 BS-6038 COc1ccccc1Cn2c(=O)c3c(c4ccccc4o3)[nH]c2=S BS-6040 CCOc1ccc(c(c1)NC(=O)CNC(=O)OC(C)(C)C)OCC BS-6041 Cc1cc(cc(c1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N)C BS-6042 Cc1ccc(c(c1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N)C BS-6043 Cc1ccc(c(c1)C)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6044 CCc1ccccc1NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6045 Cc1cccc(c1C)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6046 CCc1ccc(cc1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6047 Cc1ccc(cc1C)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6048 Cc1ccc(c(c1)NC(=O)C(Cc2ccc(cc2OC)OC)C#N)C BS-6049 Cc1ccc(c(c1)C)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6050 CCc1ccccc1NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6051 Cc1cccc(c1C)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6052 CCc1ccc(cc1)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6053 Cc1ccc(cc1C)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6054 Cc1cc(cc(c1)NC(=O)C(Cc2ccc(cc2OC)OC)C#N)C BS-6055 CCc1ccc(cc1)NCc2cc3cc(c(cc3[nH]c2=O)OC)OC BS-6056 CC(C)c1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)N BS-6063 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3ccc(nc3Cl)NN BS-6069 c1cc(oc1)C(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4 BS-6070 c1c[nH]nc1C(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4 BS-6071 Cc1ccc(c(c1)C)NC(=O)CS(=O)(=O)c2cc(ccc2F)F BS-6072 COC(=O)c1c(ccs1)NC(=O)CS(=O)(=O)c2ccccc2 BS-6073 CCOC(=O)CC(=O)Nc1c(c2c(s1)CCCC2)C(=O)OCC BS-6075 Cc1ccc(cc1C)N(C)S(=O)(=O)c2ccsc2C(=O)OC BS-6077 CC(C)c1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)O BS-6078 Cc1cc(c(c(c1)C)S(=O)(=O)N(C)c2ccsc2C(=O)O)C BS-6079 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)C4CCCC4 BS-6080 c1ccc(cc1)CCC(=O)NC2(CCCCC2)c3nc(no3)C4CC4 BS-6082 CCOC(=O)N1CCC(CC1)n2c(=O)c3c(ccs3)[nH]c2=S BS-6083 c1ccc(c(c1)CN2c3cc(ccc3C(=O)CS2(=O)=O)Cl)F BS-6084 COc1ccc(cc1)N2CCN(CC2)C(=O)C3CCCCN3.Cl BS-6086 c1cc2c(cc1Cn3c(=O)c4ccc(cc4[nH]c3=O)C(=O)O)OCO2 BS-6087 c1cc(ccc1Cn2cc(nc2)C(=O)Nc3ccc(cc3)F)[N+](=O)[O-] BS-6090 c1cc(cc(c1)F)NC(=O)c2cn(cn2)Cc3ccc(cc3)[N+](=O)[O-] BS-6091 COc1ccc(cc1OC)c2nc(on2)c3cc4n(n3)CCCC4=O BS-6092 CCOc1ccc(cc1)C(=O)CS(=O)(=O)c2ccc(cc2F)F BS-6093 Cc1ccc(cc1)S(=O)(=O)c2c3[nH]c(=O)c4ccccc4n3nn2 BS-6094 CC(C)(C)OC(=O)NCC(=O)Nc1cc(c(c(c1)OC)OC)OC BS-6095 CC(=O)/C(=C\Nc1ccc(cc1)OC)/C(=O)Nc2ccc(cc2)OC BS-6096 CCOc1ccc(cc1)NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-6097 CCOc1ccccc1NC(=O)C(Cc2ccc(c(c2)OC)O)C#N BS-6098 COc1ccccc1CC(C#N)C(=O)Nc2ccc(c(c2)OC)OC BS-6099 COc1ccc(cc1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6100 COc1cccc(c1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6101 COc1ccc(c(c1)CC(C#N)C(=O)Nc2ccccc2OC)OC BS-6102 COc1ccc(cc1)NC(=O)C(Cc2ccc(c(c2)OC)OC)C#N BS-6103 COc1cccc(c1)NC(=O)C(Cc2ccc(c(c2)OC)OC)C#N BS-6104 COc1ccccc1NC(=O)C(Cc2ccc(c(c2)OC)OC)C#N BS-6105 COc1ccc(c(c1)OC)CC(C#N)C(=O)Nc2ccccc2OC BS-6106 COc1cccc(c1)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6107 COC(=O)c1c(ccs1)NC(=O)Nc2ccsc2C(=O)OC BS-6108 CCOC(=O)c1ccc(cc1)NC2=NC3CS(=O)(=O)CC3S2 BS-6109 Cc1ccccc1NC(=O)NC2(CCCCC2)c3nc(no3)C4CC4 BS-6110 c1cc(ccc1/C=C(\C#N)/c2ncc(s2)c3ccc(cc3)Cl)F BS-6112 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3ccc(cc3)Cl)C BS-6113 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3cccc(c3)Cl)C BS-6114 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3ccccc3Cl)C BS-6115 Cc1ccc(cc1NC(=O)c2cn(cn2)Cc3ccc(cc3)N)Cl BS-6116 c1ccc2c(c1)[nH]c(n2)c3cc4cc(ccc4oc3=O)Br BS-6117 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3F BS-6118 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3ccc(cc3)F BS-6119 COc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccc(cc3)F BS-6120 COc1ccccc1CC(c2n[nH]nn2)C(=O)Nc3ccc(cc3)F BS-6121 COc1ccccc1CC(c2n[nH]nn2)C(=O)Nc3ccccc3F BS-6122 Cc1ccc2c(c1)S(=O)(=O)C(=NN2c3ccc(cc3)C(=O)O)C#N BS-6123 Cc1ccc(cc1)Cn2c3cc(nn3c(=O)c(n2)C#N)c4ccccc4 BS-6124 c1ccc(cc1)Oc2ccc(cc2)Nc3c(cccn3)S(=O)(=O)N BS-6125 CN(c1ccc(cc1)OC)S(=O)(=O)c2ccsc2C(=O)OC BS-6127 CN(c1ccc(cc1)OC)S(=O)(=O)c2ccsc2C(=O)NN BS-6128 CN(c1ccsc1C(=O)NN)S(=O)(=O)c2ccc(cc2)NN BS-6129 CCc1ccc2c(c1)cc(c(=O)[nH]2)S(=O)(=O)c3ccc(c(c3)C)C BS-6130 COc1ccc(cc1OC)CC(c2[nH]c3ccccc3n2)C(=S)N BS-6131 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NC4CCCC4 BS-6133 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NC4CCCCC4 BS-6134 Cc1cc(ccc1Br)Nc2c(cccn2)S(=O)(=O)N BS-6135 CN(c1ccccc1)C(=O)CN2CCCn3c(cc(n3)C(=O)O)C2=O BS-6138 C/C(=N\Nc1c(cccn1)S(=O)(=O)N2CCOCC2)/C(=O)OC BS-6140 c1cc(cc(c1)Cl)c2nc(cc(n2)N3CCNCC3)C(F)(F)F BS-6142 COc1ccc(cc1)C(=O)/C=C/2\NCCN2Cc3ccccc3Cl BS-6143 Cc1cc(ccc1NC(=O)CNC(=O)OC(C)(C)C)Br BS-6144 Cc1cc(ccc1Br)NC(=O)CNC(=O)OC(C)(C)C BS-6145 CC(C)(C)OC(=O)NCC(=O)NCc1ccc(cc1)Br BS-6146 CSc1[nH]c(=O)c2c(n1)c(cs2)c3ccc(c(c3)Cl)Cl BS-6147 Cc1nc(on1)C2(CCCCC2)NC(=O)C3COc4ccccc4O3 BS-6149 CCc1ccc(cc1)Nc2c(cncn2)c3nc(no3)c4ccccc4 BS-6151 c1cc(cc(c1)F)CC(=O)NC2(CCCCC2)c3nc(no3)C4CC4 BS-6156 Cc1ccc(cc1)c2nc(no2)C3CCN(CC3)C(=O)OC(C)(C)C BS-6158 CCOc1ccc(cc1)CC(=O)NC2(CCCCC2)c3nc(no3)C BS-6159 Cc1nc(on1)C2(CCCCC2)NC(=O)CCc3ccccc3OC BS-6160 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccccc3 BS-6161 Cc1cccc(c1)C2=NC3(CCN(CC3)C(=O)OC(C)(C)C)NC2=O BS-6162 COC(=O)c1ccc2c(c1)cc(c(=O)o2)S(=O)(=O)c3ccccc3 BS-6163 COc1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)CC(=O)N2CCOCC2 BS-6164 CCOC(=O)c1cc(n(n1)CCC(=O)c2ccccc2)C(=O)OCC BS-6165 CCOc1cccc2c1oc(=O)c(c2)S(=O)(=O)c3ccc(cc3)C BS-6168 c1ccc(c(c1)NC(=O)NC2(CCCCC2)c3nc(no3)C4CC4)F BS-6169 Cc1ccc(cc1)CN2CC(CC2=O)C(=O)N3CCC(CC3)C(=O)O BS-6171 CCc1ccc(cc1)N2CC(CC2=O)C(=O)N3CCC(CC3)C(=O)O BS-6172 CCOc1ccc(cc1)NC(=O)NC2(CCCCC2)c3nc(no3)C BS-6175 CC(C)(C)OC(=O)NC1(CCCCC1)c2nc(no2)c3ccncc3 BS-6176 CC(C)(C)OC(=O)NC1(CCCCC1)c2nc(no2)c3cccnc3 BS-6177 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccncc3 BS-6178 Cc1cc(c(cc1Cl)OC)n2c(c(nn2)C(=O)O)c3ccncc3 BS-6180 Cc1c(cccc1Cl)NC(=O)c2c(n(nn2)c3ccc(cc3)F)C BS-6181 CC(C)(C)OC(=O)NCC(=O)Nc1cc(c(cc1OC)OC)Cl BS-6182 CC(C)(C)OC(=O)NCC(=O)Nc1cc(c(cc1OC)Cl)OC BS-6183 c1cc(c(cc1Br)F)S(=O)(=O)/C(=C/2\CCCN2)/C#N BS-6184 Cc1cc(c(cc1C)C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC)C BS-6185 CC(C)(C)OC(=O)NC1(CCCCC1)c2nc(no2)c3cnccn3 BS-6188 Cc1ccc(cc1C)S(=O)(=O)/C(=C\Nc2ccccc2)/C(=O)OC BS-6190 CCc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2)/C(=O)OC BS-6191 Cc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C BS-6192 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccccc2 BS-6193 COc1cc2c(cc1OC)ncc(c2Cl)C(=O)c3ccc(cc3)F BS-6195 Cc1cc(n(n1)C(=O)c2ncn(n2)CC(c3ccc(cc3)Cl)O)C BS-6196 CCCOc1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Cl BS-6197 CCN(c1ccsc1C(=O)O)S(=O)(=O)c2ccc(cc2)Cl BS-6198 CC(C)(C)OC(=O)NC1CCN(CC1)c2cc(ncn2)C(F)(F)F BS-6199 Cc1nc(cc(n1)N2CCN(CC2)C(=O)OC(C)(C)C)C(F)(F)F BS-6200 COc1ccc(c(c1)S(=O)(=O)c2cc3ccccc3oc2=O)OC BS-6201 COc1ccc(cc1OC)S(=O)(=O)c2cc3ccccc3oc2=O BS-6202 COc1cc(ccc1O)CC(C#N)C(=O)Nc2cccc3c2cccc3 BS-6203 Cc1ccc(cc1)N/N=C(\C(=O)C)/S(=O)(=O)c2ccc(cc2)OC BS-6204 c1cc(cc(c1)S(=O)(=O)c2cnc3ccc(cc3c2Cl)F)C#N BS-6220 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCNCC4)Cl BS-6221 CCOc1ccc(cc1)C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-6222 Cc1ccc(c(c1)Nc2c(cncn2)c3nc(no3)c4ccccc4)F BS-6225 Cc1ccc(c(c1)F)Nc2c(cncn2)c3nc(no3)c4ccccc4 BS-6227 c1cc(c(cc1C(=O)NC2(CCCCC2)c3nc(no3)C4CC4)F)F BS-6230 CCOC(=O)CNS(=O)(=O)c1ccccc1C(=O)c2ccccc2 BS-6231 COc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2)/C(=O)OC BS-6232 COc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccccc2 BS-6233 CC(C)(C)OC(=O)N1CCC2(CC1)CC(=O)c3ccc(cc3O2)OC BS-6234 CCOC(=O)c1ccc(cc1)n2c3c(c(=O)[nH]c(n3)C)sc2=S BS-6238 CCc1ccc(cc1)NC(=O)c2c(c3cccnc3s2)n4cccc4 BS-6239 COc1ccc(c(c1)CN2Cc3cc(ccc3OCC2=O)Cl)OC BS-6240 CCc1ccc(cc1)S(=O)(=O)/C(=N/Nc2ccc(cc2)Cl)/C#N BS-6241 Cc1ccc(cc1)NS(=O)(=O)c2c(cn[nH]2)c3cccc(c3)Cl BS-6242 CC(C)c1nc(on1)CC2CCN(CC2)C(=O)c3ccc(cc3)Cl BS-6243 COc1ccc(cc1)N2Cc3cc(ccc3OCC2=O)Br BS-6244 c1cc(cc(c1)C(F)(F)F)Cn2c(c(nn2)C(=O)O)c3ccncc3 BS-6245 COc1ccc(cc1)CC(C#N)C(=O)Nc2cccc(c2)C(F)(F)F BS-6246 CCOC(=O)c1cn(c(n1)C(=O)OCC)CC(=O)c2ccc(cc2)F BS-6247 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc(cc2)F)C(=O)OCC BS-6248 CCOc1cccc2c1oc(=O)c(c2)S(=O)(=O)c3ccc(cc3)F BS-6249 CN(C)/C=N/c1c(csc1C(=O)OC)c2ccc(c(c2)OC)OC BS-6257 COc1ccc(cc1OC)CCn2c(=O)c3c(ccs3)[nH]c2=S BS-6259 Cc1c(cccc1Cl)NC(=O)NC2(CCCCC2)c3nc(no3)C BS-6261 Cc1ccc(cc1C)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F BS-6262 CCc1ccc(cc1)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F BS-6263 Cc1ccc(c(c1)S(=O)(=O)c2c[nH]c3cc(c(cc3c2=O)F)F)C BS-6264 Cc1ccc(cc1)N/C=C(\C(=O)OC)/S(=O)(=O)c2ccccc2F BS-6266 Cc1ccc2c(c1)c(=O)c3c([nH]2)CCN(C3)Cc4ccc(cc4)[N+](=O)[O-] BS-6267 CC(C)(C)OC(=O)NCC(=O)N1CCN(CC1)c2ccc(cc2)OC BS-6272 Cc1ccc(cc1)NC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C BS-6273 Cc1cccc(c1)NC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C BS-6274 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NCc4ccccc4 BS-6275 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccccc4 BS-6276 CC(C)(C)OC(=O)NC1(CCCCC1)c2nc(no2)c3ccsc3 BS-6277 Cc1nc(on1)C2(CCCCC2)NC(=O)COc3ccc(cc3)Cl BS-6279 Cc1nc(on1)C2(CCCCC2)NC(=O)c3ccc(cc3OC)Cl BS-6280 c1cc(ccc1CN2Cc3cc(ccc3OCC2=O)Br)F BS-6281 c1cc2c(cc1Br)CN(C(=O)CO2)CCC3=CCCCC3 BS-6282 c1cc(ccc1n2c(c(nn2)C(=O)O)c3ccncc3)OC(F)(F)F BS-6283 c1ccc(cc1)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6284 CCOc1ccc(cc1OCC)c2c3[nH]c(=O)c4ccccc4n3nn2 BS-6286 COC(=O)c1cn(cn1)c2ccc(cn2)S(=O)(=O)N3CCCCC3 BS-6291 Cc1ccc(c(c1)C)c2cc3c(nccn3n2)N4CCC(CC4)C(=O)O BS-6299 COC(=O)C1=NN(c2ccccc2S1(=O)=O)c3ccc(cc3)Cl BS-6302 CC(=O)Nc1ccccc1/N=c\2/c(cc3cc(ccc3o2)OC)C(=O)N BS-6303 c1cnc(cn1)c2nc(on2)C3(CCCCC3)NC(=O)c4cnccn4 BS-6304 CN(C)/C=C(/C(=O)c1ccccc1)\S(=O)(=O)c2cc(ccc2F)F BS-6305 COC(=O)c1ccc2c(c1)nc3n(c2=O)N=C(CS3)c4ccccc4 BS-6306 Cc1ccccc1/N=c\2/c(cc3ccccc3o2)c4[nH]c5ccccc5n4 BS-6307 Cc1ccc(c(c1)C)NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6309 CCc1ccccc1NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6310 Cc1ccc(c(c1)NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3)C BS-6311 CCc1ccc(cc1)NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6312 Cc1cc(cc(c1)NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3)C BS-6313 Cc1ccc(cc1C)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6314 CCc1ccccc1NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6315 Cc1cc(cc(c1)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3)C BS-6316 Cc1ccc(c(c1)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3)C BS-6317 Cc1cccc(c1C)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6318 CCc1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6319 Cc1ccc(c(c1)C)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6320 CCc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6321 Cc1ccc(c(c1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3)C BS-6322 Cc1cccc(c1C)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6323 CCc1ccccc1NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6324 Cc1ccc(cc1C)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6325 Cc1cc(cc(c1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3)C BS-6326 COC(=O)/C(=C/Nc1ccccc1)/S(=O)(=O)c2ccc(cc2)Cl BS-6329 COC(=O)/C(=C/Nc1ccc(cc1)Cl)/S(=O)(=O)c2ccccc2 BS-6330 c1cc(sc1)CCN2Cc3cc(ccc3OCC2=O)Br BS-6331 c1cc(sc1S(=O)(=O)c2c[nH]c(=S)nc2N)Br BS-6332 COc1ccc(cc1)c2nc(on2)c3nc(no3)Cc4cccc(c4)F BS-6333 CCCCOc1ccc(cc1)C(=O)c2cc3cccc(c3oc2=O)OC BS-6334 Cc1ccc(cc1)CN2CC(CC2=O)C(=O)Nc3ccc(cc3)C(=O)O BS-6335 Cc1ccc(cc1)CN2CC(CC2=O)C(=O)Nc3cccc(c3)C(=O)O BS-6336 COc1ccc(cc1OC)NC(=O)c2cn(cn2)Cc3ccc(cc3)N BS-6337 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4)CCCCC3 BS-6339 Cc1ccc(cc1)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-6340 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4)CCCC3 BS-6341 COc1cccc(c1)c2cc3c(nccn3n2)N4CCC(CC4)C(=O)O BS-6342 COc1ccc(cc1)c2cc3c(nccn3n2)N4CCC(CC4)C(=O)O BS-6343 c1ccc2c(c1)cc(c(=O)o2)C(=O)NC3=C(C4CCCCC4S3)C#N BS-6344 COc1ccc(cc1)C(=O)CCC(=O)N2CCN(CC2)c3ccccc3 BS-6345 CCOC(=O)C1CCN(CC1)C(=S)Nc2cc(cc(c2)OC)OC BS-6348 COC(=O)c1c(n(nn1)CC(=O)Nc2ccc(cc2)Cl)C(=O)OC BS-6349 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(c(c1)C(F)(F)F)Cl BS-6350 CCOC(=O)N1CCC(CC1)N2Cc3cc(ccc3OCC2=O)Cl BS-6351 c1ccc(cc1)c2csc3c2ncn(c3=O)Cc4cccc(c4)Cl BS-6358 CC(C)(C)OC(=O)NC1CCN(CC1)CC(=O)c2ccc(cc2)Cl BS-6360 CSc1[nH]c(=O)c2c(n1)c(cs2)c3cccc(c3)Br BS-6361 CSc1[nH]c(=O)c2c(n1)c(cs2)c3ccc(cc3)Br BS-6362 COC(=O)/C(=C/Nc1ccc(cc1F)F)/S(=O)(=O)c2ccccc2 BS-6363 COC(=O)/C(=C/Nc1ccc(c(c1)F)F)/S(=O)(=O)c2ccccc2 BS-6364 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3OC BS-6366 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3cccc(c3)OC BS-6367 COc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3cccc(c3)OC BS-6368 COc1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6369 COc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3OC BS-6370 COc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6372 COc1ccccc1CC(c2n[nH]nn2)C(=O)Nc3ccccc3OC BS-6373 COc1cccc(c1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6374 COc1ccc(c(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3)OC BS-6375 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(cc4)F BS-6376 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cccc(c4)F BS-6377 CCOC(=O)Cc1[nH]c(nn1)CN2CCN(CC2)C(=O)OC(C)(C)C BS-6378 CN1CCC(=NNc2ccc(cn2)S(=O)(=O)N3CCOCC3)CC1 BS-6379 CC(C)c1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)OC BS-6380 CCCn1c(=O)c2c(c(cs2)c3ccccc3)nc1N4CCCCC4 BS-6382 CC(C)(C)OC(=O)NCC(=O)N1CCN(CC1)c2cccc(c2)Cl BS-6385 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3ccoc3)C(F)(F)F BS-6387 CC12CC(c3cccc(c3O1)OC)NC(=O)N2c4cccc(c4)C(=O)O BS-6394 c1cc(cc(c1)F)Cn2cnc3c(csc3c2=O)c4cccc(c4)F BS-6396 CCOc1ccc(cc1)NC(=O)C(Cc2cc(ccc2OC)OC)C#N BS-6398 CCOc1ccccc1NC(=O)C(Cc2ccc(c(c2)OC)OC)C#N BS-6399 CCOc1ccc(cc1)NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6400 CCOc1ccccc1NC(=O)C(Cc2ccc(cc2OC)OC)C#N BS-6401 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccs4 BS-6405 c1cc(cc2c1cc(c(=O)o2)S(=O)(=O)c3ccc(c(c3)Cl)F)O BS-6406 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3cc(ccc3C)Cl)C BS-6407 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3cccc(c3C)Cl)C BS-6408 CC(C)(C)OC(=O)NC1CCN(CC1)CC(c2ccc(cc2)Cl)O BS-6409 c1cc(ccc1S(=O)(=O)c2cc3cc(ccc3oc2=O)Cl)Cl BS-6410 COc1ccc(cc1CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])C=O BS-6413 c1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCCC(C4)C(=O)O BS-6415 c1cscc1C(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4 BS-6416 COc1ccccc1CC(=O)NC2(CCCCC2)c3nc(no3)C4CC4 BS-6418 COc1ccc(cc1)Cn2c(=O)c3c(c4cccnc4s3)[nH]c2=S BS-6419 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NCc4cccs4 BS-6420 CC(C)c1nc(on1)CC2CCN(CC2)C(=O)CCCc3ccccc3 BS-6421 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NC4CCCCC4 BS-6422 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)NC4CCCCC4 BS-6423 c1cc(ccc1CN2Cc3cc(ccc3OCC2=O)Cl)C(F)(F)F BS-6424 c1cc(cc(c1)C(F)(F)F)CN2Cc3cc(ccc3OCC2=O)Cl BS-6425 Cc1ccc(cc1C)C(=O)c2cnc3cc(c(cc3c2Cl)OC)OC BS-6426 COc1ccc(cc1OC)C(=O)CS(=O)(=O)c2ccc(cc2F)F BS-6427 Cc1nc(cc(n1)N2CCN(CC2)C(=O)c3cccs3)C(F)(F)F BS-6429 Cc1nc(cc(n1)N2CCN(CC2)C(=O)c3ccsc3)C(F)(F)F BS-6430 Cc1ccc(s1)C(=O)N2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6432 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)C3CCCC3)C(F)(F)F BS-6433 CC(C)(C)OC(=O)/C(=C\N(C)C)/S(=O)(=O)c1ccccc1[N+](=O)[O-] BS-6434 Cc1ccc(cc1)n2ccc(=O)c(n2)S(=O)(=O)c3ccc(cc3)OC BS-6435 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1)OCc2ccccc2 BS-6436 CC(C)(C)OC(=O)Cn1cc(ccc1=O)S(=O)(=O)N2CCCCC2 BS-6437 c1cc(ccc1Cn2cc(nc2)C(=O)Nc3ccc(cc3)Cl)[N+](=O)[O-] BS-6442 Cc1ccc(cc1)S(=O)(=O)c2c(c3cc4c(cc3[nH]c2=O)OCO4)C BS-6443 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3cccc4c3cccc4 BS-6446 Cc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)OC(C)(C)C BS-6450 CC(C)c1ccc(cc1)Sc2ccc(nn2)N3CCC(CC3)C(=O)O BS-6452 CC(C)c1ccc(cc1)Sc2ccc(nn2)N3CCCC(C3)C(=O)O BS-6453 c1cc(ccc1C(=O)O)Nc2c(nn[nH]2)C(=O)Nc3ccc(cc3)Cl BS-6454 COc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3Cl BS-6455 c1cc(ccc1Cn2cc(nc2)C(=O)Nc3cc(ccc3F)F)[N+](=O)[O-] BS-6456 c1ccc(cc1)Oc2ccc(cc2)n3c(c(nn3)C(=O)O)c4ccccn4 BS-6457 c1ccc(cc1)Oc2ccc(cc2)n3c(c(nn3)C(=O)O)c4ccncc4 BS-6458 Cc1ccc(cc1)S(=O)(=O)c2cc3cc(ccc3oc2=O)C(=O)OC BS-6459 Cc1ccc(cc1)n2ccc(=O)c(n2)c3nc(no3)c4ccc(c(c4)C)C BS-6460 CCc1ccc(cc1)S(=O)(=O)c2cc3cccc(c3oc2=O)OCC BS-6462 C=Cc1ccc(cc1)Cn2cc(ccc2=O)S(=O)(=O)N3CCCCC3 BS-6464 c1cc(ccc1Cn2c(c(nn2)C(=O)O)c3ccncc3)Br BS-6466 Cc1cc(ccc1Br)S(=O)(=O)Cc2ccc(o2)C(=O)O BS-6467 c1cc(c(cc1Br)F)S(=O)(=O)/C(=C/2\CCCCN2)/C#N BS-6468 c1ccc(cc1)c2nc(on2)c3cncnc3Nc4ccc5c(c4)OCO5 BS-6469 CC(C)(C)OC(=O)NCC(=O)Nc1ccc(cc1)NC(=O)c2ccco2 BS-6470 Cc1cccc(c1)c2ccc(=O)n(n2)CCN3C(=O)c4ccccc4C3=O BS-6471 c1ccc(c(c1)N2CCN(CC2)C(=O)Cn3c(=O)n4c(n3)CCCC4)F BS-6477 Cc1ccc(cc1)NS(=O)(=O)c2c(cn[nH]2)C(=O)n3c(cc(n3)C)C BS-6478 Cc1cc(n(n1)C(=O)c2c(n[nH]c2S(=O)(=O)Nc3ccccc3)C)C BS-6479 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2)/C(=O)OC BS-6480 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C BS-6481 c1ccc(c(c1)CC(=O)NC2(CCCCC2)c3nc(no3)C4CC4)Cl BS-6483 CCc1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Br BS-6484 c1cc(cc(c1)NC(=O)c2cn(cn2)Cc3ccc(cc3)N)C(F)(F)F BS-6485 COc1ccc(cc1)S(=O)(=O)c2cnc3c(cccn3c2=O)C(=O)O BS-6486 COc1ccc(cc1)S(=O)(=O)c2c(=O)ccn(n2)c3ccc(cc3)F BS-6487 CCOC(=O)c1cc(n(n1)CC(=O)c2cccc(c2)OC)C(=O)OCC BS-6488 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)OC(C)(C)C)C(F)(F)F BS-6489 Cc1ccc(cc1C)S(=O)(=O)c2c3[nH]c(=O)c4c(n3nn2)ccs4 BS-6492 COC(=O)c1c(c(cs1)c2ccccc2)N/C=C(/C#N)\c3ccccc3 BS-6493 COc1cc(c(cc1n2c(c(nn2)C(=O)O)c3ccncc3)Cl)OC BS-6500 COC(=O)c1c(n(nn1)CC(=O)NC(=O)Nc2ccccc2)C(=O)OC BS-6501 CCO/C=C(/C(=O)c1ccccc1)\S(=O)(=O)c2ccccc2[N+](=O)[O-] BS-6502 COC(=O)/C(=C/Nc1ccc2c(c1)OCO2)/S(=O)(=O)c3ccccc3 BS-6503 CCOc1ccc(cc1)S(=O)(=O)c2cn(c3cc(ccc3c2=O)F)C BS-6504 CCn1cc(c(=O)c2c1cc(c(c2)F)N3CCN(CC3)C)C(=O)OCC BS-6505 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccc(cc3)F BS-6507 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3cccc(c3)F BS-6508 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccccc3F BS-6509 CCOc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2)/C(=O)OC BS-6510 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)OC)/C(=O)OC BS-6511 CCOc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccccc2 BS-6512 COc1ccc(cc1OC)CCN2Cc3cc(ccc3OCC2=O)Cl BS-6520 COc1ccc(cc1)CN2Cc3cc(ccc3OCC2=O)Br BS-6522 COc1ccc(cc1OC)S(=O)(=O)c2cc3ccc(cc3oc2=O)O BS-6523 c1ccc2c(c1)cc(c(=O)o2)c3n[nH]c(=O)c4n3nc(c4)c5cccs5 BS-6524 Cc1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-6529 CCOc1ccc(cc1OCC)c2csc3c2nc([nH]c3=O)SC BS-6541 Cc1ccc(cc1)CC2Nc3c(csc3C(=O)N2C)c4ccc(cc4)C BS-6542 COc1ccc(cc1OC)C(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-6543 COc1ccc(cc1OC)S(=O)(=O)c2c[nH]c3c(c2=O)cccc3F BS-6545 Cc1cc(cc(c1)S(=O)(=O)c2cn(c3cc(c(cc3c2=O)F)F)C)C BS-6547 Cc1cccc(c1)c2nnc(s2)NC(=O)c3cc4ccccc4oc3=O BS-6549 CCc1ccc(cc1)N/C=C(\C(=O)OC)/S(=O)(=O)c2ccccc2F BS-6550 CCc1ccc(cc1)N/C=C(\C(=O)OC)/S(=O)(=O)c2ccc(cc2)F BS-6551 CCc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)F)/C(=O)OC BS-6552 Cc1ccc(cc1)c2nc(on2)C3CCCN3C(=O)c4cccc(c4)OC BS-6556 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NCc4ccccc4 BS-6557 Cc1cc(cc(c1)NC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C)C BS-6558 Cc1ccc(cc1C)NC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C BS-6559 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)NCc4ccccc4 BS-6560 Cc1ccc(cc1)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-6561 Cc1cccc(c1)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-6562 c1cc(c(cc1Cl)C(=O)NC2(CCCCC2)c3nc(no3)C4CC4)F BS-6569 CC(c1ccc(cc1)F)N2Cc3cc(ccc3OCC2=O)Br BS-6570 COc1cc(ccc1O)CC(C#N)C(=O)Nc2cccc(c2)C(F)(F)F BS-6571 Cc1ccccc1C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6574 CC1CCCN(C1)S(=O)(=O)c2ccc(nc2)n3cc(nc3)C(=O)NN BS-6577 Cc1ccc(c(c1)Cn2cnc3c(csc3c2=O)c4cccc(c4)F)C BS-6579 CCOC(=O)c1cc(n(n1)CC(=O)c2ccccc2Cl)C(=O)OCC BS-6581 CCOC(=O)CNS(=O)(=O)c1ccccc1C(=O)c2ccccc2F BS-6586 CCOC(=O)c1ccc(cc1)NC(=O)CS(=O)(=O)c2ccccc2F BS-6587 CCOC(=O)C(CC(=O)c1ccc(cc1)OC)(C(=O)OCC)NC(=O)C BS-6588 c1cc(cnc1)c2nc(on2)C3(CCCCC3)NC(=O)c4cccnc4O BS-6589 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4cccc(c4)F BS-6590 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc(cc4)F BS-6591 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)NCc4ccco4 BS-6594 CC(C)c1ccc(cc1)NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6595 CC(C)c1ccc(cc1)NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6596 CC(C)c1ccc(cc1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6597 Cc1ccccc1CSc2nc3c4cc(ccc4[nH]c3c(=O)n2C)OC BS-6598 Cc1cc(n(n1)C(=O)c2cn(nc2S(=O)(=O)N3CCCCCC3)C)C BS-6599 CCn1cc(c(n1)S(=O)(=O)N2CCCCC2)C(=O)n3c(cc(n3)C)C BS-6600 c1cc(ccc1S(=O)(=O)c2cc3cc(ccc3oc2=O)[N+](=O)[O-])Cl BS-6601 Cc1ccc(cc1C)c2nc(on2)c3nc(n(n3)c4ccc(cc4)Cl)C BS-6602 c1cc(ccc1Cn2cc(nc2)C(=O)Nc3ccc4c(c3)OCO4)[N+](=O)[O-] BS-6605 COc1cc2c(cc1OC)-c3nc4cc(ccc4c(=O)n3CC2)C(=O)OC BS-6607 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)F BS-6609 COc1cccc(c1)Cn2cnc3c(csc3c2=O)c4cccc(c4)F BS-6614 c1ccc(cc1)c2csc3c2ncn(c3=O)CCOc4ccc(cc4)F BS-6616 Cc1ccc(cc1C)n2c(c(nn2)C(=O)Nc3ccc(cc3OC)OC)C BS-6617 Cc1cccc(c1)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-6618 Cc1ccccc1Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-6619 Cc1ccc(cc1)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-6620 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4)CCCCC3 BS-6621 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)C)CCCC3 BS-6622 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4C)CCCC3 BS-6623 Cc1ccc(cc1)c2nc(on2)CCN3CCN(CC3)c4ccc(cc4)F BS-6624 c1cc(ccc1CN2Cc3cc(ccc3OCC2=O)Br)Cl BS-6627 c1cc(cc(c1)Br)CN2Cc3cc(ccc3OCC2=O)Cl BS-6628 COc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)Cl)/C(=O)OC BS-6629 Cc1ccc(cc1)N/N=C(\C(=O)OC)/S(=O)(=O)c2ccc(cc2)Cl BS-6630 Cc1cccc(c1)S(=O)(=O)/C(=C/Nc2ccc(c(c2)F)F)/C(=O)OC BS-6646 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)F)F)/C(=O)OC BS-6647 Cc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3ccc(c(c3)OC)OC BS-6650 Cc1cc(cc(c1)NC(=O)C(Cc2ccc(c(c2)OC)O)c3n[nH]nn3)C BS-6651 CCc1ccccc1NC(=O)C(Cc2ccc(c(c2)OC)O)c3n[nH]nn3 BS-6652 Cc1ccc(c(c1)NC(=O)C(Cc2ccc(c(c2)OC)O)c3n[nH]nn3)C BS-6653 CCOc1ccc(cc1)NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6654 CCOc1ccccc1NC(=O)C(Cc2ccc(cc2)OC)c3n[nH]nn3 BS-6655 CCOc1ccccc1NC(=O)C(Cc2cccc(c2)OC)c3n[nH]nn3 BS-6656 Cc1ccc(cc1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-6657 Cc1ccccc1NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-6658 Cc1cccc(c1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-6659 CCOc1ccccc1NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6660 CCOc1ccc(cc1)NC(=O)C(Cc2ccccc2OC)c3n[nH]nn3 BS-6661 Cc1ccccc1NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3 BS-6662 Cc1cccc(c1)NC(=O)C(Cc2cccc(c2OC)OC)c3n[nH]nn3 BS-6663 Cc1ccccc1NC(=O)C(Cc2cccc(c2OC)OC)c3n[nH]nn3 BS-6664 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(cc4)F BS-6666 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cccc(c4)F BS-6667 Cc1ccc(cc1F)NC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C BS-6668 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(cc4)F BS-6669 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4cccc(c4)F BS-6670 Cc1ccsc1C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-6672 c1ccc(cc1)c2nc(on2)C3CCCN3C(=O)Cc4ccccc4Cl BS-6678 c1ccc(cc1)CC(=O)N2CCCC2c3nc(no3)c4ccccc4Cl BS-6679 CCN(CC)c1ccc2cc(c(=O)oc2c1)c3[nH]c4ccc(cc4n3)Cl BS-6680 c1cc(ccc1CC(=O)N2CCN(CC2)c3cc(ncn3)C(F)(F)F)F BS-6682 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NCc3ccco3)C(F)(F)F BS-6683 c1cc(oc1)CNC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4 BS-6685 CC(C)c1ccc(cc1)S(=O)(=O)c2c3[nH]c(=O)c4ccccc4n3nn2 BS-6686 CCOc1ccccc1CNC(=O)C2CC(=O)N(C2)c3ccc(cc3)OC BS-6687 Cc1ccc(cc1)NC(=O)c\2cc3ccccc3o/c2=N\c4ccc(cc4)C BS-6688 Cc1ccc(s1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-6690 Cc1ccsc1C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-6691 Cc1ccccc1c2ccc(nn2)N3CCC(CC3)NC(=O)OC(C)(C)C BS-6692 c1cc(c(cc1n2c(c(nn2)C(=O)O)c3ccncc3)C(F)(F)F)Cl BS-6693 c1cc(c(cc1C(F)(F)F)n2c(c(nn2)C(=O)O)c3ccncc3)Cl BS-6694 COc1ccc2c(c1)cc(c(=O)o2)S(=O)(=O)c3ccc(c(c3)Cl)F BS-6695 COc1cccc2c1oc(=O)c(c2)S(=O)(=O)c3ccc(c(c3)Cl)F BS-6696 COc1ccc2cc(c(=O)oc2c1)S(=O)(=O)c3ccc(c(c3)Cl)F BS-6697 COc1cccc(c1)NC(=O)C(Cc2ccc(c(c2)OC)O)c3n[nH]nn3 BS-6699 Cc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCCC(C4)C(=O)O BS-6705 c1cc(sc1)CC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4 BS-6706 Cn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cccc(c3)Cl BS-6708 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cccc(c4)Cl BS-6709 c1cc(oc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-6711 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)F)CCCCC3 BS-6712 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)F)CCCCC3 BS-6713 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)F)CCCC3 BS-6714 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4F)CCCC3 BS-6715 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)F)CCCC3 BS-6716 Cc1ccsc1C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6720 Cc1ccc(s1)C(=O)N2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-6722 Cc1ccc(cc1)C2Cn3c(c(nn3)C(=O)N4CCC(CC4)C(=O)O)CO2 BS-6723 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NC3CCCCC3)C(F)(F)F BS-6724 CC1CCC(CC1)NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6725 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)C3CCCCC3)C(F)(F)F BS-6726 Cc1ccc(cc1)N/N=C(\C(=O)OC)/S(=O)(=O)CC(=O)OC(C)(C)C BS-6727 CCOC(=O)C1=CN(S(=O)(=O)N=C1c2ccccc2)Cc3ccccc3 BS-6728 Cc1ccc(cc1)N2c3c(cccn3)S(=O)(=O)C(=N2)C(=O)N4CCCC4 BS-6729 c1ccc(cc1)c2nc(on2)C3(CCCCC3)NC(=O)NCC4CCCO4 BS-6730 Cc1ccc(cc1)CSc2c(cccn2)S(=O)(=O)Nc3ccccc3 BS-6731 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc(s2)Cl)C(=O)OCC BS-6733 c1cc(cc(c1)Cl)c2csc3c2ncn(c3=O)Cc4ccc(cc4)F BS-6734 Cc1ccc(cc1)CNC(=O)c2ncn(n2)CC(c3ccc(cc3)Cl)O BS-6739 COC(=O)/C(=C\Nc1ccc(c(c1)F)F)/S(=O)(=O)c2ccccc2F BS-6740 COc1ccc(c(c1)OC)CC(c2n[nH]nn2)C(=O)Nc3ccccc3F BS-6741 COc1ccc(c(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3F)OC BS-6742 COc1ccc(c(c1)CC(c2n[nH]nn2)C(=O)Nc3ccc(cc3)F)OC BS-6743 COc1cccc(c1OC)CC(c2n[nH]nn2)C(=O)Nc3ccccc3F BS-6744 COc1cccc2c1o/c(=N\c3ccccc3)/c(c2)C(=O)Nc4ccccn4 BS-6745 COc1ccc2cc(c(=O)oc2c1)S(=O)(=O)N3CCc4ccccc4C3 BS-6746 CCN(CC)c1ccc2cc(c(=O)oc2c1)S(=O)(=O)c3ccc(cc3)C BS-6747 c1cc2c(cc1F)[nH]cc(c2=O)S(=O)(=O)c3cc(cc(c3)Cl)Cl BS-6749 c1cc2c(c(c1)F)[nH]cc(c2=O)S(=O)(=O)c3ccc(c(c3)Cl)Cl BS-6750 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NCC3CCCO3)C(F)(F)F BS-6751 CC(C)(C)OC(=O)NCc1nc(no1)C2CC(=O)N(C2)Cc3ccccc3 BS-6752 CC(C)(C)OC(=O)NC1CCN(CC1)c2ccc(nn2)c3ccccc3F BS-6754 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)Cl)CCCC3 BS-6758 c1ccc(cc1)c2nc(on2)c3cncnc3NCc4ccc5c(c4)OCO5 BS-6760 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C#N BS-6763 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3cccc4c3cccc4 BS-6764 COc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3cccc4c3cccc4 BS-6765 c1ccc2c(c1)cc(c(=O)o2)c3cn4cnc5c(c4n3)c6c(s5)CCCC6 BS-6766 CCc1ccc(cc1)NS(=O)(=O)c2c(cn[nH]2)C(=O)n3c(cc(n3)C)C BS-6767 Cc1ccc(cc1)NS(=O)(=O)c2c(c(n[nH]2)C)C(=O)n3c(cc(n3)C)C BS-6768 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccc(cc3)OC BS-6769 CCOc1ccc(cc1)N(C)/C=C(\C(=O)C)/S(=O)(=O)c2ccc(cc2)C BS-6770 Cc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C(C)C BS-6771 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)CC BS-6772 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2)/C(=O)OC BS-6773 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCc5ccccc5C4 BS-6774 Cc1ccc(cc1)CNC(=O)CCCn2c(=O)c3c(ccs3)[nH]c2=S BS-6775 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(c(c4)F)F)CCCC3 BS-6776 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc3c(c2)OCO3)C(=O)OCC BS-6777 CCOc1ccc(cc1)C(=O)Cn2c(cc(n2)C(=O)OCC)C(=O)OCC BS-6778 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cccc(c4)C#N BS-6782 c1ccc(cc1)/C=C\C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-6783 COC(=O)/C(=C/Nc1ccc2c(c1)OCCO2)/S(=O)(=O)c3ccccc3 BS-6790 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)OC BS-6791 Cc1ccc(cc1C)S(=O)(=O)/C(=C\Nc2ccc(cc2)OC)/C(=O)OC BS-6792 CCc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)OC)/C(=O)OC BS-6793 CCOc1ccc(cc1)N/C=C(\C(=O)OC)/S(=O)(=O)c2ccc(cc2)C BS-6794 CN(c1ccccc1)C(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-6797 Cc1ccc(cc1)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-6798 Cc1ccccc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-6800 c1ccc(cc1)CNC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-6801 Cc1ccc(cc1C)NS(=O)(=O)c2c3ccccc3sc2C(=O)OC BS-6803 Cc1cccc(c1)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-6804 Cc1ccc(c(c1)C)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-6805 Cc1ccc(cc1)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-6806 Cc1cc(n(n1)C(=O)c2c(ccs2)N(C)S(=O)(=O)c3ccccc3)C BS-6808 CCOc1ccc(cc1OCC)CN2Cc3cc(ccc3OCC2=O)Cl BS-6809 CCOc1cccc(c1)CN2Cc3cc(ccc3OCC2=O)Br BS-6810 COc1ccc(c(c1)S(=O)(=O)c2cc3cccc(c3oc2=O)OC)OC BS-6811 COc1ccc2cc(c(=O)oc2c1)S(=O)(=O)c3ccc(c(c3)OC)OC BS-6812 COc1ccc2c(c1)cc(c(=O)o2)S(=O)(=O)c3ccc(c(c3)OC)OC BS-6813 COc1cccc2c1oc(=O)c(c2)S(=O)(=O)c3ccc(c(c3)OC)OC BS-6814 Cc1ccc(c(c1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4)C BS-6821 Cc1cccc(c1)CC(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-6822 Cc1cc(cc(c1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4)C BS-6824 Cc1ccccc1NC(=O)NC2(CCCCC2)c3nc(no3)c4ccccc4 BS-6833 Cc1ccc(cc1)NC(=O)CN2CCC3(CC2)NC(=O)C(=N3)c4ccccc4 BS-6834 CCOc1ccc(cc1OCC)c2csc(c2/N=C/N(C)C)C(=O)OC BS-6835 CC(C)(C)c1ccc(cc1)S(=O)(=O)c2cc3cc(ccc3oc2=O)Cl BS-6838 Cc1cc(n(n1)C(=O)c2c(n[nH]c2S(=O)(=O)Nc3ccc(cc3)F)C)C BS-6840 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)C#N)CCCCC3 BS-6841 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)C#N)CCCC3 BS-6842 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)C#N)CCCC3 BS-6843 CCn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cc(cc(c3)C)C BS-6844 COc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)OC BS-6845 COc1ccc(cc1OC)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccccc2 BS-6846 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)F)/C(=O)OC BS-6847 c1ccc2c(c1)CCN(C2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)F BS-6848 COc1ccccc1C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-6849 CCOc1ccc(cc1)CC(=O)N2CCCC2c3nc(no3)c4ccccc4 BS-6858 COc1ccc(cc1)c2nc(on2)C3CCCN3C(=O)CCc4ccccc4 BS-6859 Cc1cc(cc(c1)C(=O)N2CCCC2c3nc(no3)c4ccc(cc4)OC)C BS-6860 Cc1ccc(cc1C)C(=O)N2CCCC2c3nc(no3)c4ccc(cc4)OC BS-6861 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cc(cc(c4)C)C BS-6863 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)C)C BS-6864 Cc1ccc(cc1)CCNC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C BS-6865 Cc1cccc(c1)CNC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-6866 CCc1ccc(cc1)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-6867 Cc1ccc(cc1C)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-6868 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccc(cc3)Cl BS-6870 COC(=O)/C(=C\1/CCCN1)/S(=O)(=O)c2ccc(cc2F)Br BS-6871 COc1ccc(c(c1)CC(C#N)C(=O)Nc2cccc(c2)C(F)(F)F)OC BS-6872 COc1ccc(c(c1)OC)CC(C#N)C(=O)Nc2cccc(c2)C(F)(F)F BS-6873 CC(c1ccccc1)NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6874 Cc1ccc(c(c1)C)NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6876 CCc1ccc(cc1)NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6877 Cc1ccc(cc1)C(=O)NC2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-6878 Cc1ccc(cc1C)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6880 Cc1ccc(cc1)CC(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6881 Cc1ccc(c(c1)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F)C BS-6882 Cc1ccc(c(c1)C(=O)N2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F)C BS-6883 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(cc4)C(=O)N BS-6884 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)C=C)CCCC3 BS-6885 CCOC(=O)c1c[nH]nc1S(=O)(=O)N2CCN(CC2)c3cccc(c3)C BS-6891 COC(=O)c1ccc2c(c1)cc(c(=O)o2)S(=O)(=O)c3ccc(cc3)Cl BS-6895 COC(=O)c1c(n(nn1)CC(=O)NC(=O)Nc2ccccc2F)C(=O)OC BS-6896 COC(=O)/C(=C\Nc1ccc2c(c1)OCO2)/S(=O)(=O)c3ccc(cc3)F BS-6897 c1ccnc(c1)CCNC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6898 CCOc1ccc(cc1)N/C=C(\C(=O)OC)/S(=O)(=O)c2ccc(cc2)F BS-6899 CCOc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)F)/C(=O)OC BS-6900 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4ccccc4F BS-6903 c1ccc(cc1)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-6907 COc1cc(cc(c1)OC)NC(=O)c2c(c3cccnc3s2)n4cccc4 BS-6908 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4cccc(c4)OC BS-6909 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(cc4)OC BS-6910 Cc1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3ccsc3C(=O)N)C BS-6912 CCOC(=O)c1cc(n(n1)CC(=O)Nc2ccc(cc2)Cl)C(=O)OCC BS-6913 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)Cl BS-6915 Cc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2nc(cs2)c3ccc(cc3)Cl BS-6916 c1cc(oc1C(=O)NC2(CCCCC2)c3nc(no3)C4CC4)Br BS-6917 COC(=O)/C(=N\Nc1ccc(cc1)C(=O)O)/S(=O)(=O)c2ccccc2F BS-6918 COc1cc(cc(c1OC)OC)c2nc(on2)c3nc(no3)c4ccccc4 BS-6919 COc1ccc(cc1)NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6920 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)/C=C/c3ccco3)C(F)(F)F BS-6921 COc1ccccc1C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6922 c1ccc(cc1)OCC(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6923 Cc1nc(cc(n1)N2CCN(CC2)C(=O)c3ccccc3OC)C(F)(F)F BS-6924 Cc1nc(cc(n1)N2CCN(CC2)C(=O)COc3ccccc3)C(F)(F)F BS-6925 Cc1cccc(c1)OCC(=O)N2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6926 COc1cccc(c1)CC(=O)N2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6927 c1ccc(cc1)C(=O)N/N=c\2/c(cc3ccccc3o2)c4[nH]c5ccccc5n4 BS-6929 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccccc4F BS-6935 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4cccc(c4)F BS-6937 c1ccc(cc1)c2nc(on2)C3(CCCCC3)NC(=O)Nc4ccccc4F BS-6939 c1cc(cc(c1)F)CC(=O)NC2(CCCCC2)c3nc(no3)c4cccnc4 BS-6940 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4C)C)CCCC3 BS-6942 Cc1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3ccsc3C(=O)O)C BS-6946 c1ccc2c(c1)cc(c(=O)o2)c3csc(n3)c4c5c(sc4N)CCCC5 BS-6947 c1cc(ccc1CCN2Cc3cc(ccc3OCC2=O)Br)Cl BS-6948 COc1ccc(cc1OC)S(=O)(=O)c2cc3cc(ccc3oc2=O)Cl BS-6949 Cc1ccc(cc1Cl)N2C(=O)NC3(N2)CCN(CC3)C(=O)OC(C)(C)C BS-6950 c1cc(ccc1S(=O)(=O)c2cc3ccc(cc3oc2=O)O)Br BS-6952 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4)CCCC3 BS-6953 Cc1cccc(c1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccnc5 BS-6957 Cc1ccc(c(c1)C)S(=O)(=O)/C(=C\Nc2ccc(c(c2)F)F)/C(=O)OC BS-6959 CCc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)F)F)/C(=O)OC BS-6960 c1ccnc(c1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-6965 Cc1ccc(c(c1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3)C BS-6966 CCc1ccc(cc1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-6967 Cc1ccc(cc1C)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-6968 Cc1cc(cc(c1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3)C BS-6969 Cc1ccc(c(c1)C)NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3 BS-6970 CCc1ccccc1NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3 BS-6971 Cc1cccc(c1C)NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3 BS-6972 Cc1ccc(c(c1)NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3)C BS-6973 CCc1ccc(cc1)NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3 BS-6974 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)F)C BS-6975 Cc1ccc(cc1F)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-6976 CCOC(=O)C1CCN(CC1)c2c(cccn2)S(=O)(=O)N3CCCCC3 BS-6977 CCc1ccc(cc1)Nc2c(cccn2)S(=O)(=O)Nc3ccc(cc3)CC BS-6978 CCOC(=O)CNS(=O)(=O)c1ccc(cc1C(=O)c2ccccc2)Cl BS-6979 COc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Cl)/C(=O)OC BS-6980 COc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)Cl BS-6981 Cc1ccc(cc1)c2nc(on2)C3CCCN3C(=O)Cc4ccccc4Cl BS-6986 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3ccccc3F)C(F)(F)F BS-6987 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3cccc(c3)F)C(F)(F)F BS-6988 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3ccc(cc3)F)C(F)(F)F BS-6989 Cc1ccc(cc1F)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-6990 c1cc(ccc1CC(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F)F BS-6991 Cc1ccc(cc1F)C(=O)N2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-6992 Cc1nc(cc(n1)N2CCN(CC2)C(=O)Cc3cccc(c3)F)C(F)(F)F BS-6993 c1ccc(c(c1)NC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4)F BS-6994 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)OC)CCCCC3 BS-6996 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4OC)CCCC3 BS-6997 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)OC)CCCC3 BS-6998 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)OC)CCCC3 BS-6999 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccsc4 BS-7003 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccs4 BS-7004 Cc1ccccc1NC(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4 BS-7005 Cc1cccc(c1)CNCCNC(=O)C(=O)NCCNCc2cccc(c2)C BS-7006 CCN(c1cccc(c1)C)C(=O)COc2cc(nc(n2)N3CCCCCC3)C BS-7007 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)Cl BS-7008 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)Cl BS-7009 c1cc(ccc1F)S(=O)(=O)c2cc3cc(ccc3oc2=O)Br BS-7019 CCOC(=O)c1ccc(cc1)NC(=O)CS(=O)(=O)c2cc(ccc2F)F BS-7020 COc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)F)F)/C(=O)OC BS-7021 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4cc(ccc4F)F BS-7022 CCOc1ccc(cc1)NC(=O)C(Cc2ccc(c(c2)OC)O)c3n[nH]nn3 BS-7023 CCOc1ccccc1NC(=O)C(Cc2ccc(c(c2)OC)O)c3n[nH]nn3 BS-7024 COc1ccc(cc1)NC(=O)C(Cc2cccc(c2OC)OC)c3n[nH]nn3 BS-7025 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3ccc(c(c3)OC)OC BS-7026 COc1cccc(c1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-7027 COc1ccc(cc1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-7028 COc1cccc(c1)NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3 BS-7029 COc1ccc(c(c1)CC(c2n[nH]nn2)C(=O)Nc3ccccc3OC)OC BS-7030 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)CCC(=O)NCc3ccc(cc3)C(=O)O BS-7031 CCOC(=O)CNS(=O)(=O)c1c(csc1C(=O)OC)c2ccccc2 BS-7032 CCOC(=O)C1CCN(CC1)C(=O)c2c(c3cccnc3s2)n4cccc4 BS-7034 CCn1cc(c(n1)S(=O)(=O)N2CCSCC2)C(=O)n3c(cc(n3)C)C BS-7037 COc1ccc(cc1)c2nc(on2)C3CCCN3C(=O)c4cccc(c4)Cl BS-7038 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cccc(c4)Cl BS-7040 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(cc4)Cl BS-7041 Cc1ccc(cc1Cl)NC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C BS-7042 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4cccc(c4)Cl BS-7043 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(cc4)Cl BS-7044 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)F BS-7046 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(ccc4F)F BS-7047 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)F)F BS-7048 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4F)CCCCC3 BS-7050 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)F)CCCCC3 BS-7051 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NCc3cccs3)C(F)(F)F BS-7052 CCOC(=O)c1c(cc(=O)n2c1CCCC2)OCC(=O)Nc3ccc(cc3)C BS-7057 c1cc2c(cc1NC(=O)NC3(CCCCC3)c4nc(no4)C5CC5)OCCO2 BS-7058 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NCC3CCCCC3)C(F)(F)F BS-7062 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NC3CCCCCC3)C(F)(F)F BS-7063 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NC3CCC(CC3)C)C(F)(F)F BS-7064 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)CCC3CCCC3)C(F)(F)F BS-7065 CC(C)(C)OC(=O)NC1CCN(CC1)c2ccc(nn2)c3ccccc3OC BS-7067 c1cc(c(cc1F)Cl)CN2Cc3cc(ccc3OCC2=O)Br BS-7068 c1ccc(c(c1)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F)Cl BS-7069 c1ccc(c(c1)CC(=O)N2CCN(CC2)c3cc(ncn3)C(F)(F)F)Cl BS-7071 Cc1ccc(cc1)COc2cc(=O)n(nc2C(=O)OC)c3ccc(cc3)Cl BS-7073 c1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3c(c[nH]n3)C(=O)NN)Cl BS-7074 Cc1ccc(c(c1)C)NC(=O)c2c(n(nn2)c3ccc(cc3)Br)C BS-7076 CCOC(=O)c1cc(n(n1)CCN2C(=O)c3ccccc3C2=O)C(=O)OCC BS-7079 COc1ccc(cc1)C(=O)Cn2c3cc(nn3c(=O)c(n2)C#N)c4ccccc4 BS-7080 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(c(c4)F)F BS-7081 c1cc(cc(c1)F)CC(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4 BS-7083 Cc1ccc(cc1)S(=O)(=O)N/N=C(\c2ccccc2)/C(=O)N3CCCCC3 BS-7086 Cc1ccc(cc1)n2c(=O)n(c(=O)c(n2)C(=O)OC)Cc3ccc(cc3)Cl BS-7087 c1cc(c(c(c1)F)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F)F BS-7091 Cc1nc(cc(n1)N2CCN(CC2)C(=O)c3cc(ccc3F)F)C(F)(F)F BS-7092 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(c(c4)F)OC)CCCC3 BS-7093 c1ccc(cc1)c2csc3c2ncn(c3=O)Cc4cccc(c4)C(F)(F)F BS-7094 Cc1nc(on1)C2(CCCCC2)NC(=O)C3CC(=O)N(C3)c4cccc(c4)F BS-7095 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4ccc(cc4)C#N BS-7096 c1cc(ccc1Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccsc4)F BS-7099 c1cc(sc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-7100 Cc1ccc(cc1)CN2c3ccccc3S(=O)(=O)C(=N2)C(=O)OC(C)(C)C BS-7105 Cc1ccc(cc1)Cn2c(=O)n3cccc(c3n2)S(=O)(=O)N4CCCCC4 BS-7107 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccc(cc3)N(C)C BS-7108 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)Cl)CCCCC3 BS-7111 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4Cl)CCCCC3 BS-7112 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)Cl)CCCC3 BS-7113 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccccc4Cl)CCCC3 BS-7114 Cc1c(nnn1c2ccc(cc2)Br)C(=O)Nc3ccc(cc3)OC BS-7115 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccc4c(c3)OCO4 BS-7117 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NC4CCCC4)CCCC3 BS-7119 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NC4CCCCC4)CCCC3 BS-7120 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C#N BS-7121 CCOc1ccccc1c2nc(on2)CC3CCN(CC3)C(=O)OC(C)(C)C BS-7127 Cc1ccc(cc1)N(C)S(=O)(=O)c2c(csc2C(=O)O)c3ccccc3 BS-7128 Cc1ccc(cc1)NS(=O)(=O)c2c(csc2C(=O)NN)c3ccccc3 BS-7129 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C(C)C BS-7130 Cc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C(C)(C)C BS-7131 COC(=O)/C(=C\Nc1ccc(c(c1)F)F)/S(=O)(=O)c2cccc(c2)Cl BS-7132 COC(=O)/C(=C/Nc1ccc(c(c1)F)F)/S(=O)(=O)c2ccc(cc2)Cl BS-7133 COC(=O)/C(=C/Nc1ccc(cc1F)F)/S(=O)(=O)c2ccc(cc2)Cl BS-7134 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)Cl)F BS-7135 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(c(c4)F)F)CCCC3 BS-7136 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4F)F)CCCC3 BS-7137 CC(C)(C)OC(=O)N1CCC(CC1)c2n[nH]c(=O)n2Cc3ccc(cc3)OC BS-7139 c1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5 BS-7143 c1ccc2c(c1)ccc3c2cc(c(=O)o3)S(=O)(=O)c4ccc(c(c4)Cl)F BS-7144 Cc1ccc(cc1)NC(=O)c\2cc3ccccc3o/c2=N\c4ccc(cc4)Cl BS-7145 COc1ccc(cc1Cn2c(c(nn2)C(=O)O)c3cccnc3)Br BS-7146 CCOC(=O)c1c(n(nn1)CC(=O)NC(=O)Nc2ccccc2)C(=O)OCC BS-7147 Cc1cccc(c1C)NC(=O)NC(=O)Cn2c(c(nn2)C(=O)OC)C(=O)OC BS-7148 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3ccc(cc3)C#N)C(F)(F)F BS-7149 COc1cc(ccc1O)CC(c2n[nH]nn2)C(=O)Nc3cccc4c3cccc4 BS-7150 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCCO3)/C(=O)OC BS-7151 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)c2cn(nn2)c3ccc(cc3)F BS-7152 Cc1cc(n(n1)C(=O)c2c(n[nH]c2S(=O)(=O)Nc3ccc(cc3)OC)C)C BS-7153 CCOc1ccc(cc1)NS(=O)(=O)c2c(cn[nH]2)C(=O)n3c(cc(n3)C)C BS-7154 Cc1ccc(cc1)N/N=C(\C(=O)N2CCCC2)/S(=O)(=O)c3ccccc3F BS-7155 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)OCC BS-7156 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)OC)/C(=O)OC BS-7157 CCOc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(c(c2)C)C BS-7158 CCc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)OCC)/C(=O)OC BS-7159 CCc1ccc(cc1)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7166 Cc1ccc(cc1C)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7168 Cc1cccc(c1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4)C BS-7169 Cc1ccc(c(c1)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4)C BS-7170 Cc1ccc(c(c1)C)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7171 c1ccc(cc1)CCNC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7172 Cc1ccc(cc1)CNC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7173 Cc1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)n3c(cc(n3)C)C BS-7175 CCN(c1ccsc1C(=O)n2c(cc(n2)C)C)S(=O)(=O)c3ccccc3 BS-7176 c1ccc(c(c1)c2nc(on2)C3CCCN3C(=O)c4ccc(c(c4)F)F)Cl BS-7178 CN(c1ccsc1C(=O)OC)S(=O)(=O)c2ccc(cc2)Br BS-7179 c1ccc2c(c1)CCC2NC(=O)C3CCN(CC3)c4cc(ncn4)C(F)(F)F BS-7180 CC(C)(C)OC(=O)NCc1nc(no1)C2CC(=O)N(C2)Cc3ccc(cc3)F BS-7181 Cc1ccc(cc1)N2c3ccc(cc3S(=O)(=O)C(=N2)C(=O)OC(C)(C)C)F BS-7182 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)CCc4ccccc4 BS-7187 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccccc4C BS-7188 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)C)C BS-7191 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)C BS-7192 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C BS-7194 CCOC(=O)N1CCc2c(cc(=O)n(n2)CC(=O)Nc3ccccc3Cl)C1 BS-7196 COc1ccc(cc1)CC(c2n[nH]nn2)C(=O)Nc3cccc(c3)C(F)(F)F BS-7198 COc1cccc(c1)CC(c2n[nH]nn2)C(=O)Nc3cccc(c3)C(F)(F)F BS-7199 COc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCO3)/C(=O)OC BS-7200 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc5c(c4)OCO5 BS-7202 CCCn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cc(cc(c3)C)C BS-7203 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccc(c(c3)F)OC BS-7204 CCOc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)OC BS-7205 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)OC)OC)/C(=O)OC BS-7206 Cc1cccc(c1)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7208 Cc1ccccc1NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7209 c1ccc2c(c1)cc(c(=O)o2)C(=O)Cn3cnc4c(c3=N)c5c(s4)CCCC5 BS-7210 COc1cccc(c1)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7212 COc1ccccc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7213 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)F)/C(=O)OC BS-7214 Cc1ccc(cc1)OCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7215 CCOc1ccccc1C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7216 COc1ccccc1CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7217 CCOc1ccc(cc1)CC(=O)N2CCCC2c3nc(no3)c4ccc(cc4)C BS-7221 c1ccc(cc1)CCNC(=O)NC2(CCCCC2)c3nc(no3)c4cccnc4 BS-7223 CN(C)c1cccc(c1)C(=O)NC2CCN(C2)Cc3nc(on3)c4ccccc4 BS-7225 Cc1ccc(cc1C)CNC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-7226 CC(C)c1ccc(cc1)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-7227 CC(C)c1nc(on1)CC2CCN(CC2)C(=O)Cc3ccc(c(c3)Cl)OC BS-7228 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NCCc3ccccc3)C(F)(F)F BS-7230 Cc1cc(cc(c1)NC(=O)C2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F)C BS-7231 Cc1ccc(cc1C)C(=O)NC2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-7232 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)CCc3ccccc3)C(F)(F)F BS-7233 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)C(C)c3ccccc3)C(F)(F)F BS-7234 Cc1ccc(cc1)CC(=O)NC2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-7235 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(cc4)C(=O)N BS-7238 COc1cccc(c1)CC(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-7241 CCOc1ccccc1C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-7242 Cc1ccc(cn1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-7246 COc1cccc(c1)NC(=O)NC2(CCCCC2)c3nc(no3)c4ccccc4 BS-7247 CCc1ccccc1NC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4 BS-7251 c1ccc(cc1)c2nc(on2)Cn3cccc3C(=O)NCc4cccc(c4)Cl BS-7255 COC(=O)/C(=C\Nc1ccc2c(c1)OCCO2)/S(=O)(=O)c3ccc(cc3)F BS-7257 CCc1ccc(cc1)NC(=O)N2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-7259 c1cc(ccc1NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCCCC3)F BS-7260 Cc1ccc(cc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4)F BS-7265 Cc1ccc(cc1F)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7266 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)NCc4ccc(cc4)F BS-7267 COc1ccc(cc1OC)c2nc(on2)C3CCCN3C(=O)Cc4ccccc4 BS-7274 Cc1ccc(cc1)OCC(=O)N2CCC(CC2)Cc3nc(no3)c4cnccn4 BS-7276 COc1ccccc1NC(=O)NC2(CCCCC2)c3nc(no3)c4cccnc4 BS-7277 Cc1cccc(c1)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-7278 CCc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-7279 Cc1cc(cc(c1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F)C BS-7280 c1cc(c2n[nH]c(=S)n2c1)S(=O)(=O)N3CCN(CC3)c4ccc(cc4)F BS-7281 CCOc1ccc(cc1)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-7282 CCc1ccc(cc1)c2cc3c(=O)n(ccn3n2)CC(c4ccc(cc4)Cl)O BS-7284 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Cl)/C(=O)OC BS-7285 c1ccc2c(c1)CCN(C2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)Cl BS-7287 Cc1cccc(c1)OCC(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7293 CC(C(=O)NC1CCN(CC1)c2cc(ncn2)C(F)(F)F)Oc3ccccc3 BS-7295 COc1cccc(c1)CC(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7296 COc1ccccc1NC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4 BS-7306 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccccc4F BS-7312 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)F BS-7313 CCOc1cccc2c1oc(=O)c(c2)c3[nH]c(=O)c4c5c(sc4n3)CCCC5 BS-7314 Cc1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3ccsc3C(=O)OC)C BS-7318 Cc1nc(on1)C2(CCCCC2)NC(=O)Nc3cc(c(cc3OC)OC)Cl BS-7319 COc1ccc(cc1OC)N/C=C(\C(=O)OC)/S(=O)(=O)c2ccc(cc2)F BS-7320 c1ccc(c(c1)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3)F BS-7322 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4)CCCCC3 BS-7323 Cc1cccc(c1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-7324 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccccc4)CCCC3 BS-7325 CCc1ccc(cc1)N/C=C(\C(=O)OCC)/S(=O)(=O)c2ccc(cc2F)F BS-7328 CC(C)(C)OC(=O)/C(=C\Nc1ccc(cc1)F)/S(=O)(=O)c2ccccc2F BS-7329 CCOC(=O)/C(=C/Nc1ccc(c(c1)F)F)/S(=O)(=O)c2cc(cc(c2)C)C BS-7330 Cc1ccc(cc1F)NC(=O)NC2(CCCCC2)c3nc(no3)c4ccncc4 BS-7334 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)OC)OC BS-7337 CC(C)c1ccc(cc1)NC(=O)C(Cc2ccc(cc2OC)OC)c3n[nH]nn3 BS-7338 COC(=O)/C(=C/Nc1ccc2c(c1)OCO2)/S(=O)(=O)c3ccc(cc3)Cl BS-7341 CCOc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)Cl BS-7342 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)Cc4ccccc4Cl BS-7344 c1ccc(cc1)CCCC(=O)N2CCCC2c3nc(no3)c4ccccc4Cl BS-7346 Cc1cc(n(n1)C(=O)c2c(ccs2)NS(=O)(=O)c3ccc(cc3)Cl)C BS-7347 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)Cc3ccc(cc3)F)C(F)(F)F BS-7349 COc1ccc(cc1)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5ccccc5 BS-7351 COc1ccc(cc1OC)S(=O)(=O)c2cc3c4ccccc4ccc3oc2=O BS-7352 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4ccc(cc4)F BS-7353 COc1ccc(cc1F)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-7354 Cc1ccc(c(c1)C)N2CC(CC2=O)C(=O)NC3(CCCCC3)c4nc(no4)C BS-7357 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(s4)C BS-7359 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4c(ccs4)C BS-7360 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4cccs4 BS-7361 c1cc(c(nc1)NNC(=O)c2ccc(cc2)Cl)S(=O)(=O)N3CCOCC3 BS-7363 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)Cl BS-7366 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccc(cc4)Cl BS-7367 c1ccc(c(c1)CC(=O)NC2(CCCCC2)c3nc(no3)c4ccncc4)Cl BS-7370 c1ccc(cc1)c2nc(on2)C3(CCCCC3)NC(=O)Nc4ccccc4Cl BS-7371 CCOC(=O)/C(=C\Nc1ccc(cc1)OC)/S(=O)(=O)c2cc(ccc2F)F BS-7376 CCOc1ccccc1NC(=O)C(Cc2cc(ccc2OC)OC)c3n[nH]nn3 BS-7380 CCc1ccc(cc1)n2cc(c3ccccc3c2=O)C(=O)OCc4ccc(cc4)C BS-7381 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)Cc4ccsc4 BS-7382 COc1ccccc1CC(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4 BS-7383 CCCn1cc(c(n1)S(=O)(=O)N2CCSCC2)C(=O)n3c(cc(n3)C)C BS-7384 c1cc2c(cc1C#N)ncc(c2Cl)S(=O)(=O)c3cc(cc(c3)Cl)Cl BS-7385 Cc1ccc(cc1Cl)N2C(=O)C3C(C2=O)N(N=N3)CC(=O)Nc4ccccc4 BS-7387 CCCn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cccc(c3)Cl BS-7388 Cc1ccc(cc1)c2nc(on2)C3CCCN3C(=O)c4cc(ccc4OC)Cl BS-7393 COc1ccc(cc1)CC(=O)N2CCCC2c3nc(no3)c4ccccc4Cl BS-7394 c1ccc(c(c1)CC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4)Cl BS-7395 c1cc(cc(c1)Cl)NC(=O)NC2(CCCCC2)c3nc(no3)c4ccncc4 BS-7396 Cc1cc(ccc1Cl)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-7397 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)NCc4cccc(c4)Cl BS-7398 c1cc(ccc1OCC(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F)F BS-7400 Cc1cccc(c1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc(cc5)F BS-7402 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)F)F BS-7405 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NCCc3cccs3)C(F)(F)F BS-7406 Cc1nc(on1)C2(CCCCC2)NC(=O)C3CC(=O)N(C3)c4ccc(cc4)OC BS-7407 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NC3CCCCCCC3)C(F)(F)F BS-7409 Cc1ccc(cc1)CNC(=O)c2cn[nH]c2S(=O)(=O)N(C)c3ccc(cc3)C BS-7410 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccsc4 BS-7411 CCc1ccc(cc1)c2cc([nH]n2)C(=O)N3CCC(CC3)NC(=O)OC(C)(C)C BS-7413 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3cccc(c3)Cl)C(F)(F)F BS-7415 c1cc(ccc1CC(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F)Cl BS-7417 c1ccc(c(c1)NC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4)Cl BS-7418 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)F)CCCC3 BS-7420 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4F)CCCC3 BS-7421 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)F)CCCC3 BS-7422 c1cc(cnc1)c2nc(on2)C3(CCCCC3)NC(=O)Nc4ccc(cc4F)F BS-7423 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc5ccccc5n4 BS-7426 c1ccc2c(c1)ccc(n2)C(=O)NC3(CCCCC3)c4nc(no4)c5cccnc5 BS-7427 CC(C)(C)c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)OC(C)(C)C BS-7429 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)Cl)OC BS-7430 c1cc(ccc1CN2Cc3cc(ccc3OCC2=O)Br)C(F)(F)F BS-7431 c1cc(cc(c1)C(F)(F)F)CN2Cc3cc(ccc3OCC2=O)Br BS-7432 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(o4)C(=O)OC)CCCC3 BS-7436 Cc1cc(no1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-7437 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(on4)C)CCCC3 BS-7438 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(c(c4)F)OC)CCCC3 BS-7439 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CCOc4ccc(cc4)F)CCCC3 BS-7440 CCOC(=O)C1=CN(S(=O)(=O)N=C1c2ccccc2)Cc3ccc(cc3)OC BS-7443 Cc1cc(n(n1)C(=O)c2cn(cn2)c3ccc(cn3)S(=O)(=O)N4CCCC4)C BS-7445 Cc1ccc(s1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-7446 CCCCCCc1cc2cc(c(=O)oc2cc1O)S(=O)(=O)c3ccc(cc3)C BS-7451 CC1CCN(CC1)C(=O)CNS(=O)(=O)c2ccccc2C(=O)c3ccccc3 BS-7452 Cc1ccc(cc1)/N=C/c2cc3ccc(cc3nc2S(=O)(=O)c4ccccc4)C BS-7453 CCN1CCc2c(sc3c2c(=O)n(c(n3)SCC(=O)c4ccccc4)N)C1 BS-7455 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)Cl)F BS-7458 c1ccc(cc1)c2nc(no2)CN3CCC(C3)NC(=O)c4cc(ccc4F)Cl BS-7459 CCOc1ccc(cc1)NC(=O)c2c(n(nn2)c3ccc(cc3)Br)C BS-7461 c1cc(ccc1c2nc(on2)CC3CCN(CC3)C(=O)c4cc(ccc4F)F)F BS-7462 c1ccc(cc1)Nc2c3ccccc3n4c(n2)c(nn4)S(=O)(=O)c5ccccc5 BS-7463 CCOC(=O)C1CCN(CC1)c2[nH]c(=O)c3c(n2)c(cs3)c4ccccc4F BS-7464 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NC4CCCC4)CCCCC3 BS-7465 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NC4CCCCC4)CCCC3 BS-7466 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C#N BS-7467 CCn1c(ccn1)c2nc(no2)C3CCN(CC3)S(=O)(=O)c4ccc(cc4)C BS-7468 Cc1ccc(cc1)N(C)S(=O)(=O)c2c(csc2C(=O)OC)c3ccccc3 BS-7469 Cc1ccc(cc1C)N(C)S(=O)(=O)c2c(csc2C(=O)O)c3ccccc3 BS-7470 Cc1ccc(cc1)N(C)S(=O)(=O)c2c(csc2C(=O)NN)c3ccccc3 BS-7471 CCc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C(C)(C)C BS-7472 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)Cl)F BS-7477 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(c(c4)Cl)F BS-7478 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(c(c4)F)F)CCCCC3 BS-7482 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4F)F)CCCCC3 BS-7483 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cc(ccc4F)F)CCCCC3 BS-7484 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cc(cc(c4)F)F)CCCCC3 BS-7485 COc1ccc(cc1)NC(=O)C2CCCN(C2)c3c4c(c5ccccc5o4)ncn3 BS-7486 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4c5ccccc5[nH]n4 BS-7487 Cn1c2ccccc2c(n1)C(=O)N3CCC(CC3)c4n[nH]c(=O)n4c5ccccc5 BS-7488 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5 BS-7497 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccccc5 BS-7499 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cccc(c4)C(F)(F)F BS-7500 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3cccc4c3cc[nH]4)C(F)(F)F BS-7501 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3cc4ccccc4[nH]3)C(F)(F)F BS-7502 COc1ccc(c(c1)OC)CC(c2n[nH]nn2)C(=O)Nc3cccc4c3cccc4 BS-7504 COc1ccc(c(c1)CC(c2n[nH]nn2)C(=O)Nc3cccc4c3cccc4)OC BS-7505 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCO3)/C(=O)OC BS-7506 CCOc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C(C)C BS-7507 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)OC)/C(=O)OC BS-7508 Cc1cccc(c1C)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCCCC3 BS-7509 CCc1ccc(cc1)NS(=O)(=O)c2cccnc2N3CCC4(CC3)OCCO4 BS-7512 CCc1cccc(c1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4)C BS-7521 Cc1cc(c(c(c1)C)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4)C BS-7522 c1ccc(cc1)CCCNC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7523 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccn5 BS-7524 COc1ccc(cc1)NC(=O)CCCCCn2c(=O)c3c(ccs3)[nH]c2=S BS-7526 CCc1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)n3c(cc(n3)C)C BS-7527 Cc1ccc(cc1C)S(=O)(=O)N(C)c2ccsc2C(=O)n3c(cc(n3)C)C BS-7528 CCN(c1ccsc1C(=O)n2c(cc(n2)C)C)S(=O)(=O)c3ccc(cc3)C BS-7529 Cc1cc(cc(c1)N(C)S(=O)(=O)c2ccsc2C(=O)n3c(cc(n3)C)C)C BS-7530 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCC5(CC4)OCCO5)Cl BS-7531 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)Cl)Cl BS-7532 c1ccc(c(c1)CC(=O)NC2(CCCCC2)c3nc(no3)C4CC4)Br BS-7533 c1cc(cc(c1)C(F)(F)F)Cn2cnc3c(csc3c2=O)c4cccc(c4)F BS-7534 COc1ccc(cc1OC)c2nc(on2)C3CCCN3C(=O)c4ccc(cc4)C#N BS-7536 Cc1nc(cc(n1)N2CCC(CC2)C(=O)NC3CCc4c3cccc4)C(F)(F)F BS-7537 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)C3(CC3)c4ccccc4)C(F)(F)F BS-7538 COc1ccc(cc1)/C(=N/OC(=O)c2c3n(c(n2)c4ccccc4)CCCCC3)/N BS-7542 Cc1ccc(cc1)N/C=C\2/C(=O)c3ccccc3N(S2(=O)=O)Cc4ccccc4 BS-7543 CCc1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)C BS-7545 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)C)C BS-7547 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4c(cccc4Cl)F)CCCC3 BS-7551 CCOc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCO3)/C(=O)OC BS-7553 COc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCCO3)/C(=O)OC BS-7554 CC(=O)Nc1cccc(c1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-7556 CCCCn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cc(cc(c3)C)C BS-7557 CCOc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)OCC BS-7558 Cc1ccc(cc1C)S(=O)(=O)/C(=C\Nc2ccc(c(c2)OC)OC)/C(=O)OC BS-7559 Cc1ccc(c(c1)C)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7560 CCc1ccc(cc1)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7562 Cc1ccc(cc1C)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7565 CCOc1ccccc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7577 COc1cccc(c1)CNC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7579 COc1ccccc1CNC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7580 COc1ccc(cc1)NS(=O)(=O)c2cccnc2N3CCC(CC3)C(=O)NN BS-7581 COc1ccccc1CCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7583 COc1ccc(cc1)CCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7584 COc1cccc(c1)c2nc(on2)CC3CCN(CC3)C(=O)CCc4ccccc4 BS-7585 Cc1ccc(c(c1)C)C(=O)N2CCC(CC2)Cc3nc(no3)c4cccc(c4)OC BS-7586 CCc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-7588 Cc1cc(n(n1)C(=O)c2c(ccs2)N(C)S(=O)(=O)c3ccc(cc3)OC)C BS-7589 CC(C)c1ccc(cc1)CNC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7593 CCC(c1ccccc1)C(=O)NC2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-7594 CC(C)(C)c1ccc(cc1)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7595 Cc1ccc(cc1NC(=O)COc2cc(nc(n2)N3CCc4ccccc4C3)C)F BS-7596 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)NNC(=O)NCc2ccc(cc2)OC BS-7598 c1ccc(cc1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)F BS-7599 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4cccc(c4)C BS-7605 Cc1cccc(c1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-7607 Cc1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-7608 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)OC BS-7609 COc1ccccc1CCC(=O)NC2CCN(C2)Cc3nc(on3)c4ccccc4 BS-7610 COc1cc(ccc1O)CC(c2n[nH]nn2)C(=O)Nc3cccc(c3)C(F)(F)F BS-7617 CCOC(=O)c1c(n(nn1)CC(=O)NC(=O)Nc2ccccc2F)C(=O)OCC BS-7618 c1cc2c(cc1CNC(=O)c3ccc4c(c3)[nH]c(=O)n(c4=O)C5CCCC5)OCO2 BS-7620 c1ccc2c(c1)OCC(O2)C(=O)NC3(CCCCC3)c4nc(no4)c5cnccn5 BS-7621 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3cccc(c3)N(C)C)C(F)(F)F BS-7622 COc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)OC)OC)/C(=O)OC BS-7623 COc1ccc(cc1)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7624 COc1ccccc1NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7626 Cc1cc(ccc1NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCCCC3)F BS-7627 COc1ccc(cc1OC)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7638 COc1ccc(c(c1)OC)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7639 COc1cc(cc(c1)OC)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-7640 COc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4cccc(c4)OC BS-7642 COc1ccc(cc1OC)c2nc(on2)C3CCCN3C(=O)CCc4ccccc4 BS-7650 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc5c(c4)OCCO5 BS-7651 c1ccnc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)F BS-7652 COc1ccc(cc1)CCC(=O)N2CCC(CC2)Cc3nc(no3)c4cnccn4 BS-7653 Cc1cc(ccc1NC(=O)NC2(CCCCC2)c3nc(no3)c4ccncc4)OC BS-7654 Cc1ccc(cc1F)N(C)S(=O)(=O)c2ccsc2C(=O)n3c(cc(n3)C)C BS-7656 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccccc4 BS-7658 CSc1cccc(c1)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7659 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Cl)/C(=O)OC BS-7661 CCOC(=O)c1ccc(cc1)N/N=C(\C(=O)OC)/S(=O)(=O)c2ccccc2F BS-7662 CC(c1ccc(cc1)OC)NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7663 CCOc1ccccc1C(=O)NC2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-7664 Cc1cc(ccc1C(=O)NC2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F)OC BS-7665 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)C(C)Oc3ccccc3)C(F)(F)F BS-7666 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)Cc3cccc(c3)OC)C(F)(F)F BS-7667 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)Cc3ccccc3OC)C(F)(F)F BS-7668 CC(C)(C)OC(=O)N1CCN(CC1)c2cc(nc(n2)c3ccccc3)C(F)(F)F BS-7669 COc1cc(cc(c1)OC)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4 BS-7672 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc(nc4)OC BS-7676 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)F)C BS-7686 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4cccc(c4)F BS-7687 CCOC(=O)c1c(n[nH]c1S(=O)(=O)N2CCN(CC2)c3ccc(cc3)OC)C BS-7688 CCOC(=O)c1cc(n(n1)CC(=O)c2ccc(cc2)Br)C(=O)OCC BS-7694 Cc1cc(ccc1NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3)F BS-7695 COc1cccc(c1)C(=O)N2CCCC2c3nc(no3)c4ccc(c(c4)OC)OC BS-7705 COc1cc(cc(c1OC)OC)C(=O)N2CCCC2c3nc(no3)c4ccccc4 BS-7706 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4)CCCCC3 BS-7707 Cc1cccc(c1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-7708 Cc1ccccc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-7709 Cc1ccc(cc1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-7710 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccccc4)CCCCC3 BS-7711 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccccc4)CCCC3 BS-7712 Cc1ccc(c(c1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C)C BS-7713 Cc1cccc(c1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C)C BS-7714 Cc1ccc(cc1)CNC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-7715 CCc1ccccc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-7716 Cc1ccc(cc1C)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-7717 CCc1ccc(cc1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-7718 Cc1ccc(cc1)OCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-7719 CCOc1ccccc1C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-7720 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)OC)OC BS-7722 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(cc4OC)OC BS-7723 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(c(c4)OC)OC BS-7724 COC(=O)/C(=C/Nc1ccc2c(c1)OCCO2)/S(=O)(=O)c3ccc(cc3)Cl BS-7730 CCN(CC)c1ccc2cc(c(=O)oc2c1)S(=O)(=O)c3ccc(c(c3)Cl)F BS-7731 Cc1ccc(cc1)S(=O)(=O)c2c(c3cc(ccc3[nH]c2=O)Cl)c4ccccc4 BS-7732 Cc1ccc(cc1)N/N=C(\C(=O)OC(C)(C)C)/S(=O)(=O)c2cccnc2Cl BS-7733 c1cc(cc(c1)Cl)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCCCC3 BS-7734 Cc1ccc(c(c1)Cl)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7739 Cc1ccc(cc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4)Cl BS-7740 Cc1c(cccc1Cl)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7741 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)NCc4ccc(cc4)Cl BS-7742 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)NCc4ccccc4Cl BS-7743 Cc1cc(n(n1)C(=O)c2c(ccs2)N(C)S(=O)(=O)c3ccc(cc3)Cl)C BS-7745 Cc1cc(n(n1)C(=O)c2c(ccs2)N(C)S(=O)(=O)c3cccc(c3)Cl)C BS-7746 c1cc(ccc1S(=O)(=O)c2cc3cc(ccc3oc2=O)[N+](=O)[O-])Br BS-7747 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Br)/C(=O)OC BS-7748 COc1ccc(cc1)c2nc(on2)c3nc(no3)c4cc(c(c(c4)OC)OC)OC BS-7749 COc1cc(cc(c1)OC)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7752 COc1cccc(c1OC)C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7753 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)C(=O)OC)CCCC3 BS-7754 COc1ccc2c(c1)cc(/c(=N/NC(=O)c3ccccc3)/o2)c4[nH]c5ccccc5n4 BS-7755 CCOc1ccc(cc1)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5ccccc5 BS-7763 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4ccc(cc4)F BS-7764 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)F)OC BS-7765 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccccc4F BS-7766 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)F BS-7767 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)F BS-7768 c1ccc(cc1)OCC(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-7769 COc1cccc(c1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-7771 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccc(cc4)Cl BS-7782 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)Cl BS-7784 c1cc(cc(c1)Br)CN2Cc3cc(ccc3OCC2=O)Br BS-7785 Cc1ccc(c(c1)S(=O)(=O)/C(=N/Nc2ccc(cc2)C(=O)n3ccnc3)/C#N)F BS-7789 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)OC)CCCC3 BS-7790 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4OC)CCCC3 BS-7791 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)OC)CCCC3 BS-7792 CC(C)(C)OC(=O)N1CCC(CC1)Cc2nc(no2)c3ccc(cc3)C(F)(F)F BS-7793 c1cc(c(cc1F)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCCCC3)F BS-7794 COc1ccc(cc1)CC(c2[nH]c3ccccc3n2)c4ncc(s4)c5ccccc5 BS-7806 CCCCn1cc(c(=O)c2c1cc(c(c2)F)F)S(=O)(=O)c3cccc(c3)Cl BS-7808 COc1ccc(cc1OC)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)Cl BS-7809 c1cc(cc(c1)Cl)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7810 c1ccc(c(c1)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3)Cl BS-7811 COc1cc(ccc1C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4)Cl BS-7812 COc1ccc(cc1C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4)Cl BS-7813 COc1cccc(c1)c2nc(on2)CC3CCN(CC3)C(=O)c4cccc(c4)Cl BS-7814 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)COc3ccc(cc3)F)C(F)(F)F BS-7816 Cc1ccc(cc1F)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-7820 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4c(cccc4F)F BS-7823 CCOC(=O)c1cccc(c1)NC(=O)C2CC(=O)N(C2)c3ccc(c(c3)OC)OC BS-7824 CCOC(=O)c1ccc(cc1)NC(=O)C2CC(=O)N(C2)c3ccc(c(c3)OC)OC BS-7825 CCc1ccc(cc1)NS(=O)(=O)c2c(c(n[nH]2)C)C(=O)NCc3ccc(cc3)C BS-7830 Cc1ccsc1C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-7832 COc1cccc(c1)CNC(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4 BS-7833 c1cc(ccc1c2csc3c2nc([nH]c3=O)N4CCN(CC4)C5CCCCC5)F BS-7834 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)Cc3ccc(cc3)Cl)C(F)(F)F BS-7836 CC(C)(C)OC(=O)/C(=N\Nc1ccc(cc1)Cl)/S(=O)(=O)c2ccccc2F BS-7837 c1cc(c(cc1F)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3)F BS-7840 c1cc(c(cc1F)F)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3 BS-7841 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)F)CCCCC3 BS-7842 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4F)CCCCC3 BS-7843 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)F)CCCCC3 BS-7844 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)F)CCCC3 BS-7845 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)F)CCCC3 BS-7847 Cc1ccc(cc1F)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-7848 COc1cccc(c1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc(c(c4)F)F BS-7849 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4cc(ccc4F)F BS-7850 Cc1c(c(on1)C)CC(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-7853 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2c3n(nn2)CC(OC3)c4ccccc4 BS-7854 CCOc1ccc(cc1OCC)CC(=O)NC2(CCCCC2)c3nc(no3)C4CC4 BS-7856 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4ccc(cc4Cl)F BS-7860 COc1ccc(cc1)c2nc(on2)C3CCCN3C(=O)c4cc(ccc4OC)Cl BS-7865 c1ccc(c(c1)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F)Cl BS-7866 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(c(c4)Cl)OC BS-7867 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CCCOc4ccc(cc4)F)CCCC3 BS-7871 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)C)CS(=O)(=O)c3ccccc3 BS-7875 CCOc1ccc(cc1)NC(=O)c2cn[nH]c2S(=O)(=O)N(C)c3ccc(cc3)C BS-7876 CC(C)c1ccc(cc1)NC(=O)C2CCCN(C2)c3c4c(c5ccccc5o4)ncn3 BS-7878 COc1ccc(cc1Cl)NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F BS-7882 COc1ccc(cc1C(=O)NC2CCN(CC2)c3cc(ncn3)C(F)(F)F)Cl BS-7883 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)c4ccc(cc4)Cl)CCCC3 BS-7884 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(ccc4F)Cl BS-7900 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4Cl)F BS-7901 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)Cl)F BS-7902 c1ccc2c(c1)cc(c(=N)o2)Sc3nc4ccccc4c(=O)n3c5ccc(cc5)F BS-7908 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4cccs4)CCCCC3 BS-7910 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4cccs4)CCCC3 BS-7911 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NC4CCCCC4)CCCCC3 BS-7913 Cc1c(nnn1c2cc(ccc2OC)OC)S(=O)(=O)c3ccc(cc3)C(C)(C)C BS-7914 CCc1ccc(cc1)N2CC(CC2=O)C(=O)N3CCC(CC3)NC(=O)OC(C)(C)C BS-7916 Cc1ccc(cc1)CN(c2ccsc2C(=O)OC)S(=O)(=O)c3ccc(cc3)C BS-7917 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCC(CC4)Cc5ccccc5 BS-7918 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)Cl)CCCC3 BS-7920 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C(F)(F)F BS-7922 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)C(F)(F)F BS-7923 COc1ccc(cc1)c2nc(on2)c3cc4n(n3)CCCC4OC(=O)c5ccccc5 BS-7925 CCOc1ccc(cc1)NC(=O)C2CCCN(C2)c3c4c(c5ccccc5o4)ncn3 BS-7931 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4c5ccccc5n(n4)C BS-7932 CCc1ccc(cc1)NCc2cc3ccc(cc3n(c2=O)Cc4ccc(cc4)F)OC BS-7933 Cc1cc(nc(n1)N2CCc3ccccc3C2)OCC(=O)Nc4ccc(cc4)C(C)C BS-7934 COc1ccc(cc1)N2CCN(CC2)c3c(cccn3)S(=O)(=O)N4CCCCC4 BS-7936 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)Cc5ccccc5 BS-7937 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(o4)Br BS-7942 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)Cl)Cl BS-7943 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4F)F)CCCC3 BS-7944 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4F)F)CCCC3 BS-7945 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4cccc(c4)C(F)(F)F BS-7947 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCCO3)/C(=O)OC BS-7949 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCO3)/C(=O)OC BS-7950 COc1ccc(cc1)C2(CC2)C(=O)N3CCC(CC3)Cc4nc(no4)c5ccccc5 BS-7951 CCOc1ccc(cc1)N/C=C(/C(=O)OC)\S(=O)(=O)c2ccc(cc2)C(C)(C)C BS-7953 CCCCc1ccc(cc1)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7957 Cc1cc(c(c(c1)C)S(=O)(=O)N(C)c2ccsc2C(=O)n3c(cc(n3)C)C)C BS-7958 CCCc1ccc(cc1)S(=O)(=O)N(C)c2ccsc2C(=O)n3c(cc(n3)C)C BS-7959 Cc1cc(n(n1)C(=O)c2c(ccs2)N(C)S(=O)(=O)c3ccc(cc3)C(C)C)C BS-7960 Cc1cc(n(n1)C(=O)c2c(ccs2)S(=O)(=O)N(C)c3ccc(cc3)C(C)C)C BS-7961 c1cc(ccc1c2nc(on2)CC3CCN(CC3)C(=O)c4cc(ccc4Cl)F)F BS-7962 c1cc(ccc1c2nc(on2)CC3CCN(CC3)C(=O)c4ccc(cc4Cl)F)F BS-7964 COc1cc(ccc1C(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4)Cl BS-7965 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(c(c4)Cl)Cl BS-7966 COc1ccc(cc1OC)c2nc(on2)C3CCCN3C(=O)c4cc5ccccc5[nH]4 BS-7968 CC(=O)Nc1ccc(cc1)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-7969 CCCC/N=c\1/c(cc2ccccc2o1)C(=O)Nc3nnc(s3)c4cccc(c4)C BS-7974 COc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5 BS-7975 Cc1cc(n(n1)C(=O)N2CCN(CC2)c3c(cccn3)S(=O)(=O)N4CCCC4)C BS-7976 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C(C)(C)C BS-7977 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)N4CCN(CC4)c5ccccc5 BS-7978 COc1ccc(cc1NC(=O)c2c(n(nn2)CC(=O)Nc3ccccc3F)N)Cl BS-7981 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(cc4)OC(F)(F)F BS-7982 CCOc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc3c(c2)OCCO3)/C(=O)OC BS-7984 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)NC(=O)C BS-7990 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)OC)OC)/C(=O)OC BS-7991 CCCCOc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-8007 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)CCCc4ccccc4 BS-8009 CCN(c1ccsc1C(=O)n2c(cc(n2)C)C)S(=O)(=O)c3ccc(cc3)OC BS-8010 CCOc1ccc(cc1OCC)CN2Cc3cc(ccc3OCC2=O)Br BS-8011 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)C(F)(F)F)CCCC3 BS-8012 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)C(F)(F)F)CCCC3 BS-8014 COc1ccc(c(c1)OC)/N=c\2/c(cc3ccc(cc3o2)O)C(=O)NCc4ccco4 BS-8015 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)C#N)CCCC3 BS-8016 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cc(=O)n5ccccc5n4)CCCC3 BS-8017 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc5c(c4)OCO5 BS-8019 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3ccc(cc3)C(C)(C)C)C(F)(F)F BS-8020 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)F BS-8024 Cc1ccccc1c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5F BS-8025 Cc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccc(cc5)F BS-8027 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)CCc4cccc(c4)OC BS-8029 CCc1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-8033 Cc1cc(cc(c1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC)C BS-8034 Cc1ccc(cc1C)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-8035 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccccc4OC BS-8036 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4cccc(c4)C BS-8037 CN(C)c1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4cccc(c4)OC BS-8038 c1ccn2c(c1)nc(cc2=O)Cn3cnc4c(csc4c3=O)c5cccc(c5)Cl BS-8045 CC(C)(C)c1ccc(cc1)S(=O)(=O)c2cc3cc(ccc3oc2=O)Br BS-8047 COc1cccc(c1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc5c(c4)OCO5 BS-8049 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc5c(c4)OCO5 BS-8050 CCOc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)OC)OC)/C(=O)OC BS-8051 Cc1ccc(c(c1)NC(=O)Cn2cc(ccc2=O)S(=O)(=O)N3CCOCC3)OC BS-8052 Cc1ccc(cc1)COC(=O)C2=NN(c3c(cccn3)S2(=O)=O)c4ccc(cc4)C BS-8053 COc1ccc(cc1OC)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-8057 COc1ccc(cc1OC)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-8061 CCOc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4cccc(c4)OC BS-8062 Cc1ccc(cc1)OCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8063 CCOc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8064 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)Cc4ccccc4OC BS-8065 Cc1cccc(c1)OCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8066 CCCCOc1ccc(cc1)C(=O)N2CCCC2c3nc(no3)c4ccc(cc4)OC BS-8067 CCOc1ccccc1C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8068 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8069 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)OC(F)(F)F)CCCC3 BS-8079 c1cc2c(cc1NC(=O)NC3(CCCCC3)c4nc(no4)c5cnccn5)OCCO2 BS-8083 CCOc1cccc(c1)CNC(=O)C2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-8084 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)CCc3ccc(cc3)OC)C(F)(F)F BS-8085 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)CCc3ccccc3OC)C(F)(F)F BS-8087 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(cc(c4)OC)OC BS-8091 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4ccccc4 BS-8092 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)OC BS-8093 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)N4CCN(CC4)c5ccccc5F BS-8097 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)N4CCN(CC4)c5ccc(cc5)F BS-8098 c1cc(c(nc1)N2CCCCC2)S(=O)(=O)N3CCC(CC3)C(=O)N4CCOCC4 BS-8099 c1cc2c(cc1Cl)cc([nH]2)C(=O)NC3(CCCCC3)c4nc(no4)c5cnccn5 BS-8103 Cc1cc(nc(n1)N2CCc3ccccc3C2)OCC(=O)Nc4cccc(c4C)Cl BS-8106 c1ccc(cc1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)Cl BS-8109 c1ccc(cc1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccccc5Cl BS-8110 CCOc1ccc(cc1)C(=O)Cn2c(=O)c(nn(c2=O)c3ccc(cc3)C)C(=O)OC BS-8113 Cc1cccc(c1)OCC(=O)N2CCCC2c3nc(no3)c4ccc(c(c4)OC)OC BS-8126 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)C)CCCCC3 BS-8127 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4C)CCCCC3 BS-8128 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)C)CCCCC3 BS-8129 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccccc4)CCCCC3 BS-8130 Cc1ccc(c(c1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C)C BS-8131 Cc1cc(cc(c1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C)C BS-8132 CCc1cccc(c1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8133 Cc1ccc(c(c1)C)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8134 Cc1ccc(cc1)CNC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8135 CCc1ccccc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8136 Cc1ccc(cc1C)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8137 CCc1ccc(cc1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8138 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4C)C)CCCC3 BS-8139 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4c(cccc4C)C)CCCC3 BS-8140 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)C)CCCC3 BS-8141 CCc1ccccc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)CC BS-8142 CCc1ccc(cc1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)CC BS-8143 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCCCc4ccccc4)CCCC3 BS-8144 Cc1cc(c(c(c1)C)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C)C BS-8145 COc1ccccc1CCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8147 COc1ccc(cc1)CCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8148 c1ccnc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl BS-8159 c1ccnc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)Cl BS-8160 Cc1ccc(cc1Cl)S(=O)(=O)N(C)c2ccsc2C(=O)n3c(cc(n3)C)C BS-8161 CCN(c1ccsc1C(=O)n2c(cc(n2)C)C)S(=O)(=O)c3ccc(cc3)Cl BS-8162 COc1cc(cc(c1OC)OC)c2nc(on2)c3nc(no3)c4ccc5c(c4)OCO5 BS-8163 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3ccc(cc3OC)OC)C(F)(F)F BS-8167 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3cc(cc(c3)OC)OC)C(F)(F)F BS-8168 COc1ccc(cc1Cn2cnc3c(csc3c2=O)c4cccc(c4)F)C(=O)OC BS-8169 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)F)F BS-8175 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)F)F BS-8176 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5F)F BS-8177 Cc1cccc(c1)OCC(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-8178 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)F)OC BS-8179 COc1cccc(c1)NC(=O)CSc2nc(cs2)c3cc4ccccc4oc3=O BS-8183 COc1ccc2c(c1)sc3n2c(=O)c(cn3)S(=O)(=O)c4ccc(c(c4)Cl)F BS-8187 COc1ccc(cc1OC)S(=O)(=O)c2cc3cc(ccc3oc2=O)Br BS-8188 CC(C)(C)OC(=O)N1CCC(CC1)N2Cc3cc(ccc3OCC2=O)Br BS-8189 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4OC)CCCCC3 BS-8191 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)OC)CCCCC3 BS-8192 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4OC)CCCC3 BS-8193 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)OC)CCCC3 BS-8194 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)OC)CCCC3 BS-8195 CCOc1ccccc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-8196 CCOc1ccc(cc1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-8197 Cc1cccc(c1)S(=O)(=O)c2cn(c3cc(c(cc3c2=O)F)F)Cc4ccccc4 BS-8198 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc(c(c4)F)OC BS-8199 COc1ccc(c(c1)OC)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8200 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)F BS-8202 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccccc4F BS-8204 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4ccco4 BS-8212 COc1ccc(cc1Cl)NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-8216 COc1ccc(cc1Cl)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-8217 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)Cc4ccccc4Cl BS-8218 COc1ccc(cc1OC)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5ccccc5 BS-8222 c1cc(ccc1n2c(=O)c3ccc(cc3nc2S)C(=O)N4CCC(CC4)C(=O)N)F BS-8225 c1cc2c(cc1NC(=O)NC3(CCCCC3)c4nc(no4)c5ccsc5)OCCO2 BS-8227 Cc1cccc(c1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc(cc5)SC BS-8230 Cc1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc(cc5)SC BS-8231 Cc1cc(nc(n1)N2CCc3ccccc3C2)OCC(=O)Nc4ccc(cc4Cl)F BS-8234 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(ccc4OC)Cl BS-8235 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4ccc(cc4)Cl BS-8236 Cc1cc(ccc1OCC(=O)N2CCC(CC2)c3n[nH]c(=O)n3c4ccccc4)Cl BS-8237 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccccc4Cl BS-8238 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)Cl BS-8239 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)Br BS-8242 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccccc4Br BS-8243 CCOC(=O)/C(=C\Nc1ccc(c(c1)OC)OC)/S(=O)(=O)c2ccc(cc2F)F BS-8246 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4F)CCCCC3 BS-8249 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)F)CCCCC3 BS-8250 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)F)CCCCC3 BS-8251 Cc1ccc(cc1F)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8252 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)F)CCCC3 BS-8253 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(c(c4)F)C)CCCC3 BS-8254 COc1ccc(cc1)/N=c\2/c(cc3c4ccccc4ccc3o2)C(=O)Nc5nccs5 BS-8255 Cc1cc(ccc1Br)NC(=O)c2ccc3c(c2)N(C4CCCCN4C3=O)C BS-8267 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(cc4)Br BS-8269 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(ccc4F)F BS-8271 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)F)F BS-8273 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4c(cccc4F)F BS-8274 COc1ccc(cc1F)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-8275 Cc1cc(n(n1)C(=O)c2cn(cn2)c3ccc(cn3)S(=O)(=O)N4CCCC(C4)C)C BS-8279 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3cc(ccc3OC)Cl)C(F)(F)F BS-8281 Cc1nc(cc(n1)N2CCC(CC2)NC(=O)c3ccc(cc3OC)Cl)C(F)(F)F BS-8282 c1cc(ccc1CC(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F)Cl BS-8287 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(ccc4F)Cl BS-8289 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)Cl)F BS-8290 c1cc(c(cc1S(=O)(=O)c2cnc3n(c2=O)c4ccc(cc4s3)Cl)Cl)F BS-8291 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4cccs4)CCCCC3 BS-8294 Cc1ccc(cc1)NC(=O)Cn2c(=O)n3cccc(c3n2)S(=O)(=O)N4CCCCC4 BS-8295 Cc1cccc(c1)c2csc(c2n3cccc3)c4nc(no4)c5ccc(cc5)SC BS-8303 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)Cl)CCCCC3 BS-8304 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)Cl)CCCCC3 BS-8305 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4Cl)CCCCC3 BS-8306 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)Cl)CCCC3 BS-8307 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4Cl)CCCC3 BS-8308 Cc1c(cccc1Cl)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-8309 Cc1ccc(c(c1)Cl)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-8310 Cc1ccc(cc1Cl)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)C BS-8311 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccccc4Cl)CCCC3 BS-8312 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4cc(ccc4Cl)F BS-8313 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc(cc4Cl)F BS-8314 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C(F)(F)F BS-8316 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)C(F)(F)F BS-8317 Cc1cc(n(n1)C(=O)c2c(ccs2)S(=O)(=O)N3CCN(CC3)c4ccccc4)C BS-8325 CCc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4cccc(c4)Br)CCCC3 BS-8331 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4F)F)CCCC3 BS-8332 COc1ccc(cc1OC)c2nc(on2)Cn3cnc4c(c3=O)nnn4c5ccccc5 BS-8333 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cccc(c4)OC(F)(F)F BS-8344 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)OC(F)(F)F BS-8345 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccccc4OC(F)(F)F BS-8346 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4)C#N BS-8348 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)OC BS-8350 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)NC4CCN(CC4)Cc5ccccc5 BS-8353 COc1ccc(cc1Cl)NC(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4 BS-8354 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(cc4)OC(F)(F)F BS-8356 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(cc4)OC(F)(F)F BS-8357 CCOC(=O)c1ccccc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-8362 CCc1ccc(cc1)N(C)S(=O)(=O)c2c(csc2C(=O)OC)c3cccc(c3)F BS-8363 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)OC)OC)/C(=O)OC BS-8364 Cc1cc(n(n1)C(=O)C2CCN(CC2)c3c(cccn3)S(=O)(=O)N4CCOCC4)C BS-8368 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4cccc(c4)OC BS-8369 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8370 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(c(c4)Cl)F)CCCC3 BS-8371 Cc1ccc(cc1)c2nc(on2)Cn3cnc4c(c3=O)nnn4Cc5cccc(c5)Cl BS-8372 CCC(=O)Nc1c(nsc1C(=O)NCc2ccc(cc2)C(F)(F)F)c3ccccn3 BS-8375 CN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)N4CCN(CC4)c5ccc(cc5)OC BS-8378 c1ccc2c(c1)c3c(o2)c(ncn3)N4CCCC(C4)C(=O)NCCc5ccc(cc5)Cl BS-8380 c1ccc2c(c1)c3c(o2)c(ncn3)N4CCC(CC4)C(=O)NCCc5ccc(cc5)Cl BS-8381 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4cccc(c4)C(=O)OC BS-8384 CCOc1ccccc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccc(cc4)OC BS-8388 COc1cccc(c1OC)CNC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4 BS-8394 CCOc1ccc(cc1)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8396 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)CCc4cccc(c4)OC BS-8397 COc1ccc(cc1)CCC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8398 CC(C)(C)c1ccc(cc1)C(=O)N2CCCC2c3nc(no3)c4ccc(c(c4)OC)OC BS-8399 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccccc4C BS-8408 Cc1cccc(c1NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4)C BS-8412 Cc1ccc(c(c1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4)C BS-8413 Cc1ccc(c(c1)C)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-8414 Cc1ccc(cc1)CNC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-8416 Cc1c(nnn1c2ccc(cc2)Br)C(=O)Nc3ccc(cc3)Br BS-8420 Cc1nc(no1)c2c3n(c(=O)n(c2=O)Cc4ccc(cc4)OC(F)(F)F)CCCCC3 BS-8421 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc5c(c4)OCO5 BS-8422 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4cccc(c4)OC BS-8425 CCOc1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-8426 Cc1cccc(c1)OCC(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-8429 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-8430 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)N4CCN(CC4)c5ccc(cc5)F BS-8431 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)N4CCN(CC4)c5ccc(cc5)F BS-8432 c1ccc(cc1)N2CC(CC2=O)C(=O)NC3(CCCCC3)c4nc(no4)c5ccsc5 BS-8435 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl BS-8439 c1ccc(cc1)CN2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl BS-8440 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)Cl BS-8441 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccccc5Cl BS-8442 Cc1ccccc1c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5Cl BS-8443 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cccc(c5)Cl BS-8444 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5Cl BS-8445 Cc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cccc(c5)Cl BS-8446 Cc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5Cl BS-8447 COc1cc(cc(c1OC)OC)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-8450 COc1cccc(c1)c2nc(on2)CC3CCN(CC3)C(=O)c4cc(cc(c4)OC)OC BS-8451 COc1ccc(cc1)CCC(=O)N2CCCC2c3nc(no3)c4ccc(c(c4)OC)OC BS-8454 CCOc1ccc(cc1OCC)C(=O)N2CCCC2c3nc(no3)c4ccc(cc4)OC BS-8455 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4C)C)CCCCC3 BS-8456 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4c(cccc4C)C)CCCCC3 BS-8457 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4C)C)CCCCC3 BS-8458 CCc1ccccc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)CC BS-8459 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)C(C)C)CCCCC3 BS-8460 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCCCc4ccccc4)CCCC3 BS-8461 CCc1cccc(c1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCC3)c4nc(on4)CC)C BS-8462 CCCCOc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8464 CCc1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)C3CC(=O)N(C3)c4ccc(cc4)F BS-8465 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4)OC BS-8467 c1cc(c(cc1S(=O)(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4)Cl)F BS-8469 CCOc1ccc(cc1)NC(=O)Cn2c(=O)c(nn(c2=O)c3ccc(cc3)C)C(=O)OC BS-8470 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)c4ccc(nc4OC)OC BS-8473 CCOc1ccc(cc1)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5ccc(c(c5)C)C BS-8474 Cc1cccc(c1)c2nnc(s2)NC(=O)c\3cc4ccccc4o/c3=N\c5ccccc5 BS-8475 CCOc1ccc2c(c1)sc3n2c(=O)c(cn3)S(=O)(=O)c4ccc(c(c4)Cl)F BS-8478 Cc1cc(nc(n1)N2CCc3ccccc3C2)OCC(=O)Nc4ccc(c(c4)Cl)OC BS-8483 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc5c(c4)OCO5)CCCCC3 BS-8486 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc5c(c4)OCO5)CCCC3 BS-8487 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)OC)CCCCC3 BS-8494 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4OC)CCCCC3 BS-8495 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)OC)CCCCC3 BS-8496 Cc1ccc(c(c1)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C)OC BS-8497 CCOc1ccccc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8498 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4OC)C)CCCC3 BS-8499 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4cccc(c4)OC)CCCC3 BS-8500 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)OC)CCCC3 BS-8501 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4OCC)CCCC3 BS-8502 Cc1ccc(cc1C)S(=O)(=O)c2cn(c3cc(c(cc3c2=O)F)F)Cc4ccccc4 BS-8503 Cc1cccc(c1)Cn2cc(c(=O)c3c2cc(c(c3)F)F)S(=O)(=O)c4cccc(c4)C BS-8504 Cc1ccc(cc1)Cn2cc(c(=O)c3c2cc(c(c3)F)F)S(=O)(=O)c4cccc(c4)C BS-8505 COc1ccc(cc1OC)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8506 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4cc(c(c(c4)OC)OC)OC BS-8508 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4ccc(cc4)F BS-8517 c1c2cc(c(=N)oc2c(cc1I)I)C(=O)N BS-8535 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4ccc(cc4)Br BS-8536 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4cccc(c4)Br BS-8537 COc1ccc(cc1OC)c2nc(on2)c3nc(no3)c4cc(c(c(c4)OC)OC)OC BS-8538 Cc1cccc(c1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cc(cc(c5)OC)OC BS-8542 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)F)OC BS-8547 COc1cc(cc(c1)OC)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-8548 COc1ccc(cc1Cn2cnc3c(csc3c2=O)c4ccc(cc4)Cl)C(=O)OC BS-8554 COc1ccc(cc1Cn2cnc3c(csc3c2=O)c4cccc(c4)Cl)C(=O)OC BS-8555 c1cc(oc1)C(=O)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl BS-8556 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl)F BS-8557 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)Cl)F BS-8558 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccc(cc5)F)Cl BS-8559 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5F)Cl BS-8560 c1cc(cc(c1)F)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cccc(c5)Cl BS-8561 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)F)Cl BS-8562 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4ccc(cc4C)Cl BS-8563 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccc(c(c4)Cl)OC BS-8564 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccccc4Cl BS-8565 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccc(cc4)Br BS-8570 c1ccc(c(c1)CC(=O)NC2(CCCCC2)c3nc(no3)c4ccncc4)Br BS-8572 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(c(c4)OC)OC)CCCC3 BS-8573 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4OC)OC)CCCC3 BS-8574 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4OC)OC)CCCC3 BS-8575 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)F)CCCCC3 BS-8576 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(c(c4)F)C)CCCCC3 BS-8577 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)SC)CCCCC3 BS-8579 CN1c2cc(ccc2C(=O)N3C1CCCCC3)C(=O)Nc4ccc(cc4)Oc5ccccc5 BS-8580 CC1CCCN(C1)c2c3cc(ccc3n4c(n2)c(nn4)S(=O)(=O)c5ccccc5)Cl BS-8587 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)Cl BS-8588 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4)Cl BS-8589 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccccc4Cl BS-8590 c1ccc(c(c1)CC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4)Br BS-8593 c1ccc(c(c1)NC(=O)NC2(CCCCC2)c3nc(no3)c4cccnc4)Br BS-8594 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)Nc4ccc(c(c4)C)Br BS-8595 Cc1cc(ccc1Br)NC(=O)c2ccc3c(c2)N(C4CCCCCN4C3=O)C BS-8596 c1ccc(cc1)Oc2ccc(cc2)NC(=O)C3CCN(CC3)c4cc(ncn4)C(F)(F)F BS-8597 CC(C)(C)OC(=O)N1CCN(CC1)c2cc(nc(n2)c3cccc(c3)Cl)C(F)(F)F BS-8605 Cc1cc(ccc1NC(=O)C2CCN(CC2)c3cc(ncn3)C(F)(F)F)Br BS-8606 c1ccc(c(c1)NC(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4)Br BS-8607 Cc1cccc(c1)S(=O)(=O)c2cn(c3cc(c(cc3c2=O)F)F)Cc4ccc(cc4)F BS-8608 CCOC(=O)N1CCC(CC1)NC(=O)C2CCN(CC2)c3cc(nc(n3)C)C(F)(F)F BS-8610 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4F)F BS-8612 COc1cc(cc(c1OC)OC)C(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4 BS-8614 Cc1ccc(c(c1)C)S(=O)(=O)c2c3nc(c4ccccc4n3nn2)NCc5ccccc5 BS-8617 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4)Cl)CCCCC3 BS-8620 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)Cl)CCCCC3 BS-8621 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4Cl)CCCCC3 BS-8622 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)Cl)CCCCC3 BS-8623 Cc1c(cccc1Cl)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8624 Cc1ccc(c(c1)Cl)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8625 Cc1ccc(cc1NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C)Cl BS-8626 Cc1ccc(cc1Cl)NC(=O)Cn2c(=O)c(c3n(c2=O)CCCCC3)c4nc(on4)C BS-8627 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccc(cc4)Cl)CCCC3 BS-8628 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4C)Cl)CCCC3 BS-8629 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4Cl)C)CCCC3 BS-8630 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)NCc4ccccc4Cl)CCCC3 BS-8631 c1ccc(cc1)S(=O)(=O)c2cc3cc(cc(c3oc2=O)Br)Br BS-8632 Cc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C(F)(F)F BS-8633 c1ccc(cc1)C(=O)N/N=c\2/c(cc3c4ccccc4ccc3o2)C5=NCc6ccccc6N5 BS-8635 CCCOc1ccc(cc1)CNC(=O)C2CCCN(C2)c3c4c(c5ccccc5o4)ncn3 BS-8638 c1ccc2c(c1)c(nn(c2=O)c3cccc(c3)Cl)c4nc(no4)c5ccc6c(c5)OCO6 BS-8643 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(ccc4F)Cl BS-8646 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4Cl)F BS-8647 COc1ccc(cc1)Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(c(c4)Cl)F BS-8648 c1cc(ccc1Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)COc4ccc(cc4)Cl)F BS-8649 COc1cc(ccc1C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F)Cl BS-8650 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccccc5Br BS-8652 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)Br BS-8653 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4F)F)CCCCC3 BS-8655 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4F)F)CCCCC3 BS-8656 Cc1ccc(c(c1)Nc2c3ccccc3n4c(n2)c(nn4)S(=O)(=O)c5ccccc5)OC BS-8663 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cc(ccc4OC)Cl)CCCC3 BS-8671 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(c(c4)Cl)OC)CCCC3 BS-8672 c1ccc(cc1)Cn2cc(c(=O)c3c2cc(c(c3)F)F)S(=O)(=O)c4cccc(c4)Cl BS-8673 COc1ccccc1/N=c\2/c(cc3cc(ccc3o2)Br)c4[nH]c5ccccc5n4 BS-8683 c1ccc(c(c1)CC(=O)NC2(CCCCC2)c3nc(no3)c4ccsc4)Br BS-8684 c1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)Cc4ccc(cc4)OC(F)(F)F BS-8687 Cc1ccc(cc1)n2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4cc(n[nH]4)c5ccc(cc5)F BS-8688 CN(c1ccc(cc1)OC)S(=O)(=O)c2ccsc2C(=O)Nc3ccc(cc3)C(=O)O BS-8691 Cc1cc(n(n1)C(=O)c2cn(nc2S(=O)(=O)N3CCN(CC3)c4ccccc4F)C)C BS-8692 COc1ccc(c(c1)CNC(=O)C2CCCN(C2)c3c4c(c5ccccc5o4)ncn3)OC BS-8693 Cc1cccc(c1)N2CCN(CC2C)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)OC BS-8700 Cc1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)OC)C BS-8701 CSc1ccc(cc1)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5cccc(c5)Cl BS-8702 Cc1ccc(cc1C)S(=O)(=O)c2c3nc(c4ccccc4n3nn2)Nc5ccc(cc5)F BS-8705 c1ccc(cc1)CN2CCC(CC2)NC(=O)C3CCN(CC3)c4cc(ncn4)C(F)(F)F BS-8706 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)C4(CC4)c5ccc(cc5)OC BS-8710 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)N4CCCc5c4cccc5 BS-8714 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(c(c4)Cl)F)CCCCC3 BS-8717 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4F)Cl)CCCCC3 BS-8718 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(c(c4)Cl)F)CCCC3 BS-8719 CCc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccc(cc4F)Cl)CCCC3 BS-8720 c1cc(ccc1Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(cc4)C(F)(F)F)F BS-8725 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)F BS-8726 CCOC(=O)c1ccc(cc1)n2c3ccccc3c(=O)c(n2)S(=O)(=O)c4ccc(cc4)C BS-8729 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)N4CCN(CC4)c5ccc(cc5)F BS-8731 Cc1cc(n(n1)C(=O)c2c(ccs2)S(=O)(=O)N3CCN(CC3)c4ccc(cc4)F)C BS-8733 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)OC BS-8734 CCCCOc1ccc(cc1)C(=O)N2CCC(CC2)c3n[nH]c(=O)n3Cc4ccc(cc4)C BS-8735 CCN1c2cc(ccc2C(=O)N3C1CCCC3)C(=O)N4CCN(CC4)c5ccc(cc5)OC BS-8736 c1cc(ccc1Cn2c(n[nH]c2=O)C3CCN(CC3)C(=O)c4ccc(o4)Br)F BS-8737 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4ccccc4C(F)(F)F)CCCC3 BS-8738 Cc1nc(no1)c2c3n(c(=O)n(c2=O)CC(=O)Nc4cccc(c4)C(F)(F)F)CCCC3 BS-8739 CCOc1ccc(cc1OCC)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccccc4 BS-8745 CCCCOc1ccc(cc1)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-8746 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4cc(cc(c4)C)C BS-8757 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(cc4C)C BS-8759 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)NCCc4ccccc4 BS-8761 Cc1ccc(cc1)CNC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccc(cc4)C BS-8762 CCc1cccc(c1)NC(=O)CSc2nc3c(csc3c(=O)n2CC)c4ccccc4 BS-8764 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(cc(c4)C)C BS-8765 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4c(cccc4C)C BS-8767 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(ccc4C)C BS-8768 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4C)C BS-8770 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4ccc(cc4)C BS-8771 CCc1cccc(c1NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4)C BS-8773 Cc1cc(c(c(c1)C)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4)C BS-8774 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCCCc4ccccc4 BS-8775 COc1ccc(cc1)c2nc(on2)Cn3cnc4c(c3=O)nnn4Cc5cccc(c5)Cl BS-8776 CC(C)(C)OC(=O)C1=NN(c2ccccc2S1(=O)=O)CC(=O)Nc3ccc(cc3)Cl BS-8777 COc1ccc(cc1S(=O)(=O)NC2(CCCCC2)c3nc(no3)c4cnccn4)Cl BS-8778 CCOC(=O)c1c(n(nn1)c2ccc(cc2)C)c3cc[n+](cc3)C.[I-] BS-8782 Cc1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl)C BS-8788 Cc1cccc(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cc(ccc5C)Cl BS-8790 Cc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cc(ccc5C)Cl BS-8791 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)Cc4ccc(c(c4)OC)OC BS-8797 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc5c(c4)OCO5 BS-8798 Cc1cc(n(n1)C(=O)c2c(c(cs2)c3ccccc3)S(=O)(=O)N(C)c4ccccc4)C BS-8803 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)OC BS-8804 Cc1ccc(c(c1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4)OC BS-8806 CCOc1ccc(cc1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-8807 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4ccc(cc4)OC BS-8809 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Br)/C(=O)OC BS-8811 CCOC(=O)c1ccc(cc1)N2c3cc(ccc3S(=O)(=O)C(=N2)C(=O)c4ccccc4)F BS-8812 Cc1cccc(c1)c2nnc(s2)NC(=O)c\3cc4ccccc4o/c3=N\Cc5ccccc5 BS-8814 COc1ccccc1N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccccc5Cl BS-8816 COc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cccc(c5)Cl BS-8817 COc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5Cl BS-8818 COC(=O)C1=C2CCCCCN2C(=O)C(C1=O)(Cc3ccc(cc3)F)Cc4ccc(cc4)F BS-8819 CCOc1ccc(cc1OCC)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8822 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4ccc(cc4)Oc5ccccc5 BS-8825 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccccc4F BS-8828 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)NCc4ccc(cc4)F BS-8831 Cc1ccc(cc1)N2CC(CC2=O)C(=O)N3CCC(CC3)C(=O)NCc4cccc(c4)Cl BS-8840 CCc1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)C3CC(=O)N(C3)c4ccc(cc4)Cl BS-8841 CCOc1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc6c(c5)OCO6 BS-8845 c1ccc(c(c1)CNC(=O)C2CCCN(C2)c3c4c(c5ccccc5o4)ncn3)C(F)(F)F BS-8846 CC(C)Oc1ccc(cc1OC)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5ccccc5 BS-8849 Cc1cc([nH]n1)NC(=O)CSc2nc3ccccc3c(=O)n2CCCN4CCC(CC4)C BS-8860 Cc1ccc(cc1N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)F)Cl BS-8861 COc1cc(cc(c1OC)OC)C(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)F BS-8864 c1cc(ccc1NC(=O)CN2CCn3c(c(nn3)c4nc(no4)c5ccsc5)C2=O)Cl BS-8882 Cc1cc(nc(n1)N2CCN(CC2)c3ccccc3)OCC(=O)Nc4ccc(c(c4)Cl)F BS-8883 COc1cc(c(cc1NC(=O)Cn2cnc3c(csc3c2=O)c4ccccc4)Cl)OC BS-8887 COc1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)Cc4ccc(c(c4)Cl)OC BS-8888 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccccc4Cl BS-8892 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4)Cl BS-8894 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccccc4Cl BS-8895 Cc1ccc(c(c1)Cl)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-8896 Cc1ccc(cc1NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4)Cl BS-8897 c1ccc(cc1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-8903 c1cc(cc(c1)Cl)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl BS-8906 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Cl)Cl BS-8907 c1cc(cc(c1)Cl)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cccc(c5)Cl BS-8908 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)Cl)Cl BS-8909 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cccc(c5)Cl)Cl BS-8910 c1ccc(c(c1)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5Cl)Cl BS-8911 CCc1ccc(cc1)C(=O)/C(=C/Nc2ccc(cc2)OC)/S(=O)(=O)c3cc(ccc3F)F BS-8912 COc1ccc2c(c1)cc(/c(=N/c3ccc(cc3)c4ccccc4)/o2)C5=NCc6ccccc6N5 BS-8917 CCN(CCCNC(=O)C1CCCN(C1)c2c3c(c4ccccc4o3)ncn2)c5ccccc5 BS-8929 Cc1ccc(cc1)S(=O)(=O)c2cc3cc(cc(c3oc2=O)Br)Br BS-8934 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4ccc(cc4F)Br BS-8937 c1ccnc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(c(c5)Cl)Cl BS-8938 c1ccc(cc1)c2nc(on2)CC3CCN(CC3)C(=O)C4CCN(CC4)C(=O)c5ccccc5 BS-8941 Cc1cccc(c1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)Br BS-8952 Cc1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc(cc5)Br BS-8955 c1ccc(cc1)S(=O)(=O)c2c3nc(c4ccccc4n3nn2)Nc5ccc6c(c5)OCCO6 BS-8959 c1ccc2c(c1)c3c(o2)c(ncn3)N4CCC(CC4)C(=O)N5CCN(CC5)c6ccccc6F BS-8963 Cc1ccc(cc1)N(CC(=O)OC)S(=O)(=O)c2c(csc2C(=O)OC)c3ccccc3 BS-8972 Cc1ccc(cc1)c2csc3c2nc([nH]c3=O)N4CCCC(C4)C(=O)NCc5ccccn5 BS-8978 Cc1ccc(cc1)Cn2cc(c(=O)c3c2cc(c(c3)F)F)S(=O)(=O)c4cccc(c4)Cl BS-8979 Cc1cccc(c1)Cn2cc(c(=O)c3c2cc(c(c3)F)F)S(=O)(=O)c4cccc(c4)Cl BS-8980 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4Cl)F BS-8981 Cc1cc(n(n1)C(=O)c2c(ccs2)S(=O)(=O)N3CCN(CC3)c4cccc(c4)OC)C BS-8991 COc1cc(cc(c1)OC)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5cccc(c5)Cl BS-8996 COc1ccc(cc1OC)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5cccc(c5)Cl BS-8998 COc1ccc(cc1)n2c(=O)c3ccc(cc3nc2S)C(=O)NCc4ccc(cc4)C(=O)O BS-8999 COc1ccc(cc1OC)c2nc(on2)Cn3cnc4c(c3=O)nnn4Cc5cccc(c5)F BS-9021 CCc1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)C3CC(=O)N(C3)Cc4ccc(cc4)OC BS-9028 CCc1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)C3CC(=O)N(C3)c4cc(ccc4OC)C BS-9029 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(cc4)C(=O)C BS-9030 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4cccc(c4)C(=O)C BS-9031 Cc1ccc2c(c1)N(CCO2)C(=O)CSc3nc4c(csc4c(=O)n3C)c5ccccc5 BS-9034 CCc1cccc(c1)NC(=O)CSc2nc3c(csc3c(=O)n2CC)c4ccc(cc4)C BS-9036 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4cc(cc(c4)C)C BS-9037 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(c(c4)C)C BS-9038 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)NCc4ccc(cc4)C BS-9043 CCc1cccc(c1NC(=O)CSc2nc3c(csc3c(=O)n2CC)c4ccccc4)C BS-9047 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4c(cc(cc4C)C)C BS-9048 CCCCc1ccc(cc1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-9050 c1cc(cc(c1)F)Cn2cc(c(=O)c3c2cc(c(c3)F)F)S(=O)(=O)c4cccc(c4)Cl BS-9051 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4ccc(c(c4)C(F)(F)F)Cl BS-9052 c1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4cc(ccc4Cl)C(F)(F)F BS-9053 CCc1ccc(cc1)Nc2c3cc(ccc3n4c(n2)c(nn4)S(=O)(=O)c5ccccc5)Cl BS-9055 Cc1ccc(cc1)CNc2c3ccccc3n4c(n2)c(nn4)S(=O)(=O)c5ccc(cc5)Cl BS-9057 Cc1cc(n(n1)C(=O)c2c(ccs2)S(=O)(=O)N3CCN(CC3)c4ccc(cc4)Cl)C BS-9074 Cc1cc(n(n1)C(=O)c2c(ccs2)S(=O)(=O)N3CCN(CC3)c4ccccc4Cl)C BS-9075 Cc1cc(n(n1)C(=O)c2c(ccs2)S(=O)(=O)N3CCN(CC3)c4cccc(c4)Cl)C BS-9076 CC1=NS(=O)(=O)N(C=C1C(=O)O)C.c1cc(ccc1c2nc(on2)CC3CCNCC3)F BS-9080 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)C(=O)OC BS-9083 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc5c(c4)OCCO5 BS-9085 CCOc1ccc(cc1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccc(cc4)C BS-9091 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)NCc4ccc(cc4)OC BS-9092 Cc1ccc(cc1)N(C)S(=O)(=O)c2c(csc2C(=O)n3c(cc(n3)C)C)c4ccccc4 BS-9095 Cc1cccc(c1)N(C)S(=O)(=O)c2c(csc2C(=O)n3c(cc(n3)C)C)c4ccccc4 BS-9096 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(ccc4OC)C BS-9097 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4ccc(cc4)OC BS-9099 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4cccc(c4)OC BS-9100 COc1ccc(c(c1)OC)c2nc(on2)Cn3cnc4c(c3=O)nnn4c5cccc(c5)Cl BS-9104 CSc1ccc(cc1)c2nc(on2)Cn3cnc4c(c3=O)nnn4Cc5ccc(cc5)Cl BS-9107 CCOc1ccc(cc1)NS(=O)(=O)c2cccnc2N3CCN(CC3)c4cc(ccc4C)C BS-9114 Cc1ccc(cc1N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)OC)Cl BS-9117 COc1cccc(c1)c2nc(on2)CC3CCN(CC3)C(=O)c4cc(c(c(c4)OC)OC)OC BS-9120 Cc1ccc(cc1)CNC(=O)c2ccc(cc2)NC(=O)C3CCC(=O)N3Cc4ccc(cc4)C=C BS-9123 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(c(c4)OC)OC BS-9124 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(cc(c4)OC)OC BS-9125 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4OC)OC BS-9126 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4cc(ccc4C)F BS-9127 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(cc4C)F BS-9128 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(c(c4)F)C BS-9129 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)NCc4ccc(cc4)F BS-9130 c1ccnc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Br BS-9137 Cc1cc(n(n1)C(=O)c2c(c(cs2)c3ccccc3)S(=O)(=O)N(C)c4ccc(cc4)F)C BS-9154 Cc1cc(n(n1)C(=O)c2c(c(cs2)c3cccc(c3)F)S(=O)(=O)N(C)c4ccccc4)C BS-9155 c1ccc(cc1)CN2CCC(CC2)NC(=O)C3CCCN(C3)c4c5c(c6ccccc6o5)ncn4 BS-9160 Cc1ccc(cc1)c2csc3c2ncn(c3=O)CC(=O)Nc4cc(c(cc4OC)OC)Cl BS-9169 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(cc4)Cl BS-9170 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4cccc(c4)Cl BS-9171 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccccc4Cl BS-9172 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(cc4Cl)C BS-9173 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)NCc4ccc(cc4)Cl BS-9177 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)NCc4ccccc4Cl BS-9178 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4Cl)C BS-9179 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(ccc4C)Cl BS-9180 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4C)Cl BS-9182 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4ccc(cc4)Cl BS-9183 Cc1cccc(c1)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cc(c(c(c5)OC)OC)OC BS-9189 Cc1ccc(cc1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9191 Cc1cccc(c1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9192 CCn1cc(c(n1)S(=O)(=O)N2CCN(CC2)c3cccc(c3C)C)C(=O)n4c(cc(n4)C)C BS-9194 CCc1ccc(cc1)CNC(=O)C2CCN(CC2)S(=O)(=O)c3cccnc3N4CCCCC4 BS-9195 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(c(c5)Cl)Cl BS-9197 Cc1ccc(cc1N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5cccc(c5)Cl)Cl BS-9198 Cc1ccc(cc1N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccccc5Cl)Cl BS-9199 c1cc2c(c(c1)F)ncc(c2N3CCC(CC3)N4CCCCC4)S(=O)(=O)c5ccc(cc5)F BS-9217 Cc1ccc(cc1C)S(=O)(=O)c2cc3cc(cc(c3oc2=O)Br)Br BS-9223 Cc1ccc(cc1C)n2c(=O)c3ccccc3c(n2)c4nc(no4)c5cccc(c5)Br BS-9236 c1cc(ccc1c2csc3c2nc([nH]c3=O)N4CCN(CC4)C5CCCCC5)Br BS-9239 Cc1ccc(c(c1)C)S(=O)(=O)c2c3nc(c4ccccc4n3nn2)NCc5ccc(cc5)OC BS-9245 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(cc4Cl)F BS-9254 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4Cl)F BS-9256 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4F)Cl BS-9257 CCOc1ccc(cc1OC)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5cccc(c5)Cl BS-9265 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(c(c5)Cl)Cl)F BS-9270 COc1cc(cc(c1OC)OC)c2nc(on2)Cn3cnc4c(c3=O)nnn4Cc5ccccc5 BS-9271 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccccc4C(F)(F)F BS-9274 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)N4CCCc5c4cccc5 BS-9281 c1ccc2c(c1)c3c(o2)c(ncn3)N4CCC(CC4)C(=O)N5CCN(CC5)c6cccc(c6)Cl BS-9289 c1ccc2c(c1)c3c(o2)c(ncn3)N4CCC(CC4)C(=O)N5CCN(CC5)c6ccccc6Cl BS-9290 c1ccc(cc1)C(=O)N2CCC(CC2)C(=O)N3CCC(CC3)Cc4nc(no4)c5ccc(cc5)F BS-9303 CCOc1ccc(cc1OCC)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5 BS-9311 CCn1cc(c(n1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)Cl)C(=O)n4c(cc(n4)C)C BS-9318 CCOc1ccc(cc1OCC)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccn5 BS-9326 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(cc4)C(=O)C BS-9327 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)N4CCOc5c4cc(cc5)C BS-9329 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)N4CCOc5c4cc(cc5)C BS-9330 CCCCc1ccc(cc1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccc(cc4)C BS-9336 CC(C)c1ccc(cc1)Nc2c3cc(ccc3n4c(n2)c(nn4)S(=O)(=O)c5ccccc5)Cl BS-9341 Cc1cccc(c1)Cn2c3c(c(=O)n(cn3)Cc4nc(no4)c5cccc(c5)Br)nn2 BS-9346 c1cc(ccc1S(=O)(=O)c2cc3cc(cc(c3oc2=O)Br)Br)Cl BS-9350 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(cc4)NC(=O)C BS-9351 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)NC(=O)C BS-9352 CCc1ccc(cc1)NC(=O)Cn2c(=O)c3ccccc3c(n2)c4nc(no4)c5ccc(c(c5)C)C BS-9360 CCOc1ccc(cc1OCC)CC(=O)N2CCC(CC2)Cc3nc(no3)c4ccc(cc4)OC BS-9362 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)C(=O)OC BS-9364 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-9366 CCOC(=O)c1cccc(c1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-9367 CCOC(=O)c1ccccc1NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-9368 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc5c(c4)OCCO5 BS-9370 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4cc(ccc4OC)C BS-9372 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)NCc4ccccc4OC BS-9377 Cc1ccc(cc1C)N(C)S(=O)(=O)c2c(csc2C(=O)n3c(cc(n3)C)C)c4ccccc4 BS-9378 CCc1ccc(cc1)N(C)S(=O)(=O)c2c(csc2C(=O)n3c(cc(n3)C)C)c4ccccc4 BS-9379 Cc1ccc(cc1)c2csc(c2S(=O)(=O)N(C)c3ccc(cc3)C)C(=O)n4c(cc(n4)C)C BS-9380 COc1ccc(cc1OC)c2nc(on2)Cn3cnc4c(c3=O)nnn4Cc5cccc(c5)Cl BS-9381 COc1cc(cc(c1)OC)c2nc(on2)Cn3cnc4c(c3=O)nnn4Cc5ccc(cc5)Cl BS-9382 Cc1c(cccc1Cl)NC(=O)CSc2nc3c4ccccc4oc3c(=O)n2Cc5ccco5 BS-9383 COc1cccc(c1)CNc2c3ccccc3n4c(n2)c(nn4)S(=O)(=O)c5ccc(cc5)Cl BS-9385 CCOC(=O)c1ccc(cc1)NS(=O)(=O)c2c(csc2C(=O)OC)c3ccc(cc3)Cl BS-9386 Cc1cccc(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Br BS-9406 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4cc(cc(c4)OC)OC BS-9409 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(cc4OC)OC BS-9411 Cc1cc(n(n1)C(=O)c2c(c(cs2)c3ccccc3)S(=O)(=O)N(C)c4ccc(cc4)OC)C BS-9412 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(c(c4)OC)OC BS-9413 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(ccc4OC)OC BS-9415 c1cc(cc(c1)F)Cn2c3c(c(=O)n(cn3)Cc4nc(no4)c5ccc(cc5)Br)nn2 BS-9423 c1ccc(cc1)C(=O)Cn2cc(c(=O)c3c2ccc(c3)Br)S(=O)(=O)c4ccccc4 BS-9425 Cc1cccc(c1)N(C)S(=O)(=O)c2c(csc2C(=O)n3c(cc(n3)C)C)c4cccc(c4)F BS-9439 Cc1ccc(cc1)N(C)S(=O)(=O)c2c(csc2C(=O)n3c(cc(n3)C)C)c4cccc(c4)F BS-9440 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(cc4Cl)C BS-9443 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4cc(ccc4C)Cl BS-9444 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(c(c4)Cl)C BS-9445 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)NCc4ccc(cc4)Cl BS-9447 COc1cc(=O)n2c(c1C(=O)O)CCCC2.c1cc(ccc1c2nc(on2)CC3CCNCC3)F BS-9455 Cc1cc(cc(c1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5)C BS-9456 Cc1cccc(c1C)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9457 Cc1ccc(cc1C)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9458 c1ccc(c(c1)N2CCN(CC2)c3[nH]c(=O)c4c(n3)c(cs4)c5ccc(cc5)Br)F BS-9460 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(c(c4)Cl)OC BS-9485 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(ccc4OC)Cl BS-9486 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(c(c4)Cl)OC BS-9487 Cc1cc(c(cc1Cl)OC)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4 BS-9488 CC(C)c1ccc(cc1)S(=O)(=O)c2cc3cc(cc(c3oc2=O)Br)Br BS-9489 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)Br BS-9490 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4)Br BS-9491 COc1cccc2c1o/c(=N\c3ccccc3)/c(c2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9493 COc1cccc(c1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9494 COc1ccc(cc1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9495 COc1ccccc1/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9496 Cc1ccc(c(c1)C)NC(=O)/C(=C\NCc2ccccc2OC)/S(=O)(=O)c3cc(ccc3F)F BS-9497 CCc1ccc(cc1)N2C(=C(C(NC2=S)c3ccc(cc3)Cl)c4nc(no4)c5ccccc5)C BS-9501 Cc1ccc(c(c1)C)S(=O)(=O)c2c3nc(c4ccccc4n3nn2)NCc5ccc6c(c5)OCO6 BS-9505 Cc1cc(n(n1)C(=O)c2c(c(cs2)c3ccc(cc3)F)S(=O)(=O)N(C)c4cccc(c4)F)C BS-9506 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(cc4Cl)F BS-9516 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4)C(F)(F)F BS-9531 CCOc1ccc(cc1OCC)c2csc3c2nc([nH]c3=O)N4CCC(CC4)Cc5ccccc5 BS-9542 CCOc1ccc(cc1OCC)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5cccc(c5)C BS-9565 CCOc1ccc(cc1OCC)c2csc3c2nc([nH]c3=O)N4CCN(CC4)Cc5ccccc5 BS-9566 COc1cc(cc(c1OC)OC)c2nc(on2)c3c4ccccc4c(=O)n(n3)c5cccc(c5)Cl BS-9570 CCCCc1ccc(cc1)NC(=O)CSc2nc3c(csc3c(=O)n2CC)c4ccc(cc4)C BS-9577 Cc1ccc(cc1C)S(=O)(=O)c2c3nc(c4cc(ccc4n3nn2)Cl)Nc5cc(cc(c5)C)C BS-9582 Cc1ccc(cc1C)Nc2c3cc(ccc3n4c(n2)c(nn4)S(=O)(=O)c5ccc(c(c5)C)C)Cl BS-9583 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(cc4)NC(=O)C BS-9596 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(cc4)C(=O)OC BS-9609 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccc(cc4)C BS-9610 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)C(=O)OCC BS-9611 c1ccc2c(c1)c(nc3n2nnc3S(=O)(=O)c4ccc(cc4)Cl)NCc5ccc6c(c5)OCO6 BS-9616 Cc1ccc(cc1C)S(=O)(=O)c2c3nc(c4cc(ccc4n3nn2)Cl)Nc5ccc(cc5)OC BS-9617 Cc1ccc(cc1C)S(=O)(=O)c2c3nc(c4cc(ccc4n3nn2)Cl)Nc5cccc(c5)OC BS-9618 CCOc1ccc(cc1OCC)c2csc3c2nc([nH]c3=O)N4CCN(CC4)c5ccccc5F BS-9634 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)N4CCN(CC4)c5ccc(cc5)F BS-9638 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)N4CCN(CC4)c5ccccc5F BS-9639 Cc1ccc(cc1Cl)N2C(=O)C3C(C2=O)N(N=N3)CC(=O)Nc4ccc(cc4F)Br BS-9641 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)NCc4cccc(c4OC)OC BS-9648 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)NCc4cccc(c4OC)OC BS-9649 CCOc1ccc(c(c1)NC(=O)CSc2nc3c(csc3c(=O)n2C)c4ccccc4)OCC BS-9650 c1cc(cc(c1)Cl)CNC(=O)C2CCN(CC2)C(=O)c3c4n(cn3)CC(OC4)c5ccc(cc5)F BS-9661 CCOc1ccc(cc1)c2nc(c(o2)C)Cn3c(=O)n4cccc(c4n3)S(=O)(=O)N5CCCCC5 BS-9667 Cn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)Oc5ccccc5 BS-9685 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4cc(ccc4OC)Cl BS-9689 CCn1c(=O)c2c(c(cs2)c3ccc(cc3)C)nc1SCC(=O)Nc4ccc(c(c4)Cl)OC BS-9690 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cc(c(cc4OC)Cl)C BS-9691 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4ccc(cc4)Br BS-9692 Cc1ccc(cc1)c2csc3c2nc(n(c3=O)C)SCC(=O)Nc4cccc(c4)Br BS-9693 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4ccc(cc4)Br BS-9694 CCn1c(=O)c2c(c(cs2)c3ccccc3)nc1SCC(=O)Nc4cccc(c4)Br BS-9695 Cc1ccccc1/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9696 Cc1cccc(c1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9697 Cc1ccc(cc1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9698 CCOc1ccc(cc1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9699 CCOc1ccccc1/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9700 CCCn1cc(c(n1)S(=O)(=O)N2CCN(CC2)c3ccccc3OCC)C(=O)n4c(cc(n4)C)C BS-9701 c1cc(cc(c1)F)C2CCCN2c3c4ccc(cc4ncc3S(=O)(=O)c5ccc(c(c5)Cl)F)F BS-9702 C([C@@H]1[C@@H]([C@@H]([C@H]([C@H](O1)OC[C@@H]2[C@H]([C@@H]([C@H]([C@H](O2)O[C@]3([C@H]([C@@H]([C@H](O3)CO)O)O)CO)O)O)O)O)O)O)O BS-9703 Cc1cc(cc(c1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5)C BS-9704 Cc1cccc(c1C)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9705 Cc1ccc(c(c1)C)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9706 Cc1ccc(cc1)CN2CC(CC2=O)C(=O)Nc3cccc(c3)C(=O)N4CCN(CC4)c5ccc(cc5)F BS-9707 COc1cccc(c1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9708 COc1ccc(cc1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9709 COc1ccccc1/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9710 COc1ccc(c(c1)OC)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9711 COc1ccc(c(c1)/N=c\2/c(cc3ccccc3o2)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5)OC BS-9712 CCOC(=O)c1cn(nc1S(=O)(=O)N2CCN(CC2)c3cc(ccc3C)C)Cc4ccc(cc4)Cl BS-9713 CCOC(=O)c1c2c(sc1N=c3c(cc4ccc(cc4o3)O)C(=O)Nc5ccc(cc5)OC)CCCC2 BS-9714 CC(C)c1ccc(cc1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9715 CCOc1ccc(cc1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9716 CCOc1ccccc1/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9717 COc1ccc(c(c1)OC)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5 BS-9718 COc1ccc(c(c1)/N=c\2/c(cc3cccc(c3o2)OC)C(=O)Nc4ccc(cc4)c5[nH]c6ccccc6n5)OC BS-9719 CCOc1ccc(cc1)NC(=O)CN(c2ccc(cc2)C)S(=O)(=O)c3c(csc3C(=O)OC)c4ccccc4 BS-9720 CCN1C(=C(C(N=C1SCC(=O)Nc2ccc(cc2)Cl)c3ccc(cc3)Cl)c4nc(no4)c5ccccc5)C BS-9721 c1ccc(cc1)CN2CCC(CC2)(C(=O)O)N BS-9742 c1ccc2c(c1)CC(C2)(C(=O)O)N BS-9775 Cc1ccc(cc1)S(=O)(=O)NCC(=O)OC CA-0008 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2F)[N+](=O)[O-] CA-0603 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2F)N CA-0604 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNC(=O)c3cc(cc(n3)C(F)(F)F)C(F)(F)F CA-0607 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNC(=O)c3cc(cc(n3)C(F)(F)F)C(F)(F)F CA-0608 c1ccc(c(c1)S(=O)(=O)NNC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F)Cl CA-0609 c1cc(ccc1F)S(=O)(=O)NNC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0610 CC(=O)c1ccc(c(c1)OC)N CA-0700 c1cc(ccc1C=O)c2ccc(c(c2)F)Cl CA-0701 c1ccc(c(c1)C=O)c2ccc(c(c2)F)Cl CA-0702 c1ccc(c(c1)c2ccc(o2)CO)Cl CA-0703 c1ccc(c(c1)c2ccc(o2)/C=C/C(=O)O)Cl CA-0705 Cc1c(c[nH]n1)c2cccs2 CA-0706 c1cc(ccc1C=O)c2ccc(c(c2)Cl)Cl CA-0707 c1ccc(c(c1)C=O)c2ccc(c(c2)Cl)Cl CA-0708 c1ccc(c(c1)c2ccc(cc2)Cl)C(=O)O CA-0709 c1cnn(c1)c2ccc(cc2)CO CA-0710 c1ccc(c(c1)C=O)c2ccc(cc2)[N+](=O)[O-] CA-0714 c1cnn(c1)c2ccc(cc2)/C=C/C(=O)O CA-0715 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)O)Cl CA-0716 c1cc(ccc1C(=O)c2cc([nH]c2)C(=O)O)F CA-0717 c1cc(cc(c1)Br)C(=O)c2cc([nH]c2)C(=O)O CA-0718 Cc1c(nc(s1)c2cccc(c2)C(F)(F)F)CC(=O)O CA-0719 CC(C(=O)c1cccs1)Br CA-0720 Cc1c(nc(s1)c2ccc(cc2)C(F)(F)F)CC(=O)O CA-0721 Cc1c(nc(s1)c2cccs2)CC(=O)O CA-0722 CCOC(=O)C1CCN(CC1)C(C)C(=O)c2cccs2 CA-0723 Cc1cc(n2c(n1)nc(n2)N)C CA-0724 c1ccc(cc1)c2c(nc(s2)c3ccccc3)O CA-0725 CC(C)c1ccc(cc1)/N=C\2/c3cc(ccc3NC2=O)Br CA-0800 CCc1ccc(c(c1)CN(C)C)O CA-0803 c1cc(cc(c1)Br)N2CCNC2=O CA-0804 c1cc(cc(c1)NC(=O)c2cc(cc(n2)C(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F CA-0805 CSc1ccc(cc1)/N=C\2/c3cc(ccc3NC2=O)Br CA-0807 CCCC(C)c1cc(c(c(c1)CN(C)C)O)CN(C)C CA-0810 Cc1cc(c(c(c1)CN(C)C)O)C CA-0811 c1ccc(cc1)NC(=O)c2cc(cc(n2)C(=O)Nc3ccccc3)C(F)(F)F CA-0812 c1cc(ccc1NC(=O)c2cc(cc(n2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F)Cl CA-0813 c1ccc(c(c1)NC(=O)c2cc(cc(n2)C(=O)Nc3ccccc3Cl)C(F)(F)F)Cl CA-0814 COc1cccc(c1)NC(=O)c2cc(cc(n2)C(=O)Nc3cccc(c3)OC)C(F)(F)F CA-0815 CCC(C)Cc1cc(c(c(c1)CN(C)C)O)CN(C)C CA-0820 CNC(=O)c1cc(cc(n1)C(F)(F)F)C(F)(F)F CA-0822 c1c(cc(nc1C(=O)NC2CC2)C(F)(F)F)C(F)(F)F CA-0823 Cc1cc(c(c(c1)Br)O)C CA-0824 CC1=NNC=Cc2c1ccc(=O)[nH]2 CA-0825 CCOC(=O)C1(C(=O)Nc2cc(ccc2O1)[N+](=O)[O-])C CA-0826 CCOC(=O)C1(C(=O)Nc2ccc(cc2O1)[N+](=O)[O-])C CA-0827 Cc1ccc2c(c1)/C(=N/c3cccc(c3)Br)/C(=O)N2 CA-0828 Cc1cc(c(c(c1)C(C)(C)C)O)CN(C)C CA-0831 COc1ccc(c(c1)C(CC(=O)O)N)OC CA-0832 Cc1c(c(n(n1)c2ccc(cc2)C(C)C)C)C(=O)O CA-0833 c1ccc(cc1)NC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0834 c1cc(ccc1NC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F)Cl CA-0835 c1cc(cc(c1)NC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F)C(F)(F)F CA-0836 Cc1c(c(n(n1)c2ccc(cc2)OC)C)C(=O)O CA-0837 c1ccnc(c1)CNC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0838 c1cc(cnc1)CNC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0839 c1ccc(c(c1)NC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F)Cl CA-0840 c1c(cc(nc1C(=O)NN)C(F)(F)F)C(F)(F)F CA-0841 CN(C)Cc1cc(cc(c1O)Cl)Br CA-0842 CC(=O)NNC(=O)c1cc(cc(n1)C(F)(F)F)C(F)(F)F CA-0845 c1ccc(cc1)C(=O)NNC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0846 COc1cccc(c1)NC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0847 CCc1c(c2cc(ccc2n1Cc3cccc(c3)Cl)OC)C(=O)OC CA-0851 CC(C)(C)c1ccc(c(c1)C=O)OC CA-0854 COC(=O)c1ccc(cc1)NC(=O)NCCCl CA-0855 CC1(C(=O)Nc2cc(ccc2O1)[N+](=O)[O-])C(=O)O CA-0858 CC1(C(=O)Nc2ccc(cc2O1)[N+](=O)[O-])C(=O)O CA-0859 CCOC(=O)c1ccc(cc1)N2C(=O)CC(CC2=O)(C)C CA-0860 CCOC(=O)c1cc(c(nc1O)C)C#N CA-0862 c1ccc2c(c1)ccc3c2CC(=O)O3 CA-0864 CC(C)(C)OC(=O)N1CCC(=O)/C(=C/N(C)C)/C1 CA-0865 c1cc(cc(c1)N2CCN(CC2)C(=O)c3cc(cc(n3)C(F)(F)F)C(F)(F)F)C(F)(F)F CA-0866 c1ccc(cc1)N2CCN(CC2)C(=O)c3cc(cc(n3)C(F)(F)F)C(F)(F)F CA-0867 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cc(cc(n3)C(F)(F)F)C(F)(F)F CA-0868 CN1CCN(CC1)C(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0869 CC(C)c1cc(cc(c1O)C(C)C)CN(C)C CA-0871 CC(C)(C)C(=O)/C(=C/N(C)C)/C(=O)OC CA-0872 CCOC(=O)C(=O)CC(=O)c1cc(cc(c1O)[N+](=O)[O-])C CA-0874 CCOC(=O)c1ccc(cc1)N2CCC(CC2)(C)C CA-0875 COC(=O)c1ccc(cc1)N2CCNC2=O CA-0876 CC(=O)c1ccc(c(c1O)CN(C)C)O CA-0877 c1ccc2c(c1)nc(o2)C3CCNCC3 CA-0879 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2cc(cc(n2)C(F)(F)F)C(F)(F)F CA-0882 CC(C)(C)OC(=O)N1CCN(CC1)CCO CA-0884 Cc1cc(cc(c1O)CN(C)C)Cl CA-0888 CC(C)(C)c1c(c[nH]n1)C(=O)OC CA-0890 CC(C)(C)c1c(c([nH]n1)O)Br CA-0893 c1cc(cnc1)c2nccc(n2)c3c(cc(cn3)C(F)(F)F)Cl CA-0896 CC(C)(C)OC(=O)N1CCN(CC1)CCCl CA-0897 c1cnccc1NC(=O)NCCCl CA-0921 CC1=NS(=O)(=O)NC2=C1CCCC2 CA-0923 CCOC(=O)c1ccc2c(c1)sc(n2)Cl CA-0925 CCOC(=O)c1ccc2c(c1)sc(=N)n2C CA-0926 c1cc2c(cc1[N+](=O)[O-])sc(n2)NN CA-0927 CCOC(=O)C1=NS(=O)(=O)NC(=C1)C CA-0929 c1cc(oc1)C(CN)O CA-5050 COC(=O)c1ccccc1C(=O)c2ccc3c(c2)[nH]c(n3)NC(=O)OC CA-7003 c1cc(ncc1C(F)(F)F)C(=O)CC#N CB-0023 c1cc(ccc1CSc2[nH]cc(c(=O)n2)CN3CCCCC3)Br CB-0024 CCc1ccc(cc1)CSc2[nH]cc(c(=O)n2)CN3CCCCC3 CB-0025 c1cc(ccc1CSc2[nH]cc(c(=O)n2)CN3CCCCC3)F CB-0026 Cc1ccc(cc1)CSc2[nH]cc(c(=O)n2)CN3CCCCC3 CB-0027 Cc1cc(cc(c1)CSc2[nH]cc(c(=O)n2)CN3CCCCC3)C CB-0028 c1ccnc(c1)CSc2[nH]cc(c(=O)n2)CN3CCCCC3.Cl CB-0029 c1cc(ccc1CSc2[nH]cc(c(=O)n2)CN3CCOCC3)Br CB-0030 Cc1ccc(cc1)CSc2[nH]cc(c(=O)n2)CN3CCOCC3 CB-0033 Cc1cc(cc(c1)CSc2[nH]cc(c(=O)n2)CN3CCOCC3)C CB-0034 CN1CCN(CC1)Cc2c[nH]c(nc2=O)SCc3ccc(cc3)F CB-0044 Cc1ccc(cc1)CSc2[nH]cc(c(=O)n2)CN3CCN(CC3)C CB-0045 Cc1cc(cc(c1)CSc2[nH]cc(c(=O)n2)CN3CCN(CC3)C)C CB-0046 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccc(cc4)Br)OC)OC CB-0048 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccc(cc4)F)OC)OC CB-0050 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4cc(cc(c4)C)C)OC)OC CB-0052 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccccn4)OC)OC.Cl CB-0053 CCOC(=O)c1cnc2c(c1NCc3ccc(cc3)Cl)cnn2C CB-0058 CCOC(=O)c1cnc2c(c1NCCCOC)cnn2C CB-0059 CCOC(=O)c1cnc2c(c1NCc3ccc(cc3)C)cnn2C CB-0060 CCOC(=O)c1cnc2c(c1NCc3ccccc3)cnn2C CB-0061 CCOC(=O)c1cnc2c(c1NCc3cccs3)cnn2C CB-0062 CCOC(=O)c1cnc2c(c1NCc3ccc(cc3Cl)Cl)cnn2C CB-0063 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4ccc(c(c4)Cl)Cl)OC)OC CB-0072 CCc1nc2c3cc(c(cc3nc(n2n1)SCc4c(cccc4Cl)F)OC)OC CB-0074 CCc1nc2c3cc(c(cc3nc(n2n1)SCCc4ccccc4)OC)OC CB-0075 CC(C)(C)OC(=O)NNC(=O)c1ccc(cn1)C(F)(F)F CB-0109 CC(C)(C)OC(=O)N1CCCCN1C(c2ccccc2)C(=O)OC CB-0203 CC(C)(C)OC(=O)N1CCCCN1CC(=O)O CB-0204 CC(C)(C)OC(=O)N1CCCCN1C(c2ccccc2)C(=O)O CB-0208 CC(C)(C)OC(=O)N1CCCCCN1 CB-0210 CC(C)(C)OC(=O)N1CCCN1C(c2ccccc2)C(=O)OC CB-0216 CC(=O)c1ccnc(c1)Cl CB-0608 Cc1[nH]cc(n1)CO CB-0700 c1cc(ncc1Cl)S CB-0702 CCc1ccc(cc1)/C(=C\C#N)/N CB-0706 c1cc(cc(c1)F)Cn2cc(nn2)CO CB-0707 CCc1ccc(cc1)C(=O)CC#N CB-0711 c1c(cnc(c1C=O)N)Br CB-0712 c1ccc(cc1)c2[nH]cc(n2)CO CB-0713 c1ccc(cc1)Cn2cc(nn2)CO CB-0715 c1cc(c(cc1N2CCCC2)Cl)C(=O)NCCO CB-0716 c1cc(c(cc1Br)F)C(=O)CC#N CB-0717 c1cnn(c1)c2ccc(c(c2)Cl)C(=O)NCCO CB-0718 c1ccc(cc1)Cn2cc(nn2)C=O CB-0719 c1cc(ccc1Cn2cc(nn2)CO)Cl CB-0723 c1cc(cc(c1)C(F)(F)F)Cn2cc(nn2)CO CB-0724 Cc1ccc(cc1)Cn2cc(nn2)CO CB-0725 c1c(c[nH]c(=O)c1C=O)Cl CB-0729 c1cc(ccc1C(=O)NCCO)N2CCCC2 CB-0730 c1cc(c(cc1N2CCCCC2)Cl)C(=O)NN CB-0731 c1cc(cc(c1)C(F)(F)F)Cn2cc(nn2)C=O CB-0734 c1cc(ccc1Cn2cc(nn2)C=O)Cl CB-0735 c1ccc(cc1)c2[nH]cc(n2)C=O CB-0736 Cc1ccc(cc1)Cn2cc(nn2)C=O CB-0737 c1ccc(c(c1)C(=O)CC#N)F CB-0738 CS(=O)(=O)CC(=O)c1ccc(cc1)S(=O)(=O)C CB-0739 c1c(sc(n1)Cl)Cn2cc(nn2)CO CB-0740 c1cnn(c1)c2ccc(cc2)C(=O)NCCO CB-0742 c1cc(ccc1C(=O)NCCO)n2ccnc2 CB-0743 c1cc(ncc1C=O)O CB-0744 CN(C)c1ccc(cn1)C=O CB-0745 Cc1nc(cs1)C(=O)O CB-0747 c1c(c[nH]c(=O)c1Br)C=O CB-0748 c1c(c[nH]c(=O)c1Cl)C=O CB-0749 CNc1ccc(cn1)C=O CB-0750 c1c(c[nH]c(=O)c1I)C=O CB-0751 c1cc(c(c(c1)Cl)Cn2cc(ccc2=O)C=O)F CB-0752 Cn1cc2ccc(cc2n1)N CB-0800 Cn1c2c(cc(=O)[nH]c2c(=O)n(c1=O)C)C(F)(F)F CB-0802 c1cc2cn[nH]c2cc1Br CB-0803 c1cc2cn[nH]c2cc1NS(=O)(=O)CCCCl CB-0804 Cn1c2c(cc(cc2Br)[N+](=O)[O-])cn1 CB-0805 CC(C)(C)OC(=O)N1CCC(CC1)c2nnc(n2C)S CB-0809 c1cnc(nc1C(F)(F)F)N2CCCNCC2 CB-0810 Cn1c2cc(ccc2cn1)N CB-0812 COC(=O)c1ccc(o1)Oc2ccc(cc2)Br CB-0815 Cn1c2cccc(c2cn1)[N+](=O)[O-] CB-0816 Cc1c2c(cc(=O)[nH]c2n(n1)C)C(F)(F)F CB-0817 CCOC(=O)c1cc2cc(ccc2o1)N CB-0818 Cn1c2ccc(cc2c(n1)Br)[N+](=O)[O-] CB-0820 c1cc(ccc1Oc2ccc(o2)C(=O)O)Br CB-0821 c1cc2c(cn[nH]2)c(c1)Cl CB-0825 c1cn2cc(cc(c2n1)Cl)Cl CB-0827 c1cc2cn[nH]c2cc1N3CCCS3(=O)=O CB-0829 c1cc(c(cc1Br)/C=N/N)F CB-0830 COC(=O)c1cc2c(s1)ccs2 CB-0831 c1cc2cn[nH]c2c(c1)Cl CB-0833 c1csc2c1sc(c2)C(=O)NCCO CB-0839 c1csc2c1sc(c2)C(=O)NN CB-0840 CC(C)(C)OC(=O)N1CCC(CC1)c2nnc(n2C)SC CB-0847 CCOC(=O)C(=O)C[n+]1ccccc1N.[Br-] CB-0849 Cc1ccc(c2c1cn[nH]2)N CB-0850 CCOC(=O)C1=CC2C=CC=CC2=C1 CB-0853 c1ccc(c(c1)Oc2ccc(o2)C(=O)O)Br CB-0854 Cc1c(cc(c2c1cn[nH]2)Br)[N+](=O)[O-] CB-0855 Cc1c2c(cc(nc2n(n1)C)Cl)C(F)(F)F CB-0857 c1cc2c(c(c1)Cl)c(n[nH]2)Br CB-0860 c1c(cn2c(cnc2c1Cl)Br)Cl CB-0861 CC1Cc2cc(ccc2N1C(=O)C)S(=O)(=O)Cl CB-0863 c1c(cnc(c1Cl)c2csc(n2)NC3CCCCC3)C(F)(F)F CB-5001 c1ccc(c(c1)C(=O)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl CB-5007 COC(=O)Nc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl CB-5008 CC(=O)Nc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl CB-5009 c1cc(ccc1C(=O)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl CB-5010 c1ccc(cc1)C(=O)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl CB-5011 c1cc(c(nc1)Cl)C(=O)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl CB-5028 c1cc(ccc1NC(=O)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl CB-5030 c1c(cnc(c1Cl)c2csc(n2)NC(=O)C3CCCCC3)C(F)(F)F CB-5036 Cc1ccccc1C(=O)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl CB-5042 c1cc(c(nc1)C(=O)Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F CB-5046 c1ccc(cc1)NC(=S)N2CC(CC(C2)C(F)(F)F)C(F)(F)F CC-0004 C[Si](C)(C)C#Cc1cc(cnc1N)Cl CC-0010 c1ccc(cc1)CS/C(=N\c2ccccc2Cl)/N3CC(CC(C3)C(F)(F)F)C(F)(F)F CC-0031 Cc1c(cccn1)[N+](=O)[O-] CC-0602 c1c(c(cc(c1[N+](=O)[O-])Br)F)C=O CC-0606 c1cc(ccc1c2c(c[nH]n2)N)Br CC-0610 c1cc2c(cc1[N+](=O)[O-])cc(o2)C=O CC-0611 c1cc2c(cn[nH]2)c(c1)Br CC-0702 c1cc(cc(c1)[N+](=O)[O-])c2ccc(cc2)CO CC-0703 c1ccc(c(c1)CO)c2ccc(cc2)[N+](=O)[O-] CC-0704 COC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccccc2C=O CC-0710 COC(=O)c1ccc(c(c1)[N+](=O)[O-])NC2CCCCC2 CC-0711 COC(=O)c1ccc(c(c1)[N+](=O)[O-])SC CC-0712 c1ccc(c(c1)S(=O)(=O)NCCCN2CCCC2=O)Cl CC-0719 CC(=O)Nc1ccc(c(c1)OCc2ccc(cc2)[N+](=O)[O-])C(=O)OC CC-0721 c1cc(ccc1S(=O)(=O)NCCCN2CCCC2=O)Cl CC-0722 c1ccc2c(c1)nc(o2)N3C(=C(CN3)C#N)N CC-0724 CCC(c1ccc(cc1)[N+](=O)[O-])C(=O)OC CC-0725 c1cc(c(cc1[N+](=O)[O-])O)F CC-0726 c1ccc2c(c1)nc(s2)N(CCC#N)N CC-0727 Cc1cccc2c1nc(s2)N(CCC#N)N CC-0729 c1c(cn2c(cnc2c1Cl)I)Cl CC-0732 c1cc(ccc1n2c3c(cn2)c(ncn3)N)[N+](=O)[O-] CC-0733 CS(=O)(=O)/C(=C/c1cc(c[nH]1)C(=O)CN2CCC(CC2)C(F)(F)F)/C#N CC-0737 c1cc2cc[nH]c2c(c1)C(=O)O CC-0741 c1cc(c(c(c1)Cl)CO/N=C/c2cnc(s2)N3CCC(CC3)C(F)(F)F)F CC-0742 c1cc(c(cc1Cl)Cl)CO/N=C/c2cnc(s2)N3CCC(CC3)C(F)(F)F CC-0743 COC(=O)c1cccc2c1[nH]cc2 CC-0744 c1c(c[nH]c1C(=O)O)I CC-0801 c1cc2c(nc1)NCC2 CC-0803 c1c(cnc(c1I)N)Cl CC-0804 c1cc2c(c[nH]c2nc1)C(=O)O CC-0806 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)C(=O)O CC-0808 c1cn2cc(cc(c2n1)I)Cl CC-0809 COC(=O)c1ccc(nc1)N2CCNCC2 CC-0811 C#Cc1cc(cnc1N)Cl CC-0812 c1cc(ccc1C(=O)N/N=C/c2cnc(s2)N3CCC(CC3)C(F)(F)F)Cl CC-0814 c1cc(ccc1/C(=C/c2cnc(s2)N3CCC(CC3)C(F)(F)F)/C#N)Cl CC-0815 CS(=O)(=O)/C(=C/c1cnc(s1)N2CCC(CC2)C(F)(F)F)/C#N CC-0816 c1c[nH]c2c1cc(cn2)Cl CC-0823 c1ccc(c(c1)NC(=O)c2ccc(cc2)OCCN3CCC(CC3)C(F)(F)F)Cl CC-0824 c1c(cnc2c1c(c[nH]2)Br)Cl CC-0827 c1cc2c(cc1Cl)/C(=C/c3cnc(s3)N4CCC(CC4)C(F)(F)F)/C(=O)N2 CC-0832 CCOC(=O)c1c(nc(nn1)c2c(cc(cn2)C(F)(F)F)Cl)Nc3ccccc3 CC-5008 CCOC(=O)c1c(nc(nn1)c2c(cc(cn2)C(F)(F)F)Cl)N(C)C CC-5013 COC(=O)c1c(c(nc(n1)O)O)Cl CD-0006 CN(C)CC(=O)NCc1c(cc(cn1)C(F)(F)F)Cl CD-0011 Cc1c(c(nc(n1)N)N)I CD-0020 Cc1c(c(nc(n1)N)Cl)I CD-0041 c1cc(ccc1[C@H]2N(CCS2)C(=O)Nc3ccc(cc3)Cl)OCc4c(cc(cn4)C(F)(F)F)Cl CD-0053 c1c(cnc(c1Cl)CNC(=O)CN2CCC(CC2)C(F)(F)F)C(F)(F)F CD-0061 Cc1c(c(nc(n1)N)O)I CD-0062 COC(=O)c1c(c(nc(n1)Cl)Cl)Cl CD-0064 c1cc(cc(c1)C(F)(F)F)/C(=C/O)/C#N CD-0065 c1ccc(cc1)C(C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)N3CCC(CC3)C(F)(F)F CD-0073 c1cc(sc1)/C(=C/O)/C#N CD-0084 c1cc(ccc1/C(=C/O)/C#N)Br CD-0085 Cn1c2c(c(cc(=O)n2Cc3c(cccc3F)F)C(F)(F)F)c(=O)n(c1=O)C CD-0092 c1ccc(cc1)C(C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Oc3ccc(cc3)Cl CD-0097 c1cc(c(cc1/C(=C\O)/C#N)Cl)Cl CD-0105 Cc1ccccc1S(=O)(=O)Nc2ccc(nc2)Cl CD-0107 Cc1ccccc1S(=O)(=O)Nc2ccc(nc2)OC CD-0111 CC(C)(C)OC(=O)N1CCC[C@H]1C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl CD-0114 CCOC(=O)c1c(nc(o1)N)C(F)(F)F CD-0201 c1c(ncnc1O)C(F)(F)F CD-0251 CCOC(=O)c1c(c2cc(ccc2o1)Br)NC(=O)OC(C)(C)C CD-0252 CCOC(=O)c1c(nc2n1cccc2Br)C(F)(F)F CD-0279 c1cc(nc(c1C(=O)O)Br)C(F)(F)F CD-0293 CC(C)(C)OC(=O)Nc1c2cc(ccc2oc1C(=O)O)Br CD-0294 COc1c(cc(cn1)Cl)C(=O)OC CD-0700 c1c[nH]nc1I CD-0702 COc1c(c(c(cn1)C(F)(F)F)C(=O)OC)Cl CD-0705 COC(=O)c1cc2cccnc2s1 CD-0707 COc1cnc(nc1O)c2cccc(c2)[N+](=O)[O-] CD-0710 c1c(c(c(c(n1)Cl)Cl)C(=O)O)Cl CD-0714 COc1cnc(nc1Cl)c2cccc(c2)[N+](=O)[O-] CD-0715 COC(=O)c1cnc(nc1C(F)(F)F)Cl CD-0717 CCOC(=O)c1cccnc1N(C)C2CCCCC2 CD-0721 COc1c(c(c(cn1)Cl)C(=O)O)Cl CD-0723 CCOC(=O)c1cnc(nc1)n2cccc2 CD-0724 Cc1cc(nc(c1C#N)OC)C CD-0725 CC(C)(C)C(=O)Nc1cccc(c1C=O)OC CD-0726 Cc1ccc(cc1)c2cc[nH]n2 CD-0728 c1ccc(cc1)CNc2cc(ccc2[N+](=O)[O-])C#N CD-0730 COC(=O)c1c(cnc(c1Cl)Cl)C(F)(F)F CD-0731 c1cnc(nc1Br)N CD-0732 CC(=O)Nc1c(cc(s1)Br)C(=O)OC CD-0734 c1c(c(c(c(n1)Cl)Cl)CO)Cl CD-0737 COc1ccc(cc1[N+](=O)[O-])CC(=O)NN CD-0739 COC(=O)c1c(cnc(c1Cl)N2CCNCC2)C(F)(F)F CD-0741 c1cc(c(cc1CC(=O)NN)N)O CD-0742 c1cc2c(cc1[N+](=O)[O-])OCCN2 CD-0744 c1c(n[nH]c1[N+](=O)[O-])C(=O)O CD-0745 COc1cc(cc2c1oc(=O)[nH]2)C(=O)OC CE-0007 c1cc(ccc1CNc2cc(nc(n2)N)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl CE-0014 COc1cc(c2c(c1)nco2)C(=O)OC CE-0023 Cc1nc2cc(cc(c2o1)C(=O)OC)OC CE-0024 COc1cc(c2c(c1)[nH]c(=O)o2)C(=O)OC CE-0026 COc1cc(c2c(c1)NC(=O)CO2)C(=O)OC CE-0027 c1ccc(cc1)C(=O)Oc2cc(cc3c2oc(=O)[nH]3)Cl CE-0039 COc1cc(c(c(c1)[N+](=O)[O-])OCc2ccccc2)C(=O)OC CE-0042 COc1cc(cc(c1Cl)[N+](=O)[O-])C(=O)OC CE-0044 Cn1c(n[nH]c1=S)c2cccc(c2)Br CE-0047 COc1c(cc(cc1I)Br)C(=O)NN CE-0049 Cn1c(n[nH]c1=S)c2ccc(cc2)Br CE-0050 Cn1c(n[nH]c1=S)c2ccc(c(c2)F)Br CE-0052 COc1cc(c(c(c1)N)OCc2ccccc2)C(=O)OC.Cl CE-0053 COc1cc(c(c(c1)[N+](=O)[O-])OCc2ccccc2)C(=O)O CE-0054 CCc1nc2cc(cc(c2o1)OC)C(=O)OC CE-0061 CCc1nc2cc(cc(c2o1)C(=O)OC)OC CE-0062 CC(C)CC(=O)OC(=O)[C@H]1CCCN1C(=O)OC(C)(C)C CE-0075 c1cc(ccc1c2cn(nn2)COc3c(cc(cn3)C(F)(F)F)Cl)Cl CE-0078 CC(=O)c1cc2c(cc1NC(=O)c3ccccc3F)OCO2 CE-0083 c1cc(ccc1C(=O)N2CC(C2)c3c(cc(cn3)C(F)(F)F)Cl)Cl CE-0084 c1cc(cc(c1)O)Nc2ccnc3c2ccc(c3)Cl.Cl CE-0093 COc1cc(cc(c1Cl)N)C(=O)OC CE-0094 c1cc(c(cc1Cl)Cl)C(=O)N2CCN(CC2)c3cc(nc(c3)C(F)(F)F)C(F)(F)F CE-0095 CC(=O)c1c2ccccn2nc1c3ccccc3 CE-0100 C[C@@H]1CN(C[C@@H](O1)C)c2ccc(cn2)[N+](=O)[O-] CE-0111 C[C@@H]1CN(C[C@@H](O1)C)c2ccc(cn2)N.Cl.Cl CE-0117 c1cc(cc(c1)Cl)COc2ccc3c(cc(=O)oc3c2)CCl CE-0118 CCOC(=O)[C@H]1[C@H]2[C@@H]1C(=O)N(C2=O)Cc3ccccc3 CE-0202 c1ccc(cc1)CCc2cnccn2 CE-0203 Cc1cncn1CCCNC(=S)Nc2ccc(c(c2)OC)OC CE-0205 Cc1cncn1CCCn2c(=O)c3ccccc3[nH]c2=S CE-0206 c1ccc(cc1)CN2C[C@@H]([C@H](C2)C(=O)O)c3ccccn3 CE-0208 CCOC(=O)/C=C/c1cccnc1 CE-0210 c1ccc2c(c1)C(=O)CCCN2 CE-0212 c1ccc(cc1)CCC2CNCCN2 CE-0213 c1c(cnc(c1Cl)C2CNC2)C(F)(F)F CE-0214 CC(C)(C)OC(=O)N1CCC(CC1)(C#N)N CE-0216 c1cc2ncc(n2cc1C(F)(F)F)Cl CE-0217 c1ccnc(c1)C2CNC2.Cl.Cl CE-0219 c1c(cc(c(c1Cl)OCCBr)Cl)Cl CE-0221 c1ccc(cc1)CN2C[C@@H]3[C@H](C2)[C@H]3CO CE-0223 CCCNCCOc1c(cc(cc1Cl)Cl)Cl CE-0228 CCOC(=O)C=C1CCN(CC1)C(=O)OC(C)(C)C CE-0229 COC(=O)C(C(c1ccccc1)(c2ccccc2)OC)O CE-0230 CCOC(=O)C1CC12CCN(CC2)C(=O)OC(C)(C)C CE-0233 CC(C)(C)OC(=O)N1CCC2(CCC(CC2)C#N)CC1 CE-0240 COC(c1ccccc1)(c2ccccc2)C(C(=O)O)O CE-0241 C1C2C1C(NC2)C(F)(F)F CE-0244 CCOC(=O)CNCc1ccc(cc1)OC CE-0701 COc1cc(c(cc1C(=O)O)I)N CE-0702 CCOC(=O)c1c(cc(cn1)Cl)C(=O)C CE-0703 C1CCC(CC1)N2CCC3(CC2)NCCS3.Cl CE-0704 c1cc(ccc1N)Sc2c(cc(cn2)C(F)(F)F)Cl CE-0705 C1CCC(CC1)N2CCC3(CC2)NC(CS3)C(=O)O CE-0706 c1cc(ccc1S(=O)(=O)c2ccc(cn2)N)Cl CE-0708 COc1ccc(cc1)S(=O)(=O)c2ccc(cn2)N CE-0709 c1ccc(cc1)SCCN CE-0710 c1cc(ccc1S(=O)(=O)c2ccc(cn2)[N+](=O)[O-])Br CE-0712 CC(=O)c1cc(cnc1C(=O)O)Cl CE-0714 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl CE-0715 c1cc(ccc1Sc2ccc(cn2)N)Br CE-0716 c1cc(ccc1N)Sc2ccc(cn2)C(F)(F)F CE-0718 c1cc(ccc1[N+](=O)[O-])S(=O)c2c(cc(cn2)C(F)(F)F)Cl CE-0719 C1CC2(CCC13NCCS3)NCCS2.Cl.Cl CE-0720 c1ccc(cc1)C2(CCC3(CC2)NCCS3)C#N.Cl CE-0721 c1cnc2nc(nn2c1N)N CE-0724 c1cc(ccc1S(=O)c2ccc(cn2)[N+](=O)[O-])Br CE-0725 c1cc(ccc1S(=O)(=O)c2ccc(cn2)N)Br CE-0727 c1cc(c(nc1)Sc2ccc(cc2)N)C#N CE-0728 c1cc(ccc1S(=O)c2ccc(cn2)N)Br CE-0729 COC(=O)c1cc(ccc1NCc2ccc(cc2)N)[N+](=O)[O-] CE-0730 c1cc(ccc1N)S(=O)(=O)c2c(cc(cn2)C(F)(F)F)Cl CE-0731 c1cc(ccc1N)S(=O)c2c(cc(cn2)C(F)(F)F)Cl CE-0732 CS(=O)(=O)c1ccc(cn1)[N+](=O)[O-] CE-0735 CS(=O)(=O)c1c(cccn1)[N+](=O)[O-] CE-0737 CS(=O)(=O)c1ccc(cn1)N CE-0738 CNc1c(cc(cn1)N)Cl CE-0739 c1cc(ncc1[N+](=O)[O-])N2CCSC2=O CE-0740 COC(=O)CSc1ccc(cn1)[N+](=O)[O-] CE-0742 CCOC(=O)C1CCN(CC1)CCNC(=O)OC(C)(C)C CE-0744 c1cc(ncc1N)N2CCSC2=O CE-0745 CS(=O)(=O)c1c(cccn1)N CE-0746 C1CCC2(CC1)NC(CS2)C(=O)O CE-0747 CS(=O)(=O)c1ccc(s1)C=O CE-0749 CS(=O)(=O)c1ccc(cn1)C=O CE-0750 c1ccc(cc1)C2(CCC3(CC2)NC(CS3)C(=O)O)C#N CE-0752 CCOC(=O)c1c(ccc(n1)C2CC2)C#N CE-0754 c1cc(nc(c1C#N)C(=O)O)C2CC2 CE-0755 Cc1ccc(cc1)CC(CCNC(=O)OC(C)(C)C)C(=O)O CE-0756 CCOC(=O)CN1CCSC1=O CE-0758 CNc1cc(ccc1[N+](=O)[O-])CO CE-0761 c1cc(ccc1NC2(CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl)C(=O)N)Cl CF-0001 c1ccc(c(c1)NC2(CCN(CC2)Cc3c(cc(cn3)C(F)(F)F)Cl)C(=O)N)Cl CF-0017 c1ccc(c(c1)N2C(=O)NC(=O)C23CCN(CC3)Cc4c(cc(cn4)C(F)(F)F)Cl)Cl CF-0018 COC(=O)c1cc(=O)n(c(=O)[nH]1)CCc2ccc3c(c2)OCO3 CF-0041 CS(=O)(=O)N(Cc1c(cccc1F)F)[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl CF-0046 CN(C)C(=O)c1cn(nn1)Cc2c(cc(cn2)C(F)(F)F)Cl CF-0048 COC(=O)c1c(ccs1)NC(=O)c2ccc(cc2)C#N CF-0049 c1cc(c(c2c1c(n[nH]2)N)F)F CF-0051 c1cc(ccc1NC(=S)N)Cl CF-0053 COC(=C(C#N)C#N)c1cccc2c1cccc2 CF-0079 Cc1cccc(c1NC(=O)C(C)C)C CF-0081 c1ccc(cc1)C(=O)c2cccnc2C(=O)O.Cl CF-0091 CCNCc1ccccn1 CF-0240 CC1Cc2ccccc2O1 CF-0246 Cc1cc(ccc1[N+](=O)[O-])N2CCNCC2 CF-0280 c1cnc(cc1C(F)(F)F)N.Cl CF-0281 c1ccc2c(c1)ncn2c3ccc(cc3)[N+](=O)[O-] CF-0282 c1cc(ccc1C=O)c2ccc3c(c2)nco3 CF-0701 COc1ccc(cc1)c2c(c([nH]n2)N)F CF-0702 CC(C)(C)c1csc(n1)NC.Br CF-0703 CCOC(=O)Cc1nc2cc(ccc2o1)Cl CF-0704 CNc1nc(cs1)c2ccc(cc2)Br.Br CF-0705 CCOC(=O)c1c(c2ccccc2[nH]1)C(=O)O CF-0707 CCOC(=O)c1c(nc(s1)NC)C(F)(F)F CF-0708 CNc1nc(cs1)c2ccc(cc2)OC.Br CF-0709 CCOC(=O)Cc1[nH]c2ccc(cc2n1)Br CF-0710 CC(C)(C)OC(=O)N1CCC(CC1)Nc2cc(ccc2[N+](=O)[O-])C(=O)OC CF-0711 CCOC(=O)c1nc(cs1)c2ccc(cc2)Cl CF-0712 CCOC(=O)c1nc(cs1)c2ccc(cc2)OC CF-0715 c1ccc2c(c1)cc(c(c2C=O)Cl)C=O CF-0716 CCOC(=O)c1c(c2cc(ccc2s1)C=O)N CF-0719 CCOC(=O)c1nc(cs1)c2ccc(cc2)[N+](=O)[O-] CF-0720 CCOC(=O)c1nc(cs1)c2cccc(c2)Br CF-0721 COC(=O)c1ccc(c(c1)F)/N=C/c2ccccc2O CF-0723 c1cc2c(cc1Br)nc([nH]2)CC(=O)O CF-0724 CCOC(=O)Cc1nc2ccc(cc2o1)[N+](=O)[O-] CF-0725 COC(=O)c1ccc(c(c1)F)/N=C/c2cc(ccc2O)Br CF-0728 CC(C)(C)C(=O)C=CN(C)C CF-0730 c1c(cc(c(c1Cl)OC(=O)CC(=O)Oc2c(cc(cc2Cl)Cl)Cl)Cl)Cl CF-0733 CCOC(=O)c1cc2cc(cnc2[nH]c1=O)Br CF-0735 CCOC(=O)c1cc2cccnc2[nH]c1=O CF-0736 CCOC(=O)c1cc2cc(cnc2nc1C(F)(F)F)Br CF-0739 c1cc2cc(c(=O)[nH]c2nc1)C#N CF-0740 c1cc2cc(sc2c(c1)Br)CO CF-0742 c1c[nH]c2c1c(ncn2)N3CCOCC3 CF-0743 c1cc(c(cc1C=O)C(=O)O)F CF-0744 c1cc(c2cc(sc2c1)CO)F CF-0745 CCOC(=O)c1nc(c(s1)C)C CF-0746 COc1c(cc(cn1)CO)Cl CF-0749 CC(C)(C)OC(=O)N(c1ccc(cn1)C(=O)OC)C(=O)OC(C)(C)C CF-0752 CCc1csc(n1)C(=O)OCC CF-0753 CC(C)(C)Sc1ccc(cc1)CO CF-0754 c1c(cnc(c1Cl)Cl)CCl CF-0755 CC(C)(C)OC(=O)N1CCc2c(c(=O)n(cn2)Cc3cc(c(c(c3)F)F)F)C1 CF-0756 Cc1ccc(cc1)NC(=S)NC(=O)c2ccccc2 CF-0757 CCOC(=O)C1C(CC(=CC1=O)c2cccc(c2)OC)c3ccsc3 CF-0758 Cn1c(cnc1CO)Cl CF-0759 COC(=O)c1ccc(c(c1)F)/N=C/c2cc(ccc2O)Cl CF-0761 c1cc(ccc1SCCN)Br CF-0764 Cn1c(nc(c1Cl)Cl)CO CF-0765 c1ccc2c(c1)cc([nH]2)C=O CF-0774 CCOC(=O)c1c(cc(cn1)Cl)C#N CF-0776 CC(C)(C#N)NCc1ccc(cc1)Cl CG-0004 [C-]#[N+]CC(=O)NCCNc1c(cc(cn1)C(F)(F)F)Cl CG-0005 c1c(cc(cc1CBr)Br)CBr CG-0013 CC(C)(C#N)Nc1ccc(cc1)OC CG-0014 c1cc2c(nc1)ncn2C3CCNCC3.Cl CG-0018 c1cc(c(nc1)N)NC2CCCCC2 CG-0019 CC(C)(C#N)NCc1ccc(cc1)F CG-0023 c1cc2c([nH]c(=O)n2C3CCCCC3)nc1 CG-0044 c1cc2c(nc1)ncn2C3CCCCC3 CG-0045 c1ccc(cc1)NC(=O)CCCCCCC(=O)O CG-0046 CC(C)(C#N)Nc1ccccc1 CG-0047 CC(C)(C#N)Nc1ccc(cc1)F CG-0050 Cc1ccc(cc1)CNC(C)(C)C#N CG-0051 Cc1c2ccccc2oc1C(=O)OC CG-0200 CC(C)(C)OC(=O)N1CCN(CC1)Cc2c[nH]c3c2cccn3 CG-0207 c1cc(nc(c1N)F)Br CG-0211 c1cn2ccnc2cc1C(=O)NN CG-0212 c1cc2c(c[nH]c2nc1)CN3CCCCC3 CG-0215 CCOC(=O)C(Cc1c[nH]c2c1cccn2)[N+](=O)[O-] CG-0221 c1cc2c(c[nH]c2nc1)C(=O)C(Cl)(Cl)Cl CG-0229 COC(=O)c1c[nH]c2c1cccn2 CG-0232 Cc1cc2ccccc2[nH]1 CG-0500 c1ccc2c(c1)cc[nH]2 CG-0501 Cc1c[nH]c2c1cccc2 CG-0502 COc1ccc2c(c1)cc[nH]2 CG-0503 c1cc2c(cc[nH]2)cc1Cl CG-0504 c1cc2c(nc1)N=CC2 CG-0505 c1ccc(cc1)c2cc3ccccc3[nH]2 CG-0506 Cc1cc2c([nH]1)cccc2O CG-0507 Cc1cccc2c1[nH]cc2 CG-0508 Cc1ccc2c(c1)cc[nH]2 CG-0510 c1ccc(cc1)COc2ccc3c(c2)cc[nH]3 CG-0512 c1ccc2c(c1)CC(=O)N2 CG-0513 c1cc2c(cc[nH]2)cc1C#N CG-0514 c1ccc2c(c1)cc([nH]2)C(=O)O CG-0515 c1cc2c(cc[nH]2)cc1C(=O)O CG-0516 c1cc2c(cc1Cl)cc([nH]2)C(=O)O CG-0517 c1ccc2c(c1)c(c[nH]2)CCCC(=O)O CG-0518 Cn1c2ccccc2cc1C(=O)O CG-0519 CCOC(=O)c1cc2ccccc2[nH]1 CG-0521 c1ccc2c(c1)c(c[nH]2)CC(=O)O CG-0522 CC(=O)c1c[nH]c2c1cccc2 CG-0523 Cc1ccc(nc1)C(=O)O CG-0700 Cc1ccc(nc1)CO CG-0704 c1ccc(cc1)Cn2cc(cc2N)C#N CG-0705 Cc1ccc(nc1)C=O CG-0707 CCOC(=O)c1cc(c(cn1)Cl)C(F)(F)F CG-0708 COc1ccc(cc1)c2ccc(cn2)C=O CG-0710 CC(=O)Nc1ccc(cc1OC(F)(F)F)I CG-0711 CC(C)c1cc(on1)N CG-0713 c1c(c(cnc1C(=O)O)Cl)C(F)(F)F CG-0714 c1c(ncc(c1C(F)(F)F)Cl)CO CG-0716 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2cc(ccc2F)[N+](=O)[O-] CG-0717 COc1ccc(cc1)c2ccc(cn2)CO CG-0718 c1ccc2c(c1)c(c([nH]2)C#N)Cl CG-0720 c1ccc(cc1)Cn2cc(nn2)CCl CG-0721 c1ccc2c(c1)c(c([nH]2)C#N)Br CG-0723 COc1ccc(cc1)Cc2ccc(nc2)Cl CG-0724 c1cc(ccc1Cc2ccc(nc2)Cl)C=O CG-0726 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2cc(ccc2Cl)[N+](=O)[O-] CG-0728 c1cc(c2ncc(n2c1)I)[N+](=O)[O-] CG-0729 c1cc(c2ncc(n2c1)Br)[N+](=O)[O-] CG-0730 c1ccc(cc1)COc2cccn3c2ncc3Cl CG-0731 CC(=O)c1cnc(cc1Cl)Cl CG-0732 COC(=O)c1cc(c(c(c1)Br)O)N CG-0733 c1cc(c(cc1I)OC(F)(F)F)N CG-0735 c1c(cc(nc1Cl)Cl)CCl CG-0737 c1cncc2c1c(=O)[nH]cn2 CG-0739 Cc1cccc2c1[nH]c(=O)oc2=O CG-0740 Cc1cc(cc2c1[nH]c(=O)oc2=O)I CG-0741 c1ccc2c(c1)c(c([nH]2)C#N)I CG-0745 COc1cc2c(c(c1)Br)OCCN2 CG-0746 Cn1c2ccc(cc2c(n1)N)C3OCCCO3 CG-0747 B(c1ccc(nc1)OC)(O)O CH-0005 Cc1c(cnn1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3cccc(c3)Oc4ccccc4 CH-0017 Cc1c(cnn1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Oc4ccccc4 CH-0018 Cc1c(c(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)C)C(=O)Nc3cccc(c3)Oc4ccccc4 CH-0019 Cc1c(c(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)C)C(=O)Nc3ccc(cc3)Oc4ccccc4 CH-0020 Cc1c(cnn1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)C(C)(C)C CH-0021 Cc1c(c(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)C)C(=O)Nc3ccc(cc3)C(C)(C)C CH-0022 c1ccnc(c1)c2ccc(=O)[nH]c2 CH-0026 Cc1c(c(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)C)C(=O)NCc3ccccc3 CH-0041 c1ccc(cc1)n2cc(ccc2=O)c3ccccn3 CH-0042 c1ccc(cc1)n2cc(cc(c2=O)Br)c3ccccn3 CH-0052 CCOc1cc2c(cc1Br)CCC(=O)N2 CH-0701 CN1c2cc(c(cc2CCC1=O)Br)OC CH-0703 Cc1ccc(c(c1)C(=O)C)[N+](=O)[O-] CH-0704 CN1c2cc(c(cc2CCC1=O)c3cccnc3)OC CH-0706 CC(C)(C)c1c(nco1)C(=O)O CH-0708 CC(C)(C)c1c(nco1)C(=O)NN CH-0709 CC(C)(C)c1c(nc[nH]1)C(=O)O CH-0711 c1c2c(cc(c1Br)O)NCCC2 CH-0712 CCc1csc(n1)C(=O)O CH-0713 CCOc1cc2c(cc1Br)CCC(=O)N2C CH-0714 c1ccc(cc1)n2cc(cn2)I CH-0717 CCOc1cc2c(cc1Br)CCCN2 CH-0719 c1cc(c(cc1N)C#N)Cl CK-0025 CC(=O)SCC1(CCOCC1)C(=O)OC CK-0031 CCCC1CCC(CC1)c2ccc(cc2)N.CCCC1CCC(CC1)c2ccc(cc2)N.OS(=O)(=O)O CK-0036 CC(C)(C)OC(=O)N1CCc2c(c(=O)n(cn2)Cc3ccc(c(c3)F)F)C1 CK-0039 CC(C)(C)OC(=O)N1CCCC(C1)N2C(=O)c3ccccc3C2=O CK-0040 Cc1c(sc(n1)c2cccc(c2)C(F)(F)F)C(=O)/C=C/N(C)C CK-0043 Cc1cccc(c1)Nc2ccncc2S(=O)(=O)N CK-0211 CC(C)NC(=O)Oc1ccccc1 CK-0214 [2H]C([2H])([2H])C([2H])(C([2H])([2H])[2H])NC(=O)Oc1ccccc1 CK-0215 CN(C)c1ccc(cc1)c2nc3ccc(cc3s2)Br CK-0220 COc1ccc2c(c1F)[nH]nc2N CK-0224 Cc1ccc(cn1)Oc2cnn(c(=O)c2Cl)C CK-0228 C1CN2C(=N1)SSC2=S CK-0237 c1cc(cc(c1)Oc2c(cccn2)C(=O)Oc3cccc(c3)C(F)(F)F)C(F)(F)F CK-0240 CC(C)(C)OC(=O)NCCCC[C@@H](C=O)NC(=O)OCC1c2ccccc2-c3c1cccc3 CK-0700 CN(C(=O)[C@H](CCC(=O)NC(c1ccccc1)(c2ccccc2)c3ccccc3)NC(=O)OCC4c5ccccc5-c6c4cccc6)OC CK-0701 CN(C(=O)[C@H](CC(=O)NC(c1ccccc1)(c2ccccc2)c3ccccc3)NC(=O)OCC4c5ccccc5-c6c4cccc6)OC CK-0702 COC(=O)[C@H](Cc1c[nH]c2c1cc(cc2)O)N.Cl CK-0703 c1c2c(ncnc2Cl)n(n1)CCO CK-0704 c1cc(c(cc1C(F)(F)F)O)N CK-0705 CCOC(=O)Cc1[nH]c(=O)cc(n1)N2CCOCC2 CK-0706 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)NC(=O)CC[C@@H](C=O)NC(=O)OCC4c5ccccc5-c6c4cccc6 CK-0707 c1c(cc(c(c1Cl)C=O)Cl)O CK-0709 c1c(cc(c(c1Cl)CO)Cl)O CK-0710 c1ccc(cc1)COc2cc(c(c(c2)Cl)C=O)Cl CK-0712 CC(=O)Oc1cc(c(c(c1)Cl)C=O)Cl CK-0713 COc1cc(c(c(c1)Cl)C=O)Cl CK-0714 CC(=O)N/C(=C\c1ccc(c(c1)Br)F)/C(=O)OC CK-0717 COc1ccc2c(c1)c(ccn2)[C@@H](C3CC4CCN3CC4C=C)N.Cl.Cl.Cl CK-0720 c1cc2c(cc1C(F)(F)F)oc(n2)CCl CK-0721 COC(=O)c1cc(c([nH]1)C#N)Br CK-0723 c1cc(c(cc1C(F)(F)F)O)O CK-0724 CC(=O)NC(=Cc1ccc(cc1)OC(=O)C)C(=O)OC CK-0725 CC(=O)N/C(=C\c1c(cccc1Cl)Cl)/C(=O)OC CK-0727 CC(C)(C(=O)Nc1ccccc1C(=O)c2ccccc2)Br CK-0728 c1cc2c(cc1C(F)(F)F)oc(n2)S CK-0729 c1ccc(cc1)C(=O)c2ccccc2NC(=O)CCl CK-0730 c1cc2c(cc1[N+](=O)[O-])CCO2 CL-0049 COc1ccc(cc1)C=C CL-0053 C=Cc1c(cccc1Cl)Cl CL-0056 c1cnc(cn1)C(=N)NO CL-0076 C=CCCCC(CCCC=C)O CL-0727 CCc1ccc(cc1)F CL-0737 CCn1c(c(c(=O)n(c1=O)CC)N)N CL-0799 CCC(CC)C(=O)OC CM-0016 COc1cccc(c1)n2c(c(cn2)C#N)N CM-0749 C/[N+](=C\c1ccccc1[N+](=O)[O-])/[O-] CS-0001 C/[N+](=C\c1ccccc1Cl)/[O-] CS-0002 C/[N+](=C\c1ccc(o1)Br)/[O-] CS-0003 C/[N+](=C\c1ccc2ccccc2c1)/[O-] CS-0004 CC(C)(C)n1cc[n+](c1)C(C)(C)C.[Cl-] CS-0005 CC(c1c(c(ccc1)C(C)C)/N=C/C=N/c2c(cccc2C(C)C)C(C)C)C CS-0006 c1ccc(cc1)/C=[N+](/Cc2cccc(c2)Cl)\[O-] CS-0012 c1ccc(cc1)/C=[N+](/Cc2cccc(c2)Br)\[O-] CS-0013 c1ccc2cc(ccc2c1)CNO CS-0015 c1ccc(cc1)/C=[N+](/Cc2ccc3ccccc3c2)\[O-] CS-0016 c1ccc(cc1)/C=[N+](/Cc2ccc(cc2)Cl)\[O-] CS-0018 c1ccc2cc(ccc2c1)C/[N+](=C/c3ccncc3)/[O-] CS-0019 c1cc(cc(c1)Cl)C/[N+](=C/c2ccc(cc2)Cl)/[O-] CS-0020 c1ccc(cc1)/C=[N+](/Cc2ccc(o2)Br)\[O-] CS-0021 c1ccc(cc1)/C=[N+](/Cc2ccccc2Br)\[O-] CS-0023 c1ccc(cc1)/C=[N+](/Cc2ccccc2Cl)\[O-] CS-0024 c1ccc(cc1)CCC/[N+](=C/c2ccccc2)/[O-] CS-0026 c1ccc(cc1)C/[N+](=C/c2ccccc2)/[O-] CS-0027 c1ccc(cc1)/C=[N+](/CC2CCCCC2)\[O-] CS-0028 c1ccc(c(c1)C/[N+](=C/c2ccncc2)/[O-])Cl CS-0029 c1cc(cc(c1)Cl)C/[N+](=C/c2ccncc2)/[O-] CS-0030 c1ccc(cc1)C2C=CN(O2)Cc3ccccc3Br CS-0031 c1ccc(cc1)C2C=CN(O2)Cc3ccccc3Cl CS-0032 c1ccc(cc1)C2C=CN(O2)Cc3cccc(c3)Br CS-0033 c1ccc(cc1)CN2C=CC(O2)c3ccccc3 CS-0034 c1ccc2cc(ccc2c1)C/[N+](=C/c3ccccc3Br)/[O-] CS-0035 c1ccc(c(c1)C/[N+](=C/c2ccc(cc2)Cl)/[O-])Br CS-0036 c1ccc(c(c1)C/[N+](=C/c2ccncc2)/[O-])Br CS-0037 c1ccc(cc1)C/[N+](=C/c2ccncc2)/[O-] CS-0038 c1cnccc1/C=[N+](/CC2CCCCC2)\[O-] CS-0039 c1cc(ccc1C/[N+](=C/c2ccc(cc2)Cl)/[O-])Cl CS-0040 c1cc(cc(c1)Br)C/[N+](=C/c2ccncc2)/[O-] CS-0041 C/[N+](=C\C1CC1)/[O-] CS-0043 C/[N+](=C\c1ccc(cc1)OCC=C)/[O-] CS-0044 C/[N+](=C\c1cccc(c1)Br)/[O-] CS-0045 COc1ccc(cc1)C/[N+](=C/c2ccc(cc2)Cl)/[O-] CS-0046 c1ccc(c(c1)C/[N+](=C/c2ccc(cc2)[N+](=O)[O-])/[O-])Br CS-0048 c1cc(ccc1C/[N+](=C/c2ccc(cc2)[N+](=O)[O-])/[O-])Cl CS-0049 COc1ccc(cc1)C/[N+](=C/c2ccccc2)/[O-] CS-0051 c1ccc(cc1)NC2(CCCCC2)C(=O)N CS-10005 CC(C)(C)OC(=O)N1CCCC(C1)(Cc2ccc(cc2)Cl)C=O CS-1001 COC(=O)CCNCC(=O)OC CS-10018 CCOC(=O)CCNCC(=O)OCC CS-10019 CC(C)(C)OC(=O)N1CCCC(C1)(Cc2ccc(c(c2)Cl)Cl)C=O CS-1002 CCOC(=O)CN1CCCCC1 CS-10023 CCOC(=O)CCN1CCC(CC1)Cc2ccccc2 CS-10027 CCOC(=O)CCN1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl CS-10028 CC(C)(C)OC(=O)N1CCCC(C1)(Cc2ccc(cc2)Cl)C(=O)O CS-1003 CC(C)(C)OC(=O)N1CCCC(C1)(Cc2ccc(c(c2)Cl)Cl)C(=O)O CS-1004 CC(C)C1CC(=O)CCN1C(=O)OCc2ccccc2 CS-1006 c1ccc(cc1)C(C#N)N2CCOCC2.Cl CS-10087 CNC(C#N)c1ccccc1.Cl CS-10093 CN(C)C(C#N)c1ccccc1.Cl CS-10098 c1ccc(cc1)CNC(C#N)c2ccccc2.Cl CS-10113 c1ccc(cc1)CCNC(C#N)c2ccccc2.Cl CS-10118 CCCC(C#N)NC.Cl CS-10143 CC(C)C(C#N)N1CCCCC1.Cl CS-10144 c1ccc(cc1)C(C(=O)N)N2CCOCC2.Cl CS-10147 c1c(cnc(c1Cl)CC(=O)O)C(F)(F)F CS-10154 CC(c1c(cc(cn1)C(F)(F)F)Cl)C(=O)O CS-10155 COC(=O)C(c1c(cc(cn1)C(F)(F)F)Cl)Br CS-10161 COC(=O)C(C=O)Cl CS-10165 CCOC(=O)C(C)(C)Sc1ccc(cc1)Br CS-10172 CC(=C(C#N)C(=O)OC)C CS-10175 C/C(=C(\C#N)/C(=O)OC)/c1ccccc1 CS-10179 CC(C)(C)OC(=O)N(CCC(=O)OC)CC(=O)OC CS-10181 CC(C)(C)OC(=O)Cc1c(cc(cn1)C(F)(F)F)Cl CS-10188 CCOC(=O)Cn1cc(cc(c1=O)Cl)C(F)(F)F CS-10189 CC(=O)O.c1ccc(cc1)CN=C(N)N CS-10193 CC(=O)O.c1ccc(cc1)CC2CCN(CC2)C(=N)N CS-10200 CN(C)C(=N)N.Cl CS-10201 CCN(CC)C(=N)N.Cl CS-10202 CC(C)(C)NC(=N)N.Cl CS-10203 c1ccc(cc1)CCNC(=N)N.Cl CS-10204 C1CCN(C1)C(=N)N.Cl CS-10205 Cc1ccc(cc1)/C=C/C(=O)C CS-10217 c1ccc(c(c1)C2CC(=CC(=O)C2)O)C(F)(F)F CS-10218 c1cc(cc(c1)C(F)(F)F)C2CC(=CC(=O)C2)O CS-10220 c1cc(ccc1C2CC(=CC(=O)C2)O)Br CS-10222 c1c(cnc(c1Cl)CC(=S)N)C(F)(F)F CS-10238 c1c(cn(c(=O)c1Cl)CC(=O)N)C(F)(F)F CS-10243 COC(=N)c1ccccc1.Cl CS-10310 c1cc2c(cc1[N+](=O)[O-])nc(s2)Cl CS-10369 Cc1cc(nc2c1c(c(s2)C(=O)O)N)C CS-10372 CCOC(=O)c1c(c2c(s1)cc(cn2)C(F)(F)F)N CS-10376 c1c(cn2c(c1Cl)nnc2S)C(F)(F)F CS-10382 Cc1cc(no1)CBr CS-10406 CC(C)(C)OC(=O)N1CCN(CC1)c2cc(cc(n2)Cl)C(F)(F)F CS-10516 CNc1cc(cnc1C#N)C(F)(F)F CS-10526 c1c(cnc(c1N(CCO)CCO)C#N)C(F)(F)F CS-10529 CCOC(=O)CNc1cc(cnc1C#N)C(F)(F)F CS-10532 CN(C)c1cc(cnc1C#N)C(F)(F)F CS-10533 c1c(cnc(c1N2CCOCC2)C#N)C(F)(F)F CS-10536 c1c(cnc(c1C(=O)O)O)Br CS-10551 c1cc(ncc1CBr)C#N CS-10642 c1c(cnc(c1Cl)CBr)C(F)(F)F CS-10657 c1c(cnc(c1Cl)C(Br)Br)C(F)(F)F CS-10659 c1ccc(cc1)Sc2cc(cnc2C#N)C(F)(F)F CS-10686 c1ccc(cc1)Oc2cc(cnc2C#N)C(F)(F)F CS-10702 Cn1cc(cc(c1=O)Cl)C(F)(F)F CS-10719 Cn1cc(cc(c1=O)Br)C(F)(F)F CS-10720 c1ccc(cc1)n2c(cc(n2)C(F)(F)F)O CS-10775 CCOC(=O)C1CN1Cc2ccccc2 CS-10811 C(C1C(=O)NC(=O)S1)C(=O)O CS-10846 CCOC(=O)C1CCNC(=O)C1=O CS-10858 COC(=O)C1CC(=O)N(C1)CCc2ccccc2 CS-10864 C1=C(C(=O)NC1=O)Br CS-10874 c1cc(cc(c1)[N+](=O)[O-])c2nnc(s2)N CS-10900 Cc1csnn1 CS-10903 c1cc(ccc1c2[nH]nnn2)Cl CS-10906 c1cc(cc(c1)[N+](=O)[O-])c2[nH]nnn2 CS-10907 c1c(cc(cc1Cl)Cl)Nc2cc(nc(n2)N)Cl CS-2002 CC(C)(C)c1ccc(c(c1)/N=N/c2ccc(cc2)C(=O)O)O CS-2006 CC(=O)c1cccc(c1)Nc2cc(nc(n2)SC)Cl CS-2007 CCNc1cc(nc(n1)N)Cl CS-2009 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3C(=O)c4ccccc4S3(=O)=O CS-2016 c1cc2ccc3cc([nH]c3c2nc1)C(=O)O CS-2017 CSc1nc(cc(n1)Cl)N2CCN(CC2)c3ccccc3 CS-2019 CC(=O)c1ccc(c(c1)[N+](=O)[O-])Cl CS-2021 c1cc(c(cc1Cl)Cl)Nc2cc(nc(n2)N)Cl CS-2027 COc1ccc2c(c1)[nH]c(n2)Sc3ccc(cn3)[N+](=O)[O-] CS-2028 c1c(cc(c(c1Br)O)Br)c2csc(n2)N CS-2036 CC(c1ccccc1)Nc2cc(nc(n2)N)Cl CS-2037 CCNc1ccncc1[N+](=O)[O-] CS-2042 CN(C)CCNC1=C(C(=O)c2ccccc2C1=O)Cl.Cl CS-2045 c1ccc(cc1)c2ccc(cc2)C(=O)Nc3ccccc3F CS-2062 CSc1nc(cc(n1)Cl)NCCc2ccccc2 CS-2072 Cc1cc(no1)C(=O)CBr CS-4004 Cc1ccc(o1)C(=O)CBr CS-4005 c1ccc2c(c1)cc(cn2)CCl CS-4006 c1ccc(cc1)S(=O)(=O)c2cc3cccc(c3nc2)N CS-4007 CC(C)(C)OC(=O)N1CCC(CC1)OC2CCNCC2 CS-4009 c1c2c(cc(c1F)O)C(=O)CC2 CS-4014 COc1ccc(nc1[N+](=O)[O-])Br CS-4015 COC(=O)c1ccc2c(c1)cc(o2)CCO CS-4016 c1cc2c(cc1F)NCC2 CS-4017 c1cc2c(cc1C=O)CCN(C2)C(=O)C(F)(F)F CS-4018 CC(C)(C)OC(=O)N1CCc2cc(c(cc2C1)N)OC CS-4019 c1cc2c(cc1I)[nH]c(=O)[nH]2 CS-4020 COC(=O)c1c[nH]c2c1c(ccc2)I CS-4023 Cc1nc(on1)c2ccc(cc2)Br CS-4024 Cc1nccn1c2ccc(cc2)I CS-4025 C[C@H]1CNCCN1C(C)C.Cl.Cl CS-4026 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)CCC3=O CS-4027 C[C@@H]1CNC[C@@H](N1C(=O)OC(C)(C)C)C CS-4028 Cc1nc(on1)c2ccc(cn2)Br CS-4030 Cn1c(ncn1)CCl.Cl CS-4031 C1CC(C1)N2CCNCC2.Cl.Cl CS-4033 CC(C)(C)OC(=O)N1CCC(CC1)N2CCc3c2ccc(c3)Br CS-4034 CC(=O)c1cc(c(cc1O)Cl)F CS-4040 Cc1c(ccc(n1)c2ccc(cc2)F)C(=O)O CS-4041 CC(C)(C)OC(=O)N1CCN(CC1)c2cccc(c2)C(=O)O CS-4044 CC1(CC(=O)c2ccccc2O1)C CS-4045 COc1c(ccc(c1C=O)F)Br CS-4046 COc1ccc(c(c1F)C(=O)O)Br CS-4048 c1cc(c(c(c1F)C(=O)O)F)Br CS-4049 c1cc(c(c(c1)C(=O)O)F)C#N CS-4050 c1cc(c2cn[nH]c2c1)C#N CS-4051 c1cc(c(c(c1C#N)F)Br)F CS-4053 c1cc(c(c(c1C(=O)O)F)Br)F CS-4054 c1cc2cc(cnc2c(c1)Br)I CS-4055 Cc1cc(n2c(n1)nc(n2)CO)C CS-4057 Cc1nc(on1)c2ccc(cc2F)Br CS-4058 c1cc(ccc1S(=O)(=O)Nc2cc(ccc2F)F)Cl CS-4059 c1cc(ccc1c2ncco2)Br CS-4060 Cc1nc(no1)c2ccc(cc2)Br CS-4061 c1cc(c(c(c1)O)Cl)C(=O)O CS-4062 c1cc2cc(cc(c2nc1)Br)F CS-4063 c1cc2c(ccc(c2nc1)Br)F CS-4064 c1cc2cc(cc(c2nc1)[N+](=O)[O-])F CS-4065 Cc1c(ccc(n1)Cl)C#N CS-4066 Cc1cc2cccnc2c(c1)Br CS-4067 c1c[nH]c2c1cc(nc2)Cl CS-4078 C1CC1CN2CCNCC2.Cl.Cl CS-4080 c1ccc(cc1)CN2CCc3c(ccc(n3)Cl)C2 CS-4081 COC(=O)c1c(ccc(c1F)Br)F CS-4082 Cc1cc2cc(ccc2[nH]1)CN CS-4083 C[C@H]1CNCCN1C2CCC2.Cl.Cl CS-4084 Cc1nc(c(s1)c2ccc(cc2)F)C(=O)O CS-4086 c1c(c(nc(n1)N)N)Cl CS-4090 c1cc2c(cc1F)cc(o2)CO CS-4099 c1ccc(c(c1)COc2ccc(cc2)Br)F CS-4100 COc1ccc2c(n1)c(c(cn2)F)Br CS-4103 c1cc2c(cc1Br)C[C@H](C2)N.Cl CS-4104 c1cc2c(cc1Br)C[C@@H](C2)N.Cl CS-4105 c1c[nH]c2c1c(ncc2Br)Br CS-4106 Cc1c(ccc2c1[nH]c(=O)cc2)I CS-4107 Cc1ccc(c(n1)N)C=O CS-4110 C=CC(c1ccccc1)N.Cl CS-4112 COc1ccc(nc1N)Br CS-4115 Cc1c(c(nc(n1)C)N)C=O CS-4116 C1CCC(C1)CBr CS-4118 Cc1ccc2c(c1)c(no2)N CS-4119 c1cc(c(cc1C#N)F)C#N CS-4120 COC(=O)c1ccc(c(c1)F)N2CCNC2=O CS-4121 CC(C)(C)OC(=O)N1CCc2c(sc(n2)Br)C1 CS-4124 c1cc2c(cc1C3(CC3)C(=O)O)OCO2 CS-4125 COc1cc(ccc1Cl)CC#N CS-4126 COc1ccc2cnc(nc2c1)Cl CS-4128 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2ncnc3I CS-4130 Cc1cc2c(cccc2N)cn1 CS-4131 c1cc2cc(cnc2c(c1)Cl)I CS-4134 c1cc2cc(cnc2c(c1)[N+](=O)[O-])Br CS-4135 c1cc2cc(cnc2c(c1)N)Br CS-4136 Cc1cn(cn1)c2ccc(cc2OC)Br CS-4137 Cc1cn(cn1)c2ccc(cc2)Br CS-4138 CC(C)(c1cccc(c1)Br)C(=O)O CS-4143 c1ccc(cc1)C2(CC2)C=O CS-4145 c1c(c(nc(n1)N)N)Br CS-4147 CNc1cccc(c1)CO CS-4148 CC(C)c1cc(c(cc1O)I)OC CS-4149 c1cc(c(c2c1cc[nH]2)Cl)C(=O)O CS-4150 c1c(c(cc(c1[N+](=O)[O-])O)F)C#N CS-4151 Cc1ccc(c(c1N)C)Br CS-4152 c1cc(nc2c1CC(CC2)C(=O)O)C(F)(F)F CS-4153 COc1ccc(cc1C(=O)O)C(=O)OC CS-4160 Cn1cc(cn1)c2cccc(c2)N CS-4161 COc1cc(c(cc1[N+](=O)[O-])F)Br CS-4162 Cc1c(ccc(c1OC)Br)C(=O)O CS-4166 c1c(c(c(c(c1F)N)Br)F)C#N CS-4168 c1cc(c(cc1[N+](=O)[O-])C(F)(F)F)C=O CS-4169 COC(=O)c1cccc(c1Cl)[N+](=O)[O-] CS-4172 c1ccc(cc1)COc2coc(cc2=O)C(=O)O CS-4175 c1c(cnc(c1C#N)Cl)F CS-4176 c1cc2c(cc1Br)cns2 CS-4178 Cc1cc(c(cc1Cl)F)I CS-4179 CC(C)Cc1ncc(s1)Br CS-4180 CCOc1cc(ccc1N)C(=O)N CS-4182 COc1cc(c(cc1F)Br)C(=O)O CS-4186 c1c(c(cnc1Br)Cl)C(=O)O CS-4188 CC(C)(C)OC(=O)N1CCc2c(ccc(n2)Cl)C1=O CS-4192 c1cc(nc2c1C(=O)NCC2)Cl CS-4193 CC(C)(C)NS(=O)(=O)c1cc(cnc1)Br CS-4195 COC(=O)c1ccc(c2c1[nH]cc2)Br CS-4197 c1ccc2c(c1)c(c[nH]2)C(=O)CN.Cl CS-4198 c1c(c(cnc1Cl)N)Cl CS-4199 c1cc2c(cc1Br)C(=O)CCCN2 CS-4201 c1cc(nc(c1O)[N+](=O)[O-])Br CS-4206 Cc1cc(c(cc1Br)F)O CS-4212 COC(=O)c1cccc(c1F)Br CS-4213 COc1cc(ccc1Cl)CBr CS-4220 COc1ccc(c(c1)N)C=O CS-4221 c1cc2cc(cnc2c(c1)[N+](=O)[O-])Cl CS-4222 c1cc2cc(cnc2c(c1)N)Cl CS-4223 c1c(cc(cc1C(F)(F)F)Cl)CO CS-4224 COC(=O)c1cc(cc(c1)N)CO CS-4225 c1cc(c(cc1F)I)[N+](=O)[O-] CS-4226 CS(=O)(=O)Nc1ccc(c(c1)C#N)Br CS-4230 c1cc2cc(cnc2c(c1)F)I CS-4233 COc1ccc(c(c1)O)[N+](=O)[O-] CS-4236 c1c2c(c(c(c1Br)Br)C(=O)O)OCCO2 CS-4238 COc1ccc(c(c1)Oc2cnc(nc2N)N)Br CS-4239 c1cc(c(cc1F)Br)Oc2cnc(nc2N)N CS-4243 CC(C)(C)OC(=O)N1Cc2ccc(cc2C1)C(=O)O CS-4247 c1ccc(c(c1)COc2cccc(c2)[C@@H]3CCC[C@H]3NCC(=O)N)F CS-4250 CC(C)(C)OC(=O)N1CCC(CC1)Oc2cc[n+](cc2)Cc3ccccc3.[Br-] CS-4251 CC(C)(C)OC(=O)N1CCC(CC1)Oc2ccncc2 CS-4252 c1cc(c(cc1OC2CCNCC2)Cl)C#N.Cl CS-4253 c1ccc(c(c1)COc2ccc(cc2)[C@@H]3CCC[C@@H]3NCC(=O)N)F CS-4255 CC(=O)N1CC(c2c1cccc2)(C)C CS-4256 CN(C)C=C(C#N)Oc1cc(ccc1Br)F CS-4259 c1cc(c(cc1F)Oc2cnc(nc2N)N)Br CS-4260 CC(C)(C)OC(=O)c1ccc(cn1)Br CS-4261 CC(C)(C)OC(=O)N1CCc2ccc(cc2CC1)[N+](=O)[O-] CS-4264 CC(C)(C)OC(=O)N1CCc2ccc(cc2CC1)N CS-4265 CC(=O)Nc1c(cc(c2c1C=CCO2)C(=O)OC)Cl CS-4266 COc1ccc(cc1)[C@@H]2CCC[C@H]2O CS-4267 CC(C)(C)OC(=O)N[C@H]1CCC[C@@H]1O CS-4268 CC(=O)Nc1cc(c(cc1Cl)C(=O)OC)OCC#C CS-4271 CC(C)(CC(=O)OC)c1ccc(cc1)OC CS-4272 c1c(c2c(c(c1Br)N)CCCO2)C(=O)O CS-4274 CC(=O)Nc1c(cc(c2c1CCCO2)C(=O)OC)Br CS-4275 C[C@@H]1CN(C[C@@H](N1)C)c2ccc(c(n2)NS(=O)(=O)c3ccc(c(c3)F)Br)OC CS-4279 c1cc(ccc1S(=O)(=O)Cc2cc(ccc2F)F)Cl CS-4282 CC(C)(C)OC(=O)N1CC[C@H](C1)OC2CCNCC2 CS-4286 c1cc2c(cc1C#N)CCC2O CS-4288 COc1cc(cc(c1N)C(=O)O)Br CS-4291 c1c(cc(c(c1F)N)I)I CS-4292 c1cc(ncc1Br)NC(=S)NC(=O)O CS-4293 COC(=O)c1cccc(c1[N+](=O)[O-])O CS-4294 Cn1ccc(n1)c2cccc3c2ccc(c3)C(=O)O CS-4295 c1c(c(c[n+](c1Br)[O-])Br)[N+](=O)[O-] CS-4299 COc1cc(ccc1NC(=O)C(F)(F)F)Br CS-4300 c1cc(nc2c1CNCC2)Cl.Cl CS-4303 CC(C)(C)OC(=O)N1CCc2c(ccc(n2)Cl)C1 CS-4304 CC(C)(C)OC(=O)N1CCc2c(ccc(c2[N+](=O)[O-])OC)C1 CS-4307 Cc1ccc(cc1)S(=O)(=O)Oc2cc(c(cc2C(C)C)OC)I CS-4308 COc1ccc(cc1C=O)C(=O)OC CS-4309 Cc1ccc(c(c1[N+](=O)[O-])C)Br CS-4310 CNN=Cc1c(cc(cc1F)F)F CS-4312 c1ccc(cc1)S(=O)(=O)c2cc3cccc(c3nc2)[N+](=O)[O-] CS-4313 c1c(cc(cc1[N+](=O)[O-])Br)[N+](=O)[O-] CS-4314 COC(=O)c1ccc(c(c1F)Br)F CS-4315 COc1ccc2c(c1)CCNC2.Cl CS-4316 c1c(cc(c(c1Cl)O)Br)Br CS-4317 COc1cc2c(cc1F)CCC2=O CS-4319 c1cc2c(cc1Br)CC(C2)N.Br CS-4320 CC(C)(C)OC(=O)N1CCc2cc(c(cc2C1)[N+](=O)[O-])OC CS-4326 Cc1c(ccc(c1C(=O)OC)Br)O CS-4328 c1cc(ncc1Br)C(F)(F)F CS-4330 c1ccc(cc1)C2(CCCC2)CO CS-4332 c1cc(c(c(c1)O)Br)[N+](=O)[O-] CS-4333 CN(C)c1c(ccc(c1C=O)F)C#N CS-4336 CC(C)(C)Oc1ccc(cc1)C[C@@H](C(=O)O)N(C)C(=O)OCc2ccccc2 CS-4339 c1cc(c(cc1C(=O)O)Br)O CS-4340 CC(=O)c1ccc2c(c1)CCN(CC2)C(=O)OC(C)(C)C CS-4341 c1cc2c(cc1O)CCNC2.Br CS-4343 c1cc(c(c(c1C#N)F)C(=O)O)F CS-4344 Cc1ncc(c(n1)N)C#N CS-4345 c1ccc(cc1)CN2C3CCC2CC(=O)C3.Cl CS-4347 C1CC(C1)N2CCN(CC2)C(=O)C3CCNCC3 CS-4348 Cc1cccc(n1)NC(=O)C(C)(C)C CS-4349 C[C@H]1CN(CCN1)C(=O)OCc2ccccc2 CS-4350 COC(=O)c1ccc(c(c1)I)O CS-4351 C1CCN(CC1)CCCC(=O)O.Cl CS-4355 c1cc(ccc1C(=O)N2CCNCC2)OCCCN3CCCCC3.Cl.Cl CS-4359 c1ccc(cc1)CN2CCC3=C(C2)CCC(=O)N3 CS-4360 COc1cc(cc2c1nc(nc2)Cl)Br CS-4364 COC(=O)C1Cc2ccccc2CN1.Cl CS-4365 C1CC(C1)N2CCC(CC2)C(=O)O CS-4366 C1CC(C1)N2CCCN(CC2)C(=O)C3CCNCC3 CS-4368 COc1ccc(cc1)C23CC2C(=O)NC3=O CS-4369 c1cc(ncc1N2CCC(CC2)C(=O)O)C(F)(F)F CS-4371 c1cc2c(cc1Br)CCN2C3CCN(CC3)C4CCC4 CS-4372 CN1C(=O)[C@H]2[C@H](N3CCc4c5ccccc5[nH]c4[C@H]3[C@H]2C1=O)c6ccccc6 CS-4373 Cn1c2cc(c(c(c2cn1)F)C=O)F CS-4374 CC(C)(C)c1ccc(c(c1)Br)C(=O)O CS-4375 c1cc2c(cc1O)CCNC2 CS-4376 c1cc(c(nc1)ON)C(F)(F)F CS-4379 COC(=O)/C=C/c1cccnc1Br CS-4380 c1ccc(cc1)COc2c3ccccc3c(cc2I)Cl CS-4382 c1cn2c(n1)C(CC2)O CS-4383 c1ccc2c(c1)nc(o2)c3cccc(c3)F CS-4385 c1ccc(cc1)COc2c(cc(c3c2nccc3)I)I CS-4386 CN1c2ccccc2/C(=C/c3ccccc3I)/C1=O CS-4387 c1cc(c(nc1)Br)/C=C/C#N CS-4388 c1ccc(cc1)NNC(=O)C(F)(F)F CS-4389 c1ccc(c(c1)/C=C\2/c3ccccc3NC2=O)I CS-4390 CN1CCN(CC1)C(=O)/C=C/c2ccccc2I CS-4391 CN1C(=O)C(=Cc2ccccc2I)C(=O)N(C1=O)C CS-4393 c1ccc(c(c1)/C=C/C(=O)O)I CS-4394 COC(=O)C#CCO CS-4395 C1C(O1)C(=O)[O-].[K+] CS-4397 COc1cc(cc(c1)Br)[N+](=O)[O-] CS-4400 c1ccc(cc1)P(=O)(c2ccccc2)N CS-4401 c1cc2cc(cnc2c(c1)I)Br CS-4404 COC(=O)c1ccc(c(c1)F)C#N CS-4406 c1cc(c(c(c1C#N)F)C=O)F CS-4410 c1c(nc(cn1)Cl)CC(=O)O CS-4411 c1c(c(cnc1Cl)F)C(=O)O CS-4413 c1cc2c(cc1I)nc(o2)S CS-4417 Cc1ccc2cccnc2c1Br CS-4418 CC(C)(C)OC(=O)NN=C1CCOC1 CS-4421 COc1ccc2c(c1)OCC(=O)N2O CS-4422 COc1ccc2c(c1)c(c(cn2)N)Br CS-4423 Cc1c(ccc2c1nc(cn2)OC)F CS-4424 COc1ccc2c(n1)c(=O)cc[nH]2 CS-4425 COc1ccc2c(n1)c(c(cn2)N)Br CS-4426 COc1cc2c(c(c1)F)ncc(c2Br)N CS-4428 c1cc(nc2c1OCC(=O)N2)Br CS-4429 COc1ccc2c(n1)c(c(cn2)F)O CS-4430 c1cc2c(nc1C=O)NC(=O)CS2 CS-4431 c1ccc(c(c1)C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F DA-0024 CC(C)(C)OC(=O)N1C(=O)C=CC1=O DA-0025 c1cc2cc(ncn2c1)C(=O)O.O.Cl DA-0600 COC(=O)c1ccc(cc1O)Br DA-0608 c1cc(c(nc1)S)C(F)(F)F DA-0609 c1ccc2c(c1)nc(s2)c3ccc(nc3)O DA-0611 COc1ccc(cc1O)C(=O)OC DA-0613 c1ccc(c(c1)c2ccc(cn2)C(F)(F)F)C(=O)O DA-0700 c1ccc(c(c1)c2ccc(cc2)[N+](=O)[O-])C(=O)O DA-0701 Cc1c(nc(s1)N)c2cccs2 DA-0703 CCc1c(nc2nc(nn2c1C)N)C DA-0704 c1ccc(cc1)n2cc(nn2)CCl DA-0705 c1ccc(cc1)c2c(nc(s2)c3cccc(c3)C(F)(F)F)O DA-0706 c1ccc(cc1)c2c(nc(s2)c3ccc(cc3)Cl)O DA-0708 c1ccc(cc1)c2c(nc(s2)N)O DA-0709 CCOC(=O)c1c(nc(s1)c2cccc(c2)C(F)(F)F)O DA-0710 CCOC(=O)c1c(nc(s1)c2ccccc2)O DA-0712 c1cc(ccc1Oc2ccc(cn2)C(F)(F)F)S(=O)(=O)Cl DA-0718 Cc1c(nc(s1)c2ccc(cc2)Cl)CC(=O)O DA-0720 CCOC(=O)c1c(nc(s1)c2ccc(cc2)C(F)(F)F)O DA-0721 CCOC(=O)c1c(nc(s1)c2ccc(c(c2)OC)OC)O DA-0722 CCOC(=O)c1c(nc(s1)c2cccs2)O DA-0723 CCOC(=O)c1c(nc(s1)c2ccc(cc2)OC)O DA-0724 CC(=O)NC(CSc1ccc(cc1)Br)C(=O)O DA-0725 c1cc(ccc1NC(=O)NCCCl)Br DA-0802 COC(=O)Cc1ccc2c(c1)nc(o2)CCl DA-0807 c1ccc(cc1)c2cc3nccc(n3n2)c4c(cc(cn4)C(F)(F)F)Cl DA-0810 c1c(cc(c(c1Cl)Oc2c(cc(cn2)C(F)(F)F)Cl)Cl)N DA-0811 c1cc(ncc1CN2C(=O)CCC2=O)Cl DA-0812 c1cc2c(cc1CC(=O)NN)nco2 DA-0813 c1cc(ccc1N2CCNC2=O)Br DA-0815 c1ccc(cc1)CN2CCN(CC2)C(=O)c3c(cccn3)C(F)(F)F DA-0816 CCOC(=O)c1cc(c(nc1Cl)C)C#N DA-0819 c1cc(cnc1)C(=O)CC#N DA-0820 c1cc2c(cc1CN3CCC(CC3)C(=O)O)CCO2 DA-0822 COC(=O)c1cccn2c1nc(c2)c3ccc(cc3)Br DA-0824 c1cc(cc(c1)C(F)(F)F)C(=O)CC#N DA-0827 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F DA-0830 c1cc(ccc1C(=O)CC#N)C(F)(F)F DA-0831 c1cc(ccc1c2cc3nccc(n3n2)c4c(cc(cn4)C(F)(F)F)Cl)Cl DA-0832 c1cc(ncc1CN2C(=O)CCC2=O)N3CCOCC3 DA-0834 Cc1cc(cc(c1N)C(=O)NN)Br DA-0835 c1ccc2c(c1)nc(o2)C3CCN(CC3)CCC(=O)O DA-0836 c1cc(c2nc(cn2c1)c3ccc(cc3)Br)C(=O)NN DA-0837 c1cc2c(cc1S(=O)(=O)Cl)CCO2 DA-0838 CC(C)(C)OC(=O)N1CCN(CC1)c2cccc(c2)C#N DA-0839 c1cc(cc(c1)C(F)(F)F)c2cc(on2)N DA-0841 c1cc(cc(c1)C(F)(F)F)c2cc([nH]n2)N DA-0842 c1ccc(c(c1)S(=O)(=O)NNC(=O)c2cc(nc(c2)C(F)(F)F)C(F)(F)F)Cl DA-0843 CN(C)/C=C/C(=O)c1ccc(cn1)C(F)(F)F DA-0844 CSc1nc2nccc(n2n1)c3ccc(cn3)C(F)(F)F DA-0847 c1ccnc(c1)C(=O)CC#N DA-0848 c1cc(ccc1c2cc(on2)N)C(F)(F)F DA-0854 c1cc(ccc1N2CCNC2=O)[N+](=O)[O-] DA-0855 c1cc(ccc1c2cc([nH]n2)N)C(F)(F)F DA-0856 c1cc(c2nc(cn2c1)c3ccc(cc3)Br)C(=O)O DA-0860 CC(C)(C)OC(=O)N1CCN(CC1)CCc2cccc(c2)c3ccn[nH]3 DA-0861 c1cc2c(cc1S(=O)(=O)N)CCO2 DA-0862 Cc1cc(cc2c1ncn(c2=O)N)Br DA-0867 Cc1c(cccc1[N+](=O)[O-])c2nnco2 DA-0868 c1ccc2c(c1)c(c([nH]2)C(=O)NN)Br DA-0869 c1ccc2c(c1)c(c([nH]2)C(=O)NCCCO)Br DA-0871 CNC(=O)c1cccc(c1)c2ccc(cn2)C(F)(F)F DA-0873 c1ccc(cc1)CN2C[C@@H]3[C@H](C2)C(=O)N(C3=O)c4ccccc4 DA-0875 COC(=O)Cc1ccc2c(c1)nc(o2)CN3CCC(CC3)Cc4ccccc4 DA-0876 CC(C)(C)OC(=O)NCCCN DA-0878 CCOC(=O)c1cc(c(nc1N2CCN(CC2)CCO)C)C#N DA-0879 CCOC(=O)c1ccc2c(c1)sc(n2)C DA-0920 CC1=NS(=O)(=O)NC(=C1)C(=O)O DA-0921 Cc1nc2ccc(cc2s1)C(=O)O DA-0922 c1cc2c(ccc(=O)[nH]2)c(c1)O DA-0923 c1cc2c(cc1C(=O)O)NC(=O)CS2 DA-0924 c1cc2c(cc1C(=O)NN)sc(n2)NN DA-0925 c1cc2c(cc1C(=O)O)sc(n2)O DA-0926 c1c(cc(nc1NN)Cl)C(F)(F)F DA-5014 c1cc(c(cc1C#N)Cl)N2CCNCC2 DA-7004 CC(C)(C)OC(=O)NC(c1cccs1)S(=O)(=O)c2ccccc2 DB-0031 CN(C)C(=O)c1ccc(c(c1)[N+](=O)[O-])n2cccn2 DB-0099 CC(=O)c1cccnc1Cl DB-0602 Cc1c2cccnc2[nH]n1 DB-0603 CCOC(=O)c1ccc(c(c1)F)C#N DB-0604 c1cc(c(cc1CO)F)C#N DB-0605 CC(=O)c1ccc(nc1)Cl DB-0607 c1cc(c(cc1C=O)F)C#N DB-0608 CC(=O)c1ccc2nnnn2c1 DB-0609 CCNc1cc(ccc1[N+](=O)[O-])C(=O)OC DB-0700 Cc1ccc(cc1)Cn2cc(ccc2=O)C=O DB-0701 c1cc(c(cc1Cn2cc(ccc2=O)C=O)Cl)Cl DB-0702 c1cc(cc(c1)C(F)(F)F)Cn2cc(ccc2=O)C=O DB-0704 CCc1ccc(cc1)Nc2ncc(s2)C(=O)C DB-0711 CC(=O)c1cnc(s1)Nc2cc(ccc2OC)OC DB-0712 Cc1c(sc(n1)Nc2cc(ccc2OC)OC)C(=O)C DB-0714 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C=O DB-0719 Cc1c(sc(n1)Nc2cccnc2)C(=O)C DB-0720 CC(=O)c1cnc(s1)Nc2cccnc2 DB-0721 c1cc2c(cc1S(=O)(=O)Cl)CCC2 DB-0800 Cc1c2c(cc(nc2n(n1)C)N3CCNCC3)C(F)(F)F DB-0810 c1c(cnc(c1Cl)C(=N)N)C(F)(F)F.Cl DB-0812 CNC1CCN(CC1)Cc2ccccc2 DB-0816 Cc1ccc(cc1C(=O)O)S(=O)(=O)Cl DB-0820 c1ccc(cc1)S(=O)(=O)N(c2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)S(=O)(=O)c4ccccc4 DB-5006 c1cnc(nc1C(=O)OCC2CC2)c3c(cc(cn3)C(F)(F)F)Cl DC-0018 c1ccc(cc1)OC(=O)c2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl DC-0022 C=CCc1c(=O)[nH]cnc1O DC-0032 C[C@@H](C(=O)OC)Nc1c(cc(cn1)C(F)(F)F)Cl DC-0203 c1c(cnc(c1Cl)N2CCC3(CC2)NCCS3)C(F)(F)F.Cl.Cl DC-0204 c1ccc(cc1)CN2CC(C(C2)c3ccccc3O)CO DC-0205 CC(C(=O)NN)Nc1c(cc(cn1)C(F)(F)F)Cl DC-0207 c1cc(cc(c1)Br)c2c(c[nH]n2)N DC-0604 c1cc(cc(c1)Br)c2c(c[nH]n2)C#N DC-0605 c1cc(nc(c1)Cl)CO DC-0607 c1cc(nc(c1)Cl)n2c(c(cn2)C#N)N DC-0700 c1c(cnc(c1Cl)n2c(c(cn2)C#N)N)C(F)(F)F DC-0706 CCOC(=O)c1cc2ccc(cc2[nH]1)Br DC-0707 CCOC(=O)c1c(nc2n1cccc2N)C DC-0710 c1c(cnc(c1I)N)[N+](=O)[O-] DC-0717 Cc1c(sc(n1)Cc2ccc(cc2)Cl)C(=O)O DC-0718 c1cc(ccc1c2ccc(cn2)C(F)(F)F)C(=S)N3CCCCC3 DC-0719 c1cc2cn[nH]c2c(c1)Br DC-0720 CCOC(=O)c1c(nc2n1ccc(c2)C)C(F)(F)F DC-0721 c1c(cnc(c1N)N)I DC-0722 c1c(cnc(c1Cl)C(=O)NN)C(F)(F)F DC-0725 c1c(cnc(c1Cl)C(=O)O)C(F)(F)F DC-0726 Cc1cccn2c1nc(c2C(=O)O)C DC-0729 c1c(cnc(c1Cl)CO)C(F)(F)F DC-0730 c1cc(ccc1C(=O)/C=C/c2cc(ccc2N3CCC(CC3)C(F)(F)F)[N+](=O)[O-])Cl DC-0732 c1cc(ccc1S(=O)(=O)NCCCN2CCCC2)Cl DC-0735 c1ccc(c(c1)S(=O)(=O)NCCCN2CCCC2)Cl DC-0736 COC(=O)C1(CCC1)CN.Cl DC-0800 C1CC(C1)(C#N)C(=O)O DC-0801 COC(=O)c1ccc2c(c1)[nH]c(=O)[nH]2 DC-0805 COC(=O)C1(CC1)C#N DC-0807 c1cc(ccc1CCC2CNCCN2)C(F)(F)F DC-0809 c1c(cnc2c1c(c[nH]2)[N+](=O)[O-])Cl DC-0810 c1ccc(c(c1)N2CCN(CC2)C(=O)c3ccc(cc3)OCCN4CCC(CC4)C(F)(F)F)Cl DC-0812 CCOC(=O)c1cn2cc(cc(c2n1)I)Cl DC-0813 COC(=O)C1(CCCC1)CN.Cl DC-0815 c1c(cnc(c1C(F)(F)F)N)Br DC-0818 CC(C)(C#N)C(=O)OC DC-0819 c1ccn2c(c1)nc(c2I)C(=O)O DC-0820 COC(=O)C1(CC1)CN.Cl DC-0821 c1cc(ncc1C(=O)O)N2CCC(CC2)C(F)(F)F DC-0823 CC(C)(CN)C(=O)OC.Cl DC-0826 c1cc(c(cc1[N+](=O)[O-])C=O)N2CCC(CC2)C(F)(F)F DC-0827 c1cc(c(cc1[N+](=O)[O-])C=O)N2CCC(CC2)CO DC-0828 c1ccc(c(c1)NC(=O)c2ccc(nc2)N3CCC(CC3)C(F)(F)F)Cl DC-0829 c1ccc(c(c1)CNC(=O)c2ccc(nc2)N3CCC(CC3)C(F)(F)F)Cl DC-0832 c1cc(ccc1N2CCN(CC2)C(=O)c3ccc(nc3)N4CCC(CC4)C(F)(F)F)Cl DC-0833 CC(C)(C#N)C(=O)O DC-0839 COC(=O)C1(CCCCC1)C#N DC-0840 c1c(cnc(c1Cl)CNC(=O)[C@@H]2CCC[NH2+]2)C(F)(F)F.[Cl-] DD-0001 c1c(cnc(c1Cl)CN\2CCN/C2=N/[N+](=O)[O-])C(F)(F)F DD-0003 CS(=O)(=O)N1CCC[C@H]1C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl DD-0011 c1cc(ccc1S(=O)(=O)N2CCC[C@H]2C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)Cl DD-0012 CC(=O)N1CCC[C@H]1C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl DD-0013 COC(=O)c1cc(ccc1[N+](=O)[O-])N2CCN(CC2)c3ccc(cn3)C(F)(F)F DD-0017 COC(=O)c1cc(ccc1[N+](=O)[O-])N2CCC(CC2)C(F)(F)F DD-0020 CC(C)N1C(=O)C2(CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)NC1=O DD-0023 c1cc(ccc1[C@H]2N(CCS2)C(=O)c3ccc(cc3)Cl)OCc4c(cc(cn4)C(F)(F)F)Cl DD-0042 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)C2CC2C(=O)O DD-0044 CCOC(=O)C1CCCN(C1)c2ccc(cc2C(F)(F)F)[N+](=O)[O-] DD-0045 CCOC(=O)c1c(c2cc(ccc2[nH]1)Cl)C(F)(F)F DD-0047 c1ccc(cc1)CNC(=O)C2CC2C(=O)O DD-0051 c1cc(c(cc1[N+](=O)[O-])C(F)(F)F)N2CCCC(C2)C(=O)O DD-0052 CN(C(=O)C1CCCN(C1)c2ccc(cc2C(F)(F)F)[N+](=O)[O-])OC DD-0056 COc1cc(c(cc1C(F)(F)F)[N+](=O)[O-])CC#N DD-0057 c1cnn(c1)c2ccc(cc2C(F)(F)F)[N+](=O)[O-] DD-0060 c1c(cnc(c1Cl)Cn2c(=O)c(c(cn2)Cl)Cl)C(F)(F)F DD-0061 c1cc(ccc1CN2C(=O)C3(CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)N(C2=O)Cc5ccc(cc5)Cl)Cl DD-0067 CCOC(=O)C1=Cc2ccccc2OC1C(F)(F)F DD-0210 c1nc(c(c(n1)O)Br)C(F)(F)F DD-0212 c1cc2nc(cn2cc1Br)C(F)(F)F DD-0214 CCOC(=O)C1=Cc2cc(ccc2OC1C(F)(F)F)Cl DD-0219 CCOC(=O)C1=Cc2cc(ccc2OC1C(F)(F)F)Br DD-0220 CC(=O)CCCN1C(=O)c2ccccc2C1=O DD-0234 CCOC(=O)C1CNc2cc(ccc2O1)C DD-0236 CCOC(=O)C1=Cc2cc(cc(c2OC1C(F)(F)F)Cl)Cl DD-0238 c1c(c(c(c(n1)Cl)Cl)I)C(F)(F)F DD-0700 CNc1c(cc(cn1)[N+](=O)[O-])Cl DD-0701 CCNc1c(cc(cn1)[N+](=O)[O-])Cl DD-0702 c1c(cnc(c1Cl)NCCO)[N+](=O)[O-] DD-0703 c1c(cnc(c1Cl)S)[N+](=O)[O-] DD-0704 COC(=O)c1ccc2c(c1)N(CCO2)S(=O)(=O)C DD-0705 CC(C)(C)OC(=O)N1CCOc2c1cc(cc2)C(=O)OC DD-0706 CN1CCOc2c1cc(cc2)C(=O)OC DD-0707 c1ccc2c(c1)CC(C(=O)N2)N.Cl DD-0708 CC(=O)Nc1c(cc(s1)Br)C(=O)O DD-0709 c1c(n[nH]c1N)C(=O)O DD-0710 COC(=O)c1cc([nH]n1)N DD-0712 c1cc2c(cc1Cl)NCCO2 DD-0714 c1c(c(cc(c1F)[N+](=O)[O-])F)CO DD-0715 c1c(c(c(c(n1)Cl)Cl)CO)C(F)(F)F DD-0716 c1c(n[nH]c1[N+](=O)[O-])C(=O)NN DD-0719 c1cc2c(cc1CO)NCCO2 DD-0721 Cn1c2ccccc2c(c(c1=O)N)O.Cl DD-0722 COC(=O)c1ccnc(c1Cl)Cl DD-0723 c1c(c(cc(c1F)[N+](=O)[O-])F)C=O DD-0725 c1c(n[nH]c1[N+](=O)[O-])CO DD-0726 C[N+]1(CCOc2c1cc(cc2)C(=O)OC)C.[I-] DD-0727 COc1c(cc(cn1)C(=O)OC)Cl DD-0729 c1cc(c(cc1[N+](=O)[O-])N2CCNCC2)C#N DD-0731 c1c(cnc2c1COC(=O)N2)Br DD-0732 CCOC(=O)c1cc([nH]n1)[N+](=O)[O-] DD-0733 c1cnc(c(c1I)Cl)Cl DD-0734 c1cc2c(c(c1)Cl)[nH]nc2Br DD-0735 COC(=O)c1ccc(cc1)c2ccnc(c2Cl)Cl DD-0736 CN1CCOc2c1cc(cc2)C(=O)NN DD-0737 CN1CCOc2c1cc(cc2)C(=O)O DD-0738 c1cc(ccc1CO)c2cnco2 DD-0740 COC(=O)c1c(cnc(n1)S(=O)(=O)C)Br DD-0741 CS(=O)(=O)c1ncc(c(n1)C(=O)O)Br DD-0742 c1cc2c(c(c1)[N+](=O)[O-])c(n[nH]2)Br DD-0744 Cc1cc2c(cc1[N+](=O)[O-])cnn2C(=O)C DD-0747 Cn1c(nc(c1Br)Br)CO DD-0748 CC(C)(C)OC(=O)N1CCCCC12CCNCC2.Cl DE-0006 COc1ccc(cc1F)c2nnc3n2cc(cc3Cl)C(F)(F)F DE-0014 Cc1c(cccc1Br)C(=O)Nc2ccc(nc2)N3C[C@H](O[C@H](C3)C)C DE-0018 c1ccc(cc1)c2c(c3ccccn3n2)c4cc(c(=O)[nH]n4)C(=O)O DE-0023 COc1cccc(c1)Cn2c(c(nn2)COc3c(cc(cn3)C(F)(F)F)Cl)I DE-0024 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)C=[N+]=[N-] DE-0031 c1ccc(cc1)CN2CCC3(CCCCN3)CC2 DE-0038 CC(C)(C)OC(=O)N1CCC[C@@H]1C(=O)OC DE-0044 CC1(Cc2c(c(n[nH]2)C(F)(F)F)C(=O)C1)C DE-0046 CC(C)(C)OC(=O)N1CCC2(CCCCN2)CC1 DE-0047 c1ccc(cc1)c2c(c3ccccn3n2)c4cc(c(=O)[nH]n4)C(=O)N DE-0050 c1cc(c2cnccc2c1Cl)Cl DE-0056 c1ccc2c(c1)c(nc(n2)Cl)Cl DE-0057 c1ccc(cc1)C2C(=O)Nc3c(cccn3)O2 DE-0060 c1ccc(cc1)c2c(c3ccccn3n2)c4cc(c(nn4)Cl)C#N DE-0069 c1ccc2c(c1)c(nc(n2)Cl)CC(=O)N DE-0070 CC1(Cc2c(c(nn2c3ccc(c(c3)Br)C#N)C(F)(F)F)C(=O)C1)C DE-0071 CC(C)(C)OC(=O)N1CCC2(CCC(CC2)CN)CC1 DE-0207 CC(C)(C)OC(=O)N1CCC2(CC1)CC2C(=O)O DE-0209 c1ccc(cc1)C2CN(C2)C(c3ccccc3)c4ccccc4 DE-0211 COc1ccc2c(c1)C(=O)C(C2)Br DE-0228 c1cc2c(cc1Cl)cc(s2)CO DE-0700 c1cc2c(cc1Cl)cn[nH]2 DE-0701 c1cc2c(cc1Cl)cc(s2)C=O DE-0702 c1cc2c(cc1Cl)cc(s2)CBr DE-0703 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2C=O)Cl DE-0704 c1cc(cnc1)c2nc(sn2)N DE-0705 CC(C)(C)OC(=O)NC1CCCN(C1)c2ccc(cc2C=O)Cl DE-0707 c1c(c(cnc1NN)Cl)C(=O)O.Cl DE-0714 c1c(cnc(c1C(=O)O)Cl)[N+](=O)[O-] DE-0715 c1ccc(cc1)c2c(cc(c(=O)[nH]2)C#N)Br DE-0716 CNc1c(cc(cn1)[N+](=O)[O-])C(=O)NC DE-0717 COc1ccc-2c(c1)NC3(CCNCC3)c4n2ccc4.Cl DE-0718 COC(=O)c1cc(cnc1O)[N+](=O)[O-] DE-0720 C/N=C/c1cc(ccc1Cl)[N+](=O)[O-] DE-0721 c1ccc(cc1)c2c(cc(c(n2)Cl)C#N)Br DE-0722 CS(=O)(=O)c1c(cccn1)C#N DE-0725 CS(=O)(=O)OCC1CCC(=C)CC1 DE-0728 COc1cc(ccc1[N+](=O)[O-])N2CCC(CC2)OS(=O)(=O)C DE-0729 c1cc(c(c(c1)F)C(=O)N2CC3(CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)OC2=O)F DF-0044 c1cc(ccc1NC(=O)N2CC3(CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)OC2=O)Cl DF-0053 c1cc(ccc1c2cnc([nH]2)c3c(cc(cn3)C(F)(F)F)Cl)Cl DF-0054 c1ccc(cc1)COC(=O)N2CCC(CC2)N3CCCNC3=O DF-0055 c1ccc(cc1)COC(=O)N2CCC(CC2)N3CCNC3=O DF-0056 C1CNC(=O)N(C1)C2CCNCC2 DF-0059 CC(C)(C)OC(=O)N1CCN(C1=O)C2CCN(CC2)C(=O)OCc3ccccc3 DF-0060 CCCN(CCOc1c(cc(cc1Cl)Cl)Cl)C(=O)NC(=O)N DF-0064 c1c[nH]c2c1c(ncn2)N3CC4CC4C3C(=O)O DF-0700 CCCCCCNc1c2cc[nH]c2ncn1 DF-0703 c1ccc2c(c1)c(c([nH]2)C=O)I DF-0704 CCOC(=O)c1nc(cs1)C(=O)O DF-0707 CCOC(=O)c1c(c(c(cn1)Cl)C#N)Cl DF-0712 COC(=O)c1ccc(c(c1)NCC(=O)O)[N+](=O)[O-] DF-0713 COC(=O)c1ccc(c(c1)F)/N=C/c2cccnc2Cl DF-0715 COC(=O)c1cc(ccc1F)C=O DF-0718 CC(C)(C)OC(=O)N1CCC(CC1)NC(=O)c2cc(c(nc2)Cl)Cl DF-0719 c1cc(c(cc1CCl)C#N)F DF-0720 c1cc(c(cc1CO)C(=O)O)F DF-0721 CC(=O)c1ccc(c2c1ccc(=O)[nH]2)O DF-0723 CCOC(=O)c1cc(c[nH]1)I DF-0725 CC(=O)c1ccc(c2c1ccc(=O)[nH]2)OCc3ccccc3 DF-0726 c1c(c2c(nc1O)CCCC2=O)O DF-0729 CC(C)OC(=O)c1cc(c[nH]1)I DF-0735 CC(C)(C)OC(=O)Oc1c(cc(cc1OC)C=O)OC DG-0008 Cc1nc2c(n1C3CCN(CC3)C(=O)OC(C)(C)C)cccn2 DG-0020 Cc1nc2c(n1C3CCNCC3)cccn2.Cl.Cl DG-0024 COc1ccc(cc1OC)C(=O)c2ccc(c(c2)OC)OC DG-0030 CC(C)(C#N)NCc1ccccc1.Cl DG-0035 Cc1ccc(cc1)NC(C)(C)C#N DG-0038 COc1ccc2c(c1)C(=O)CCC2 DG-0040 CC1(CNC(=O)N1Cc2ccccc2)C DG-0042 CC(C(=O)c1ccc(c(c1)OC)O)Cl DG-0046 CCOC(=O)c1c2c([nH]n1)CCC2 DG-0049 CC(C(=O)c1ccc(c(c1)OC)O)O DG-0050 CC(C)(CN)NCc1ccccc1.Cl.Cl DG-0051 C1Cc2c([nH]nc2C(=O)O)C1 DG-0059 c1c(nc(nc1Cl)N2CCOCC2)N3CCOCC3 DG-0060 c1ccc(cc1)S(=O)(=O)n2ccc3c2ccc(c3)C=O DG-0062 c1cnc(cc1C(F)(F)F)N DG-0065 Cc1ccc(cc1)NC(C)(C)C(=O)OC DG-0067 Cc1ccc(cc1)NC(C)C DG-0068 CCOC(=O)Cn1cc(nn1)C#N DG-0069 COc1ccc2c(c1Br)C(=O)CCC2 DG-0073 C1Cc2c([nH]nc2C(=O)N)C1 DG-0075 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCCC(=O)O DG-0077 c1ccc(cc1)S(=O)(=O)n2ccc3c2ccc(c3)/C=C/C(=O)O DG-0080 CCOC(=O)/C(=C\N(C)C)/n1cc(nn1)C#N DG-0081 COc1ccc(cc1OC)c2cn[nH]c2N DG-0223 Cc1cccc(c1N)C(=O)N2CCN(CC2)C(=O)OC(C)(C)C DG-0700 c1cnc(c2c1c(c[nH]2)Br)Cl DG-0704 c1cc(c2ncc(n2c1)Cl)[N+](=O)[O-] DG-0706 c1cc(ccc1c2ccc(nc2)N)Cl DG-0708 c1cc(c2nccn2c1)N DG-0709 c1cc(c(cc1Cl)N2CCCCC2)N DG-0710 CC(C)(C)OC(=O)N1CCCCC12CCN(CC2)Cc3ccccc3 DG-0712 c1cc(ccc1c2cc(c(nc2)N)I)Cl DG-0713 CCOC(=O)c1ccc2cc[nH]c2c1 DG-0716 Cn1cc(c(cc1=O)Cl)C(=O)O DG-0718 COC(=O)c1coc2c1C(=O)NCCC2 DG-0719 c1c(cc(c2c1OCO2)Br)C=O DG-0721 Cn1ccc2c1ncnc2Cl DG-0725 c1cc(nnc1C(=O)O)Cl DH-0006 c1cc(nnc1C(=O)NCCC2CC2)Cl DH-0024 c1cc(nnc1C(=O)NCCC2CC2)N3CCN(CC3)c4ccc(nn4)C(=O)NCCC5CC5 DH-0034 Cn1c(c(c(n1)c2ccccc2)C=O)O DH-0500 c1c(c(cnc1Cl)Br)C=O DH-0700 COc1cc2c(cc1Br)CCCN2 DH-0701 c1cc2c(cc1Br)CCCN2 DH-0702 COc1cc(c(cn1)Br)C(=O)OC DH-0703 c1c(c(cnc1Cl)Br)CO DH-0704 CCOc1cc2c(cc1c3cccnc3)CCC(=O)N2C DH-0705 Cc1cccnc1C(=O)NC(C)(C)C DH-0711 CC(=O)/C(=C\N(C)C)/c1ccc(cc1)Cl DH-0712 CC(C)(C)c1c(nc[nH]1)CO DH-0713 COC(=O)c1ccc2nc(c(n2c1)I)C(F)(F)F DH-0716 c1cc(cc(c1)[N+](=O)[O-])c2c3c(cccn3)cc(n2)N DH-0717 CN1c2ccc(cc2CCC1=O)Br DH-0718 CC(C)(C)c1c(nc[nH]1)C=O DH-0720 c1cc(cc(c1)c2c3c(cccn3)cc(n2)N)C#N DH-0722 CC(C)(C)OC(=O)N1CCC(=CC1)OS(=O)(=O)C(F)(F)F DH-0724 Cc1ccc(c(c1O)C)[N+](=O)[O-] DH-0726 Cc1ccc(c(c1I)C)[N+](=O)[O-] DH-0728 c1nc(c(c(n1)Cl)CO)N DH-0730 COc1ccc(c(c1CO)[N+](=O)[O-])OC DH-0732 C=C(c1ccccc1)c2cccc(c2)N DK-0003 c1cc(ccc1C(=O)NNc2cc(cc(n2)Cl)C(F)(F)F)[N+](=O)[O-] DK-0005 COC(=O)c1c(ccs1)NC(=O)c2ccncc2 DK-0008 c1cc(cc(c1)NC(=O)/C=C/C(=O)O)C(F)(F)F DK-0010 c1cc(ncc1C(Cl)(Cl)Cl)Cl DK-0013 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)n4c5cccc(c5cn4)Br DK-0015 c1ccc(cc1)Sc2c(cc(cn2)C(F)(F)F)Cl DK-0016 c1cc(cc(c1)I)/C=C/C(=O)O DK-0019 CCOC(=O)C1CC1c2ccc(cc2)c3ccccc3 DK-0020 Cn1cccc(c1=O)c2nc3ccccc3n2C DK-0021 c1cc(ccc1C(=O)NCCOc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] DK-0022 COC(=O)C1=C(CCC1)NC(=O)NC2CCC(CC2)O DK-0024 Cc1ccc2c(n1)cc(cc2Cl)Cl DK-0025 CC(C)(C)OC(=O)N1CCC(CC1)c2[nH]cc(n2)c3ccc(c(c3)C(F)(F)F)F DK-0039 Cn1cnc2c1cccc2Br DK-0044 CSc1ccc(c(c1)O)C(=O)O DK-0201 CS(=O)(=O)c1ccc(c(c1)O)C(=O)O DK-0206 COc1ccc(cc1)CC(=O)NCc2ccccc2c3ccccc3C(=O)NCc4cc(cc(c4)F)F DK-0221 c1ccc2cc(c(cc2c1)C(=O)[O-])O.[Na+] DK-0222 Cc1cccnc1c2nc(on2)c3ccc(cc3O)OC DK-0224 C1C[C@H](NC[C@@H]1O)C(=O)O.Cl DK-0229 COc1c(c(=O)c1=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F DK-0701 c1cc(ccc1C=O)n2cc(cn2)C(F)(F)F DK-0703 C[C@@H](c1ccccc1)NCC(=O)Nc2ccccc2C(=O)c3ccccc3 DK-0704 Cc1c(cc(cn1)Cl)C(=O)O DK-0705 Cc1cc(cc(c1C=O)C)O DK-0706 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2nccc3Br DK-0707 Cc1cc(cc(c1C=O)C)OC(=O)C DK-0709 c1cc2c(cc1C(F)(F)F)oc(n2)Cl DK-0710 Cc1cc(cc(c1CO)C)O DK-0713 Cc1ccc(c(c1N)C)[N+](=O)[O-] DK-0714 Cc1cc(cc(c1C=O)C)OCc2ccccc2 DK-0715 CC(=O)Nc1ccc(cc1)C=C(C(=O)OC)NC(=O)C DK-0716 c1cc(ccc1C(=O)O)n2cc(cn2)C(F)(F)F DK-0720 CC(=O)NC(Cc1c(cccc1Cl)Cl)C(=O)OC DK-0721 Cc1cc(cc(c1C=O)C)OC DK-0722 CCOC(=O)Cn1cc(nn1)Cc2ccccc2 DK-0723 CCOC(=O)Cn1cc(nn1)CO DK-0724 Cc1cc(cc(c1/C=C(/C(=O)OC)\NC(=O)C)C)OCc2ccccc2 DK-0725 Cc1cc(cc(c1CO)C)OC DK-0726 c1cc(ccc1n2cc(cn2)C(F)(F)F)[N+](=O)[O-] DK-0728 CCOC(=O)c1cc(c(cn1)C(=O)OCC)C#N DK-0729 Cc1cc(cc(c1/C=C(/C(=O)OC)\NC(=O)C)C)O DK-0730 C[C@H](c1ccccc1)NCC(=O)Nc2ccccc2C(=O)c3ccccc3 DK-0731 CC(=O)NC(Cc1ccc(cc1)N2CCOCC2)C(=O)OC DK-0732 CC1(CCCCC1=O)C(=O)OC DL-0027 CC1=C(C(C(=C(N1)C)C(=O)OC)c2cccc(c2)[N+](=O)[O-])C(=O)O DL-0029 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=N/OC DL-0030 CC(C)(C)OC(=O)N1CCc2c(c(=O)n(cn2)Cc3ccc(cc3)F)C1 DL-0033 c1cc(ccc1C2CC2C(=O)O)Br DL-0034 COC(=O)C1=CN2C=CC=CC2N1 DL-0038 CN1CCN(CC1)c2ccc(cc2)c3nc4ccc(cc4s3)Br DL-0039 CS(=O)(=O)c1ccc(cc1)Cn2cnc3c(c2=O)CNCC3 DL-0050 c1ccc(cc1)CC(=O)O DL-0063 Cc1c(c(n[nH]1)C)N DL-0069 COCCON1C(=O)c2ccccc2C1=O DL-0070 CCCS(=O)(=O)Nc1[nH]c(nn1)N DL-0074 CC(C)(C)OC(=O)NC1CCN(C1)Cc2ccccc2 DL-0075 Cc1ccc(c(c1)C)CS(=O)(=O)N DL-0708 Cc1cc(c(c(c1)C)/c/2c\3/nc(/c(c/4\[nH]/c(c(\c5n/c(c(\c6[nH]c2cc6)/c7c(cc(cc7C)C)C)/C=C5)/c8c(cc(cc8C)C)C)/cc4)/c9c(cc(cc9C)C)C)C=C3)C DL-0709 c1cc(c(c(c1F)F)[N+](=O)[O-])Br DM-0711 Cc1c(c(n(n1)C(=O)C)C)N DM-0736 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)C#N)C=O DS-0052 CC(C)(C)OC(=O)n1ccc2c1cc(c(c2)Cl)C(F)(F)F DS-0333 CC(C)(C)OC(=O)N1CCC(=O)C(C1)Br DS-0375 c1ccc2c(c1)c(cc(=O)[nH]2)CBr DS-1133 COC(=O)c1cccc(c1CBr)Cl DS-1195 Cc1cccc(c1CBr)C DS-1240 c1ccc(cc1)C2CC(=O)N(C2)CC(=O)N DS-1993 c1ccc(cc1)CNc2c3c(cc[nH]3)nc(n2)Cl DS-2907 Cc1ccc(cc1)C(=O)C(C)Br DS-3156 COC(=O)C(c1ccc(cc1)Cl)Br DS-3169 c1ccc(cc1)CN2C[C@@H]3[C@H](C2)C(=O)NC3=O EA-0003 c1ccc(c(c1)C(=O)N2C(NN=N2)c3c(cc(cn3)C(F)(F)F)Cl)Cl EA-0019 c1ccc(c(c1)C(=O)N2[C@H](NN=N2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F EA-0020 c1ccc(cc1)COC(=O)c2cc(cc(n2)C(=O)OCc3ccccc3)C(F)(F)F EA-0030 COC(=O)/C=C/c1ccc(c(c1)Cl)OS(=O)(=O)C(F)(F)F EA-0038 Cc1cn(c(=O)[nH]c1=O)Cc2nnc(o2)C EA-0201 c1ccc2c(c1)nc(s2)c3ccc(nc3)Cl EA-0600 c1ccc2c(c1)nc(o2)c3cccnc3O EA-0601 c1ccc2c(c1)nc(o2)c3ccc(nc3)O EA-0602 c1ccc2c(c1)nc(o2)c3cccnc3Cl EA-0603 c1ccc2c(c1)nc(o2)c3ccc(nc3)Cl EA-0604 CCOC(=O)CNc1ccc(c(c1)Cl)F EA-0605 COc1cc(c(cc1F)F)[N+](=O)[O-] EA-0606 c1ccc(cc1)c2nc(cs2)O EA-0700 COC(=O)c1ccc(cc1)n2cccn2 EA-0702 c1ccc(cc1)S(=O)(=O)N2CCCC(C2)CO EA-0703 c1cc(c(nc1)c2ccc(cc2)C(=O)O)[N+](=O)[O-] EA-0706 CC(C)(C)OC(=O)N1CCC(CC1)CCl EA-0707 COC(=O)c1ccc(cc1)N2CCCC2 EA-0708 COC(=O)c1ccc(cc1)n2cncn2 EA-0709 COC(=O)c1ccc(cc1)N2CCCCC2 EA-0710 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCCC(C2)CO EA-0711 c1cc(ccc1S(=O)(=O)N2CCCC(C2)CO)Br EA-0712 CCOC(=O)C(C(=O)c1ccccc1)Br EA-0713 COC(=O)c1ccc(c(c1)F)[N+](=O)[O-] EA-0714 COC(=O)c1ccc(cc1F)[N+](=O)[O-] EA-0715 c1cc2c(cc1[N+](=O)[O-])c(=O)[nH][nH]2 EA-0717 COC(=O)C(c1ccc(cc1)C(F)(F)F)N.Cl EA-0720 CCOC(=O)N1CCN(CC1)CC(c2cccc(c2)Cl)O EA-0721 c1cc(ccc1S(=O)(=O)N2CCCC(C2)CO)Cl EA-0722 CCOc1c(cnc(n1)c2ccccc2)C(=O)OCC EA-0723 CC(=O)NC(CSc1ccc(cc1)Cl)C(=O)O EA-0724 c1ccc(c(c1)n2cccc2C=O)[N+](=O)[O-] EA-0727 c1c(c(cc(c1NC(=O)C(F)(F)F)[N+](=O)[O-])Cl)C(F)(F)F EA-0728 COc1ccc(cc1)c2ccc3c(c2)cc(s3)C(=O)OC EA-0729 CCOC(=O)N1CCN(CC1)c2ccc(cc2)C(=O)OC EA-0730 c1c(c(cc(c1N)[N+](=O)[O-])Cl)C(F)(F)F EA-0732 Cc1c(sc(n1)N)C EA-0734 c1ccc-2c(c1)Cc3c2nc(s3)N EA-0736 c1cc(ccc1c2csc(n2)N)N3CCCC3 EA-0738 Cn1c(cnc1SCc2ccc(c(c2)Cl)Cl)C=O EA-0740 c1cc(cc(c1)N2CCOCC2)C#N EA-0800 Cc1c(cccc1N)c2nnco2 EA-0801 c1cc(cc(c1)C(=O)Nc2ccc(cc2)Cl)c3ccc(cn3)C(F)(F)F EA-0802 c1ccnc(c1)CNC(=O)c2cccc(c2)c3ccc(cn3)C(F)(F)F EA-0803 c1c(cncc1Br)c2nnco2 EA-0805 c1cc(cc(c1)C(=O)NCc2ccncc2)c3ccc(cn3)C(F)(F)F EA-0806 c1ccc2c(c1)cc([nH]2)C(=O)NCCCO EA-0811 CNC(=O)c1ccccc1c2ccc(cn2)C(F)(F)F EA-0812 c1ccc(c(c1)c2ccc(cn2)C(F)(F)F)C(=O)Nc3ccc(cc3)Cl EA-0813 c1ccc(c(c1)c2ccc(cn2)C(F)(F)F)C(=O)NCc3ccccn3 EA-0814 c1ccc(c(c1)c2ccc(cn2)C(F)(F)F)C(=O)NCc3ccncc3 EA-0815 c1ccc(c(c1)c2ccc(cn2)C(F)(F)F)C(=O)N3CCN(CC3)c4ccc(cc4)Cl EA-0817 c1ccc2c(c1)cc([nH]2)C(=O)NCCO EA-0819 c1cc2nccn2cc1C(=O)NCCO EA-0820 c1ccc2c(c1)c(=O)n(cn2)N EA-0822 c1cc(cc(c1)C(=O)N2CCN(CC2)c3ccc(cc3)Cl)c4ccc(cn4)C(F)(F)F EA-0824 CN1CCN(CC1)C(=O)c2cccc(c2)c3ccc(cn3)C(F)(F)F EA-0825 CC(c1c(cc(cn1)C(F)(F)F)Cl)Sc2c(cccn2)C(F)(F)F EA-0833 CCOC(=O)c1cccc(c1)N2C(=O)CC(CC2=O)(C)C EA-0836 CC(C)(C)OC(=O)N1CCN(CC1)CCN2CCC(CC2)C(=O)O EA-0838 CC(C)(C)OC(=O)N1CCN(CC1)CCN EA-0839 COC(=O)c1c(c2ccccc2n1CC#N)Br EA-0841 CC(c1ccc(cn1)C(F)(F)F)Sc2ccc(cn2)C(F)(F)F EA-0842 c1c(cc(c(c1Cl)Oc2c(cc(cn2)C(F)(F)F)Cl)Cl)N3CCNC3=O EA-0843 COc1cccc(c1)OCCBr EA-0844 c1ccc(cc1)CN2CCN(C2=O)c3cc(c(c(c3)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl)Cl EA-0846 CN1CCN(C1=O)c2cc(c(c(c2)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl EA-0848 c1cc2c(cc1[N+](=O)[O-])c(n[nH]2)Br EA-0849 c1ccc(cc1)c2cnn3c2nccc3c4c(cc(cn4)C(F)(F)F)Cl EA-0851 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2ccsc2C(=O)O EA-0852 COC(=O)c1ccc2c(c1)nco2 EA-0853 COC(=O)c1ccc(c(c1)N)O EA-0857 Cc1ccc(c2c1cn[nH]2)[N+](=O)[O-] EA-0859 COC(=O)c1ccc(cc1)/C(=N\O)/N EA-0861 Cc1nc2cc(ccc2o1)C(=O)OC EA-0862 c1cc2c(cc1[N+](=O)[O-])c(n[nH]2)Cl EA-0864 c1cc(ncc1C(=O)NC2CC2)C(F)(F)F EA-0869 COC(=O)c1ccc(nc1)C(F)(F)F EA-0870 c1c(c2c(o1)CCCC2=O)C(=O)O EA-0872 COCCCNC(=O)c1ccc(nc1)C(F)(F)F EA-0873 COC(=O)c1cc(c(c(c1)Br)O)[N+](=O)[O-] EA-0875 c1cc2c(cc1[N+](=O)[O-])[nH]nc2Br EA-0876 c1cc(ncc1C(=O)NCC#N)C(F)(F)F EA-0880 c1cc(ncc1C(=O)NN)C(F)(F)F EA-0881 C=CCNC(=S)n1c2ccccc2nn1 EA-0921 COC(=O)c1cc(nc(c1)Cl)Cl EA-0927 c1cc(ccc1/C=N\Nc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl EB-0003 c1ccc(c(c1)/C=C(\C#N)/c2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl EB-0030 c1c(cnc(c1Cl)N2CCC(CC2)/C(=N/O)/N)C(F)(F)F EB-0064 c1cc(ccc1CC(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl EB-0082 c1cc(c(c(c1)Cl)CC(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl EB-0083 CCOC(=O)CC1=C(C(NC(=O)N1)c2ccccc2)C(=O)OCC EB-0084 COC(=O)CC1=C(C(NC(=O)N1)c2ccc(cc2)Cl)C(=O)OC EB-0085 CC(C)(C)c1ccc(cc1)C2C(=C(NC(=O)N2)CC(=O)OC)C(=O)OC EB-0086 COc1ccc(cc1)C2C(=C(NC(=O)N2)CC(=O)OC)C(=O)OC EB-0087 c1cc(ccc1C=C2C(=O)NC(=O)NC2=O)c3ccc(cn3)C(F)(F)F EB-0701 CN1C(=O)C(=Cc2ccc(cc2)c3ccc(cn3)C(F)(F)F)C(=O)N(C1=O)C EB-0702 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)Cl)c3ccc(cn3)C(F)(F)F EB-0703 c1ccc(c(c1)/C(=C/c2ccc(cc2)c3ccc(cn3)C(F)(F)F)/C#N)Cl EB-0704 CC1(OC(=O)C(=Cc2ccc(cc2)c3ccc(cn3)C(F)(F)F)C(=O)O1)C EB-0705 CNS(=O)(=O)c1ccc(cc1)Cl EB-0706 CNS(=O)(=O)c1ccccc1Cl EB-0707 c1cc(ccc1/C=C\2/C(=O)NC(=O)S2)c3ccc(cn3)C(F)(F)F EB-0709 CN(c1ccc(cn1)C(F)(F)F)S(=O)(=O)c2ccccc2 EB-0711 c1cc(c(cc1Cn2cc(cc(c2=O)Br)C=O)Cl)Cl EB-0716 c1cc(c(c(c1)Cl)Cn2cc(cc(c2=O)Br)C=O)F EB-0717 CN(c1ccc(cn1)C(F)(F)F)S(=O)(=O)c2ccccc2Cl EB-0718 Cc1c(sc(n1)Nc2ccc(cc2)F)C(=O)C EB-0720 Cc1c(sc(n1)Nc2ccc(cn2)Cl)C(=O)C EB-0721 CC(=O)c1cnc(s1)Nc2ccc(cc2)F EB-0722 CN(c1ccc(cn1)C(F)(F)F)S(=O)(=O)c2ccc(cc2)Cl EB-0724 CC(=O)c1cnc(s1)Nc2ccc(cn2)Cl EB-0725 CN(c1ccc(cn1)C(F)(F)F)S(=O)(=O)c2cccc(c2)C(F)(F)F EB-0726 CNS(=O)(=O)c1cccc(c1)C(F)(F)F EB-0727 CNS(=O)(=O)c1ccc(cc1)OC EB-0728 CNS(=O)(=O)c1ccc(cc1)F EB-0731 CNS(=O)(=O)c1ccccc1[N+](=O)[O-] EB-0733 c1cc(ccc1CO)c2ccc(cn2)C(F)(F)F EB-0735 c1ccc(cc1)/C(=C/c2ccc(cc2)c3ccc(cn3)C(F)(F)F)/C#N EB-0736 c1cc(ccc1/C=N/NC(=O)c2ccc(cc2)Cl)c3ccc(cn3)C(F)(F)F EB-0737 CS(=O)(=O)/C(=C/c1ccc(cc1)c2ccc(cn2)C(F)(F)F)/C#N EB-0738 c1cc(ccc1/C=C/C(=O)O)c2ccc(cn2)C(F)(F)F EB-0739 c1ccc(cc1)CN2CCN(CC2)Cc3ccc(cc3)c4ccc(cn4)C(F)(F)F EB-0741 c1cc(ccc1CN2CCN(CC2)c3ccc(cc3)C#N)c4ccc(cn4)C(F)(F)F EB-0742 c1cc(ccc1CN2CCCCC2)c3ccc(cn3)C(F)(F)F EB-0743 c1cc(ccc1CN2CCN(CC2)c3ccc(cc3)C(F)(F)F)c4ccc(cn4)C(F)(F)F EB-0744 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Cl)c3ccc(cn3)C(F)(F)F EB-0745 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)c3ccc(cn3)C(F)(F)F)Cl EB-0746 c1cc(cc(c1)C(F)(F)F)C(=O)/C=C/c2ccc(cc2)c3ccc(cn3)C(F)(F)F EB-0750 Cc1ccc(cc1)Cn2cc(cc(c2=O)Br)C=O EB-0752 CNS(=O)(=O)c1ccc(cc1)Oc2ccc(cn2)C(F)(F)F EB-0754 Cc1c2c(cc(nc2n(n1)C)N3CCN(CC3)CCO)C(F)(F)F EB-0800 CCOC(=O)c1cn2cc(cc(c2n1)Br)Cl EB-0803 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)Sc3ccccc3 EB-0804 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)Nc3ccccc3 EB-0805 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)N(C)C EB-0811 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)SCC(=O)OC EB-0813 CCC(C)C(C(=O)OC)N EB-0818 c1cc(c(c(c1)[N+](=O)[O-])O)C(=O)NN EB-0820 c1cc(c(cc1/C(=N/O)/N)[N+](=O)[O-])O EB-0821 CCOC(=O)C1CCN(CC1)c2cn[nH]c(=O)c2Cl EB-0822 Cc1cccn2c1nc(c2)c3ccc(cc3)N EB-0824 CC(C)(C)OC(=O)NS(=O)(=O)NCc1ccccc1 EB-0827 Cc1c2c(cc(nc2n(n1)C)N3CCCNCC3)C(F)(F)F EB-0828 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)NC EB-0832 c1c(cnc(c1Cl)c2nc(cc(n2)O)C(F)(F)F)C(F)(F)F EB-0835 c1ccc(cc1)COC(=O)N2CCN(CC2)c3cn[nH]c(=O)c3Cl EB-0836 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)Oc3ccccn3 EB-0847 CCOC(=O)c1cn2cc(ccc2n1)Br.Br EB-0851 c1cc(ccc1c2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl EB-5000 c1ccnc(c1)c2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl EB-5002 c1cc(cc(c1)Cl)c2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl EB-5004 c1ccc(c(c1)c2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl)Cl EB-5005 Cc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl EB-5006 c1cc(ccc1C=C(C#N)C#N)c2ccc(cn2)C(F)(F)F EB-5007 CCOC(=O)/C(=C/c1ccc(cc1)c2ccc(cn2)C(F)(F)F)/C#N EB-5009 COc1cccc(c1)c2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl EB-5021 c1cc(ccc1SCc2nc(no2)c3c(cc(cn3)C(F)(F)F)Cl)Cl EC-0042 c1cc(c(c(c1)Cl)C(=O)NNC(=O)[C@@H]2CCCN2c3c(cc(cn3)C(F)(F)F)Cl)Cl EC-0201 c1ccc(cc1)C(=O)NNC(=O)[C@@H]2CCCN2c3c(cc(cn3)C(F)(F)F)Cl EC-0202 COc1ccc(cc1)C(=O)NNC(=O)[C@@H]2CCCN2c3c(cc(cn3)C(F)(F)F)Cl EC-0204 c1cc(c(c(c1)Cl)C(=O)N2CCSC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl EC-0208 C[C@@H](C(=O)NNC(=O)c1ccccc1)Nc2c(cc(cn2)C(F)(F)F)Cl EC-0209 c1cc(ncc1Cl)c2[nH]nc(n2)N EC-0602 c1cnc(c(c1C=O)Cl)Cl EC-0603 c1ccc(cc1)c2ncc3n2cc(cc3Cl)C(F)(F)F EC-0605 COC(=O)C1(CCCCC1)CN.Cl EC-0705 c1c(cnc(c1Br)N)C(F)(F)F EC-0707 c1c(cnc(c1I)N)C(F)(F)F EC-0713 CCOC(=O)c1cn2cc(ccc2n1)C(F)(F)F EC-0714 c1cc(c(cc1[N+](=O)[O-])Br)CBr EC-0717 c1cc2nc(cn2cc1C(F)(F)F)C(=O)O EC-0718 c1ccc(c(c1)CO/N=C/c2cc(ccc2N3CCC(CC3)C(F)(F)F)[N+](=O)[O-])Cl EC-0721 c1cc(ccc1CO/N=C/c2cc(ccc2N3CCC(CC3)C(F)(F)F)[N+](=O)[O-])Cl EC-0722 COc1cnc(nc1O)C(F)(F)F EC-0723 c1cc2c(c(c1)[N+](=O)[O-])CNC2=O EC-0724 c1cc2c(c(c1)N)CNC2=O EC-0727 CC(C)(C)OC(=O)NC1CCCNC1 EC-0728 c1cc(ccc1S(=O)(=O)NCCO)Cl EC-0729 c1cc(ccc1c2ccc(cn2)C(F)(F)F)C(=S)N3CCN(CC3)c4ccc(cc4)Cl EC-0734 COc1cnc(nc1Cl)C(F)(F)F EC-0736 C1CC1c2c(c(c(c(n2)O)C#N)C(F)(F)F)Br EC-0737 c1cc2nc(cn2cc1C(F)(F)F)C(=O)NN EC-0739 c1ccc(cc1)S(=O)(=O)NCCO EC-0740 c1ccc2c(c1)nc(s2)NCCO EC-0741 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCCO EC-0742 COc1cnc(nc1N2CCNCC2)C(F)(F)F EC-0743 c1ccc(cc1)c2c(nc3n2cc(cc3Cl)C(F)(F)F)/C=N/NC(=O)c4ccc(cc4)Cl EC-0819 CN1C(=O)N(C(=O)C12CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cc4ccc(cc4)Cl ED-0003 Cc1ccccc1c2nc3ccc(cc3c(=O)n2Cc4c(cc(cn4)C(F)(F)F)Cl)Br ED-0014 CC(C)N1C(=O)C2(CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)N(C1=O)C ED-0018 c1cc(c(cc1[N+](=O)[O-])C=O)Br ED-0022 c1cc(ccc1n2c(=O)c3cc(ccc3[nH]c2=O)N4CCN(CC4)c5ccc(cn5)C(F)(F)F)Cl ED-0024 c1cc(ccc1NC(=O)NS(=O)(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl ED-0025 c1cc(ccc1OCC2COCCO2)Cl ED-0026 c1cc(c(cc1[N+](=O)[O-])CO)Br ED-0027 CCn1c(=O)c2cc(ccc2[nH]c1=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F ED-0031 c1ccc(cc1)COc2coc(cc2=O)CO ED-0040 COc1cc2cc[nH]c2cc1C(F)(F)F ED-0041 c1ccc(cc1)COc2cnc(cc2O)CO ED-0044 c1cc(ccc1c2nc3cc(c(cc3c(=O)n2Cc4c(cc(cn4)C(F)(F)F)Cl)F)F)C(F)(F)F ED-0045 c1c[nH]c2c(cc(cc2c1=O)Br)C#N ED-0048 c1cc(c(nc1CO)Cl)O ED-0050 c1c[nH]c2c(c1=O)cc(cc2I)Cl ED-0051 c1cc(nc(c1O)Cl)I ED-0052 c1c(nc(c(c1I)O)Cl)CO ED-0058 c1cc(ccc1n2c(=O)c3cc(ccc3[nH]c2=O)N4CCC(CC4)C(F)(F)F)Cl ED-0061 CCn1c(=O)c2cc(ccc2[nH]c1=O)N3CCC(CC3)C(F)(F)F ED-0062 c1ccc(cc1)COc2cnc(cc2O)CCl ED-0065 COc1cc(nc(n1)NC(=O)NS(=O)(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)OC ED-0069 c1c(c(cc(c1N)I)[N+](=O)[O-])C(F)(F)F ED-0070 c1cc(cc(c1)Cl)C(=O)Cc2c(cc(cn2)C(F)(F)F)Cl ED-0200 c1ccc2c(c1)C(=O)N(C2=O)CCCC(=O)CBr ED-0201 CC1(OCCO1)CCCN ED-0211 Cc1cc(cnc1Cl)C=O ED-0221 c1ccn2cc(nc2c1)C(F)(F)F ED-0228 c1cc2nc(cn2cc1Cl)C(F)(F)F ED-0229 CCOC(=O)C1CCC(=C)CC1 ED-0231 CCOC(=O)c1cc(c2cc(ccc2n1)Cl)C(F)(F)F ED-0233 CCOC(=O)C1CCC2(CC1)CO2 ED-0237 c1nc(c(c(n1)Cl)Br)C(F)(F)F ED-0241 c1cc(c2cc(sc2c1)C(=O)NN)F ED-0249 c1ccn2c(c1)nc(c2Br)C(F)(F)F ED-0250 c1cc2nc(c(n2cc1Cl)Br)C(F)(F)F ED-0251 CCOC(=O)c1c(nc(o1)NC(=O)OC(C)(C)C)C(F)(F)F ED-0252 c1c2c(sc1C(=O)NN)CCC2 ED-0254 c1c(cc(nc1C(=O)O)C(=O)O)Cl ED-0255 CCOC(=O)C1CCCc2c1c(c(s2)N)C#N ED-0256 Cn1c(nc(c1Br)Br)C=O ED-0700 c1cc(ncc1Cl)CO ED-0701 COC(=O)c1c(c2ccc(cc2s1)[N+](=O)[O-])N ED-0704 CN(C)c1c(c(ccn1)Cl)C=O ED-0705 COC(=O)c1cc(c(nc1)F)Cl ED-0706 Cc1nnc(o1)c2ccncc2 ED-0707 c1cc(c(cc1[N+](=O)[O-])NC(=O)CCl)O ED-0717 CC(=O)Nc1cc(ccc1O)N ED-0718 c1cc(c(cc1Br)C=O)N ED-0721 c1cc(ncc1Cl)C=O ED-0722 c1cc(ccc1CO)c2cnccn2 ED-0723 c1c(c(c(nc1Cl)Cl)C(=O)O)C(F)(F)F ED-0724 c1cc2c(cc1Br)cc(c(=O)[nH]2)C#N ED-0725 COC(=O)c1cc2c([nH]1)ccnc2Cl ED-0726 c1cc2c(cc1Br)cc(c(n2)N)C#N ED-0727 c1c(c(c(c(n1)Cl)Cl)I)Cl ED-0728 CCOC(=O)c1c(n2cc(ccc2n1)C(F)(F)F)Br ED-0729 c1cc2c(cc1Cl)cc(s2)C(=O)O ED-0730 COC(=O)c1c(cc(nc1Cl)Cl)C(F)(F)F ED-0733 c1ccc2c(c1)c(c(s2)C(=O)O)n3cccc3 ED-0735 Cn1c(c2ccc(cc2n1)[N+](=O)[O-])Br ED-0736 Cc1cc(cc2c1[nH]nc2)Br ED-0740 COC(=O)c1cc2ccc(nc2[nH]1)Cl ED-0741 Cn1c2cc(ccc2c(n1)Br)[N+](=O)[O-] ED-0742 c1cc(cc2c1cc([nH]2)CO)Br ED-0743 CCOC(=O)c1cc2ccc(cc2n1C(=O)OC(C)(C)C)Br ED-0744 c1cc(cc2c1cc([nH]2)C=O)Br ED-0747 c1cc2c(c(c1)[N+](=O)[O-])c(n[nH]2)I ED-0749 CCOC(=O)c1c(nc2n1cc(cc2I)C(F)(F)F)C(F)(F)F ED-0752 c1cc2c(cc1Br)cc(c(n2)Cl)C#N ED-0757 c1ccc(c(c1)CO)N2CCCCC2 ED-0758 c1cc(cc(c1)F)CNc2cccc(c2C#N)F EE-0001 Cc1c(cc(cc1I)C(=O)O)F EE-0002 CC(=O)Nc1ccc(cc1C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)N3CCN(CC3)C(=O)C EE-0004 c1cncc2c1c(cc(c2Cl)[N+](=O)[O-])Cl EE-0006 CC(C)(C)OC(=O)N1CCN(CC1)c2cccc(c2C#N)NCc3cccc(c3)F EE-0009 c1cc(ccc1/C=N/NC(=N)N)Cl EE-0010 C1COCCN1c2nc(nc(n2)Cl)N3CCOCC3 EE-0011 CCOC(=O)CNc1ccc(cc1)F EE-0012 c1cc(ccc1NCC(=O)NN)F EE-0015 CC(=O)N1CCN(CC1)c2ccc(c(c2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)NS(=O)(=O)c4ccccc4Cl EE-0018 CN1CCN(CC1)c2nc3ccccc3c(n2)CC(=O)N EE-0020 c1nc(c(c(n1)Cl)CC=O)Cl EE-0022 CC(C)(C)OC(=O)N1CCN(CC1)c2cccc3c2CNC(=O)N3Cc4cccc(c4)F EE-0023 c1cc(ccc1n2cc(nn2)COc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] EE-0026 c1cc(sc1)n2cc(nn2)COc3c(cc(cn3)C(F)(F)F)Cl EE-0027 Cc1c(cnc(n1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)O EE-0030 Cc1nc2ccccc2c(n1)O EE-0034 COc1ccc(cc1)n2cc(nn2)COc3c(cc(cn3)C(F)(F)F)Cl EE-0038 CC(C)CCn1cc(nn1)COc2c(cc(cn2)C(F)(F)F)Cl EE-0039 c1c(cnc(c1Cl)OCc2c(n(nn2)CCC3OCCO3)I)C(F)(F)F EE-0040 Cc1c(cnc(n1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)OC(C)(C)C EE-0044 CC(=O)Nc1ccc(cc1C(=O)NC)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl EE-0045 CC(C)(C)OC(=O)Nc1cnc(cc1F)Cl EE-0046 CC(C)(C)OC(=O)N(C)C1CCN(CC1)c2cc(nc(c2)C(F)(F)F)C(F)(F)F EE-0047 CC(C)(C)OC(=O)N1CC[C@H](C[C@H]1C(=O)OC)O EE-0204 CC(C)(C)OC(=O)N1CC[C@H](C[C@H]1C(=O)O)O EE-0206 c1cc2c(cc1O)C(=O)NC23CC3 EE-0208 COc1ccc2c(c1)CC(C2=O)Br EE-0215 c1ccnc(c1)C2CCNCC2.Cl.Cl EE-0216 c1c(cnc(c1Cl)N2CC(CO2)O)C(F)(F)F EE-0700 COC(=O)c1cccc2c1c(=O)[nH]c(=O)[nH]2 EE-0703 COC(=O)c1cc(cnc1Cl)[N+](=O)[O-] EE-0704 c1ccn(c1)c2ccc(cc2[N+](=O)[O-])O EE-0705 CCOC(=O)c1cc(cnc1Cl)[N+](=O)[O-] EE-0706 c1cc2c3c(c1)[nH]c(=O)nc3NNC2=O EE-0707 c1cc(c2c(c1)[nH]c(=O)[nH]c2=O)C(=O)O EE-0708 COC(=O)c1ccc(cn1)Cl EE-0710 CNc1c(cc(cn1)[N+](=O)[O-])C(=O)OC EE-0711 c1cc(ncc1C(F)(F)F)CO EE-0713 CC(C)(C)OC(=O)c1ccc(cn1)C#N EE-0714 c1cc(c(cc1Br)F)c2cc([nH]n2)N EE-0719 CS(=O)(=O)c1ccc(cn1)C#N EE-0721 c1cc2c(cc1Cl)cc(s2)C(=O)Cl EE-0723 c1c(cnc2c1c(c[nH]2)I)C(F)(F)F EE-0724 c1cc(ccc1n2cc(nn2)CBr)Cl EE-0726 c1ccn(c1)c2ccc(cc2N)O EE-0730 c1cc(ncc1C#N)N2CC(CO2)O EE-0732 C=C1CCC(CC1)CN EE-0733 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cc(cn2)[N+](=O)[O-])C(=O)O EE-0736 CC(C)(C)OC(=O)n1cc(c2c1ncc(c2)C(F)(F)F)I EE-0737 C[C@@H]1CN(C[C@@H](O1)C)c2ccc(cc2C=O)Cl EE-0738 C[C@@H]1CN(C[C@@H](O1)C)c2ccc(cc2C=O)F EE-0739 c1c(c(c(c(n1)Cl)Br)N)Br EE-0741 COC(=O)c1cc2cnc(cc2[nH]1)Cl EE-0744 C1CCc2c(c(=O)[nH]c(=O)[nH]2)C1 EE-0745 c1cnc(c(c1C(F)(F)F)Cl)CO EE-0747 c1cc2c(cc1F)cc(s2)C(=O)NN EE-0749 CS(=O)(=O)c1ccc(cc1)C(CN)O EE-0750 CC(=O)Nc1cc2c(cc1[N+](=O)[O-])OCO2 EE-0752 c1cnc(cc1C(F)(F)F)CO EE-0755 c1c(c(cc2c1OCO2)[N+](=O)[O-])N EE-0756 CC(C)(C)OC(=O)Nc1cccc(n1)N EE-0758 c1c(c(cnc1Cl)C=O)Cl EF-0002 C1CNCCC1N2CCNC2=O EF-0006 c1cc(ccc1NC(=O)c2c(c(ccn2)C(F)(F)F)Cl)Cl EF-0007 CC(C)(C)OC(=O)N1CCCN(C1=O)C2CCN(CC2)C(=O)OCc3ccccc3 EF-0010 c1cc(ccc1S(=O)(=O)N2CCN(CC2)C(=O)c3c(c(ccn3)C(F)(F)F)Cl)Cl EF-0016 c1cnc(c(c1C(F)(F)F)Cl)C(=O)N2CCN(CC2)S(=O)(=O)C(F)(F)F EF-0024 c1ccc(c(c1)S(=O)(=O)N2CC3(CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)OC2=O)Cl EF-0025 c1cnc(c(c1C(F)(F)F)Cl)C(=O)N EF-0027 CC(C)(C)OC(=O)N1CCN(C1=O)C2CCNCC2 EF-0037 CC(C)(C)OC(=O)N1CCCN(C1=O)C2CCNCC2 EF-0044 c1cc2c(cc1F)CC(=NO)C2=O EF-0048 COc1ccc2c(c1)C(=O)C(=NO)C2 EF-0052 COc1cc2c(cc1OC)C(=O)C(=NO)C2 EF-0054 c1cc(ccc1NC(=O)NC(=O)c2c(c(ccn2)C(F)(F)F)Cl)Cl EF-0056 COc1ccc2c(c1)CC(C2)N.Cl EF-0060 CC(=O)Nc1cc(ccc1[N+](=O)[O-])Cl EF-0226 CC(=O)Nc1cccc(c1)Cl EF-0227 c1cc(c(nc1)C#N)C(F)(F)F EF-0235 c1ccc2c(c1)C(=O)N(C2=O)c3ccc(cn3)C(=O)O EF-0248 CC(=O)c1c(cccn1)C(F)(F)F EF-0259 Cc1cc(cc(c1NC)C)O EF-0701 COC(=O)c1cc(ccc1F)CO EF-0702 Cc1c(sc(n1)NC(=O)CCl)C EF-0703 COc1cc(cc(n1)Cl)CO EF-0706 COC(=O)c1cc(ccc1N2CCOCC2)C=O EF-0710 COC(=O)c1cc(ccc1N2CCCCC2)C=O EF-0713 COC(=O)c1cc(ccc1N2CCCC2)C=O EF-0714 COc1cc(cc(n1)Cl)C=O EF-0715 CN(C)c1ccc(cc1C(=O)OC)C=O EF-0716 CC(C)(C)OC(=O)NC1CCCN(C1)c2ccc(cc2C(=O)OC)C=O EF-0717 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2C(=O)OC)C=O EF-0718 CC(C)(C)OC(=O)Nc1cc2c(s1)CCC2 EF-0721 c1c2cnc(cc2[nH]c1C(=O)O)Cl EF-0722 COc1cc(cc(n1)Cl)CCl EF-0723 c1cc2c(cc1/C=N/N)c(n[nH]2)N EF-0726 CC1(C(OC(O1)c2ccc(cc2)O)(C)C)C EF-0727 c1c(cnc(c1C#N)C(=O)O)Cl EF-0728 Cc1cc(c(cc1F)[N+](=O)[O-])NC EF-0731 CCOC(=O)c1cc(c(nc1)C(=O)OCC)C#N EF-0732 c1cc(c(nc1C=O)Cl)O EF-0733 CC(=O)c1ccc(c2c1ccc(=O)[nH]2)OCc3ccc(cc3)F EF-0734 CC(=O)c1ccc(c2c1ccc(=O)[nH]2)OCc3ccccc3C(F)(F)F EF-0740 c1cc2c(cc(s2)CO)c(c1)Br EF-0744 Cc1nc(on1)c2ccc(cc2)C(=O)O EF-0745 c1cc2c(cc1CCO)OCO2 EF-0746 c1c(cnc(c1C(=O)O)F)Br EF-0747 Cc1cc(c(cc1F)[N+](=O)[O-])O EF-0748 COc1c(ccc(n1)Cl)C(=O)OC EF-0750 c1cc2c(cc(s2)C=O)c(c1)Br EF-0753 COc1cc(ncc1C(=O)OC)Cl EF-0754 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCCCCC(=O)O EG-0001 CNC(=O)c1c2c([nH]n1)CCC2 EG-0002 CCOC(=O)c1c2c([nH]n1)CCCC2 EG-0003 COC(=O)[C@@H]1CCCN1.Cl EG-0005 c1cc(cc(c1)Br)n2c3c(cn2)C(=O)CCC3 EG-0012 CC1(CNC(=O)N1Cc2ccc(cc2)Cl)C EG-0014 C1CCc2c(c(n[nH]2)C(=O)O)C1 EG-0015 c1c(c(cnc1N)Br)C(F)(F)F EG-0018 C1Cc2c([nH]nc2C#N)C1 EG-0019 C1CCc2c(c(n[nH]2)C(=O)NN)C1 EG-0025 c1ccc(cc1)COC(=O)N2CCC(=O)C=C2 EG-0027 c1cc(c(c(c1)F)C#N)O EG-0028 COC(=O)[C@@H]1CCCN1C(=O)C(=O)OC EG-0031 C1CCc2c(c(n[nH]2)C(=O)N)C1 EG-0033 Cc1c(cccc1O)O EG-0038 c1ccc(cc1)S(=O)(=O)n2ccc3c2ccc(c3)/C=C/C(=O)NOC4CCCCO4 EG-0039 CC(C)(C(=O)OC)NCc1ccc(cc1)Cl EG-0042 CC1(CNCN1Cc2ccc(cc2)Cl)C EG-0043 CCC(C)(C)C(=O)C(=O)N1CCC[C@H]1C(=O)OC EG-0048 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCCCCC(=O)NOC4CCCCO4 EG-0051 CCC(C)(C)C(=O)C(=O)N1CCC[C@H]1C(=O)O EG-0058 c1cc(cnc1)CCCO EG-0061 COc1cc2c(c(c1O)OC)C3Cc4cc(c(c(c4C(C2)O3)OC)O)OC EG-0073 c1cnc2ccsc2c1C#N EG-0082 c1cc(c(nc1)N)NC2CCCC2 EG-0085 CC(C)/C=N/NC(=O)c1ccccc1 EG-0086 c1cc2c([nH]c(=O)n2C3CCCC3)nc1 EG-0087 c1cc(cc(c1)C(F)(F)F)c2[nH]c(=O)ccn2 EG-0091 CC(C)c1nnc(o1)c2ccccc2 EG-0092 COC(=O)N1CCC(CC1)O EG-0095 CC(C)C1N(N=C(O1)c2ccccc2)C(=O)C EG-0101 CC(C)(C)/C=N/NC(=O)c1ccccc1 EG-0102 c1ccc(cc1)P(=C2CC(=O)NC2=O)(c3ccccc3)c4ccccc4 EG-0103 c1cc(cc(c1)Nc2ncnc(n2)N)C(F)(F)F EG-0220 c1cc(ccc1CS(=O)(=O)N)Br EG-0222 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)O)Cl EG-0224 CCOC(=O)c1c2c(cc[nH]2)ccn1 EG-0700 c1cc(c2c(c1)OCC(=O)N2)[N+](=O)[O-] EG-0701 Cn1ccc2c1ncnc2OC EG-0702 c1c[nH]c2c1ccnc2C(=O)O EG-0703 CCOC(=O)c1c(c([nH]n1)C(F)(F)F)Cl EG-0704 c1c[nH]c2c1ccnc2CO EG-0705 c1c[nH]c2c1ccnc2C=O EG-0706 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2C(=O)OC)[N+](=O)[O-] EG-0709 CCOC(=O)c1ccnc(c1)C EG-0710 c1cc(c2c(c1)OCCN2)[N+](=O)[O-] EG-0713 Cc1cc(ccn1)C(=O)O EG-0714 CCOC(=O)c1ccc2c(cc(nc2n1)C(F)(F)F)C(F)(F)F EG-0715 c1cc(c2c(c1)OCC(=O)N2)N EG-0717 c1cc(nc2c1c(cc(n2)C(F)(F)F)C(F)(F)F)C(=O)O EG-0718 CCOC(=O)c1cccc(n1)C(C#N)c2ccccc2 EG-0719 Cc1cc(ccn1)CO EG-0720 c1ccc(cc1)C(C#N)c2cccc(n2)C(=O)O EG-0721 CC(C)(C)OC(=O)n1cc(cc1C(=O)OC)I EG-0723 Cc1cc(ccn1)C=O EG-0724 Cc1c2cc(c(nc2ccn1)OC)Br EG-0726 CCOC(=O)c1c2ccn(c2ncn1)C EG-0727 Cn1cc(c2c1ncnc2Cl)Br EG-0728 c1c(cc(c2c1CCO2)Br)CO EG-0729 Cc1cc(nc(c1C#N)CO)C EG-0730 c1c2c(cnc1Cl)C(C(=O)N2)(Br)Br EG-0732 c1c2c(cnc1Cl)CC(=O)N2 EG-0734 Cn1cc(cc1C(=O)OC)I EG-0735 c1cc2cc(nc(c2nc1)O)C3CCC(CC3)C(=O)O EH-0703 c1cc2cc(nc(c2nc1)Cl)C3CCC(CC3)C(=O)O EH-0706 CN(C(=O)c1cc(c(nc1)Cl)Cl)OC EH-0710 CC(=O)c1cc(c(nc1)Cl)Cl EH-0711 CC(c1cn(nn1)Cc2ccccc2)O EH-0712 CC(=O)c1cn(nn1)Cc2ccccc2 EH-0713 CC(C)[C@H](C(=O)O)N1Cc2ccccc2C1=O EH-0715 CC(c1cn(nn1)Cc2ccc(cc2)Cl)O EH-0716 CC(c1cn(nn1)Cc2ccc(cc2)F)O EH-0717 c1cc(cc(c1)F)c2c3c(cccn3)cc(n2)C4CCC(CC4)C(=O)O EH-0718 CC(c1cn(nn1)Cc2ccc(cc2)OC)O EH-0719 CC(c1cn(nn1)Cc2cccc(c2)C(F)(F)F)O EH-0720 CC(=O)c1cn(nn1)Cc2ccc(cc2)F EH-0721 CC(=O)c1cn(nn1)Cc2ccc(cc2)Cl EH-0722 CC(c1cn(nn1)Cc2ccc(cc2Cl)Cl)O EH-0723 c1cnc(c(c1Cl)C(=O)N)Cl EH-0725 CC(=O)c1cn(nn1)Cc2ccc(cc2)OC EH-0727 CC(=O)c1cn(nn1)Cc2cccc(c2)C(F)(F)F EH-0728 c1cc(oc1CO)Br EH-0729 C[C@H](c1cc(no1)c2ccc(cc2)Cl)O EH-0730 C[C@@H](c1cc(no1)c2ccc(cc2)Cl)O EH-0731 CC(=O)c1cn(nn1)Cc2ccc(cc2Cl)Cl EH-0732 CC1=N/C(=C\c2ccccc2)/C(=O)O1 EH-0734 CC(C)[C@H](C(=O)O)N1Cc2ccccc2C1=O EH-0735 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)CBr)Cl EK-0009 C[C@H](c1ccccc1)NCC(=O)Nc2ccc(cc2C(=O)c3ccccc3)Cl EK-0015 C[C@@H](c1ccccc1)NCC(=O)Nc2ccc(cc2C(=O)c3ccccc3)Cl EK-0016 CC(COc1ccccc1)NCCO EK-0035 [2H]c1c(c(c(c(c1[2H])[2H])CCl)[2H])[2H] EK-0040 c1cc(cc(c1)F)C(=O)CC#N EK-0059 Cn1nc(nn1)c2cccc(c2)N EK-0202 CNc1ccc(cc1)C#N EK-0203 Cn1cc(c2c1ncnc2N)Br EK-0205 CC(C)(C)OC(=O)N1CCc2c1ccc(c2)c3cn(c4c3c(ncn4)N)C EK-0207 Cn1cc(c2c1ncnc2N)c3ccc4c(c3)CCN4.Cl.Cl EK-0212 COc1ccc(cc1)CC(=O)NCc2ccccc2c3ccccc3C(=O)NCc4ccc(cc4F)F EK-0218 CC(=O)N[C@@H](Cc1ccc(cc1)N2CCOCC2)C(=O)OC EK-0702 CCOC(=O)Cn1cc(nn1)C(=O)C EK-0704 CCOC(=O)c1c(c(ccn1)C#N)Cl EK-0705 Cn1c2cccc(c2[nH]c1=O)Br EK-0706 Cn1c2cccc(c2[nH]c1=S)Br EK-0707 CC(=O)NC(=Cc1ccc(cc1)N2CCN(CC2)C)C(=O)OC EK-0710 c1cc2nc(cn2cc1Cl)C=O EK-0712 c1c(cnc(c1C(F)(F)F)O)I EK-0716 c1cc2c(cc1Br)nc(o2)S EK-0718 c1cc2c(cc1F)oc(n2)S EK-0719 c1cc2c(cc1F)oc(n2)CCl EK-0720 CCOC(=O)c1cc2ccccc2[nH]c1=O EK-0722 CC(=O)N/C(=C\c1c(ccc(c1F)F)F)/C(=O)OC EK-0723 CC(=O)N/C(=C\c1cc(ccc1Cl)[N+](=O)[O-])/C(=O)OC EK-0726 c1cc2c(cc1N(=O)=O)nc(o2)S EK-0727 CC(C)(C)OC(=O)n1c(cc(n1)c2ccc(cc2)Cl)N EL-0015 Cc1c(c(n(n1)C(=O)C)C)[N+](=O)[O-] EM-0020 c1ccc(cc1)CNC(=O)Oc2ccccc2 FA-0003 COC(=O)[C@@H]1CCCN1c2ccc(cn2)[N+](=O)[O-] FA-0006 c1ccc(cc1)OC(=O)N2CCCC2 FA-0016 C(C(=O)NNC(=O)C(F)(F)F)Cl FA-0212 C1CC1CC(=O)NNC(=O)CCl FA-0214 CC(=O)NNC(=O)c1ccc(nc1)C(F)(F)F FA-0215 COc1ccc(cc1)C(=O)NNC(=O)c2ccc(nc2)C(F)(F)F FA-0216 c1cc(ncc1C(=O)NNC(=O)C2CCCCC2)C(F)(F)F FA-0218 c1ccc(cc1)S(=O)(=O)NNC(=O)c2ccc(nc2)C(F)(F)F FA-0219 c1cc(n(c1)c2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NNC(=O)c3ccc(nc3)C(F)(F)F FA-0220 c1ccc(cc1)CN2CCC(CC2)N3C(C(CCC3=O)C(=O)O)c4ccccc4 FA-0223 c1cc(ccc1Oc2ccc(cn2)C(F)(F)F)S(=O)(=O)NNC(=O)c3ccc(nc3)C(F)(F)F FA-0226 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2ccc(nc2)C(F)(F)F FA-0227 CS(=O)(=O)NNC(=O)c1ccc(nc1)C(F)(F)F FA-0228 c1cc(c(c(c1)Cl)C(=O)NNC(=O)c2ccc(nc2)C(F)(F)F)Cl FA-0229 CCc1nnc(o1)Cn2cc(c(=O)[nH]c2=O)C FA-0233 CC(=O)c1cccc(n1)Br FA-0234 C(c1nnc(o1)C(F)(F)F)Cl FA-0235 Cc1cn(c(=O)[nH]c1=O)Cc2nnc(o2)C(C)C FA-0237 Cc1cn(c(=O)[nH]c1=O)Cc2nnc(o2)C(F)(F)F FA-0238 COc1ccc(cc1)C2C(CCC(=O)N2Cc3ccccc3)C(=O)O FA-0239 COCCC(=O)NNC(=O)CCl FA-0240 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNC(=O)c3ccc(nc3)C(F)(F)F FA-0242 CCOC(=O)c1cn[nH]c1C(F)(F)F FA-0246 c1cc2c(cc1Br)c(=O)[nH]c(=O)[nH]2 FA-0247 Cc1ccnc(n1)Cl FA-0251 c1c[nH]c(=O)nc1/C=N/O FA-0252 COc1ccc(cc1)C2C(CCC(=O)N2Cc3ccccc3)CO FA-0253 CCOC(=O)c1cnn(c1C(F)(F)F)C(=O)OC(C)(C)C FA-0255 CC(C)c1ccc(cc1)C2C(CCC(=O)N2Cc3ccccc3)C(=O)O FA-0257 c1ccc(cc1)CNC(=O)CC#N FA-0601 Cc1ccc(cc1)CNC(=O)CC#N FA-0602 c1ccc(cc1)n2c(=O)c3ccc(cc3[nH]c2=S)Cl FA-0603 c1ccc(cc1)n2c(=O)c3cc(ccc3[nH]c2=S)Cl FA-0604 c1ccc(cc1)n2c(=O)c3c(cccc3Cl)[nH]c2=S FA-0605 c1ccc(cc1)n2c(=O)c3cc(cc(c3[nH]c2=S)Cl)Cl FA-0606 c1cc(cnc1)CNC(=O)CC#N FA-0607 COc1cc2c(cc1OC)[nH]c(=S)n(c2=O)c3ccccc3 FA-0609 Cc1cccc2c1c(=O)n(c(=S)[nH]2)c3ccccc3 FA-0610 COc1ccc(cc1)CNC(=O)CC#N FA-0611 c1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=O FA-0613 c1cc2c(cc1CNC(=O)CC#N)OCO2 FA-0614 c1cc(ccc1CNC(=O)CC#N)C(F)(F)F FA-0615 c1cc(c(cc1CO)F)[N+](=O)[O-] FA-0618 COc1cccc(c1)n2c(=O)c3ccccc3[nH]c2=S FA-0619 CCOC(=O)c1cccnc1C(=O)OCC FA-0620 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3Br)F FA-0622 Cc1c(cccc1Cl)n2c(=O)c3ccccc3[nH]c2=S FA-0623 COc1cc(c(cc1F)F)N FA-0625 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccccc3F FA-0626 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)[N+](=O)[O-] FA-0627 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)Br FA-0629 c1cc(c(cc1C=O)F)[N+](=O)[O-] FA-0630 c1cc(c(cc1CO)F)N FA-0632 Cc1cc(ccc1Br)n2c(=O)c3ccccc3[nH]c2=S FA-0633 COc1ccc(c(c1)n2c(=O)c3ccccc3[nH]c2=S)OC FA-0634 Cc1cccc2c1c(=O)n(c(=S)[nH]2)c3ccc(cc3)Br FA-0635 c1cc(ccc1n2c(=O)c3cc(cc(c3[nH]c2=S)Cl)Cl)[N+](=O)[O-] FA-0636 COC(=O)c1ccc(cc1)c2c(cccn2)N FA-0700 COC(=O)c1ccc(c(c1)F)N FA-0701 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCC(=O)CC2 FA-0704 c1cc(ccc1S(=O)(=O)N2CCC(=O)CC2)Cl FA-0706 CNc1cc(ccc1[N+](=O)[O-])C(=O)OC FA-0707 CCOC(=O)N1CCN(CC1)CC(=O)c2ccc(cc2)S(=O)(=O)C FA-0708 c1cc(cnc1)/C(=N/O)/N FA-0709 c1cc2c(c[nH]c2nc1)Cl FA-0710 COc1cc(ccc1[N+](=O)[O-])C(=O)OC FA-0711 CCOC(=O)N1CCC(CC1)C(=O)O FA-0712 COc1cc(ccc1N)C(=O)OC FA-0713 CCOC(=O)N1CCN(CC1)CC(c2ccc(cc2)S(=O)(=O)C)O FA-0714 c1c2cc(c(nc2c(cc1Br)Br)N)C(=O)N FA-0716 COc1ccc(cc1)c2ccc(cc2C(=O)OC)[N+](=O)[O-] FA-0718 COc1ccc(cc1)c2cc3c(cc2C=O)OCO3 FA-0719 c1cc(cc(c1)[N+](=O)[O-])c2c(cccn2)C(=O)O FA-0721 c1cc2c(c[nH]c2nc1)I FA-0722 c1c(cnc(c1CO)Cl)Br FA-0723 c1ccc2c(c1)[nH]/c(=N/O)/c(=O)[nH]2 FA-0724 c1c(cnc(c1C=O)Cl)Br FA-0725 c1c2cc(c(nc2c(cc1Br)Br)N)C#N FA-0726 c1cc(ncc1C(=O)O)C(F)(F)F FA-0727 c1ccc(cc1)C(=O)C2CC(=O)OC2 FA-0728 COC(=O)CCCOc1ccc(cc1Cl)Cl FA-0729 Cc1cc2c(cc1C)[nH]c(=O)/c(=N\O)/[nH]2 FA-0730 CCOC(=O)c1cc2cc(ccc2[nH]1)Br FA-0732 c1ccc(cc1)NC(=O)c2ccc(nc2)C(F)(F)F FA-0800 Cc1ccc(cc1NC(=O)NCCCl)C(=O)OC FA-0801 c1cc2c(cc1[N+](=O)[O-])[nH]nc2Cl FA-0802 c1cc(ccc1NC(=O)NCCCl)OC(F)(F)F FA-0803 COc1ccc(cc1)NC(=O)NCCCl FA-0804 c1ccc(cc1)c2nc(c(s2)CC(=O)O)O FA-0805 CC(C)(C)c1ccc(cc1)NC(=O)NCCCl FA-0806 c1ccnc(c1)CN(Cc2ccccn2)C(=O)c3ccc(nc3)C(F)(F)F FA-0807 CNC(=O)c1ccc(nc1)C(F)(F)F FA-0808 c1cc(ccc1NC(=O)c2ccc(nc2)C(F)(F)F)Cl FA-0809 c1cc(cc(c1)NC(=O)c2ccc(nc2)C(F)(F)F)C(F)(F)F FA-0810 CCCc1nc2cc(ccc2o1)C(=O)OC FA-0811 c1cc(ccc1Oc2ccc(cc2CO)N)Cl FA-0812 CCOC(=O)C1CCN(CC1)c2ccc(cc2C=O)[N+](=O)[O-] FA-0813 CC(C)(C)OC(=O)N1CCc2c(c[nH]n2)C1 FA-0815 c1cc2cnn(c2cc1[N+](=O)[O-])CCO FA-0819 c1ccnc(c1)CNC(=O)c2ccc(nc2)C(F)(F)F FA-0822 c1cc2c(cc1F)c3c([nH]2)C(CCC3)C(=O)N FA-0823 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2cccc(c2)C=O FA-0825 COC(=O)c1ccc2c(c1)nc(o2)CCl FA-0826 c1ccc(c(c1)NC(=O)c2ccc(nc2)C(F)(F)F)F FA-0828 c1cc(ncc1C(=O)NCc2ccncc2)C(F)(F)F FA-0829 c1cc(ccc1Oc2ccc(cc2CCl)[N+](=O)[O-])Cl FA-0830 CCc1nc2cc(ccc2o1)C(=O)OC FA-0832 c1cc(ccc1N2CCNC2=O)OC(F)(F)F FA-0833 c1c(cc(c2c1CCO2)[N+](=O)[O-])S(=O)(=O)Cl FA-0834 COC(=O)c1ccc(c(c1)O)N FA-0837 c1cc(c(c(c1)F)C#N)OCC(F)(F)F FA-0838 CC(C)(C)OC(=O)N1CCN(CC1)CCN2CCC(CC2)C(=O)NN FA-0842 COc1ccc(cc1)N2CCNC2=O FA-0844 COC(=O)c1ccc2c(c1)oc(n2)CCl FA-0845 Cc1ccc(cc1Cl)NC(=O)NCCCl FA-0848 CSc1ccc(cc1)NC(=O)NCCCl FA-0849 CSc1cccc(c1)NC(=O)NCCCl FA-0850 c1ccc(cc1)CN2CCN(CC2)C(=O)c3ccc(nc3)C(F)(F)F FA-0851 CN1CCN(CC1)C(=O)c2ccc(nc2)C(F)(F)F FA-0853 CC(=O)N1CCc2c1ccc(c2)S(=O)(=O)Cl FA-0854 Cc1ccc(c(c1)C)NC(=O)NCCCl FA-0855 COC(=O)c1cccn2c1ncc2 FA-0856 c1cc(ccc1N2CCN(CC2)C(=O)c3ccc(nc3)C(F)(F)F)Cl FA-0857 c1cc(ncc1C(F)(F)F)n2cc(cn2)S(=O)(=O)Cl FA-0858 c1cc(cnc1)NC(=O)NCCCl FA-0861 c1ccnc(c1)CN2CCN(C2=O)c3cc(c(c(c3)Cl)Oc4c(cc(cn4)C(F)(F)F)Cl)Cl FA-0862 Cc1cnc2c(c1c3cccc(c3)OC)cccc2C(F)(F)F FA-0863 CCOC(=O)C=C1CCN(CC1)Cc2ccccc2 FA-0864 CCOC(=O)CC1CCNCC1 FA-0865 c1c(cnc(c1Cl)Cn2c(nc(n2)Br)Br)C(F)(F)F FA-0866 c1cc(c(cc1NC(=O)NCCCl)Cl)Cl FA-0874 c1nncn1CCCO FA-0875 c1cc(cnc1)N2CCNC2=O FA-0877 c1cc(c2nccn2c1)C(=O)NN FA-0879 CCOC(=O)c1nnnn1Cc2c(cc(cn2)C(F)(F)F)Cl FA-0880 c1ccc(cc1)CN2CCC3(CC2)CC(=O)NN3 FA-0881 Cc1nc(nn1Cc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F FA-0882 c1cc(ccc1C#N)NC(=O)NCCCl FA-0884 c1ccnc(c1)CCNC(=O)NCCCl FA-0886 c1cc(c(cc1N2CCNC2=O)Cl)Cl FA-0887 CSc1ccc(cc1)N2CCNC2=O FA-0888 COC(=O)c1cc2c(s1)CCC2 FA-0889 Cc1ccc(c(c1)C)N2CCNC2=O FA-0890 CC(C)(C)c1ccc(cc1)N2CCNC2=O FA-0891 c1c(cnc(c1Cl)Cn2cnc(n2)[N+](=O)[O-])C(F)(F)F FA-0893 CSc1cccc(c1)N2CCNC2=O FA-0894 c1c2c(sc1C(=O)O)CCC2 FA-0897 c1cc(ccc1C#N)N2CCNC2=O FA-0898 c1cc2c(c(c1)F)c(nc(n2)N)N FA-0899 Cc1ccc2c(c1)sc(n2)Cl FA-0920 Cc1ccc2c(c1)sc(n2)NN FA-0921 c1cc2c(cc1Br)sc(n2)Cl FA-0922 COc1cc(cc(n1)Cl)C(=O)O FA-0923 c1cc2c(cc1C(=O)O)sc(n2)Cl FA-0926 COC(=O)c1cc2cc(ccc2s1)F FA-0928 CC(C)(C)OC(=O)n1cc(c2c1nccc2)Br FA-0931 COC(=O)c1cc2c(s1)cccc2Br FA-0932 COC(=O)c1cc2cccc(c2s1)Br FA-0933 c1cc2c(cc1Br)sc(n2)NN FA-0934 c1ccnc(c1)CNC(=O)c2c(ccs2)Oc3c(cc(cn3)C(F)(F)F)Cl FB-0014 CC(C)(C)N(C(=O)c1ccccc1)NC(=O)c2ccc(cn2)C(F)(F)F FB-0017 c1c(cnc(c1Cl)c2nc(cc(n2)Cl)C(F)(F)F)C(F)(F)F FB-0056 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)OC FB-0057 Cc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)OCc3ccccc3 FB-0058 CNc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F FB-0069 c1ccc(cc1)C2=C(SC3=NCCN23)Br.Br FB-0210 c1ccc(cc1)C2=C(SC3=NCCN23)C=O FB-0218 COc1cccc(c1O)C#N FB-0600 CC(=O)c1cccnc1N FB-0601 c1cc(c(cc1Cl)Cl)C(=O)NNC(=O)CCl FB-0701 c1cc(ccc1Oc2ccc(cn2)C(F)(F)F)S(=O)(=O)N3CCCCC3 FB-0706 c1coc(n1)N FB-0707 c1cc(ccc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F FB-0708 c1cc(ccc1Oc2ccc(cn2)C(F)(F)F)S(=O)(=O)NCCN3CCCC3 FB-0709 CCOC(=O)/C(=N\Nc1ccc(cc1[N+](=O)[O-])C)/Cl FB-0713 c1cc(c(nc1)Cl)C(=O)N2CCC(CC2)C(F)(F)F FB-0714 Cc1c(c(no1)c2cc(ccc2F)Cl)C(=O)N3CCC(CC3)C(F)(F)F FB-0715 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCC(CC2)C(F)(F)F FB-0716 c1cnccc1C(=O)N2CCC(CC2)C(F)(F)F FB-0719 c1cc(ncc1C(=O)N2CCC(CC2)C(F)(F)F)C(F)(F)F FB-0720 c1cc(ccc1C(=O)N2CCC(CC2)C(F)(F)F)Cl FB-0721 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCNCC2 FB-0723 CN(C)/C=C(\C#N)/C(=O)c1ccccc1Cl FB-0724 Cc1ccc(cc1)C(=O)/C(=C/N(C)C)/C#N FB-0725 CN(C)/C=C(\C#N)/C(=O)c1cccs1 FB-0726 CN(C)/C=C(\C#N)/C(=O)c1ccc(cc1)Cl FB-0727 c1ccc(cc1)n2c(c(cn2)C(=O)N)N FB-0729 c1ccc(c(c1)NC(=O)N2CCC(CC2)C(F)(F)F)Cl FB-0730 c1cc(ccc1NC(=O)N2CCC(CC2)C(F)(F)F)Cl FB-0731 CCOC(=O)CC(=O)C1CCN(CC1)C(=O)OC(C)(C)C FB-0733 c1cc(c(cc1C(C(=O)O)N)Cl)Cl FB-0734 c1cc(ccc1C(C(=O)O)N)O FB-0735 CCCOc1ccc(cc1)C(C(=O)O)O FB-0736 c1cc(ccc1/C=C/2\C(=O)NC(=S)N2)c3c(cc(cn3)C(F)(F)F)Cl FB-5005 CSC1=N/C(=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)/C(=O)N1 FB-5007 c1cc(cc(c1)NCc2ccc(cc2)c3ccc(cn3)C(F)(F)F)C(F)(F)F FB-5008 C=CCSC1=N/C(=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)/C(=O)N1 FB-5013 C#CCSC1=N/C(=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)/C(=O)N1 FB-5014 CSC1=NC(=O)/C(=C\c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)/S1 FB-5015 c1cc(ccc1CSC2=N/C(=C/c3ccc(cc3)c4c(cc(cn4)C(F)(F)F)Cl)/C(=O)N2)Cl FB-5016 c1ccnc(c1)CSC2=N/C(=C/c3ccc(cc3)c4c(cc(cn4)C(F)(F)F)Cl)/C(=O)N2 FB-5017 CC(=O)CSC1=N/C(=C/c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)/C(=O)N1 FB-5018 CC(=O)NCc1nc(no1)c2c(cc(cn2)C(F)(F)F)Cl FC-0004 c1ccc(cc1)S(=O)(=O)Cc2nc(no2)c3c(cc(cn3)C(F)(F)F)Cl FC-0025 c1cc(ccc1S(=O)(=O)Cc2nc(no2)c3c(cc(cn3)C(F)(F)F)Cl)Cl FC-0029 Cc1cn(c(=O)[nH]c1=O)Cc2c(cc(cn2)C(F)(F)F)Cl FC-0047 Cc1cn(c(=O)n(c1=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cc3c(cc(cn3)C(F)(F)F)Cl FC-0049 Cc1cn(c(=O)n(c1=O)Cc2ccc(cc2)Cl)Cc3c(cc(cn3)C(F)(F)F)Cl FC-0050 Cc1cn(c(=O)[nH]c1=O)Cc2ccc(cc2)Cl FC-0061 Cc1cn(c(=O)[nH]c1=O)Cc2ccccc2 FC-0066 Cc1cn(c(=O)n(c1=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cc3ccc(cc3)Cl FC-0077 Cc1cn(c(=O)n(c1=O)Cc2nnc(o2)c3ccc(cc3)Cl)Cc4c(cc(cn4)C(F)(F)F)Cl FC-0080 c1cc(c(c(c1)Cl)NC(=O)N2CCSC23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl FC-0202 c1cc(c(c(c1)Cl)c2nc(c3n2cc(cc3Cl)C(F)(F)F)Br)Cl FC-0203 c1ccc(cc1)c2nc(c3n2cc(cc3Cl)C(F)(F)F)Br FC-0204 c1cc(c(c(c1)Cl)C(=O)N2CC[S@](=O)C23CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl FC-0207 c1c(c(cnc1Cl)Cl)C=O FC-0601 c1ccc(cc1)c2nc(c3n2cc(cc3Cl)C(F)(F)F)C=O FC-0602 c1cc(nc(c1)Cl)C=O FC-0603 c1cc2c(cc1Cl)NCC(O2)CO FC-0604 c1c(cnc(c1Cl)O)[N+](=O)[O-] FC-0605 c1ccc(c(c1)c2ccc(cn2)[N+](=O)[O-])C(=O)O FC-0606 c1ccc(c(c1)c2ccc(cn2)Cl)C(=O)O FC-0608 c1cc(ncc1C(F)(F)F)C(=O)O FC-0609 CC(C)(C)OC(=O)N1CCC2(CC1)c3cccn3-c4ccccc4N2 FC-0612 CCOC(=O)c1cc(cn2c1cnc2c3ccccc3)C(F)(F)F FC-0613 c1c(cnc(c1Cl)Cl)[N+](=O)[O-] FC-0614 CC(C)(C)OC(=O)N1CCN(CC1)c2c(c(ccn2)C(=O)O)Cl FC-0616 c1cc(c(cc1C=O)I)F FC-0617 c1c(c(nc(n1)N)O)Br FC-0700 COC(=O)C(C#N)(Cl)Cl FC-0708 COC(=O)c1c(ccnc1Cl)Cl FC-0713 CCOC(=O)c1cnc(nc1O)C(F)(F)F FC-0720 CCc1nc2cc(ccc2o1)Br FC-0721 Cc1nc2cc(ccc2o1)Br FC-0722 CCOC(=O)Cn1ccc2c1nccc2 FC-0723 CCOC(=O)c1c(nc(s1)Br)C(F)(F)F FC-0727 CCOC(=O)c1cnc(nc1O)c2ccccn2 FC-0729 c1cc(ccc1/C=N/NC(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl FC-0730 c1cc2ccn(c2nc1)CC(=O)O FC-0734 c1c(cnc(c1Cl)C(=O)N2CCCCC2)C(F)(F)F FC-0738 c1ccnc(c1)c2ccc(c(=O)[nH]2)C#N FC-0739 c1ccc(cc1)CN2CCN(CC2)C(=O)c3c(cc(cn3)C(F)(F)F)Cl FC-0743 c1cc(c(c(c1)Cl)c2nc(c3n2cc(cc3Cl)C(F)(F)F)/C=N/OCc4ccc(cc4)Cl)Cl FC-0808 Cn1c(c(cn1)c2c(cc(cn2)C(F)(F)F)Cl)N FC-0809 c1ccc(cc1)c2nc(c3n2cc(cc3Cl)C(F)(F)F)/C=N/OCc4ccc(cc4)Cl FC-0817 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2c3c(cc(cn3c(n2)c4ccccc4)C(F)(F)F)Cl FC-0818 CC(=O)N/N=C/c1c2c(cc(cn2c(n1)c3ccccc3)C(F)(F)F)Cl FC-0821 Cn1c(c(cn1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)Nc3ccc(cc3)Cl FC-0824 COC(=O)c1cc(cc2c1[nH]ccc2=O)Br FD-0006 Cn1c2ccc(cc2c(=O)n(c1=O)c3ccc(cc3)Cl)N4CCN(CC4)c5ccc(cn5)C(F)(F)F FD-0007 c1ccc(cc1)COc2cnc(cc2Cl)CCl FD-0010 c1c(c(c(nc1I)Cl)O)I FD-0011 COc1ccc(nc1Cl)I FD-0014 c1c[nH]c2c(c1=O)cc(cc2[N+](=O)[O-])Br FD-0016 c1c(c(cc(c1I)N)C(F)(F)F)C#N FD-0019 c1cc(ccc1Oc2cnn(c(=O)c2Cl)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl FD-0023 CCn1c(=O)c2cc(ccc2n(c1=O)C)N3CCN(CC3)c4ccc(cn4)C(F)(F)F FD-0026 Cn1c2ccc(cc2c(=O)n(c1=O)c3ccc(cc3)Cl)N4CCC(CC4)C(F)(F)F FD-0027 c1cc(nc(c1O)Br)I FD-0029 c1cc2cccc(c2c(c1)CO)CO FD-0033 COc1cc2c(cc1C(F)(F)F)NCC2 FD-0035 CC(C)(C)OC(=O)n1c2ccccc2nc1CCl FD-0036 COc1cc2c(cc1C(F)(F)F)[nH]cc2I FD-0039 COc1ccc(nc1Br)I FD-0041 c1cc(ccc1CNc2cnn(c(=O)c2Cl)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl FD-0042 c1cc(ccc1CNc2c(cnn(c2=O)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl FD-0047 c1cnc2c(c1Cl)cc(cc2[N+](=O)[O-])Br FD-0056 COc1coc(cc1=O)CO FD-0057 c1cnc2c(c1Cl)cc(cc2I)Cl FD-0067 COC(=O)c1c2cc(ccc2[nH]n1)OC(F)(F)F FD-0068 COc1cc(nc(n1)NC(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)OC FD-0070 COC(=O)c1cc(cc2c1nccc2Cl)Br FD-0072 c1cc(ccc1C(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F FD-0073 c1c(cnc(c1Cl)N2CCC(CC2)C#N)C(F)(F)F FD-0075 COc1c[nH]c(cc1=O)CO FD-0078 CCNC(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl FD-0079 c1cc(c(cc1Cl)Cl)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl FD-0081 c1c(c(cc(c1N)I)Cl)C(F)(F)F FD-0083 c1c[nH]c2c(c1=O)cc(cc2[N+](=O)[O-])C(F)(F)F FD-0086 CCOC(=O)c1cnn(c1N)c2ccc(cc2F)F FD-0087 c1cc(ccc1c2cc([nH]n2)NC(=O)c3ccc(cc3)Cl)Cl FD-0090 c1cc(c(cc1[N+](=O)[O-])C(F)(F)F)O FD-0093 c1cc(ccc1/C(=N\O)/Cc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F FD-0101 CO/N=C(/Cc1c(cc(cn1)C(F)(F)F)Cl)\c2ccc(cc2)C(F)(F)F FD-0102 CCOC(=O)c1cnn(c1N)c2ccc(cn2)Cl FD-0105 c1cc(c(nc1CO)Br)O FD-0107 CCOC(=O)c1cnn(c1N)c2ccc(c(c2)C(F)(F)F)Br FD-0109 C[Si](C)(C)C#Cc1cc(c(cc1N)C(F)(F)F)[N+](=O)[O-] FD-0110 c1cc(c(nc1CCl)Br)O FD-0111 CC(C)(C)n1c(=O)c(c(cn1)Cl)Cl FD-0113 c1c[nH]c2c(c1=O)cc(cc2Cl)C(F)(F)F FD-0114 c1c(nc(s1)Cl)Cl FD-0206 CC1CN(CCN1Cc2cc3ccccc3nc2)C(=O)OC(C)(C)C FD-0214 c1(c(sc(n1)Cl)[N+](=O)[O-])Cl FD-0215 COC(=O)C1Cc2cc(ccc2OC1)Cl FD-0220 C=C1CCC(CC1)CO FD-0222 CC(C)(C)OC(=O)NCC(CNC(=O)OC(C)(C)C)O FD-0231 c1ccc(cc1)CCNC(=O)c2c(cccc2F)F FD-0232 c1ccc(cc1)CCNC(=O)Cn2cnnn2 FD-0233 CC(C)(C)OC(=O)NCC1CNC(=O)O1 FD-0238 CCOC(=O)c1c(cc(nc1C(F)(F)F)O)O FD-0250 c1c(noc1N)C(F)(F)F FD-0252 c1(c(sc(n1)N)[N+](=O)[O-])Cl FD-0253 c1c(c(c(c(n1)Cl)I)N)I FD-0700 c1ccc(cc1)c2nc(cc(n2)Cl)N FD-0704 COc1ccc(cc1)COc2cc(nc(n2)c3ccccc3)Cl FD-0705 CCOC(=O)c1ccc(nc1)n2ccnc2 FD-0707 COc1ccc(cc1)c2cc(cc(n2)c3ccccc3)OC FD-0708 COC(=O)c1cc(c(nc1)C#N)Cl FD-0709 c1c[nH]c2c1cnc(c2I)Cl FD-0711 c1cnc(cc1I)C(=O)O.I FD-0712 c1cncc(c1C(=O)NO)O FD-0713 c1cnc2c(c1Cl)c(c[nH]2)Br FD-0714 CCOC(=O)c1c(n2cc(ccc2n1)C(F)(F)F)[N+](=O)[O-] FD-0716 CCOC(=O)c1cc(ccn1)C(F)(F)F FD-0717 c1c(c(cnc1Cl)Br)N FD-0719 c1cncc2c1c(no2)O FD-0722 CSc1nc(cc(n1)N)C(F)(F)F FD-0724 c1cc2c(c(c1)[N+](=O)[O-])C(=O)CC2=O FD-0726 COC(=O)c1ccc2c(c1)[nH]c(=O)o2 FD-0728 c1c(nc(nc1N)Cl)C(=O)N FD-0729 COC(=O)c1c(cnc(c1Cl)N)C(F)(F)F FD-0730 COC(=O)c1c(c(=O)[nH]c(=O)[nH]1)I FD-0731 COC(=O)C(C#N)c1ncc(cn1)Br FD-0732 c1cnc(c(c1N)Br)Cl FD-0733 CCOC(=O)c1ccc(s1)c2ccc3ccccc3n2 FD-0734 CCOC(=O)c1c(n2cc(ccc2n1)C(F)(F)F)N FD-0738 c1cnc(cc1C(F)(F)F)C(=O)O FD-0739 Cc1c(c(c(c(n1)NC)C#N)C(F)(F)F)Br FD-0740 COC(=O)c1ccc2c(c1)oc(=O)[nH]2 FD-0742 c1cc(nc(c1CO)Cl)Cl FD-0743 COC(=O)c1c(cn2ccnc2c1Cl)C(F)(F)F FD-0745 Cn1c2cc(ccc2c(n1)N)O FD-0747 Cc1cc(cc(n1)Cl)Cl FD-0748 c1cc2c(csc2nc1)N FD-0749 CCOC(=O)c1c(cc([nH]1)C)N FD-0751 CNC(=O)c1cc(ccc1NC(=O)CCl)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl FE-0007 CNC(=O)c1cc(ccc1NS(=O)(=O)c2ccccc2Cl)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl FE-0008 CNC(=O)c1cc(ccc1NS(=O)(=O)C)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl FE-0009 c1cc2c(cc1F)[nH]c(=O)oc2=O FE-0012 Cc1cc(cc(c1Oc2cc(nc(n2)Cl)Cl)C)C#N FE-0020 Cc1c2c(cc(cc2oc(=O)c1Cl)O)O FE-0021 c1cc(c(cc1N2CCN(CC2)S(=O)(=O)C(F)(F)F)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)N FE-0026 CCCOCCNc1cc(ncc1NC(=O)OC(C)(C)C)Cl FE-0033 c1cnc(cn1)n2cc(nn2)COc3c(cc(cn3)C(F)(F)F)Cl FE-0037 c1ccc(cc1)S(=O)(=O)NC(=O)Nc2nnc(s2)c3c(cc(cn3)C(F)(F)F)Cl FE-0038 CN1CC(=O)N(C1=O)c2cc(cc(c2)Cl)Cl FE-0041 c1cc2c(cc1N3CCN(CC3)S(=O)(=O)C(F)(F)F)c(=O)n(cn2)Cc4c(cc(cn4)C(F)(F)F)Cl FE-0043 c1ccc(c(c1)C(=O)Nc2ccc(cc2C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)N4CCN(CC4)S(=O)(=O)C(F)(F)F)Cl FE-0044 c1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)N4CCN(CC4)S(=O)(=O)C(F)(F)F)Cl FE-0045 CCCOCCNc1cc(ncc1N)Cl FE-0047 COc1cccc(c1)NC(=O)Cc2cccs2 FE-0048 c1cc(c(cc1N2CCN(CC2)S(=O)(=O)C(F)(F)F)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)NC(=O)C(F)(F)F FE-0050 CS(=O)c1c[nH]c2cc(ccc2c1=O)F FE-0052 Cc1cc(cc(c1Oc2cc(cc(c2)Cl)Nc3ccc(cc3)C#N)C)C#N FE-0066 Cc1c(cc(cc1I)C(=O)NC2CC2)F FE-0067 CCCOCCn1c2cc(ncc2nc(c1=O)Cl)Cl FE-0074 COc1ccc(cc1)c2cc3ccc(cc3nc2Cl)OCc4ccccc4 FE-0078 COc1cccc(c1)NC(=O)Cc2cccc(c2)C(F)(F)F FE-0079 c1c(cnc(c1Cl)OC2CCCNC2)C(F)(F)F FE-0207 COc1c(cccn1)C(=O)NN FE-0210 COc1cc(ccn1)F FE-0211 c1cc(ccc1COC(=O)c2c(cnc(c2Cl)Cl)C(F)(F)F)Cl FE-0214 c1cc(ccc1NC(=O)C2CN(C2)c3c(cc(cn3)C(F)(F)F)Cl)Cl FE-0215 c1cc(cc(c1)Cl)NC(=O)C2CN(C2)c3c(cc(cn3)C(F)(F)F)Cl FE-0216 c1c(cnc(c1Cl)N2CC(C2)C(=O)N3CCCC3)C(F)(F)F FE-0217 COC(=O)N1CCN(CC1)C(=O)C2CN(C2)c3c(cc(cn3)C(F)(F)F)Cl FE-0218 c1ccnc(c1)OC2CCNCC2 FE-0219 c1c(c(cnc1Cl)Br)C(=O)O FE-0223 c1c(cnc(c1Cl)CNC(=O)N)C(F)(F)F FE-0224 c1c(c(cnc1Cl)Br)C(=O)N FE-0230 c1cn(cn1)C(=O)NCc2c(cc(cn2)C(F)(F)F)Cl FE-0232 c1ccc(cc1)N2CCOCC2=O FE-0234 c1c(c(cnc1Cl)Br)C#N FE-0237 c1c(cc(nc1C(F)(F)F)C(F)(F)F)Br FE-0239 CCOC(=O)c1cc(ncc1Br)Cl FE-0247 CC(C)C(=O)N[C@H]1CCCN(C1)c2c(cc(cn2)C(F)(F)F)Cl FE-0248 c1cc(ccc1C(=O)N[C@H]2CCCN(C2)c3c(cc(cn3)C(F)(F)F)Cl)Cl FE-0249 c1cc(ccc1S(=O)(=O)N[C@H]2CCCN(C2)c3c(cc(cn3)C(F)(F)F)Cl)Cl FE-0251 CC(C)(C)OC(=O)NC1CCN(C1)c2c(cc(cn2)C(F)(F)F)Cl FE-0702 COC(=O)c1cc(ccc1N2CC(CO2)O)[N+](=O)[O-] FE-0703 CC(C)(C)OC(=O)N1CCCC(C1)CCl FE-0705 c1cc(c(nc1)C(=O)NN)Br FE-0706 CC(C)(C)C(=O)Nc1cccc2n1ccn2 FE-0707 c1cnc2ncc(n2c1)Cl FE-0708 c1cc2c(cc1Cl)cc(s2)C#N FE-0709 CC(C)(C)OC(=O)NC1CCN(C1)c2c(cc(cn2)[N+](=O)[O-])C(=O)OC FE-0711 CC1(CCNC1=O)C FE-0712 CCOC(=O)c1c(cc(c(n1)C)C(=O)C)C#N FE-0713 c1cc(c(nc1)CO)Br FE-0714 COC(=O)C(C#N)c1c(cc(cn1)C(F)(F)F)Cl FE-0716 c1c(cnc(c1Cl)CC#N)C(F)(F)F FE-0718 c1ccn(c1)c2cc3c(cc2[N+](=O)[O-])OCO3 FE-0721 COC(=O)C(C#N)c1ccc(cn1)C#N FE-0722 c1ccc(cc1)c2c(cc3c(n[nH]c3n2)N)Br FE-0724 c1c(c(cc2c1OCO2)N)N FE-0725 c1cc(ncc1C#N)CC#N FE-0726 C1CC1(C#N)C(=O)NN FE-0728 c1cc(ccc1C(=O)CC#N)Cl FE-0729 C=C1CCC(CC1)CBr FE-0731 c1cc(ncc1Cl)C(=O)NN FE-0732 CCOC(=O)c1[nH]c2ccccc2n1 FE-0733 CC(C)(C)OC(=O)NC1CCN(C1)c2ccc(cc2C(=O)OC)[N+](=O)[O-] FE-0734 COc1cc(ccc1[N+](=O)[O-])N2CCC(CC2)Br FE-0735 c1cc2c(cc1F)cc(s2)C=O FE-0738 c1ccn(c1)c2cc3c(cc2N)OCO3 FE-0740 COc1cc(ccc1N)C#N FE-0741 CNCc1cc(ccc1Cl)[N+](=O)[O-] FE-0742 CC(C)(C)OC(=O)N1CCc2cc(ccc2C1)O FE-0745 c1cc2n(c1)-c3cc4c(cc3NC25CCNCC5)OCO4.Cl FE-0748 c1cc(oc1)c2ccc(c(=O)[nH]2)C#N FE-0750 c1cc(ncc1Cl)CCl FE-0751 COC(=O)c1ccc(c(c1O)I)N FE-0752 CCCCCCOc1cccc(c1)C#N FE-0753 CC(C)C1CN(CCN1Cc2ccccc2)Cc3ccccc3 FE-0755 CCOC(=O)c1c(=O)[nH]c2ccccc2n1 FE-0756 COC(=O)c1c(c2c(s1)cccn2)O FE-0758 c1ccc(cc1)c2nc(cc(n2)Cl)C(=O)N FE-0761 CN(C)/C=C(\C#N)/c1c(cc(cn1)C(F)(F)F)Cl FE-0762 COc1cc(nc(n1)c2ccccc2)C(=O)OC FE-0763 CC(=O)Nc1ccc(c(c1)OC)OC FE-0764 c1c(cnc(c1Cl)c2c[nH]nc2N)C(F)(F)F FE-0765 c1cc(oc1)c2ccc(c(n2)Cl)C#N FE-0767 c1ccc(cc1)c2nc(cc(n2)Cl)C#N FE-0768 c1cc(ccc1Sc2ccc(cc2C=O)F)Cl FE-0769 COC(=O)c1ccc(c(c1)O)I FE-0770 COC(=O)c1cc(c(cc1O)N)Br FE-0772 COc1cc(c(cc1OC)[N+](=O)[O-])N FE-0773 CC(C)(C)OC(=O)N1CCc2cc(ccc2C1)C#N FE-0775 c1cc2c(cc1N)NCCO2.Cl FE-0777 c1cc(cc(c1)C(F)(F)F)c2cnc([nH]2)c3c(cc(cn3)C(F)(F)F)Cl FF-0004 C1CC(CC=C1)C(=O)Cl FF-0009 Cc1cc(cc(c1N)Cl)c2ccco2.Cl FF-0013 c1cc(ccc1C(=O)NC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl FF-0022 c1ccc(c(c1)C(=O)NC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl FF-0024 COc1ccc(cc1)C(=O)O[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl FF-0036 COc1cc2c(cc1OC)CC(C2)N FF-0041 c1ccc(cc1)COC(=O)N2CCC3(CC2)CO3 FF-0054 c1ccc(c(c1)C(=O)NC(=S)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl FF-0055 C1CN(C(=O)N1)CCCl FF-0057 c1cc(ccc1C(=O)NC(=S)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl FF-0066 c1cc(ccc1NC(=O)O[C@H]2CCN(C2)c3c(cc(cn3)C(F)(F)F)Cl)Cl FF-0070 c1ccc(cc1)COC(=O)N2CCC(CC2)(CNc3cccc(c3)F)O FF-0071 c1ccc(cc1)COC(=O)N2CCC(CC2)(CNc3ccccc3)O FF-0072 C[C@@H]1CN(C[C@@H](O1)C)CCN2CCNC2=O FF-0081 C1CCN(CC1)CCN2CCNC2=O FF-0082 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=S)NC(=O)c2ccc(cc2)Cl FF-0086 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=S)NC(=O)c2ccccc2Cl FF-0104 c1ccc(cc1)NCC2(CCNCC2)O FF-0107 c1cc(cc(c1)F)NCC2(CCNCC2)O FF-0122 Cc1cc(c2c(c1)[nH]c(n2)N)C FF-0208 CCn1c2ccc(cc2cc1C(=O)OCC)[N+](=O)[O-] FF-0209 c1ccc(cc1)CC(=O)Nc2ccccc2C(=O)O FF-0211 CC(C)(C)OC(=O)N1CCC(CC1)(c2ccccc2)C(=O)N FF-0212 CC(C)(C)OC(=O)Nc1cc(cc(c1)I)[N+](=O)[O-] FF-0264 COC(=O)Cc1cc2c(cc1Br)OCO2 FF-0703 CCOC(=O)c1ccc(cc1)NC(=O)NC2CCCCC2 FF-0707 CCOC(=O)c1ccc(cc1)NC(=S)Nc2cccnc2 FF-0708 COc1cc(ncc1C(=O)N)Cl FF-0709 c1c(cnc(c1C(=O)N)Cl)Br FF-0711 c1c2cc([nH]c2ncc1C(F)(F)F)C(=O)O FF-0713 c1cc2c(cc(s2)CBr)c(c1)Br FF-0719 COc1ccc(c(n1)OC)C(=O)OC FF-0720 c1cc(c(cc1[N+](=O)[O-])F)CO FF-0723 c1c(cnc(c1C#N)Cl)Br FF-0725 c1cc2c(cc(s2)C#N)c(c1)Br FF-0726 CCOC(=O)c1ccc(cc1)NC(=S)NC(=O)OCC FF-0727 CCOC(=O)c1ccc(cc1)NC(=O)Nc2ccc3c(c2)CCC3 FF-0728 COc1ccc(cc1)N2CCCC2 FF-0732 COc1cc(c(cn1)C(=O)O)Cl FF-0733 c1ccc(cc1)Cn2c(cc3c2CCC3)C(=O)O FF-0736 CCOC(=O)c1ccc(cc1)NS(=O)(=O)C FF-0742 COc1c(ccc(n1)Cl)C(=O)O FF-0743 COc1cc(ncc1C#N)Cl FF-0744 c1c2cc([nH]c2ncc1Cl)C(=O)O FF-0745 C1[C@H](O1)C(F)(F)F FF-0746 c1cc(c(cc1[N+](=O)[O-])F)C=O FF-0748 c1c(cc(nc1Cl)Cl)CO FF-0750 CCOC(=O)c1c(cccn1)F FF-0751 CC(C)(C)n1c(c(cn1)C#N)N FF-0752 CCOC(=O)C1C2CC2CN1 FF-0755 CC(C)(C)OC(=O)NN=C1C2CC3CC(C2)CC1C3 FG-0025 c1ccc2c(c1)[nH]c(n2)c3c(cc(cn3)C(F)(F)F)Cl FG-0027 c1cnc2cc(sc2c1C(=O)O)Br FG-0049 c1ccc(c(c1)NC2CC2)[N+](=O)[O-] FG-0053 c1c(cnc(c1NC2CCCC2)N)Br FG-0063 COc1ccc(cc1)COC2CCNCC2 FG-0203 c1c[nH]c2c1c(ccn2)Br FG-0210 c1cnc2c(c1Br)c(c[nH]2)Cl FG-0213 C1CC(=O)N(C1)CCCN FG-0400 CN1CCCC1CCCl FG-0401 c1cc(c(cc1Br)F)CN2CCCC2 FG-0402 C1CNCC1O.Cl FG-0403 COC1=CC(=O)NC1 FG-0404 COC1CCC(=O)N1 FG-0405 c1c[nH]c2c1cc(cn2)Br FG-0406 C1CC(=O)N(C1)CCO FG-0408 c1ccn(c1)c2ccc(cc2)O FG-0410 c1cc([nH]c1)C(=O)O FG-0411 c1c[nH]cc1C(=O)O FG-0412 Cn1cccc1C(=O)O FG-0414 c1ccc(c(c1)C(=O)O)n2cccc2 FG-0415 c1ccn(c1)c2cccc(c2)N FG-0417 C=CN1CCCC1=O FG-0420 C1CC(=O)NC1 FG-0424 c1ccn2cc(nc2c1)CO FG-0428 c1cc(cnc1)CCO FG-0429 Cc1ccc(c(=O)[nH]1)C(=O)O FG-0430 Cc1ccc(c(=O)[nH]1)C#N FG-0431 Cc1cc(cc(n1)C)O FG-0432 c1ccnc(c1)CCCO FG-0433 c1cnccc1CCCO FG-0434 c1cc(cnc1)CO FG-0435 c1ccnc(c1)CO FG-0436 c1ccnc(c1)C(=O)C(=O)c2ccccn2 FG-0437 c1c(cncc1Cl)O FG-0438 c1ccnc(c1)/C=N/O FG-0440 CC(=O)c1ccncc1 FG-0441 c1ccnc(c1)C(=O)c2ccccn2 FG-0442 c1cc(=O)[nH]nc1C(=O)O FG-0444 c1cnc(c(c1C(=O)O)F)Cl FG-0445 c1cc(cc(c1)C(=O)O)c2cccnc2 FG-0446 c1cc(cc(c1)C(=O)O)c2cccc(n2)Br FG-0447 c1ccnc(c1)c2cccc(c2)C(=O)O FG-0448 CCOC(=O)Cc1ccccn1 FG-0449 CCOC(=O)Cc1ccncc1 FG-0450 c1cnccc1CCS(=O)(=O)O FG-0451 Cc1cccc(n1)C(=O)O FG-0452 c1cc(cnc1)CC(=O)O FG-0453 CCOC(=O)Cc1cccnc1 FG-0454 c1cc(nc(c1)O)C(=O)O FG-0455 c1ccnc(c1)CCS(=O)(=O)O FG-0456 c1cc(ncc1C(=O)O)C(=O)O FG-0457 c1cncc(c1C(=O)O)C(=O)O FG-0458 c1cc(cnc1)CCC(=O)O FG-0459 c1cc(cnc1)S(=O)(=O)O FG-0460 c1cc(c(nc1)C(=O)O)C(=O)O FG-0461 c1c(cncc1C(=O)O)C(=O)O FG-0462 c1ccnc(c1)CC#N FG-0464 c1cc(nc(c1)Cl)C#N FG-0465 c1ccnc(c1)C#N FG-0466 c1cc(c(nc1)Cl)C#N FG-0467 c1cc(cnc1)C#N FG-0468 c1c(cnc(c1N)N)Br FG-0469 c1c(cnc2c1OCCN2)Br FG-0470 c1cc(ncc1Br)Cl FG-0471 c1cc(ncc1Cl)Br FG-0472 Cc1c2cc(ncc2[nH]n1)Cl FG-0474 c1cc(c(nc1)C#N)F FG-0475 Cc1cccc(n1)CO FG-0476 CCc1ccnc(c1)Br FG-0477 c1cc(ncc1C(F)(F)F)Br FG-0478 COc1cccc(n1)Br FG-0479 c1cc(ncc1F)Br FG-0480 Cc1ccnc(c1)Br FG-0481 c1cc(c(nc1)Br)[N+](=O)[O-] FG-0482 c1cc(nc(c1)Br)C(F)(F)F FG-0483 COc1cccnc1Br FG-0484 c1c(cnc(c1F)F)Cl FG-0488 c1cnccc1S FG-0489 c1cc(cnc1)CBr.Br FG-0490 c1cnccc1CBr.Br FG-0492 c1cc(nc(c1)Cl)C(F)(F)F FG-0493 c1cc(c(nc1)O)[N+](=O)[O-] FG-0494 Cc1ccc(nc1)Br FG-0495 c1ccnc(c1)CCl.Cl FG-0496 c1cc(nc(c1)Cl)Cl FG-0497 c1cc(ncc1[N+](=O)[O-])Cl FG-0498 c1cc(nc(c1)Br)C#N FG-0499 c1ccnc(c1)C(=S)N FG-0502 c1c(cnc(c1Cl)Cl)Cl FG-0503 c1cnccc1Cl.Cl FG-0504 c1cc(c(nc1)Cl)Cl FG-0505 c1c(c(c(cn1)Cl)Cl)Cl FG-0506 c1cc(ncc1Br)Br FG-0507 c1cc(ncc1[N+](=O)[O-])Br FG-0508 c1c(cncc1Cl)Cl FG-0510 c1cncc(c1O)[N+](=O)[O-] FG-0511 c1cc(nc(c1)Br)Br FG-0512 c1cc(nc(c1)Br)CO FG-0513 C1CC1(C#N)C(=O)O FG-0700 c1c(c(cnc1Cl)[N+](=O)[O-])N FG-0701 CC(C)(C)OC(=O)N(c1c(cc(cn1)C(=O)OC)Br)C(=O)OC(C)(C)C FG-0702 C1CC(C1)(C(=O)N)C(=O)O FG-0705 c1ccc(cc1)C2C=CN(N=C2C(F)(F)F)c3ccccc3 FG-0706 Cn1cc(cc1C(=O)O)I FG-0709 CC1C=NN(C=C1C(F)(F)F)c2ccccc2 FG-0710 COC(=O)c1c[nH]c(c1N)C(=O)OC FG-0711 CN1c2c(cccc2OCC1=O)N FG-0714 Cn1c2ccc(cc2nc1Cl)[N+](=O)[O-] FG-0715 Cn1cc(c2c1ncnc2OC)Br FG-0716 CC(=O)c1c(cc([nH]1)C(=O)OC)Br FG-0717 CC(=O)c1c(cc([nH]1)C(=O)OC)I FG-0718 CCOC(=O)c1ccnc(n1)Nc2ccc(cc2)C#N FG-0719 c1cc(ccc1C#N)Nc2nccc(n2)C(=O)O FG-0723 CC(C)Nc1ncc2n1cc(cc2Cl)C(F)(F)F FH-0011 Cc1cc(nc(n1)NC(=O)NCC(CO)O)C FH-0027 CC(C)N1CCN(CC1)c2ccc(cn2)C(F)(F)F FH-0204 c1cc(c(c(c1)F)CN2CCN(CC2)c3ccc(c(n3)Cl)C(F)(F)F)F FH-0205 c1ccc(cc1)C(=O)CN2CCN(CC2)c3ccc(c(n3)Cl)C(F)(F)F FH-0211 c1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(c(n3)Cl)C(F)(F)F FH-0212 c1c(c(n[nH]1)N)Cl FH-0225 CC(=O)CC(=O)Nc1cccc(c1)Br FH-0227 c1c[nH]nc1C2CC2 FH-0702 c1cnc(c(c1Cl)C(F)F)Cl FH-0707 c1ccc(cc1)CN2CCC(CC2)NCc3ccccc3[N+](=O)[O-] FH-0709 CC(C)(C)OC(=O)NC(c1ccc(cc1)Br)C(=O)O FH-0710 C[C@@H](c1cn(nn1)Cc2ccccc2)O FH-0712 c1ccc(cc1)CN2CCC(CC2)NCc3ccccc3N FH-0715 C[C@H](c1cn(nn1)Cc2ccccc2)O FH-0716 c1cc(nc(c1)Cl)C(F)F FH-0717 CN(C(=O)c1c(ccnc1Cl)Cl)OC FH-0719 c1cnc(c(c1Cl)C#N)Cl FH-0720 c1ccc(cc1)CN2CCC(CC2)N3Cc4ccccc4NC3=O FH-0721 Cc1ccc(cc1)S(=O)(=O)OC(C)C#C FH-0722 c1nc(c(c(n1)Cl)C(F)F)Cl FH-0725 CNc1c(c(ncn1)Cl)C=O FH-0726 COc1cc(cc(n1)Cl)C(F)F FH-0727 COC(=O)c1cc2cc(ccc2o1)Br FH-0731 c1ccc(cc1)CN2CCC(CC2)N3Cc4ccccc4N=C3N FH-0732 c1ccc(cc1)CN2CCC(CC2)N3Cc4ccccc4NS3(=O)=O FH-0733 c1cnc(c(c1I)C(F)F)F FH-0736 c1cnc(cc1Cl)C(F)F FH-0738 CCOC(=O)c1cc(c(nc1O)O)C#N FH-0739 CN1CCN(CC1)c2ccc3c(c2)[nH]c(=O)[nH]3 FH-0740 Cc1ccc(cc1)C2(CO2)c3ccccc3 FK-0001 c1ncn(n1)CCC#N FK-0003 c1nncn1CCC#N FK-0012 c1c(cnc2c1onc2N)C(F)(F)F FK-0026 CC(=O)n1cncn1 FK-0043 Cn1cnnc1 FK-0046 COc1ccc(c(n1)OC)[N+](=O)[O-] FK-0055 c1cc(ccc1N)n2cc(cn2)C(F)(F)F FK-0700 CC(=O)N/C(=C/c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl)/C(=O)OC FK-0703 Cc1ccc2c(c1)nc(o2)S FK-0705 Cc1ccc2c(c1)oc(n2)S FK-0706 c1cc2c(cc1F)oc(n2)Cl FK-0709 Cc1c(ccc(c1O)Br)C(=O)OC FK-0710 Cc1ccc2c(c1)oc(n2)Cl FK-0712 Cc1ccc2c(c1)nc(o2)Cl FK-0713 CC(=O)N/C(=C\c1ccc(cc1)N(C)C)/C(=O)OC FK-0715 Cc1cc(cc(c1/C=C(/C(=O)OC)\NC(=O)C)C)OC FK-0716 CC(=O)NC(Cc1cccc(c1)N)C(=O)OC FK-0719 c1cc2c(cc1Br)nc(o2)Cl FK-0720 c1cc2c(cc1[N+](=O)[O-])nc(o2)Cl FK-0723 CCOc1cc(ccc1OC)C(CS(=O)(=O)C)N FK-0724 CCOc1cc(ccc1OC)[C@@H](CS(=O)(=O)C)N FK-0726 CC(=O)NC(Cc1ccc(cc1)N(C)C)C(=O)OC FK-0730 Cc1cc(cc(c1CC(C(=O)OC)NC(=O)C)C)OC FK-0734 c1c(ncc(n1)N)C(F)(F)F FK-0736 C1C[C@@H](CNC1)C(F)(F)F FK-0737 C1C[C@H](CNC1)C(F)(F)F FK-0738 c1c(cnc(c1C(=O)O)C(F)(F)F)Br FK-0739 C[C@H](c1c(cc(cc1C(C)C)C(C)C)C(C)C)O FS-0001 C[C@@H](c1c(cc(cc1C(C)C)C(C)C)C(C)C)O FS-0002 c1cc(ccc1C(=N)N)C(=O)N.Cl FS-1000 CSc1ccc(cc1)C(=N)N.Cl FS-1001 c1cc(cc(c1)Cl)CC(=N)N FS-1002 COc1cccc(c1)CC(=N)N.Cl FS-1003 c1cc(ccc1CC(=N)N)Cl.Cl FS-1004 COc1ccc(cc1)CC(=N)N.Cl FS-1005 c1ccc(cc1)CCC(=N)N.Cl FS-1006 c1ccc(cc1)OCC(=N)N.Cl FS-1007 c1cc(cc(c1)Cl)OCC(=N)N.Cl FS-1008 COc1cccc(c1)OCC(=N)N.Cl FS-1009 COc1ccc(cc1)OCC(=N)N.Cl FS-1010 c1cc(cc2c1cc(nc2)N)Br FS-1011 c1c(cnc2c1c(n[nH]2)N)Br FS-1012 c1cc2c(cc1Br)c(no2)N FS-1013 c1cc2c(cc1Br)onc2N FS-1014 c1ccc(cc1)c2ccnc(c2)N FS-1015 COc1ccc2c(c1)ccnc2N FS-1017 CC(=O)Nc1cc(ccc1C(=O)O)F FS-1018 c1cc2c(cc1Cl)CCC2=O FS-1019 c1cc2c(cc1F)CCC2=O FS-1020 CC(=O)c1ccc(s1)Br FS-1021 CC(=O)c1ccc(s1)Cl FS-1022 Cc1ccc(cc1)S(=O)(=O)C FS-1023 Cc1ccccc1CC(=O)O FS-1024 Cc1ccc(cc1)CC(=O)O FS-1025 CC(=O)c1ccc(cc1)OC(F)(F)F FS-1026 c1cc(ccc1CN)OC(F)(F)F FS-1027 c1cc2c(cc1F)C(=O)CCO2 FS-1028 c1cc2c(cc1Br)CCC2=O FS-1029 c1cc2c(cc1Cl)C(=O)C(=O)N2 FS-1030 CC(=O)c1ccc(cc1)C(F)(F)F FS-1031 c1cc(ccc1CO)C(F)(F)F FS-1032 c1cc(ccc1CC(=O)O)C(F)(F)F FS-1033 Cc1ccc(cc1C(=O)O)F FS-1034 Cc1cc(c(nc1)N)Br FS-1035 Cc1c(ccc(n1)N)Br FS-1036 CC(=O)c1ccc(cc1)C(C)(C)C FS-1037 CCOc1ccc(cc1)CC#N FS-1038 c1cc(cc(c1)F)n2ccnc2 FS-1039 c1cc(ccc1n2ccnc2)F FS-1040 Cc1ccc2cc(ccc2n1)F FS-1041 Cc1ccc2cc(ccc2n1)OC FS-1042 c1cc2c(cc1CC#N)OCO2 FS-1043 c1ccc(cc1)n2cc[nH]c2=S FS-1044 CSc1ccccc1C(=O)O FS-1045 CC(=O)Nc1ccc(cc1)C(F)(F)F FS-1046 CCc1c(nccn1)C(=O)C FS-1047 CCc1c(nccn1)SC FS-1048 c1cc2c(cc1Br)OCO2 FS-1049 CC(=O)c1ccc(cc1O)F FS-1050 c1c(c(=O)[nH]c(=O)[nH]1)C(F)(F)F FS-1051 c1ccc(cc1)C(=O)C2CCC2 FS-1052 c1ccc2c(c1)c(c[nH]2)C(=O)O FS-1053 c1cc(ncc1Br)N FS-1054 Cc1cccc(c1C(=O)O)C FS-1055 c1ccnc(c1)c2ccccn2 FS-1056 CN(C)c1cccc2c1cccc2 FS-1057 c1ccc(cc1)CS(=O)(=O)c2ccccc2 FS-1058 Cc1ccc(cc1)SCC(=O)C FS-1059 Cc1ccc(cc1)S(=O)(=O)CC(=O)C FS-1060 Cc1ccc(cc1)S(=O)(=O)CC#N FS-1061 c1ccc(cc1)C(=O)n2ccnc2 FS-1062 c1cc2c(cc1F)C3(CCO2)C(=O)NC(=O)N3 FS-1063 c1cc2c(cc1F)C(=O)CCS2 FS-1064 c1ccc(c(c1)Nc2ncnc(n2)N)F FS-1065 c1cc2c(c(c1)F)c(ncn2)N FS-1066 c1c(nc(nc1O)N)C(F)(F)F FS-1067 c1cc(ncc1C(F)(F)F)N FS-1068 c1cncc(c1C(F)(F)F)N FS-1069 CC(=O)Nc1ccc(cc1OC(F)(F)F)C#N FS-1070 CC(=O)Nc1ccc(cc1C(F)(F)F)C#N FS-1071 CC(=O)Nc1ccc(c(c1)C(F)(F)F)C#N FS-1072 c1cncc(c1C(F)(F)F)C#N FS-1073 CN(C)c1cccc(c1C#N)F FS-1075 c1cc2c(cc1F)nc(s2)S FS-1076 c1cc(c(cc1Br)C#N)O FS-1077 COc1ccc(cc1F)C(=O)O FS-1078 c1cc(cc2c1cc[nH]2)C(F)(F)F FS-1080 c1cc2c(cc1C(F)(F)F)c(ccn2)N FS-1081 c1cc2c(ccnc2cc1C(F)(F)F)N FS-1082 c1cc2c(ccnc2c(c1)C(F)(F)F)N FS-1083 c1cc2c(cc1F)c(ccn2)O FS-1084 c1cc2c(ccnc2c(c1)F)O FS-1085 Cn1c(c(cn1)Br)N FS-1086 c1c(c([nH]n1)N)Br FS-1087 CC(C)(C)C1=NN(C(=O)C1)C FS-1088 CCOC(=O)c1cnn(c1N)C FS-1089 c1cc(sc1S(=O)(=O)N)Br FS-1090 c1cc(ccc1OC(F)(F)F)S(=O)(=O)N FS-1091 c1cc2c(cc1C(F)(F)F)sc(n2)N FS-1092 c1ccc(c(c1)C(=O)O)SC(F)F FS-1093 Cc1ccc(cc1F)C(=O)C FS-1094 Cc1ccc(cc1F)C(=O)N FS-1095 Cc1cc(ccc1F)C(=O)N FS-1096 Cc1cc(ccc1F)C(=O)O FS-1097 Cc1ccc(cc1F)CC(=O)O FS-1098 Cc1ccc(cc1CC(=O)O)F FS-1099 Cc1cc(ccc1F)C(C(=O)O)N FS-1100 COc1ccc(cc1C(F)(F)F)C(=O)N FS-1101 COc1ccc(cc1C(F)(F)F)C(=O)O FS-1102 COc1ccc(cc1C(F)(F)F)C#N FS-1103 COc1ccc(cc1C(F)(F)F)CO FS-1104 c1cc(ccc1c2cc[nH]n2)Cl FS-1105 c1cc(sc1S(=O)(=O)N)Cl FS-1106 c1c(cncc1Br)C#N FS-1107 c1cc2c(cc1C(=O)O)scn2 FS-1108 CCOC(=O)c1c[nH]c(n1)S FS-1109 Cc1c(ccc(n1)C(F)(F)F)C(=O)O FS-1111 c1cnc(nc1C(F)(F)F)N2CCNCC2 FS-1112 c1cc(sc1)c2cc[nH]n2 FS-1113 c1cc(ccc1c2cc[nH]n2)F FS-1114 Cc1cc(n(n1)c2ccccc2)N FS-1115 CCOC(=O)c1c(cc([nH]1)C)C FS-1116 CCOC(=O)c1cn[nH]c1N FS-1117 CCOC(=O)c1c(n[nH]c1N)C FS-1118 c1ccc(cc1)n2c(c(cn2)C#N)N FS-1119 c1ccc2c(c1)nc(s2)F FS-1120 c1cc(ccc1C(=O)N2CCCCC2)F FS-1121 c1cc(c(c(c1)F)C(=O)O)O FS-1122 CC(=O)c1ccc(cc1F)OC FS-1123 CC(=O)c1ccc(cc1OC)F FS-1124 COc1cccc(c1C#N)F FS-1125 c1ccc2c(c1)c(ccc2F)C(=O)O FS-1126 c1cc2c(cc(=O)oc2cc1O)C(F)(F)F FS-1127 c1cc(c(nc1)O)C(F)(F)F FS-1128 c1cc(ncc1C(F)(F)F)S FS-1129 COc1c(cccn1)C(F)(F)F FS-1130 COc1ccc(cn1)C(F)(F)F FS-1131 COc1cc(c(cn1)C(=O)N)C(F)(F)F FS-1132 CNc1nnc(s1)C(F)(F)F FS-1133 COC(=O)c1c(cccc1F)O FS-1134 CNc1ccc(cc1)OC(F)(F)F FS-1135 CC(c1ccc(cc1)C(F)(F)F)O FS-1136 Cc1ccc(cc1)C(=O)C(F)(F)F FS-1137 c1cn(cn1)S(=O)(=O)C(F)(F)F FS-1138 CC(=O)Nc1ccc(cc1)OC(F)(F)F FS-1139 c1cc(ccc1CN)C(F)(F)F FS-1140 c1cc(ccc1C(C(=O)O)O)C(F)(F)F FS-1141 c1cncc(c1C(F)(F)F)C(=O)O FS-1142 c1cc(ccc1CC#N)C(F)(F)F FS-1143 CCC(=O)c1ccc(cc1)C(F)(F)F FS-1144 c1cc2c(cc1C(F)(F)F)c(ccn2)O FS-1145 c1cc2c(ccnc2c(c1)C(F)(F)F)O FS-1146 c1ccc(c(c1)CO)OC(F)F FS-1147 c1cc(cc(c1)OC(F)F)CO FS-1148 c1cc(ccc1CO)OC(F)F FS-1149 c1ccc(c(c1)CN)OC(F)F FS-1150 c1cc(cc(c1)OC(F)F)CN FS-1151 c1cc(ccc1CN)OC(F)F FS-1152 c1ccc(c(c1)CC#N)OC(F)F FS-1153 c1cc(cc(c1)OC(F)F)CC#N FS-1154 c1cc(ccc1CC#N)OC(F)F FS-1155 c1cc(ccc1CC(C(=O)O)N)C(F)(F)F FS-1156 Cc1ccc(cc1)S(=O)(=O)CCO FS-1158 CS(=O)(=O)c1ccc(cc1)OC(F)(F)F FS-1159 c1cc2c(cc1F)sc(n2)N FS-1160 c1cc(ccc1n2c(c(cn2)C#N)N)F FS-1161 c1cc(ccc1c2cc(c(s2)C#N)N)F FS-1162 c1cc(c(=O)n(c1)CCC#N)C(F)(F)F FS-1163 c1cc(=O)n(cc1C(F)(F)F)CCC#N FS-1164 CCOC(=O)c1c[nH]c2c(c1=O)cccc2F FS-1165 CCOC(=O)c1cc(oc1C(F)(F)F)C FS-1166 CCOC(=O)c1c[nH]nc1C(F)(F)F FS-1167 c1cc2c(cc1F)nsn2 FS-1168 c1cc2c(c(c1)F)c(ncn2)O FS-1169 Cc1ccc(cc1C(=O)N)F FS-1170 c1cc2c3c([nH]c2c(c1)F)CCNC3 FS-1172 c1cc2c(cc1C(F)(F)F)nc([nH]2)CCCO FS-1173 Cc1cc(c(o1)C(F)(F)F)C(=O)CC#N FS-1174 c1cc(sc1)c2cc(on2)C(F)(F)F FS-1175 c1cc(ncc1C#N)OCC(F)(F)F FS-1176 c1cc(ncc1C(=S)N)OCC(F)(F)F FS-1177 c1cc2c(cc1OC(F)(F)F)cc([nH]2)C(=O)O FS-1178 c1cc(cc(c1)C(F)(F)F)c2cnco2 FS-1179 c1cc(ccc1c2[nH]nnn2)C(F)(F)F FS-1180 CN(c1ccc(cn1)C(F)(F)F)N FS-1181 CC1CC(=O)c2cc(ccc2O1)F FS-1183 C#CC(c1ccccc1)(C(F)(F)F)O FS-1184 c1ccc(cc1)C2CC(C(=O)O2)C(F)(F)F FS-1185 c1cc2c(cc1CO)OCO2 FS-1186 CN(C)c1cccc(c1)CO FS-1187 COc1cccc(c1O)OC FS-1188 c1ccc2c(c1)[nH]c(n2)CCCO FS-1189 CC(C)(C)c1ccc(cc1)CN FS-1190 c1cc2c(cc1CN)OCO2 FS-1191 c1ccc(c(c1)CCN)Cl FS-1192 COc1cc(c(c(c1)OC)Br)OC FS-1193 Cc1cc(cc(c1)OC)OC FS-1194 CC(=O)Nc1ccc(cc1C(=O)O)F FS-1195 c1cc(ncc1CN)C(F)(F)F FS-1196 c1cncc(c1N)C(F)(F)F FS-1197 c1cc(ncc1N)C(F)(F)F FS-1198 c1c(cncc1Br)C(=O)O FS-1199 c1cc2c(cc1Br)C(=O)OC2=O FS-1200 CC(=O)c1ccc(cc1F)O FS-1201 c1cc(c(cc1C(=O)O)O)F FS-1202 c1cc(cc(c1)F)n2cc[nH]c2=S FS-1203 COC(c1ccccc1)(C(=O)O)C(F)(F)F FS-1204 CSc1ccc(cc1)CN FS-1205 c1ccc(cc1)Oc2ccc(cc2)CN FS-1206 c1cc(ncc1C#N)C(F)(F)F FS-1207 CC(=O)C(=O)c1ccc(cc1)C(F)(F)F FS-1208 CC(C)(c1ccc(cc1)C(F)(F)F)O FS-1209 CCOC(=O)Nc1ccc(cc1)C(F)(F)F FS-1210 c1cc(ncc1C(=S)N)C(F)(F)F FS-1211 c1cc(nc(c1)N)C(F)(F)F FS-1212 c1cc(ccc1NC(=O)C(F)(F)F)O FS-1213 c1cc(oc1)CSc2cnccn2 FS-1214 c1cc(oc1)CSc2nccs2 FS-1215 Cc1c(sc(n1)C(C)C)C FS-1216 COC(=O)c1c(ccs1)N FS-1217 Cc1c(sc(n1)C(=O)C)C FS-1218 c1ccc(cc1)CSc2nc(ns2)N FS-1219 CSc1nc2ccccc2c(n1)N FS-1220 COC(=O)c1c(nc(s1)SC)N FS-1221 c1ccc2c(c1)nc(s2)O FS-1222 c1ccc(c(c1)C(C(=O)O)O)F FS-1223 C=CCNc1nc(ns1)N FS-1224 c1ccc(cc1)Nc2nc(ns2)N FS-1225 c1cc(ccc1N2CCNCC2)Cl FS-1226 c1ccc(cc1)/C=C/C(=O)N2CCNCC2 FS-1227 c1ccc(c(c1)C#N)N2CCNCC2 FS-1228 Cc1cccc(c1C)N2CCNCC2 FS-1229 Cc1ccc(cc1C)N2CCNCC2 FS-1230 c1cc(oc1)C(=O)N2CCNCC2 FS-1231 c1ccc(c(c1)N2CCNCC2)O FS-1232 c1cc(cc(c1)O)N2CCNCC2 FS-1233 Cc1ccccc1N2CCNCC2 FS-1234 Cc1cccc(c1)N2CCNCC2 FS-1235 Cc1ccc(cc1)N2CCNCC2 FS-1236 c1ccc2c(c1)cccc2CN3CCNCC3 FS-1237 c1ccc(cc1)CCN2CCNCC2 FS-1238 CN(c1ccccc1)C(=O)CN2CCNCC2 FS-1239 c1cnc(cn1)N2CCNCC2 FS-1240 c1ccnc(c1)CN2CCNCC2 FS-1241 c1cc(cnc1)CN2CCNCC2 FS-1242 c1cnccc1N2CCNCC2 FS-1243 c1cnc(nc1)N2CCNCC2 FS-1244 c1c([nH]c(=O)[nH]c1=O)C(F)(F)F FS-1245 c1c(nc(s1)N)C(F)(F)F FS-1246 CCSc1nnc(s1)S FS-1247 c1ccc(cc1)Cc2[nH]c(nn2)N FS-1248 c1(nnc(n1N)S)C(F)(F)F FS-1249 c1ccc(cc1)Cc2nnc(o2)N FS-1250 c1ccc(cc1)c2c[nH]nc2N FS-1251 Cc1c(c([nH]n1)N)c2ccccc2 FS-1252 c1ccc(cc1)C[C@@H]2C(=O)OC(=O)N2 FS-1253 CN(C)Cc1c[nH]c2c1cc(cc2)F FS-1254 CN(C)Cc1c[nH]c2c1ccc(c2)F FS-1255 c1cc2c(cc1F)c(c[nH]2)CC(=O)O FS-1256 c1cc2c(cc1F)[nH]cc2CC(=O)O FS-1257 c1cc2c(cc1F)cc([nH]2)C(=O)O FS-1258 CCOC(=O)c1cc2cc(ccc2[nH]1)F FS-1259 c1cc2c(cc1F)[nH]cc2CCN FS-1260 c1cc2c(c(c1)F)NC(=O)C2=O FS-1261 c1ccc(cc1)C[C@@H]2CCCN2 FS-1262 c1cc(c(cc1F)O)C(=O)O FS-1263 Cc1cc(n[nH]1)C(F)(F)F FS-1264 c1c(cnc(n1)N2CCNCC2)Br FS-1265 c1cncc(c1C(F)(F)F)SCC(=O)O FS-1266 c1cc(c(nc1)C(=O)O)Cl FS-1267 c1ccc(cc1)CN2CCN(CC2)C(=S)N FS-1268 Cc1ccc2c(c(sc2n1)C(=O)OC)N FS-1269 CN1c2ccccc2C(=O)C1=O FS-1270 c1ccc(c(c1)C(=O)O)NC2=CC(=O)CCC2 FS-1271 c1ccc(cc1)COC(=O)N2CCCC(C2)N FS-1272 c1ccc(cc1)CN2CCC(C2)N FS-1273 c1cc2c(c(c1)C(=O)O)OCC2 FS-1274 c1ccc(cc1)CN2CCNC(C2)CO FS-1275 c1ccc(cc1)CN2CCC(C2)O FS-1276 c1cc2c(c(c1)Br)CCC2=O FS-1277 c1cc(ccc1C2CCNCC2)Br FS-1278 c1ccc(cc1)COC(=O)N2CCCC(=O)C2 FS-1279 c1ccc(cc1)COC(=O)N2CCC(=O)C2 FS-1280 Cc1c(cccc1Cl)C(=O)O FS-1281 c1cc2c(cc1Cl)NC(=O)CN2 FS-1282 c1cc2c(cc1Cl)[nH]c(=O)oc2=O FS-1283 c1cc2c(cc1Cl)c(=O)oc(=O)[nH]2 FS-1284 c1ccc(c(c1)C(C(=O)O)N)Cl FS-1285 c1ccc(c(c1)C(C(=O)O)N)Cl FS-1286 c1cc2c(cc1O)CCC(=O)N2 FS-1287 CC1C(=O)OC(=N1)c2ccccc2 FS-1288 c1ccc(c(c1)c2cccnc2)C(=O)O FS-1289 c1cc(cnc1)c2ccc(cc2)C(=O)O FS-1290 COC(=O)C1CCc2ccccc2N1 FS-1291 c1cc2c(cc1Br)c(=O)c(co2)C#N FS-1292 c1cc2c(cc1F)c(=O)cco2 FS-1293 CC(=O)c1cc(ccc1O)Br FS-1294 Cc1cc(c(cc1Cl)C(=O)C)O FS-1295 CCc1ccc(c(c1)C(=O)C)O FS-1296 Cc1cc(c(c(c1)C(=O)C)O)C FS-1297 Cc1cc(c(cc1C)O)C(=O)C FS-1298 CCC(=O)c1cc(ccc1O)C FS-1299 CCC(=O)c1cc(ccc1O)Br FS-1300 c1cc2c(cc1Br)c(cc(=O)o2)O FS-1301 CCc1ccc2c(c1)c(cc(=O)o2)O FS-1302 c1cc(c(cc1F)c2ccno2)O FS-1303 c1cc(c(cc1Cl)c2ccn[nH]2)O FS-1304 c1ccc(cc1)c2[nH]nc(n2)S FS-1305 c1cnccc1c2nnc(s2)N FS-1306 c1cc2c(cc1F)NC(=O)CO2 FS-1307 CC(=O)c1ccc2c(c1)OCCO2 FS-1308 Cc1ccc(cc1)c2cc([nH]n2)N FS-1309 c1cc(c(nc1)C(=O)O)Br FS-1310 c1cc(cc(c1)Br)C[C@@H](C(=O)O)N FS-1311 COc1ccc2c(c1)C(=O)CC2 FS-1312 COc1ccc2c(c1)CCC2=O FS-1313 CC(=O)c1c(cccc1F)OC FS-1314 CC(=O)c1ccc(c(c1)OC)F FS-1315 c1cc(c(c(c1)F)O)C(=O)O FS-1316 c1cc(c(cc1C(=O)O)F)O FS-1317 c1cc(c(cc1C(=O)O)C(F)(F)F)O FS-1318 c1cc(c(cc1CC(=O)O)F)O FS-1319 c1ccc(cc1)c2ccc(nc2)N FS-1320 CNCc1cccc2c1cccc2 FS-1321 COC(=O)c1ccc2ccccc2c1 FS-1322 c1cc(c(cc1O)C(=O)O)F FS-1323 COc1ccc(c(c1)F)C(=O)O FS-1324 COc1cc(ccc1C(=O)O)F FS-1325 COc1ccc(c(c1)F)C#N FS-1326 COc1ccc(c(c1)C#N)F FS-1327 COc1cc(ccc1C#N)F FS-1328 COc1cc(ccc1F)CO FS-1329 COc1ccc(c(c1)CN)F FS-1330 COc1cc(ccc1F)CN FS-1332 CC(c1ccc(c(c1)F)OC)N FS-1333 c1cc2c(c(c1)Cl)nc(s2)N FS-1334 c1cc2c(cc1Br)sc(=O)[nH]2 FS-1335 c1ccc2c(c1)nc(s2)Cl FS-1336 c1cc2c(c(c1)Cl)C(=O)OC2=O FS-1337 COc1ccc2c(c1)sc(n2)C#N FS-1338 c1ccc2c(c1)[nH]c(n2)CC#N FS-1339 c1cc(cc2c1cc(cc2)O)C(=O)O FS-1340 c1ccn(c1)c2ccc(c(c2)C(=O)O)O FS-1341 c1cc(ccc1n2ccnc2)O FS-1342 COc1ccc(cc1)n2cccc2 FS-1343 CCOC(=O)c1c(c2ccccc2o1)C FS-1344 c1ccc(cc1)c2ccc(o2)C(=O)O FS-1345 Cc1ccc(c(c1)C(=O)O)F FS-1346 c1cc(ccc1C(F)(F)F)S(=O)(=O)N FS-1347 CC(=O)c1ccc(c(c1)Cl)OC FS-1348 c1c(cc(cc1C(=O)O)F)C#N FS-1349 COC(=O)c1cnccc1N FS-1350 CC1CCc2c(sc(c2C(=O)OC)N)C1 FS-1351 COC(=O)c1c2c(sc1N)CCCC2 FS-1352 COC(=O)c1c2c(sc1N)CCC2 FS-1353 Cc1c(sc(c1C(=O)OC)N)C FS-1354 CCc1c(sc(c1C(=O)OC)N)C FS-1355 CCC1CCc2c(sc(c2C(=O)OC)N)C1 FS-1356 COC(=O)c1c2c(sc1N)CCCCCC2 FS-1357 Cc1cc(c(s1)N)C(=O)OC FS-1358 CCc1cc(c(s1)N)C(=O)OC FS-1359 CC(C)c1cc(c(s1)N)C(=O)OC FS-1360 COC(=O)c1cc(sc1N)c2ccccc2 FS-1361 COC(=O)c1c(csc1N)c2ccccc2 FS-1362 Cc1ccc(cc1)c2csc(c2C(=O)OC)N FS-1363 Cc1cccc(c1)c2csc(c2C(=O)OC)N FS-1364 Cc1cccc(c1)c2csc(n2)N FS-1365 c1cc(ccc1C#N)c2csc(n2)N FS-1366 COC(=O)c1ccc(cc1)c2csc(n2)N FS-1367 c1cc(cc(c1)F)c2csc(n2)N FS-1368 c1cc(cc(c1)c2csc(n2)N)C#N FS-1369 c1cc2c(cc1c3csc(n3)N)OCCO2 FS-1370 CSc1ccc(cc1)c2csc(n2)N FS-1371 COc1ccc(cc1F)c2csc(n2)N FS-1372 c1cc(sc1c2csc(n2)N)Cl FS-1373 Cc1c(nc(s1)N)c2ccccc2 FS-1374 CCc1ccc(s1)c2csc(n2)N FS-1375 Cc1c(sc(n1)N)C(=O)OC FS-1376 c1ccc2c(c1)c(c3c(n2)CCC3)C(=O)O FS-1377 c1cc(sc1C(=O)O)Cl FS-1378 CCc1ccc(s1)C(=O)O FS-1379 Cn1c(c(cn1)Br)C(=O)O FS-1380 Cn1cc(c(n1)C(=O)O)Br FS-1381 Cn1cc(c(n1)C(=O)O)Cl FS-1382 Cc1c(c(n(n1)C)C(=O)O)Cl FS-1383 CCn1c(c(cn1)Cl)C(=O)O FS-1384 Cc1c(n(c2c1cc(cc2)C(=O)O)C)C FS-1385 Cc1cc(nn1CC(=O)O)C(F)(F)F FS-1386 c1cc(cc(c1)C(=O)O)Cn2cc(cn2)Cl FS-1387 c1cc(ccc1Cn2cc(cn2)Cl)C(=O)O FS-1388 Cn1c(cc(n1)C(F)(F)F)C(=O)O FS-1389 Cc1c(c(nn1C)C(=O)O)Br FS-1390 Cc1cc(c2ccccc2n1)C(=O)O FS-1391 c1ccc2c(c1)c(c(s2)C(=O)O)Cl FS-1392 COc1ccc2c(c1)sc(c2Cl)C(=O)O FS-1393 c1ccc(c(c1)CN2CCNCC2)Cl FS-1395 Cc1ccc(c(c1)CN2CCNCC2)C FS-1396 Cc1ccc2ccccc2c1CN3CCNCC3 FS-1397 c1csc2n1cc(n2)C(=O)O FS-1398 Cc1cccn2c1nc(c2)C(=O)O FS-1399 Cc1cc(n(n1)CC(=O)O)C FS-1400 CCOc1ccc(cc1)c2csc(n2)N FS-1401 c1cc(ccc1c2csc(n2)N)O FS-1402 c1cc2c(cc1O)sc(n2)N FS-1403 CC(=O)c1ccc(c(c1)Br)OC FS-1404 c1cc(sc1)C(=O)c2[nH]ccn2 FS-1405 COC(=O)c1c(c2cc(ccc2o1)Cl)N FS-1406 COc1ccc(cc1Cl)CN FS-1407 c1cc2c(cc1Cl)nc([nH]2)N FS-1408 Cc1ccc(cc1)c2nnc(s2)N FS-1409 c1ccc(cc1)CCc2nnc(s2)N FS-1410 CCCn1c2ccccc2nc1N FS-1411 Cc1cc(cc(c1OCCN)C)Br FS-1412 CNC(=O)c1ccc2c(c1)sc(n2)N FS-1413 CC(C)(C)C(=O)Nc1ccc(cc1)C(=O)O FS-1414 CC(C)(C)C(=O)Nc1cccc(c1)C(=O)O FS-1415 CC(C)(C)Sc1ccccc1C(=O)O FS-1416 Cc1cc(n(n1)c2ccc(cc2)C(=O)O)N FS-1417 c1ccc(cc1)c2[nH]c3ccc(cc3n2)C(=O)O FS-1418 c1ccc(cc1)c2c(n3ccccc3n2)CN FS-1419 Cc1c(nc(s1)N)c2ccc(cc2)F FS-1420 c1cc(ccc1c2c[nH]nc2)Br FS-1422 c1ccc2c(c1)c(ccn2)c3c[nH]nc3 FS-1423 c1ccc2c(c1)ccc(n2)c3c[nH]nc3 FS-1424 Cc1csc(n1)Br FS-1425 c1c(nc(s1)Br)C(=O)O FS-1426 c1c(sc(n1)Br)C(=O)O FS-1427 c1c(nc(s1)Br)CO FS-1428 COC(=O)c1csc(n1)Br FS-1429 COC(=O)c1cnc(s1)Br FS-1430 c1c(onc1Br)CO FS-1432 COc1ncc(cn1)Br FS-1433 c1cc2c(cc[nH]2)c(c1)Cl FS-1434 COC(=O)c1ccc2cc[nH]c2c1 FS-1436 COC(=O)c1cc(cs1)c2ccccc2 FS-1437 Cc1c(ccc(n1)C(F)(F)F)C#N FS-1438 Cc1c(ccc(n1)C(F)(F)F)CO FS-1439 c1ccc(cc1)c2cc(c(o2)N)C#N FS-1440 CC1=CS(=O)(=O)c2c1cc(cc2)Cl FS-1441 Cc1cc(c(o1)C(F)(F)F)C(=O)O FS-1442 Cc1csc2c1c(=O)[nH]cn2 FS-1443 c1ccc(cc1)c2cc3c(s2)c(=O)[nH]cn3 FS-1444 c1cc(ccc1c2cc3c(s2)c(=O)[nH]cn3)F FS-1445 Cc1c(cc(c(n1)N)C#N)C#N FS-1446 COC(=O)c1c(c(cs1)c2ccccc2)N FS-1447 c1ccc(cc1)c2cc(sc2)C(=O)O FS-1448 c1ccc(cc1)n2c(cc(n2)C3CC3)N FS-1449 Cc1c(c(n[nH]1)C)Br FS-1450 c1cc(sc1)S(=O)(=O)N FS-1451 c1cc2c(cc1Br)c(ccn2)N FS-1452 CC(C)(C)c1ccc(cc1)S(=O)(=O)N FS-1453 c1cc(ccc1SCc2[nH]nnn2)Cl FS-1454 c1cnc(cc1C(F)(F)F)O FS-1455 c1cc(c(cc1C#N)Cl)O FS-1456 Cc1c(c(on1)C)Br FS-1457 CCOC(=O)c1ccsc1N FS-1458 c1cc(sc1)C(=O)N2CCCNCC2 FS-1459 CC(=O)c1ccc(s1)C#N FS-1460 Cc1c(ccc(n1)C(F)(F)F)C(=O)C FS-1461 COC(=O)c1c(cc(s1)c2ccccc2)N FS-1462 Cc1c(cnn1c2ccccc2)C(=O)O FS-1463 Cc1c(cc(o1)c2ccccc2)C(=O)O FS-1464 c1cc(ncc1C(F)(F)F)N2CCCNCC2 FS-1465 c1cc(c(nc1)N2CCCNCC2)C(F)(F)F FS-1466 c1ccc(cc1)CN2CCCNCC2 FS-1467 Cc1c(c(no1)N)Br FS-1468 CN(C)c1cccc(c1)C(=O)N FS-1469 Cn1cc(nc1)S(=O)(=O)N FS-1470 Cc1nc(cn1C)S(=O)(=O)N FS-1471 CN1CCN(CC1)c2ccccc2CO FS-1472 Cn1c(cc(n1)C(F)(F)F)c2cccs2 FS-1473 Cc1c(cc(o1)C(C)(C)C)C(=O)O FS-1477 CC(C)(C)c1cc(c(s1)C(=O)OC)N FS-1478 c1cc(c(nc1)Oc2ccc(cc2)F)N FS-1479 COC(=O)c1c(ccs1)Cl FS-1480 Cc1c(sc(n1)C)C(=O)O FS-1481 c1cc(ncc1C#N)N2CCCNCC2 FS-1483 c1ccnc(c1)c2csc(n2)N FS-1484 Cn1c(cc(n1)c2ccccc2)N FS-1485 Cn1c(cc(n1)c2cccs2)N FS-1486 c1cc(sc1)c2cc([nH]n2)N FS-1487 c1cc(cnc1)c2csc(n2)N FS-1488 c1cnccc1c2csc(n2)N FS-1489 CCOC(=O)c1c(c(sc1N)C)C FS-1490 Cc1c(sc2c1c(=O)[nH]cn2)C FS-1491 Cc1c(sc2c1c(ncn2)N3CCNCC3)C FS-1492 Cc1c(cccc1Cl)S(=O)(=O)N FS-1493 Cc1c(nc(o1)c2ccccc2)CCO FS-1494 Cc1c(nc(s1)c2ccccc2)CCO FS-1495 CCn1c(cc(n1)C)C(=O)O FS-1496 c1ccc2c(c1)OCC(O2)CN FS-1497 c1ccn(c1)c2ccsc2CO FS-1498 c1cc2c(cc1Br)CCO2 FS-1499 c1ccc2c(c1)cc(s2)CO FS-1500 c1csc2c1[nH]cnc2=O FS-1501 c1csc2c1ncnc2N3CCNCC3 FS-1502 CC(C)(C)c1cc2c(s1)c(=O)nc[nH]2 FS-1503 CC(=O)c1c(cc(s1)C(C)(C)C)N FS-1504 c1ccnc(c1)c2ccc(s2)C(=O)O FS-1505 Cc1c(c(n[nH]1)C)c2ccccc2C(=O)O FS-1506 CC(=O)Nc1ccc(cn1)N FS-1507 COc1ccc(c(c1)OC)F FS-1508 Cc1csc(c1Cl)C(=O)O FS-1509 Cc1csc(c1N)C(=O)OC FS-1510 Cc1csc(c1Cl)C(=O)OC FS-1511 c1cc(cc(c1)Br)N2CCNCC2 FS-1512 c1cn(cn1)CCN2CCNCC2 FS-1514 Cc1cccnc1N2CCNCC2 FS-1515 c1cc(ccc1C(F)(F)F)N2CCNCC2 FS-1516 CC(=O)Nc1ccc(cc1)CO FS-1517 CC(=O)Nc1ccc(cc1)CC#N FS-1518 c1ccc2c(c1)cc(s2)C(=O)O FS-1519 COc1ccc(c(c1)OC)Br FS-1520 COc1ccc(cc1Br)CC#N FS-1521 c1ccc(c(c1)CCC(=O)O)Br FS-1522 c1cc2c(cc1Cl)cc(o2)C(=O)O FS-1523 COc1ccc(c(c1)OC)Cl FS-1524 c1cc(c(cc1Cl)O)C(=O)O FS-1525 c1cc(c(cc1Cl)CO)O FS-1526 COc1ccc(cc1Cl)C(=O)O FS-1527 Cc1ccc(c(c1)Cl)OC FS-1528 Cc1cccc(c1C(=O)O)Cl FS-1529 Cc1cc(ccc1C(=O)O)Cl FS-1530 Cc1cc(ccc1Cl)C(=O)O FS-1531 Cc1ccc(cc1C(=O)O)Cl FS-1532 Cc1c(cccc1Cl)CN FS-1533 Cc1cc(ccc1CN)Cl FS-1534 Cc1ccc(cc1CN)Cl FS-1535 c1ccc(c(c1)n2ccnc2)Cl FS-1536 c1cc(cc(c1)Cl)n2ccnc2 FS-1537 c1cc(ccc1n2ccnc2)Cl FS-1538 c1ccc(c(c1)CCC(=O)O)Cl FS-1539 c1ccc(c(c1)CCC#N)Cl FS-1540 COc1cc(cc(c1)OC)CC#N FS-1541 Cc1ccc(c(c1)C)NC(=O)N FS-1542 CCOc1ccc(cc1)C(=O)C FS-1543 COc1ccc(cc1F)CC#N FS-1544 Cc1cc(ccc1O)C(=O)O FS-1545 c1ccc(c(c1)CCC(=O)O)O FS-1546 Cc1cc(ccc1OC)C(=O)O FS-1547 Cc1cc(ccc1OC)CC(=O)O FS-1548 COc1ccc(cc1)n2cc[nH]c2=S FS-1549 CNc1ccccc1C(=O)N FS-1550 COC(=O)c1ccccc1C#N FS-1551 Cc1cccc(c1)CCC(=O)O FS-1552 Cc1ccc(cc1)CCC(=O)O FS-1553 Cc1cccc(c1)NC(=O)N FS-1554 CSc1ccc(cc1)CC#N FS-1555 c1ccc2c(c1)cccc2C(=O)N FS-1556 CC(=O)c1ccc(cc1)Oc2ccccc2 FS-1557 c1ccc(c(c1)C(=O)N)C(=O)O FS-1558 CCCOc1ccccc1C#N FS-1559 Cc1cccc(c1)n2ccnc2 FS-1560 COc1cc(cc(c1)OC)N2CCNCC2 FS-1561 CC(c1ccccc1)N2CCCNCC2 FS-1562 CCc1ccccc1N2CCNCC2 FS-1563 CC(C)(C)c1ccc(cc1)N2CCNCC2 FS-1564 c1ccc(c(c1)C(=O)O)N2CCNCC2 FS-1565 c1ccc(c(c1)N2CCNCC2)Cl FS-1566 c1cc(ccc1CN2CCNCC2)Cl FS-1567 Cc1cccc(n1)N2CCNCC2 FS-1568 c1cc(sc1)CCN2CCNCC2 FS-1569 c1cnccc1CCN2CCNCC2 FS-1570 c1ccc2c(c1)ccnc2C(=O)O FS-1571 c1cc(ccc1N2CCNCC2)Br FS-1572 CCc1ccc(c(c1)C(=O)C)OC FS-1573 Cc1ccnc2c1cc(cc2)OC FS-1574 Cc1cc(c(c(c1)C)CN2CCNCC2)C FS-1575 Cc1cc(cc(c1)N2CCNCC2)C FS-1576 Cc1ccc(cc1)CN2CCNCC2 FS-1577 c1cc(ccc1CN2CCNCC2)F FS-1578 Cc1cccc(c1)C(C(=O)O)O FS-1579 c1ccc(c(c1)F)S(=O)(=O)CCO FS-1580 Cc1cc(c(cc1Cl)C(=O)C)OC FS-1581 CC(=O)c1cc(ccc1OC)Cl FS-1582 CC(=O)c1cc(ccc1OC)F FS-1583 CC(=O)c1cc(ccc1OC)Br FS-1584 Cc1cc(c(cc1C)OC)C(=O)C FS-1585 Cc1cc(c(c(c1)C(=O)C)OC)C FS-1586 c1ccc(c(c1)S(=O)(=O)CCO)Cl FS-1587 c1cc2c(cc1C#N)OC(O2)(F)F FS-1588 COc1cccc(c1C(=O)O)F FS-1589 C1COCCN1c2nnc(s2)S FS-1590 COCc1nnc(s1)S FS-1591 Cc1cc(n(n1)CCN(C)C)N FS-1592 Cc1ccc(c(c1)C)S(=O)(=O)C FS-1594 Cc1ccc(c(c1)S(=O)(=O)C)C FS-1595 Cc1cccc(c1S(=O)(=O)C)C FS-1596 Cc1ccc(cc1C)S(=O)(=O)C FS-1597 CS(=O)(=O)c1ccc(cc1)C(F)(F)F FS-1598 CCc1ccc(cc1)S(=O)(=O)C FS-1599 Cc1cccc(c1)S(=O)(=O)C FS-1600 Cc1cccc(c1SCCO)C FS-1601 Cc1cc(cc(c1)SCCO)C FS-1602 c1cc(ccc1C(F)(F)F)SCCO FS-1603 Cc1cccc(c1)SCCO FS-1604 Cc1c(csc1C(=O)O)Br FS-1605 c1csc(c1Br)C(=O)O FS-1606 c1ccc(c(c1)N2CCNCC2)Br FS-1607 c1ccc2c(c1)CC(C2)C(=O)O FS-1608 c1ccc(cc1)C2CCCNC2 FS-1609 c1ccn(c1)CCN2CCNCC2 FS-1610 c1ccc(c(c1)c2[nH]nnn2)Br FS-1611 c1ccc2c(c1)cc(s2)C(CN)O FS-1612 c1cc(ccc1C(=S)N)C(F)(F)F FS-1613 CCOc1ccc(cc1)c2cc([nH]n2)N FS-1614 Cc1c(c(sc1c2ccccc2)C(=O)OC)N FS-1615 c1cc(ccc1C(=O)N2CCNCC2)O FS-1616 c1ccc(c(c1)C(=O)N2CCNCC2)Cl FS-1617 CC(C)c1ccc(cc1)C(C)N2CCNCC2 FS-1618 CC(C)c1ccc(cc1)N2CCNCC2 FS-1619 Cc1ccc(cc1)S(=O)(=O)N2CCNCC2 FS-1620 c1cocc1C(C(F)(F)F)O FS-1621 c1cc(oc1)C(C(F)(F)F)O FS-1622 C1CCc2c(c(n[nH]2)C(F)(F)F)C1 FS-1623 C1CCc2c(c(nc(n2)N)C(F)(F)F)C1 FS-1624 Cc1ccc(cc1)c2cc(c(s2)C(=O)OC)N FS-1625 Cc1c(c(sc1C(=O)O)SC)C=C FS-1627 c1cc(sc1c2ccno2)Br FS-1628 Cc1ccc(cc1)NC(C)C(=O)O FS-1629 Cc1ccc(cc1C)NC(C)C(=O)O FS-1630 c1ccc(cc1)NC2(CCCCC2)C(=O)O FS-1631 c1cc(oc1C(=O)O)Br FS-1632 c1ccc(cc1)C(=O)C2CC=CCC2C(=O)O FS-1633 c1ccc(cc1)C(=O)N2CCNCC2 FS-1634 c1csc(n1)N2CCNCC2 FS-1635 CC(=O)c1cc(cc(c1)O)O FS-1636 c1ccc(c(c1)C(=S)N)F FS-1637 c1ccc(c(c1)C(=S)N)O FS-1638 COc1ccc(c(c1)OC)C(=S)N FS-1639 COc1cc(cc(c1)OC)C(=S)N FS-1640 Cc1ccc(cc1)C(=S)N FS-1641 Cc1cccc(c1)C(=S)N FS-1642 Cc1ccccc1C(=S)N FS-1643 c1ccc(cc1)c2csc3c2nc[nH]c3=O FS-1644 Cc1cc2c(=O)[nH]cnc2s1 FS-1645 CC(C)c1cc2c(=O)[nH]cnc2s1 FS-1646 c1ccc(cc1)c2cc3c(=O)[nH]cnc3s2 FS-1647 c1[nH]c(=O)c2c3c(sc2n1)CCCC3 FS-1648 CCOC(=O)c1c2c(sc1N)CCC2 FS-1649 c1[nH]c(=O)c2c3c(sc2n1)CCC3 FS-1650 CCOC(=O)c1c(csc1N)C FS-1651 c1cc(ccc1c2csc3c2c(=O)[nH]cn3)F FS-1652 Cc1csc(c1C(=O)OC)N FS-1653 c1ccc(cc1)c2csc3c2c(=O)[nH]cn3 FS-1654 CC(C)(C)c1cc(n(n1)C)N FS-1655 CCOc1ccc(cc1)N2CCNCC2 FS-1656 CCOc1ccccc1N2CCNCC2 FS-1657 Cc1cccc(c1N2CCNCC2)C FS-1658 c1ccc(cc1)CCN2CCCNCC2 FS-1659 c1ccc(cc1)C2CNCCN2 FS-1660 CN1CCNC(C1)c2ccccc2 FS-1661 c1cc(cc(c1)C#N)CN2CCNCC2 FS-1662 Cc1ccc(cc1C)CN2CCNCC2 FS-1663 Cc1cc(nc(n1)N2CCNCC2)C FS-1664 CC(C)(C)c1cc(c(s1)C(=O)O)N FS-1665 c1ccc(c(c1)C(=O)O)Nc2cccc(c2)F FS-1666 Cn1c(c(cn1)c2ccccc2)N FS-1667 CC(=O)Nc1cccc(c1Cl)C(=O)O FS-1668 CC(C)(C)C(=O)c1ccsc1N FS-1669 CC(C)(C)c1ccc(s1)C(=O)OC FS-1670 C=CCOc1ccccc1F FS-1671 CC(C)(C)c1ccc(s1)C(=O)O FS-1672 CC(C)(C)c1ccc(s1)C#N FS-1673 CC(C)(C)c1ccc(s1)C(=O)N FS-1674 CC(=O)c1ccc2c(c1)CCO2 FS-1675 CC(=O)c1cc(cc(c1)OC)OC FS-1676 CC(C)C(=O)c1ccsc1N FS-1677 CC(C)C(=O)c1c2c(sc1N)CCCC2 FS-1678 Cc1cccnc1/C(=N/O)/N FS-1679 c1cc(cc(c1)F)N2C(=O)CCC2=O FS-1680 c1cc(ccc1C(F)(F)F)N2C(=O)CCC2=O FS-1681 COC(=O)c1c(c2c(cccc2s1)F)N FS-1682 COc1ccc(cc1F)CC(=O)O FS-1683 COC(=O)c1c(cc(s1)C(F)(F)F)O FS-1684 c1c(c(sc1C(F)(F)F)C(=O)O)O FS-1685 Cc1ccc(c(c1)C(=O)C(F)(F)F)O FS-1686 COc1ccc(cc1)C(=O)C(F)(F)F FS-1687 c1ccc(cc1)C2CCCCN2 FS-1688 c1ccc(cc1)S(=O)(=O)N2CCNCC2 FS-1689 Cc1ccc(cc1)c2ccc(s2)C(=O)OC FS-1690 c1ccnc(c1)SCC#N FS-1691 c1ccc(c(c1)OCC#N)Cl FS-1692 c1ccc2c(c1)c3c(s2)c(=O)[nH]cn3 FS-1693 CCCc1cc2c(=O)[nH]cnc2s1 FS-1694 COC(=O)c1c(c2cc(ccc2s1)F)N FS-1695 COc1ccc(cc1F)CCO FS-1696 Cc1cc(ccc1Cl)CO FS-1697 Cc1ccc(c(c1)OC)CO FS-1698 Cc1cc(ccc1CO)OC FS-1699 CCCc1ccc(cc1)CO FS-1700 Cc1cc(ccc1CCO)Cl FS-1701 Cc1cc(cc(c1OC)C)C(=O)C FS-1702 CCSc1ccc(cc1)C(=O)C FS-1703 Cc1cc(cc(c1OC)C)C(=O)O FS-1704 Cc1ccc(c(c1)OC)C(=O)O FS-1705 COc1ccc2cc(ccc2c1)C(=O)O FS-1706 Cc1cccc(c1)C(=O)C(F)(F)F FS-1707 CCSc1ccc(cc1)C(=O)C(F)(F)F FS-1708 CC(C)Oc1cccc(c1)C(=O)C(F)(F)F FS-1709 CSc1ccc(cc1)C(=O)C(F)(F)F FS-1710 CC(=O)c1ccc(cc1)Oc2ccccc2F FS-1711 CC(=O)c1ccc(cc1)Oc2ccc(cc2)F FS-1712 C1CNC=C(C1C(F)(F)F)C#N FS-1713 c1ccc(cc1)CN2CCC(=O)CC2 FS-1714 c1ccc(cc1)CN2C[C@H]3C[C@@H]2CN3 FS-1715 c1cc(ccc1CN2C[C@@H]3C[C@H]2CN3)Cl FS-1716 c1cc(cc(c1)Cl)CN2C[C@H]3C[C@@H]2CN3 FS-1717 c1cc(ccc1CN2C[C@@H]3C[C@H]2CN3)F.C(=O)(C(F)(F)F)O.C(=O)(C(F)(F)F)O FS-1718 c1cc(ccc1CN2C[C@H]3C[C@@H]2CN3)C#N FS-1719 COc1ccc(cc1)CN2C[C@H]3C[C@@H]2CN3 FS-1720 c1cc(c(nc1)N)C(F)(F)F FS-1722 c1cc(cc2c1cc[nH]2)C(=O)O FS-1724 CS(=O)(=O)c1ccc2ccn(c2c1)O FS-1725 c1cc2c(cc1CC(=O)O)CCO2 FS-1726 CC(C)Oc1cccc(c1)CN FS-1727 CC(C)Oc1ccc(cc1)CN FS-1728 CS(=O)(=O)c1cccc(c1)CN FS-1729 c1cc2c(cc1Cl)CCN2 FS-1730 c1cncc(c1C(F)(F)F)C(=O)N FS-1731 c1cc(cc2c1cc[nH]2)Cl FS-1732 CN(C)c1cccc(c1)CN FS-1733 CN(C)c1ccccc1CN FS-1734 CS(=O)(=O)c1ccc(cc1)CC#N FS-1735 COC(=O)c1cccc(c1)C(=O)N FS-1736 Cn1ccc2c1cc(cc2)C(=O)OC FS-1737 CC(C)(C)Oc1c(cccn1)CN FS-1738 c1ccc(cc1)C(=O)Cc2ccncn2 FS-1739 c1ccc(cc1)C(Cc2cnccn2)O FS-1740 c1ccc(cc1)C(Cc2cnc3ccccc3n2)O FS-1741 c1cc2c(cc1C(=O)O)CCCC2=O FS-1742 c1ccc2c(c1)c(c[nH]2)C3=CCNCC3 FS-1743 c1csc2c1sc(c2)C(=O)O FS-1744 Cc1c(c2ccccc2n1C)C#N FS-1745 c1cc2c(cc1CCC(=O)O)CCO2 FS-1746 CN(C)c1ccc(cc1)CN FS-1747 Cc1c(c(c(nc1C)S)C#N)C FS-1749 Cc1ccc(cc1S(=O)(=O)C)Br FS-1750 Cc1cc(ccc1S(=O)(=O)C)F FS-1751 CS(=O)(=O)c1ccc2cc[nH]c2c1 FS-1752 CS(=O)(=O)c1ccc(cc1)N2CCNCC2 FS-1753 Cc1c(cc2cnccc2n1)C(=O)C FS-1754 c1ccc2c(c1)n3cc(nc3s2)CO FS-1755 c1cc2cc3c(nc2nc1)CCNC3 FS-1756 COc1ccc(cc1)c2cc(sc2)C(=O)O FS-1757 c1cc2c(cc1F)CCN2C(=O)CCC(=O)O FS-1758 CC(C)(CC(=O)O)n1cccc1 FS-1759 c1ccc(cc1)CN2CCC(=O)NCC2 FS-1760 CS(=O)(=O)c1ccc2c(c1)CCN2 FS-1761 CC(c1ccc(cc1)S(=O)(=O)C)N FS-1762 c1ccc2c(c1)c(c[nH]2)C3CCNCC3 FS-1763 c1ccc2c(c1)CC(=O)N2C3CCNCC3 FS-1764 Cc1cc(n(n1)c2ccccc2)C(=O)O FS-1765 CC(=O)c1ccc(cc1)SC FS-1766 c1ccc(cc1)CN2CCCC(C2)(F)F FS-1767 c1ccc(c(c1)C(=O)C(F)(F)F)O FS-1768 CCc1cc(ccn1)C(=S)N FS-1770 Cc1cc(sc1)C(=O)OC FS-1771 Cc1cc(sc1)/C(=N/O)/N FS-1772 c1ccc(cc1)c2csc(n2)O FS-1773 CCN1CCc2c(sc(c2C(=O)OC)N)C1 FS-1774 COc1ccc(cc1)C(=O)N2CCNCC2 FS-1775 CN1CCc2c(sc(c2C(=O)OC)N)C1 FS-1776 Cc1ccc(cn1)C(=O)OC FS-1777 c1ccc2c(c1)nc(s2)Br FS-1778 c1cc2c(cc1Cl)nco2 FS-1779 c1cc2c(cc1Cl)CC(=O)N2 FS-1780 Cc1cc(sc1C)C(=O)O FS-1781 CCCC(=O)c1cccs1 FS-1782 Cc1ccc(cc1)S(=O)(=O)n2ccnc2 FS-1783 CS(=O)(=O)Cc1ccc(cc1)C(F)(F)F FS-1784 c1cc(ccc1CS)C(F)(F)F FS-1785 CS(=O)(=O)c1ccc(cn1)C(F)(F)F FS-1786 CS(=O)(=O)c1c(cccn1)C(F)(F)F FS-1787 CS(=O)(=O)c1ccc(c2c1cccc2)F FS-1788 c1cc2c(ccc3c2c(c1)C(=O)OC3=O)Cl FS-1789 CCOc1ccc(cn1)Br FS-1790 Cc1ccc(c(c1)O)C(=O)O FS-1791 Cc1nnc(s1)Br FS-1792 CCOc1cccc(c1C#N)F FS-1794 Cc1ccc(c(c1)OC)C(=O)OC FS-1795 c1ccc2c(c1)CCNC2c3ccncc3 FS-1796 c1ccc2c(c1)CCNC2CC3CCNCC3 FS-1797 c1ccnc(c1)NCc2cccnc2 FS-1798 Cc1ccnc(c1)NC(=O)c2ccncc2 FS-1799 c1ccc2c(c1)cccc2CCO FS-1800 c1ccc2c(c1)nc(s2)S FS-1801 c1cc(ccc1C2CNCCN2)F FS-1802 Cc1cc(ccc1O)C(=O)C FS-1803 c1cc2c(c(c1)C(F)(F)F)NC(=O)C2=O FS-1804 c1cc2c(cc[nH]2)cc1Br FS-1805 CC1CN(CCN1)Cc2ccccc2 FS-1806 Cc1cccc(c1)C(=O)N2CCNCC2 FS-1807 Cc1ccc(cc1)C(=O)N2CCNCC2 FS-1808 c1cc(ccc1C#CCO)C#N FS-1809 c1cc(c(cc1Cl)C#N)O FS-1810 c1ccc2c(c1)nc(s2)CCC(=O)O FS-1813 c1ccc(cc1)C(=O)NC2CCNCC2 FS-1814 Cc1cc(n2c(n1)nc(n2)N)c3ccccc3 FS-1815 c1ccc(cc1)c2ccc(o2)CO FS-1816 COc1ccc2c(c1)nc([nH]2)CO FS-1817 c1ccc(cc1)c2cc([nH]n2)O FS-1818 c1cc2c(cc1Cl)nc(cc2O)O FS-1819 CCc1c(cc(c(n1)S)C#N)C FS-1820 CCC(=O)c1ccc2c(c1)OCCO2 FS-1821 c1cnccc1c2[nH]c(nn2)S FS-1822 c1cc(sc1)C2NCCS2 FS-1823 Cn1c(nnc1S)c2ccc(cc2)F FS-1824 C1CC1c2nnc(n2C3CC3)S FS-1825 c1c([nH]nc1C(F)F)C2CC2 FS-1826 CCn1c(nnc1S)C2CC2 FS-1827 Cc1ccc(cc1)N2C(=O)C=CC2=O FS-1828 c1ccc2c(c1)nc3n2CCN3 FS-1829 CC1CNc2ccccc2NC1=O FS-1830 COc1cccc(c1)C2=NNC(=O)C2 FS-1831 c1ccc2c(c1)NC(=O)C3N2CCC3 FS-1832 c1cc2c(cc1Br)C(=O)OC2 FS-1833 COC(=O)c1c(c[nH]n1)Cl FS-1834 CCOC(=O)c1c(c(nn1C)C)Br FS-1835 CCOC(=O)c1c(c(n(n1)C)C)Cl FS-1836 Cn1cc(c(n1)C(=O)OC)Br FS-1837 Cn1c(c(cn1)Cl)C(=O)OC FS-1838 CCOC(=O)c1ccc2c(c1)c(c([nH]2)C)C FS-1839 c1cc(cc(c1)C(=O)O)c2c[nH]nc2 FS-1840 c1cc(c(cc1C(=O)O)N2CCCCC2)Cl FS-1841 c1cc(ccc1c2csc(n2)N)C(=O)O FS-1842 c1ccc(c(c1)c2csc(n2)N)C(=O)O FS-1843 c1cnccc1CCC(=O)O FS-1845 c1ccc2c(c1)ncn2CCC(=O)O FS-1846 Cc1ccc(cc1)C2CC2C(=O)O FS-1847 CCn1c(cc(n1)C(=O)O)C(F)(F)F FS-1848 CCn1c(cc(n1)C(F)(F)F)C(=O)O FS-1849 CCCn1c(ccn1)C(=O)O FS-1850 Cc1c(c(n(n1)C(C)C(=O)O)C)Br FS-1851 Cc1c(c(n(n1)CC(=O)O)C)Cl FS-1852 CC(C(=O)O)n1cc(cn1)Br FS-1853 c1c(nn2c1NCCC2C(F)(F)F)C(=O)O FS-1854 CCC(C(=O)O)n1cc(cn1)Br FS-1855 CC(C)(C(=O)O)n1cc(cn1)Br FS-1856 Cc1cc(nn1CC(C)C(=O)O)C(F)(F)F FS-1857 c1c(csc1C(=O)O)Br FS-1858 c1cc(ccc1c2cc([nH]n2)C(=O)O)Cl FS-1859 c1cn(nc1C(=O)O)C(F)F FS-1860 Cn1c(cc(n1)C(=O)O)C(F)(F)F FS-1861 c1c(n(nc1C(F)(F)F)CC(=O)O)C2CC2 FS-1862 Cc1cc(n(n1)CCC(=O)O)C FS-1863 c1c(cn(n1)CCC(=O)O)Br FS-1864 Cc1c(cn(n1)C(C)C(=O)O)Br FS-1865 Cc1ccn(n1)CCC(=O)O FS-1866 c1c(c(n[nH]1)C(=O)O)Br FS-1867 c1cc(cc(c1)C(=O)O)Cn2cccn2 FS-1868 Cc1ccccc1C(C(=O)O)O FS-1869 Cc1c(cc(o1)C2CC2)C(=O)O FS-1870 c1ccc(cc1)c2cc([nH]n2)C(=O)O FS-1871 CC(C)(C)c1cc([nH]n1)C(=O)O FS-1872 Cc1nc2cc(ccc2s1)C(=O)O FS-1873 c1ccc(cc1)C(C(=O)O)N2CCCC2 FS-1874 c1ccc(cc1)C(C(=O)O)N2CCCCC2 FS-1875 c1ccc2c(c1)[nH]c(n2)CC(=O)O FS-1876 c1cc(ccc1c2cc([nH]n2)C(=O)O)F FS-1877 c1ccc(c(c1)c2cc([nH]n2)C(=O)O)Cl FS-1878 CN1Cc2cccc(c2C1=O)C(=O)O FS-1880 c1cc2c(cc1CC(=O)O)sc(n2)N FS-1881 Cn1c2ccc(cc2n(c1=O)C)C(=O)O FS-1882 Cc1nc2ccccc2n1CCC(=O)O FS-1884 CCc1nc2ccccc2n1C(C)C(=O)O FS-1885 COc1ccc(c2c1cccc2)C(=O)O FS-1886 Cc1ccc(n1c2ccc(c(c2)C(=O)O)O)C FS-1887 Cc1ccc(cc1)c2ccc([nH]2)C(=O)O FS-1888 c1ccc2c(c1)ccc(n2)SCC(=O)O FS-1889 Cc1ccc2c(c1)C3C=CCC3C(N2)C(=O)O FS-1890 Cc1ccc(n1c2cccc(c2)C(=O)O)C FS-1891 c1ccnc(c1)SCC(=O)O FS-1892 c1ccc2c(c1)cnn2CCC(=O)O FS-1893 c1ccnc(c1)CCC(=O)O FS-1895 c1ccc(cc1)C2CC2C(=O)O FS-1896 CCn1c(c(cn1)CN2CCNCC2)C FS-1897 CCn1c(c(cn1)Cl)CNC FS-1898 CCn1cc(c(n1)CNC)Cl FS-1899 CNCc1c(cnn1C)Cl FS-1900 CCn1c(c(c(n1)C)CNC)C FS-1901 COc1cccc(c1)CN2CCNCC2 FS-1902 c1cc(sc1)C(=O)N2CCNCC2 FS-1903 c1cc(cc(c1)Cl)C(=O)N2CCNCC2 FS-1904 CCn1c(c(cn1)CNC)C FS-1905 CN(Cc1ccccc1)C2CCNCC2 FS-1906 c1ccc2c(c1)nc(o2)N3CCNCC3 FS-1907 c1ccc(cc1)CNC2CCS(=O)(=O)C2 FS-1908 c1ccc(cc1)NCc2ccncc2 FS-1909 c1ccc(cc1)NCc2cccnc2 FS-1910 c1ccc(cc1)NCc2ccccn2 FS-1911 c1ccc(cc1)CN2CCCNC2 FS-1912 c1ccc(cc1)C2CCC(CC2)N3CCNCC3 FS-1913 c1cc2n(c(=O)c1)C[C@@H]3C[C@H]2CNC3 FS-1914 CCOC(=O)C1c2ccccc2CCN1 FS-1915 c1cc(cc(c1)F)C(=O)NC2CCNCC2 FS-1916 c1cc(ccc1C(=O)NC2CCNCC2)F FS-1917 Cc1ccc(o1)CNC(C)C FS-1918 CC(C)NCc1nccn1C FS-1919 COc1ccc(c(c1)F)c2csc(n2)N FS-1920 CC(=O)Nc1cccc(c1)c2csc(n2)N FS-1921 Cc1ccccc1c2csc(n2)N FS-1922 CN(c1ccc(cc1)O)C(=S)N FS-1923 Cc1cc2c(cc1NC(=O)C)nc(s2)N FS-1924 c1c(=O)[nH]c(nc1N2CCOCC2)N FS-1925 c1cc2c(cc1CNC(=N)N)OCO2 FS-1926 c1cnccc1C(=O)NCCN FS-1927 CCC(c1ccc(c(c1)C)C)N FS-1928 CCOC(=O)c1c(cn[nH]1)N FS-1929 c1cc(cc(c1)Cl)Cn2cc(cn2)N FS-1930 Cc1cccc(c1)Cn2cc(cn2)N FS-1931 CC(C)(C)c1cc(n[nH]1)CN FS-1932 Cc1cc(n(n1)Cc2ccccc2)N FS-1933 c1cn(nc1C2CC2)CCN FS-1934 CCn1c(c(cn1)c2csc(n2)N)C FS-1935 Cc1c(cn(n1)C)c2csc(n2)N FS-1936 CCn1cc(cn1)c2csc(n2)N FS-1937 CCn1cc(c(n1)C)c2csc(n2)N FS-1938 Cc1cc(nc2c1c(c(s2)C#N)N)C FS-1939 CCn1cc(c(n1)C(=O)NC)N FS-1940 c1ccc(cc1)Cn2cnc(n2)N FS-1941 CC(c1cccc(c1)n2cccc2)N FS-1942 Cc1ccc(cc1)Cn2cnc(n2)N FS-1943 c1ccc(c(c1)Cn2cnc(n2)N)Cl FS-1944 c1cc(ccc1Cn2cnc(n2)N)Cl FS-1945 CCn1cc(c(n1)C)C(C)N FS-1946 Cc1c(cn(n1)CCCN)Br FS-1947 CCn1c(c(cn1)Cl)CN FS-1948 CCn1cc(c(n1)CN)Cl FS-1949 Cc1c(c2ccccc2[nH]1)CCN FS-1950 c1ccc(c(c1)Cn2cc(cn2)N)Cl FS-1951 Cc1ccccc1Cn2ccc(n2)N FS-1952 c1cc(ccc1Cn2cc(cn2)N)Cl FS-1953 c1ccc(c(c1)Cn2cc(cn2)N)F FS-1954 C1CCc2c(sc(c2C#N)N)CC1 FS-1955 c1ccc(cc1)Cn2cc(cn2)N FS-1956 C1Cc2c(sc(c2C#N)N)C1 FS-1957 Cc1c(c(n(n1)Cc2ccccc2)C)N FS-1958 CCn1c2ccccc2nc1N FS-1959 c1cc(ccc1c2cnnc(n2)N)F FS-1960 c1ccc(cc1)CN2CCCC(C2)CN FS-1961 Cc1cnn(c1N)Cc2ccccc2 FS-1962 Cc1cc2c(cc1Cl)nc(s2)N FS-1963 COC(=O)c1c(c2cc(ccc2[nH]1)F)N FS-1964 CCC(C)n1c(cc(n1)O)N FS-1965 CC(C)CC(c1[nH]c2ccccc2n1)N FS-1966 CC(c1[nH]c2ccccc2n1)N FS-1967 c1ccc(c(c1)c2csc(n2)N)O FS-1968 c1c(nc(s1)N)CN2CCCCC2 FS-1969 Cc1cc(=O)n2c([nH]1)nc(n2)N FS-1970 c1ccc2c(c1)nc(n2CCN3CCCCC3)N FS-1971 CC(C)Cc1nnc(s1)N FS-1972 c1cnc(nc1)N2CCC(CC2)N FS-1973 CC(=O)c1ccc(s1)Cc2ccccc2 FS-1974 CC(=O)c1cccc(c1)OC(F)F FS-1975 c1cc(oc1)c2ccc(cc2)C#N FS-1976 c1cc(cc(c1)C(F)(F)F)C2CCCN2 FS-1977 c1ccc(cc1)CN2CCCC2C(=O)O FS-1978 CC(=O)Nc1ccc2c(c1)sc(n2)N FS-1979 CC(=O)c1ccc(cc1)OC(F)F FS-1980 c1cc(cc(c1)Br)C#CCO FS-1981 c1cc(c(nc1)c2ccc(cc2)C(=O)O)N FS-1982 c1ccc(c(c1)c2ccsc2)C(=O)O FS-1983 c1cc(sc1)c2ccc(o2)C(=O)O FS-1984 c1cc(oc1c2ccsc2)C(=O)O FS-1985 Cc1ccc(cc1C)NC(=O)C(=O)O FS-1986 c1cc(oc1)c2ccc(cc2)C(=O)O FS-1987 c1cc(ccc1c2ccc(o2)C(=O)O)F FS-1989 c1cc(ccc1NC2CCNC2)Cl FS-1990 c1cc(ccc1NC2CCNCC2)Cl FS-1991 c1ccc(cc1)CC2CCCCN2 FS-1992 c1ccc2c(c1)cccc2C3CCCN3 FS-1993 c1cc(cc(c1)F)C2CCCN2 FS-1994 Cc1ccc(cc1)C2CCCN2 FS-1995 Cc1cccc(c1)C2CCCN2 FS-1996 Cc1ccccc1C2CCCN2 FS-1997 c1cnccc1C2CCNCC2 FS-1998 Cc1ccc(cc1F)NC2CCNCC2 FS-1999 c1cc(ccc1C(F)(F)F)NC2CCNCC2 FS-2000 c1cc(cc(c1)F)NC2CCNCC2 FS-2001 c1cc2c(cc1NC3CCNCC3)OCO2 FS-2002 c1cc(cc(c1)NC2CCNC2)C(F)(F)F FS-2003 c1cc(c(nc1)c2ccc(cc2)F)N FS-2004 Cc1ccccc1c2c(cccn2)N FS-2005 CC(=O)c1ccc(cc1)c2ccsc2 FS-2006 c1ccc(cc1)NC(=O)C2CCCN2 FS-2007 c1ccc(cc1)NC(=O)[C@@H]2CCCN2 FS-2008 Cc1ccc(s1)C(=O)C(F)(F)F FS-2010 Cc1cc(c(cc1Cl)C)S(=O)(=O)N FS-2011 c1cc2c(cc1Br)COC2=O FS-2012 c1ccc(cc1)C(C2CCCCN2)O FS-2013 Cc1cc(cc(n1)C)C2CCOCC2 FS-2014 Cc1ccnc(c1)NCc2cccnc2 FS-2015 Cc1cc(ccn1)CCCO FS-2017 CC(=O)NCc1ccncc1 FS-2018 CCC(CO)c1ccccn1 FS-2019 c1ccnc(c1)NC(=O)c2ccncc2 FS-2020 Cc1cc(ccn1)C2CCOCC2 FS-2021 Cc1cccc(n1)C(=O)OC FS-2022 CC1(CCOCC1)c2ccncc2 FS-2023 CC(C)CC(C)(c1ccccn1)O FS-2024 c1ccc(cc1)CN2CCC(CC2)CN FS-2025 c1cc2c(cc1C(=O)C(F)(F)F)CCO2 FS-2026 Cn1ccnc1CCC(=O)O FS-2027 Cc1ccc(o1)C(F)(F)F FS-2028 Cc1cc(ccc1CC(=O)O)F FS-2029 c1cc(cc(c1)C(=O)O)C2CCNCC2 FS-2030 c1c(nc(o1)N)C(F)(F)F FS-2031 Cc1cc(nc(c1)O)C(F)(F)F FS-2032 c1cc(ncc1Br)C(=O)O FS-2034 c1cc(c(cc1O)F)C(=O)O FS-2035 CCc1cccc2c1NC(=O)C2=O FS-2036 c1c(cncc1Br)N FS-2037 c1c(n[nH]c1N)C(F)(F)F FS-2038 c1cc2c(cc1Cl)S(=O)(=O)NC2=O FS-2039 Cc1ccc(cc1)c2c(n3ccccc3n2)CN FS-2040 CC(=O)c1cc(cs1)Cl FS-2041 c1cc(ccc1C2CNCCN2)Br FS-2042 c1cc(cc(c1)Br)C2CNCCN2 FS-2043 COC(=O)c1ccc(cc1)c2ccncc2 FS-2044 COc1ccc(c(c1)Cl)C(=O)O FS-2045 c1cc(nc(c1)N2CCOCC2)C(F)(F)F FS-2046 c1cc(nc(c1)N2CCNCC2)C(F)(F)F FS-2047 c1cc(ccc1c2cnoc2N)Cl FS-2048 COC(=O)c1ccc2c(c1)CCO2 FS-2050 c1cnc(cc1C(F)(F)F)N2CCNCC2 FS-2051 CC(C)(C)c1cccc(c1)N2CCNCC2 FS-2052 COc1ccc(c(c1)Cl)C#N FS-2053 c1cc(cc(c1)S(=O)(=O)N2CCNCC2)F FS-2054 c1cc(ccc1CN)CN2CCOCC2 FS-2055 c1cc(cc(c1)N2CCOCC2)CN FS-2056 c1c(cc(cc1C(F)(F)F)O)C(=O)O FS-2057 c1cc2c(c(c1)Br)nc(s2)N FS-2058 CCc1cccc2c1nc(s2)N FS-2059 Cc1ccc(c2c1nc(s2)N)Cl FS-2060 Cc1c(ccc2c1nc(s2)N)Cl FS-2061 Cc1ccc(c2c1nc(s2)N)C FS-2062 Cc1cc2c(c(c1)Br)nc(s2)N FS-2063 Cc1ccc(c2c1sc(n2)N)Br FS-2064 Cc1cc(cc2c1nc(s2)N)Br FS-2065 c1cc(cc(c1)F)C2CNCCN2 FS-2066 c1ccc(c(c1)C2CNCCN2)Cl FS-2068 c1cc(cc(c1)Cl)C2CNCCN2 FS-2069 Cc1ccccc1c2cc([nH]n2)N FS-2070 Cc1ccc(cc1)c2c[nH]nc2N FS-2071 c1cc(ccc1c2c[nH]nc2N)Cl FS-2072 c1cc(ccc1c2c[nH]nc2N)Br FS-2073 COc1ccc(cc1)c2c[nH]nc2N FS-2074 c1cc(ccc1c2ccno2)Cl FS-2075 c1cc(ccc1c2ccno2)F FS-2076 CCn1c(cc(n1)C(=O)O)C FS-2077 Cc1cc(nn1Cc2ccccc2)C(=O)O FS-2078 Cc1cc(n(n1)c2ccccc2F)C(=O)O FS-2079 c1cc(ccc1c2ccon2)F FS-2080 COc1ccc(cc1)c2ccon2 FS-2081 c1cc(c(cc1CO)Br)O FS-2082 c1ccc2c(c1)[nH]c(n2)Br FS-2083 COc1cccc(c1C(=O)N)F FS-2084 COc1ccc(c(c1)C(=O)O)Cl FS-2085 CC(=O)c1c(cccc1F)O FS-2086 CC(=O)c1ccc(c(c1)C(F)(F)F)O FS-2087 CC(=O)c1ccc(c(c1)C(F)(F)F)OC FS-2088 COc1ccc(c(c1)C(F)(F)F)C(=O)O FS-2089 COc1cc(ccc1F)C#N FS-2090 COc1ccc(cc1Br)CO FS-2091 c1ccc2c(c1)nc(s2)C(=O)O FS-2092 CN1CCN(CC1)c2ccc(cc2)CN FS-2093 CN1CCN(CC1)c2ccc(cc2)C#N FS-2094 c1cc(c(cc1O)C(=O)O)Cl FS-2095 c1cc(c(cc1O)C(F)(F)F)C#N FS-2096 c1cc(c(cc1C#N)C(F)(F)F)O FS-2097 CCC(c1ccccc1F)O FS-2098 c1ccc(cc1)C(=O)N2CCC(CC2)C(=O)O FS-2099 c1cc(ccc1CN2CCNCC2)C#N FS-2100 c1cc(cc(c1)N2CCNCC2)C#N FS-2101 c1cc(ccc1C#N)N2CCC(CC2)C(=O)O FS-2102 c1c[nH]c(=O)c2c1scc2 FS-2103 c1cnc(c2c1scc2)N3CCNCC3 FS-2104 Cc1cc(nn1c2ccccc2)C(=O)O FS-2105 CC(=O)c1coc2c1cccc2 FS-2106 CS(=O)(=O)c1ccccc1N2CCNCC2 FS-2107 Cc1cc2ccc(cc2[nH]1)Cl FS-2108 CCS(=O)(=O)c1ccc(cc1)C(=O)C FS-2109 CCOC(=O)c1cc(cnc1)Br FS-2110 CC(=O)c1cc(ccc1O)OC FS-2111 c1cc2c(cc1F)c(=O)oc(=O)[nH]2 FS-2112 c1ccc(cc1)CN2CCC[C@H](C2)O FS-2115 c1cc(ccc1[C@H](CCO)N)Cl FS-2116 c1cc(ccc1c2ccncc2)C(=O)O FS-2117 Cc1cc(ccc1Br)S(=O)(=O)N FS-2118 Cc1ccc(c(c1)F)S(=O)(=O)N FS-2119 Cc1ccc(cc1F)S(=O)(=O)N FS-2120 Cc1ccc(cc1S(=O)(=O)N)F FS-2121 CC(C)c1ccc(cc1)S(=O)(=O)N FS-2122 c1ccc(cc1)Oc2ccc(cc2)S(=O)(=O)N FS-2123 CCCc1ccc(cc1)S(=O)(=O)N FS-2124 Cc1cccc(c1)S(=O)(=O)N FS-2125 Cc1ccc(c(c1)S(=O)(=O)N)F FS-2126 Cc1c(cccc1S(=O)(=O)N)F FS-2127 Cc1cc(ccc1F)S(=O)(=O)N FS-2128 Cc1cc(ccc1S(=O)(=O)N)Br FS-2129 Cc1ccc(cc1)CS(=O)(=O)N FS-2130 c1cc(ccc1OC(F)F)S(=O)(=O)N FS-2131 COc1cccc(c1CN)F FS-2132 c1cc2c(cc1C(F)(F)F)n(nn2)O FS-2133 Cc1cc(cc(c1)Cl)C#N FS-2134 Cc1cccc(c1F)C(=O)O FS-2135 Cc1c(sc(n1)c2cccc(c2)F)C(=O)O FS-2136 c1ccc2c(c1)cc(s2)CN FS-2137 c1ccc(cc1)C2(CCCNC2)O FS-2138 Cc1ccccc1C(=O)N2CCNCC2 FS-2139 c1cc(ccc1C(=O)O)N2CCNCC2 FS-2140 c1cc(nnc1N)N2CCOCC2 FS-2141 COc1cccc(c1F)C(=O)O FS-2142 CS(=O)(=O)c1ccc(c(c1)F)O FS-2143 c1cc(cnc1)N2CCNCC2 FS-2144 c1ccnc(c1)N2CCC(CC2)C(=O)O FS-2145 c1cnccc1N2CCCC(C2)C(=O)O FS-2146 c1cnccc1N2CCC(CC2)C(=O)O FS-2147 COc1c(cccc1F)C(=O)OC FS-2148 Cc1cc(cnc1O)Br FS-2149 Cc1cc(ncc1Br)O FS-2150 Cc1cnn(c1N)C2CCN(CC2)C FS-2151 COc1ccc2c(c1)C(=O)NC2 FS-2152 COC(=O)c1ccc(cn1)Br FS-2153 C1CNC(CN1)C(F)(F)F FS-2154 C[C@@H](CCc1ccccc1)O FS-2155 c1ccc2c(c1)ccc(n2)C(=O)O FS-2156 c1ccc2c(c1)cc(cn2)C(=O)O FS-2157 C1CC2(CCC(=O)CC2)OC1 FS-2158 COc1ccc(c(c1)Cl)O FS-2159 COC(=O)c1c(c[nH]n1)Br FS-2160 COc1c(cc(cn1)N)Br FS-2161 Cc1c(ccc(n1)OC)Br FS-2162 CCCn1cc(cn1)C(C)N FS-2163 c1cc(c(nc1)O)Br FS-2164 COc1c(cccn1)Br FS-2165 c1ccc2c(c1)nc(n2CCN3CCOCC3)N FS-2166 c1cc(ncc1Br)CO FS-2167 c1cc2c(c(c1)Cl)NC(=O)C2=O FS-2168 c1c(cnc(n1)O)Br FS-2169 c1cc(ccc1C(F)(F)F)N2CCC(CC2)O FS-2170 c1ccc2c(c1)c(n[nH]2)C(=O)O FS-2171 Cn1c2ccccc2c(n1)C(=O)O FS-2172 COc1ccc2c(c1)CC(=O)CC2 FS-2173 Cc1cc(c(s1)C(=O)OC)N FS-2174 Cc1c(sc(=S)[nH]1)CC(=O)O FS-2175 CC(=O)c1c2ccccc2[nH]n1 FS-2176 CC(=O)c1cc2ccccc2s1 FS-2177 c1c(ncc(n1)Br)N FS-2178 c1ccc(cc1)[C@@H]([C@@H](c2ccccc2)O)N FS-2179 CCC(=O)N1[C@@H](COC1=O)Cc2ccccc2 FS-2180 c1ccc(cc1)C(=O)N2CCC(=O)CC2 FS-2181 c1ccc(cc1)CNC2CCC(=O)CC2 FS-2182 c1ccc(cc1)CN2C[C@H]([C@@H](C2)O)O FS-2183 c1ccc(cc1)CN2CCOC[C@H]2CO FS-2184 c1cc2c(c(c1)Br)C(=O)OC2=O FS-2185 Cc1cc(cc(c1Br)C(=O)O)OC FS-2186 c1cc2cnccc2cc1Br FS-2187 COc1ccc2c(c1)sc(n2)Br FS-2188 c1cc2c(cc1Br)C(=O)CC2 FS-2189 c1cc2c(cc1Br)nccn2 FS-2190 c1cc(ccc1C2CCCN2)Br FS-2191 CCOC(=O)c1cnc(s1)Br FS-2192 c1cc2c(cc1Br)c(c[nH]2)C(=O)O FS-2193 Cc1ccc(c(c1)F)C(=O)O FS-2194 Cc1cccc(c1C(=O)O)F FS-2195 Cc1c(cccc1F)C(=O)O FS-2196 Cc1cc(cc(c1)F)C(=O)O FS-2197 Cc1cc(ccc1C(=O)O)F FS-2198 CC(C)n1c(ccn1)C(=O)O FS-2200 c1cc(ccc1CN)N2CCCC2 FS-2201 c1ccnc(c1)C2CC2C(=O)O FS-2202 c1ccc(cc1)CN2CCOCC2=O FS-2203 Cc1cc(cc(c1)C(=O)O)C FS-2204 CC(C)c1ccccc1C(=O)O FS-2206 Cc1cc(cc(c1)Cl)C(=O)O FS-2207 Cc1cc(ccc1Cl)C(=O)OC FS-2208 CN(C)c1ccc(c(c1)Cl)C(=O)O FS-2209 COc1c(cn(n1)CC(F)F)N.Cl FS-2210 Cc1cc(ccc1OC)S(=O)(=O)N FS-2211 COc1ccc(cc1Cl)S(=O)(=O)N FS-2212 Cc1ccc(c(c1)Cl)C(=O)O FS-2213 Cc1ccc(cn1)C(F)(F)F FS-2214 COc1ccc2c(c1)NC(=O)C2=O FS-2215 C#Cc1ccc(s1)C(=O)O FS-2216 CS(=O)(=O)c1ccc(cc1)CO FS-2217 c1ccc(c(c1)CN)C(=O)O FS-2218 COc1cc(ccc1C(=O)O)Br FS-2219 c1cc2c(cc1C(=O)N)nc[nH]2 FS-2220 Cc1c(cn(n1)CCC#N)Br FS-2221 c1cc(ccc1N2CC(CC2=O)N)F.Cl FS-2222 c1cc(ccc1C2(CCOCC2)C(=O)O)F FS-2223 c1ccc(cc1)OC2CCCC2 FS-2224 CN(C)c1ccc(cc1)CCN FS-2225 c1cc2cnccc2c(c1)Br FS-2226 c1cc(cc2c1ccnc2)Br FS-2227 c1cc2ccncc2c(c1)Br FS-2228 Cc1cc(cc(c1)OC)C(=O)O FS-2229 Cc1ccc(cc1C(=O)O)OC FS-2230 c1cc(ccc1N2CCOCC2)Br FS-2231 COc1ccc(c(c1)Br)C(=O)O FS-2232 COc1ccc(c(c1)Br)C(=O)OC FS-2233 COc1c(cccc1Br)C(=O)O FS-2234 Cc1ccccc1c2[nH]c(nn2)S FS-2235 c1cc(cc(c1)F)c2ccc(nc2)N FS-2236 c1cc(ccc1C#N)c2ccc(nc2)N FS-2237 Cc1ccc(cc1)c2ccc(nc2)N FS-2238 c1cc(cc(c1)C(=O)O)C2CC2 FS-2239 c1cc2c(c(c1)F)NC(=O)C2 FS-2240 c1cc2cc[nH]c2c(c1)Cl FS-2241 c1cc2c(cc1C#N)CNCC2 FS-2242 c1cc2ccc(nc2c(c1)O)O FS-2243 c1ccc2c(c1)C[C@H](N2)C(=O)O FS-2244 CSc1ccc2c(c1)cc[nH]2 FS-2245 c1ccc2c(c1)ccnc2Cl FS-2246 c1cc2c(cc1O)CNCCN2 FS-2247 c1cc2c(c(c1)Cl)C(=O)CC2 FS-2248 CCOC(=O)c1c(c[nH]c1C)C FS-2249 C[C@@H](c1cccc2c1cccc2)O FS-2250 c1ccc2c(c1)nc(s2)CC#N FS-2251 Cn1ccc2c1ccc(c2)C(=O)O FS-2252 Cc1cccc(c1)C2CCNCC2 FS-2253 COc1cccc2c1CC(=O)CC2 FS-2254 Cc1ccc2c(c1)c(=O)oc(=O)[nH]2 FS-2255 COc1ccc2c(c1)CCC(=O)N2 FS-2256 c1ccc2c(c1)CCNC2C(=O)O FS-2257 COc1cccc2c1nc(s2)N FS-2258 c1cc2c(c(c1)Cl)C(=O)CCC2 FS-2259 c1cc2c(cc1Cl)NC(=O)C2=O FS-2260 c1ccc2c(c1)c(c3c(n2)CCC3)N FS-2261 c1cc(cc(c1)Cl)[C@H](CCO)N FS-2262 Cc1c(c2ccccc2[nH]1)CC(=O)O FS-2263 COc1ccc2c(c1)CCCCC2=O FS-2264 COc1cccc2c1cc([nH]2)C(=O)O FS-2265 COc1cccc2c1[nH]cc2C(=O)O FS-2266 COc1ccc2c(c1)c(c[nH]2)C(=O)O FS-2267 c1ccc(cc1)CN2CC(C2)C(=O)O FS-2268 CN1CCC(CC1)(c2ccccc2)O FS-2269 COc1ccc2c(ccnc2c1)Cl FS-2270 c1cc2c(cc1Cl)c(c[nH]2)C(=O)O FS-2271 c1cc2c(cco2)cc1Br FS-2272 c1cc(ccc1[C@@H](CC(=O)O)N)Cl FS-2273 COC(=O)[C@@H](c1ccc(cc1)Cl)N FS-2274 c1ccc(cc1)CN2CCC[C@H]2C(=O)O FS-2275 c1cc(ccc1C2CCCNC2)C(=O)O FS-2276 c1cc(ccc1C2CCNCC2)C(=O)O FS-2277 C[C@H]([C@H](c1ccccc1)O)N2CCCC2 FS-2278 c1cc2cccnc2c(c1)Br FS-2279 c1cc(ccc1[C@@H]2CCNC[C@H]2CO)F FS-2280 c1cc2c(c(c1)Br)C(=O)CC2 FS-2281 c1c(cnc2c1oc(=O)[nH]2)Br FS-2282 CC(=O)Nc1ccc(cn1)Br FS-2283 CN1CCN(CC1)C(=O)c2ccc(cc2)O FS-2284 c1ccc(cc1)CN2CC[C@H]([C@@H](C2)CO)N FS-2285 CCOC(=O)c1c([nH]c2c1ccc(c2)F)C FS-2286 CCOC(=O)c1c([nH]c2c1cc(cc2)F)C FS-2287 c1cc2c(c(c1)Br)NC(=O)C2=O FS-2288 c1cc2c(cc1Br)CNCCN2 FS-2289 COC(=O)C1Cc2c3ccccc3[nH]c2CN1 FS-2290 c1ccc(cc1)COC(=O)N2CCC(CC2)N FS-2291 C[C@H]1CNCCN1C(=O)OCc2ccccc2 FS-2292 c1ccc(cc1)COC(=O)N2CCCC(C2)O FS-2293 CC(=O)Nc1ccc(cc1OC)Br FS-2294 c1ccc(cc1)COC(=O)N2CCCC(C2)C#N FS-2295 c1ccc(cc1)COC(=O)N2CCC(CC2)C#N FS-2296 c1cc(ccc1c2cncnc2)O FS-2297 c1cc(cc(c1)C(=O)O)c2ccc(nc2)N FS-2298 Cn1ccc(cc1=O)C(=O)O FS-2299 CC(C)Oc1ccccc1C(=O)O FS-2300 c1cc2n(c1)CCNC2c3ccc(cc3)F FS-2301 c1ccn2cc(nc2c1)C(=O)O FS-2303 CC(=O)CCN1CCOCC1 FS-2304 Cn1c(cc(n1)c2cccs2)C(=O)O FS-2305 c1ccc(c(c1)N2CC(CC2=O)N)F FS-2306 CCCc1[nH]c2ccccc2n1 FS-2307 c1cc(cc(c1)N2CCOCC2)C(=O)O FS-2308 Cc1cc(ccc1Br)OCC(=O)O FS-2309 Cc1ccc(cc1)c2cc(nn2C)C(=O)O FS-2310 CN(c1ccccc1)C(=O)CC#N FS-2311 c1ccc(cc1)C2CC(=O)NC(=N2)N FS-2312 c1cc2c(c(c1)F)c(no2)N FS-2313 c1cc(ccc1C2CCCN2)Cl FS-2314 c1cc(c2cccnc2c1)CN FS-2316 c1cc2c(ccnc2c(c1)Br)CO FS-2317 c1c(cnc2c1CC(=O)N2)Br FS-2318 c1cc(sc1C(=O)O)C(F)(F)F FS-2319 c1cc(oc1C(=O)O)C(F)(F)F FS-2320 c1ccc2c(c1)[nH]c(n2)N3CCNCC3 FS-2321 c1cc2c(c(c1)Br)COC2=O FS-2322 c1cc(c(cc1O)C(F)(F)F)C(=O)N FS-2323 CC1(CNCCN1c2ccc(cc2)OC)C FS-2324 CN(C)c1cccc(n1)C(F)(F)F FS-2326 CC(C)Oc1ccc(cc1)NC(=O)C FS-2327 CN1CCC(CC1)C(=O)c2ccccc2F FS-2328 CNc1cccc(n1)C(F)(F)F FS-2329 CN(C)c1cc(cc(c1)F)OC FS-2330 c1cc(c(cc1C(F)(F)F)O)C(=O)O FS-2331 COc1ccc2c(c1)C(=O)C(=O)N2 FS-2332 c1cc(nc2c1ccc(n2)O)N FS-2333 c1cncc(c1C(=O)O)Cl FS-2334 c1ccc(cc1)C2CCC(CC2)N FS-2335 c1c(csc1C#N)Br FS-2336 COc1ccc(cc1O)Br FS-2337 Cc1cccc(n1)C(F)(F)F FS-2338 CC(=O)c1ccc(cc1)S(=O)(=O)N FS-2339 c1cc(ccc1c2ccc(nc2)C(=O)O)F FS-2340 c1cc(cc(c1)F)C2(CC2)C(=O)O FS-2341 CC(C)Oc1ccc(cc1)S(=O)(=O)N FS-2342 Cn1c(cc(n1)N)C(F)(F)F FS-2343 CC(=O)c1cc(cnc1)Br FS-2344 CC(C)(C)c1cccc(c1)S(=O)(=O)N FS-2345 Cc1ccc(c(c1)C)S(=O)(=O)N FS-2346 Cc1ccc(cc1C)S(=O)(=O)N FS-2347 Cn1c(cc(n1)C(F)(F)F)N FS-2348 Cc1ccc(c(c1)C)C(=O)O FS-2349 Cc1ccc(c(c1)S(=O)(=O)N)OC FS-2350 Cc1ccc(cc1C)C(=O)O FS-2351 Cc1ccc(c(c1)C(=O)O)C FS-2352 COc1cccc(c1C(=O)OC)F FS-2353 COc1cc(ccc1F)CC#N FS-2354 c1cc(c2cc[nH]c2c1)C(=O)O FS-2355 Cc1c(c(ccc1C(=O)O)OC)C FS-2356 c1cc(ccc1CCC(=O)O)C(F)(F)F FS-2357 c1cc(ncc1Br)C#N FS-2358 c1ccc(cc1)c2nccs2 FS-2359 c1(nnc(o1)N)C(F)(F)F FS-2360 c1cc(ccc1c2nnc(s2)N)Cl FS-2361 Cc1cc(ccc1Br)NC FS-2362 CNc1cccc(c1)C(F)(F)F FS-2363 CNc1ccc(cc1)C(F)(F)F FS-2364 C#Cc1ccc2c(c1)CCC2=O FS-2365 CS(=O)(=O)c1ccc(cc1)C#C FS-2366 c1ccc2c(c1)c(ccc2F)O FS-2367 c1ccc(c(c1)C2CC2)C(=O)O FS-2368 CC(=O)c1ccc(nc1)OC FS-2369 c1cc(ccc1c2nccs2)C(=O)O FS-2370 c1c[nH]c2c1c(nc(n2)N)O FS-2371 c1cc2c(cc1Br)[nH]c(=O)[nH]2 FS-2372 c1c(cnc2c1nc[nH]2)Br FS-2373 c1cnc2c(n1)cc(cn2)Br FS-2374 c1cc2c(cc1Br)nn[nH]2 FS-2375 CCc1nc2ccccc2c(=O)o1 FS-2376 Cc1cc(=O)[nH]c(n1)SC FS-2377 CC(=O)c1cccc(c1OC)F FS-2378 c1c(ncc(n1)Br)O FS-2379 c1cc2ccc3cc[nH]c3c2nc1 FS-2380 CCOC(=O)C1=CNC(=O)NC1 FS-2381 c1cc(ccc1CN)n2ccnc2 FS-2382 C[C@@H](c1cccc2c1cccc2)N FS-2383 Cn1c2cc(ccc2cn1)Br FS-2384 Cn1cc2ccc(cc2n1)Br FS-2385 CC(=O)c1cccc(c1O)F FS-2386 CC(=O)c1ccc(c(c1)O)F FS-2387 CC(=O)c1csc(n1)Cl FS-2388 c1cc(nc(c1)C(F)(F)F)C(=O)O FS-2389 CCOC(=O)c1cncs1 FS-2390 Cc1nc2cc(ccc2s1)Br FS-2391 c1cc2c(cc1Br)C(=O)NC2=O FS-2392 CCOC(=O)c1cc(c[nH]1)C FS-2393 c1ccc2c(c1)ccc(c2C#N)C#N FS-2394 CC1=CC=CC(CC1=O)(C)C FS-2395 Cc1c(cc(cn1)Cl)C(=O)OC FS-2396 c1ccn2c(c1)c(cn2)Br FS-2397 CS(=O)(=O)c1ccc2cn[nH]c2c1 FS-2398 Cc1cc2c([nH]1)ccc(c2F)O FS-2399 CC(C)c1cc(n[nH]1)C(C)C FS-2400 c1ccc2cc(c(cc2c1)C(=O)O)O FS-2401 Cc1nc2c3ccccc3ccc2s1 FS-2402 Cc1nc2cc3ccccc3cc2o1 FS-2403 Cc1cccc(c1Cl)C#N FS-2404 Cc1cc(ncc1Br)OC FS-2405 c1cc(c(c(c1)O)Br)O FS-2409 Cc1ccc2cc([nH]c2c1)C(=O)O FS-2410 CCOC(=O)c1cc([nH]n1)C FS-2411 CN1CCN(CC1)c2cccc(c2)C(=O)O FS-2412 CCOC(=O)c1cc2cc(ccc2[nH]1)Cl FS-2413 CCOC(=O)c1cc2ccc(cc2[nH]1)Cl FS-2414 Cc1cc(cc(c1)O)C(=O)O FS-2415 c1ccc(cc1)CN2CCCC2=O FS-2416 COC(=O)c1cccc(c1)C#C FS-2417 CC(=O)c1ccccc1C(=O)O FS-2418 c1ccc(cc1)CN2CCC(CC2)C(=O)N FS-2419 C1CC1C(=O)N2CCNCC2 FS-2420 c1ccc2c(c1)ccc(n2)CN FS-2421 c1ccc(cc1)S(=O)(=O)c2ccccn2 FS-2422 c1ccc2c(c1)[nH]c(n2)CCN FS-2423 c1ccc(cc1)Cn2c3ccccc3nc2CN FS-2424 c1ccc(cc1)Cn2cc(cn2)C#N FS-2425 c1ccc(cc1)CN2CCC(=O)C2 FS-2426 c1cc(cnc1)Cn2cc(cn2)Br FS-2427 c1cc(c(nc1)C#N)Br FS-2428 c1cc(c(cc1C#N)F)C(=O)O FS-2429 CC(=O)c1ccc(cn1)Br FS-2430 c1ccc2c(c1)cc(nc2Cl)C(=O)O FS-2431 c1cc2c(cc1Br)CCNC2=O FS-2432 c1c(cnc2c1[nH]c(=O)c(=O)[nH]2)Br FS-2433 c1c2c(c(cn1)Br)[nH]cn2 FS-2434 c1cc(c(cc1C(=O)O)O)Br FS-2435 c1ccc2c(c1)c(c[nH]c2=O)Br FS-2436 COc1cc(ccc1Br)C(=O)O FS-2437 Cc1cc(cnc1C(=O)O)Br FS-2438 c1cc2c(cc1Br)NC(=O)CO2 FS-2439 C[C@@H](c1ccccc1Br)N FS-2440 c1cc2c(c(c[nH]2)Br)nc1 FS-2441 c1cc2c(cc1Br)cncn2 FS-2442 c1ccc2c(c1)c(ccn2)Br FS-2443 c1c(n2c(n1)CNCC2)Br FS-2444 c1cc2ncnn2cc1Br FS-2445 c1ccc(cc1)COC(=O)N2CC(C2)O FS-2446 c1ccc(cc1)COC(=O)N2CCC(C2)O FS-2447 c1ccc(cc1)COC(=O)N2CC[C@H](C2)O FS-2448 c1ccc(cc1)COC(=O)N2CCNCC2 FS-2449 c1cc2c(ccs2)cc1Cl FS-2450 c1cc(nn2c1ncc2)Cl FS-2451 c1cc2c(cc1Cl)c(n[nH]2)C(=O)O FS-2452 c1cc2c(c(c1)Cl)C(=O)C(=O)N2 FS-2453 c1cc2cnccc2cc1Cl FS-2454 c1cc2cnccc2c(c1)Cl FS-2455 c1ccc(c(c1)C(C(=O)O)O)Cl FS-2456 c1cc(ccc1C[C@H](C(=O)O)N)Cl FS-2457 c1cc(cc(c1)Cl)C[C@H](C(=O)O)N FS-2458 c1cc(ccc1C2CNCCN2)Cl FS-2459 c1cc(cc(c1)Cl)C2CSCCN2 FS-2460 c1cc2c(cc1Cl)[nH]c(=O)[nH]c2=O FS-2461 c1cc(sc1C#N)Br FS-2462 c1cc2c(cc1O)sc(n2)C#N FS-2463 c1cc2cnccc2cc1C#N FS-2464 c1cc(cc(c1)C#N)CC(=O)O FS-2465 Cc1cc(ncc1Br)N FS-2466 Cc1cc(cnc1C(=O)OC)Br FS-2467 c1cc(c(nc1)N)Br FS-2468 CC1(Cc2c(nc(s2)N)C(=O)C1)C FS-2469 c1ccc2c(c1)C(=O)NC(N2)c3ccncc3 FS-2470 C1[C@@H]2C[C@@]3(C[C@H]1C[C@](C2)(C3)N)C(=O)O FS-2471 Cc1cc(c2c(c1)NC(C3C2C=CC3)C(=O)O)C FS-2472 C1CCC2(CCNCC2C1)O FS-2473 Cc1cc(n(n1)c2cccc(c2)C(=O)O)C FS-2474 CCC1c2c(c3ccccc3[nH]2)CC(N1)C(=O)O FS-2475 CC(c1nc2ccccc2s1)N FS-2476 c1cc2cc(ccc2nc1)C(=O)O FS-2477 c1cn(ccc1=O)CC(=O)O FS-2478 c1ccc2c(c1)CC(O2)CO FS-2479 c1cc(ccc1c2nnc(o2)S)F FS-2480 Cn1c2ccccc2nc1CCN FS-2481 c1ccc(cc1)c2cc(c(s2)N)C(=O)O FS-2482 COc1ccc(cc1)C2(CCCC2)CN FS-2483 C1CNCCC12C(=O)NC(=O)N2 FS-2484 Cc1ccc(n1c2ccc(c(c2)O)C(=O)O)C FS-2485 c1cc(sc1)c2cc([nH]n2)C(=O)O FS-2486 Cc1ccc2nc(cn2c1)C(=O)O FS-2487 CNC[C@@]12C[C@H]3C[C@@H](C1)C[C@@H](C2)C3 FS-2488 COc1ccc2ccccc2c1CN FS-2489 Cc1ccc2c(c1)c(n[nH]2)C(=O)O FS-2490 C1CCC(CC1)(C(=O)O)N2CCCCC2 FS-2491 c1ccc2c(c1)NC(C(=O)N2)CC(=O)O FS-2492 CN1CCN(CC1)CC(c2ccccc2)N FS-2493 c1cc2c(cc1Cl)nc([nH]2)CN.Cl.Cl FS-2494 Cc1csc(n1)N2CCNCC2 FS-2495 c1ccc(cc1)C2(CCCC2)N FS-2496 c1cc2cc([nH]c2c(c1)F)C(=O)O FS-2497 CCc1c(c([nH]n1)C(=O)O)C FS-2498 Cc1c(n[nH]c1C(=O)O)c2cccs2 FS-2499 Cc1c(sc(n1)N(C)C)C(=O)O FS-2500 Cn1cc(c2c1cccc2)CCO FS-2501 c1ccc(c(c1)C2(CC2)CN)Cl FS-2502 Cc1cc(c2c(c1)cc(n2C)C(=O)O)C FS-2503 c1ccc(cc1)C2c3cccn3CCN2 FS-2504 Cc1cc(c2c(c1)nc([nH]2)CCC(=O)O)C FS-2505 c1cnn(c1N)C2CCNCC2 FS-2506 Cn1c2ccccc2n(c1=O)CC(=O)O FS-2507 Cc1nc(c(s1)c2ccccc2)C(=O)O FS-2508 c1cc(ccc1CN)N2CCCCC2 FS-2509 CC(c1ccc(cc1)N2CCCCC2)N FS-2510 c1cc(ccc1CN)CN2CCCCC2 FS-2511 c1ccc(cc1)Cn2c(nnn2)S FS-2512 c1cc2c(cc1C(=O)O)CCC2 FS-2513 COc1ccc2c(c1)C(C(=O)N2)CCN FS-2514 COc1cccc(c1)c2cc([nH]n2)N FS-2515 CC(C)c1cc(cs1)C(=O)O FS-2516 c1cc2c(cc1S(=O)(=O)N)CCN2 FS-2517 c1cc(ccc1CCN)C(F)(F)F FS-2518 Cn1c2ccccc2nc1Cl FS-2519 c1cc2c(cc1Br)C(=O)C(=O)N2 FS-2520 Cc1c(c(sc1C(=O)C)N)C(=O)OC FS-2521 Cc1c(sc2c1c(nc(n2)C)S)C FS-2522 C1CCc2c(c(c(s2)N)C(=O)O)C1 FS-2523 CC1(Cc2cc(ccc2O1)CO)C FS-2524 c1cc2cccnc2c(c1)CC(=O)O FS-2525 c1ccc(cc1)C2COCCN2 FS-2526 Cc1cccc(c1Br)S(=O)(=O)N FS-2527 Cc1cc2c(o1)cc(n2C)C(=O)O FS-2528 Cc1ccc(c(c1)Cl)C#N FS-2529 Cc1cc(ccc1Cl)C#N FS-2530 Cc1ccc(cc1Cl)C#N FS-2531 Cc1cc(ccc1C(=O)N)Br FS-2532 Cc1cc(cc(c1)Cl)CN FS-2533 C1[C@@H]2C[C@]3(C[C@@H](C2)C[C@@H]1C3)C(=O)O FS-2534 COc1ccc(cc1Br)CC(=O)O FS-2535 COc1ccc(cc1CC(=O)O)Br FS-2536 COc1ccc(cc1CC#N)Br FS-2537 c1cc(sc1C(=O)O)Br FS-2538 Cc1cccc(c1Cl)C(=O)O FS-2539 Cc1ccc(c(c1)C(=O)O)Cl FS-2540 Cc1ccc(cc1Cl)C(=O)O FS-2541 Cc1c(cccc1Cl)C#N FS-2542 Cc1cc(ccc1C#N)Cl FS-2543 Cc1ccc(cc1C#N)Cl FS-2544 c1cc2c(cc1Cl)C(=O)OC2=O FS-2545 CC(=O)c1c(cccc1O)O FS-2546 Cc1ccc(cc1OC)CC#N FS-2547 c1ccc2c(c1)cccc2CC(=O)O FS-2548 c1ccc(cc1)c2cccc(=O)[nH]2 FS-2549 c1cc2c(cc1Cl)nn[nH]2 FS-2550 c1cc2c(cc1Cl)n(nn2)O FS-2552 Cc1ccc(cc1)C[C@H](C(=O)O)N FS-2553 c1cc2ccc3cccnc3c2nc1.O FS-2554 c1cc(=O)[nH]cc1C(F)(F)F FS-2555 CC1=CC(=O)c2ccccc2C1=O FS-2556 CCOC(=O)c1cnc([nH]1)N FS-2557 CCOC(=O)c1ccncc1N FS-2558 CCOC(=O)c1cc(cnc1C)Br FS-2559 c1c(sc(n1)Br)CO FS-2560 c1cc2c(c(c1)F)C(=O)CC2 FS-2561 c1cc(cc(c1)F)N2C[C@@H](OC2=O)CO FS-2562 CN1CC[C@H]([C@@H](C1)CO)c2ccc(cc2)F FS-2563 Cc1c(cc(cn1)N)Br FS-2564 Cc1c(cc(cn1)Br)N FS-2565 c1cncc(c1N)Br FS-2566 COc1c(ncc(n1)Br)N FS-2567 c1c[nH]c2c1cncc2Br FS-2568 c1cc2c(cc1Cl)C(=O)CC2 FS-2569 Cc1cc(sc1C(=O)O)Br FS-2570 Cc1c(c[nH]n1)Br FS-2571 c1cc(nnc1N)Br FS-2572 c1cc(ccc1CN)OC2COC2 FS-2573 c1cc2c(cc1C(=O)O)nc[nH]2 FS-2574 c1cc(c2c(c1)[nH]cn2)C(=O)O FS-2575 c1cc(c2cccnc2c1)C(=O)O FS-2576 c1ccc2cnc(cc2c1)C(=O)O FS-2577 c1cc2c(c(c1)C(=O)O)CCCC2 FS-2578 c1cc2c(cc1C(=O)O)cn[nH]2 FS-2579 c1ccc(c(c1)CS(=O)(=O)N)F FS-2581 Cc1ccc(cc1C(=O)O)O FS-2582 c1cn2cc(nc(c2n1)N)Br FS-2583 Cc1ccc(cc1)S(=O)(=O)NN FS-2584 Cc1ccc(cc1C(=O)OC)OC FS-2585 c1cnc(cc1N)C(F)(F)F FS-2586 c1ccc(c(c1)CC(=O)O)O FS-2587 c1ccc(cc1)c2ccnc(c2)C(=O)O FS-2588 Cc1ccc(cn1)CC(=O)O FS-2589 c1cc(c(nc1)S)C(=O)O FS-2590 c1cnc(cc1C(=O)O)C(F)(F)F FS-2591 c1ccc(cc1)c2cccc(n2)C(=O)O FS-2592 c1c(cncc1C(F)(F)F)C(=O)O FS-2593 c1cc2c(cc1F)CCC(O2)C(=O)O FS-2594 Cc1ccc(cc1C)C(=O)OC FS-2595 Cc1ccc(cc1Cl)C(=O)OC FS-2596 Cc1ccncc1C(=O)OC FS-2597 c1cc(c(cc1O)Cl)C(=O)O FS-2598 c1cc(cc(c1)C(=O)O)c2ccncc2 FS-2599 COc1cc(cc(c1)Cl)C(=O)O FS-2600 COc1cc(ccc1Cl)C(=O)O FS-2601 c1ccnc(c1)c2ccc(cc2)C(=O)O FS-2602 Cc1cccc(c1C(=O)O)O FS-2603 c1c(cncc1Cl)C(=O)O FS-2604 c1ccc(c(c1)CN)N2CCOCC2 FS-2606 Cc1c(nc(s1)N)C(=O)C FS-2607 CC(C)(C#N)c1cccc(c1)OC FS-2608 Cc1cc(ccc1F)C(=O)C FS-2609 c1ccc(cc1)C2(CCC2)C#N FS-2610 c1c(cc(cc1O)Cl)C#N FS-2611 c1cc(ccc1C#N)N2CCCCC2 FS-2612 CC(=O)c1ccc(cc1C(F)(F)F)O FS-2613 c1cc2c(ccnc2N)cc1Br FS-2614 c1cn2cc(cc(c2n1)N)Br FS-2616 CNc1cccc2c1cccc2 FS-2617 c1ccc2c(c1)c(no2)Cl FS-2618 Cn1cc2cc(ccc2n1)Br FS-2619 c1c(n2c(n1)CCCC2)Br FS-2620 c1c(cnc2c1CCC2)Br FS-2621 c1cc2c(cc1Br)nc[nH]c2=O FS-2622 c1cn2cc(ncc2n1)Br FS-2623 c1cn2c(n1)cncc2Br FS-2624 c1c(cnc2c1ncs2)Br FS-2626 c1cc(c(cc1Br)CO)O FS-2627 Cc1cnc(c(c1OC)C)CO FS-2628 CC(=O)c1ccc(cc1)N(C)C FS-2629 c1cc(ccc1C#N)N2CCOCC2 FS-2630 c1cc(ncc1C#N)N2CCCCC2 FS-2631 Cc1cc(cnc1OC)Br FS-2632 Cn1ccc(cc1=O)Br FS-2633 Cc1cnc(s1)Br FS-2634 CC1CCc2cc(ccc2N1)F FS-2635 c1ccc2c(c1)cncc2Br FS-2636 c1cnc2ccsc2c1O FS-2637 c1cc2cc(ccc2cc1C#N)O FS-2638 c1cc2c(cc1F)nc[nH]c2=O FS-2639 c1cc2c(cc1C(F)(F)F)cn[nH]2 FS-2640 Cc1c(ccs1)C(=O)OC FS-2641 CCOC(=O)c1ccc(s1)Cl FS-2642 COC(=O)c1ccoc1Br FS-2643 COC(=O)c1csc(n1)N FS-2644 CCOC(=O)c1cc([nH]n1)N FS-2645 COC(=O)c1ccc2c(c1)nc[nH]2 FS-2646 CCOC(=O)c1cc2ccccc2cn1 FS-2647 c1cc2c(cc1F)[nH]c(=O)[nH]2 FS-2648 c1ccc(cc1)CC2CCCNC2 FS-2649 Cc1ccc(cc1N2CCNCC2)Cl FS-2650 Cc1cccc(c1NC(=O)CN2CCNCC2)C FS-2651 COc1cccc2c1CCC(=O)C2 FS-2652 c1ccc2c(c1)cccc2CC#N FS-2653 c1ccc(cc1)CN2C3CCC2CC(=O)C3 FS-2654 CC1CN(NC1=O)c2ccccc2 FS-2655 c1ccc(cc1)Cn2ccnc2 FS-2656 c1ccc(cc1)C2C(=O)NC(=O)N2 FS-2657 c1ccc2c(c1)[nH]c(n2)S FS-2658 CC(C)(C)OC(=O)c1c[nH]nc1 FS-2659 c1(=O)c(n[nH]c(=O)[nH]1)Br FS-2660 c1cc(ncc1Br)C(=O)N FS-2661 c1c(cnc(c1C(=O)O)N)Cl FS-2662 COc1cnc(cn1)Br FS-2663 COc1ccc(cc1)Cn2c(ccn2)N FS-2664 c1cc2c(cc1CN)OCCO2 FS-2665 CCOC(=O)c1ccc([nH]1)N FS-2666 Cc1c(c(nc(n1)N)C)Br FS-2667 COc1ccc(cc1C#N)Cl FS-2668 Cc1ccc(cc1O)C(=O)O FS-2669 Cc1cccc2c1nc([nH]2)C(=O)O FS-2670 c1ccc2c(c1)CC(O2)C(=O)O FS-2671 Cc1c(c(ncn1)C)Br FS-2672 c1cc2c(cc1Cl)[nH]c(=O)[nH]2 FS-2673 c1ccc(cc1)COc2cc[nH]c(=O)c2 FS-2674 c1ccc(c(c1)C(=O)O)NC2=CCCCC2 FS-2675 COC(=O)c1c(cccn1)N FS-2676 c1c(cncc1Br)C(=O)N FS-2677 c1cc2c(cc1C(=O)O)ncs2 FS-2678 c1cc2c(c(c1)Br)C(=O)C(=O)N2 FS-2679 CC(=O)c1ccc(nc1)C(F)(F)F FS-2680 Cc1cc(cc(c1C(=O)O)C)F FS-2681 c1cc2c(cc1O)CCC(=O)C2 FS-2682 c1ccc2c(c1)[nH]c(n2)C(F)F FS-2683 COC(=O)c1c(ccs1)Br FS-2684 COC(=O)c1cnc(s1)N FS-2685 COc1ccc(cc1)C2(CCC2)C#N FS-2686 c1cc2c(cc1Br)scn2 FS-2687 c1ccn2c(c1)cc(n2)C(=O)O FS-2688 Cc1ccc(cc1O)C(=O)OC FS-2689 c1cc(c(cc1C(=O)O)O)Cl FS-2690 c1cc2c(cc1Br)nc[nH]2 FS-2692 CCOC(=O)c1ccccc1C#N FS-2693 c1cc(cc(c1)F)CN2CC(CC2=O)C(=O)O FS-2694 c1cc(ccc1CN)N2CCOCC2 FS-2695 Cc1cnc(c(n1)Br)N FS-2696 COc1cc(ccc1C#N)Br FS-2698 c1cc2c(c(c1)Br)ncs2 FS-2699 c1ccc(cc1)CN2CCOC(C2)C#N FS-2700 c1ccc2c(c1)c(c[nH]2)CC(=O)N FS-2701 COc1cc(ccc1O)CC=C FS-2702 CC1COc2ccc(cc2N1)Br FS-2703 c1ccc2c(c1)C(=O)C=CC2=O FS-2704 c1cc2c(cc1C(F)F)OCCO2 FS-2705 c1cc2c(c(c1)F)c(=O)[nH][nH]2 FS-2706 c1ccc2c(c1)c(ccc2F)CN FS-2707 COc1ccc(c(c1)Cl)CN FS-2708 CCOc1cccc(c1CN)F FS-2709 c1cc(ccc1C#N)N2CCCC2 FS-2710 c1ccc(cc1)N2CCCC2=O FS-2711 c1cc(ccc1CCN)OC(F)(F)F FS-2712 Cc1cnc(cn1)C(F)(F)F FS-2713 c1cc(ccc1C#N)NC2CCCCC2 FS-2714 CCOc1ccccc1CN FS-2715 CCOC(=O)c1c(ccnc1C)C FS-2716 c1cc(ccc1CO)N2CCOCC2 FS-2718 CC1(C(=O)Nc2c(cccn2)O1)C FS-2719 c1cc(ncc1Br)CC(=O)O FS-2720 COCc1ccc(cc1)CN FS-2721 c1cc2nc(nn2c(c1)Br)N FS-2722 C1COCc2c1nc(s2)N FS-2723 c1cc(nnc1)N2CCNCC2 FS-2724 c1cc2c(cc1Br)nc(s2)N FS-2725 c1ccc(cc1)CN2CC3CNCC3C2 FS-2726 c1ccc(cc1)CN2CC3CCCNC3C2 FS-2727 c1ccc(cc1)c2cc3c([nH]2)cccn3 FS-2728 c1ccc2c(c1)cncc2C#N FS-2729 c1cnc(nc1)n2cc(cn2)Br FS-2730 c1cnn(c1)c2ncc(cn2)Br FS-2731 c1cc(nc2c1cc(cn2)Br)N FS-2732 c1c(nc(s1)Br)C#N FS-2733 c1c(sc(n1)Br)C#N FS-2734 c1c(ncc(n1)Br)C#N FS-2735 c1c(c(ncn1)O)Br FS-2736 c1csc2c1[nH]c(=O)[nH]c2=O FS-2737 c1c(cnc(n1)N2CCC2)Br FS-2738 c1c(cnc2c1c(=O)[nH]c(n2)N)Br FS-2739 c1cc2nncn2cc1Br FS-2740 c1c(cnc2c1NC(=O)CO2)Br FS-2741 COc1ncc(c(n1)N)Br FS-2742 c1ccc(cc1)COc2nccc(n2)N FS-2743 c1[nH]c(=O)c2c(n1)[nH]nc2Br FS-2744 c1c(c2c(s1)c(=O)nc[nH]2)Br FS-2745 COc1ccc2c(c1)scn2 FS-2746 c1cnc(c(n1)N)Br FS-2747 Cc1[nH]c(=O)c2cc(ccc2n1)Cl FS-2748 Cc1[nH]c(=O)c2cc(ccc2n1)Br FS-2749 c1c(nc2c(n1)nc(s2)N)Br FS-2750 c1cc2c(cc1Cl)c(ncn2)N FS-2751 c1nc(c(s1)CO)Br FS-2752 COc1ccc(c(n1)OC)N FS-2753 Cc1cccc(c1NC(=O)C2CCCCN2)C FS-2754 Cc1ccc(nc1)N2CCNCC2 FS-2755 COc1ccc2c(c1)sc(=O)[nH]2 FS-2756 c1cc(c(cc1O)C#N)Br FS-2757 c1cc2c(cc1F)c(no2)N FS-2758 c1cc2c(cc1F)onc2N FS-2759 C#Cc1c(ncc(n1)Br)N FS-2760 c1cc2c(cc1Br)cno2 FS-2761 Cc1c2cc(ccc2[nH]n1)Br FS-2762 Cc1c2cc(ccc2[nH]n1)Cl FS-2763 Cc1c2ccc(cc2[nH]n1)OC FS-2764 CN1CCC2(CC1)CNc3c2cccc3 FS-2765 c1ccc2c(c1)ccnc2N3CCNCC3 FS-2766 c1ccc2c(c1)n(c(=O)o2)C3CCNCC3 FS-2767 c1cc(c2c(c1)OCC(=O)N2)O FS-2768 COc1cccc(c1C#N)Cl FS-2769 COc1cccc(c1C(=O)O)Cl FS-2770 c1ccc2cnc(cc2c1)Cl FS-2771 CCOC(=O)c1cnc(s1)Cl FS-2772 c1cc2cc(ccc2c(c1)C(=O)O)F FS-2773 c1ccc(cc1)C2CC(=O)c3ccccc3N2 FS-2774 c1ccc2c(c1)C(=O)CC(N2)c3ccc(cc3)F FS-2775 c1c(nc(s1)N)Br FS-2776 c1cc2c(cc1F)ncc(=O)[nH]2 FS-2777 c1cc2c(c[nH]c2nc1)CN3CCNCC3 FS-2778 c1c(c2cncnc2[nH]1)Br FS-2779 CN1CCN(CC1)c2nccc(n2)N FS-2780 c1cn2cnnc2c(n1)Cl FS-2781 Cc1nc(c2n1ccnc2)Br FS-2782 Cc1cn2ccnc(c2n1)Cl FS-2783 CCOC(=O)c1cc2c(s1)CCNC2 FS-2784 c1c(c2c([nH]1)c(=O)nc[nH]2)Br FS-2785 COC(=O)c1ccc(cn1)N FS-2786 Cc1c(cnc(n1)N)Br FS-2787 c1cc2c(cc1C#N)onc2N FS-2788 c1cc(c(cc1Br)CC#N)C#N FS-2789 c1cc(c(cc1Br)C#N)CC#N FS-2790 CCOC(=O)c1c(cc[nH]1)N FS-2791 c1ccc2cnc(cc2c1)CO FS-2792 c1cc(c2c(c1)OCCO2)O FS-2793 c1c(ncnc1N2CCOCC2)N FS-2794 CN1CCN(CC1)c2cc(ncn2)N FS-2795 c1c(nc2n1CCNC2)C(F)(F)F FS-2796 c1c(cnc2c1CCC(=O)N2)Br FS-2797 c1c(c2c([nH]1)nc[nH]c2=O)Br FS-2798 c1cc(c(c(c1)Br)O)C(=O)O FS-2799 COc1cccc2c1nc(nc2)N FS-2800 c1cc2c(c(c1)Cl)ncs2 FS-2801 c1cc(nn2c1ncc2N)Cl FS-2802 c1c(c(nn1C2CCCC2)N)C#N FS-2803 c1cc2c(cc1C#N)sc(n2)Cl FS-2804 c1cc2c(cc1F)C(=O)CCC2 FS-2805 c1cc2c(cc[nH]c2=O)cc1Br FS-2806 c1cc2c(c(c1)Br)[nH]cnc2=O FS-2807 Cc1c(c(ncn1)N)Br FS-2808 c1cn2c(cn1)ncc2Br FS-2809 CCCOc1ccc(nn1)N FS-2810 Cc1c(ncc(n1)Br)N FS-2811 c1ccc2c(c1)cnc(c2N)Br FS-2813 c1ccc2c(c1)cnc(c2N)Cl FS-2814 c1c(ncnc1Br)N FS-2815 Cc1cc(nc(n1)N)Br FS-2816 c1cc2c(cc1Br)C(=O)CCN2 FS-2817 c1c(ncnc1N)C(F)(F)F FS-2818 c1c(nc(cn1)Br)C#N FS-2819 Cc1nc2ccc(cc2s1)Br FS-2820 c1c(ncnc1N2CCNCC2)C(F)(F)F FS-2821 c1ccc(cc1)COc2cnc(nc2)Cl FS-2822 c1c(cnc(c1C#N)N)Br FS-2823 c1cc2cc(ccc2nc1)C#N FS-2824 c1cc2cc(ccc2nc1)CO FS-2825 c1c2c(cncc2Br)[nH]n1 FS-2826 c1cc2c(cc1Br)CCNC2 FS-2827 COc1ccc(cc1Br)O FS-2828 CCOC(=O)c1ccc2c(c1)cn[nH]2 FS-2829 c1ccc2c(c1)c(n[nH]2)Cl FS-2830 c1cnn2c1nc(cc2)Cl FS-2831 COc1cccc2c1CCCC2=O FS-2832 c1ccc2c(c1)COC23CCNCC3 FS-2833 c1ccc(cc1)n2c3c(cn2)CNCC3 FS-2834 c1cc(ccc1C2CNCCN2)C(F)(F)F FS-2835 c1ccc2cc(ccc2c1)C3CNCCN3 FS-2836 c1cc(sc1C2CNCCN2)Br FS-2837 c1cc(ccc1C2CNCCN2)O FS-2838 c1cc(ccc1C2CNCCN2)N3CCOCC3 FS-2839 COc1ccc2cc(ccc2c1)C3CNCCN3 FS-2840 c1cc(sc1)C2CNCCN2 FS-2841 c1ccc2c(c1)CCCC(=O)N2 FS-2842 COC(=O)c1ccc(c(c1)C#N)F FS-2843 c1cc(cc2c1ccc(n2)O)O FS-2844 c1cc2c(cc1C(=O)O)CCC(=O)N2 FS-2845 CCOC(=O)c1ccc(cn1)Br FS-2846 CCc1cc([nH]n1)C(=O)OC FS-2847 c1cc2c(ccnc2cc1Cl)N3CCNCC3 FS-2848 c1cc2c(cc[nH]2)c(c1)N3CCNCC3 FS-2849 c1ccc(cc1)c2cccnc2N FS-2850 c1c(cnc(c1N)CC(=O)O)Br FS-2851 c1cc2c(cc1Br)NC(=O)C2 FS-2852 c1c(nc(cn1)Br)N FS-2853 C1Cn2c(nc(n2)C(F)(F)F)CN1 FS-2854 CN1CCN(CC1)c2ccc(nc2)N FS-2855 c1cc2c(cc1Br)[nH]c(=O)cn2 FS-2856 c1ccc2c(c1)c(cc(=O)[nH]2)N FS-2857 Cn1c2cc(ccc2ncc1=O)Br FS-2858 c1cc2c(cc1Br)c(=O)ocn2 FS-2859 Cn1cc2cccc(c2n1)Br FS-2860 c1cc2ncc(n2nc1N)Br FS-2861 c1ccc2c(c1)c(ns2)N FS-2862 c1cnc(nc1N2CCOCC2)N FS-2863 COc1c2ncc(n2ccn1)Br FS-2864 Cc1ccc2c(c1)nc(cn2)Cl FS-2865 c1cc2c(cc1F)NCCO2 FS-2866 c1ccc2c(c1)c(=O)[nH]c(=O)[nH]2 FS-2867 c1cc2ncc(n2nc1)Br FS-2868 c1cc2c(cc1O)CC(=O)CC2 FS-2869 c1ccn2cc(nc2c1)Br FS-2870 c1cc(cc2c1ccnc2N)Br FS-2871 c1cc2c(cc1Br)ocn2 FS-2872 c1cc2cnc(cc2cc1Br)O FS-2873 Cc1cccc(c1NC(=O)[C@@H]2CCCCN2)C FS-2874 c1c2c(sc1C(=O)O)CCNC2 FS-2875 Cn1cnc2c1cc(cc2)C(=O)O FS-2876 CN1CCc2c(cc(cn2)N)C1 FS-2877 c1ccc2c(c1)CCCC2C(=O)O FS-2878 c1cc2c(c(n[nH]2)Br)nc1 FS-2879 c1cncc2c1[nH]nc2Br FS-2880 c1cc(=O)[nH]c2c1cc(cc2)Br FS-2881 c1c(cnc2c1CCN2)Br FS-2882 c1cc(cc2c1cc(cn2)C(=O)O)C(F)(F)F FS-2883 c1cc2c(cncn2)c(c1)Br FS-2884 COC(=O)c1cc2cc(cnc2[nH]1)Cl FS-2885 c1cncc2c1c(=O)[nH]c(=O)[nH]2 FS-2886 c1ccc2c(c1)cnc(n2)Cl FS-2887 c1cc2c(cc1Br)ncc(n2)O FS-2888 Cn1c2c(cccc2Br)cn1 FS-2889 c1cc2cn[nH]c2c(c1)C(=O)N FS-2890 c1cc2cn[nH]c2cc1Cl FS-2891 c1cnc2c(cnn2c1)Br FS-2892 c1cc2cc([nH]c2nc1)C(=O)O FS-2893 Cc1c(cccn1)C(=O)OC FS-2894 c1cc2c(cc1Br)C(=O)CCO2 FS-2895 Cc1cc(c(nc1)N)C(=O)OC FS-2896 Cc1cn2cc(ncc2n1)Br FS-2898 c1cc(c2nccn2c1)Br FS-2899 c1cc2c(cc1Br)C(=O)CO2 FS-2900 CCOc1ccc2ccc(cc2c1)O FS-2901 Cc1nc(cc(n1)Br)N FS-2902 c1ccc2c(c1)ccc(n2)CCO FS-2903 c1cn2c(cc1Br)ncn2 FS-2904 c1cc2ncnn2c(c1)Br FS-2905 Cc1c(ccc2n1ncn2)Br FS-2906 c1cc(c2nncn2c1)Cl FS-2907 Cn1ccc2c1ncc(n2)Br FS-2908 c1cc2c(cc1Br)OCCC2=O FS-2909 c1c(c(n[nH]c1=O)O)Br FS-2910 c1ccc2c(c1)c3c(o2)CNCC3 FS-2911 c1c2ncnn2cc(n1)Br FS-2912 COC(=O)c1cc(cnc1)N FS-2913 c1c(csc1Br)C(=O)O FS-2914 CCOC(=O)c1c(cccc1Cl)O FS-2915 CC(=O)c1c[nH]c2c1ccc(c2)OC FS-2916 c1cnc(nc1)N2CCC(CC2)O FS-2917 c1cc(ccc1CO)N2CCC(CC2)O FS-2918 c1ccnc(c1)CN2CCC(CC2)CO FS-2919 Cc1ccc(cc1)c2cnc(nc2)N FS-2920 COc1ccc(cc1)c2cnc(nc2)N FS-2921 c1cc(cc(c1)Cl)c2cc(n[nH]2)C(=O)O FS-2922 c1ccc2cc(ccc2c1)c3cc(n[nH]3)C(=O)O FS-2923 CCOC(=O)c1cn2cc(ccc2n1)N FS-2924 Cc1cccc2n1cc(n2)C(=O)O FS-2926 CCOC(=O)c1cn2cccc(c2n1)C FS-2927 Cc1ccc2cccc(c2n1)O FS-2928 c1cc2c(cc1C#N)scn2 FS-2929 c1cc2c(cc1Br)c(n[nH]2)C(=O)O FS-2930 c1cc2c(cc1C(F)(F)F)CCC2=O FS-2931 c1cc2c(c(c1)Cl)CCC2=O FS-2932 c1ccc2c(c1)cncc2Cl FS-2933 Cc1ccc2c(c1)c(cc(n2)O)O FS-2934 Cn1c2ccccc2c3c1CCCC3=O FS-2935 c1cnccc1N2CCCCC2 FS-2936 c1ccc2c(c1)c(ncn2)Br FS-2937 c1c(csc1Cl)C(=O)O FS-2938 c1c(cncc1Br)CO FS-2939 CCOC(=O)C1CCc2ccccc2N1 FS-2940 c1ccc(cc1)COc2cncc(n2)Cl FS-2941 C[C@@H]1CCN(C[C@@H]1NC)Cc2ccccc2 FS-2942 Cn1c2ccccc2n(c1=O)C3CCNCC3 FS-2943 c1csc(c1C(=O)O)Cl FS-2944 c1ccc2c(c1)cc(s2)C#N FS-2945 c1cn2cncc2cc1C(=O)O FS-2947 c1ccc(c(c1)C2CCCN2)F FS-2948 c1cc2c(cc1Br)c(c[nH]2)C#N FS-2949 c1c(cnc(c1N)O)Br FS-2950 Cc1cc(cnc1C(=O)O)Cl FS-2951 COc1ccc2c(n1)nc([nH]2)S FS-2952 Cc1cc(c(cn1)C(=O)O)N FS-2953 c1cc2c(cc1Cl)[nH]nc2C(=O)O FS-2954 c1ccc(c(c1)C2CCCN2)Br FS-2955 c1cncc(c1C(=O)N)Br FS-2957 COC(=O)c1ccc2c(c1)CCN2 FS-2958 c1cc2c(cc1Cl)C(=O)CCCN2 FS-2959 c1cc2c(cc1C#N)CCC2=O FS-2960 CC(C)CC1C(=O)NC(=O)N1 FS-2961 c1cc2c(cc1Br)CCCC2=O FS-2962 COC(=O)c1cc[nH]c(=O)c1 FS-2963 C1CCC(C1)N2CCCC(=O)C2 FS-2964 c1cc(c2cncn2c1)C(=O)O FS-2965 COC(=O)c1ccn2cccc2c1 FS-2967 c1cc2cc(cc(c2nc1)C(=O)O)Cl FS-2968 c1cc2c(cc1Br)ncs2 FS-2969 Cn1ccc2cc(ccc2c1=O)Br FS-2970 Cc1cc(nc(n1)N)N2CCCCC2 FS-2971 c1ccc(cc1)CN2C3CCC2CC(C3)N FS-2972 c1ccc(cc1)COc2ccc(nc2)N FS-2973 CCOC(=O)c1cc2cccnc2[nH]1 FS-2974 Cc1nc2c(o1)cc(cn2)Br FS-2975 Cc1cnc(s1)N2CCNCC2 FS-2976 c1cnc2c(n1)c(ns2)Br FS-2977 c1cnc2c(n1)c(cs2)Br FS-2978 Cc1c(cc2ccccc2n1)N FS-2979 c1cc2c(cc1Br)c(ns2)N FS-2980 c1cc2c(cc1F)C3(CC3)CN2 FS-2981 CN1CCN(CC1)c2ncc(cn2)N FS-2982 c1cc2c(cc1Br)CNC(=O)C2 FS-2983 c1cncc2c1sc(n2)Cl FS-2984 c1cc2c(nc1)nc(s2)Cl FS-2985 COc1ccc2c(n1)NCCN2 FS-2986 CN1CCN(CC1)c2cccc(c2)CO FS-2988 c1cc2c(cno2)c(c1)Br FS-2989 c1ccc(cc1)n2cc(nc2)C(=O)O FS-2990 Cc1c(sc2n1ccn2)C(=O)O FS-2991 c1cc2nc(nn2cc1Br)N FS-2992 COc1ccc(nn1)Br FS-2993 c1ccc2c(c1)C(=O)NC3(N2)CCNCC3 FS-2994 c1cc2c(c(c1)Br)[nH]nc2C(=O)O FS-2995 c1c(cnc2c1c(n[nH]2)Br)N FS-2996 c1ccc2c(c1)C3(CCNCC3)C(=O)N2 FS-2997 COC(=O)c1cccc2c1sc(n2)N FS-2998 c1cc(c2c(c1)nc(s2)N)C(=O)O FS-2999 c1cc(c2c(c1)ncs2)C(=O)O FS-3000 c1c2c([nH]nc2Br)ncn1 FS-3001 c1nc(c2c(n1)[nH]nc2Br)N FS-3002 Cc1cc(ncn1)Br FS-3003 c1cc2cc[nH]c(=O)c2c(c1)Br FS-3004 c1cc2c(cc1Br)OCCN2 FS-3005 CNc1nccc(n1)Br FS-3006 CNc1c(cncn1)Br FS-3007 c1c(cnc2c1nc(s2)N)Br FS-3008 c1cc(ncc1Br)CN FS-3009 CC(=O)c1nc2ccccc2o1 FS-3010 c1cnn2c1nc(cc2)Br FS-3011 CC(=O)n1c2ccc(cc2cn1)Cl FS-3012 CC(C#N)c1cccc(c1)C(=O)O FS-3013 c1cc2c(c(c1)Br)nc[nH]2 FS-3014 CC1=C(SCCO1)C(=O)Nc2ccccc2 FS-3015 c1cc(ccc1c2nc[nH]n2)Br FS-3016 c1ccc2c(c1)c(cc(n2)Cl)O FS-3017 c1ccc2c(c1)C(=O)Nc3ccccc3S2 FS-3018 c1cc(ccc1C2CCC(=O)CC2)O FS-3019 COc1ccc(c(c1)OC)O FS-3021 c1cc(sc1C(=O)C(O)O)Br FS-3022 Cc1nccn1c2ccccc2CO FS-3023 Cc1nccn1c2ccc(cc2)CO FS-3024 c1ccc(c(c1)CO)N2CCOCC2 FS-3025 c1ccc(c(c1)CO)n2ccnc2 FS-3026 CCN1CCN(CC1)c2ccccc2CO FS-3027 CCN1CCN(CC1)c2ccc(cc2)CO FS-3028 CCN1CCN(CC1)c2ccc(cc2)C(=O)O FS-3029 c1cncc(c1O)Br FS-3030 c1ccc(cc1)C2CSCCN2 FS-3031 COc1ccc(cc1)C2CSCCN2 FS-3032 c1ccc2c(c1)cccc2C3CNCCN3 FS-3033 c1ccc(cc1)C2CC(=O)CCO2 FS-3034 COC(=O)c1ccc2cn[nH]c2c1 FS-3035 CS(=O)(=O)c1ccc2c(c1)sc(n2)N FS-3036 c1cc2c(cc1Cl)OCCC2=O FS-3037 C[C@@]12C[C@H]3C[C@@](C1)(C[C@](C3)(C2)N)C.Cl FS-3038 Cc1ccc2c(c1)[nH]cc2C(=O)O FS-3039 c1cc(c(cc1C#N)Br)O FS-3040 c1cc2cc(ccc2c(c1)C(=O)O)O FS-3041 c1cc2c(c(c1)Cl)c(c[nH]2)CC(=O)O FS-3042 c1c(cc2c(c1C(=O)O)nc[nH]2)Br FS-3043 c1cc(ncc1Br)CC#N FS-3044 COc1cccc(c1C(=O)O)Br FS-3045 COc1c(cccc1Cl)C(=O)O FS-3046 CCOC(=O)c1ccc([nH]1)C FS-3047 Cn1cc(c2ccccc2c1=O)Br FS-3048 c1cc2c(c(c1)F)C(=O)C(=O)N2 FS-3049 COc1ccc2c(c1)c(c[nH]2)CC(=O)O FS-3050 CC(=O)c1cc(ccc1O)C#N FS-3051 c1ccc2c(c1)[nH]c(n2)C3CCNCC3 FS-3052 CC(=O)c1ccc2cc(ccc2c1)OC FS-3053 c1c2c(sc1C(=O)O)CCCC2 FS-3054 COc1ccc2cnccc2c1 FS-3055 C1C2CC3CC(C2)(CC1C3=O)C(=O)O FS-3056 c1cc(cc(c1)C(=O)O)CC#N FS-3057 COc1cc(ccc1C(=O)O)Cl FS-3058 CC(=O)c1cc(sc1)Br FS-3059 CCOC(=O)c1c(scn1)Br FS-3060 c1ccc2c(c1)cc(o2)CC(=O)O FS-3061 c1ccc(cc1)CN2CCC(CC2)C#N FS-3062 COc1ccc(c(c1)O)Br FS-3063 c1cc(c(cc1O)F)CC(=O)O FS-3065 CC(C)(C)C(=O)Nc1cccnc1 FS-3066 c1cc2c(cc1Cl)[nH]cc2C(=O)O FS-3067 COc1ccc2c(c1)CC(=O)N2 FS-3068 COc1cc(ccc1F)CC(=O)O FS-3069 C1CCC2C(C1)CC(N2)C(=O)O FS-3070 c1cc2c(cc1Br)CC(C2)O FS-3071 Cn1c(ccc1Br)C(=O)O FS-3072 COc1cc(cc(c1)Br)C#N FS-3073 COc1ccc(c(c1)F)CC(=O)O FS-3074 c1cc2c(cc1Br)[nH]nc2O FS-3075 c1ccc2c(c1)C(=O)Nc3cccnc3N2 FS-3076 Cc1cc(ncc1Br)C(=O)OC FS-3077 COC(=O)c1cc(cs1)N FS-3078 CCOC(=O)c1cc[nH]c1C FS-3079 c1c[nH]c2c1ncc(c2)Br FS-3080 COc1nccc(n1)Br FS-3081 Cc1cc(ncc1Br)C(=O)O FS-3082 c1c(cnc2c1[nH]nc2)Br FS-3083 COC(=O)c1cccc(n1)N FS-3084 CCOC(=O)c1c(cc[nH]1)C FS-3085 c1ccc(cc1)COC(=O)N2CCCC(=O)CC2 FS-3087 c1ccc(cc1)COC(=O)N2CCCC(CC2)O FS-3088 C1CC2(CCNC2=O)CNC1 FS-3089 c1csc2c1cc(cn2)N FS-3090 Cc1cc(c(s1)C(=O)OC)O FS-3091 c1ccc(cc1)CN2CCCCC2C(=O)O FS-3092 Cn1cc(ncc1=O)Br FS-3093 c1cc2c(cc1Br)c(n[nH]2)O FS-3094 COc1cccc2c1C(=O)CCC2 FS-3095 CCOc1ccc2cc[nH]c2c1 FS-3096 CC(=O)Nc1ccc(c(c1)Cl)O FS-3097 c1cc(c(c(c1)Cl)C(=O)O)O FS-3098 c1ccc2cnc(cc2c1)CN FS-3099 CC1(c2ccccc2NC1=O)C FS-3100 c1cc(cnc1)C(=O)NCCO FS-3101 CCc1ncc(cn1)Br FS-3102 c1cc2c(c(c1)F)[nH]nc2C(=O)O FS-3103 COC(=O)c1cccc(c1)c2nccs2 FS-3104 CN1CCN(CC1)Cc2ccccc2CN FS-3105 c1c(cnc(n1)C#N)Br FS-3106 CCOc1ccc2c(c1)cc[nH]2 FS-3107 c1cc(ccc1c2nccs2)O FS-3108 COC(=O)c1csc(n1)Cl FS-3109 c1cc(ccc1c2ccc(nc2)C#N)F FS-3110 Cc1cc2ccccc2n1CC(=O)O FS-3111 Cc1cc(nc(n1)C(F)(F)F)O FS-3112 Cc1nc(cc(n1)O)C(F)(F)F FS-3113 COc1cccc(c1Cl)O FS-3114 CCOC(=O)c1ccc2c(c1)cccn2 FS-3115 c1ccn2c(c1)nnc2Br FS-3116 COc1cc2ccccc2nc1 FS-3117 COc1cncc2c1cccc2 FS-3118 Cc1cc(cnc1)C(=O)OC FS-3119 COc1cccc2c1cccn2 FS-3120 COc1cccc2c1ccnc2 FS-3121 c1cc2ccc(cc2nc1)Cl FS-3122 Cc1ccc(cc1F)C(=O)OC FS-3123 COc1ccc(c(c1)CC#N)F FS-3124 c1cnc(nc1Br)NC2CCCC2 FS-3125 c1cc(sc1)N2CCNCC2 FS-3126 Cc1nc2cc(cnc2s1)Br FS-3127 COC(=O)c1cc(co1)Br FS-3129 C#CCN[C@@H]1CCc2c1cccc2 FS-3130 c1c(c(n[nH]1)C(=O)N)Br FS-3131 CC(=O)c1ccc(cc1O)Br FS-3132 COC(=O)c1cc2ccc(cc2[nH]1)C#N FS-3133 c1cc(c2ccc(nc2c1)Cl)C(=O)O FS-3134 CC(=C)c1cc(cnc1)Br FS-3135 c1c(cc2c(c1C(=O)O)cn[nH]2)Br FS-3136 COC(=O)c1cccc(c1O)Cl FS-3137 C#Cc1ccnc2c1cccc2 FS-3138 Cc1c(sc(n1)Br)C FS-3139 c1cc2cnoc2cc1Br FS-3140 COc1ccc(c(c1)Br)C#N FS-3141 c1ccc2c(c1)nc(s2)N FS-3142 COC(=O)c1ccc(cc1F)O FS-3143 COc1cc(cnc1N)Br FS-3144 Cc1ccc(nc1)S(=O)(=O)N FS-3145 c1c2n(nc1C(=O)O)CCC2 FS-3146 Cc1ccc(c(c1)CC(=O)O)C FS-3147 c1cc(c(cc1Cl)C(=O)N)O FS-3148 c1cc(c(cc1Br)C(=O)O)O FS-3149 C1CCC2(CC1)CC(=O)NC(=O)C2 FS-3150 c1ccc(cc1)Oc2ccncc2 FS-3151 c1cc(c(cc1CC#N)C#N)F FS-3152 CCOC(=O)C1(CCNCC1)C FS-3153 c1cc2c(cc1Cl)nc(s2)N FS-3154 Cc1ccccc1[C@H](CC(=O)O)N FS-3155 COc1cccc2c1[nH]c(=O)s2 FS-3156 Cc1c(cccc1O)C(=O)O FS-3157 c1ccc2c(c1)c(c[nH]2)CCC(=O)O FS-3158 c1c(cnc2c1nco2)Br FS-3159 CNc1ccc(cn1)Br FS-3160 Cc1cc(ccc1F)C(=O)OC FS-3161 Cc1c2ccccc2nc(n1)C FS-3162 c1ccc2c(c1)c(=O)[nH]s2 FS-3163 c1cc2cnccc2c(c1)C#N FS-3164 COC(=O)c1c(sc(n1)N)Cl FS-3165 c1c(nc(c(n1)N)C#N)Br FS-3166 CN(C)c1ncc(cn1)Br FS-3167 COC(=O)c1c(scn1)Br FS-3168 c1nc(c(s1)Br)C(=O)O FS-3169 COC(=O)c1cc(c(s1)Cl)N FS-3170 Cc1ncc(c(n1)O)Br FS-3171 COc1c(cnc(n1)N)Br FS-3172 COc1ccc(cc1O)CO FS-3173 COC(=O)c1ccc(c(c1)O)Br FS-3174 c1ccc2c(c1)CC(=C2)Br FS-3175 c1ccc(cc1)C(=O)Nc2cccc(c2)C#N FS-3176 c1ccc2c(c1)nc(o2)Cl FS-3177 CCOc1ccccc1C(=O)O FS-3178 c1ccc(cc1)COc2ccnc(c2)N FS-3179 c1cc2cc(ccc2c(c1)O)O FS-3180 COc1cc(cc(c1)OC)CO FS-3181 COc1ccc(cc1C(=O)O)Cl FS-3182 c1cc2c(cc1Cl)OCCN2 FS-3183 CCOC(=O)c1cnc(s1)C(F)(F)F FS-3184 c1ccc2c(c1)C(=O)N(C2=O)O FS-3185 COc1cc2c(ccnc2cc1O)Cl FS-3186 COC(=O)c1cc2cc[nH]c2nc1 FS-3187 CCOC(=O)c1cccc2c1[nH]nc2 FS-3188 CC(=O)c1cccc2c1cccc2 FS-3189 COc1cc(cc(c1)F)C(=O)O FS-3190 Cc1cccc(c1O)C(=O)O FS-3191 CCOC(=O)c1ccccn1 FS-3192 c1ccc2c(c1)cccc2CC(=O)N FS-3193 c1ccc2cc(ccc2c1)CO FS-3194 c1cncc2c1[nH]c(c2)C(=O)O FS-3195 COc1ccc2cccc(c2c1)O FS-3196 c1cc2c(c(c1)Br)OCC2=O FS-3197 c1ccc(cc1)C(C2CCCCN2)C(=O)O FS-3198 c1cc(ccc1C#N)NCC(=O)O FS-3199 COC(=O)c1ccc(cc1O)F FS-3200 Cc1cc(n[nH]1)Br FS-3201 COc1c(cccc1F)CO FS-3202 CC(=O)c1ccc(c(c1)O)OC FS-3203 COc1cc(cc(c1)OC)CN FS-3204 c1cc(c2nc(cn2c1)C(F)(F)F)C(=O)O FS-3205 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)O FS-3206 Cc1cc(ncc1Br)C#N FS-3207 Cc1ccc(cc1)S(=O)(=O)NNC(=O)N FS-3208 Cc1cn2ccnc2c(n1)SC FS-3209 CNCc1cc(cnc1)Br FS-3210 CC(=O)c1cc(ccc1O)O FS-3211 Cc1cccc2c1[nH]cc2C(=O)O FS-3212 Cc1c(cc(cn1)Br)O FS-3213 Cc1cc(ccc1C#N)C(=O)O FS-3214 CCc1c(sc(n1)C)C(=O)O FS-3215 c1ccc(c(c1)C(=O)CC#N)Cl FS-3216 c1ccc(c(c1)CC(C(=O)O)N)Cl FS-3217 Cc1cc(cc(c1)OCC2CNC(=O)O2)C FS-3218 COC(=O)c1cnc(s1)Cl FS-3219 CCOC(=O)c1c2ccccc2[nH]n1 FS-3220 c1cc(ccc1c2nc(cs2)C(=O)O)F FS-3221 c1cc2c(cc1Cl)ncc(=O)[nH]2 FS-3222 c1ccc(cc1)CN2CCC3C2CNC3 FS-3223 c1ccc(cc1)C(=O)C2(CCCCC2)O FS-3226 c1cc2cccc(c2c(c1)O)O FS-3227 COc1cc(cc(c1)OC)C#N FS-3228 c1cc2cc(ccc2nc1)CC(=O)O FS-3229 c1cc2c(cc1Cl)NC(=O)CC2 FS-3230 c1[nH]c2c(n1)c(=O)[nH]c(=O)[nH]2 FS-3231 c1c(cnc(n1)C(=O)N)Br FS-3232 CN1CCN(CC1)Cc2cccc(c2)CN FS-3233 CC(=O)c1c[nH]c2c1cccn2 FS-3234 c1cc2c(c(c1)Br)c(no2)N FS-3235 CC(=O)c1c(cccc1Cl)O FS-3236 c1cc(cn2c1cnc2)C(=O)O FS-3237 Cc1c(ncc(n1)N)Br FS-3238 Cn1c2cc(ccc2c(n1)N)Br FS-3239 c1cc2c(cc([nH]2)C(=O)O)c(c1)F FS-3240 Cc1cccc(c1C(=O)O)OC FS-3241 Cc1c2cc(ccc2[nH]n1)C#C FS-3242 CCOC(=O)c1ccsc1C FS-3243 COc1c(nc2ccccc2n1)Cl FS-3244 COc1ccc(c(c1)OC)CN FS-3245 c1cc(c(c(c1)Cl)O)C(=O)O FS-3246 CN1CCN(CC1)c2[nH]nc(n2)N FS-3247 CCc1cc(n(n1)c2ccccc2)N FS-3248 COc1c(csc1Br)C(=O)O FS-3249 c1ccc(c(c1)C(=O)NO)O FS-3250 Cc1cnc(s1)C(=O)OC FS-3251 c1cc2c(cc1F)OCCC2=O FS-3252 c1csc2n1c(cn2)C(=O)O FS-3253 c1cc2c(c(c1)Br)OCO2 FS-3254 COC(=O)c1ccc2c(c1)nc([nH]2)N FS-3255 Cc1c(ccc2c1cn[nH]2)Br FS-3256 c1cc(nc2c1cc(cc2)O)O FS-3257 c1ccc(cc1)c2cc(ccn2)N FS-3258 CCOC(=O)c1c([nH]cn1)C FS-3259 Cc1cc2c(cc1Br)cn[nH]2 FS-3260 CCn1cc2cc(ccc2n1)N FS-3261 c1cc(c(cc1C(F)(F)F)C#N)O FS-3263 COC(=O)Cc1ccc(cc1)C#N FS-3264 COC(=O)c1ccc(c(c1)C(F)(F)F)O FS-3265 c1c(cnc(n1)C(F)(F)F)N FS-3266 c1ccc(cc1)C(=O)c2cccnc2 FS-3267 c1cc2c(cc1Cl)CNC2=O FS-3268 c1cnc(c2c1occ2)N3CCNCC3 FS-3269 c1cc(c(cc1Cl)C(=O)O)O FS-3270 Cc1c(sc(n1)N)Br FS-3271 c1ccc(cc1)COc2c(nccn2)N FS-3272 c1cnc2c(n1)c(c[nH]2)Br FS-3273 c1ccc2c(c1)c(n[nH]2)Br FS-3275 c1ccc2c(c1)c(c(cn2)Br)N FS-3276 c1cc2c(cc([nH]2)C(=O)O)c(c1)Br FS-3277 c1ccc(cc1)C2CC(=O)NC2 FS-3278 c1c[nH]c2c1nc(cn2)Br FS-3280 c1cc2c(cc1Br)cnc(n2)N FS-3282 c1cc2c(cc1O)scn2 FS-3284 COc1ccc2c(c1)CCNC2=O FS-3285 c1cc2cc([nH]c2c(c1)Br)C(=O)O FS-3286 COC(=O)c1c(cccn1)Cl FS-3287 c1c(nc(c(n1)N)N2CCCC2)Br FS-3288 CCNc1c(ncc(n1)Br)N FS-3289 CN(C)c1c(ncc(n1)Br)N FS-3290 CCN(CC)c1c(ncc(n1)Br)N FS-3291 c1c(c(ncn1)N)Br FS-3292 c1ccc(cc1)c2cc3c([nH]2)nccn3 FS-3293 Cc1ccc(cc1)C2CNCCN2 FS-3294 CCc1ccc(cc1)C2CNCCN2 FS-3295 c1c(cnc(c1O)N)Br FS-3296 c1cc2c(cc1F)c(n[nH]2)C(=O)O FS-3297 Cc1nc2c(s1)CNCC2 FS-3298 c1cc2c(cc1Br)[nH]cc2C(=O)O FS-3299 CC1CCN(CC1)c2ccc(cc2)C#N FS-3300 CC1CCN(CC1)c2ccc(cc2)CN FS-3301 Cc1cc(ccc1Br)C(=O)N FS-3302 c1ccc(cc1)c2c(c(n[nH]2)N)Br FS-3303 c1ccc(cc1)C2CCNC2=O FS-3305 c1c(cnc(n1)N)C(F)(F)F FS-3306 Cc1cc(cc(c1OC)C)C(C)N FS-3307 CN[C@@H]1CCCN(C1)Cc2ccccc2 FS-3308 c1cc(c2c(c1)OCCO2)CO FS-3309 c1cnc(nc1C(F)(F)F)N2CCC(CC2)O FS-3310 c1ccc2c(c1)c(=O)oc(=O)[nH]2 FS-3311 CCc1nnc2n1cc(cc2)Br FS-3312 c1cc(c(cc1O)O)Br FS-3313 CC(=O)N1CC(=O)c2c1cccc2 FS-3314 CC1CN(CCC1=O)Cc2ccccc2 FS-3315 COC(=O)c1ccnc(c1)C(F)(F)F FS-3316 c1ccc2c(c1)c(c[nH]2)CCN FS-3317 COC(=O)c1cccc2c1[nH]cc2C#N FS-3318 c1cc2c(cc[nH]2)cc1N3CCOCC3 FS-3319 c1cc2c(cc1C#N)[nH]cc2C(=O)O FS-3320 Cc1cc(ccc1C#N)C(=O)OC FS-3321 Cc1nc2ccc(cn2n1)Br FS-3322 c1cc(c2cc[nH]c2c1)C(F)(F)F FS-3323 c1c(c2c([nH]c1=O)CCC2)O FS-3324 CCOC(=O)c1cccc2c1cc[nH]2 FS-3325 c1c(csc1CN)Br FS-3326 c1c(cnc2c1CNCC2)O FS-3327 CN1CCc2c1cccc2C(=O)O FS-3328 c1cc(c(cc1O)C(=O)O)Br FS-3329 Cc1cc(c(nc1)C#N)Br FS-3330 c1cc2c(c(c1)Br)CCN2 FS-3331 c1cc(c(cc1Br)O)C#N FS-3332 c1cnc(c2c1scc2Br)N FS-3333 c1cc(c2c(c1)NCC2)C(F)(F)F FS-3334 c1cc(c(cc1C(F)(F)F)C(=O)O)O FS-3335 COc1c(c2c(cc[nH]2)cn1)Br FS-3336 c1ccc(cc1)COC(=O)N2CC(=O)C2 FS-3337 COc1ccc2c(c1)CCC2C(=O)O FS-3338 c1cc2c(c(c1)Br)c(ncn2)O FS-3339 COC(=O)c1cc(ccc1C#N)Cl FS-3340 c1cc(c(cc1Br)C#N)C#N FS-3341 c1ccc2cc(ccc2c1)C(=O)O FS-3342 c1cc2c(cc1Cl)c(c[nH]2)CCO FS-3343 c1cn2c(cc1Br)nc(n2)N FS-3344 CC(=O)c1ccc(cc1Cl)O FS-3345 COc1ccc(c(c1)C(=O)O)Br FS-3346 c1cc2c(cc1Br)CCN2 FS-3347 COc1ccc2c(c1)ccc(n2)Cl FS-3348 c1ccc(cc1)CN2Cc3c([nH]c(=O)[nH]c3=O)C2 FS-3349 c1cc2c(cc1F)NC(=O)C2 FS-3350 CCOc1c(ncc(n1)Br)N FS-3351 c1ccc(cc1)COC(=O)N2CC=CC2 FS-3352 c1cc2c(c(c1)Br)OCC2 FS-3353 c1cc2c(cc(cn2)Br)nc1 FS-3354 c1c(nc[nH]1)C2CCNCC2 FS-3355 c1cc2c(cc1Br)NCC2 FS-3356 c1c(nc(s1)Cl)C(=O)O FS-3357 c1cc2c(cc1C#N)c(n[nH]2)N FS-3358 CCCc1c[nH]c(=O)[nH]c1=O FS-3359 c1cc2c(ccnc2cc1O)Cl FS-3360 CCOC(=O)c1cc2cc(ccc2[nH]1)C#N FS-3361 c1ccnc(c1)C2(CC2)C(=O)O FS-3362 COC(=O)c1ccc([nH]1)Br FS-3363 CCc1c(cccc1OC)C(=O)O FS-3364 COc1cc(cc(c1)Br)OC FS-3365 c1c[nH]c2c1cc(cn2)C(=O)O FS-3366 COC(=O)c1ccc(o1)Br FS-3367 c1cc2c(cc1C(=O)N3CCCCC3)nccn2 FS-3368 c1c[nH]c2c1c(cnc2)Br FS-3369 Cc1c2ccc(cc2[nH]n1)Br FS-3370 CCOC(=O)c1cccc(n1)N FS-3371 c1ccc(cc1)c2cccc(n2)N FS-3372 c1cnn(c1)C2CCCCO2 FS-3373 c1cc2c(cc1C(F)(F)F)NC(=O)C2=O FS-3374 Cc1ccc2c(c1)cc([nH]2)C(=O)O FS-3375 COc1cc(ccc1Br)C(=O)OC FS-3376 c1cc2c(cccn2)c(c1)Cl FS-3377 Cn1c2cccc(c2cn1)C(=O)OC FS-3378 c1ccc2c(c1)CCC2C(=O)O FS-3379 c1cncc(c1CO)Br FS-3380 CN(C)c1ccc(cc1)c2nc(cs2)C(=O)O FS-3381 c1c(cn(n1)C2CCCCO2)Br FS-3382 c1ccc2c(c1)cncc2C(=O)O FS-3383 c1ccc2c(c1)c(co2)CC(=O)O FS-3384 c1ccn2c(c1)cc(n2)Cl FS-3385 CCOC(=O)c1ccc(s1)Br FS-3386 COC(=O)c1ccc2c(c1)cn[nH]2 FS-3387 c1cc2c(c(c1)Cl)CCN2 FS-3388 COc1cc2c(cc1Br)cn[nH]2 FS-3390 c1ccc(cc1)n2cc(cn2)C(=O)O FS-3391 c1ccc2c(c1)c(co2)CCN FS-3392 c1ccc(cc1)C(c2ccccn2)N FS-3393 c1cnc(cc1O)C(F)(F)F FS-3394 c1coc2c1c(=O)[nH]cc2Br FS-3395 c1cc2c(cc1Br)C3(CC3)CN2 FS-3396 c1cc2c(nsc2nc1)N FS-3397 c1cc2c(c(c1)Br)CCNC2 FS-3398 c1ccn2c(c1)ncc2C(=O)O FS-3399 c1cc(c2cn[nH]c2c1)C(=O)O FS-3400 c1cc2c(cc1Cl)OCC(=O)N2 FS-3402 c1cc2c(c(c1)Br)scn2 FS-3403 Cc1c2cc(cnc2[nH]n1)Br FS-3404 Cc1nnc2n1ccc(c2)Br FS-3405 c1cn2cnnc2cc1Br FS-3406 c1cc2c(c(c1)Br)[nH]nc2N FS-3407 c1cc2cn[nH]c2c(c1)C(=O)O FS-3408 Cc1c(ccc(n1)O)Br FS-3409 c1c2c(c(cs2)Br)[nH]c1C(=O)O FS-3410 c1cc2cccnc2c(c1)C(=O)O FS-3411 c1cn2ccnc2cc1Br FS-3412 c1cc2cnccc2c(c1)C(=O)O FS-3413 c1cc2c(cc1O)CCNC2=O FS-3414 c1c[nH]c2c1c(ncn2)Br FS-3415 c1cn2ccnc2cc1Cl FS-3416 COc1c2nccn2cc(n1)Br FS-3417 c1cc2c(cc1Cl)c(ncn2)O FS-3418 Cc1cc(c(nc1)C(=O)O)Br FS-3419 CC(=O)c1c[nH]c2c1cc(cc2)Cl FS-3420 c1cc(c2c(c1)OCO2)CN FS-3421 c1cc2c(c(c1)Cl)c(c[nH]2)C(=O)O FS-3422 C1C2C=CC1C3C2C(=O)NC3=O FS-3423 c1cc2c(cc1Br)cn[nH]c2=O FS-3424 Cc1ccc2c(c1)C(=O)C(=O)N2 FS-3425 c1cc(c(cc1Cl)O)C#N FS-3426 Cc1cc2c([nH]1)cccc2Br FS-3427 Cc1cc(ccc1C(=O)OC)F FS-3428 Cc1cc(c(nc1)O)Br FS-3429 c1ccc(cc1)CN2C3CC(=O)CC2COC3 FS-3430 c1c(nc(s1)N)CC(=O)O FS-3431 Cc1ccc(cc1)C(=O)Cc2ccncc2 FS-3432 COC(=O)c1cc2c([nH]1)ccs2 FS-3433 c1ccnc(c1)c2csc(n2)Br FS-3434 COc1cccc2c1CCC2=O FS-3435 Cc1cc(cnc1C#N)Br FS-3436 COc1ccc2cccnc2c1 FS-3437 COc1cc(ccc1O)CCO FS-3438 c1cc2c(cc1Br)OCC(=O)N2 FS-3439 c1cc2c(cc1Br)C(=O)NCC2 FS-3440 c1cc(c2c(c1)C(=O)CC2)C#N FS-3441 c1cc2c(ncnn2c1)Cl FS-3442 c1c(nc2n1CCCC2)C(=O)O FS-3443 c1c(c2c(ncnc2[nH]1)N)Br FS-3445 COC(=O)c1cncc2c1cccc2 FS-3446 C#Cc1cc(cnc1N)Br FS-3447 c1ccc(cc1)C(CC(F)(F)F)N FS-3448 c1cc2c(c(c1)CO)CCCC2 FS-3449 c1cc(ccc1CN2CCCNCC2)F FS-3450 C=CCc1ccc2c(c1)OCO2 FS-3451 Cc1cc(nc(c1)C(=O)O)C FS-3452 CCOC(=O)c1cccnc1 FS-3453 Cc1ccc(nc1)C(=O)OC FS-3454 c1csc2c1ncc(c2)O FS-3455 CC(=O)c1ccc(cc1O)O FS-3456 c1cc2c(cc1O)OCCO2 FS-3457 C#Cc1c2ccccc2ccn1 FS-3458 C#Cc1cccc2c1ccnc2 FS-3459 c1cc(cc2c1ccnc2)C#N FS-3460 c1c(cnc2c1[nH]nn2)Cl FS-3461 CC(=O)c1ccc(cn1)Cl FS-3462 c1c(cc(cc1O)F)C(=O)O FS-3463 c1cc2c(cc1C#N)C(=O)CC2 FS-3464 COC(=O)c1ccc(s1)N FS-3465 Cc1csc(n1)C(=O)OC FS-3466 COC(=O)c1c(ncs1)N FS-3467 c1ccc2c(c1)cccc2CO FS-3468 COc1cc(cc(c1)Cl)O FS-3469 c1cc2c(cc1F)c(c[nH]2)C#N FS-3470 Cc1c([nH]cn1)Br FS-3471 c1ccc(c(c1)CC(=O)O)C#N FS-3472 c1cc(ccc1CC(=O)O)C#N FS-3473 c1cc2c(cc([nH]2)C(=O)O)nc1 FS-3474 c1cncc2c1[nH]cc2C(=O)O FS-3475 c1cc2c(c(c[nH]2)C(=O)O)nc1 FS-3476 c1c[nH]c2c1cnc(c2)C(=O)O FS-3477 COc1cccc2c1C(=O)CC2 FS-3478 c1ccc2c(c1)C(=O)NCCN2 FS-3479 c1ccc2c(c1)C(CN2)CCN FS-3480 COc1ccc2c(c1)NC(=O)C2 FS-3481 c1cc(=O)[nH]nc1C(F)(F)F FS-3482 c1cc2c(cc1F)CCCC2=O FS-3483 COc1cc(cc(c1)F)CC#N FS-3484 Cc1c(nn(c1C(=O)OC)C)C FS-3486 c1cc2c(cc1Cl)OCC2=O FS-3487 c1c(cnc2c1CC(=O)N2)Cl FS-3488 Cc1c(cc(cc1F)C(=O)O)O FS-3489 CC(C)c1nc(cs1)CNC FS-3490 c1cc(c(nc1)CC(=O)O)Cl FS-3491 c1ccc2c(c1)cccc2C(=O)O FS-3492 Cc1ccc2c(c1)c(c[nH]2)C(=O)O FS-3493 c1cc2c(cc1F)c3c([nH]2)CCC3 FS-3494 c1cc2c(cc1C(=O)O)C(=O)CC2 FS-3495 COC(=O)c1c[nH]c2c1ccnc2 FS-3496 COC(=O)c1c[nH]c2c1nccc2 FS-3497 COc1ccc2c(c1)NC(=O)CC2 FS-3498 c1cc(cc(c1)O)N2CCCCC2 FS-3499 CCOC(=O)c1cc2n(n1)CCC2 FS-3500 CC1(CCCC2(C1=CC(=O)O2)C)C FS-3501 C#Cc1ccc(cc1)S(=O)(=O)N FS-3502 COc1cccc(c1CC(=O)O)F FS-3503 Cc1ccc(cc1)c2ccc(cn2)N FS-3504 Cc1cccc(c1)c2cnc(nc2)N FS-3505 c1c[nH]c2c1ncc(c2)C(F)(F)F FS-3506 c1ccc2cc(ccc2c1)CC(=O)O FS-3507 COc1ccncc1Br FS-3508 CNc1ncc(cn1)Br FS-3509 c1c(c(c(cn1)Br)O)N FS-3510 CCOC(=O)c1cc2c([nH]1)cccn2 FS-3511 c1c(coc1C(=O)O)Br FS-3512 COC(=O)c1cccc2c1NC(=O)C2 FS-3513 c1cc(ccc1C2CSCCN2)F FS-3514 c1ccc(cc1)CNc2cnccc2N FS-3515 CC(=O)c1c(cccn1)Br FS-3516 c1cc(ccc1CN2CCOCC2)C#N FS-3517 COc1cc(ccc1O)Br FS-3518 c1cc(c(cc1CO)O)Br FS-3519 COC(=O)C(=O)c1c[nH]c2c1cccc2 FS-3520 c1ccc(cc1)n2cc(c(n2)C(=O)O)N FS-3521 c1cnccc1CN2CCC(CC2)CO FS-3522 COc1cccc(c1)C2CSCCN2 FS-3523 Cc1c(cc2cc[nH]c2n1)Br FS-3524 COc1cccc(c1C#N)Br FS-3525 c1cc2c(c(c1)Br)NC(=O)C2 FS-3526 Cc1ccc(cc1)S(=O)(=O)NC(=O)N FS-3527 CC(=O)c1cccc(c1O)Br FS-3528 CC(=O)c1ccc(cc1Br)O FS-3529 CC(=O)c1c(cccc1Br)O FS-3530 c1ccc(cc1)COC(=O)N2CC(C2)C#N FS-3531 COC(=O)Cn1cc(cn1)Br FS-3532 c1c(c(sc1C(=O)O)Br)N FS-3533 c1cc(cc(c1)Cl)C(=O)C2CCNCC2 FS-3534 c1cc2c(ccnc2cc1Br)O FS-3535 c1cc2c(c(c1)Br)ncnc2N FS-3536 c1cc2c(cc1Br)ncnc2N FS-3537 c1cc2c(cc1Br)c(ncn2)N FS-3538 c1cc2c(c(c1)Br)CCC(=O)N2 FS-3539 c1cc(cc(c1)Br)N2CCCC2 FS-3540 COc1c2cc(ccc2[nH]n1)Br FS-3541 COc1cc2c(cc1Br)nc[nH]2 FS-3542 c1c[nH]c(=O)c2c1scc2Br FS-3543 COC(=O)c1ccc(c(c1)Br)O FS-3544 COc1cc(cc(c1)Br)C(=O)O FS-3545 COc1ccc(cc1C(=O)O)Br FS-3546 c1c[nH]c2c1c(cc(c2)Br)C(=O)O FS-3547 c1cc2c(cc1Br)c(cc(=O)[nH]2)O FS-3548 c1c(cc(c2c1[nH]nc2)Br)C(=O)O FS-3549 c1c(cnc2c1c(c[nH]2)C(=O)O)Br FS-3550 c1c(cnc(n1)N2CCC(C2)O)Br FS-3551 Cc1ccc(cc1Br)S(=O)(=O)C FS-3552 C[C@@H](c1ccc(cc1)C(=O)OC)N FS-3553 COC(=O)c1ccncc1Br FS-3554 Cc1cccc(c1C(=O)N)Cl FS-3555 Cc1ccc(cc1Br)C(=O)N FS-3556 CCc1cc(ccc1C#N)C#N FS-3557 Cc1c(cccc1Cl)C(=O)OC FS-3558 c1cncc2c1cc([nH]2)C(=O)O FS-3559 CC(C)(C#N)c1nc2ccccc2o1 FS-3560 Cc1cc(ccc1C(=O)O)O FS-3561 CC(=O)c1cccc(c1O)Cl FS-3562 CCOC(=O)c1cc2cnccc2[nH]1 FS-3563 COC(=O)c1ccc2c(n1)cc[nH]2 FS-3564 COc1cccc2c1NC(=O)C2=O FS-3565 COc1ccc2c(c1)C(=O)NCC2 FS-3566 CCOC(=O)c1cccc2c1[nH]cc2 FS-3567 c1cc(c2c(c1)NC(=O)C2)C(=O)O FS-3568 Cc1cccc2c1c(c[nH]2)C(=O)O FS-3569 CN1CCC(=CC1)c2c[nH]c3c2cccn3 FS-3570 c1cc2c(c(c1)F)CC(=O)N2 FS-3571 c1cc2c(cc1C#N)ncs2 FS-3572 c1ccnc(c1)c2ccc(cc2)O FS-3573 COC(=O)c1cc2cc[nH]c2cn1 FS-3574 C#Cc1cccc2c1nccc2 FS-3575 CN(C)c1ccc(cc1)CCO FS-3576 c1cc2c(cc1C#N)NC(=O)C2 FS-3577 c1cc2c(cc[nH]2)cc1C(F)(F)F FS-3578 Cc1c(nc(s1)Br)C(=O)O FS-3579 Cc1cccc2c1cc[nH]c2=O FS-3580 COc1ccc(cc1)c2ccncc2 FS-3581 c1cc2c(cc1F)CCC(=O)C2 FS-3582 c1ccc2c(c1)CCOC23CCNCC3 FS-3583 c1ccc(cc1)c2cnc(s2)N FS-3584 Cc1ccc(cc1)S(=O)(=O)N FS-3585 Cc1c(cccc1F)CC(=O)O FS-3586 c1cc2c(cc1Cl)c(n[nH]2)CC(=O)O FS-3587 c1cc2c(cc1Br)OCC2=O FS-3588 c1cc2c(cc1C#N)sc(n2)Br FS-3589 COc1ccc(c2c1[nH]cc2)Br FS-3590 CCOC(=O)c1c(c(n[nH]1)Br)C FS-3591 CCOC(=O)c1c(cn[nH]1)C FS-3592 COc1cccc2c1CNC2=O FS-3593 COC(=O)c1cc2cccnc2[nH]1 FS-3594 Cc1[nH]c2ccc(cc2n1)Br FS-3595 COC(=O)Cc1c[nH]c2c1cccc2 FS-3596 c1cc2c(cc1Br)CC(=O)C2 FS-3597 COc1ccc2c(c1)cccn2 FS-3598 Cc1ccc(cc1)C2(CNCCO2)C FS-3599 CCOC(=O)c1cccc(n1)C(F)(F)F FS-3600 c1ccc(cc1)CO[C@H]2CCCC[C@@H]2N FS-3601 Cc1ccnc(c1Br)O FS-3602 c1cc2c(cc1F)sc(=O)[nH]2 FS-3603 CC(=O)c1c(cncn1)Br FS-3604 Cn1c2ccccc2nc1C(=O)O FS-3605 c1cnc(cc1CO)C(F)(F)F FS-3606 COC(=O)c1c(cccn1)C(F)(F)F FS-3607 CCc1cccc(n1)C(=O)O FS-3608 c1cc(c2ccsc2c1)C(=O)O FS-3609 c1cc2c(nc1)sc(n2)Cl FS-3610 CC(C)(C#N)c1cccc(c1)C(=O)O FS-3611 c1ccc(cc1)N2CCC(CC2)C(=O)O FS-3612 c1cc(cc2c1ccnc2)CO FS-3614 c1cc2cn[nH]c2cc1C(F)(F)F FS-3615 c1ccc(cc1)C(=O)Cc2ccncc2 FS-3616 c1cc2c(cc1F)o[nH]c2=O FS-3617 c1cc2c(cc1F)c(=O)[nH]o2 FS-3618 CCOc1c(cc(cn1)N)F FS-3619 c1c(cn(n1)C2CC2)Br FS-3620 CCOC(=O)c1cc(cs1)Cl FS-3621 COc1ccc(c(n1)C#N)Br FS-3622 c1c[nH]c2c1cc(nc2)C(=O)O FS-3623 c1cc2c(cc1Br)cc([nH]2)C#N FS-3624 COc1c(cccc1Br)C(=O)OC FS-3625 c1cc(c2c(c1)[nH]nc2N)C#N FS-3626 Cc1c(cc(cn1)Cl)C#N FS-3627 c1ccn2cnc(c2c1)C(=O)O FS-3628 CCOC(=O)c1ccsc1 FS-3629 c1c(cnc2c1[nH]cc2C#N)Br FS-3630 Cc1nc2ccc(cc2o1)Br FS-3631 Cc1c[nH]c2c1c(ccc2)C(=O)O FS-3632 c1cc(c2c(c1)scn2)O FS-3633 CCOC(=O)c1c2ccccn2cn1 FS-3634 c1ccc(cc1)CN2CC(=O)Nc3c2cccc3 FS-3635 c1cc(cc2c1ccc(=O)[nH]2)Br FS-3636 c1cc2c(c(c1)Br)C(=O)NC2=O FS-3637 c1cc2c(cc1Cl)C(=O)NC2=O FS-3638 C[C@H]1CNCCN1Cc2ccccc2 FS-3639 CC(=O)Nc1ccc(s1)Br FS-3640 c1cc(c2c(c1)sc(n2)N)F FS-3641 COc1ccc2c(c1)[nH]c(n2)C(F)(F)F FS-3642 COC(=O)c1ccccc1N2CCNCC2 FS-3643 Cc1ccn2c(cnc2n1)Br FS-3644 c1cc(ccc1C#CC(=O)O)Cl FS-3645 c1cc2c(cc1F)[nH][nH]c2=O FS-3646 Cn1c2cc(ccc2cn1)F FS-3647 c1cc2c(cc1Br)[nH]c(=O)oc2=O FS-3648 c1cc(ccc1N2CCCC2)Br FS-3649 CC(=O)c1c2ccccc2n(n1)C FS-3650 c1csc(c1Br)C#N FS-3651 c1ccc2c(c1)c(n[nH]2)CC(=O)O FS-3652 c1cc2c(cc[nH]c2=O)c(c1)Br FS-3653 c1cc2c(cc1Br)c(=O)[nH]o2 FS-3654 c1cncc2c1c(c[nH]2)Br FS-3655 c1cc2cncnc2c(c1)Br FS-3656 c1c([nH]c(n1)C(F)(F)F)C(=O)O FS-3657 COC(=O)c1ccc(cc1Cl)O FS-3658 c1cc2c(cc1Br)[nH]nc2C#N FS-3659 CC(=O)c1ccc2c(c1)OCO2 FS-3660 C#Cc1ccc(cn1)Br FS-3661 c1cc2c(cc1Cl)[nH]cc2CC(=O)O FS-3662 c1ccc(cc1)c2cnc(o2)Cl FS-3663 c1cc(cc2c1cc[nH]2)CC(=O)O FS-3664 COC(=O)c1cccc2c1nc[nH]2 FS-3665 Cn1c(ccn1)c2cccc(c2)C(=O)O FS-3666 Cn1c(cccc1=O)C(=O)O FS-3667 c1ccc2c(c1)cc(nn2)Br FS-3668 c1cc2c(c(c1)Cl)nc(s2)S FS-3669 c1ccc2c(c1)c(nc(n2)O)N FS-3670 c1c(nc2c(n1)[nH]c(=O)[nH]2)Br FS-3671 c1cc(cc(c1)F)OCC2(CCCNC2)O FS-3672 CC(=O)c1ccc(c(c1)OC)O FS-3673 Cc1cc(cnc1C#N)Cl FS-3674 COc1cc(cc(c1)Cl)OC FS-3675 c1cc2c(cc1Br)[nH]cc2CCO FS-3676 Cc1cc(nc2c1c(=O)[nH]s2)C FS-3677 c1ccc2c(c1)cc(c(n2)N)Br FS-3678 Cc1cccc(c1NC(=O)C2CCCCN2C)C FS-3679 c1cc(nc2c1cc(cc2)C(=O)O)Cl FS-3680 c1c(c(n[nH]1)C(F)(F)F)CO FS-3681 COC(=O)c1cc(cs1)Br FS-3682 Cc1ccc2c(c1)c(ncn2)O FS-3683 COC(=O)c1cscc1Br FS-3684 c1cc(ccc1c2cocn2)C(F)(F)F FS-3685 c1c(cc(=O)[nH]c1C(F)(F)F)O FS-3686 c1cc2c(cc[nH]2)cc1CCN FS-3687 COc1cc(cc(c1)O)C(F)(F)F FS-3689 c1cc2c(cc1Cl)cc(cn2)C(=O)O FS-3690 c1cc2c(ccnc2cc1C(=O)O)Cl FS-3691 c1cc2c(cc1Cl)sc(n2)C(=O)O FS-3692 COC(=O)c1cccc2c1scn2 FS-3693 c1cc2c(cc1Br)oc(n2)N FS-3694 Cc1c2cc[nH]c2ncc1Br FS-3695 CCOC(=O)c1cc(sc1)Br FS-3696 c1cc2c(cc(cn2)Br)c(c1)O FS-3697 CCOC(=O)c1ccc2c(c1)NCC2 FS-3698 Cc1cc2c(cc1C)C(=O)CC2 FS-3699 Cc1c(ccc(n1)C#N)Br FS-3700 Cc1nc2cncc(c2o1)Br FS-3701 CC(=O)c1c(cccn1)OC FS-3702 COc1ccc(cc1)c2ccc(=O)[nH]c2 FS-3703 Cc1nc2cc(ccc2s1)C#N FS-3704 c1cc(ccc1c2cnc(s2)N)Cl FS-3705 c1ccc2c(c1)[nH]c(n2)C(=O)N FS-3706 c1cc2c(cc1O)cc(cn2)Br FS-3707 c1cc2c(cc1Cl)CC(=O)CO2 FS-3708 CSc1[nH]c(=O)c2c(n1)CCCC2 FS-3709 COC(=O)c1ccc2c(=O)cc[nH]c2c1Cl FS-3710 C=CCN1C(=O)c2ccccc2C1=O FS-3712 CSc1nc2ccccc2o1 FS-3713 CNc1ccc(cc1C(=O)OC)Br FS-3714 c1cc2c(cc1C(=O)O)OCC2 FS-3715 COC(=O)c1c[nH]nc1C(F)(F)F FS-3716 c1ccnc(c1)N2CCC(CC2)N FS-3717 CN1Cc2cc(ccc2C1=O)Br FS-3718 c1ccc2c(c1)nc(o2)C(F)(F)F FS-3719 CC(=O)c1cc2ccccc2[nH]1 FS-3720 c1cc2c(cc1O)OCCC2=O FS-3721 c1c(cnc2c1c(c[nH]2)C(=O)O)Cl FS-3722 Cc1cc2ccc(cc2[nH]1)Br FS-3723 c1cc2c(c(c1)Br)ocn2 FS-3724 Cc1ccc(cc1F)CC(=O)OC FS-3725 COC(=O)c1ccc(c(c1)O)Cl FS-3726 c1ccc(cc1)Oc2cccc(c2)[C@@H](C#N)O FS-3727 c1cc2c(cc(cc2O)Br)nc1 FS-3728 Cc1cn2c(n1)ccc(n2)Cl FS-3729 c1cc2c(cc1Br)cc(cn2)O FS-3730 CCOC(=O)c1c(cccn1)N FS-3731 c1cc(cnc1)c2cc(n[nH]2)CO FS-3732 C1CNCCC12CC(=O)NC2 FS-3733 c1ccc2c(c1)c(cc(n2)Cl)N FS-3735 c1c(cnc(n1)CN)Br FS-3736 CCC(=O)c1ccc(c(c1)OC)O FS-3737 c1ccc2c(c1)CC(NC2)C(=O)O FS-3738 COc1ccc2c(c1)nc([nH]c2=O)Cl FS-3739 Cn1cc(cnc1=O)Br FS-3740 COC(=O)c1cc([nH]n1)Br FS-3741 COC(=O)c1c(cc[nH]1)Cl FS-3742 COC(=O)c1ccc(c(c1)Cl)C#N FS-3743 c1ccc(cc1)c2c(nccn2)O FS-3744 c1cc2c(cc1F)C(CC2)CC(=O)O FS-3745 COc1cc(ccn1)C(F)(F)F FS-3746 c1cc2c(c(c1)Br)CCNC2=O FS-3747 Cc1cc2ccccc2nc1C#N FS-3748 c1c(c(c(cn1)Br)N)C(=O)O FS-3749 c1c(cnc(n1)C(F)(F)F)O FS-3750 c1cc(c(cc1Br)C(=O)O)C#N FS-3751 c1cc2c(c(c1)Cl)CC(=O)C2 FS-3752 COC(=O)c1cc2c(cc[nH]2)c(c1)O FS-3753 c1cc(cc(c1)c2cn[nH]n2)C#N FS-3754 c1cc2cc(cc(c2nc1)O)F FS-3756 c1cc2c(cc1Br)NC(=O)C2=O FS-3757 c1c(c(cs1)Br)C(=O)O FS-3758 CCOC(=O)c1cnc(n1C)N FS-3759 Cn1cc(c2c1cccc2)CC#N FS-3760 Cc1ccc(cc1C(=O)OC)F FS-3761 COc1cccc(c1Br)C(=O)O FS-3762 COc1cc(ccc1CN)F FS-3763 c1cc2c(cc1F)c(ncn2)O FS-3764 c1ccc2c(c1)c(c[nH]2)CCCN FS-3765 Cc1cc2=NC(=O)N=c2cc1N FS-3766 c1cc2cncnc2cc1Br FS-3767 c1c(c[nH]c-2ncnc12)Br FS-3768 c1c(nc(cn1)N2CCOCC2)N FS-3769 Cc1ccc2cc(ccc2n1)C(=O)O FS-3770 c1c(c[nH]c(=O)c1C#N)Br FS-3771 c1cc(ccc1N2CCNCC2)O FS-3772 c1ccc2c(c1)[nH]c(=O)s2 FS-3774 c1c(c-2c(nc[nH]c2n1)N)Br FS-3775 Cc1cc(=O)[nH]c2c1cc(cc2)Cl FS-3776 c1cc(ncc1O)C(F)(F)F FS-3777 c1c[nH]c2c1cc(cc2C(=O)O)Br FS-3778 c1ccc2c(c1)ccc(c2O)C(=O)O FS-3779 c1csc2n1cc(n2)C(F)(F)F FS-3780 c1ccc2c(c1)CCC(C2)C(=O)O FS-3781 COc1cc(ccc1O)C=C FS-3782 c1cc(n2cc(nc2c1)C(=O)O)C(F)(F)F FS-3783 Cc1cc(n[nH]1)c2ccccn2 FS-3784 COc1c(cc(cn1)N)Cl FS-3785 c1ccc(cc1)n2c3ccccc3[nH]c2=O FS-3786 c1cc2c(cc1C#N)c(=O)[nH]cn2 FS-3787 CC(=O)c1c(cccc1Cl)OC FS-3788 COc1[nH]c(=O)cc(n1)C(F)(F)F FS-3789 c1csc2c1NC(=O)CCC2 FS-3790 CCOc1ncc(c(n1)N)F FS-3791 COc1ccc(c(c1)NC(=O)Oc2ccccc2)OC GA-0050 CN(C)/C=C/C(=O)c1cccc(n1)Br GA-0201 c1cc(ccc1c2nc(sn2)N)Cl GA-0206 CCOC(=O)c1csc(n1)n2c(=O)c(c([nH]2)C)CCO GA-0208 c1ccc(cc1)OC(=O)NCCN2CCOCC2.Cl GA-0215 c1ccc(cc1)OC(=O)NCCN2CCCCC2.Cl GA-0216 c1ccc(cc1)OC(=O)NCCN2CCCC2.Cl GA-0217 CN(C)CCNC(=O)Oc1ccccc1.Cl GA-0218 COc1cccc(c1)OCCN2C(=O)[C@@H]3CN(C[C@@H]3C2=O)S(=O)(=O)c4cccs4 GA-0219 c1ccc(cc1)OCCN2C(=O)[C@@H]3CN(C[C@@H]3C2=O)S(=O)(=O)c4cccs4 GA-0220 CC(C)(CNC(=O)Oc1ccccc1)CN(C)C.Cl GA-0221 CCOCc1nnc(o1)Cn2cc(c(=O)[nH]c2=O)C GA-0223 Cc1ccc(cc1)c2nc(sn2)N GA-0225 c1cnccc1c2nc(sn2)N GA-0226 C1COCCN1c2nc(sn2)N GA-0230 CC(C)(C)c1nc(sn1)N GA-0234 Cc1ccc(cc1F)c2nc(sn2)N GA-0235 c1cc(cc(c1)[N+](=O)[O-])c2nc(sn2)N GA-0236 c1cc(ccc1OCc2nc(sn2)N)F GA-0238 CCc1nn2cc(nc2s1)C(=O)OCC GA-0241 C1CC1c2nc(sn2)N GA-0244 c1ccc(cc1)CN2CCC(CC2)N3CCC(C3)CO GA-0600 CCn1c(=O)c2ccccc2[nH]c1=S GA-0603 CCNC(=O)CNC.Cl GA-0609 COC(=O)c1c(c(n[nH]1)C(=O)OC)I GA-0610 c1cc(ccc1S(=O)(=O)N2CCC(CC2)CO)Br GA-0701 c1cc(ccc1S(=O)(=O)N2CCC(CC2)CO)Cl GA-0703 c1cc(c(cc1Cl)Cl)OCCCC(=O)NN GA-0704 c1cc(c(cc1[N+](=O)[O-])C#N)N2CCOCC2 GA-0706 c1cc(c(cc1[N+](=O)[O-])C#N)N2CCCCC2 GA-0707 COC(=O)c1ccc(c(c1)N)F GA-0709 c1cc(ccc1C2=CSCC(N2)C(=O)O)F GA-0710 c1cc(ccc1C=O)N2CCC(CC2)CO GA-0713 COC(=O)C1CC2(c3ccccc3NC2=O)N(C1)Cc4ccccc4 GA-0714 c1cc(ccc1C#N)N2CCC(CC2)CO GA-0715 COC(=O)c1ccc(cc1)N2CCC(CC2)CO GA-0719 c1ccc(cc1)C2=NNC(=O)CC2CO GA-0720 c1ccc(c(c1)C#N)N2CCC(CC2)C(=O)O GA-0722 c1cc(c(cc1Cl)/C=C/C(=O)O)Cl GA-0723 c1cc(ncc1Cl)NN GA-0724 c1cc(c(nc1)c2ccsc2)C#N GA-0725 c1cc(ncc1C#N)c2ccsc2 GA-0726 c1cc(ccc1C=O)N2CCC(CC2)C(=O)O GA-0728 CNc1ccc(cn1)[N+](=O)[O-] GA-0729 CNc1c(cccn1)C#N GA-0730 CN(C)c1c(cccn1)C#N GA-0731 c1ccc(cc1)CNc2nc(cs2)C(=O)O GA-0732 c1ccc(cc1)/N=c\2/n(c(cs2)C(=O)O)c3ccccc3 GA-0733 C1C(NC(=CS1)C(=O)O)C(=O)O GA-0734 CNc1ccc(cn1)C#N GA-0737 CN(C)c1ccc(cn1)C#N GA-0738 CNc1c(cccn1)[N+](=O)[O-] GA-0739 COC(=O)c1ccc(c(n1)N)[N+](=O)[O-] GA-0750 COC(=O)c1ncn(n1)Cc2c(cc(cn2)C(F)(F)F)Cl GA-0800 c1cc(ccc1NS(=O)(=O)c2cnn(c2)c3ccc(cn3)C(F)(F)F)Cl GA-0801 c1ccc(cc1)COc2ccc(cc2)OCCBr GA-0802 CS(=O)(=O)c1cccc(c1)N2CCNC2=O GA-0804 c1cc(cc(c1)NS(=O)(=O)c2cnn(c2)c3ccc(cn3)C(F)(F)F)C(F)(F)F GA-0806 c1ccc2c(c1)C(=O)N(C2=O)CCCn3cnnc3 GA-0807 COC(=O)c1ccc(cc1)OCCBr GA-0808 CC(=O)N1CCc2c1ccc(c2)S(=O)(=O)N GA-0810 CCOC(=O)c1nnnn1C(C)c2c(cc(cn2)C(F)(F)F)Cl GA-0813 CN(C(=O)c1c(cccc1F)F)OC GA-0816 Cc1cccc2c1nccc2O GA-0817 CN(C(=O)c1ccc(cc1Cl)Cl)OC GA-0818 CC(C)(C)c1ccc(cc1)OCCBr GA-0819 COC(=O)c1ccc(cc1)OCCOc2cccc(c2)C=O GA-0821 COC(=O)c1ccc(cc1)OCCOc2ccc(cc2)C=O GA-0822 c1cc(cc(c1)Br)OCCBr GA-0825 CC(=O)c1cccc(c1)OCCOc2ccc(cc2)C(=O)OC GA-0826 CC(=O)c1ccc(cc1)OCCOc2ccc(cc2)C(=O)OC GA-0827 c1ccc(cc1)COc2ccc(cc2)OCCOc3cccc(c3)C=O GA-0828 c1ccc(cc1)COc2ccc(cc2)OCCOc3ccc(cc3)C=O GA-0829 CC(=O)c1cccc(c1)OCCOc2ccc(cc2)OCc3ccccc3 GA-0831 CC(=O)c1ccc(cc1)OCCOc2ccc(cc2)OCc3ccccc3 GA-0832 COC(=O)c1ccc(c(c1)[N+](=O)[O-])n2cccc2 GA-0833 c1cc(ccc1n2c(c3c(n2)CCCC3)O)Cl GA-0834 c1cc(c(cc1C(=O)NCCO)Cl)Cl GA-0835 c1c(cc(c2c1CCO2)Br)C=O GA-0836 CCOC(=O)c1c2c(sc1N)CN(CC2)C(=O)c3ccccc3 GA-0838 COC(=O)c1cccc(c1)OCCBr GA-0840 COC(=O)c1ccc(cc1)OCCN2CCN(CC2)Cc3ccccc3 GA-0841 CCOC(=O)c1ccc(cc1)OCCN2CCC(CC2)O GA-0842 c1cc2nccn2cc1C(=O)NCCCO GA-0843 CC(c1ccnn1C(=O)C)Sc2c(cccn2)C(F)(F)F GA-0847 COC(=O)c1cccc(c1)OCCOc2cccc(c2)C=O GA-0848 COC(=O)c1cccc(c1)OCCOc2ccc(cc2)C=O GA-0849 CC(=O)c1cccc(c1)OCCOc2cccc(c2)C(=O)OC GA-0850 CC(=O)c1ccc(cc1)OCCOc2cccc(c2)C(=O)OC GA-0851 Cc1ccc2c(c1)c3c([nH]2)CCNC3.Cl GA-0855 CCOC(=O)C1CCCc2c1nc(s2)N GA-0858 CCOC(=O)C1CCCc2c1[nH]c3c2cc(cc3)Cl GA-0859 Cc1ccc2c(c1)nsn2 GA-0860 CCC(CO)NC(=O)c1ccc2nccn2c1 GA-0861 c1ccc(cc1)COc2ccc(cc2)OCCCBr GA-0862 COC(=O)c1ccc(cc1)OCCCOc2cccc(c2)C=O GA-0863 COC(=O)c1ccc(cc1)OCCCOc2ccc(cc2)C=O GA-0864 CC(=O)c1cccc(c1)OCCCOc2ccc(cc2)C(=O)OC GA-0865 CC(=O)c1ccc(cc1)OCCCOc2ccc(cc2)C(=O)OC GA-0866 c1cc2c(cc1CBr)nsn2 GA-0867 c1cc(cnc1)COC(=O)c2cc(cc(n2)C(=O)OCc3cccnc3)C(F)(F)F GA-0868 c1ccc(cc1)COc2ccc(cc2)OCCCOc3cccc(c3)C=O GA-0872 c1ccc(cc1)COc2ccc(cc2)OCCCOc3ccc(cc3)C=O GA-0873 CC(=O)c1cccc(c1)OCCCOc2ccc(cc2)OCc3ccccc3 GA-0874 CC(=O)c1ccc(cc1)OCCCOc2ccc(cc2)OCc3ccccc3 GA-0875 C1CCc2c(nc(s2)Cl)C1 GA-0920 COC(=O)c1cc2cccc(c2s1)F GA-0921 c1cc2c(cc1F)cc(s2)C(=O)O GA-0923 c1cc2c(cc(s2)C(=O)O)c(c1)Br GA-0924 c1cc(cc2c1cc(s2)C(=O)O)Br GA-0925 c1cc2cc(sc2c(c1)F)C(=O)O GA-0926 COC(=O)c1cc2ccc(cc2s1)Cl GA-0927 COC(=O)c1cc2cc(ccc2s1)Cl GA-0932 COC(=O)c1cc2cccc(c2s1)Cl GA-0933 CCOC(=O)c1c(c2cc(ccc2[nH]1)Br)Br GA-0935 c1cc2c(cc1Br)cc([nH]2)CO GA-0936 c1cc2c(cc1Br)cc([nH]2)C(=O)O GA-0937 COC(=O)c1cc2c(cccc2s1)C(F)(F)F GA-0940 COC(=O)c1cc2ccc(cc2s1)C(F)(F)F GA-0941 COC(=O)c1cc2cccc(c2s1)C(F)(F)F GA-0942 c1cc2c(cc(s2)C(=O)O)c(c1)Cl GA-0943 c1cc(cc2c1cc(s2)C(=O)O)Cl GA-0945 c1cc2cc(sc2c(c1)Cl)C(=O)O GA-0946 c1cc(c2cc(sc2c1)C(=O)O)C(F)(F)F GA-0948 c1cc(cc2c1cc(s2)C(=O)O)C(F)(F)F GA-0949 c1cc2cc(sc2c(c1)C(F)(F)F)C(=O)O GA-0950 CS(=O)(=O)c1ccc(cc1)C2=C(C(=O)CC2)Br GA-7001 c1cc2c(cc1Cl)[nH]nc2N GA-7014 c1ccc(cc1)COC(=O)NC(C2CCCCC2)S(=O)(=O)c3ccccc3 GB-0033 COC(=O)CSc1cc(nc(n1)c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F GB-0039 c1cc(ccc1C(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)Cl GB-0051 Cn1c(c(cn1)C(=O)N)N GB-0603 c1cc(cc(c1)S(=O)(=O)N2CCC(CC2)C(F)(F)F)C(F)(F)F GB-0700 c1cc(c(cc1Nc2nc(cs2)C(=O)O)Cl)Cl GB-0702 c1cc(ccc1CN2CCC(CC2)C(F)(F)F)Cl GB-0703 c1ccc(c(c1)S(=O)(=O)N2CCC(CC2)C(F)(F)F)Cl GB-0704 c1ccc(cc1)Nc2nc(cs2)C(=O)O GB-0705 Cc1ccc(cc1)N2CCC(C2=O)C#N GB-0706 c1ccc(cc1)N2CCC(C2=O)C#N GB-0707 c1cc(ccc1S(=O)(=O)N2CCC(CC2)C(F)(F)F)Cl GB-0709 c1ccc(c(c1)S(=O)(=O)N2CCNCC2)Cl GB-0710 CS(=O)(=O)CC(=O)c1ccc(cc1)[N+](=O)[O-] GB-0713 CS(=O)(=O)CC(=O)c1ccc(cc1)Br GB-0714 c1cc(ccc1N2CCC(C2=O)C#N)Cl GB-0715 COc1ccc(cc1)N2CCC(C2=O)C#N GB-0716 c1ccc(cc1)N(c2ccccc2)c3nc(cs3)C(=O)O GB-0720 COC(=O)c1ccc(cc1Cl)N2CCC(CC2)C(F)(F)F GB-0721 COC(=O)C(c1ccc(c(c1)Cl)Cl)N.Cl GB-0722 c1cc2c(cc(s2)C(=O)NN)c(c1)Cl GB-0727 c1cc(ccc1/C=N/NC(=O)c2ccc(cc2)Cl)N3CCC(CC3)C(F)(F)F GB-0729 c1cc(ccc1/C=C\2/C(=O)NC(=O)S2)N3CCC(CC3)C(F)(F)F GB-0730 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)Cl)N3CCC(CC3)C(F)(F)F GB-0731 CN1C(=O)C(=Cc2ccc(cc2)N3CCC(CC3)C(F)(F)F)C(=O)N(C1=O)C GB-0734 c1cc(ccc1C=C2C(=O)NC(=O)NC2=O)N3CCC(CC3)C(F)(F)F GB-0735 CC1(OC(=O)C(=Cc2ccc(cc2)N3CCC(CC3)C(F)(F)F)C(=O)O1)C GB-0736 c1cnc(nc1C(F)(F)F)N GB-0804 c1cc(cnc1)CSC2=N/C(=C/c3ccc(cc3)c4c(cc(cn4)C(F)(F)F)Cl)/C(=O)N2 GB-5000 c1cc(ccc1/C=C/2\C(=O)N=C(S2)N3CCOCC3)c4c(cc(cn4)C(F)(F)F)Cl GB-5001 c1cc(ccc1/C=C/2\C(=O)N=C(S2)N3CCCCC3)c4c(cc(cn4)C(F)(F)F)Cl GB-5003 CN(C)C1=NC(=O)/C(=C\c2ccc(cc2)c3c(cc(cn3)C(F)(F)F)Cl)/S1 GB-5004 c1ccnc(c1)CNC2=NC(=O)/C(=C\c3ccc(cc3)c4c(cc(cn4)C(F)(F)F)Cl)/S2 GB-5005 c1ccc(cc1)CNC2=NC(=O)/C(=C\c3ccc(cc3)c4c(cc(cn4)C(F)(F)F)Cl)/S2 GB-5006 CCNc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl GB-5023 c1ccc(cc1)NCc2ccc(cc2)c3ccc(cn3)C(F)(F)F GB-5024 Cc1cn(c(=O)n(c1=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cc3ccccc3 GC-0001 Cc1cn(c(=O)n(c1=O)Cc2ccc(cc2C(F)(F)F)Cl)Cc3nnc(o3)c4ccc(cc4)Cl GC-0034 c1cc(ccc1[C@H]2NCCS2)OCc3c(cc(cn3)C(F)(F)F)Cl GC-0043 c1cc(c(c(c1)Cl)c2nc(c3n2cc(cc3Cl)C(F)(F)F)[C@H]4NCCS4)Cl GC-0044 c1cocc1C(=O)CC#N GC-0049 c1cscc1C(=O)CC#N GC-0058 CN(C)/C=C(/C=C/C(=O)C(F)(F)F)\C#N GC-0205 CC(C)(C)OC(=O)N1CCN([C@@H](C1)CO)C(=O)Cc2ccc(c(c2)Cl)Cl GC-0208 c1ccc(cc1)c2ccc(cc2)C(=O)CC#N GC-0212 Cn1c2ccccc2c(n1)N GC-0600 c1cc(ccc1c2nnco2)N GC-0604 c1cc(ccc1c2nnc(o2)O)[N+](=O)[O-] GC-0606 c1cc2c(c(c1)I)c(n[nH]2)N GC-0607 c1c(cnc(c1Cl)I)[N+](=O)[O-] GC-0608 CC(C)(C)OC(=O)N1CCC2(CC1)c3cccn3-c4ccc(cc4N2)OC GC-0610 CCOC(=O)c1c(nc(s1)N2CCNCC2)C(F)(F)F GC-0611 CCOC(=O)c1c2c(cc(cn2c(n1)c3ccccc3)C(F)(F)F)Cl GC-0612 c1cc2c(cc1N)cc(o2)C(=O)O GC-0616 c1cc2c(cc1N)cc(o2)C(=O)NN GC-0617 c1cc(ccc1c2nnc(o2)O)N GC-0618 c1ccc(cc1)CNc2c(c(ncn2)Cl)C=O GC-0619 CCOC(=O)c1cc2cc(ccc2o1)NC(=O)OC(C)(C)C GC-0620 c1cc(c(cc1Cl)Cl)Cn2cc(cc(c2=O)Cl)C=O GC-0700 c1c(cnc(c1C#N)O)Br GC-0703 c1c(cnc(c1Br)O)C#N GC-0704 Cc1ccc(cc1)Cn2cc(cc(c2=O)Cl)C=O GC-0705 B(c1cc(ccc1OC)C#N)(O)O GC-0707 CC1C(=O)Nc2cc(ccc2O1)Br GC-0710 c1c(cnc(c1C#N)O)Cl GC-0712 c1cc2c(cc1Br)nc(o2)CCl GC-0713 CC1C(=O)Nc2cc(ccc2O1)C(=O)OC GC-0717 COC(=O)c1ccc2c(c1)OCC(=O)N2 GC-0720 c1ccc(cc1)Cn2cc(cc(c2=O)Cl)C=O GC-0723 CC1C(=O)Nc2ccc(cc2O1)C(=O)OC GC-0724 c1cc(ccc1N2CCC(CC2)CO)[N+](=O)[O-] GC-0725 c1c(cnc(c1C=O)N)Cl GC-0727 c1cc2c(cc1/C=C/C(=O)O)CCO2 GC-0728 Cc1c(cnn1c2ccc(cn2)Cl)C(=O)C GC-0730 c1cc2nncn2cc1Cl GC-0731 CC(C)(C)OC(=O)N1CCC(CC1)(CN)O GC-0732 c1cn2cc(cc(c2n1)I)C(F)(F)F GC-0733 COC(=O)C1(CCOCC1)C#N GC-0734 c1c[nH]c2c1cc(cn2)C(F)(F)F GC-0735 c1cc(ncc1Cl)n2c(cc(n2)C(F)(F)F)O GC-0736 c1cc([nH]c1)/C=C(/C#N)\C(=O)O GC-0737 COC(=O)c1ccc(cc1Br)F GC-0738 c1c(cnc(c1I)O)C#N GC-0739 c1c(cnc(c1Cl)O)C#N GC-0740 c1cc2cc(sc2c(c1)F)C(=O)NN GC-0741 c1cc(cc2c1cc(s2)C(=O)NN)Cl GC-0742 CCOC(=O)/C=C/c1ccc2c(c1)CCO2 GC-0746 COC(=O)c1ccc2c(c1)NCCO2 GC-0747 c1ccnc(c1)c2nc(cc(n2)N3CCNCC3)C(F)(F)F GC-0748 C#Cc1cc(cnc1N)C(F)(F)F GC-0749 c1c(cnc2c1c(c[nH]2)Br)C(F)(F)F GC-0750 CCOC(=O)c1c(ncs1)C GC-0751 CC1CN(N=C1N)c2ccc(cn2)Cl GC-0752 c1c(c(c(cn1)F)C(=O)O)F GC-0754 c1c(cnc(c1Cl)Cl)C#N GC-0755 CC1CC(=NN1c2ccc(cn2)Cl)N GC-0756 c1ccnc(c1)c2ccc(c(n2)Cl)C#N GC-0757 c1c(c[nH]c1C(=O)NN)I GC-0758 c1c(cnc2c1c(c[nH]2)[N+](=O)[O-])C(F)(F)F GC-0759 CCOC(=O)C1CCN(CC1)c2c(cc(cn2)C(=O)O)Cl GC-0760 CCCCc1nc2cc(ccc2o1)Br GC-0764 c1ccnc(c1)c2ncc(c(n2)O)C(=O)O GC-0765 c1c(cnc(c1Br)Cl)C#N GC-0766 CCOC(=O)CCS(=O)(=O)Cl GC-0767 COC(=O)Cc1cn2cc(cc(c2n1)I)Cl GC-0768 CCOC(=O)c1cn2cc(cc(c2n1)I)C(F)(F)F GC-0769 CCOC(=O)c1c(n2cc(ccc2n1)C(F)(F)F)Cl GC-0771 c1cc(c(nc1)c2ccc(cc2)CO)C(F)(F)F GC-0772 c1ccc2c(c1)c(c([nH]2)C(=O)O)Br GC-0773 Cc1ccc(cc1)S(=O)(=O)OCC2(COC2)C GC-0776 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cc(cn2)C(=O)O)Cl GC-0777 CCOC(=O)C1CCN(CC1)c2cc(ccc2[N+](=O)[O-])Cl GC-0778 c1c(c(c(=O)[nH]n1)Cl)N2CCC(CC2)C(F)(F)F GC-0800 Cn1c(c(cn1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)c3ccccc3Cl GC-0801 CC(C)(C)OC(=O)NS(=O)(=O)NCc1c(cc(cn1)C(F)(F)F)Cl GC-0816 c1cnc2c(c1Cl)cc(cc2Cl)C(F)(F)F GD-0001 CC(C)(C)n1c(=O)c(c(cn1)NN)Cl GD-0003 c1cc(c(nc1CCl)Cl)O GD-0006 C[Si](C)(C)C#Cc1cc(nc(c1O)Cl)CO GD-0009 CC(C)(C)n1c(=O)c(ccn1)N GD-0015 c1c[nH]c2c1cc(c(c2)C(F)(F)F)Cl GD-0016 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NCc3c(cc(cn3)C(F)(F)F)Cl GD-0020 c1cc2c(cc1S(=O)(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)CCO2 GD-0021 c1c2c(cc(c1Cl)C(F)(F)F)[nH]cc2Br GD-0025 COC(=O)c1ccc(c(c1)OCc2ccccc2)[N+](=O)[O-] GD-0029 c1ccnc(c1)CNS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl GD-0033 c1cc(ccc1CNS(=O)(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)Cl GD-0034 c1cc(ccc1Oc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)N3CCC(CC3)C(F)(F)F GD-0035 c1ccc(cc1)Oc2ccc(cc2)S(=O)(=O)NCc3c(cc(cn3)C(F)(F)F)Cl GD-0036 c1ccc2c(c1)cccc2S(=O)(=O)NCc3c(cc(cn3)C(F)(F)F)Cl GD-0037 c1cc(c(c(c1)Cl)Cl)S(=O)(=O)NCc2c(cc(cn2)C(F)(F)F)Cl GD-0038 COc1ccc(cc1S(=O)(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Br GD-0039 c1ccc(c(c1)C2=N[C@@H]2c3c(cc(cn3)C(F)(F)F)Cl)Cl GD-0049 c1ccc(cc1)COc2cc(ccc2[N+](=O)[O-])C(=O)O GD-0051 c1ccc(cc1)COc2cc(ccc2[N+](=O)[O-])C(=O)NN GD-0052 COC(=O)c1ccc(c(c1)OCc2ccccc2)N GD-0053 COc1cc(c(cc1C(F)(F)F)[N+](=O)[O-])CC(=O)OC GD-0054 c1cc(ccc1c2nnc(o2)CCCCSc3c(cc(cn3)C(F)(F)F)Cl)Cl GD-0058 c1c(cc(c(c1I)N)I)Br GD-0063 Cc1ccc(cc1)C2=N[C@@H]2c3c(cc(cn3)C(F)(F)F)Cl GD-0067 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2ccc3c(c2)CCO3 GD-0069 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2cccc3c2cccc3 GD-0070 CN(c1c(cc(cn1)C(F)(F)F)Cl)NS(=O)(=O)c2cc(ccc2OC)Br GD-0072 c1cc2c(cc1I)c(=O)c(c[nH]2)C(=O)O GD-0074 C#Cc1cc(c(cc1N)C(F)(F)F)C#N GD-0076 c1c[nH]c2c1cc(c(c2)C(F)(F)F)C#N GD-0077 c1c[nH]c2c1cc(c(c2)C(F)(F)F)[N+](=O)[O-] GD-0078 COc1cc(c(cc1C(F)(F)F)[N+](=O)[O-])CC(=O)O GD-0080 COc1cc2c(cc1C(F)(F)F)NC(=O)C2 GD-0081 CCOC(=O)c1c[nH]c2c(cc(cc2c1=O)I)C GD-0084 CCOC(=O)c1c[nH]c2ccc(cc2c1=O)I GD-0085 c1c(c(cc2c1c(c[nH]2)Br)C(F)(F)F)C#N GD-0089 c1ccc(cc1)CNc2c(cc(cn2)Br)C(=O)O GD-0090 Cc1cc(cc2c1[nH]cc(c2=O)C(=O)O)I GD-0093 c1ccc(cc1)CNc2c(cc(cn2)Cl)C(=O)O GD-0094 CC(C)(C)n1cc(cc1N)C#N GD-0202 c1cc(ccc1c2ccc(c(c2)F)Cl)C(=O)NN GD-0207 Cc1cc(c2c(cn(c2n1)C(C)(C)C)C#N)C(F)(F)F GD-0209 CC(C)(C)OC(=O)Nc1nc(c(o1)C(=O)O)C(F)(F)F GD-0210 CC(C)(C)n1cc(c2c1nc(cc2C(F)(F)F)C(F)(F)F)C#N GD-0213 CC(C)(C)n1cc(c2c1nc(nc2C(F)(F)F)C(F)(F)F)C#N GD-0217 Cc1cc(c2c(cn(c2n1)C(C)(C)C)C(=O)N)C(F)(F)F GD-0220 c1c(c2c([nH]nc2O)nc1C(F)(F)F)C(F)(F)F GD-0225 CCOC(=O)C[C@H]1CNC[C@H](N1C)CC(=O)OCC.CC(=O)O GD-0226 CC(=O)O[Pd]([NH+](C1CCCCC1)C2CCCCC2)([NH+](C3CCCCC3)C4CCCCC4)OC(=O)C GD-0228 c1c(c(c(nc1C(F)(F)F)N)C(=O)N)C(F)(F)F GD-0236 CC(C)(C)n1cc(c2c1nc(nc2C(F)(F)F)C(F)(F)F)C(=O)N GD-0239 CC(C)(C)n1cc(c2c1nccc2C(F)(F)F)C#N GD-0240 Cc1c(cc(c(=O)[nH]1)Br)C(=O)C GD-0241 CCOC(=O)c1c(ccnc1Cl)Cl GD-0700 c1ccc(cc1)n2cc(c(n2)C(F)(F)F)O GD-0702 C#Cc1cnc(c(c1N)I)Cl GD-0703 c1cc(c(cc1N)CO)F GD-0704 c1ccc(cc1)/C(=C/C#N)/N GD-0705 CCOC(=O)c1cccn2c1ncc2 GD-0707 C1C[C@@H]2[C@H]1C(=O)NC(=O)N2 GD-0711 CNCc1cccnc1Cl GD-0716 c1cc2nc(c(n2cc1C(F)(F)F)[N+](=O)[O-])C(=O)O GD-0717 c1cc2c(c(c1)N)C(=O)CC2O GD-0718 COc1c(c(nc(n1)SC)C(F)(F)F)C(=O)O GD-0719 COC(=O)c1c[nH]c(n1)N GD-0723 CCOC(=O)c1cc2cccnc2s1 GD-0724 COc1c(cccn1)CO GD-0733 c1cc(nc(c1CCl)Cl)Cl GD-0735 COC(=O)CC1c2ccccc2CCN1 GD-0737 c1cc2ncc(n2cc1C(F)(F)F)[N+](=O)[O-] GD-0742 c1cc2c(cc1C(=O)O)[nH]c(=O)o2 GD-0744 c1cnc(c(c1C(F)(F)F)C(=O)O)Cl GD-0745 COC(=O)c1ccc2c(c1)[nH]c(=O)c(=O)[nH]2 GD-0747 CN(C)c1ccc(c(n1)Cl)C=O GD-0748 COC(=O)c1ccc2c(c1)nc(c(n2)Cl)Cl GD-0751 COC(=O)c1ccc2c(c1)OCCN2 GD-0753 COC(=O)c1c(ccnc1Cl)C(F)(F)F GD-0754 Cc1ccc(cc1)S(=O)(=O)O/C(=C/C#N)/c2ccccc2 GD-0756 c1cc2cc(sc2nc1)C(=O)CC#N GD-0761 CC(C)C1CN(CCN1)c2c(cc(cn2)C(F)(F)F)Cl GE-0003 CCCOCCn1c2cc(ncc2nc(c1=O)N3CCN(CC3)CCO)Cl GE-0008 Cc1cc(cc(c1Oc2cc(nc(n2)Nc3ccc(cc3)C#N)N)C)C#N GE-0012 COc1ccc2cc(c(nc2c1)N3CCCC3)c4cccc(c4)C(F)(F)F GE-0014 CC(C)(C)CNC(=O)c1ccc(nc1)Br GE-0021 Cc1ccc(c(c1)NC2CCN(CC2)C(=O)OC(C)(C)C)[N+](=O)[O-] GE-0022 c1cc(cc(c1)S(=O)(=O)Nc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F GE-0033 c1cc(ccc1NC(=O)Nc2nnc(s2)c3c(cc(cn3)C(F)(F)F)Cl)Cl GE-0035 c1c(cnc(c1Cl)N2CCC3(CC2)CNC(=O)O3)C(F)(F)F GE-0046 Cc1cc(cc(c1Oc2c(c(nc(n2)Nc3ccc(cc3Br)C#N)N)Br)C)C#N GE-0050 Cc1ccc(c(c1)NC2CCN(CC2)C(=O)OC(C)(C)C)N GE-0055 c1cc(ccc1S(=O)(=O)NC(=O)Nc2nnc(s2)c3c(cc(cn3)C(F)(F)F)Cl)Cl GE-0060 c1ccc(c(c1)NC(=O)Nc2nnc(s2)c3c(cc(cn3)C(F)(F)F)Cl)Cl GE-0061 c1ccc(c(c1)S(=O)(=O)NC(=O)Nc2nnc(s2)c3c(cc(cn3)C(F)(F)F)Cl)Cl GE-0062 c1cc(ccc1C#N)NC(=N)N.[N+](=O)(O)[O-] GE-0066 Cc1cc(c(cc1F)[N+](=O)[O-])NC2CCN(CC2)C(=O)OC(C)(C)C GE-0076 c1cc(ccc1S(=O)(=O)NCc2ccc(nc2N3CCC(CC3)C(F)(F)F)C(F)(F)F)Cl GE-0091 Cn1cc(c2c1cccc2)CC(=O)N GE-0097 c1c(cnc(c1Cl)N2CCC(CC2)CCCO)C(F)(F)F GE-0202 CCOC(=O)c1cnc(nc1NCc2ccc(c(c2)Cl)OC)SC GE-0212 CCOC(=O)c1cnc(nc1NCc2ccc(c(c2)Cl)OC)N3CCC[C@H]3CO GE-0219 CC(C)S(=O)(=O)N[C@H]1CCCN(C1)c2c(cc(cn2)C(F)(F)F)Cl GE-0225 COC(=O)c1ccncc1C(F)(F)F GE-0233 c1cnc(nc1)C(=N)N GE-0236 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(nc2)Cl GE-0237 c1cncc(c1C(=O)O)C(F)(F)F GE-0239 c1cc(ccc1N2CCOCC2=O)[N+](=O)[O-] GE-0240 c1cc2ncc(n2cc1C(F)(F)F)C(=O)O GE-0243 COC(=O)c1cc(ncc1Br)Cl GE-0244 COc1cc(nc(n1)c2ccccc2)C(=O)O GE-0701 CC(C)C1CN(CCN1c2ccc(cc2C(=O)OC)[N+](=O)[O-])Cc3ccccc3 GE-0702 COC(=O)c1cc(cnc1S(=O)(=O)C)Cl GE-0703 COc1ccc2c(c1)[nH]c(=O)c3n2ccc3 GE-0704 CC(C)C1CNCCN1c2ccc(cc2C(=O)OC)N GE-0705 c1c(cnc(c1I)Cl)C(=O)N GE-0706 CC(C)(C)OC(=O)N1CCc2c(sc3c2c(ncn3)N)C1 GE-0707 CCNc1cc(ccc1N)C(=O)OC GE-0708 CCn1cnc2c1cc(cc2)C(=O)OC GE-0709 COc1cc2c(cc1OC)-n3cccc3C4(N2)CCNCC4.Cl GE-0710 COC(=O)c1ccc(c(c1O)Br)N GE-0711 COc1ccc2c(c1)nc(c3n2ccc3)Cl GE-0712 COC(=O)c1ccc(c(c1)O)C#N GE-0714 Cn1c2ccc(cc2oc1=O)Br GE-0717 Cc1ccc-2c(c1)NC3(CCNCC3)c4n2ccc4.Cl GE-0718 c1c(cnc(c1Cl)N2CCC(C2)O)C(F)(F)F GE-0719 COC(=O)c1ccc(c(c1)N)n2cccc2 GE-0720 CCOC(=O)c1c(nc2ccccc2n1)Cl GE-0721 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2C(=O)NN)[N+](=O)[O-] GE-0723 CC(C)C1CN(CCN1c2ccc(cc2C(=O)OC)N)Cc3ccccc3 GE-0724 COC(=O)c1ccc-2c(c1)NC3(CCNCC3)c4n2ccc4.Cl GE-0725 c1cc2c(c[nH]c2nc1)CO GE-0726 c1cc2c(cc1I)oc(=O)[nH]2 GE-0727 Cn1c(cnc1c2ccccc2)C=O GE-0731 c1cc(c(nc1)CO)Cl GE-0733 CC(C)(C)OC(=O)n1cc(c2c1nccc2)C=O GE-0735 Cn1c2ccc(cc2oc1=O)I GE-0736 COC(=O)c1ccc2c(c1)[nH]c(=O)c3n2ccc3 GE-0737 Cn1cc(nc1c2ccccc2)C=O GE-0738 c1cc(c(cc1N)O)F GE-0739 CC(C)(C)OC(=O)n1cc(c2c1nccc2)CO GE-0740 COc1c(nc2ccccc2n1)C(=O)O GE-0741 COc1c(cc(cn1)C(=O)OC)I GE-0742 c1c(cnc(c1I)Cl)C#N GE-0743 Cn1cnc(n1)CO GE-0745 Cn1cnc(n1)CCl.Cl GE-0746 COC(=O)c1cc(ncc1N)I GE-0747 c1ccc2c(c1)cc([nH]2)c3c(cc(cn3)C(F)(F)F)Cl GF-0010 c1c(cn2c(nnc2c1Cl)CBr)C(F)(F)F GF-0014 Cc1ccc(c(c1)c2ccc(cc2)C(F)(F)F)C(=O)O GF-0026 CCOC(=O)c1csc(n1)Br GF-0027 c1ccc2c(c1)N(c3ccccc3S2)CCN.Cl GF-0032 c1ccc(cc1)COC(=O)N2CCC(CC2)C3CN(C(=O)O3)c4ccccc4 GF-0047 c1ccc(c(c1)c2cnc([nH]2)c3c(cc(cn3)C(F)(F)F)Cl)Cl GF-0053 C1CC2C(C1)C\3CC2C/C3=N\O GF-0055 c1c(cnc(c1Cl)n2cnc3c2ncnc3N)C(F)(F)F GF-0070 CC(C)(C)OC(=O)N1CCN(CC1)c2ccccc2/C=C\c3ccccc3N4CCN(CC4)C(=O)OC(C)(C)C GF-0075 C1CN(C(=O)N1)CCN2CCSCC2 GF-0083 c1cc(c(c(c1)Cl)CO)F GF-0090 c1ccc(cc1)COC(=O)N2CCC3(CC2)CN(C(=O)O3)c4cccc(c4)F GF-0092 c1ccc(cc1)N2CC3(CCNCC3)OC2=O GF-0106 CC(C)NC(=O)C(C)(C)Nc1c(cc(cn1)C(F)(F)F)Cl GF-0107 c1cc(cc(c1)Cl)N2CCNCC2 GF-0110 c1cc(cnc1)C2CCCN2 GF-0112 CC(=O)c1ccc(c(c1)OC)OC GF-0115 c1ccc(c(c1)Cl)Cl GF-0116 c1cc(ccc1C2(CCNCC2)O)Cl GF-0117 c1ccc(cc1)/C=C/CN2CCNCC2 GF-0118 c1ccc(cc1)C(c2ccccc2)N3CCNCC3 GF-0119 COc1cc2c(cc1OC)C(=O)CC2 GF-0120 c1cc2c(cc1Cl)[nH]c(=O)n2C3CCNCC3 GF-0121 c1cc2c(cc1O)NC(=O)CC2 GF-0122 c1ccc2c(c1)CCC(=O)N2 GF-0123 c1cc(c(c(c1)Cl)Cl)N2CCNCC2 GF-0124 c1ccc2c(c1)[nH]c(=O)n2C3=CCNCC3 GF-0125 c1ccc2c(c1)c3c([nH]2)CCCC3=O GF-0126 c1ccn2c(c1)n[nH]c2=O GF-0127 c1ccc2c(c1)c(ns2)N3CCNCC3 GF-0131 c1ccc(cc1)C(c2ccc(cc2)Cl)N3CCNCC3 GF-0133 Cc1cccc(c1)CN2CCNCC2 GF-0134 c1cc2c(cc1F)onc2C3CCNCC3 GF-0135 c1ccc2c(c1)CCc3ccccc3N2 GF-0137 c1ccc2c(c1)c(=O)[nH]c(n2)S GF-0138 COc1cc(cc(c1OC)OC)O GF-0143 CCOC(=O)C=C1CN(C1)C(=O)OC(C)(C)C GF-0212 c1cc(c(nc1)CO)F GF-0219 C1CC(CNC1)c2nc(on2)C(F)(F)F.Cl GF-0229 CC(C)(C)OC(=O)N1C[C@@H]2C[C@@H]2[C@@H]1C(=O)O GF-0238 c1ccn(c1)c2cc(c(cc2N)Cl)C(F)(F)F GF-0700 c1cc(c(nc1)C(=O)O)F GF-0701 Cn1cc(c(n1)C(F)(F)F)C#N GF-0702 c1c(cnc(c1C=O)N)I GF-0703 c1c(cc(nc1Cl)Cl)C=O GF-0706 Cn1c2ccc(cc2c(n1)I)[N+](=O)[O-] GF-0707 c1cc(c(cc1[N+](=O)[O-])F)CCl GF-0710 c1cc(cc(c1)S(=O)(=O)N)NN.Cl GF-0715 c1cc2c(cc1[N+](=O)[O-])[nH]c(=O)cn2 GF-0716 c1c(cnc2c1ocn2)Br GF-0717 c1cnc(c(c1Cl)I)N GF-0718 COC(=O)Cc1cc2c(cc1C#N)OCO2 GF-0719 COc1cc2ccccc2c(c1O)Br GF-0721 c1cc(nc2c1[nH]c(c2)C(=O)O)Cl GF-0722 CC(C)(C)n1c2c(cn1)c(ncn2)N GF-0723 c1cc2c(cc1[N+](=O)[O-])nc(cn2)Cl GF-0726 CCOC(=O)c1nc(cs1)CCl GF-0727 c1c(c(cc2c1OCO2)C#N)CC(=O)O GF-0730 CCOC(=O)c1cnc(cc1NN)Cl GF-0732 CCOC(=O)c1cc2cc(cnc2nc1O)I GF-0733 CCOC(=O)c1cc2cc(cnc2nc1Cl)I GF-0734 CC(=O)Nc1cc(c(cc1N)OC)Cl GF-0735 CCOC(=O)c1c[nH]c(=O)c(c1Cl)[N+](=O)[O-] GF-0737 c1cc(ncc1Cl)C(=O)CC#N GF-0739 c1c(cnc2c1n(c(=O)[nH]2)C3CCCC3)Br GG-0019 Cc1c(cc(n1C)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NCC#C GG-0044 Cc1ccc2c(cccc2n1)C(=O)O GG-0060 CN1CCC(=CC1)C(=O)OC GG-0063 Cc1ccc(cc1)S(=O)(=O)N/N=C(/c2ccc(cc2)OC)\c3c(cc(cn3)C(F)(F)F)Cl GG-0071 Cc1ccc(cc1)S(=O)(=O)N/N=C(\c2ccc(cc2)Cl)/c3c(cc(cn3)C(F)(F)F)Cl GG-0072 COc1ccc(cc1)c2c3c(cc(cn3nn2)C(F)(F)F)Cl GG-0073 c1cc2cc(cnc2c(c1)[N+](=O)[O-])I GG-0202 c1cnc2c(c1Br)c(c[nH]2)I GG-0205 CN1CCc2c(c3cc(ccc3n2Cc4ccc(cc4)C(=O)OC)Cl)C1 GG-0209 c1cc2cc(cnc2c(c1)N)I GG-0221 c1(c(nc(nc1O)N)N)Br GG-0242 c1cc(ccc1C#N)Nc2nccc(n2)CO GG-0701 CC(=O)C1(CC1)C(=O)O GG-0702 CCOC(=O)C1(CC1)C(=O)C GG-0703 CCOC(=O)C1(CCCC1)C(=O)C GG-0704 C1CCC(C1)(C(=O)N)C(=O)O GG-0707 C1CC1(C(=O)N)C(=O)O GG-0709 C1CCC(CC1)(C(=O)N)C(=O)O GG-0710 CCOC(=O)C1(CCC1)C(=O)C GG-0714 CC(C)(C)OC(=O)N1CCC2(C1)CCCCN2 GG-0718 COC(=O)c1cccc(c1)C(=O)NCCc2ccccc2 GH-0059 COC(=O)c1cccc(c1)C(=O)NCc2ccccc2 GH-0060 COC(=O)c1cccc(c1)C(=O)Nc2ccccc2 GH-0061 COc1ccc(cc1)NC(=O)c2cccc(c2)C(=O)OC GH-0062 COC(=O)c1cccc(c1)C(=O)NCCc2ccncc2 GH-0063 Cc1cc(=O)[nH]c2c1ccc(c2)Br GH-0204 CNC(=O)N1CCN(CC1)c2ccc(c(n2)Cl)C(F)(F)F GH-0219 COC(=O)c1ccc(cc1)c2cccc(c2)N GH-0701 c1c(c(cnc1Cl)Cl)C(F)F GH-0704 c1c(cnc(c1Cl)Cl)C(F)F GH-0705 CCc1cscn1 GH-0707 c1cnc(c(c1C(F)(F)F)CO)Cl GH-0708 CCOC(=O)c1cc(c(nc1Cl)Cl)C#N GH-0710 COC(=O)c1ccc(c(c1)[N+](=O)[O-])[N+](=O)[O-] GH-0718 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])[N+](=O)[O-] GH-0719 c1c(cnc(c1C#N)N)C(F)(F)F GH-0720 CC(=O)Nc1cc(ccc1NC)C(=O)OC GH-0722 B1(OC(C(O1)(C)C)(C)C)c2ccc3c(c2)CCCO3 GH-0724 B1(OC(C(O1)(C)C)(C)C)c2ccc(cc2)NC(C)C GH-0725 CC(=O)NC(Cc1cc(ccc1Cl)N)C(=O)OC GK-0702 CCOC(=O)c1cc2ccc(cc2o1)Br GK-0703 c1cc(ncc1COC(=O)c2ccc(nc2)C(F)(F)F)C(F)(F)F GK-0710 C=CC(C(F)(F)F)(C(F)(F)F)O GS-0001 C1C2CC(C1C=C2)CC(C(F)(F)F)(C(F)(F)F)O GS-0002 CC(=O)CC(C(F)(F)F)(C(F)(F)F)O GS-0003 C(CO)C(C(F)(F)F)(C(F)(F)F)O GS-0004 CC(CC(C(F)(F)F)(C(F)(F)F)O)O GS-0005 c1ccc(cc1)C2C3C4CCC(C4)C3c5cc(ccc5N2)C(=O)O GS-0012 c1ccc2c(c1)/c(=N/N)/[nH]nc2NN GS-0013 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)C=O GS-0015 c1ccc2cc(ccc2c1)S(=O)(=O)Nc3ccc(c4c3cccc4)NS(=O)(=O)c5ccc6ccccc6c5 GS-0017 c1ccc2c(c1)C(=O)N(C2=O)C[C@H](CNc3ccc(cc3)N4CCOCC4=O)O GS-0019 COC(=O)[C@H](Cc1cccc2c1cccc2)CC(=O)O GS-0020 c1[nH]c2c(n1)c(=O)[nH]nn2 GS-0021 CC(=O)N[C@@H](Cc1cccc(c1)O)C(=O)O GS-0024 c1ccc2cc(ccc2c1)C[C@H](C(=O)O)NC(=O)OCC3c4ccccc4-c5c3cccc5 GS-0025 c1ccc2cc(ccc2c1)C[C@H](C(=O)O)NC(=O)OCC3c4ccccc4-c5c3cccc5 GS-0026 CC(=O)N/C(=C\c1ccc(c(c1)OC)OC)/C(=O)O GS-0027 CC(=O)N[C@@H](Cc1cccc(c1)O)C(=O)O GS-0028 CC(C)(C)OC(=O)N[C@@H](Cc1ccc(cc1)Cl)C(=O)O GS-0029 CC(C)(C)OC(=O)N[C@@H](Cc1ccc(cc1)Cl)C(=O)O GS-0030 c1ccc2c(c1)-c3ccccc3C2COC(=O)N[C@H](Cc4ccc(cc4)[N+](=O)[O-])C(=O)O GS-0031 CC(=O)N/C(=C\c1cccs1)/C(=O)O GS-0032 c1ccc(cc1)COC(=O)[C@H](Cc2cccs2)N GS-0033 CC(C)(C)OC(=O)N[C@@H](Cc1ccc(cc1)[N+](=O)[O-])C(=O)O GS-0035 c1cc(ccc1C[C@H](C(=O)O)N)[N+](=O)[O-] GS-0036 CC(C)(C)OC(=O)N[C@@H](Cc1ccc(cc1)[N+](=O)[O-])C(=O)O GS-0037 c1ccc2c(c1)-c3ccccc3C2COC(=O)N[C@H](Cc4ccc(cc4)Cl)C(=O)O GS-0038 Cc1c(c2ccccc2[nH]1)C(=O)c3cccc4c3cccc4 GS-0039 CC(=O)N/C(=C/c1cc(cc(c1)F)F)/C(=O)O GS-0041 CC(=O)N/C(=C\c1ccc(cc1)[N+](=O)[O-])/C(=O)O GS-0042 CC1=N/C(=C\c2cccnc2)/C(=O)O1 GS-0043 COC(=O)NC1=Cc2cc(cc(c2OC1)F)F GS-0044 c1ccc(cc1)CN2c3ccccc3C(=O)C2=O GS-0045 c1cc(ccc1c2nc(on2)[C@@H]3C[C@H](CN3)O)F GS-0100 Cc1ccc(cc1)c2nc(on2)[C@@H]3C[C@H](CN3)O GS-0101 c1cc(ccc1c2nc(on2)[C@@H]3C[C@H](CN3)O)Cl GS-0102 c1cnc(cn1)c2nc(on2)[C@@H]3C[C@H](CN3)O GS-0103 Cc1nc(on1)[C@@H]2C[C@H](CN2)O GS-0104 c1cnccc1c2nc(on2)[C@@H]3C[C@H](CN3)O GS-0105 c1ccc(cc1)c2nc(on2)[C@@H]3C[C@H](CN3)O GS-0106 COc1ccc(cc1)c2nc(on2)[C@@H]3C[C@H](CN3)O GS-0107 CC(C)c1nc(on1)[C@@H]2C[C@H](CN2)O GS-0108 c1cc(ccc1c2nc(on2)[C@@H]3Cc4c([nH]cn4)CN3)F GS-0109 c1cnccc1c2nc(on2)[C@@H]3Cc4c([nH]cn4)CN3 GS-0110 c1ccc(cc1)c2nc(on2)[C@@H]3Cc4c([nH]cn4)CN3 GS-0111 CC(C)c1nc(on1)[C@@H]2Cc3c(nc[nH]3)CN2 GS-0112 c1ccc(cc1)Cc2nc(on2)[C@@H]3Cc4c([nH]cn4)CN3 GS-0113 c1[nH]c2c(n1)C[C@H](NC2)c3nc(no3)C4CC4 GS-0114 Cc1ccc(cc1)c2nc(on2)[C@@H]3Cc4c([nH]cn4)CN3 GS-0115 Cc1c(c(n(n1)c2ccc(cc2)OC)C)[C@@H]3C[C@@H](C=C3)O GS-0116 Cc1c(c(n(n1)c2ccccc2)C)[C@@H]3C[C@@H](C=C3)O GS-0117 Cc1c(c(n(n1)c2ccccn2)C)[C@@H]3C[C@@H](C=C3)O GS-0118 Cc1c(c(n(n1)CCO)C)[C@@H]2C[C@@H](C=C2)O GS-0119 Cc1c(c(n(n1)C)C)[C@@H]2C[C@@H](C=C2)O GS-0120 Cc1c(c(n[nH]1)C)[C@@H]2C[C@@H](C=C2)O GS-0121 Cc1c(c(n(n1)C(C)(C)C)C)[C@@H]2C[C@@H](C=C2)O GS-0122 Cc1c(c(n(n1)CC(F)(F)F)C)[C@@H]2C[C@@H](C=C2)O GS-0123 CO[C@@H]1CO[C@H]2[C@@H]1OC[C@@H]2N GS-0124 c1ccc(cc1)CO[C@@H]2CO[C@H]3[C@@H]2OC[C@@H]3N GS-0125 CC(C)NC(=O)O[C@@H]1CO[C@H]2[C@@H]1OC[C@@H]2N GS-0126 c1ccc(cc1)NC(=O)O[C@@H]2CO[C@H]3[C@@H]2OC[C@@H]3N GS-0127 COc1cccc(c1)NC(=O)O[C@@H]2CO[C@H]3[C@@H]2OC[C@@H]3N GS-0128 c1cc(cc(c1)F)NC(=O)O[C@@H]2CO[C@H]3[C@@H]2OC[C@@H]3N GS-0129 c1cc(cc(c1)F)CO[C@@H]2CO[C@H]3[C@@H]2OC[C@@H]3N GS-0130 COc1cccc(c1)CO[C@@H]2CO[C@H]3[C@@H]2OC[C@@H]3N GS-0131 C1[C@@H]([C@@H]2[C@H](O1)[C@@H](CO2)O)N GS-0132 c1ccc(cc1)c2cc(no2)C[C@H]3CNCC[C@H]3CC(=O)O GS-0133 c1c(noc1C2CC2)C[C@H]3CNCC[C@H]3CC(=O)O GS-0134 c1c(noc1CO)C[C@H]2CNCC[C@H]2CC(=O)O GS-0135 COCc1cc(no1)C[C@H]2CNCC[C@H]2CC(=O)O GS-0136 c1c(onc1C[C@H]2CNCC[C@H]2CC(=O)O)CCCC#N GS-0137 Cc1c(c(n(n1)CCC#N)C)[C@@H]2C[C@@H](C=C2)O GS-0138 C1C[C@H](N(C1)CC[C@H]2CNCC[C@H]2CC(=O)O)CO GS-0139 CN1CCN(CC1)[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0140 C1CCN(C1)[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0141 CC(=O)N1CCN(CC1)[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0142 c1ccc(cc1)S[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0143 CCN(CC)[C@@H]1[C@H]([C@@H]([C@H]2CO[C@@H]1O2)N)O GS-0144 C1COCCN1[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0145 C[C@@H]([C@@H]1CC[C@@H](O1)C(=O)NCCCn2ccnc2)N GS-0146 C[C@@H]([C@@H]1CC[C@@H](O1)C(=O)NC(C)C)N GS-0147 COC(=O)[C@@H](Cn1cc(c(=O)[nH]c1=O)Cl)N GS-0148 COC(=O)[C@@H](Cn1cc(c(=O)[nH]c1=O)Br)N GS-0149 CN1CCN(CC1)CC[C@H]2CNCC[C@H]2CC(=O)O GS-0150 CN(CC[C@H]1CNCC[C@H]1CC(=O)O)Cc2ccccc2 GS-0151 C1CNC[C@@H]([C@@H]1CC(=O)O)CCN2CCC(CC2)O GS-0152 CN(CC[C@H]1CNCC[C@H]1CC(=O)O)Cc2cccnc2 GS-0153 CN(CC[C@H]1CNCC[C@H]1CC(=O)O)c2ccc(cc2)F GS-0154 C[C@@H]([C@@H]1CC[C@@H](O1)C(=O)NCc2ccccc2)N GS-0155 C[C@@H]([C@@H]1CC[C@@H](O1)C(=O)N2CCOCC2)N GS-0156 COc1ccc(cc1)c2nnc(o2)[C@H]3CCNC3 GS-0157 c1ccc(cc1)c2nnc(o2)[C@H]3CCNC3 GS-0158 c1ccc2c(c1)c(c[nH]2)Cc3nnc(o3)[C@H]4CCNC4 GS-0159 c1cc(ccc1c2nnc(o2)[C@H]3CCNC3)Cl GS-0160 c1cnccc1c2nnc(o2)[C@H]3CCNC3 GS-0161 c1cc(ccc1c2nc(on2)[C@@H]3C[C@H](CN3)O)C(F)(F)F GS-0162 c1ccnc(c1)c2cc(no2)CC3(COC3)N GS-0163 CC(C)(c1cc(no1)CC2(COC2)N)O GS-0164 c1cc(oc1)c2cc(c(nc2C#N)C(=O)O)O GS-0165 c1cc(sc1)c2cc(c(nc2C#N)C(=O)O)O GS-0166 C1C[C@H](N(C1)[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O)CO GS-0167 CN(Cc1ccccc1)[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0168 CCN(CC)CC[C@H]1CNCC[C@H]1CC(=O)OC GS-0169 C1CNC[C@@H]([C@@H]1CC(=O)O)CCN2CCOCC2 GS-0170 COc1ccc(cc1)CCN[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0171 CN(Cc1cccnc1)[C@@H]2[C@H]([C@@H]([C@H]3CO[C@@H]2O3)N)O GS-0172 Cn1c(cc(n1)c2ccccc2)[C@H]3CN4CC[C@H]3C[C@@H]4CO GS-0173 Cn1c(cc(n1)c2ccco2)[C@H]3CN4CC[C@H]3C[C@@H]4CN GS-0174 C=C[C@H]1C[N@@]2CC[C@H]1C[C@@H]2CNC(=O)c3ccccc3 GS-0175 Cc1ccc(cc1)C(=O)NC[C@H]2C[C@@H]3CC[N@]2C[C@@H]3C=C GS-0176 C=C[C@H]1C[N@@]2CC[C@H]1C[C@@H]2CNC(=O)c3cccc(c3)F GS-0177 CCCNC(=O)NC[C@H]1C[C@@H]2CC[N@]1C[C@@H]2C=C GS-0178 c1cc(cnc1)Cn2cc(nn2)[C@H]3CN4CC[C@H]3C[C@@H]4CO GS-0179 COC(=O)c1c(cc(c(n1)C#N)c2ccco2)O GS-0180 c1cc(cc(c1)Cl)c2c[nH]c(n2)[C@@H]3COCCN3 GS-0181 CC(C)n1cc(nn1)[C@H]2CN3CC[C@H]2C[C@@H]3CO GS-0182 C1COCCN1[C@H]2[C@H](O[C@H]([C@H]2O)CO)CN GS-0183 c1ccc2c(c1)CCN(C2)[C@H]3[C@H](O[C@H]([C@H]3O)CO)CN GS-0184 COC[C@H]1CCCN1[C@H]2[C@H](O[C@H]([C@H]2O)CO)CN GS-0185 CC1CCN(CC1)[C@H]2[C@H](O[C@H]([C@H]2O)CO)CN GS-0186 CN(Cc1cccc(c1)F)[C@H]2[C@H](O[C@H]([C@H]2O)CO)CN GS-0187 CN1CCN(CC1)[C@H]2[C@H](O[C@H]([C@H]2O)CO)CN GS-0188 C1CCN(CC1)[C@H]2[C@H](O[C@H]([C@H]2O)CO)CN GS-0189 COCCN1CCN(CC1)[C@H]2[C@H](O[C@H]([C@H]2O)CO)CN GS-0190 c1cc2c(cc1F)[nH]c(n2)[C@H]3CCNC3 GS-0191 c1ccc2c(c1)[nH]c(n2)[C@H]3CCNC3 GS-0192 c1cc2c(cc1C(F)(F)F)nc([nH]2)[C@H]3CCNC3 GS-0193 COc1ccc2c(c1)[nH]c(n2)[C@H]3CCNC3 GS-0194 COC(=O)c1ccc2c(c1)nc([nH]2)[C@H]3CCNC3 GS-0195 CC(C)(C)c1cc(no1)CC2(COC2)N GS-0196 CN(Cc1ccccc1)Cc2cc(no2)CC3(COC3)N GS-0197 c1c(noc1CN2CCOCC2)CC3(COC3)N GS-0198 c1c(noc1CN2CCCCC2)CC3(COC3)N GS-0199 c1cc(ccc1c2c[nH]c(n2)[C@@H]3COCCN3)C(F)(F)F GS-0200 c1cc(sc1c2c[nH]c(n2)[C@@H]3COCCN3)Cl GS-0201 c1cc(c(cc1F)F)c2c[nH]c(n2)[C@@H]3COCCN3 GS-0202 c1c(nnn1C[C@@H](CO)O)[C@H]2CN3CC[C@H]2C[C@@H]3CO GS-0203 c1c(nnn1C2CCNCC2)[C@H]3CN4CC[C@H]3C[C@@H]4CO GS-0204 c1ccc(cc1)Cn2cc(nn2)[C@H]3CN4CC[C@H]3C[C@@H]4CO GS-0205 c1ccc2c(c1)CCN2C(=O)C[C@H]3[C@@H]([C@@H]([C@H](O3)CN)O)O GS-0206 c1cc(ccc1CNC(=O)C[C@H]2[C@@H]([C@@H]([C@H](O2)CN)O)O)F GS-0207 c1ccc(cc1)NC(=O)C[C@H]2[C@@H]([C@@H]([C@H](O2)CN)O)O GS-0208 c1ccc(c(c1)CN2C[C@@H]3[C@H](C2)OCC(=O)N3)F GS-0209 c1ccc(cc1)CCCN2C[C@@H]3[C@H](C2)OCC(=O)N3 GS-0210 c1cc2c(cc1CN3C[C@@H]4[C@H](C3)OCC(=O)N4)OCO2 GS-0211 c1ccc(c(c1)CN2C[C@@H]3[C@H](C2)OCC(=O)N3)Cl GS-0212 c1cc(ncc1C2C[C@H]([C@H]([C@@H]2N)O)O)N3CCOCC3 GS-0213 Cc1cccc(c1)C2C[C@H]([C@H]([C@@H]2N)O)O GS-0214 c1cnccc1C2C[C@H]([C@H]([C@@H]2N)O)O GS-0215 C1CCC(CC1)C2C[C@H]([C@H]([C@@H]2N)O)O GS-0216 Cc1ccc(cc1)C2C[C@H]([C@H]([C@@H]2N)O)O GS-0217 c1ccc(cc1)c2cc(no2)C[C@@H]3CC[C@@H]([C@H](O3)CN)O GS-0218 CNC(=O)[C@@H](c1ccccc1F)N2CCC[C@H]2C(=O)O GS-0219 CNC(=O)[C@@H](C1CCCCC1)N2CCC[C@H]2C(=O)O GS-0220 CNC(=O)[C@@H](Cc1ccccc1)N2CCC[C@H]2C(=O)O GS-0221 CN[C@H]1[C@H](O[C@H]([C@H]1O)CO)CN GS-0222 c1cc(cnc1)c2c[nH]c(n2)[C@@H]3COCCN3 GS-0223 COC(=O)c1coc(n1)[C@H](CO)NCc2ccccc2 GS-0224 COC(=O)c1coc(n1)[C@H](CO)NC2CCOCC2 GS-0225 COC(=O)c1coc(n1)[C@H](CO)NC(=O)c2ccccc2 GS-0226 CC(C)(C)C(=O)N[C@@H](CO)c1nc(co1)C(=O)OC GS-0227 c1c(nc(o1)[C@H](CO)N)C(=O)N2CCOCC2 GS-0228 CNC(=O)[C@@H](c1ccc(cc1)Cl)N2CCC[C@H]2C(=O)O GS-0229 Cc1ccc(cc1)S(=O)(=O)N[C@@H]2CO[C@@H]([C@H]2O)CO GS-0230 c1cc(ccc1F)S(=O)(=O)N[C@@H]2CO[C@@H]([C@H]2O)CO GS-0231 c1cc(cc(c1)F)C(=O)N[C@@H]2CO[C@@H]([C@H]2O)CO GS-0232 c1cnccc1C(=O)N[C@@H]2CO[C@@H]([C@H]2O)CO GS-0233 COCC(=O)N[C@@H]1CO[C@@H]([C@H]1O)CO GS-0234 CC(=O)NC[C@@H]1[C@H]([C@@H](CO1)N)O GS-0235 CC(C)NC(=O)NC[C@@H]1[C@H]([C@@H](CO1)N)O GS-0236 COCC(=O)NC[C@@H]1[C@H]([C@@H](CO1)N)O GS-0237 Cc1ccc(cc1)S(=O)(=O)NC[C@@H]2[C@H]([C@@H](CO2)N)O GS-0238 C1CC1C(=O)NC[C@@H]2[C@H]([C@@H](CO2)N)O GS-0239 CC(C)(C)CC(=O)NC[C@@H]1[C@H]([C@@H](CO1)N)O GS-0240 c1cnccc1C(=O)NC[C@@H]2[C@H]([C@@H](CO2)N)O GS-0241 c1cc(sc1)C(=O)NC[C@@H]2[C@H]([C@@H](CO2)N)O GS-0242 c1cc(sc1)C(=O)N[C@@H]2CO[C@@H]([C@H]2O)CO GS-0243 c1cc(ccc1C(=O)NC[C@@H]2[C@H]([C@@H](CO2)N)O)F GS-0244 c1ccc(cc1)S(=O)(=O)NC[C@@H]2[C@H]([C@@H](CO2)N)O GS-0245 c1cc(cnc1)C2C[C@H]([C@H]([C@@H]2N)O)O GS-0246 COc1ccc(cc1)C2C[C@H]([C@H]([C@@H]2N)O)O GS-0247 CN(C)[C@@H](CO)c1nc(co1)C(=O)OC GS-0248 C=C[C@H]1C[N@@]2CC[C@H]1C[C@@H]2CNC(=O)NC3CCCCC3 GS-0249 CC(=O)Nc1ccc(cc1)CN2C[C@@H]3[C@H](C2)OCC(=O)N3 GS-0250 C1CCC(CC1)N2C[C@@H]3[C@H](C2)OCC(=O)N3 GS-0251 c1ccnc(c1)c2cc(no2)C[C@H]3CNCC[C@H]3CC(=O)O GS-0252 C#CCNC(=O)C[C@H]1[C@@H]([C@@H]([C@H](O1)CN)O)O GS-0253 C1CC1NC(=O)C[C@H]2[C@@H]([C@@H]([C@H](O2)CN)O)O GS-0254 C1COCCN1C(=O)C[C@H]2[C@@H]([C@@H]([C@H](O2)CN)O)O GS-0255 CC(C)NC(=O)C[C@H]1[C@@H]([C@@H]([C@H](O1)CN)O)O GS-0256 c1ccc(cc1)CNC(=O)c2coc(n2)[C@H](CO)N GS-0257 c1ccc(cc1)NC(=O)NC[C@@H]2[C@@H]([C@H](CO2)O)N GS-0258 COCCOC[C@@]1(C[C@H]([C@H](C1)O)O)CN GS-0259 c1cc(ccc1C(F)(F)F)OC[C@]2(C[C@H]([C@H](C2)O)O)CN GS-0260 C1[C@H]([C@H](C[C@@]1(CN)CO)O)O GS-0261 COC[C@]1(C[C@H]([C@H](C1)O)O)CN GS-0262 CC(C)CCOC[C@@]1(C[C@H]([C@H](C1)O)O)CN GS-0263 Cc1cccc(n1)OC[C@@]2(C[C@H]([C@H](C2)O)O)CN GS-0264 C1[C@H]([C@H](C[C@]1(CN)CO)O)O GS-0265 Cc1cccc(n1)O[C@@H]2CNCCOC2 GS-0266 c1cc(ncc1C(F)(F)F)OC[C@@]2(C[C@H]([C@H](C2)O)O)CN GS-0267 c1ccc2c(c1)nc(o2)N3CCOC[C@@H](C3)O GS-0268 CS(=O)(=O)c1ccc(cc1)O[C@@H]2CNCCOC2 GS-0269 c1ccc(cc1)CN2CCN3[C@H](C2)COC3=O GS-0270 CC(C)NC(=O)N1CCN2[C@H](C1)COC2=O GS-0271 c1cc(cnc1)CN2CCN3[C@H](C2)COC3=O GS-0272 CC(=O)N1CCC(CC1)N2CCN3[C@H](C2)COC3=O GS-0273 CC(C)N1CCN2[C@H](C1)COC2=O GS-0274 C1COCCC1N2CCN3[C@H](C2)COC3=O GS-0275 COCC(=O)N1CCN2[C@H](C1)COC2=O GS-0276 C1COC[C@@H](CN1)O GS-0277 c1cc(ccc1C(F)(F)F)O[C@@H]2CNCCOC2 GS-0278 COc1ccc(cc1)O[C@@H]2CNCCOC2 GS-0279 c1ccc(cc1)C(=O)N2CCN3[C@H](C2)COC3=O GS-0280 c1ccc(cc1)O[C@@H]2CNCCOC2 GS-0281 CC(C)NC(=O)NC[C@H]1COCc2n1c3ccccc3n2 GS-0282 CS(=O)(=O)NCCc1ccccc1 GS-0400 c1cc(ncc1C#N)N2CCOCC2 GS-0401 CN(C)C(=O)CCN1c2ccccc2OCC1=O GS-0402 CC(=O)N1CCN(CC1)c2ccccc2 GS-0403 CNC(=O)c1c(ocn1)c2ccccc2 GS-0405 CN(C)C(=O)c1c(ocn1)c2ccccc2 GS-0406 CC(=O)NCCc1ccccc1 GS-0407 CC(=O)N1CCC(CC1)C#N GS-0408 CN(CCO)c1ccc(cn1)C#N GS-0409 CC(=O)NCc1ccc(cc1)OC GS-0410 CC(=O)NCc1ccc(cc1)Cl GS-0411 COc1ccc(cc1)CNS(=O)(=O)C GS-0412 CC(=O)NCc1cccc(c1)C(F)(F)F GS-0413 C[C@@H](c1ccccc1)NC(=O)C GS-0414 CC(=O)NCc1cccc(c1)Cl GS-0415 CC(=O)NCc1ccccc1Cl GS-0416 CCOC(=O)c1c2c(sc1NC(=O)C)CCC(C2)(C)C GS-0417 CS(=O)(=O)NCc1ccccc1Cl GS-0419 Cc1cccnc1CNC(=O)C GS-0420 CC(=O)NC1CCc2c1cccc2 GS-0421 CC(=O)NC1CCN(CC1)Cc2ccccc2 GS-0422 CC(=O)NCc1ccc(cc1)C#N GS-0423 CC(=O)NC1CCN(CC1)C(=O)Cc2ccccc2 GS-0424 CS(=O)(=O)NC1Cc2ccccc2C1 GS-0426 CS(=O)(=O)NC1CCc2c1cccc2 GS-0427 CS(=O)(=O)NC1CCN(CC1)Cc2ccccc2 GS-0428 CS(=O)(=O)NCc1ccc(cc1)C#N GS-0429 CNC(=O)NC1CCN(CC1)Cc2ccccc2 GS-0430 CNC(=O)NCc1ccccc1OC GS-0431 CNC(=O)C1(CC1)c2ccccc2F GS-0432 CNC(=O)C1(CC1)c2ccccc2 GS-0433 CNC(=O)C1CCC(CC1)(F)F GS-0434 CN(C)C(=O)Cc1ccc(cc1)C#N GS-0435 CNC(=O)Cc1ccc(cc1)C#N GS-0436 Cc1ccc(o1)c2cc(c3cc(ccc3n2)F)C(=O)N(C)C GS-0437 CNC(=O)c1ccc2ccccc2n1 GS-0438 CNC(=O)c1c(nccn1)N GS-0439 CNC(=O)c1cc2ccccc2nc1 GS-0440 CN(C)C(=O)c1ccc(o1)c2ccccc2 GS-0441 CNC(=O)c1ccc(o1)c2ccccc2 GS-0442 Cc1c(cn(n1)c2ccccc2)C(=O)NC GS-0444 CC(C)(C)n1cc(c(n1)c2cccnc2)C(=O)NC GS-0445 Cn1c2ccccc2c(n1)C(=O)N(C)C GS-0446 CNC(=O)c1c2ccccc2n(n1)C GS-0447 CC(=O)N1CCN(CC1)c2ccc(cc2)F GS-0448 CC(=O)N1CCN(CC1)c2ccc(cn2)C#N GS-0449 CC(=O)N1CCN(CC1)c2ccc(cc2)OC GS-0450 CC(=O)N1CCc2cc(c(cc2C1)OC)OC GS-0451 CC(=O)N1CCN(CC1)S(=O)(=O)C GS-0452 CC(=O)N1CCN(CC1)c2ccccn2 GS-0453 CC(=O)N1CCN(CC1)c2ccncc2 GS-0454 CC(=O)N1CCC(CC1)N2CCOCC2 GS-0455 CC(=O)NCc1ccc(cc1OC)OC GS-0456 Cc1ccc(cc1)CNC(=O)C GS-0457 CC(=O)N[C@H]1CC2CCC1C2 GS-0458 CS(=O)(=O)NCC1CC(=O)N(C1)C2CCCC2 GS-0459 CS(=O)(=O)N[C@H]1CC2CCC1C2 GS-0460 CNC(=O)N1CCC(CC1)N2CCOCC2 GS-0461 CS(=O)(=O)N1CCN(CC1)CC2CCCO2 GS-0462 CS(=O)(=O)N(Cc1ccccn1)Cc2ccccn2 GS-0463 CS(=O)(=O)N1CCN(CC1)Cc2ccccc2 GS-0464 CS(=O)(=O)N1CCC(CC1)N2CCCCC2 GS-0465 CC1CN(CCN1C)S(=O)(=O)C GS-0466 COc1ccccc1N2CCN(CC2)S(=O)(=O)C GS-0467 CS(=O)(=O)N1CCN(CC1)c2ccccn2 GS-0468 CS(=O)(=O)N1CCN(CC1)CCc2ccccc2 GS-0469 Cn1cc(c(n1)c2cccs2)C(=O)N(C)C GS-0470 CNC(=O)C1CC(=O)N(C1)Cc2ccccc2 GS-0471 CN(C)C(=O)C1CCCN(C1)S(=O)(=O)C2CC2 GS-0472 CNC(=O)C1CCCN(C1)S(=O)(=O)C2CC2 GS-0473 CC(=O)N1CCC(CC1)c2c3cc(ccc3on2)F GS-0474 CNC(=O)NCc1ccccc1F GS-0475 CNC(=O)NCc1ccc2c(c1)OCO2 GS-0476 c1cnc(nc1)NC2CCOCC2 GS-0477 c1cnc(nc1)N2CCC(C2)CCO GS-0478 c1cnc(nc1)N2CCS(=O)(=O)CC2 GS-0479 c1[nH]c2c(n1)nc(nc2N3CCOCC3)N GS-0480 CN(C)C(=O)C1CCN(CC1)c2ccc(cn2)C#N GS-0481 CN1CCN(CC1=O)c2ccc(cn2)C#N GS-0482 CN(C)CC1CCN(CC1)c2ccnc(n2)N GS-0483 CN(C)C(=O)C1CCN(CC1)c2ccnc(n2)N GS-0484 c1cnc(nc1N)N2CCOCC2 GS-0485 CN(C)CC1CCN(CC1)c2nccc(n2)N GS-0486 c1cnccc1CNC(=O)c2cocn2 GS-0487 CS(=O)(=O)N1CCOCC1 GS-0488 CNC(=O)NCc1ccncc1 GS-0489 CNC(=O)NCc1ccc(cc1)C(F)(F)F GS-0490 CNC(=O)NCc1ccc(cc1)OC GS-0491 CC(=O)NC1Cc2ccccc2C1 GS-0492 CNC(=O)NCc1ccccc1S(=O)(=O)C GS-0493 CNC(=O)NCc1cccc(c1)Cl GS-0494 CNC(=O)NC1CCc2c1cccc2 GS-0495 CNC(=O)NCc1c(cccc1F)F GS-0496 CNC(=O)NC1Cc2ccccc2C1 GS-0497 CNC(=O)NC1CCN(CC1)c2ncccn2 GS-0498 CNC(=O)NCCN1CCc2ccccc2C1 GS-0499 CNC(=O)NCc1cccnc1 GS-0500 CNC(=O)NCc1ccc(c(c1)F)F GS-0501 CNC(=O)NCc1ccc(nc1)OC GS-0502 CNC(=O)NCCc1ccccn1 GS-0503 CNC(=O)NCCc1ccncc1 GS-0504 CNC(=O)NCCn1cccn1 GS-0505 CNC(=O)NCc1ccccn1 GS-0506 CNC(=O)NCCc1cc[nH]n1 GS-0507 CNC(=O)NCC(c1ccccc1)O GS-0508 CNC(=O)N[C@H]1CC[C@@H](CC1)O GS-0509 CC(=O)N1CCC(CC1)NC(=O)NC GS-0510 CCOC(=O)N1CCC(CC1)NC(=O)NC GS-0511 CNC(=O)NCCN1CCC(CC1)(F)F GS-0512 CNC(=O)NC1CCC(CC1)(F)F GS-0513 CNC(=O)NCC1CCN(CC1)C GS-0514 CNC(=O)NCCN1CCCCC1 GS-0515 CCN1CCCC1CNC(=O)NC GS-0516 CNC(=O)NCCC1CCCN1C GS-0517 CNC(=O)NCCN1CCCC1 GS-0518 CNC(=O)NCC(=O)N1CCOCC1 GS-0519 Cc1nc(cs1)CCNC(=O)NC GS-0520 CNC(=O)NCc1ccc(cc1)S(=O)(=O)C GS-0521 CNC(=O)NCc1ccc2c(c1)cc[nH]2 GS-0522 CNC(=O)NCc1ccc(cc1)C#N GS-0523 CNC(=O)NCCc1cccnc1 GS-0524 CNC(=O)N1Cc2ccccc2C1 GS-0525 CN(C)C(=O)N1Cc2ccccc2C1 GS-0526 CNC(=O)NCCN1CCS(=O)(=O)CC1 GS-0527 CS(=O)(=O)N1CCCC1 GS-0528 CS(=O)(=O)N1CCS(=O)(=O)CC1 GS-0529 Cc1nc(on1)CCNS(=O)(=O)C GS-0530 CS(=O)(=O)NC1CCOCC1 GS-0531 CS(=O)(=O)NCc1ccccn1 GS-0532 Cc1nc(cs1)CCNS(=O)(=O)C GS-0533 CS(=O)(=O)NCCN1CCC(CC1)(F)F GS-0534 CN(C)C(=O)CN(C)S(=O)(=O)C GS-0535 CN(C)C(=O)C1CCN(CC1)S(=O)(=O)C GS-0536 CS(=O)(=O)N1CCC(C1)CCO GS-0537 CC1COCCN1S(=O)(=O)C GS-0538 CN(CCO)S(=O)(=O)C GS-0539 CS(=O)(=O)N1CCCCC1 GS-0540 CS(=O)(=O)N1CCC(CC1)C#N GS-0541 CN(C1CCS(=O)(=O)C1)S(=O)(=O)C GS-0542 CN(C)C(=O)CNS(=O)(=O)C GS-0543 CC(=O)N1CCS(=O)(=O)CC1 GS-0544 Cc1nc(on1)CCNC(=O)C GS-0545 CC(=O)NCC1(CCCC1)CO GS-0546 CC(=O)NCC(=O)N1CCOCC1 GS-0547 CC(=O)NC1CCOCC1 GS-0548 CC(=O)NCc1ccccc1 GS-0549 Cc1nc(cs1)CCNC(=O)C GS-0550 CC(=O)NC1CCN(CC1)c2ncccn2 GS-0551 CC(=O)NCCN1CCC(CC1)(F)F GS-0552 CC(=O)NCCS(=O)(=O)N1CCOCC1 GS-0553 CC(=O)N1CCC(CC1)C(=O)N(C)C GS-0554 CC(=O)N(C)C1CCS(=O)(=O)C1 GS-0555 CC(=O)N1CCCC(C1)OC GS-0556 CC(=O)N1CCC2(CCCN(C2)C)CC1 GS-0557 COc1ccc(cc1)Cn2cc(nc(c2=O)Cl)Cl GS-0600 c1c(cnc(c1N)C(=O)N)Br GS-0601 COc1ccc(cc1)Cn2c3cc(ccc3nc(c2=O)Cl)Cl GS-0602 c1c(cnc(c1[N+](=O)[O-])C(=O)N)Br GS-0603 c1cc2c(cc1I)c(nc(n2)Cl)N GS-0604 Cc1cccc2c1nc(nc2Cl)Cl GS-0605 C1c2c([nH]c(=O)[nH]c2=O)C(=O)O1 GS-0606 c1cc2c(c(=O)[nH]c(=O)[nH]2)nc1 GS-0607 c1cc2c(cc1Cl)c(nc(n2)Cl)Cl GS-0609 c1cc2c(c(c1)F)c(nc(n2)Cl)Cl GS-0610 Cc1csc2c1[nH]c(=O)[nH]c2=O GS-0611 c1cc2c([nH]c(=O)[nH]c2=O)nc1 GS-0612 c1cc(ccc1OC2CCN(CC2)C3CCC3)Br GS-0613 c1cc2c(cc1F)c(=O)[nH]c(=O)[nH]2 GS-0614 CCOC(=O)C1=C(CCCC1)N GS-0615 C1CCc2c(c(nc(n2)Cl)Cl)C1 GS-0616 CCOC(=O)c1c(c2c([nH]c1=O)CCCC2)O GS-0617 c1c(c2c(nc1Cl)CCCC2=O)Cl GS-0618 c1cnc(c2c1CCCC2)O GS-0619 CC1(Cc2c(c(cc(n2)Cl)Cl)C(=O)C1)C GS-0620 Cc1cc(cc2c1[nH]c(=O)[nH]c2=O)Cl GS-0621 C1CC1CNS(=O)(=O)CCN.Cl GS-0622 CS(=O)(=O)OCCCc1ccc(cc1)Cl GS-0623 CC1(C(=C(CO1)C(=O)OC)N)C GS-0624 COc1ccc(cc1)CNCC#N.Br GS-0626 COc1ccc(cc1)CNCC#N.Cl GS-0627 CCCS(=O)(=O)NCC1CCC1.Cl GS-0628 c1cc2nc(cc(=O)n2cc1Br)O GS-0629 CSc1nc2ccc(cc2c(n1)O)Cl GS-0630 c1ccc(cc1)CN2CCC(CC2)Br GS-0631 COc1c(nc(nc1O)O)O GS-0632 c1cc(c2c(c1)nc(nc2Cl)Cl)C(F)(F)F GS-0633 C1c2c(nc(nc2Cl)Cl)C(=O)O1 GS-0634 C1Cc2c(c(nc(n2)Cl)Cl)SC1 GS-0635 c1ccn2c(c1)nc(cc2=O)O GS-0636 c1cc2c(c(ncn2)O)nc1 GS-0637 CC1(Cc2c(ccc(=O)[nH]2)C(=O)C1)C GS-0638 CC1(Cc2c(c(n[nH]2)Nc3ccccc3)C(=O)C1)C GS-0639 CCOC(=O)c1c2c([nH]n1)CNCC2.Cl GS-0641 c1cc2c(c(nc(n2)Cl)Cl)nc1 GS-0642 c1ccnc(c1)CNS(=O)(=O)CCN.Cl GS-0643 CCOC(=O)C1=C(C(OC1=O)(C)C)N GS-0644 CCOC(=O)c1c2c([nH]n1)CN(CC2)C(=O)OC(C)(C)C GS-0646 CCOC(=O)c1c2c([nH]n1)COCC2 GS-0647 c1ccc(cc1)c2c(=O)[nH]c3ccccc3n2 GS-0648 CC(C)(C)OC(=O)N1CCc2c([nH]nc2C(=O)O)C1 GS-0650 c1ccc(cc1)Nc2c3c([nH]n2)CCCC3=O GS-0651 c1ccc(cc1)NS(=O)(=O)CCN GS-0652 CC1(C(=C(C(=O)O1)C(=O)O)N)C GS-0653 c1ccc2c(c1)c3ccc(cc3[nH]2)Cl GS-0700 c1cc(c(cc1N)N)Br GS-0702 c1cnc(nc1N)CCl GS-0703 c1ccc(cc1)S(=O)(=O)n2c3cc(ccc3cc2C4(C=CC(=O)C=C4)O)F GS-1301 CCOC(=O)Cc1ccc(cc1)F GS-4515 Cc1c(nnn1Cc2ccccc2)C(=O)Cl H-20003 Cc1ccc2c(c1)cc(c(=O)[nH]2)C=O H-20019 CCOC(=O)c1c(n(nn1)Cc2ccc(cc2)Br)C H-20029 CCOC(=O)C1Cc2cc(ccc2CN1C(=O)OC)O H-20039 Cc1c(nnn1Cc2ccc(cc2)Br)C(=O)N H-20044 Cc1c(nnn1Cc2ccccc2)C(=O)N H-20045 Cc1c(nnn1Cc2ccc(cc2)Br)C(=O)Cl H-20047 c1cc(ccc1Cn2c3c(c(ncn3)O)nn2)Br H-20077 c1ccc2c(c1)cc(c(=O)[nH]2)C=O H-2008 c1ccc2c(c1)cc(c(=O)[nH]2)C#N H-2011 c1ccc2c(c1)cc(c(=O)[nH]2)/C=N/O H-2012 c1cc(ccc1Cn2c(c(nn2)C(=O)N)N)Cl H-20130 c1ccnc(c1)Cn2c(c(nn2)C(=O)N)N H-20135 c1ccc2c(c1)cc(c(=O)[nH]2)C(=O)O H-2016 CCOC(=O)c1c(n(nn1)Cc2ccc(cc2)C)C H-20170 Cc1ccc(cc1)Cn2c(c(nn2)C(=O)O)C H-20171 Cc1c(nnn1Cc2ccc(cc2)Br)C(=O)N3CCOCC3 H-20172 Cc1c(nnn1Cc2ccc(cc2)Br)C(=O)NC H-20173 Cc1c(nnn1Cc2ccc(cc2)Br)C(C)O H-20195 c1cc(ccc1Cn2c3c(c(ncn3)O)nn2)Cl H-20212 Cc1ccc(cc1)Cn2c3c(c(ncn3)O)nn2 H-20213 Cc1c(nnn1Cc2ccc(cc2)Cl)C(=O)O H-20228 CCOC(=O)c1c(n(nn1)Cc2ccc(cc2)Cl)C H-20231 Cc1c(nnn1Cc2ccc(cc2)Cl)C(=O)C H-20234 CCOC(=O)C1Cc2cc(ccc2CN1)O.Cl H-20242 c1cc2c(cc1O)CC(NC2)C(=O)O H-20243 C[C@H](c1cc(cc(c1)C(F)(F)F)C(F)(F)F)NC.C(C(C(=O)O)O)C(=O)O H-20244 CC(C)OC(=O)N[C@H]1Cc2c3cc(ccc3[nH]c2C1)Br H-20253 CCOC(=O)c1c(nc(s1)c2ccc(cc2F)C(F)(F)F)C H-20255 COc1cnc(nc1Cl)c2cc(ccc2F)Cl H-20257 Cc1c(sc(n1)c2ccc(cc2F)C(F)(F)F)C(=O)O H-20260 CC1(OCC(CO1)(C=C)O)C H-20267 C1CC(CCC1C(=O)O)(F)F H-20299 c1ccc2c(c1)cc(c(=O)[nH]2)CO H-2032 Cc1ccc2c(c1)cc(c(=O)[nH]2)CO H-21008 COc1ccc2c(c1)cc(c(n2)Cl)/C=N/O H-28012 Cc1c(nnn1Cc2ccc(cc2)Br)C(=O)C H-31006 CCOC(=O)c1c(n(nn1)Cc2ccc(cc2)F)C H-32003 Cc1c(nnn1Cc2ccc(cc2)F)C(=O)O H-32004 CCOC(=O)c1c(n(nn1)Cc2ccccc2)C H-33001 Cc1c(nnn1Cc2ccccc2)C(=O)C H-33006 c1ccc(cc1)Cn2c(c(nn2)c3ccccc3)N H-33007 c1ccc(cc1)c2c(n(nn2)Cc3ccc(cc3)Br)N H-33008 c1ccc(cc1)Cn2c(c(nn2)C(=O)N)N H-34005 c1cc(ccc1Cn2c(c(nn2)C(=O)N)N)Br H-34006 c1ccc(cc1)Cn2c3c(c(ncn3)O)nn2 H-38001 CCOC(=O)c1cn2c(n1)sc(n2)C(F)(F)F HA-0202 Cc1cn(c(=O)[nH]c1=O)Cc2nnc(o2)CC3CC3 HA-0205 CCOC(=O)c1cn2c(n1)scn2 HA-0207 CC(C)c1nc(sn1)N HA-0210 CCOC(=O)c1cn2c(n1)sc(n2)C3CC3 HA-0212 c1cc(nc(c1)Br)c2csc(n2)N HA-0213 c1ccc(cc1)c2nc(sn2)N HA-0214 Cc1nc(sn1)N HA-0217 CCOC(=O)C1=C(N(C(=O)NC1c2cccc(c2)Cl)C)C HA-0231 CCOC(=O)C1=C(N(C(=O)NC1c2ccccc2F)C)C HA-0232 CCOC(=O)C1=C(N(C(=O)NC1c2ccccc2)C)C HA-0233 CCOC(=O)C1=C(N(C(=O)NC1c2ccc(cc2)C(C)C)C)C HA-0234 CCOC(=O)C1=C(N(C(=O)NC1c2ccc(cc2)C(C)(C)C)C)C HA-0235 CCOC(=O)C1=C(N(C(=O)NC1c2ccc(cc2)Cl)C)C HA-0236 CCOC(=O)C1=C(N(C(=O)NC1c2cccc(c2)F)C)C HA-0237 CCOC(=O)C1=C(N(C(=O)NC1c2ccc(cc2)OC)C)C HA-0238 CCOC(=O)C1=C(N(C(=O)NC1c2ccc(cc2)C)C)C HA-0240 CCOC(=O)C1=C(N(C(=O)NC1c2ccccc2OC)C)C HA-0241 CCOC(=O)C1=C(N(C(=O)NC1c2cccc(c2)C)C)C HA-0242 CCOC(=O)C1=C(N(C(=O)NC1c2ccccc2Cl)C)C HA-0243 CCOC(=O)C1=C(N(C(=O)NC1c2ccccc2C)C)C HA-0244 CCOC(=O)C1=C(N(C(=O)NC1c2cccc(c2)OC)C)C HA-0245 CCOC(=O)C1=C(N(C(=O)NC1c2cccnc2)C)C HA-0247 CCOC(=O)c1cn2c(n1)sc(n2)C(C)(C)C HA-0260 c1ccc2c(c1)[nH]/c(=N/O)/c(=O)o2 HA-0700 CNc1ccc(cn1)C(F)(F)F HA-0702 Cc1ccc2c(c1)[nH]/c(=N/O)/c(=O)o2 HA-0703 c1c2c(cc(c1Cl)Cl)[nH]c(=O)/c(=N\O)/[nH]2 HA-0704 c1cc2c(cc1Cl)[nH]/c(=N/O)/c(=O)o2 HA-0705 c1ccc2c(c1)[nH]/c(=N/O)/c(=O)s2 HA-0706 COc1ccc2c(c1)c(c[nH]2)C(=S)N3CCCCC3 HA-0713 c1cc(ccc1C(=O)CSC#N)Br HA-0720 COc1ccc(cc1)C(=O)CSC#N HA-0721 c1cc(ccc1C(=O)CSC#N)Cl HA-0726 CS(=O)(=O)c1ccc(cc1)C(=O)CSC#N HA-0727 c1cc(c(cc1C(=S)N)F)C(F)(F)F HA-0801 CC(c1ccnn1C(=O)c2ccc(cc2)Cl)Sc3c(cccn3)C(F)(F)F HA-0802 CC(c1ccnn1C(=O)Cc2ccccc2)Sc3c(cccn3)C(F)(F)F HA-0803 CC(c1ccnn1C(=O)c2ccccc2Cl)Sc3c(cccn3)C(F)(F)F HA-0804 c1cc2nc(c(n2cc1Cl)Br)C(=O)NCCO HA-0805 CN(C(=O)c1ccc(cc1)C(F)(F)F)OC HA-0808 c1ccc(c(c1)OC(=O)c2cc(cc(n2)C(=O)Oc3ccccc3Cl)C(F)(F)F)Cl HA-0809 COC(=O)c1ccc(cc1)OCc2ccc3c(c2)nsn3 HA-0810 c1cc(ccc1C=O)OCc2ccc3c(c2)nsn3 HA-0811 CCOC(=O)C1CCCN(C1)CCCOc2ccc(cc2)OCc3ccccc3 HA-0812 CCOC(=O)C1CCN(CC1)CCCOc2ccc(cc2)OCc3ccccc3 HA-0813 CCOC(=O)C1CCN(CC1)Cc2ccc3c(c2)nsn3 HA-0815 c1cc(cc(c1)OC(=O)c2cc(cc(n2)C(=O)Oc3cccc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F HA-0817 c1cc(ccc1C(=O)O)OCc2ccc3c(c2)nsn3 HA-0818 COC(=O)c1ccc2c(c1)NC(=O)CO2 HA-0820 CC(C)(C)c1ccc(cc1)C(=O)N(C)OC HA-0821 c1cc(c(cc1NS(=O)(=O)CCCCl)Cl)Cl HA-0822 Cc1cc(cc(c1N)C(=O)OC)Cl HA-0823 c1ccnc(c1)COC(=O)c2cc(cc(n2)C(=O)OCc3ccccn3)C(F)(F)F HA-0825 Cn1cccc(c1=S)C(=O)OC HA-0827 COCCOC(=O)c1cc(cc(n1)C(=O)OCCOC)C(F)(F)F HA-0828 CCOC(=O)c1c(nc(s1)c2ccc(c(c2)F)C(F)(F)F)C HA-0829 COC(=O)c1cccc(c1)OCCOc2ccc(cc2)OCc3ccccc3 HA-0830 CN(C(=O)c1c(cc(cc1F)F)F)OC HA-0833 Cc1c(sc(n1)c2ccc(c(c2)F)C(F)(F)F)CO HA-0834 c1cnccc1COC(=O)c2cc(cc(n2)C(=O)OCc3ccncc3)C(F)(F)F HA-0835 CN(C(=O)c1cccs1)OC HA-0837 COC(=O)c1ccc(cc1)OCCOc2ccc(cc2)OCc3ccccc3 HA-0838 c1cc2c(cc1CN3CCN(CC3)CCO)nsn2 HA-0839 Cc1c(sc(n1)c2ccc(c(c2)F)C(F)(F)F)CCl HA-0841 CN(C(=O)c1ccc(cc1)C#N)OC HA-0842 c1cc2c(cc1C=O)nsn2 HA-0843 CCOC(=O)C1CCCc2c1nc(s2)c3ccc(cc3)Cl HA-0844 c1cc(c(cc1N2CCCS2(=O)=O)Cl)Cl HA-0845 c1ccc(cc1)CN2CCN(CC2)CCOc3ccc(cc3)C(=O)O HA-0847 CSc1ccc(cc1)NS(=O)(=O)CCCCl HA-0850 c1ccc(cc1)CN2CCN(CC2)CCOc3ccc(cc3)C(=O)NN HA-0852 CCOC(=O)c1cc(cc(n1)C(=O)Nc2ccccc2)C(F)(F)F HA-0854 CCOC(=O)c1cc(cc(n1)C(=O)NCc2ccccn2)C(F)(F)F HA-0858 c1c(cnc(c1Br)N)C(=O)O HA-0859 COc1cc(cc(n1)Cl)C(=O)OC HA-0921 COc1ccc2c(c1)sc(n2)Cl HA-0923 COc1ccc2c(c1)sc(n2)NN HA-0925 CCNC(=O)N(Cc1c(cc(cn1)C(F)(F)F)Cl)NC(=O)OC(C)(C)C HB-0012 CC(C)(C)OC(=O)NN(Cc1c(cc(cn1)C(F)(F)F)Cl)C(=O)Nc2ccc(cc2)Cl HB-0025 c1cc(ccc1NC(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)Cl HB-0026 c1cc(c(c(c1)Cl)C(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)Cl HB-0047 c1ccc(c(c1)C(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)C(F)(F)F HB-0048 c1cc(cc(c1)NC(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)C(F)(F)F HB-0061 c1ccc(c(c1)C(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)Cl HB-0062 c1cc(ccc1S(=O)(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)Cl HB-0074 c1ccc(c(c1)S(=O)(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)Cl HB-0075 c1cc(cc(c1)S(=O)(=O)N2CC(CC(C2)C(F)(F)F)C(F)(F)F)C(F)(F)F HB-0076 CN(C)C(=O)[C@H](c1ccccc1)N.Cl HB-0078 CS(=O)(=O)/C(=C\c1ccc(cc1)N2CCC(CC2)C(F)(F)F)/C#N HB-0703 c1cc(ccc1CNC(=O)c2ccc(cc2Cl)N3CCC(CC3)C(F)(F)F)Cl HB-0707 CC(=O)c1ccc(c(c1)[N+](=O)[O-])O HB-0708 c1cc(ccc1C(F)(F)F)N2CCN(CC2)C(=O)c3ccc(cc3Cl)N4CCC(CC4)C(F)(F)F HB-0711 c1cc(ccc1C=C(C#N)C#N)N2CCC(CC2)C(F)(F)F HB-0715 c1ccc(cc1)CN2CCN(CC2)Cc3ccc(cc3)N4CCC(CC4)C(F)(F)F HB-0718 c1cc(ccc1CN2CCCCC2)N3CCC(CC3)C(F)(F)F HB-0719 c1cc(cc2c1cc([nH]2)C(=O)O)Br HB-0721 c1ccc(c(c1)NC(=O)c2ccc(cc2Cl)N3CCC(CC3)C(F)(F)F)Cl HB-0723 c1cc(ccc1/C=N\NC(=O)c2ccc(cc2)Cl)OCCN3CCC(CC3)C(F)(F)F HB-0728 CC(C)(C)OC(=O)n1cc(cc1C(=O)OC)Br HB-0733 c1c(c[nH]c1C(=O)O)Br HB-0734 CC(=O)c1cnc(nc1O)S HB-0803 c1c(cnc(c1Cl)Cn2cc(cn2)[N+](=O)[O-])C(F)(F)F HB-0806 CCOC(=O)Cn1c(=O)c(c(cn1)N2CCN(CC2)C(=O)OCc3ccccc3)Cl HB-0807 CC(C)Nc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl HB-5000 C=CCNc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl HB-5001 CCCCCCNc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl HB-5002 c1ccc(c(c1)NCc2ccc(cc2)c3ccc(cn3)C(F)(F)F)Cl HB-5003 c1cc(ccc1CNc2ccc(cc2)Cl)c3ccc(cn3)C(F)(F)F HB-5006 c1cc(c(c(c1)F)NCc2ccc(cc2)c3ccc(cn3)C(F)(F)F)F HB-5007 c1c(cnc(c1Cl)c2csc(n2)NC3CC3)C(F)(F)F HB-5008 c1ccc(cc1)CNc2nc(cs2)c3c(cc(cn3)C(F)(F)F)Cl HB-5009 COCCNc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl HB-5010 CN(C)CCNc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl HB-5012 C#CCNc1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl HB-5015 CN(C)c1nc(cs1)c2c(cc(cn2)C(F)(F)F)Cl HB-5016 c1c(cnc(c1Cl)c2csc(n2)N3CCCCC3)C(F)(F)F HB-5017 c1c(cnc(c1Cl)c2csc(n2)N3CCOCC3)C(F)(F)F HB-5018 c1c(cnc(c1Cl)c2csc(n2)NCC(F)(F)F)C(F)(F)F HB-5021 CN1CCN(CC1)Cc2cccc(c2)N HB-5027 CCOC(=O)c1c(nc(nn1)c2c(cc(cn2)C(F)(F)F)Cl)O HB-5033 c1cc(c(cc1n2cncn2)Cl)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl HC-0024 c1ccc(cc1)c2ccc(cc2)c3cc([nH]n3)N HC-0201 c1ccc(cc1)c2ccc(cc2)c3cc(on3)N HC-0202 CCOC(=O)c1c(cc([nH]1)c2ccccc2)N HC-0206 CCOC(=O)[C@H]1C[C@H](C(N1)c2ccco2)C(=O)OC(C)(C)C HC-0209 c1cc2c(cc1C(=O)CC#N)OCO2 HC-0214 c1cncc(c1C(=O)NN)N HC-0600 CC1(COC1)CI HC-0700 c1cc2c(cc1C(=O)O)OCC(=O)N2 HC-0701 CC(C)(C)OC(=O)N/N=C/c1ccc(cc1F)Br HC-0702 c1cc(c(cc1Cl)N2CCC(CC2)C(=O)O)[N+](=O)[O-] HC-0703 CN1c2ccc(cc2OCC1=O)C(=O)OC HC-0704 CC1C(=O)Nc2ccc(cc2O1)C(=O)O HC-0705 CC1C(=O)N(c2ccc(cc2O1)C(=O)OC)C HC-0707 C/C(=N\O)/c1cccnc1 HC-0709 C/C(=N\O)/c1ccncc1 HC-0710 c1cc(ncc1Cl)n2c(c(cn2)C#N)N HC-0711 c1cc(c(cc1Cl)N2CCOCC2)[N+](=O)[O-] HC-0714 COC(=O)Cc1cn2cc(cc(c2n1)I)C(F)(F)F HC-0715 CN1c2ccc(cc2OCC1=O)C(=O)O HC-0716 CC1C(=O)N(c2ccc(cc2O1)C(=O)O)C HC-0717 c1ccnc(c1)c2c(cc(c(=O)[nH]2)C#N)Br HC-0718 C1CC1c2c(c(c(c(n2)O)C#N)C(F)(F)F)Cl HC-0722 c1ccnc(c1)c2c(cc(c(=O)[nH]2)C#N)Cl HC-0725 c1cc(c(cc1Cl)N2CCCC2)[N+](=O)[O-] HC-0727 c1cc(c(cc1Cl)N2CCCCC2)[N+](=O)[O-] HC-0728 c1ccnc(c1)c2c(cc(c(=O)[nH]2)C#N)I HC-0731 CCOC(=O)c1cnc(s1)NC2CCCCO2 HC-0732 CCOC(=O)c1cnc(s1)NC(=O)OC(C)(C)C HC-0734 COc1ccc(cc1)n2c(=O)cc(c(n2)C(=O)O)O HC-0735 CCOC(=O)Cn1cc(nn1)C(=O)O HC-0736 c1cc(cnc1)/C(=N\C#N)/N HC-0737 CC(C)(C)OC(=O)N1CCN(CC1)c2cc(ccc2[N+](=O)[O-])Cl HC-0738 Cc1cc(c(c(n1)Cl)C#N)C(F)(F)F HC-0739 c1cnccc1/C(=N\C#N)/N HC-0741 c1cn2cc(cnc2n1)Br HC-0742 CC(C)(C)OC(=O)Nc1ccc2c(c1)cc(o2)CO HC-0743 c1ccnc(c1)c2c(cc(c(n2)Cl)C#N)Br HC-0744 CC(C)(CCC(=O)OC)C(=O)OC HC-0746 CC(C)(C)OC(=O)Nc1ncc(s1)C(=O)O HC-0747 CC1C(=O)Nc2cc(ccc2O1)C(=O)O HC-0749 COC(=O)c1cc(ccc1OCc2ccccc2)[N+](=O)[O-] HD-0002 CN(C(=O)c1ccc(c(c1)OCc2ccccc2)[N+](=O)[O-])OC HD-0004 CC(C)(C)n1c(=O)c(c(cn1)Br)Br HD-0005 c1ccc(cc1)COc2ccc(cc2C(=O)O)[N+](=O)[O-] HD-0007 CCOC(=O)c1cc(cnc1NCc2ccccc2)Br HD-0016 c1c(c(cc2c1c(c[nH]2)C=O)C(F)(F)F)C#N HD-0019 COC(=O)c1cc(ccc1OCc2ccccc2)[NH3+].[Cl-] HD-0021 c1c(cc(c(c1C(=O)O)O)Br)[N+](=O)[O-] HD-0025 CCOC(=O)c1cc(cnc1NCc2ccccc2)Cl HD-0026 c1ccc(cc1)COc2c(cc(nc2Cl)CO)I HD-0031 COC(=O)c1cc(c(c(c1)I)N)OCc2ccccc2 HD-0040 CCCC(CCO)O HD-0041 c1ccc(cc1)COc2c(cc(nc2Cl)C=O)I HD-0049 COC(=O)c1cc(c(c(c1)Br)N)OCc2ccccc2 HD-0055 CCOC(=O)c1c(c2cc(cnc2n(c1=O)Cc3ccccc3)Br)O HD-0073 CC(C)(C)OC(=O)n1cc(c2c1cc(c(c2)C#N)C(F)(F)F)C=O HD-0077 COC(=O)c1cc(ccc1O)C#C[Si](C)(C)C HD-0078 Cn1cc(c(c1)C(F)(F)F)C(=O)NNC(=S)Nc2ccc(cc2)Cl HD-0083 Cn1cc(c(c1)C(F)(F)F)C(=O)Nc2ccccc2Cl HD-0089 COC(=O)c1cc(c(c(c1)OCc2ccccc2)N)C#C[Si](C)(C)C HD-0092 COC(=O)c1cc2cc[nH]c2c(c1)OCc3ccccc3 HD-0094 CCOC(=O)c1c(c2cc(cnc2n(c1=O)Cc3ccccc3)Cl)O HD-0095 COc1ccc(c(c1)OCc2ccccc2)C=O HD-0097 c1cc(c(cc1c2nc(cs2)CCCN)F)C(F)(F)F HD-0205 c1c(cnc(c1C(F)(F)F)Cl)Cl HD-0213 c1cnc(c(c1Cl)C(F)(F)F)Cl HD-0214 c1c(c(nc(n1)Cl)Cl)CI HD-0230 CCOC(=O)C1C2CN(CC(N2C)CC1=O)C(=O)OC(C)(C)C HD-0231 CSc1nc(cc(n1)N2CCNCC2)C(F)(F)F HD-0233 COC(=O)c1c(c(=O)[nH]c(=O)[nH]1)C(F)(F)F HD-0237 CC1(CC(=O)C(C(=O)C1)Br)C HD-0700 C1CC(=O)C(C(=O)C1)Br HD-0701 C1CC(=O)C(C1=O)Br HD-0702 c1c(cnc2c1[nH]c(=O)[nH]2)Br HD-0706 c1c(c(=O)[nH]c(=O)[nH]1)CO HD-0707 c1cc2c(cc1Br)oc(=O)[nH]2 HD-0708 c1ccc(cc1)c2cc(c(nn2)Cl)Cl HD-0710 CC(c1cccc(n1)Br)O HD-0715 CNc1c2ccccc2nc(n1)C(F)(F)F HD-0716 CC(C)(C)OC(=O)NCCCl HD-0717 CCOC(=O)c1cnc(c(c1O)[N+](=O)[O-])O HD-0719 c1c(c(nc(n1)Cl)Cl)CCl HD-0720 Cc1cc(cc(c1N)C(=O)O)I HD-0722 CCOC(=O)C1CNc2cc(ccc2O1)[N+](=O)[O-] HD-0723 C1C[C@H]2[C@@H]1C(=O)NC2=O HD-0725 c1cc2c(cc1C(=O)O)oc(=O)[nH]2 HD-0726 c1c(c(c(nc1Cl)Cl)I)C(F)(F)F HD-0728 c1cnc(c(c1C(F)(F)F)I)Cl HD-0730 COc1c(c(ccn1)N)Br HD-0734 Cc1cc(cc(c1NC(=O)C(F)(F)F)C(=O)O)I HD-0735 CNc1ccc(cc1[N+](=O)[O-])C(=O)OC HD-0736 c1c(c(cnc1O)C(=O)O)O HD-0738 COC(=O)c1ccc(nc1N)Cl HD-0739 Cc1c(cc(c(n1)Cl)Br)C(=O)C HD-0740 CC(=O)c1cc(c(=O)[nH]c1/C=C/N(C)C)Br HD-0742 Cc1cc(cc(c1NC(=O)C(F)(F)F)C(=O)C)I HD-0743 CNc1ccc(c(n1)OC)C(=O)OC HD-0744 CCOC(=O)c1cnc(c(c1Cl)[N+](=O)[O-])Cl HD-0745 Cc1cc(cc(c1N)C(=O)C)I HD-0746 CC(=O)n1c2ccc(cc2c(n1)Cl)[N+](=O)[O-] HD-0747 c1cc(c(cc1Cl)Cl)C(=O)Cc2c(cc(cn2)C(F)(F)F)Cl HE-0003 c1cc(ccc1C#N)Nc2[nH]ccc(=O)n2 HE-0007 c1cc(c(cc1C(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cl)Cl HE-0008 c1ccc(cc1)CNc2cccc(c2C#N)F HE-0011 CC(C)(C)OC(=O)N1CCN(CC1)c2cccc(c2C#N)NCc3ccccc3 HE-0012 CC(C)(C)OC(=O)N1CCN(CC1)c2cccc3c2CNC(=O)N3Cc4ccccc4 HE-0013 c1ccc(cc1)CN2c3cccc(c3CNC2=O)N4CCNCC4.Cl HE-0014 CC(C)(C)OC(=O)c1ccc(nc1)Cl HE-0017 Cc1ccc2c(c1)n(c(=O)[nH]2)C3CCN(CC3)C(=O)OC(C)(C)C HE-0020 CC1(C2CCC1(CC2)CS(=O)(=O)O)C.c1ccnc(c1)CN2CCC(=O)CC2 HE-0021 c1cc(ccc1C#N)Nc2nccc(n2)Cl HE-0022 CC1(CC(=O)c2c(nn(c2C1)c3cc(c(cc3)C(=O)O)N[C@H]4CC[C@@H](CC4)O)C(F)(F)F)C HE-0024 COC(Cc1ccccc1[N+](=O)[O-])OC HE-0029 Cc1cc(c(cc1F)[N+](=O)[O-])N HE-0034 c1c(cc(cc1Cl)Cl)/C(=N/O)/Cc2c(cc(cn2)C(F)(F)F)Cl HE-0035 CC(C)(C)OC(=O)c1ccc(cc1)N2C[C@H](C3(C2)C(=O)N(C(=O)N3C)c4cc(cc(c4)Cl)Cl)c5ccc(cc5)C#N HE-0037 c1cc(ccc1N2CCCCC2=O)I HE-0041 c1cc(nc(c1CNS(=O)(=O)C(F)(F)F)N2CCC(CC2)C(F)(F)F)C(F)(F)F HE-0043 c1cc(c(cc1/C(=N\O)/Cc2c(cc(cn2)C(F)(F)F)Cl)Cl)Cl HE-0044 Cc1ccc2c(c1)n(c(=O)[nH]2)C3CCNCC3.Cl HE-0046 COC(Cc1ccccc1N)OC HE-0069 c1cc(cc(c1)F)C2=N[C@@H]2c3c(cc(cn3)C(F)(F)F)Cl HE-0076 Cc1cc(cc(c1Nc2ccnc(n2)Nc3ccc(cc3)C#N)C)Br HE-0078 c1cc(c2c(c1Cl)CCNC2)Cl.Cl HE-0079 Cc1cc(c(cc1F)N)N HE-0085 Cc1cc2c(cc1F)[nH]c(=O)n2C3CCN(CC3)C(=O)OC(C)(C)C HE-0086 CC(C)(C)c1cc(c(cc1[N+](=O)[O-])O)C(C)(C)C HE-0089 c1cc2c(cc1CO)OCCO2 HE-0207 c1cc(ccc1N)N2CCOCC2=O HE-0208 c1cc(c(c(c1)Cl)c2ncc3n2cc(cc3C(F)(F)F)Cl)Cl HE-0210 Cc1c(cnc(n1)c2c(cc(cn2)C(F)(F)F)Cl)NC(=O)N(C)C HE-0213 c1cc(ccc1C(=O)O[C@H]2CN(OC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl HE-0216 CC(C)C(=O)O[C@H]1CN(OC1)c2c(cc(cn2)C(F)(F)F)Cl HE-0219 COC(=O)c1ccnc(c1)N HE-0224 c1cc(ccc1/C=N/c2ccc(c(c2)[N+](=O)[O-])N)F HE-0226 c1cnc(nc1)c2nc(cc(n2)O)C(F)(F)F HE-0227 C1[C@@H]2[C@@H]([C@H]2CO)CN1 HE-0228 COC(=O)c1cc(ncc1Br)N HE-0229 COC(=O)c1ccn2ccnc2c1 HE-0231 CC(C)(C)OC(=O)N1C[C@@H]2[C@H](C1)[C@H]2CO HE-0233 c1cc(ccc1CNc2ccc(c(c2)[N+](=O)[O-])N)F HE-0235 c1cnc(nc1)c2nc(cc(n2)Cl)C(F)(F)F HE-0237 c1cnc2c(c1C(F)(F)F)c(=O)[nH][nH]2 HE-0239 c1cn2ccnc2cc1C(=O)O HE-0336 c1c(cnc(c1Cl)N2CCCCCC2)C(F)(F)F HE-0701 CC(C)(C)OC(=O)N1CCN(CC1)c2c(ccc(n2)Cl)[N+](=O)[O-] HE-0702 COC(=O)c1cc2ncc(cn2n1)Br HE-0708 Cc1c(c2ncc(cn2n1)Br)C#N HE-0711 CCOC(=O)C1CCCN(C1)c2c(cc(cn2)C(F)(F)F)Cl HE-0713 CCOC(=O)C1CCCN(C1)c2c(cccn2)[N+](=O)[O-] HE-0714 c1c(cnc(c1Cl)Cl)CO HE-0716 c1c(cnc(c1Cl)Cl)C=O HE-0717 c1c(cnc(c1Cl)N2CC(C2)O)C(F)(F)F HE-0718 c1c(cnc(c1Cl)N2CCC3(CC2)NCCS3)C(F)(F)F.Cl HE-0720 Cn1c2c(c(cc(n2)C3CC3)C(F)(F)F)c(n1)N HE-0724 c1c(c2c(n[nH]c2nc1C3CC3)N)C(F)(F)F HE-0725 CCOC(=O)c1c(nc(s1)N(c2ccccc2)c3ccccc3)C HE-0726 CCOc1c(nc2ccccc2n1)C(=O)O HE-0727 Cn1c2ccc(cc2[nH]c(=O)c1=O)C(=O)OC HE-0728 c1ccc(cc1)CN2CCC(CC2)Nc3c(cc(cn3)C(F)(F)F)Cl HE-0729 Cc1c(sc(n1)N(c2ccccc2)c3ccccc3)C(=O)O HE-0730 Cn1c2ccc(cc2nc1CCl)C(=O)OC HE-0732 CCOC(=O)C1CCCN(C1)c2c(cccn2)N HE-0733 Cn1c2ccc(cc2[nH]c1=O)C(=O)O HE-0735 CC(C)(C)OC(=O)N1CCC(C1=O)C(=O)OC HE-0736 Cc1c(=O)n(c2ccc(cc2n1)C(=O)OC)C HE-0737 COC(=O)C1CCNC1=O.Cl HE-0738 COC(=O)c1cc2c(ncnc2s1)N HE-0739 Cn1c2ccc(cc2[nH]c(=O)c1=O)C(=O)O HE-0740 c1cc(c(cc1[N+](=O)[O-])Br)CO HE-0741 Cn1c2ccc(cc2nc(c1=O)Cl)C(=O)OC HE-0744 c1cc(ccc1C2c3ccc(cc3CO2)C#N)F HF-0004 CC(=O)Nc1nc(cs1)C(C)(C)C HF-0005 CC(C)(C)c1cc([nH]n1)O HF-0006 CC(C)(C)c1cc(cc(c1O)[N+](=O)[O-])[N+](=O)[O-] HF-0007 CC(C)(C)c1c(c([nH]n1)O)[N+](=O)[O-] HF-0008 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=N/NC(=S)Nc2ccccc2 HF-0009 c1ccc2c(c1)CCN(C2)c3cc(sc3)[N+](=O)[O-] HF-0010 CCOC(=O)CCC(=O)Nc1ccc(cc1)C(=O)C HF-0011 Cc1ccc(cc1)Sc2c3c([nH]cn3)nc(n2)N HF-0012 CCOC(=O)N1CCN(CC1)c2cc(ccc2[N+](=O)[O-])C(F)(F)F HF-0013 Cc1csc(c1NC(=O)Nc2ccc(cc2)Cl)C(=O)OC HF-0014 CCOC(=O)C1CCN(CC1)C(=O)Nc2ccccc2 HF-0015 CCOC(=O)C(CC(C)C)NS(=O)(=O)c1ccc(cc1)CSc2ccc(cc2)F HF-0016 c1ccc(cc1)NC(=O)NNC(=O)c2ccncc2 HF-0017 c1ccc(cc1)NC(=O)Nc2nc(cc(n2)Cl)Cl HF-0019 CCOC(=O)c1ccc(cc1)NC(=O)/C=C\C(=O)O HF-0020 c1ccc(cc1)NC(=O)Nc2ccc(cn2)[N+](=O)[O-] HF-0021 c1ccc(cc1)NC(=O)Nc2cc(cc(c2)Cl)Cl HF-0022 c1ccc2c(c1)nc(s2)Sc3ccc(cn3)[N+](=O)[O-] HF-0023 C[n+]1ccc(cc1)c2nnc(s2)c3cc[n+](cc3)C.[I-].[I-] HF-0024 c1c(ccnc1)/C=N/N=C/c2ccncc2 HF-0025 c1ccc(cc1)NC(=S)N2CCCc3c2cccc3 HF-0026 CCOC(=O)c1c(nc(s1)NC(=O)CCl)c2ccccc2 HF-0027 c1ccc2c(c1)[nH]c(n2)SCC(=O)N HF-0029 CC(C)(C)c1c(c([nH]n1)O)C(=O)Nc2ccccc2 HF-0030 CCOC(=O)CNC(=O)Nc1nc(cs1)c2ccc(cc2)C HF-0031 c1ccc(cc1)SCC(=O)N HF-0032 c1ccc(cc1)S(=O)(=O)CC(=O)N HF-0033 c1ccc(c(c1)Nc2cc(nc(n2)N)Cl)F HF-0034 c1ccc(cc1)NC(=O)N2CCCc3c2cccc3 HF-0035 C(C(=O)N)Sc1nnc(s1)SCC(=O)N HF-0036 CSc1nc(cc(n1)Sc2cccc(c2)F)Sc3cccc(c3)F HF-0037 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Sc3[nH]c4ccccc4n3 HF-0038 c1cc(cc(c1)F)N2CC3(CCNCC3)OC2=O HF-0048 C1CN(CCC1C(F)(F)F)CCN2CCNC2=O HF-0050 c1ccc(cc1)N2CC3(CCNCC3)OC2=O.Cl HF-0055 c1ccc(cc1)COC(=O)N2CCC(CC2)(CNc3ccc(cc3)F)O HF-0058 c1ccc(cc1)COC(=O)N2CCC(CC2)(CNc3ccc(cc3F)Cl)O HF-0059 CC(C)(C(=O)OC)Nc1c(cc(cn1)C(F)(F)F)Cl HF-0065 c1ccc(cc1)COC(=O)N2CCC3(CC2)CN(C(=O)O3)c4ccc(cc4)F HF-0068 c1cc(ccc1NCC2(CCNCC2)O)F HF-0069 c1cc(ccc1NC(=O)OC[C@H]2CCCCN2c3c(cc(cn3)C(F)(F)F)Cl)Cl HF-0133 c1cc(c(cc1Cl)F)NCC2(CCNCC2)O HF-0150 Cc1cc(cc(c1O)C)C(=O)CN2CCCCC2 HF-0155 c1ccc(cc1)COC(=O)N2CCC3(CC2)CN(C(=O)O3)c4ccc(cc4F)Cl HF-0160 COC(=O)c1ccc(cc1)CN2CCSCC2 HF-0164 C[C@@H]1CN(C[C@@H](O1)C)Cc2ccc(cc2)C(=O)OC HF-0168 COC(=O)c1ccc(cc1)CN2CCOCC2 HF-0170 COC(=O)c1ccc(cc1)CN2CCCC2 HF-0172 C[C@@H]1CN(C[C@@H](O1)C)Cc2ccc(cc2)C(=O)O HF-0173 c1cc(ccc1CN2CCSCC2)C(=O)O HF-0177 c1cc(ccc1CN2CCOCC2)C(=O)O.Cl HF-0179 COC(=O)c1ccc(cc1)C[N+]2(CCCC2)Cc3ccc(cc3)C(=O)OC.[Br-] HF-0180 COC(=O)CC(c1ccc(cc1)Cl)N.Cl HF-0207 CC(C)(C)OC(=O)N1CCC(=CC#N)CC1 HF-0215 CC(C)(C)OC(=O)N1CCC(CC1)CC#N HF-0217 C1CNCCC1CC#N HF-0228 C(CSC[C@@H](C(=O)O)N)C(=O)O HF-0229 c1cn2ccnc2c(c1Cl)I HF-0723 c1cc2c(cc1NC(=O)C(F)(F)F)OCO2 HF-0726 CCOC(=O)c1cc2cc(cnc2nc1Cl)Br HF-0728 COc1cc(c(cc1Cl)N)N HF-0730 CCOC(=O)c1cc2cc(cnc2nc1O)Cl HF-0731 c1cn2cc(nc2c(c1Cl)I)C(F)(F)F HF-0736 CCOC(=O)c1cn2ccc(c(c2n1)I)Cl HF-0737 c1c2cc(c(nc2ncc1Cl)O)C#N HF-0748 c1cc2c(cc1Cl)C(CS2(=O)=O)O HF-0751 c1c2cc(c(nc2ncc1Cl)Cl)C#N HF-0753 c1cc2c(cc1Cl)c(n[nH]2)Br HF-0754 c1cc2c(cc1Cl)c(n[nH]2)Cl HF-0755 CCOC(=O)c1cc2cc(cnc2nc1NN)Br HF-0759 CNC(=O)c1ccccc1O HF-0760 c1c2cc3c(n[nH]c3nc2ncc1Cl)N HF-0761 c1cn2cc(nc2c(c1Cl)I)C(=O)O HF-0762 COc1c(c(c2ccccc2c1Br)Br)O HF-0764 CCCc1ccc2c(c1)sc(n2)N HG-0005 c1ccc(cc1)CN2CC3C(C2)C(=O)NC3=O HG-0008 c1cc(oc1C(=O)O)Cl HG-0015 c1cc(c(cc1F)CCl)Br HG-0023 COC(=O)/C(=N/O)/Cc1ccc(cc1)O HG-0044 COC(=O)CCc1ccc(cc1)OCc2cc(ccc2Br)F HG-0047 COC(=O)C(=NO)Cc1ccc(c(c1)Br)O HG-0050 CC(C)(C)OC(=O)N1CC2CN(CC2C1)Cc3ccccc3 HG-0052 Cc1ccc(cc1)c2ccc(cc2COc3ccc(cc3)CCC(=O)OC)F HG-0062 c1(c(nc(nc1O)N)N)Cl HG-0204 c1(c(nc(nc1O)N)N)I HG-0206 CC(=O)Nc1cccc2c1ncc(c2)I HG-0213 Cc1ccc(cc1)CNC(=O)CCCCCBr HG-0216 c1cc(ccc1CNC(=O)CCCCCBr)C#N HG-0220 CC(=O)n1ccc2c1nccc2I HG-0221 CC(C)(C)OC(=O)NNC1CCOCC1 HG-0222 Cc1ccc(cc1)CNC(=O)CCCCCN2CCN(CC2)CCCCCC(=O)NCc3ccc(cc3)C HG-0227 C1COCCC1NN.Cl.Cl HG-0229 CCOC(=O)c1c(nc(s1)Nc2ccc(cc2)OC)C HG-0703 COC(=O)c1ccc(c(c1)F)NCc2ccccc2O HG-0704 Cc1c(cccc1OC)C(=O)NN HG-0706 CC(C)(C)OC(=O)N1CCCCC12CCNC2.Cl HG-0707 COC(=O)c1c(c(nc(n1)Cl)N)Cl HG-0708 c1ccc(cc1)CN2CCCCC23CCNC3 HG-0710 CNC(=O)NCc1c(cc(cn1)C(F)(F)F)Cl HH-0200 c1ccc(cc1)CNC(=O)NCc2c(cc(cn2)C(F)(F)F)Cl HH-0202 CCOC(=O)C=Cc1ccc(cc1)c2ccc(cc2)Br HH-0211 c1c(c(cnc1Cl)[N+](=O)[O-])C(=O)N HH-0700 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])NN HH-0701 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])N(C)C HH-0704 CNc1ccc(cc1[N+](=O)[O-])C#N HH-0705 c1cc(c(cc1CO)[N+](=O)[O-])[N+](=O)[O-] HH-0706 c1cc(c(cc1C=O)[N+](=O)[O-])[N+](=O)[O-] HH-0707 c1cnc(c(c1C(F)(F)F)C=O)Cl HH-0708 c1cc(c(cc1C(=O)N)[N+](=O)[O-])[N+](=O)[O-] HH-0716 CCn1c2c(c(n1)C)c(cc(=O)[nH]2)C(F)(F)F HK-0033 COC(=O)C(=O)Nc1cc(no1)c2ccc(cc2)Cl HK-0215 COc1cccc(c1)c2cc(on2)NC(=O)C(=O)OC HK-0216 C[C@@H]1[C@H](N(C(O1)(C)C)C(=O)OC(C)(C)C)C=O HK-0238 CC(=O)N[C@@H](Cc1ccc(cc1)N(C)C)C(=O)OC HK-0701 CC(=O)NC(Cc1ccc(cc1)N2CCN(CC2)C)C(=O)OC HK-0702 CC(=O)N[C@@H](Cc1ccc(cc1)N2CCN(CC2)C)C(=O)OC HK-0703 CC(=O)N[C@@H](Cc1c(ccc(c1F)F)F)C(=O)OC HK-0704 Cc1cnc(c(c1OC)C)CCl.Cl HL-0755 CCOC(=O)C1(CC1)C(=O)OCC HL-0756 c1ccc(cc1)C(=O)c2cc(c([nH]2)Br)Br HL-0757 CC(=O)N1CCC(CC1)c2ccc(cc2)O HL-0758 c1c([nH]cn1)/C=C/C(=O)O HS-0075 C/C=C/C#CCCO HS-0078 c1c(cnc(c1N)Br)Br HS-3000 Cc1cc(cnc1)CCl.Cl HS-3001 Cc1c(cc(cn1)Br)Br HS-3002 Cc1c(cncc1Br)Br HS-3003 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CSc2ccc(cc2)Br JS-0001 c1ccnc(c1)SCC(=O)Nc2cccc(c2)[N+](=O)[O-] JS-0002 Cc1ccc(cc1C)NC(=O)CSc2ccc(cc2)Br JS-0003 Cn1cnnc1SCC(=O)Nc2cccc(c2)[N+](=O)[O-] JS-0004 Cc1ccc(cc1C)NC(=O)CSc2ccccn2 JS-0006 CCOC(=O)CNC(=O)CSc1ccc(cc1)Br JS-0007 Cc1cc(nc(n1)SCC(=O)Nc2ccc(cc2)OC)C JS-0008 Cc1ccc(cc1C)NC(=O)CSc2nncn2C JS-0010 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CSC2CCCCC2 JS-0011 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)Cl)F JS-0012 c1ccnc(c1)SCC(=O)Nc2ccc3c(c2)OCO3 JS-0013 c1cc(ccc1SCC(=O)Nc2ccc3c(c2)OCO3)Br JS-0014 Cn1cnnc1SCC(=O)Nc2cccc(c2)C(F)(F)F JS-0015 c1cc(ccc1C2CCCCC2)NC(=O)CSc3ccc(cc3)Br JS-0016 Cn1cnnc1SCC(=O)Nc2ccc(c(c2)Cl)F JS-0017 c1ccnc(c1)SCC(=O)Nc2cccc(c2)C(F)(F)F JS-0018 Cn1cnnc1SCC(=O)Nc2ccc3c(c2)OCCO3 JS-0019 c1cc(c(cc1C=O)[N+](=O)[O-])N2CCCC2 JS-001C Cn1cnnc1SCC(=O)Nc2ccc(cc2)C3CCCCC3 JS-0020 c1ccnc(c1)SC2CC(=O)N(C2=O)c3ccc(cc3)Br JS-0021 c1ccc(cc1)CN(Cc2ccccc2)C3CC(=O)N(C3=O)c4ccc(cc4)Br JS-0022 CCOc1ccc(cc1)NC(=O)C(=S)NCc2ccccc2 JS-0023 c1cc(c(cc1NC(=O)CCC(=O)N2CCCC2)[N+](=O)[O-])F JS-0024 CCCCc1ccc(cc1)NC(=O)C(=S)NCc2ccccc2 JS-0025 Cc1ccc(cc1NC(=O)CSc2nnnn2C)F JS-0026 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)Cl)Cl JS-0027 c1cc(ccc1N2C(=O)CC(C2=O)Sc3ccc(cc3)Cl)Br JS-0028 Cc1cc(ccc1NC(=O)CSc2ccccn2)Br JS-0029 c1cc(c(cc1[N+](=O)[O-])C=O)N2CCCCC2 JS-002C Cc1cc(nc(n1)SCC(=O)Nc2ccc(c(c2)Cl)Cl)C JS-0030 Cc1cc(ccc1NC(=O)CSc2nc(cc(n2)C)C)Br JS-0031 Cn1c(nnn1)SCC(=O)Nc2ccc(c(c2)Cl)Cl JS-0032 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)C(F)(F)F)Cl JS-0033 c1cc(c(cc1NC(=O)C(=S)NC2CCCCC2)Cl)Cl JS-0034 c1cc(c(cc1NC(=O)C(=O)NC2CCCCC2)Cl)Cl JS-0035 c1cc(c(cc1NC(=O)CN2CCOCC2)Cl)F JS-0036 c1cc(ccc1C2CCCCC2)NC(=O)C(=S)NC3CCCCC3 JS-0037 Cc1ccc(cc1)NC(=O)CSc2nc(cc(n2)C)C JS-0038 Cc1ccc(cc1)NC(=O)CN2CCCc3c2cccc3 JS-0039 Cc1ccc(cc1)NC(=O)CN2CCOCC2 JS-0040 Cc1ccc(cc1)NC(=O)CN2CCCCC2 JS-0041 c1cc(ccc1C2CCCCC2)NC(=O)C(=O)NC3CCCCC3 JS-0042 c1ccc(c(c1)NC(=O)CN2CCCCC2)[N+](=O)[O-] JS-0043 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(c(c2)C(F)(F)F)Cl JS-0044 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(c(c2)Cl)F JS-0045 CCCCc1ccc(cc1)NC(=O)CSc2nnnn2C JS-0046 Cc1cc(nc(n1)SCC(=O)Nc2ccccc2[N+](=O)[O-])C JS-0047 c1ccc(cc1)CNC(=O)C(=O)Nc2ccc(c(c2)C(F)(F)F)Cl JS-0049 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C=O)Br JS-004C CCOC(=O)C(CSC1CC(=O)N(C1=O)c2ccc(cc2)Br)N.Cl JS-0050 c1ccc(cc1)CNC(=O)C(=O)Nc2ccc(c(c2)Cl)F JS-0051 CCOc1ccc(cc1)NC(=O)C(=O)NCc2ccccc2 JS-0052 c1cc(ccc1SC2CC(=O)N(C2=O)c3ccc(cc3F)F)Cl JS-0053 CCOc1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cc2)Cl JS-0054 c1cc(c(cc1F)F)N2C(=O)CC(C2=O)N3CCOCC3 JS-0055 COc1ccccc1c2c(c(=O)c3ccccc3o2)OC(=O)c4cccs4 JS-0056 CCOC(=O)COc1c(=O)c2ccccc2oc1c3ccc(cc3)OC JS-0057 CCOC(=O)COc1c(=O)c2ccccc2oc1c3cccc(c3OC)OC JS-0058 CCOc1ccc(cc1)C(=O)CC(C(=O)O)N JS-0059 c1cc(ccc1Sc2ccc(cc2C=O)[N+](=O)[O-])Cl JS-005C c1ccc(c(c1)NC(=O)CSc2ccccn2)Br JS-0061 Cn1c(nnn1)SCC(=O)Nc2ccccc2Br JS-0062 Cc1cc(nc(n1)SCC(=O)Nc2ccccc2Br)C JS-0063 Cc1cccc(c1C)NC(=O)C(=S)NCc2ccccc2 JS-0064 c1ccc(c(c1)NC(=O)CSc2ccc(cc2)Cl)Br JS-0065 Cn1c(nnn1)SCC(=O)Nc2cccc(c2)C(F)(F)F JS-0066 c1ccnc(c1)SC2CC(=O)N(C2=O)c3ccc(cc3F)F JS-0067 c1ccc(cc1)CNC(=S)C(=O)Nc2cccc(c2)C(F)(F)F JS-0068 Cn1c(nnn1)SCC(=O)Nc2ccc(c(c2)Cl)F JS-0069 Cc1cccc(c1C)NC(=O)C(=O)NCc2ccccc2 JS-0070 Cn1c(nnn1)SCC(=O)Nc2ccccc2[N+](=O)[O-] JS-0071 Cc1ccc(cc1)NC(=O)C(=S)NCc2ccco2 JS-0072 CCOc1ccc(cc1)NC(=O)CSc2nnnn2C JS-0074 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cc2)Cl JS-0075 c1ccc(cc1)CNC(=O)C(=O)Nc2cccc(c2)C(F)(F)F JS-0076 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)N2CCCCC2 JS-0077 Cc1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)C JS-0078 CC(=O)Oc1c(=O)c2ccccc2oc1c3cccc(c3OC)OC JS-0079 c1ccc(cc1)Sc2ccc(cc2C=O)[N+](=O)[O-] JS-007C Cc1ccc(cc1)C(=O)CC(C(=O)O)N2CCCC2 JS-0080 Cc1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccco2.Cl JS-0081 Cc1ccc(cc1)Sc2ccc(cc2/C=C\3/C(=O)N(C(=S)S3)c4ccccc4Cl)[N+](=O)[O-] JS-0083 Cc1ccc(cc1C#N)/N=C/c2cccs2 JS-0084 COc1ccc(cc1NC(=O)CSc2ccccn2)Cl JS-0085 Cc1ccc(cc1)NC(=O)CSc2ccccn2 JS-0086 Cc1ccc(cc1)NC(=O)CSc2nncn2C JS-0087 COc1ccc(cc1[N+](=O)[O-])CNc2ccc(cc2)Br JS-0088 Cc1cccc(c1C)NC(=O)CSc2ccccn2 JS-0089 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C=O JS-008C c1cc(ccc1CSCC(=O)Nc2ccc(c(c2)Cl)Cl)Cl JS-0090 Cc1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccccc2.Cl JS-0091 c1cc(oc1)CNC(=S)C(=O)Nc2ccc(c(c2)Cl)F JS-0092 c1ccc(cc1)CN2C(=O)/C(=C\c3ccccc3SC4CCCCC4)/SC2=S JS-0093 COc1ccc(cc1[N+](=O)[O-])CNc2cc(c(cc2F)F)F JS-0094 COc1ccc(cc1[N+](=O)[O-])/C=C/2\C(=O)N(C(=S)S2)Cc3ccccc3 JS-0095 Cc1ccc(cc1)Sc2ccc(cc2/C=C\3/C(=O)N(C(=S)S3)Cc4ccccc4)[N+](=O)[O-] JS-0096 Cc1ccc(c(c1)NC(=O)CSc2ccccn2)OC JS-0097 c1ccc(c(c1)NC(=O)CSCc2ccc(cc2)Cl)Br JS-0098 c1cc(oc1)CNC(=S)C(=O)Nc2ccc(c(c2)C(F)(F)F)Cl JS-0099 c1cc(c(cc1[N+](=O)[O-])C=O)SC2CCCCC2 JS-009C Cc1ccc(c(c1)NC(=O)C(=S)NCc2ccco2)OC JS-0101 c1cc(ccc1SCC(=O)NNC(=O)NC2CCCCC2)Cl JS-0103 Cc1ccc(c(c1)NC(=O)C(=S)NCc2ccccc2)OC JS-0104 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)/C=C\C(=O)c3ccccc3 JS-0105 CC(C)(C)C(=O)Oc1ccc(cc1)/C=C/C(=O)c2ccccc2 JS-0106 c1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OC(=O)c3cccs3 JS-0107 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nnnn2c3ccccc3 JS-0108 Cc1ccc(cc1)C(=O)Oc2ccc(cc2[N+](=O)[O-])F JS-0109 c1cc(ccc1C(=O)Oc2ccc(cc2[N+](=O)[O-])F)[N+](=O)[O-] JS-0110 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)Sc3ccc(cc3)OC(=O)c4ccc(cc4)C JS-0111 c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccs3 JS-0112 c1cc(c(cc1[N+](=O)[O-])C2SCCS2)SC3CCCCC3 JS-0113 c1cc(ccc1C(=O)Oc2ccc(cc2[N+](=O)[O-])F)Cl JS-0114 c1cc(sc1)C(=O)Oc2ccc(cc2)Sc3ccc(cc3)OC(=O)c4cccs4 JS-0115 CC(C)(C)C(=O)Oc1ccc(cc1)Sc2ccc(cc2)OC(=O)C(C)(C)C JS-0116 Cc1ccc(cc1)C(=O)O/N=C/c2cc(ccc2OC)Br JS-0117 CC(C)(C)c1ccc(cc1)C(=O)O/N=C/c2cc(ccc2OC)Br JS-0118 Cc1cc(ccc1Br)NC(=O)CSc2nnc(s2)C JS-0119 Cc1ccc(cc1)Sc2ccc(cc2C=O)[N+](=O)[O-] JS-011C Cc1ccc(cc1)Sc2ccc(cc2C3SCCS3)[N+](=O)[O-] JS-0121 c1cc(sc1)C(=O)O/N=C/c2ccc3c(c2)OCO3 JS-0122 COc1ccc(cc1[N+](=O)[O-])C2SCCS2 JS-0123 c1cc(oc1)CSc2ccc(cc2C3SCCS3)[N+](=O)[O-] JS-0125 Cc1cc(ccc1Br)NC(=O)CSc2nnnn2c3ccccc3 JS-0127 CCCCCCCC(=O)Oc1ccc(cc1)/C=C/C(=O)c2ccccc2 JS-0129 C#CCSc1nnc(s1)N JS-012C Cc1ccc(cc1)C(=O)OCc2cc(ccc2Sc3ccccc3)[N+](=O)[O-] JS-0130 c1cc(c(cc1F)[N+](=O)[O-])OC(=O)CCCC(=O)Oc2ccc(cc2[N+](=O)[O-])F JS-0131 c1ccc(cc1)CC(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccccc3 JS-0132 CC(C)(C)c1ccc(cc1)C(=O)OCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0133 Cc1ccc(cc1)C(=O)OCc2cc(ccc2OC)Br JS-0134 c1c(c(cc2c1OCO2)[N+](=O)[O-])COC(=O)CCCC(=O)OCc3cc4c(cc3[N+](=O)[O-])OCO4 JS-0135 c1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)CCCC(=O)Oc3ccc(cc3)/C=C/C(=O)c4ccccc4 JS-0136 COc1ccc(cc1COC(=O)c2ccc(cc2)[N+](=O)[O-])Br JS-0137 c1ccc(cc1)Sc2ccc(cc2/C=C\3/C(=O)N(C(=S)S3)c4ccccc4Cl)[N+](=O)[O-] JS-0139 Cc1ccc(cc1C#N)N JS-013C Cc1ccc(cc1)C(=O)OCc2cc(ccc2Cl)[N+](=O)[O-] JS-0140 CC(C)(C)c1ccc(cc1)C(=O)OCc2cc(ccc2Cl)[N+](=O)[O-] JS-0141 c1ccc(cc1)/C=C\C(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccccc3 JS-0142 COc1ccc(cc1COC(=O)/C=C/c2ccccc2)Br JS-0143 c1ccc(cc1)/C=C/C(=O)OCc2cc(ccc2Cl)[N+](=O)[O-] JS-0144 Cc1ccc(cc1C#N)NC(=S)NCc2ccccc2 JS-0145 Cc1ccc(cc1C#N)NC(=S)NC JS-0146 c1cc(c(cc1[N+](=O)[O-])C=O)SCCSc2ccc(cc2C=O)[N+](=O)[O-] JS-0148 c1ccc(cc1)CC(=O)OCc2cc(ccc2Cl)[N+](=O)[O-] JS-0149 Cc1ccc(cc1C)Nc2[nH]nc(n2)N JS-014C COc1ccc(cc1)C(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccccc3 JS-0151 COc1ccc(cc1)C(=O)OCc2cc(ccc2Cl)[N+](=O)[O-] JS-0153 CC(C1C/C(=C/c2ccc(cc2)OC)/C(=O)/C(=C\c3ccc(cc3)OC)/C1)(C)C JS-0155 Cc1ccc(cc1)Sc2ccc(cc2COC(=O)c3cccs3)[N+](=O)[O-] JS-0157 Cc1ccc(cc1)C(=O)OCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0159 Cc1ccc(cc1)C(=O)ON=C2CCCCCCCCCCC2 JS-0160 CC(C)(C)c1ccc(cc1)C(=O)ON=C2CCCCCCCCCCC2 JS-0161 c1cc(sc1)C(=O)ON=C2CCCCCCCCCCC2 JS-0162 COc1ccc(cc1)C(=O)ON=C2CCCCCCCCCCC2 JS-0163 CCC(C)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl JS-0164 CCC(C)c1ccc(cc1)NC(=O)CSc2nnnn2C JS-0165 Cc1ccc(cc1)Sc2ccc(cc2COC(=O)/C=C/c3ccccc3)[N+](=O)[O-] JS-0166 CCC(C)c1ccc(cc1)NC(=O)CSc2nc(cc(n2)C)C JS-0167 c1cc(ccc1C(=O)ON=C2CCCCCCCCCCC2)[N+](=O)[O-] JS-0168 CCC(C)c1ccc(cc1)NC(=O)CSc2nncn2C JS-0169 Cc1cccc(c1)CSc2nnc(s2)N JS-016C c1cc(ccc1C(=O)OCc2cc3c(cc2[N+](=O)[O-])OCO3)[N+](=O)[O-] JS-0170 CCC(C)c1ccc(cc1)NC(=O)CSCc2ccc(cc2)Cl JS-0172 CCC(C)c1ccc(cc1)NC(=O)CSc2nnnn2c3ccccc3 JS-0173 c1cc(sc1)C(=O)OCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0175 c1cc(ccc1C(=O)ON=C2CCCCCCCCCCC2)Cl JS-0176 Cc1ccc(cc1)C(=O)Oc2c(=O)c3ccccc3oc2c4ccc(cc4)OC JS-0178 CCC(C)c1ccc(cc1)NC(=O)CSc2nccn2C JS-0179 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OC(=O)c4cccs4 JS-0182 c1c(c(cc2c1OCO2)[N+](=O)[O-])COC(=O)C=C3C=CCC=C3 JS-0183 Cc1nnc(s1)SCC(=O)Nc2ccc(c(c2)Cl)F JS-0186 Cc1ccc(cc1NC(=O)CSc2nnc(s2)C)F JS-0187 c1cc(ccc1C(=O)ON=C2CCCCCCCCCCC2)F JS-0188 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OC(=O)/C=C/c4ccccc4 JS-0189 Cc1ccc(cc1)C(c2ccccc2)OC(=O)c3ccc(cc3)[N+](=O)[O-] JS-0190 c1ccc(cc1)/C=C\C(=O)ON=C2CCCCCCCCCCC2 JS-0191 Cc1ccc(cc1)C(=O)Oc2ccc3c(cc(=O)oc3c2)C JS-0193 Cc1nnc(s1)SCC(=O)Nc2ccc(c(c2)C(F)(F)F)Cl JS-0194 c1cc(sc1)C(=O)OCc2cc(ccc2SC3CCCCC3)[N+](=O)[O-] JS-0196 c1cc(ccc1C(=O)OCc2cc3c(cc2[N+](=O)[O-])OCO3)F JS-0197 c1cc(ccc1C(=O)OCc2cc(ccc2SC3CCCCC3)[N+](=O)[O-])[N+](=O)[O-] JS-0198 CCC(C)c1ccc(cc1)NC(=O)C(=S)NCc2ccccc2 JS-0199 Cc1ccc(cc1)C(=O)O/N=C/c2ccc(cc2)N(C)C JS-0200 CCC(C)c1ccc(cc1)NC(=O)C(=O)NCc2ccccc2 JS-0201 c1cc(ccc1C(=O)OCc2cc(ccc2Cl)[N+](=O)[O-])[N+](=O)[O-] JS-0202 Cc1ccc(cc1)C(=O)Oc2ccccc2C(=O)/C=C\c3ccccc3OC JS-0204 c1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OC(=O)c3ccc(cc3)F JS-0205 c1ccc(cc1)/C=C/C(=O)OCc2cc(ccc2SC3CCCCC3)[N+](=O)[O-] JS-0206 CCC(C)c1ccc(cc1)NC(=O)C(=S)NC2CCCCC2 JS-0207 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(cc2)C(F)(F)F JS-0210 Cc1cc(ccc1Br)NC(=O)C(=S)NCc2ccccc2 JS-0211 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)Br)Cl JS-0212 Cc1cc(ccc1Br)NC(=O)C(=O)NCc2ccccc2 JS-0213 CC(C)(C)C1CCC(=NOC(=O)c2ccc(cc2)[N+](=O)[O-])CC1 JS-0214 COc1ccc(cc1COC(=O)c2cccs2)Br JS-0216 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)Sc3ccc(cc3)OC(=O)c4ccc(cc4)C(C)(C)C JS-0218 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)/C=C\C(=O)c3ccccc3 JS-0219 c1cc(ccc1N)SCc2ccc(cc2Cl)Cl JS-021C Cc1ccc(c(c1)NC(=O)C(=O)NCc2ccccc2)OC JS-0220 CC(C)(C)c1ccc(cc1)C(=O)OCc2cc(ccc2OC)Br JS-0221 c1ccc(cc1)/C=C\C(=O)Oc2ccc(cc2)Sc3ccc(cc3)OC(=O)/C=C\c4ccccc4 JS-0222 c1cc(ccc1C(=O)Oc2ccc(cc2)Sc3ccc(cc3)OC(=O)c4ccc(cc4)F)F JS-0223 COc1ccc(cc1)C(=O)OCc2cc(ccc2OC)Br JS-0225 COc1ccc(cc1COC(=O)c2ccc(cc2)F)Br JS-0226 COc1ccccc1/C=N/OC(=O)c2ccc(cc2)F JS-0227 CC(C)(C)c1ccc(cc1)C(=O)O/N=C/c2ccccc2OC JS-0228 CN(C)c1ccc(cc1)/C=N/OC(=O)c2ccc(cc2)OC JS-0229 c1cc(ccc1CSc2ccc(cc2)N)F JS-022C COc1ccccc1/C=N/OC(=O)c2ccc(cc2)[N+](=O)[O-] JS-0230 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C\c3ccc(cc3Cl)Cl JS-0231 CC(C)(C)C(=O)Oc1ccc(cc1)C(=O)/C=C\c2ccc(cc2Cl)Cl JS-0233 CC(C)c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)[N+](=O)[O-] JS-0234 CN(C)c1ccc(cc1)/C=N/OC(=O)c2ccc(cc2)F JS-0235 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)OC)C(=O)OCC)C)C JS-0236 c1cc(ccc1NC(=O)CCCC(=O)O)OC(F)(F)F JS-0237 CCOC(=O)c1c(nc(c(c1c2ccc(cc2)OC)C(=O)OCC)C)C JS-0238 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc(cc3)C(C)C JS-0239 C(C(=O)Nc1c(c(c(c(c1F)F)F)F)F)Cl JS-023C Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-0240 COc1ccc(c(c1OC)OC)/C=C/C(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)[N+](=O)[O-] JS-0241 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cc(ccc3OC)Br JS-0242 COc1ccc(c(c1OC)OC)/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccs3 JS-0243 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc(c(c3OC)OC)OC JS-0244 CC(C)c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccs3 JS-0245 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C\c3cccc4c3cccc4 JS-0246 c1c(c(cc(c1F)F)F)NC(=O)CCCC(=O)O JS-0247 c1cc(sc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc(cc3Cl)Cl JS-0248 c1cc(sc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-0249 c1c(c(cc(c1F)F)F)NC(=O)CCl JS-024C c1cc(ccc1C(=O)CC(C(=O)O)Sc2ccc(cc2)Cl)Br JS-0250 c1ccc2c(c1)cccc2/C=C/C(=O)c3ccc(cc3)OC(=O)c4cccs4 JS-0251 COc1ccc(cc1/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccs3)Br JS-0252 CN1CCN(CC1)C(CC(=O)c2ccc(cc2)Br)C(=O)O JS-0253 c1cc(ccc1C(=O)CC(C(=O)O)SC2CCCCC2)Br JS-0254 c1cc(c(cc1NC(=O)CCCC(=O)O)Cl)F JS-0255 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cc(ccc3OC)Br JS-0257 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc(c(c3OC)OC)OC JS-0258 c1cc(c(cc1NC(=O)CCl)Cl)F JS-025C c1cc(ccc1CSC(CC(=O)c2ccc(cc2)Br)C(=O)O)Cl JS-0260 c1cc(sc1)CNC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-0261 c1cc(ccc1C(=O)CC(C(=O)O)NC2CCCCC2)Br JS-0262 c1ccc(cc1)CNC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-0263 CCCCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C\c2ccc(cc2Cl)Cl JS-0264 CCCCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C\c2ccc3c(c2)OCO3 JS-0265 CCCCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C\c2cccc3c2cccc3 JS-0266 CCCCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C\c2ccc(cc2)C(C)C JS-0267 c1cc(c(cc1F)F)N2C(=O)CC(C2=O)N3CCCCC3 JS-0268 c1cc(c(cc1F)NC(=O)CCl)F JS-026C CC(C)c1ccc(cc1)/C=C\C(=O)c2ccc(cc2)OC(=O)/C=C/c3ccccc3 JS-0270 CC(C)(C)C(=O)Oc1ccc(cc1)C(=O)/C=C\c2ccc3c(c2)OCO3 JS-0271 c1ccc(cc1)/C=C/C(=O)Oc2ccc(cc2)C(=O)/C=C\c3ccc4c(c3)OCO4 JS-0272 Cc1cccc(c1)SC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-0273 c1cc(ccc1C(=O)/C=C\c2ccc3c(c2)OCO3)OC(=O)c4ccc(cc4)F JS-0274 c1cc(c(cc1F)F)Nc2nc(nc(n2)Cl)Cl JS-0275 Cc1cccc(c1)SC2CC(=O)N(C2=O)c3ccc(cc3)Br JS-0276 CCN(CC)CCCNc1nc(nc(n1)Cl)Nc2ccc(cc2F)F.Cl JS-0277 COc1ccc(cc1/C=C\C(=O)c2ccc(cc2)OC(=O)/C=C/c3ccccc3)Br JS-0278 COc1ccc(cc1/C=C\C(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl)Br JS-0279 c1cc(ccc1NC(=O)CCl)OC(F)(F)F JS-027C Cc1cc(ccc1Br)NCc2ccc(cc2O)OC JS-0280 CC(C)(C)C(=O)Oc1ccc(cc1)C(=O)/C=C\c2cccc3c2cccc3 JS-0281 c1cc(ccc1CNc2ccc(cc2)OC(F)(F)F)OCc3ccc(cc3)F JS-0282 Cc1ccnc(c1)NCc2ccc(cc2O)OC JS-0283 Cc1cc(ccc1Br)NCc2ccc(cc2)OCc3ccc(c(c3)Cl)Cl JS-0284 c1cc(c(cc1CNc2ccc(cc2F)F)[N+](=O)[O-])Cl JS-0285 c1cc(c(cc1F)F)NCc2cc3c(cc2Br)OCO3 JS-0286 c1cc(c(cc1F)F)NCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0287 Cc1cc(cnc1NCc2cccc(c2O)OC)Br JS-0288 COc1cccc(c1O)CNc2ccc(cc2)C#N JS-0289 COc1cccc(c1O)CNc2ccc(c(c2)[N+](=O)[O-])F JS-0290 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)C JS-0291 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2cccs2 JS-0292 c1cc(ccc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)Cl JS-0294 Cn1cnnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl JS-0295 c1c(cc(cc1Cl)Cl)NC(=O)C(=S)NC2CCCCC2 JS-0296 c1c(cc(cc1Cl)Cl)NC(=O)C(=O)NC2CCCCC2 JS-0297 Cc1nnc(s1)SCC(=O)Nc2cc(cc(c2)Cl)Cl JS-0298 Cc1ccc(cc1)SCC(=O)Nc2cc(cc(c2)Cl)Cl JS-0299 c1c(cc(cc1Cl)Cl)NC(=O)CSC2CCCCC2 JS-0300 c1c(cc(cc1Cl)Cl)NC(=O)C(=S)N2CCOCC2 JS-0301 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc(cc3)F JS-0303 c1ccc(cc1)CNC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O JS-0304 CN1CCN(CC1)C(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O JS-0305 CC(C)(C)C(=O)Oc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)F JS-0306 c1c(cc(cc1Cl)Cl)NC(=O)C(=O)N2CCOCC2 JS-0307 c1cc(sc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc(cc3)F JS-0308 Cc1cc(nc(n1)SCC(=O)Nc2cc(cc(c2)Cl)Cl)C JS-0309 c1cc2c(cc1NC(=O)CCl)OCCO2 JS-030C Cc1ccc(cc1NCc2cccc(c2O)OC)F JS-0310 COc1cccc(c1O)CNc2ccc(cc2)OC(F)(F)F JS-0311 CC(C)(C)C(=O)Oc1ccc(cc1)C(=O)/C=C/c2cccs2 JS-0312 c1ccc(c(c1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cccs3)Cl JS-0313 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cccs3 JS-0314 CC(C)(C)c1ccc(cc1)N(Cc2ccc(cc2OC)OC)C(=S)NCc3ccccc3 JS-0315 Cc1cc(ccc1Br)NCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0316 CC(C)(C)c1ccc(cc1)N(Cc2ccc(cc2OC)OC)C(=S)Nc3ccccc3Cl JS-0317 CC(C)(C)c1ccc(cc1)N(Cc2ccc(cc2OC)OC)C(=S)NC JS-0318 CC(C)(C)c1ccc(cc1)NCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0319 c1cc2c(cc1NC(=O)CCl)OCO2 JS-031C COc1cccc(c1O)CN(c2ccc(c(c2)Cl)F)C(=S)NCc3ccccc3 JS-0320 COc1ccc(c(c1)OC)CN(c2ccc(cc2)I)C(=S)NCc3ccccc3 JS-0321 CCCCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)F JS-0322 COc1ccc(c(c1)OC)CNc2ccc(cc2)I JS-0323 c1cc(c(c(c1)Cl)Cl)NCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0324 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccs3 JS-0326 CNC(=S)N(Cc1ccc(cc1OC)OC)c2ccc(cc2)I JS-0327 COc1cc(ccc1CNc2ccc(cc2)OC(F)(F)F)Br JS-0328 Cc1ccc(cc1NC(=O)CCl)F JS-032C CC(C)(C)C1CCC(=NOC(=O)c2ccc(cc2)Cl)CC1 JS-0330 Cc1ccc(cc1NCc2ccc(cc2OC)Br)F JS-0331 c1cc(ccc1C2CCCCC2)NCc3cc4c(cc3[N+](=O)[O-])OCO4 JS-0332 COc1ccc(cc1CNc2ccc(c(c2)[N+](=O)[O-])F)Br JS-0333 CC(C)(C)C1CCC(=NOC(=O)/C=C\c2ccccc2)CC1 JS-0334 COc1ccc(cc1CNc2cc(c(cc2F)F)F)Br JS-0335 COc1ccc(c(c1)OC)CN(c2ccc(cc2)I)C(=S)Nc3ccccc3 JS-0336 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OC(=O)c4ccccc4Cl JS-0337 CCCCCCCCCC(=O)Oc1c(=O)c2ccccc2oc1c3ccc(cc3)OC JS-0338 c1ccc(cc1)CNCC(=O)Nc2ccccc2[N+](=O)[O-] JS-0339 c1cc(c(cc1NC(=O)CCl)F)F JS-033C c1ccc(c(c1)NC(=O)CN2CCOCC2)[N+](=O)[O-] JS-0340 Cc1ccc(c(c1)NC(=O)CN2CCOCC2)OC JS-0341 CCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C\c2cccc3c2cccc3 JS-0342 c1ccc(c(c1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc4c(c3)OCO4)Cl JS-0343 Cc1ccc(cc1)SC2CC(=O)N(C2=O)c3ccc(cc3F)F JS-0344 CC[n+]1ccc(cc1)/C=C/c2cccc(c2OC)OC.[I-] JS-0345 Cc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl JS-0346 c1cc(c(cc1NC(=O)CN2CCOCC2)[N+](=O)[O-])Cl JS-0347 CC[n+]1ccc(cc1)/C=C/c2ccc(cc2OC)OC.[I-] JS-0348 Cn1cnnc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl JS-0349 c1cc(c(cc1F)F)NC(=O)CCl JS-034C Cc1nnc(s1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl JS-0350 Cn1ccnc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl JS-0351 Cc1ccc(cc1)SCC(=O)Nc2cccc(c2Cl)Cl JS-0352 CC[n+]1ccc(cc1)/C=C/c2ccc(c(c2OC)OC)OC.[I-] JS-0353 c1cc(c(c(c1)Cl)Cl)NC(=O)CSc2ccc(cc2)Cl JS-0354 c1cc(c(c(c1)Cl)Cl)NC(=O)CN2CCOCC2 JS-0355 Cn1ccnc1SCC(=O)Nc2cccc(c2Cl)Cl JS-0356 c1cc(c(c(c1)Cl)Cl)NC(=O)CSCc2ccc(cc2)Cl JS-0357 c1cc(ccc1N2C(=O)CC(C2=O)Sc3ccc(cc3)Cl)I JS-0359 COc1ccc(c2c1cccc2)/C=C/C(=O)O JS-035C CCc1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl JS-0360 CCc1ccc(cc1)NC(=O)CSc2ccc(cc2)C JS-0361 c1cc(ccc1N2C(=O)CC(C2=O)N3CCCCC3)I JS-0363 c1cc(ccc1N2C(=O)CC(C2=O)N3CCOCC3)I JS-0364 Cc1ccc(cc1Cl)NC(=O)CN2CCOCC2 JS-0365 Cc1ccc(cc1)SC2CC(=O)N(C2=O)c3ccc(cc3)I JS-0366 c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3cccc(c3Cl)Cl JS-0367 Cc1ccc(cc1)SC2CC(=O)N(C2=O)c3ccc(cc3)[N+](=O)[O-] JS-0368 c1cc(ccc1N2C(=O)CC(C2=O)Sc3ccc(cc3)Cl)[N+](=O)[O-] JS-0369 c1cc2c(cc1/C=C/C(=O)O)OCCO2 JS-036C c1ccc(cc1)CNC2CC(=O)N(C2=O)c3ccc(cc3)I JS-0371 Cc1ccc(cc1)C(=O)O/N=C/c2ccc3c(c2)OCO3 JS-0372 c1cc(ccc1C(=O)O/N=C/c2ccc3c(c2)OCO3)[N+](=O)[O-] JS-0373 CCc1ccc(cc1)NC(=O)CN2CCOCC2 JS-0374 Cc1cccc(c1)SCC(=O)Nc2ccc(cc2)C3CCCCC3 JS-0375 c1ccc(c(c1)C(=O)O/N=C/c2ccc3c(c2)OCO3)Cl JS-0376 c1cc(ccc1C2CCCCC2)NC(=O)CSc3ccc(cc3)Cl JS-0377 CCc1ccc(cc1)NC(=O)C(=O)NCc2ccccc2 JS-0378 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(cc2)C3CCCCC3 JS-0379 c1ccc(cc1)Oc2cccc(c2)/C=C/C(=O)O JS-037C c1cc(ccc1C2CCCCC2)NC(=O)CN3CCOCC3 JS-0380 c1ccc(cc1)CNC(=O)C(=O)Nc2ccc(cc2)C3CCCCC3 JS-0383 CCc1ccc(cc1)NC(=O)CSc2ncccn2 JS-0384 CCc1ccc(cc1)NC(=O)CSc2nncn2C JS-0386 Cc1ccc(cc1)C(=O)O/N=C/c2ccc(cc2)Cl JS-0387 c1ccc(c(c1)NC(=O)CNCc2ccc(cc2)Cl)[N+](=O)[O-] JS-0388 c1cc(ccc1/C=N/OC(=O)c2ccc(cc2)[N+](=O)[O-])Cl JS-0389 c1cc(ccc1/C=C/C(=O)O)OC(F)(F)F JS-038C CCc1ccc(cc1)NC(=O)CSCc2ccc(cc2)Cl JS-0390 Cc1cc(cnc1NCc2ccccc2O)Br JS-0393 Cc1ccc(cc1Br)NCc2ccccc2O JS-0394 c1ccc(c(c1)C(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccc(cc3)Br)Cl JS-0395 CCCCNC(=O)Nc1ccc(c(c1)C#N)C JS-0396 c1cc(ccc1SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl JS-0397 Cn1ccnc1SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F JS-0398 CSc1ccc(cc1)/C=C/C(=O)O JS-039C CCc1ccc(cc1)NC(=O)C(=S)NC2CCCCC2 JS-0400 Cc1ccc(cc1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F JS-0401 c1cnc(nc1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F JS-0402 CCc1ccc(cc1)NC(=O)C[NH+]2CCN(CC2)C.[Cl-] JS-0403 c1cc(ccc1Cc2ccc(cc2)NC(=O)CN3CCCCC3)NC(=O)CN4CCCCC4 JS-0404 Cc1cc(ccc1Br)NC(=O)CN2CCOCC2 JS-0407 Cc1cccc(c1)SCC(=O)Nc2ccc(cc2)F JS-0408 Cn1ccnc1SCC(=O)Nc2ccccc2C#N JS-0409 CCCOc1ccc(cc1)/C=C/C(=O)O JS-040C c1ccc(c(c1)NC(=O)CSc2ccc(cn2)[N+](=O)[O-])Br JS-0410 c1cnc(nc1)SCC(=O)Nc2cc(c(cc2F)F)F JS-0411 c1cnc(nc1)SCC(=O)Nc2ccc(cc2)F JS-0412 CCOc1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl JS-0413 Cn1ccnc1SCC(=O)Nc2ccc(c(c2)Cl)F JS-0414 CCCCc1ccc(cc1)NC(=O)CSc2nncn2C JS-0415 c1cc(ccc1Cc2ccc(cc2)NC(=O)CN3CCOCC3)NC(=O)CN4CCOCC4 JS-0416 c1c(cc(cc1Cl)Cl)NC(=O)CN2CCOCC2 JS-0417 CCc1ccc(cc1)NC(=O)CSc2nnnn2C JS-0418 COc1cc(c(cc1)/C=N/c2c(cc(cc2)Cl)SSc3c(ccc(c3)Cl)/N=C/c4c(cc(cc4)OC)O)O JS-0419 CC(C)Cc1ccc(cc1)/C=C/C(=O)O JS-041C c1cc(ccc1/C=N/NC(=S)Nc2ccc(cc2F)F)C#N JS-0421 CCC(C)c1ccc(cc1)NC(=O)CN2CCOCC2 JS-0422 Cc1cc(cnc1NC(=S)Nc2ccc(cc2F)F)Br JS-0423 c1cc(c(cc1Br)NC(=O)CN2CCOCC2)Br JS-0424 Cc1ccc(cc1)SCC(=O)Nc2ccccc2C#N JS-0426 c1ccc(c(c1)C#N)NC(=O)CN2CCOCC2 JS-0428 c1cc(ccc1Cc2ccc(cc2)NC(=O)CN3CCCC3)NC(=O)CN4CCCC4 JS-0429 c1ccc(cc1)c2ccc(cc2)/C=C/C(=O)O JS-042C Cn1ccnc1SCC(=O)Nc2ccc(c(c2)C(F)(F)F)Cl JS-0430 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)C(F)(F)F)Cl)Cl JS-0431 Cc1cc(ccc1NC(=O)CSc2nncn2C)Br JS-0432 c1cc(ccc1NC(=O)/C=C/C(=O)O)OC(F)(F)F JS-0433 Cc1ccc(cc1)SC2CC(=O)N(C2=O)c3ccc(cc3)OC(F)(F)F JS-0434 c1cc(sc1)C(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccc(c(c3)Cl)Cl JS-0435 CCOc1ccc(cc1)NC(=O)CSc2nnc(s2)C JS-0437 CCOc1ccc(cc1)NC(=O)CSc2nccn2C JS-0438 c1cc(ccc1N2C(=O)CC(C2=O)Sc3ccc(cc3)Cl)OC(F)(F)F JS-0439 CCOc1ccc(cc1)NC(=O)CSc2ncccn2 JS-0440 CCOc1ccc(cc1)NC(=O)CSCc2c(c(c(c(c2C)C)C)C)C JS-0441 CCOc1ccc(cc1)NC(=O)CSc2nncn2C JS-0442 CCOc1ccc(cc1)NC(=O)CNCc2ccccc2 JS-0443 CCOc1ccc(cc1)NC(=O)CN2CCOCC2 JS-0444 CCOc1ccc(cc1)NC(=O)C(=S)NCc2ccco2 JS-0445 CCOc1ccc(cc1)NC(=O)CSc2ccc(cc2)C JS-0446 c1cc(cc(c1)Cl)NC(=O)CSc2ccc(cc2)Cl JS-0447 Cc1ccc(cc1)SCC(=O)Nc2cccc(c2)Cl JS-0448 c1ccc(cc1)CNC(=S)C(=O)Nc2cccc(c2)Cl JS-0449 c1cc(ccc1C(=O)NN)F JS-044C c1cc(cc(c1)Cl)NC(=O)CN2CCOCC2 JS-0450 c1cc(cc(c1)Cl)NC(=O)CSc2ncccn2 JS-0451 Cc1c(c(c(c(c1C)C)CSCC(=O)Nc2cccc(c2)Cl)C)C JS-0452 Cn1ccnc1SCC(=O)Nc2cccc(c2)Cl JS-0453 Cc1nnc(s1)SCC(=O)Nc2cccc(c2)Cl JS-0454 Cn1cnnc1SCC(=O)Nc2cccc(c2)Cl JS-0455 c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3cccc(c3)Cl JS-0456 c1ccc(cc1)CNC(=O)C(=O)Nc2cccc(c2)Cl JS-0457 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)c3ccc(cc3)C JS-0458 Cc1cccc(c1)SCC(=O)Nc2cccc(c2)Cl JS-0459 c1cc(c(cc1NCC(=O)NN)Cl)F JS-045C CCOc1ccc(cc1)NC(=O)CSc2cccc(c2)C JS-0460 Cc1cccc(c1)SCC(=O)Nc2ccccc2[N+](=O)[O-] JS-0461 CCCCCCCCCC(=O)Oc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)C JS-0462 Cc1cccc(c1)SCC(=O)Nc2ccc3c(c2)OCCO3 JS-0463 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)Cc3ccccc3 JS-0464 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)C(C)(C)C JS-0465 c1cc(cc(c1)Cl)NC(=O)CSCCSCC(=O)Nc2cccc(c2)Cl JS-0466 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)/C=C/c3ccccc3 JS-0467 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)c3ccc(cc3)C(C)(C)C JS-0468 c1ccc2cc(ccc2c1)C(=O)/C=C/c3ccc(cc3)OC(=O)c4cccs4 JS-0469 c1cc(ccc1SCC(=O)NN)Cl JS-046C COc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)c3cccs3 JS-0470 c1ccc2cc(ccc2c1)C(=O)/C=C/c3ccc(cc3)OC(=O)c4ccco4 JS-0471 c1cc(sc1)C(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccc(cc3)Cl JS-0472 c1cc(oc1)C(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccc(cc3)F JS-0473 Cc1ccc(c(c1)C)C(=O)/C=C/c2ccc(cc2)OC(=O)c3cccs3 JS-0475 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)c3cccs3 JS-0476 c1cc(cc(c1)Cl)NC(=O)C(=S)NCc2ccco2 JS-0477 CC(C)(C)C(=O)Oc1ccc(cc1)/N=C/c2ccc(cc2)OC JS-0478 c1cc(c(cc1F)F)NCC(=O)NN JS-047C CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)/N=C/c3ccc4c(c3)OCO4 JS-0480 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)/N=C/c3cccc(c3)[N+](=O)[O-] JS-0481 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)/N=C/c3ccc(cc3)[N+](=O)[O-] JS-0482 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)/N=C/c3cccs3 JS-0483 c1ccc(c(c1)C(=O)Oc2ccc(cc2)/N=C/c3cccs3)Cl JS-0484 c1ccc(cc1)CC(=O)Oc2ccc(cc2)/N=C/c3cccs3 JS-0485 CC(C)(C)C(=O)Oc1ccc(cc1)/N=C/c2cccc(c2)[N+](=O)[O-] JS-0486 CC(C)(C)C(=O)Oc1ccc(cc1)/N=C/c2ccc3c(c2)OCO3 JS-0487 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)/N=C/c3ccc(cc3)Cl JS-0489 c1cc(cc(c1)[N+](=O)[O-])NCC(=O)NN JS-048C Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C3SCCS3 JS-0490 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)C3SCCS3 JS-0491 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)/C=N/c3ccc(c(c3)Cl)F JS-0492 c1cc(ccc1/C=N/c2ccc(cc2)Cl)OS(=O)(=O)c3ccc(cc3)Cl JS-0493 c1ccc(cc1)SCC(=O)N/N=C/c2cc(ccc2Cl)[N+](=O)[O-] JS-0494 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)/C=N/c3cccs3 JS-0495 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)/C=N/c3ccc(c(c3)OC)OC JS-0496 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)/C=N/c3ccc(c(c3)[N+](=O)[O-])F JS-0497 CS(=O)(=O)Oc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Cl JS-0499 c1cc(cc(c1)/N=C/c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F JS-0500 CS(=O)(=O)Oc1ccc(cc1)/C=N/c2cccc(c2)C(F)(F)F JS-0501 c1ccc(cc1)SCC(=O)N/N=C/c2cc3c(cc2[N+](=O)[O-])OCO3 JS-0502 c1cc(ccc1/C=N\c2ccc(cc2)F)OS(=O)(=O)c3ccc(cc3)Cl JS-0504 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OS(=O)(=O)C JS-0505 CS(=O)(=O)Oc1ccc(cc1)/C=C\C(=O)c2ccc3ccccc3c2 JS-0506 CC(C)c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)C JS-0507 COc1ccc(cc1/C=C\C(=O)c2ccc(cc2)OS(=O)(=O)C)Br JS-0508 CS(=O)(=O)Oc1ccc(cc1)C(=O)/C=C/c2cccs2 JS-0509 c1c(cc(cc1Cl)Cl)N2C(=O)C=CC2=O JS-050C COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)C JS-0510 CS(=O)(=O)Oc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)F JS-0511 CS(=O)(=O)Oc1ccc(cc1)C(=O)/C=C/c2ccc(cc2Cl)Cl JS-0512 c1ccc(cc1)CC(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccc(cc3)F JS-0513 c1cc(cc(c1)C(F)(F)F)C(=O)Oc2ccc(cc2)C3SCCS3 JS-0514 COc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)Cc3ccccc3 JS-0516 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)F)OC(=O)C3CCCCC3 JS-0517 CS(=O)(=O)Oc1ccc(cc1)C(=O)/C=C/c2ccc3c(c2)OCO3 JS-0518 COc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC(=O)C3CCCCC3 JS-0519 c1cc(c(cc1F)F)N2C(=O)C=CC2=O JS-051C c1ccc(cc1)CC(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccc4ccccc4c3 JS-0520 c1ccc(cc1)CC(=O)Oc2ccc(cc2)/C=C/C(=O)c3ccc(cc3)Cl JS-0521 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)C3SCCS3 JS-0522 COc1cc(cc(c1O)[N+](=O)[O-])C2SCCS2 JS-0523 c1cc(ccc1C(=O)/C=C/c2ccc3c(c2)OCO3)OS(=O)(=O)c4ccc(cc4)Cl JS-0524 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4)Cl JS-0525 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl)F JS-0526 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl JS-0527 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl JS-0528 c1cc(ccc1/C=N/c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] JS-0529 c1cc(ccc1N2C(=O)C=CC2=O)OC(F)(F)F JS-052C c1cc(ccc1/C=C/C(=O)c2ccc(cc2)F)OS(=O)(=O)c3ccc(cc3)Cl JS-0530 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Cl)OS(=O)(=O)c3ccc(cc3)Cl JS-0531 c1ccc2cc(ccc2c1)C(=O)/C=C/c3ccc(cc3)OS(=O)(=O)c4ccc(cc4)Cl JS-0532 CCCCCC[n+]1ccccc1/C=C/c2ccc(cc2OC)OC.[I-] JS-0533 CCCCCC[n+]1ccccc1/C=C/c2ccc(cc2)N(CC)CC.[I-] JS-0534 c1c(cc(cc1Cl)Cl)NC(=O)CCC(=O)O JS-0535 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3ccc(cc3)Cl JS-0536 COc1cc(cc(c1OS(=O)(=O)C)[N+](=O)[O-])C2SCCS2 JS-0537 c1ccc(cc1)NC(=O)Oc2ccc(cc2)C3SCCS3 JS-0538 CC1(SCCS1)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl JS-0539 c1cc(ccc1N2C(=O)C=CC2=O)I JS-053C C[n+]1ccccc1/C=C/c2cc(ccc2OC)Br.[I-] JS-0540 C[n+]1ccccc1/C=C/c2ccc(cc2OC)OC.[I-] JS-0541 CCN(CC)c1ccc(cc1)/C=C/c2cccc[n+]2C.[I-] JS-0542 c1cc(ccc1NC(=O)CCC(=O)O)SSc2ccc(cc2)NC(=O)CCC(=O)O JS-0543 C[n+]1ccccc1/C=C/c2ccco2.[I-] JS-0544 CCCCCC[n+]1ccccc1/C=C/c2ccc3c(c2)OCO3.[I-] JS-0545 C[n+]1ccccc1/C=C/c2ccc(cc2)F.[I-] JS-0547 c1cc(ccc1/C=N/c2ccc(cc2F)F)OS(=O)(=O)c3ccc(cc3)Cl JS-0548 Cc1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OC(=O)c3ccco3 JS-0549 c1ccc(cc1)NC(=S)NNC(=O)C2CCCC=C2 JS-0550 C[n+]1ccccc1/C=C/C=C/c2ccc(cc2)N(C)C.[I-] JS-0551 COC(=O)CCC(=O)Nc1ccc(c(c1)[N+](=O)[O-])F JS-0552 c1ccc(cc1)CN(Cc2ccccc2)C(=O)CCC(=O)N/N=C\c3ccc(cc3)F JS-0553 c1cc(ccc1C2SCCS2)OC(=O)c3ccc(cc3)[N+](=O)[O-] JS-0554 Cc1cc(ccc1Br)N2C(=O)CCC2=O JS-0555 c1cc2c(cc1NC(=O)CCC(=O)O)OCCO2 JS-0556 c1cc(cc(c1)/N=C/c2ccc(cc2)OC(=O)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F JS-0557 c1cc(oc1)C(=O)Oc2ccc(cc2)C3SCCS3 JS-0558 c1ccc(cc1)CNC(=S)NNC(=O)CCC(=O)N(Cc2ccccc2)Cc3ccccc3 JS-0559 c1cc(ccc1N2C(=O)CCC2=O)F JS-0560 c1cc(c(cc1N2C(=O)CCC2=O)Cl)Cl JS-0561 CCOc1ccc(cc1)N2C(=O)CCC2=O JS-0562 c1cc(c(cc1F)F)N2C(=O)CCC2=O JS-0563 CCOc1ccc(cc1)NC(=O)CCC(=O)O JS-0564 CC(C)(C)c1ccc(cc1)NC(=O)CCC(=O)O JS-0565 c1cc2c(cc1N3C(=O)CCC3=O)OCCO2 JS-0566 C[n+]1ccccc1/C=C/c2ccc(c(c2OC)OC)OC.[I-] JS-0567 CC(C)(C)c1ccc(cc1)N2C(=O)CCC2=O JS-0568 c1cc(cc(c1)Cl)N2C(=O)CCC2=O JS-0569 c1ccc(cc1)/C=C/C(=O)Oc2ccc(cc2)C3SCCS3 JS-0570 c1ccc(cc1)/C=C/C(=O)O/N=C/c2ccc3c(c2)OCO3 JS-0571 c1cc(ccc1C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc4c(c3)OCO4)[N+](=O)[O-] JS-0572 CS(=O)(=O)Oc1ccc(cc1)C2SCCS2 JS-0573 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2[N+](=O)[O-])OC JS-0575 c1ccc(cc1)CC(=O)Oc2ccc(cc2)C3SCCS3 JS-0576 c1ccc(c(c1)C(=O)Oc2ccc(cc2)C3SCCS3)Cl JS-0577 CC(C)(C)c1ccc(cc1)C(=O)Oc2c(cc(cc2OC)C3SCCS3)[N+](=O)[O-] JS-0578 Cc1ccc(cc1)C(=O)Oc2c(cc(cc2OC)C3SCCS3)[N+](=O)[O-] JS-0579 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)O JS-057C c1cc(c(cc1F)F)NC(=O)CCC(=O)O JS-0580 COc1cc(cc(c1OS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-])C3SCCS3 JS-0581 COc1cc(cc(c1OC(=O)Cc2ccccc2)[N+](=O)[O-])C3SCCS3 JS-0582 CCCCc1ccc(cc1)n2c(=O)c3ccccc3nc2C(C)(C)C JS-0583 COC(=O)CCC(=O)N1CCc2c1cccc2 JS-0584 COc1cc(cc(c1OC(=O)c2ccccc2Cl)[N+](=O)[O-])C3SCCS3 JS-0585 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccc(cc3)C(C)C)C JS-0589 c1cc(ccc1SCC(=O)NNC(=S)NC2CCCCC2)Cl JS-0590 CCCCCCCCCCCCSC1CC(=O)N(C1=O)c2ccc(cc2)Br JS-0591 COc1ccc(c(c1)OC)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl JS-0592 COC(=O)CCC(=O)Nc1ccc(c(c1)Cl)Cl JS-0593 Cc1cc(ccc1Br)n2c(=O)c3ccccc3nc2C(C)(C)C JS-0595 c1cc(sc1)C(=O)NNC(=S)NC2CCCCC2 JS-0596 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)C3SCCS3)C JS-0597 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3ccc(cc3)F JS-0598 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3ccc(cc3)Br JS-0599 CCCCCCCCCCCCSCC(=O)c1ccc(cc1)OCc2ccc(c(c2)Cl)Cl JS-0602 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3ccccc3Cl JS-0606 c1ccc(c(c1)NC(=S)NNC(=O)CNc2cccc(c2)[N+](=O)[O-])Cl JS-0607 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/C=C\C(=O)c3ccc(cc3)OC)C JS-0608 Cc1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OS(=O)(=O)c3c(cc(cc3C)C)C JS-0609 Cc1cccc(c1)CC2C(=NNC2=O)C JS-060C CCCCCCCC(=O)Oc1ccc(cc1)C2SCCS2 JS-0610 CCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)C(C)C JS-0611 c1cc(ccc1C2SCCS2)OC(=O)C3CCCCC3 JS-0614 CCCCCCCCCCCCSCC(=O)Nc1ccc(cc1)C(=O)OCC JS-0618 CSc1nc(nc(n1)SC)SC JS-061C Cc1c(c(c(c(c1Br)OC(=O)c2ccc(cc2)Cl)Br)C)Br JS-0620 COc1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OS(=O)(=O)C JS-0621 COC(=O)/C=C/c1ccc(cc1)OC(=O)c2ccc(cc2)Cl JS-0622 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)/C=C\C(=O)c3ccc(cc3)OC JS-0623 Cc1cc(cc(c1)NC(=O)CSc2nccn2C)C JS-0626 Cc1cc(cc(c1)NC(=O)CSc2ccc(cc2)Cl)C JS-0627 Cc1ccc(cc1)SCC(=O)Nc2cc(cc(c2)C)C JS-0628 Cc1cc(cc(c1)NC(=O)CN2CCOCC2)C JS-0629 CCCn1c(n[nH]c1=O)c2ccc(cc2)F JS-062C Cc1cc(cc(c1)NC(=O)CSc2nnc(s2)C)C JS-0630 COc1ccc(c(c1)OC)/C=C\C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Br JS-0630A Cc1cc(cc(c1)NC(=O)CSc2nncn2C)C JS-0631 CC(C)(C)C(=O)Oc1ccc(cc1)C(=O)/C=C\c2ccc(cc2OC)OC JS-0631A Cc1cc(cc(c1)NC(=O)CSc2nnnn2c3ccccc3)C JS-0632 Cc1cc(cc(c1)NC(=O)CSc2ccccn2)C JS-0632A COC(=O)/C=C\c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Br JS-0633 Cc1cc(cc(c1)NC(=O)C(=S)NCc2ccccc2)C JS-0634 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)F JS-0634A Cc1cc(cc(c1)NC(=O)CN2CCCCC2)C JS-0635 c1cc(ccc1/C=C\C(=O)Nc2ccc(cc2)F)Cl JS-0635A CCCCCCCCCCCCSCC(=O)Nc1cc(cc(c1)C)C JS-0636 CN1CCN(CC1)C(=O)/C=C\c2ccc(cc2)Cl JS-0636A Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/C=C\C(=O)OC)C JS-0637 c1cc(ccc1/C=C\C(=O)Sc2ccc(cc2)Cl)Cl JS-0637A Cc1cc(cc(c1)NC(=O)CSCc2c(c(c(c(c2C)C)C)C)C)C JS-0638 CC(C)(C)c1ccc(cc1)NC(=O)/C=C\c2ccc(cc2)Cl JS-0638A COc1ccc(c(c1)OC)/C=C/C(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl JS-0639 Cc1ccc(cc1NC(=O)/C=C\c2ccc(cc2)Cl)F JS-0639A c1cc(ccc1/C=C/C(=O)Nc2cc(cc(c2)Cl)Cl)Cl JS-0640 Cc1cc(cc(c1)NC(=O)CSCc2ccc(cc2)Cl)C JS-0642 c1cc(ccc1NC(=O)CN2CCOCC2)F JS-0643 CCCCCCCCCCCCSCC(=O)Nc1ccc(cc1)F JS-0644 Cn1ccnc1SCC(=O)Nc2ccc(cc2)F JS-0645 Cn1cnnc1SCC(=O)Nc2ccc(cc2)F JS-0646 Cc1nnc(s1)SCC(=O)Nc2ccc(cc2)F JS-0647 c1cc(c(cc1F)F)NC(=O)CN2CCOCC2 JS-0649 c1ccc(cc1)CNC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])Cl JS-0651 c1cc(ccc1/C=C/C(=O)Sc2ccc(cc2)Cl)C#N JS-0652 c1ccc(cc1)CNC(=O)/C=C/c2ccc(cc2)C#N JS-0653 c1cc(ccc1NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])Cl)F JS-0654 CCCCCCCCCCCCSCC(=O)Nc1ccc(cc1F)F JS-0655 c1ccc(cc1)CNCC(=O)Nc2ccc(cc2)F JS-0656 c1cc(ccc1/C=C/C(=O)SC2CCCCC2)C#N JS-0657 Cc1nnc(s1)SCC(=O)Nc2ccc(cc2F)F JS-0658 CN1CCN(CC1)C(=O)/C=C/c2ccc(cc2)C#N JS-0659 c1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S JS-066C Cc1cc(ccc1Br)NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])Cl JS-0670 CNC(=S)NNC(=S)NC1CCCCC1 JS-0671 Cc1ccc(cc1)c2nc3cc(c(cc3c(=O)o2)OC)OC JS-0672 c1cc(ccc1CNCC(=O)Nc2ccc(cc2F)F)Cl JS-0673 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccc(cc2)Cl JS-0674 c1cc(cc(c1)[N+](=O)[O-])C(=O)OCc2ccc(cc2)OCc3ccc(cc3)[N+](=O)[O-] JS-0675 CCCCCCCCCCCCSc1ccc(cc1/C=N/NC(=O)CSc2ccc(cc2)Cl)[N+](=O)[O-] JS-0676 c1cc(cc(c1)[N+](=O)[O-])C(=O)Oc2ccc(cc2)C3SCCS3 JS-0677 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)Cl)OC(=O)c3cccc(c3)[N+](=O)[O-] JS-0678 c1cc(cc(c1)[N+](=O)[O-])C(=O)O/N=C/c2ccc(cc2)Cl JS-0679 CC(C)Cn1c(=O)c2ccccc2[nH]c1=S JS-067C COc1ccc(c(c1)OC)/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccc(c3)[N+](=O)[O-] JS-0680 c1ccc(cc1)CC(=O)N/N=C/c2ccc(cc2)OCc3ccc(cc3)F JS-0681 c1cc(sc1)C(=O)N/N=C/c2ccc(cc2)OCc3ccc(cc3)F JS-0682 c1cc(ccc1COc2ccc(cc2)/C=N/NC(=O)CSc3ccc(cc3)Cl)F JS-0683 COc1cc2c(cc1OC)nc(oc2=O)c3cccc(c3)[N+](=O)[O-] JS-0684 c1cc(oc1)CSc2ccc(cc2[N+](=O)[O-])/C=N/NC(=O)c3cccs3 JS-0685 c1cc(cc(c1)[N+](=O)[O-])C(=O)ON=C2CCCCCCCCCCC2 JS-0686 c1cc(cc(c1)[N+](=O)[O-])C(=O)OCc2ccc(cc2)OCc3ccc(cc3)F JS-0687 CC(C)(C)C1CCC(=NOC(=O)c2cccc(c2)[N+](=O)[O-])CC1 JS-0688 COc1cc(c(cc1OC)Br)COC(=O)c2cccc(c2)[N+](=O)[O-] JS-0689 COC(=O)c1cc(ccc1O)I JS-068C c1ccc2c(c1)c(=O)oc(n2)c3cccc(c3)[N+](=O)[O-] JS-0690 COC(=O)/C=C/c1ccc(cc1)OC(=O)c2cccc(c2)[N+](=O)[O-] JS-0691 c1cc(cc(c1)[N+](=O)[O-])C(=O)OCc2cc3c(cc2[N+](=O)[O-])OCO3 JS-0692 c1ccc(cc1)Sc2ccc(cc2/C=N\NC(=O)COc3ccc(cc3Cl)Cl)[N+](=O)[O-] JS-0693 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)Nc2ccc(cc2)F JS-0694 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)NCc2ccc(cc2)Cl JS-0695 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)N2CCCCC2 JS-0696 Cc1cc(nc(n1)SCC(=O)Nc2ccc(cc2F)F)C JS-0697 Cc1cc(cc(c1)NC(=O)CSc2nc(cc(n2)C)C)C JS-0698 CC(C)(C)c1ccc(cc1)NC(=O)/C=C/c2cc(c(cc2[N+](=O)[O-])OC)OC JS-0699 COc1ccc(c(c1OC)OC)/C=C/C(=O)c2ccc(cc2)O JS-069C CN1CCN(CC1)C(=O)/C=C/c2cc(c(cc2[N+](=O)[O-])OC)OC JS-0700 CCc1ccc(cc1)NC(=O)/C=C/C(=O)c2ccc(cc2)OCC JS-0701 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)N2CCOCC2 JS-0702 CCOc1ccc(cc1)C(=O)/C=C/C(=O)Nc2ccc(cc2)C(C)(C)C JS-0704 CCOc1ccc(cc1)C(=O)/C=C/C(=O)Nc2ccc(cc2)OC(F)(F)F JS-0705 CCOc1ccc(cc1)C(=O)/C=C/C(=O)Nc2ccc(cc2)Br JS-0706 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)Nc2cccc(c2)Cl JS-0707 CC(C)(C)c1ccc(cc1)NCc2ccccc2O JS-0708 Cc1cc(ccc1Br)NCc2ccccc2O JS-0709 c1ccc2cc(ccc2c1)C(=O)/C=C/c3ccc(cc3)O JS-070C Cc1cc(ccc1Br)NCc2ccc(cc2)C#N JS-0710 c1cc(ccc1C(=O)CSC2CCCCC2)Br JS-0711 c1ccc(c(c1)CNc2cc(cc(c2)Cl)Cl)O JS-0712 CCOc1ccc(cc1)C(=O)/C=C\C(=O)Nc2ccc(cc2)F JS-0713 c1cc(ccc1C(=O)CSCCSCC(=O)c2ccc(cc2)Cl)Cl JS-0714 Cc1cc(nc(n1)SCC(=O)c2ccc(cc2)Cl)C JS-0715 Cc1cccc(c1)SCC(=O)c2ccc(cc2)Cl JS-0716 Cc1cccc(c1)SCC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl JS-0717 COC(=O)/C=C/c1ccc(cc1)O JS-071C c1ccc(cc1)CN2CCN(CC2)C3CC(=O)N(C3=O)c4ccc(cc4)Br JS-0720 c1cc(ccc1C(=O)CSCCSCC(=O)c2ccc(cc2)F)F JS-0721 c1ccc(cc1)CN2CCN(CC2)C3CC(=O)N(C3=O)c4ccc(cc4F)F JS-0722 c1cc(ccc1C(=O)O/N=C/c2cc(ccc2SC3CCCCC3)[N+](=O)[O-])Cl JS-0723 CCC(C)c1ccc(cc1)NC(=O)/C=C/c2ccc(cc2C)C JS-0725 Cc1ccc(c(c1)C)/C=C/C(=O)NCc2ccccc2 JS-0726 Cc1ccc(c(c1)C)/C=C/C(=O)NCc2ccc(cc2)Cl JS-0728 Cc1ccc(c(c1)C)/C=C/C(=O)Nc2ccc(cc2)F JS-0729 CC(=O)c1ccc(cc1)OCc2ccc(c(c2)Cl)Cl JS-072C Cc1ccc(c(c1)C)/C=C/C(=O)NCc2cccs2 JS-0731 Cc1ccc(c(c1)C)/C=C/C(=O)Nc2cccc(c2)C(F)(F)F JS-0732 Cc1ccc(c(c1)C)/C=C/C(=O)Nc2ccccc2F JS-0733 Cc1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)Cc3ccccc3 JS-0734 c1ccc(cc1)CN(Cc2ccccc2)C(=O)CCC(=O)NCc3cccs3 JS-0735 CC(C)(C)c1ccc(cc1)NC(=O)CCC(=O)N(Cc2ccccc2)Cc3ccccc3 JS-0736 c1ccc(cc1)CN(Cc2ccccc2)C(=O)CCC(=O)Nc3ccc(cc3)F JS-0737 Cc1ccc(c(c1)C)/C=C/C(=O)Nc2ccc3c(c2)OCO3 JS-0738 c1cc(ccc1/C=N/OC(=O)C2CCCCC2)Cl JS-0739 c1ccc(cc1)CN(Cc2ccccc2)C(=O)CCC(=O)Nc3ccc4c(c3)OCO4 JS-0740 CC(C)(C)c1ccc(cc1)C(=O)O/N=C/c2ccc(cc2)Cl JS-0741 c1cc(ccc1/C=N/OC(=O)c2ccc(cc2)Cl)Cl JS-0742 c1ccc(cc1)/C=C\C(=O)O/N=C/c2ccc(cc2)Cl JS-0743 CCCCOC(=O)c1ccc(cc1)OC(=O)c2ccc(cc2)C(C)(C)C JS-0746 CCCCOC(=O)c1ccc(cc1)OC(=O)c2ccc(cc2)Cl JS-0747 CCCCOC(=O)c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Cl JS-0748 c1ccc(cc1)CNC(=O)CCC(=O)N(Cc2ccccc2)Cc3ccccc3 JS-0749 CCCCOC(=O)c1ccc(cc1)OC(=O)/C=C/c2ccccc2 JS-0750 c1ccc(cc1)CNC(=O)/C=C/c2cccc(c2)Br JS-0751 COc1ccc(c(c1)NC(=O)/C=C/c2cccc(c2)Br)OC JS-0752 c1cc(cc(c1)Br)/C=C/C(=O)Nc2ccc(cc2)F JS-0753 CCc1ccc(cc1)NC(=O)/C=C/c2cccc(c2)Br JS-0754 c1cc(cc(c1)Br)/C=C/C(=O)Nc2ccc(cc2)Cl JS-0755 Cc1ccc(c(c1)NC(=O)/C=C/c2cccc(c2)Br)OC JS-0756 Cc1ccc(cc1Cl)NC(=O)/C=C/c2cccc(c2)Br JS-0757 Cc1ccc(cc1C)NC(=O)/C=C/c2cccc(c2)Br JS-0758 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)NCc2ccc(cc2)Cl JS-0759 c1cc(ccc1COc2ccc(cc2[N+](=O)[O-])C=O)F JS-075C COc1ccc(c(c1)NC(=O)/C=C/c2cccc(c2)[N+](=O)[O-])OC JS-0760 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)Nc2ccc(cc2)F JS-0761 c1ccc(cc1)Oc2ccc(cc2)NC(=O)/C=C/c3cccc(c3)[N+](=O)[O-] JS-0762 CC(C)(C)c1ccc(cc1)NC(=O)/C=C/c2cccc(c2)[N+](=O)[O-] JS-0763 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)Nc2cccc(c2)Cl JS-0764 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)Nc2ccc(cc2)Br JS-0765 CCOc1ccc(cc1)NC(=O)/C=C/c2cccc(c2)[N+](=O)[O-] JS-0766 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)NCc2cccs2 JS-0767 Cc1ccc(cc1C)NC(=O)/C=C/c2cccc(c2)[N+](=O)[O-] JS-0768 CCCCCCCCCCCCNC(=O)/C=C/c1cccc(c1)[N+](=O)[O-] JS-0769 c1cc(ccc1C=O)OCc2ccc(c(c2)Cl)Cl JS-076C c1ccc(cc1)CNC(=O)/C=C/c2cccc(c2)[N+](=O)[O-] JS-0770 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)Sc2ccc(cc2)Cl JS-0771 c1cc(cc(c1)Br)/C=C/C(=O)Nc2cccc(c2)C(F)(F)F JS-0772 CCC(C)c1ccc(cc1)NC(=O)/C=C/c2cccc(c2)Br JS-0773 CCc1ccc(cc1)NC(=O)/C=C/c2cccc(c2)[N+](=O)[O-] JS-0774 CCCCNC(=O)/C=C/c1cccc(c1)[N+](=O)[O-] JS-0775 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCOCCO JS-0776 CCCCNC1=C(C(=O)c2ccccc2C1=O)Cl JS-0778 Cc1ccc(cc1)C(=O)O/N=C/c2ccccc2OC JS-0779 c1cc(c(cc1COc2ccc(cc2[N+](=O)[O-])C=O)Cl)Cl JS-077C CC(C)(C)c1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl JS-0781 COc1ccccc1/C=N/OC(=O)c2cccc(c2)[N+](=O)[O-] JS-0782 CCCCOC(=O)c1ccc(cc1)OS(=O)(=O)c2c(cc(cc2C)C)C JS-0783 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCOCCOC(=O)c3ccc(cc3)Cl JS-0784 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCc3cccs3 JS-0785 CCOc1ccccc1NC2=C(C(=O)c3ccccc3C2=O)Cl JS-0786 CCCCOC(=O)c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Br JS-0788 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCc3ccc(cc3)Cl JS-0789 COC(=O)c1cc(ccc1O)Br JS-078C CCCCOC(=O)c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)F JS-0790 CCN(CC)CCCNC1=C(C(=O)c2ccccc2C1=O)Cl JS-0791 COc1ccc(c(c1)NC2=C(C(=O)c3ccccc3C2=O)Cl)OC JS-0792 c1cc(cc(c1)Br)/C=C/C(=O)Nc2cc(cc(c2)Cl)Cl JS-0793 Cc1ccc(cc1NC(=O)/C=C/c2cccc(c2)[N+](=O)[O-])F JS-0794 c1ccc(cc1)C/N=C/c2cc(ccc2SC3CCCCC3)[N+](=O)[O-] JS-0795 COc1ccc(c(c1)OC)NCc2cc(ccc2O)Br JS-0796 c1cc(ccc1NCc2cc(ccc2O)Br)F JS-0798 Cc1ccc(cc1C)NCc2cc(ccc2O)Br JS-0799 CC(C)c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)O JS-079C c1cc(c(cc1[N+](=O)[O-])C=C(C#N)C#N)SC2CCCCC2 JS-0800 c1cc2c(cc1NCc3cc(ccc3O)Br)OCO2 JS-0801 c1cc(ccc1SC(=O)/C=C/c2ccc3c(c2)OCO3)Cl JS-0802 c1cc(ccc1C2CCCCC2)NCc3cc(ccc3O)Br JS-0803 Cc1ccc(nc1)NCc2cc(ccc2O)Br JS-0804 CCOc1ccc(cc1)NCc2cc(ccc2O)Br JS-0805 c1cc(ccc1NCc2cc(ccc2O)Br)Cl JS-0807 Cc1cc(ccc1Br)NCc2cc(ccc2O)Br JS-0808 Cc1ccc(cc1)SC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0809 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)F)O JS-080C c1cc(ccc1C2CCCCC2)NC(=O)/C=C/c3ccc4c(c3)OCO4 JS-0810 c1cc(ccc1NCc2cc(ccc2O)Br)Br JS-0811 c1cc(cc(c1)NCc2cc(ccc2O)Br)C(F)(F)F JS-0812 Cc1ccc(cc1Cl)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0814 c1cc(ccc1NC(=O)/C=C/c2ccc3c(c2)OCO3)F JS-0815 c1cc2c(cc1/C=C/C(=O)Nc3ccc4c(c3)OCO4)OCO2 JS-0816 c1cc(ccc1SC2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl)Cl JS-0817 c1cc(c(cc1Br)CNc2cc(cc(c2)Cl)Cl)O JS-0818 COc1ccc(c(c1)OC)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0819 c1ccc(c(c1)/C=C/C(=O)c2ccc(cc2)O)Cl JS-081C CCCCCCCCCCCCSC1CC(=O)N(C1=O)c2cc(cc(c2)Cl)Cl JS-0820 Cc1ccc(cc1)SC2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl JS-0821 c1c(cc(cc1Cl)Cl)N2C(=O)CC(C2=O)N3CCOCC3 JS-0822 Cc1cc(cnc1NCc2cc(ccc2O)Br)Br JS-0823 c1cc(ccc1CNC(=O)/C=C/c2ccc3c(c2)OCO3)Cl JS-0824 c1ccc(cc1)CN(Cc2ccccc2)CC(=O)Nc3ccc(c(c3)Cl)Cl JS-0825 CCc1ccc(cc1)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0826 Cc1cc(ccc1Br)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0827 c1ccc2c(c1)CCCN2CC(=O)Nc3cccc(c3)C(F)(F)F JS-0828 c1ccc(cc1)CN(Cc2ccccc2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-0829 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)Cl JS-0830 c1ccc2c(c1)ccn2CC(=O)Nc3cccc(c3)C(F)(F)F JS-0831 CCC(C)c1ccc(cc1)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0832 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4cc(ccc4Cl)Cl JS-0833 c1ccc(cc1)Oc2ccc(cc2)NC(=O)/C=C/c3ccc4c(c3)OCO4 JS-0834 CC(C)(C)c1ccc(cc1)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0835 c1ccc(cc1)CNC(=O)/C=C/c2ccc3c(c2)OCO3 JS-0836 Cc1ccc(cc1C)NCC(=O)Nc2ccc(c(c2)Cl)Cl JS-0837 c1ccc2c(c1)CCCN2CC(=O)Nc3ccc(c(c3)Cl)Cl JS-0838 c1ccc2c(c1)CCN2CC(=O)Nc3ccc(c(c3)Cl)Cl JS-0839 c1cc(c(cc1/C=C/2\C(=O)NC(=S)S2)[N+](=O)[O-])SC3CCCCC3 JS-0840 c1ccc(cc1)CN2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])SC4CCCCC4)/SC2=S JS-0841 c1cc(c(cc1NC(=S)Nc2cc(cc(c2)Cl)Cl)Cl)F JS-0843 CC(C)(C)c1ccc(cc1)NC(=S)Nc2ccc(c(c2)Cl)F JS-0846 c1cc(c(cc1NC(=S)Nc2ccc(cc2F)F)Cl)F JS-0848 c1cc(ccc1C(=O)/C=C/c2ccc3c(c2)OCO3)O JS-084C c1cc(ccc1NC(=S)Nc2ccc(c(c2)Cl)F)Cl JS-0850 c1ccc(c(c1)N2C(=O)/C(=C/c3cc(ccc3SC4CCCCC4)[N+](=O)[O-])/SC2=S)Cl JS-0853 c1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)F JS-0854 c1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OS(=O)(=O)c3cc(ccc3Cl)Cl JS-0855 c1ccc(cc1)C(=O)/C=C\c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Br JS-0856 c1ccc(cc1)Sc2ccc(cc2/C=C\3/C(=O)NC(=S)S3)[N+](=O)[O-] JS-0858 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/C=C\C(=O)c3ccccc3)C JS-0859 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)O JS-085C c1ccc(c(c1)N2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])SC4CCCCC4)/SC2=S)Cl JS-0860 c1ccc(cc1)CN2C(=O)/C(=C/c3cc(ccc3Sc4ccccc4)[N+](=O)[O-])/SC2=S JS-0861 CCCCCCCC(=O)Oc1ccc(cc1)C(=O)/C=C/c2cccc(c2)Cl JS-0862 COC(=O)/C=C/c1ccc(cc1)OS(=O)(=O)c2cc(ccc2Cl)Cl JS-0863 Cc1ccc(cc1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cccc(c3)Cl JS-0864 c1cc(cc(c1)Cl)/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccs3 JS-0865 c1cc(cc(c1)Cl)/C=C/C(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl JS-0866 c1ccc(c(c1)C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cccc(c3)Cl)F JS-0867 CC(C)(C)C(=O)Oc1ccc(cc1)C(=O)/C=C/c2cccc(c2)Cl JS-0868 c1ccc(c(c1)N2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl)/SC2=S)Cl JS-0869 CC1(SCCS1)c2ccc(cc2)O JS-086C c1cc(ccc1C2SCCS2)OS(=O)(=O)c3cc(ccc3Cl)Cl JS-0871 COc1cc(cc(c1OS(=O)(=O)c2cc(ccc2Cl)Cl)[N+](=O)[O-])C3SCCS3 JS-0873 c1ccc(cc1)Sc2ccc(c(c2)/C=C/3\C(=O)N(C(=S)S3)c4ccccc4Cl)[N+](=O)[O-] JS-0874 c1cc(cc(c1)Cl)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)F JS-0875 c1cc(cc(c1)Cl)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3cc(ccc3Cl)Cl JS-0876 c1cc(cc(c1)Cl)/C=C/C(=O)c2ccc(cc2)OC(=O)c3cccc(c3)[N+](=O)[O-] JS-0877 c1cc(cc(c1)Cl)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Br JS-0878 Cc1cc(no1)/N=C/c2ccccc2O JS-0879 COc1ccc(cc1/C=C/C(=O)c2ccc(cc2)O)Br JS-087C c1ccc(cc1)/C=C/C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cccc(c3)Cl JS-0880 Cc1cc(no1)NCc2ccccc2O JS-0883 Cc1ccc(cc1)C(=O)CC(C(=O)O)NCc2cccs2 JS-0884 Cc1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccc(cc2)Cl JS-0886 Cc1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cc2)C JS-0888 Cc1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cc2)Cl JS-0889 c1cc(ccc1/C=N/c2ccc(cc2F)F)OCc3ccc(cc3Cl)Cl JS-0890 c1ccc2c(c1)CCN2C3CC(=O)N(C3=O)c4cc(cc(c4)Cl)Cl JS-0891 Cc1ccc(cc1)C(=O)Oc2cc(ccc2[N+](=O)[O-])C(=O)OC JS-0894 c1cc(ccc1/C=N/c2ccc(cc2Cl)F)OCc3ccc(cc3Cl)Cl JS-0895 c1ccc(cc1)CN2C(=O)/C(=C\c3ccc(cc3)OCc4ccc(cc4Cl)Cl)/SC2=S JS-0896 COC(=O)c1ccc(c(c1)OS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] JS-0898 c1cc(ccc1/C=N/c2ccc(cc2F)Br)OCc3ccc(cc3Cl)Cl JS-0899 c1ccc(cc1)CSc2ccc(cc2C=O)[N+](=O)[O-] JS-089C c1cc(ccc1/C=N/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)OCc3ccc(cc3Cl)Cl JS-0900 Cc1ccc(cc1C#N)/N=C/c2ccccc2O JS-0901 Cc1ccc(cc1C#N)NCc2ccccc2O JS-0903 CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)F JS-0904 CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2F)F JS-0905 CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)Oc3ccccc3 JS-0906 CCOc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)Cl JS-0907 CCOc1ccc(cc1)/C=C/C(=O)N(Cc2ccccc2)Cc3ccccc3 JS-0908 Cc1ccc(c(c1)NC(=O)/C=C/c2ccc3c(c2)OCO3)OC JS-0909 c1ccc(cc1)CSc2ccc(cc2[N+](=O)[O-])C=O JS-090C CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2OC)OC JS-0910 CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)C(C)(C)C JS-0912 CCCNC(=S)Nc1ccc(c(c1)C#N)C JS-0913 CCOc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)F JS-0914 CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)C)Br JS-0915 CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc3c(c2)OCO3 JS-0916 CCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)C3CCCCC3 JS-0917 Cc1cc(no1)NC(=O)CSc2ccccn2 JS-0918 Cc1ccc(cc1C#N)NC(=S)NC2CCCCC2 JS-0919 c1c(c(cc2c1OCO2)Br)/C=C/C(=O)O JS-091C CCOc1ccc(cc1)/C=C/C(=O)SCc2ccco2 JS-0920 Cc1cc(no1)NC(=O)CN2CCOCC2 JS-0921 Cc1cc(no1)NC(=O)CSc2ccc(cc2)Cl JS-0922 Cc1cc(no1)NC(=O)CSc2nnc(s2)C JS-0923 Cc1ccc(cc1)C(=O)Oc2ccc(cc2C(=O)OC)I JS-0924 C1CCC(CC1)N2C(=O)CSC2=S JS-0925 Cc1cc(nc(n1)SCC(=O)Nc2cc(on2)C)C JS-0926 Cc1cc(no1)NC(=O)C(=S)NCc2ccccc2 JS-0927 COC(=O)c1ccc(c(c1)OC(=O)c2cccs2)[N+](=O)[O-] JS-0928 COC(=O)c1ccc(c(c1)OS(=O)(=O)c2cc(ccc2Cl)Cl)[N+](=O)[O-] JS-0929 c1c(cc(cc1C(F)(F)F)NC(=O)CCl)C(F)(F)F JS-092C COC(=O)c1ccc(c(c1)OC(=O)c2ccccc2F)[N+](=O)[O-] JS-0930 COC(=O)c1ccc(c(c1)OS(=O)(=O)c2ccc(cc2)F)[N+](=O)[O-] JS-0931 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2cc(ccc2[N+](=O)[O-])C(=O)OC)C JS-0932 COC(=O)c1cc(ccc1OS(=O)(=O)c2ccc(cc2)Br)I JS-0933 Cc1ccc(cc1C#N)/N=C/c2ccc(cc2)OCc3ccc(cc3)F JS-0934 COC(=O)c1cc(ccc1OS(=O)(=O)c2cc(ccc2Cl)Cl)I JS-0935 COC(=O)c1cc(ccc1OC(=O)c2cccs2)Br JS-0936 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl JS-0937 c1ccc(cc1)/C=C/C(=O)Oc2ccc(cc2)C(=O)/C=C/c3cccs3 JS-0938 COC(=O)c1cc(ccc1OC(=O)/C=C/c2ccccc2)Br JS-0939 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3cc(ccc3Cl)Cl JS-0940 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)F JS-0941 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)C(=O)/C=C/c3cccs3)C JS-0942 c1cc(sc1)/C=C/C(=O)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Br JS-0943 COC(=O)c1cc(ccc1OS(=O)(=O)c2ccc(cc2)F)I JS-0944 CCOc1ccc(cc1)/C=N/OC(=O)c2ccc(cc2)Cl JS-0945 CCOc1ccc(cc1)/C=N/OC(=O)c2ccc(cc2)C JS-0946 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2C(=O)OC)I)C JS-0947 COC(=O)c1cc(ccc1OS(=O)(=O)c2ccc(cc2)Cl)I JS-0948 CCOc1ccc(cc1)/C=N/OC(=O)/C=C/c2ccccc2 JS-0949 c1cc(cc(c1)Cl)NC(=O)CCl JS-094C COC(=O)c1cc(ccc1OC(=O)/C=C/c2ccccc2)I JS-0950 COC(=O)c1cc(ccc1OC(=O)c2ccc(cc2)Cl)I JS-0951 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=N/c3ccc(c(c3)Cl)F)Br JS-0952 Cc1cc(ccc1Br)NCn2c3ccccc3nn2 JS-0954 c1ccc2c(c1)nnn2CNc3ccc(c(c3)Cl)F JS-0955 c1ccc2c(c1)nnn2CNc3ccc(cc3F)F JS-0956 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])/C=N/c3cc(cc(c3)Cl)Cl JS-0957 c1cc(oc1)CSc2ccc(cc2[N+](=O)[O-])/C=N/c3cc(cc(c3)Cl)Cl JS-0958 c1cc(ccc1c2cnc(s2)Nc3ccc(cc3)F)Cl JS-0959 c1c(cc(cc1Cl)Cl)NC(=O)CCl JS-095C Cc1ccc(cc1)Sc2ccc(cc2/C=N/c3cc(cc(c3)Cl)Cl)[N+](=O)[O-] JS-0960 COc1cc(ccc1OCc2ccc(cc2)[N+](=O)[O-])/C=N/Cc3ccccc3 JS-0961 c1cc(ccc1Nc2ncc(s2)c3ccc(s3)Br)F JS-0962 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=N/c3cc(cc(c3)Cl)Cl)Br JS-0963 c1ccc(c(c1)Nc2ncc(s2)c3ccc(cc3)Cl)F JS-0964 c1cc(ccc1c2cnc(s2)Nc3cc(cc(c3)Cl)Cl)Cl JS-0965 c1cc(ccc1COc2ccc(cc2)c3cnc(s3)Nc4ccc(cc4)F)F JS-0966 c1cc(ccc1Nc2ncc(s2)c3ccc(c(c3)Cl)Cl)F JS-0967 c1cc(ccc1c2cnc(s2)Nc3ccc(cc3)Br)Cl JS-0968 c1cc(ccc1c2cnc(s2)Nc3ccc(cc3Cl)Cl)Cl JS-0969 CCOc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4cc(ccc4Cl)Cl JS-0970 c1ccc2c(c1)nc(o2)SCC(=O)Nc3ccc(c(c3)Cl)Cl JS-0972 CCOc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4)F JS-0973 CCOc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4)Br JS-0974 Cc1cc(ccc1Br)/N=C/c2ccc(c(c2)Cl)OCc3ccc(cc3)F JS-0975 CCOc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4c(cc(cc4C)C)C JS-0976 Cc1ccc(cc1)C(=O)OCCN2C(=O)c3cccc4c3c(ccc4)C2=O JS-0977 c1cc(ccc1NC(=O)CNCCO)F JS-0978 c1cc(c(cc1C(F)(F)F)NC(=O)CN2CCOCC2)Cl JS-0979 c1cc(c(cc1Cl)Cl)NC(=O)CCl JS-097C c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cc(ccc3Cl)C(F)(F)F JS-0980 c1cc(ccc1CNCC(=O)Nc2cc(ccc2Cl)C(F)(F)F)F JS-0981 c1cc(ccc1CNCC(=O)Nc2cc(ccc2Cl)C(F)(F)F)Cl JS-0982 c1cc(ccc1COc2ccc(cc2Cl)/C=C/3\C(=O)NC(=S)S3)F JS-0983 c1cc(ccc1COc2ccc(cc2Cl)/C=N\c3ccc(cc3F)F)F JS-0984 CCOc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4)Cl JS-0986 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)F)C(F)(F)F JS-0989 c1cc(c(c(c1)Cl)Cl)NC(=O)CCl JS-098C Cc1nnc(s1)SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F JS-0990 c1ccc(cc1)N2C(=O)CC(=N2)NC(=O)CSc3ccc(cc3)Cl JS-0991 c1ccc(cc1)C(=O)NC(=S)Nc2cccc(c2)C(F)(F)F JS-0992 Cn1c(nnc1SCC(=O)Nc2ccc(cc2F)F)Cc3ccccc3 JS-0994 c1cc(ccc1NC(=O)CNCCO)I JS-0995 c1cnc(nc1)SCC(=O)Nc2ccc(cc2F)F JS-0997 Cc1cc(cc(c1)NC(=O)CSc2ncccn2)C JS-0998 COc1ccc(cc1/C=N/NC(=O)c2ccc(c(c2)OC)OC)Br JS-0999 CC(C)c1ccc(cc1)NC(=O)CCl JS-099C c1ccc(cc1)CN2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl JS-1000 c1cc(ccc1NC(=O)CN2CCOCC2)I JS-1002 CCCNC(=S)NNC(=O)c1cccs1 JS-1003 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Nc3ccc4c(c3)OCCO4 JS-1004 c1cc(ccc1CNCC(=O)Nc2ccc(cc2)I)Cl JS-1005 COc1ccc(cc1)NC(=O)CSc2ccccn2 JS-1007 CC1=C(c2ccc(cc2S1(=O)=O)Cl)Cl JS-1008 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC)C(F)(F)F JS-1009 COc1ccc(cc1)NC(=O)CSc2nnnn2c3ccccc3 JS-1010 Cn1cnnc1SCC(=O)Nc2ccc(cc2)OC JS-1011 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC)Cc3ccccc3 JS-1012 COc1ccc(cc1)NC(=O)CSc2nc3ccccc3o2 JS-1013 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)F JS-1015 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)C3CCCCC3 JS-1016 c1cc(ccc1NC(=O)CN(CCO)S(=O)(=O)c2ccc(cc2)Br)F JS-1017 c1cc(ccc1C(=O)N(CCO)CC(=O)Nc2ccc(cc2)F)Cl JS-1018 CC(C)(C)c1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)F JS-1019 c1ccc(c(c1)NC(=O)CCl)[N+](=O)[O-] JS-101C CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2F)F JS-1020 Cc1cc(ccc1Br)NC(=O)/C=C/c2ccc(cc2)CC(C)C JS-1021 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)Oc3ccccc3 JS-1022 CCOc1ccc(cc1)/C=C/C(=O)Sc2ccc(cc2)Cl JS-1023 CC(C)(C)c1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)OC JS-1025 c1ccc(cc1)C(C#N)C(CC(=O)c2ccccc2)c3ccc(cc3)Cl JS-1026 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2OC)OC JS-1027 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)Cl)F JS-1028 CNC(=S)NNC(=O)c1ccc(c(c1)OC)OC JS-1029 c1ccc(cc1)NC(=O)CCl JS-102C CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc3c(c2)OCO3 JS-1030 CCOc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)CC(C)C JS-1031 Cc1nnc(s1)SCC(=O)Nc2ccc(cc2)OC JS-1032 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc3c(c2)OCCO3 JS-1033 Cn1c(nnc1S)c2ccc(c(c2)OC)OC JS-1034 CCC(C)c1ccc(cc1)NC(=O)CSc2ccccn2 JS-1035 COc1ccc(cc1)NC(=O)C(=S)NCc2ccccc2 JS-1036 c1ccc2c(c1)nnn2CNc3ccc(cc3)C4CCCCC4 JS-1038 c1cc(ccc1C(F)(F)F)NC(=O)CCl JS-103C c1ccc2c(c1)nnn2CNc3ccc(cc3F)Br JS-1040 CCC(C)c1ccc(cc1)NC(=O)CSc2ncccn2 JS-1041 CCC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C)Cc3ccccc3 JS-1042 COc1ccc(cc1)NC(=O)CSc2ncccn2 JS-1043 c1cc(ccc1SCC(=O)Nc2ccc3c(c2)OCCO3)Cl JS-1044 c1ccc(c(c1)C#N)NCn2c3ccccc3nn2 JS-1045 c1ccc2c(c1)nnn2CNc3ccc(cc3)SSc4ccc(cc4)NCn5c6ccccc6nn5 JS-1046 COc1ccc(cc1)NC(=O)C(=O)NCc2ccccc2 JS-1047 c1ccc2c(c1)nnn2CNc3cc(cc(c3)C(F)(F)F)C(F)(F)F JS-1049 c1cc(cc(c1)NC(=O)CCl)C(F)(F)F JS-104C c1ccc2c(c1)nnn2CNc3ccc(c(c3)[N+](=O)[O-])F JS-1050 COc1ccc(cc1NCn2c3ccccc3nn2)Cl JS-1051 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC)Cc3ccc(c(c3)OC)OC JS-1052 Cc1cc(nc(n1)SCC(=O)Nc2ccc(cc2)I)C JS-1053 Cc1nnc(s1)SCC(=O)Nc2ccc3c(c2)OCCO3 JS-1055 c1ccc(c(c1)C(F)(F)F)NC(=O)CCl JS-105C Cc1cc(nc(n1)SCC(=O)Nc2cccc(c2)[N+](=O)[O-])C JS-1063 Cc1nnc(s1)SCC(=O)Nc2cccc(c2)[N+](=O)[O-] JS-1065 c1cc(cc(c1)[N+](=O)[O-])NCC(=O)N/N=C/c2ccc(cc2)OCc3ccc(cc3)F JS-1067 c1cc(ccc1SCC(=O)Nc2ccc3c(c2)OCO3)Cl JS-1068 Cn1c(nnc1SCC(=O)Nc2ccc3c(c2)OCO3)C(F)(F)F JS-1069 c1ccc(cc1)CNC(=O)CCl JS-106C Cn1cnnc1SCC(=O)Nc2ccc3c(c2)OCO3 JS-1070 c1ccc(c(c1)/C=N/NC(=O)CNc2ccc(cc2)F)O JS-1071 Cn1c(nnc1SCC(=O)Nc2cccc(c2)[N+](=O)[O-])Cc3ccccc3 JS-1073 Cc1c(cco1)C(=O)N/N=C/c2cccs2 JS-1074 c1ccc(cc1)CC(=O)N/N=C/c2ccc(o2)[N+](=O)[O-] JS-1075 c1cc(c(cc1Cl)C(=O)N/N=C/c2ccc(o2)[N+](=O)[O-])Cl JS-1076 c1cc(sc1)C(=O)N/N=C/c2ccc(o2)[N+](=O)[O-] JS-1077 CCCCc1ccc(cc1)NC(=O)Cn2c3ccccc3nn2 JS-1078 c1cc(ccc1NCC(=O)N/N=C/c2cc(ccc2O)Br)F JS-1079 c1cc(ccc1CNC(=O)CCl)F JS-107C c1ccc2c(c1)C(c3ccccc3O2)C(=O)N/N=C/c4ccc(o4)[N+](=O)[O-] JS-1081 c1cc(cc(c1)[N+](=O)[O-])NCC(=O)N/N=C/c2ccc(o2)[N+](=O)[O-] JS-1082 COc1ccc(cc1OC)C(=O)N/N=C/c2ccc(o2)[N+](=O)[O-] JS-1083 Cc1c(cco1)C(=O)N/N=C/c2ccc(o2)[N+](=O)[O-] JS-1084 c1ccc(cc1)CC(=O)N/N=C/c2cccnc2 JS-1085 CC(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccc(cc2)F JS-1087 c1cc(cnc1)/C=N/NC(=O)c2cccs2 JS-1089 COc1ccc(cc1)CNC(=O)CCl JS-108C CC(C)c1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cc2)Cl JS-1090 CC(C)c1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)C JS-1091 CC(C)c1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)Oc3ccccc3 JS-1092 c1ccc(cc1)CC(=O)N/N=C/c2ccc(c(c2)[N+](=O)[O-])N3CCCC3 JS-1093 c1cc(sc1)C(=O)N/N=C/c2ccc(c(c2)[N+](=O)[O-])N3CCCC3 JS-1094 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=O)c2cccs2 JS-1095 c1cc(ccc1C2CCCCC2)C(=O)CC(C(=O)O)Sc3ccc(cc3)Cl JS-1096 c1ccc(cc1)CC(=O)N/N=C/c2cccc(c2)C(F)(F)F JS-1097 c1cc(ccc1CNC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O)Cl JS-1098 c1cc(c(cc1/C=N/O)[N+](=O)[O-])N2CCCC2 JS-1099 COc1c(cc(cc1Br)Br)C(=O)O JS-109C c1cc(ccc1C(=O)O/N=C/c2ccc(c(c2)[N+](=O)[O-])N3CCCC3)Cl JS-1102 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NCc2cccs2 JS-1103 COc1cc2c(cc1OC)nc(oc2=O)c3cccs3 JS-1107 Cc1c(cco1)C(=O)N/N=C/c2cccc(c2)C(F)(F)F JS-1108 c1cc(ccc1/C=C/C(=O)O)OCc2ccc(c(c2)Cl)Cl JS-110C c1cc(ccc1CNC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O)F JS-1110 c1cc(sc1)CNC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O JS-1111 CCCCCCCCCCNC(CC(=O)c1ccc(cc1)C2CCCCC2)C(=O)O JS-1112 c1cc(cnc1)/C=N/NC(=O)c2cc(ccc2Cl)Cl JS-1114 c1ccc(cc1)CNC(=O)C(=O)Nc2cccc(c2Cl)Cl JS-1115 c1cc(ccc1SCC(=O)N/N=C/c2ccc(o2)[N+](=O)[O-])Cl JS-1116 c1cc(ccc1/C=N/NC(=O)CSc2ccc(cc2)Cl)OCc3ccc(c(c3)Cl)Cl JS-1117 c1cc(cnc1)/C=N/NC(=O)CSc2ccc(cc2)Cl JS-1119 c1cc(c(cc1NC(=S)NNC(=O)c2ccsc2)Cl)F JS-1120 CCCCn1c(nn(c1=O)S(=O)(=O)c2ccc(cc2)Br)c3ccccc3 JS-1121 c1cc(ccc1SCC(=O)NNC(=S)Nc2ccc(c(c2)Cl)F)Cl JS-1122 c1cc(cc(c1)Cl)C(=O)N/N=C/c2cccnc2 JS-1124 c1ccc(cc1)C(=O)NNC(=S)Nc2ccc(c(c2)Cl)F JS-1125 Cc1ccc(cc1)NC(=O)CSc2nc(nc(n2)SCC(=O)Nc3ccc(cc3)C)SCC(=O)Nc4ccc(cc4)C JS-1126 c1cc(ccc1SCC(=O)NNC(=O)Nc2ccc(cc2F)F)Cl JS-1129 COc1c(cc(cc1Cl)C(=O)O)Cl JS-112C Cc1ccccc1CC2C(=NNC2=O)C JS-1132 c1cc(ccc1NC(=O)CSc2nc(nc(n2)SCC(=O)Nc3ccc(cc3)F)SCC(=O)Nc4ccc(cc4)F)F JS-1134 Cc1ccccc1Cc2c(c3c(n[nH]c3oc2=O)C)C JS-1135 CCCNC(=O)NNC(=O)c1ccc(cc1)F JS-1136 c1cc(ccc1CSC2CC(=O)N(C2=O)c3ccc(cc3)Br)Cl JS-1137 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3ccc(cc3Cl)Cl JS-1138 COc1ccc(c(c1)S(=O)(=O)Oc2ccc(cc2)C3SCCS3)OC JS-1139 CC(=O)c1ccc(cc1)OCc2ccc(cc2)F JS-113C CCOC(=O)Cn1nc(nn1)c2ccc(cc2)C JS-1140 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2ccc(cc2)C3SCCS3)C)C JS-1141 CC(C)(C)c1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)C3SCCS3 JS-1142 c1cc(ccc1CSc2ccc(cc2C3SCCS3)[N+](=O)[O-])Cl JS-1143 Cc1ccc(cc1)c2nc3ccc(cc3c(=O)o2)C JS-1145 Cc1ccc2c(c1)c(=O)oc(n2)c3cccs3 JS-1146 Cc1ccc2c(c1)c(=O)oc(n2)c3cccc(c3)C(F)(F)F JS-1147 Cc1ccc2c(c1)c(=O)oc(n2)c3ccccc3Cl JS-1148 Cc1ccc2c(c1)c(=O)oc(n2)c3ccc(cc3)Cl JS-1149 Cc1cc(c2c(c1)c(=O)oc(n2)c3ccccc3F)C JS-1150 Cc1cc(c2c(c1)c(=O)oc(n2)c3ccc(cc3)Cl)C JS-1151 Cc1ccc(cc1)c2nc3c(cc(cc3c(=O)o2)C)C JS-1152 c1cc(oc1)CNC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-1154 COc1ccc(cc1)CNC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-1155 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2c(=O)c3ccccc3oc2c4ccc(cc4)OC)C)C JS-1156 c1cc(ccc1C(=O)CC(C(=O)O)N2CCOCC2)Br JS-1157 c1cc(ccc1C(=O)CC(C(=O)O)Sc2ccc(cc2)Br)Br JS-1159 c1cc(ccc1COc2ccc(cc2)/C=C/C(=O)O)F JS-115C COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4)OC JS-1160 CC(C)(C)c1ccc(cc1)S(=O)(=O)Oc2c(=O)c3ccccc3oc2c4ccc(cc4)OC JS-1161 CCOc1ccc(cc1)NC(=S)Nc2ccc(c(c2)C#N)C JS-1163 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4cc(ccc4OC)OC JS-1164 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4Cl)Cl JS-1165 c1cc(ccc1CSC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O)Cl JS-1166 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4)F JS-1167 c1ccc(cc1)c2nc(cs2)c3ccc(cc3)Cl JS-1168 CC(=O)c1ccc(c(c1)[N+](=O)[O-])OCc2ccc(cc2)F JS-116C c1ccc(cc1)c2nc(cs2)c3ccc(cc3)OCc4ccc(c(c4)Cl)Cl JS-1170 c1cc(ccc1C2CCCCC2)C(=O)CC(C(=O)O)NC3CCCCC3 JS-1171 c1cc(ccc1C2CCCCC2)C(=O)CC(C(=O)O)N3CCCC3 JS-1173 Cc1ccc(cc1)SC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O JS-1174 CCOc1ccc(cc1)C(=O)CC(C(=O)O)N2CCCC2 JS-1175 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccco2 JS-1176 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccccc2 JS-1177 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NC2CCCCC2 JS-1178 CCOc1ccc(cc1)C(=O)CC(C(=O)O)SCc2ccc(cc2)Cl JS-1179 c1cc(ccc1C(=O)CC(C(=O)O)NC2CCCCC2)Cl JS-1181 c1cc(oc1)CNC(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1182 c1ccc(cc1)CNC(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1183 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccccc2 JS-1184 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccc(cc2)Cl JS-1185 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NC2CCCCC2 JS-1186 Cc1ccc(cc1)SC(CC(=O)c2ccc(cc2)C(C)(C)C)C(=O)O JS-1187 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)SCc2ccc(cc2)Cl JS-1188 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)N2CCCC2 JS-1189 COc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)O JS-118C CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccco2 JS-1190 c1cc(ccc1CSC(CC(=O)c2ccc(cc2)Cl)C(=O)O)Cl JS-1191 Cc1ccc(cc1)SC(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1192 c1cc(sc1)CNC(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1193 c1cc(ccc1CNC(CC(=O)c2ccc(cc2)Cl)C(=O)O)Cl JS-1194 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc3ccccc3c2C(c4ccccc4)N5CCCCC5 JS-1195 c1ccc(cc1)c2nc(cs2)c3ccc(cc3)F JS-1196 CCN(CC)CCCNC(CC(=O)c1ccc(cc1)Br)C(=O)O JS-1197 CC(=O)c1ccc(c(c1)OC)[N+](=O)[O-] JS-119C c1ccc(c(c1)/C=N/c2c(cc(cn2)C(F)(F)F)Cl)O JS-1200 c1cc(ccc1C(=O)CC(C(=O)O)SC2CCCCC2)Cl JS-1201 c1cc(ccc1C(=O)CC(C(=O)O)Nc2ccc(cc2)F)Cl JS-1202 Cc1ccc(cc1)C(=O)CC(C(=O)O)SCc2ccc(cc2)Cl JS-1203 c1cc(ccc1C2CCCCC2)C(=O)CC(C(=O)O)SC3CCCCC3 JS-1204 CCOc1ccc(cc1)C(=O)CC(C(=O)O)SC2CCCCC2 JS-1205 Cc1ccc(cc1)C(=O)CC(C(=O)O)SC2CCCCC2 JS-1206 c1cc(cnc1)CNC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-1207 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)SC2CCCCC2 JS-1208 CCOc1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cc2)C JS-1209 COc1cc(ccc1OCc2ccc(cc2)[N+](=O)[O-])C=O JS-120C c1cc(ccc1C(=O)CC(C(=O)O)Sc2ccc(cc2)Cl)Cl JS-1210 c1cc(cc(c1)[N+](=O)[O-])NC(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1211 CCN(CC)CCCNC(CC(=O)c1ccc(cc1)Cl)C(=O)O JS-1212 c1cc(cnc1)CNC(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1214 COc1ccc(cc1)CNC(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1215 c1cc(ccc1C(=O)CC(C(=O)O)NCCCO)Br JS-1216 CN1CCN(CC1)C(CC(=O)c2ccc(cc2)Cl)C(=O)O JS-1217 c1ccc(cc1)CN2CCN(CC2)C(CC(=O)c3ccc(cc3)Cl)C(=O)O JS-1218 COc1c(cc(cc1Br)Br)C(=O)OC JS-121C c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCOC(=O)c4cccc(c4)C(F)(F)F JS-1220 c1ccc(cc1)Cc2nc3ccccc3c(=O)n2c4ccc(cc4)F JS-1221 c1cc(cnc1)CNC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O JS-1223 COc1ccc(cc1)C(=O)CC(C(=O)O)NCc2cccnc2 JS-1224 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2cccnc2 JS-1225 c1cc(ccc1C(=O)CC(C(=O)O)NCCCn2ccnc2)Cl JS-1226 c1cc(ccc1C(=O)CC(C(=O)O)NCCN2CCOCC2)Cl JS-1227 c1ccc(cc1)C(c2ccccc2)NC(CC(=O)c3ccc(cc3)Cl)C(=O)O JS-1228 c1cc(ccc1C=C(C#N)C#N)OCc2ccc(cc2Cl)Cl JS-1229 CCN1C(=O)/C(=C\c2ccc(cc2)OCc3ccc(cc3)F)/SC1=S JS-1230 CCN1C(=O)/C(=C\c2cc(ccc2OC)Br)/SC1=S JS-1231 c1cc(ccc1Sc2ccc(cc2C3SCCCS3)[N+](=O)[O-])Cl JS-1232 c1cc(c(c(c1)Cl)Cl)NC(=O)CSCCCSCC(=O)Nc2cccc(c2Cl)Cl JS-1233 CCN1C(=O)/C(=C\c2cc(ccc2SC3CCCCC3)[N+](=O)[O-])/SC1=S JS-1234 CCN1C(=O)/C(=C\c2cc(ccc2SCc3ccc(cc3)Cl)[N+](=O)[O-])/SC1=S JS-1235 CCN1C(=O)/C(=C\c2ccc(c(c2)[N+](=O)[O-])OC)/SC1=S JS-1236 CCN1C(=O)/C(=C\c2cc(ccc2Sc3ccc(cc3)C)[N+](=O)[O-])/SC1=S JS-1237 CCN1C(=O)/C(=C\c2cc(ccc2Sc3ccc(cc3)Cl)[N+](=O)[O-])/SC1=S JS-1238 c1cc(ccc1C2SCCCS2)OS(=O)(=O)c3ccc(cc3)Br JS-1239 CC(=O)c1ccc(cc1)OCc2cccc3c2cccc3 JS-123C COc1ccc(cc1C2SCCCS2)Br JS-1240 Cc1cc(ccc1Br)/N=C/C=C/c2ccccc2 JS-1241 c1cc(ccc1C(=O)CC(C(=O)O)n2ccnc2)Cl JS-1243 c1cc(ccc1CNC(CC(=O)c2ccc(cc2)Cl)C(=O)O)F JS-1244 Cc1c(cco1)C(=O)NN JS-124C COc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)C3SCCCS3 JS-1250 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)C3SCCCS3)C JS-1252 c1cc(ccc1C2SCCCS2)OS(=O)(=O)c3ccc(cc3)F JS-1253 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2ccc(cc2)C3SCCCS3)C)C JS-1255 CCN1C(=O)/C(=C\c2cc(c(cc2Br)OC)OC)/SC1=S JS-1256 c1ccc(cc1)c2nc(cs2)c3ccc(cc3)Br JS-1257 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)F JS-1258 COc1c(cc(cc1Cl)C(=O)NN)Cl JS-125C Cc1ccc(cc1)C(=O)CC(C(=O)O)NCCN2CCOCC2 JS-1260 c1cc(c(cc1C(F)(F)F)NC(=O)CSCCCSCC(=O)Nc2cc(ccc2Cl)C(F)(F)F)Cl JS-1261 CC(C)(C)c1ccc(cc1)c2nc3c(cc(cc3Cl)Cl)c(=O)o2 JS-1262 c1cc(cc(c1)C(F)(F)F)c2nc3c(cc(cc3Cl)Cl)c(=O)o2 JS-1263 c1cc(ccc1c2nc3c(cc(cc3Cl)Cl)c(=O)o2)Cl JS-1264 CCOc1ccc(cc1)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-1265 c1cc(sc1)c2nc3c(cc(cc3Cl)Cl)c(=O)o2 JS-1266 c1ccc2c(c1)nnn2CNc3cc(ccc3F)F JS-1267 c1cc(c(cc1F)NCc2cc(ccc2O)Cl)F JS-1269 COc1ccc(cc1OC)C(=O)NN JS-126C CCn1c(=O)c2ccccc2nc1SCC(=O)Nc3ccc(cc3)OC JS-1270 CCOc1ccc(cc1)NC(=O)CCC(=O)N(Cc2ccccc2)Cc3ccccc3 JS-1271 Cc1nc2ccccc2c(=O)n1c3cc(ccc3F)F JS-1272 c1cc(c(c(c1NC(=O)CCCC(=O)O)F)F)F JS-1273 c1cc(c(cc1F)NC(=O)CCCC(=O)O)F JS-1274 Cc1nc2ccccc2c(=O)n1c3ccc(c(c3F)F)F JS-1275 c1ccc2c(c1)nnn2CNc3ccc(c(c3F)F)F JS-1279 Cc1nnc(s1)SCC(=O)Nc2cc(ccc2F)F JS-1282 COc1ccc(cc1)CNC(=O)c2ccccc2C(=O)Cc3ccccc3 JS-1284 c1cc(ccc1NC(=O)CCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])F)F JS-1286 c1ccc(cc1)CC(=O)c2ccccc2C(=O)N3CCCCC3 JS-1288 c1cc(ccc1N2C(=O)CSC2=S)F JS-128C Cc1cc(cnc1NC(=S)Nc2ccccc2)Br JS-1290 CCn1c(=O)c2ccccc2nc1SCC(=O)c3ccc(cc3)Cl JS-1291 CCn1c(=O)c2ccccc2nc1SCC(=O)Nc3ccccc3Br JS-1292 COc1cccc(c1)C(=O)CSc2nc3ccccc3c(=O)n2c4ccccc4 JS-1293 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)Nc4ccc(cc4)F JS-1294 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)c4ccc(cc4)OCc5ccc(c(c5)Cl)Cl JS-1295 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)c4ccc(cc4)F JS-1296 Cc1cc(ccc1Br)NCc2ccc3c(c2)OCO3 JS-1297 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NCCN2CCOCC2 JS-1298 Cc1ccc(cc1Cl)C(=O)CSc2nc3ccccc3c(=O)n2c4ccccc4 JS-1299 c1ccc(cc1)CN2C(=O)CSC2=S JS-129C CCn1c(=O)c2ccccc2nc1SCC(=O)Nc3ccc(cc3)F JS-1300 CCn1c(=O)c2ccccc2nc1SCC(=O)Nc3cccc(c3Cl)Cl JS-1301 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NCCCn2ccnc2 JS-1302 Cn1cnnc1SCC(=O)Nc2cc(ccc2F)F JS-1303 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NC2CC2 JS-1305 CCOc1ccc(cc1)C(=O)CC(C(=O)O)NCCc2c[nH]c3c2cccc3 JS-1306 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CCC(=O)O JS-1307 c1ccc2c(c1)cc([nH]2)CCNC(CC(=O)c3ccc(cc3)Br)C(=O)O JS-1308 CC(C)(C)c1ccc(cc1)/C=C/C(=O)NCCc2c[nH]c3c2cccc3 JS-1309 c1cc(c(cc1N2C(=O)C=CC2=O)[N+](=O)[O-])F JS-130C c1cc(ccc1C(=O)CC(C(=O)O)NC2CC2)Br JS-1310 c1ccc(cc1)CC(=O)c2ccccc2C(=O)NCc3cccs3 JS-1311 c1cc(ccc1C(=O)CC(C(=O)O)NC2CC2)Cl JS-1313 c1ccc(cc1)CC(=O)c2ccccc2C(=O)NCc3ccc(cc3)Cl JS-1314 c1ccc(cc1)CC(=O)c2ccccc2C(=O)NCc3ccc(cc3)F JS-1315 c1ccc(cc1)CC(=O)c2ccccc2C(=O)N3CCOCC3 JS-1318 Cc1ccc(cc1)C(=O)CC(C(=O)O)NCCc2c[nH]c3c2cccc3 JS-1319 COc1ccc(cc1N2C(=O)C=CC2=O)[N+](=O)[O-] JS-131C Cc1ccc(cc1Cl)NC(=O)CSc2ccccn2 JS-1321 c1cc(cc(c1)Br)/C=C/C(=O)NC2CC2 JS-1322 CCN(CC)CCNC1=C(C(=O)c2ccccc2C1=O)Cl JS-1323 CCN(CC)CCNC(CC(=O)c1ccc(cc1)Cl)C(=O)O JS-1324 c1ccc2c(c1)c(c[nH]2)CC/N=C/c3cc(ccc3O)Cl JS-1325 c1cc2c(cc1/C=C/C(=O)NC3CC3)OCO2 JS-1326 CCOc1ccc(cc1)/C=C/C(=O)NCCc2c[nH]c3c2cccc3 JS-1327 c1ccc(cc1)CC(=O)N/N=C/c2ccc(c(c2)[N+](=O)[O-])SC3CCCCC3 JS-1328 C#CCNC(=O)/C=C/c1ccc2c(c1)OCO2 JS-1329 COc1ccc(cc1/C=N/NC(=O)CNc2ccccc2)Br JS-1330 c1ccc2c(c1)cccc2/C=N\c3ccc(cc3)OS(=O)(=O)c4ccc(cc4)Br JS-1332 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/N=C\c3cccc4c3cccc4)C JS-1333 COc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)/N=C\c3cccc4c3cccc4 JS-1334 COc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)/N=C/c3cc(ccc3OC)Br JS-1335 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)c3ccc(cc3)Cl JS-1337 CCN1C(=O)/C(=C\c2ccc3c(c2)OCCO3)/SC1=S JS-1338 CCN1C(=O)/C(=C\c2ccc(cc2)OCc3ccc(cc3Cl)Cl)/SC1=S JS-1339 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)c3cccc(c3)OC JS-1340 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)c3ccc(cc3)Br JS-1341 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)Nc3ccc(cc3)F JS-1342 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccc(cc2)OC JS-1343 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cn2)C(F)(F)F JS-1344 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccc(cc2)F JS-1345 c1ccc(c(c1)CNc2ccc(cc2C#N)Br)O JS-1346 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/N=C/c3cc(ccc3OC)Br)C JS-1347 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)Nc3ccc(cc3F)F JS-1348 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)Nc3cccc(c3)[N+](=O)[O-] JS-1349 Cn1c(nnc1S)c2ccc(cc2)Cl JS-134C CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)Nc3cccc(c3)C(F)(F)F JS-1350 COc1cc(cc(c1OC)OC)/C=N/c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Br JS-1352 COc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)/N=C/c3cc(c(c(c3)OC)OC)OC JS-1353 Cc1cc(no1)NC(=O)CNCc2ccccc2 JS-1355 CCN1C(=O)/C(=C\c2ccc(c(c2)Cl)OCc3ccc(cc3)F)/SC1=S JS-1356 c1ccc(cc1)CC(=O)N/N=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl JS-1358 c1ccc(cc1)CC(=O)N/N=C/c2cc(ccc2SCc3ccc(cc3)Cl)[N+](=O)[O-] JS-1359 c1ccc(cc1)c2nnc(n2c3ccccc3)S JS-135C c1ccc(cc1)NCC(=O)N/N=C/c2ccc(cc2)OCc3ccc(cc3)F JS-1360 c1ccc(cc1)NCC(=O)N/N=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl JS-1361 c1ccc(cc1)NCC(=O)N/N=C/c2ccc(c(c2)[N+](=O)[O-])SC3CCCCC3 JS-1362 c1ccc(cc1)NCC(=O)N/N=C/c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl JS-1363 c1ccc(cc1)NCC(=O)N/N=C/c2ccc(c(c2)Cl)OCc3ccc(cc3)F JS-1365 Cc1ccc(cc1C)N/C(=N/C#N)/SC JS-1367 Cc1ccc(cc1C)Nc2[nH]nc(n2)/N=C/N(C)C JS-1368 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)F JS-1369 CCn1c(nnc1S)c2ccccc2 JS-136C c1cc(ccc1C2SCCS2)OCC(=O)NN JS-1371 Cc1ccc(cc1C)Nc2[nH]nc(n2)N/C=N/O JS-1372 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCc4ccc(cc4)F JS-1374 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCc4ccc(cc4)[N+](=O)[O-] JS-1375 Cc1cc(ccc1Br)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1376 Cc1c(c(c(c(c1C)C)CSc2nc3ccccc3c(=O)n2c4ccccc4)C)C JS-1377 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCc4ccc(cc4Cl)Cl JS-1378 CC(c1ccccc1)NC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-1379 CCCCn1c(nnc1S)c2ccccc2 JS-137C c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)Cl JS-1383 c1cc2c(cc1CN3CCN(CC3)CC(=O)Nc4ccc(c(c4)Cl)F)OCO2 JS-1384 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccc(cc3)Cl JS-1385 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3)Cl JS-1386 c1cc(ccc1NC(=O)CN2CCN(CC2)Cc3ccc4c(c3)OCO4)Cl JS-1387 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3)C4CCCCC4 JS-1388 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCCO4 JS-1389 c1ccc(cc1)Cc2nnc(n2c3ccc(cc3)F)S JS-138C c1cc(cc(c1)[N+](=O)[O-])NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1390 c1cc(ccc1CNC(=O)CC#N)Cl JS-1392 COc1ccc(cc1)NCC(C#N)C(=O)NCc2ccc(cc2)Cl JS-1393 Cc1cc(ccc1Br)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1396 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)F)F JS-1397 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F)Br JS-1398 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F)[N+](=O)[O-] JS-1399 c1ccc(cc1)Cc2nnc(n2Cc3ccccc3)S JS-139C Cc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F)OC JS-1400 c1cc(ccc1CNC2CC(=O)N(C2=O)c3ccc(cc3)Br)F JS-1402 c1cc(cc(c1)Cl)N2CCN(CC2)C3CC(=O)N(C3=O)c4ccc(cc4)Br JS-1403 c1cc(ccc1N2CCN(CC2)C3CC(=O)N(C3=O)c4ccc(cc4)Br)F JS-1404 CCOc1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)c3cccc(c3)Cl JS-1405 c1ccc(c(c1)NC(=O)CSCCCCCCSCC(=O)Nc2ccccc2Br)Br JS-1406 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCN(CC3)c4cccc(c4)Cl JS-1407 CCc1ccccc1NC(=O)CSCCCCCCSCC(=O)Nc2ccccc2CC JS-1408 c1cc(cc(c1)Cl)N2CCN(CC2)C(CC(=O)c3ccc(cc3)Cl)C(=O)O JS-1409 c1ccc(cc1)Cc2nnc(n2c3ccccc3)S JS-140C c1cc(c(cc1[N+](=O)[O-])C=O)SCCCCCCSc2ccc(cc2C=O)[N+](=O)[O-] JS-1410 c1cc(ccc1C(=O)CC(C(=O)O)NCc2ccc3c(c2)OCO3)Cl JS-1412 c1cc(ccc1C(=O)CC(C(=O)O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)Cl JS-1413 c1cc(c(cc1F)F)NC(=O)CSCCCCCCSCC(=O)Nc2ccc(cc2F)F JS-1414 c1cc(ccc1NC(=O)CSCCCCCCSCC(=O)Nc2ccc(cc2)F)F JS-1415 CCOc1ccc(cc1)NC(=O)CSc2nnnn2c3ccccc3 JS-1419 Cc1ccc(cc1C#N)I JS-1420 CCCCc1ccc(cc1)NCn2c3ccccc3nn2 JS-1421 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)c3cccc(c3)Cl JS-1422 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCCCn2ccnc2 JS-1424 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)NCc2ccc3c(c2)OCO3 JS-1425 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 JS-1427 c1ccc2c(c1)nnn2CN3CCN(CC3)c4cccc(c4)Cl JS-1428 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3c(c(c(c(c3F)F)F)F)F JS-1429 CCn1c(nnc1S)c2cccc(c2)Cl JS-142C Cc1ccc(cc1)SCC(=O)Nc2c(c(c(c(c2F)F)F)F)F JS-1431 c1cc(ccc1SCC(=O)Nc2c(c(c(c(c2F)F)F)F)F)Br JS-1432 c1ccc2c(c1)nnn2CN3CCN(CC3)c4ccc(cc4)F JS-1433 c1ccc2c(c1)nnn2CN3CCN(CC3)Cc4ccc5c(c4)OCO5 JS-1434 c1cc(ccc1C2CCCCC2)C(=O)CC(C(=O)O)N3CCN(CC3)c4ccc(cc4)F JS-1435 c1cc(cc(c1)Cl)N2CCN(CC2)C(CC(=O)c3ccc(cc3)C4CCCCC4)C(=O)O JS-1437 Cc1cc(cc(c1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl)C JS-1438 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CSCCCCSCC(=O)Nc2cccc(c2)[N+](=O)[O-] JS-1439 c1ccc(c(c1)NC(=O)CSCCCCSCC(=O)Nc2ccccc2Br)Br JS-1440 c1cc(c(cc1F)F)NC(=O)CSCCCCSCC(=O)Nc2ccc(cc2F)F JS-1441 CC(C)(C)c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)F)c4ccc(cc4Cl)Cl JS-1443 CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)F JS-1444 CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2OC)OC JS-1445 CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)Cl)F JS-1446 CCOc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)C(C)(C)C JS-1447 Cc1ccc(c(c1)NC(=O)CSCCCCSCC(=O)Nc2cc(ccc2OC)C)OC JS-1449 CCCCn1c(nnc1S)c2cccc(c2)Cl JS-144C Cc1ccc(cc1C)N2C(CC(=N2)c3ccc(cc3)F)c4ccc(c(c4OC)OC)OC JS-1450 CCC(C)c1ccc(cc1)NC(=O)CSCCCCSCC(=O)Nc2ccc(cc2)C(C)CC JS-1451 Cc1cc(ccc1Br)NC(=O)CSCCCCSCC(=O)Nc2ccc(c(c2)C)Br JS-1452 CCCCc1ccc(cc1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1453 Cc1cc(no1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1454 COc1ccc(cc1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1455 Cc1ccc(cc1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1456 COc1ccc(cc1)CNC(CC(=O)c2ccc(cc2)C3CCCCC3)C(=O)O JS-1457 c1cc(ccc1C(=O)CC(C(=O)O)Sc2ccc(cc2)Br)F JS-1458 c1cc(ccc1COc2ccc(cc2)/C=C/c3ccc(cc3C#N)[N+](=O)[O-])F JS-1459 CC(C)Cn1c(nnc1S)c2cccc(c2)Cl JS-145C c1cc(ccc1C(=O)CC(C(=O)O)Sc2ccc(cc2)Cl)F JS-1460 CN1CCN(CC1)C(CC(=O)c2ccc(cc2)F)C(=O)O JS-1461 COc1ccc(cc1/C=C/c2ccc(cc2C#N)[N+](=O)[O-])Br JS-1462 c1cc(sc1)CNC(CC(=O)c2ccc(cc2)F)C(=O)O JS-1463 Cc1ccc(cc1)SC(CC(=O)c2ccc(cc2)F)C(=O)O JS-1464 CC(c1ccccc1)NC(CC(=O)c2ccc(cc2)F)C(=O)O JS-1465 c1cc(ccc1CNC(CC(=O)c2ccc(cc2)F)C(=O)O)Cl JS-1466 c1cc(oc1)CNC(CC(=O)c2ccc(cc2)F)C(=O)O JS-1467 c1ccc2c(c1)c(c[nH]2)CCNC(CC(=O)c3ccc(cc3)F)C(=O)O JS-1468 COc1ccc(cc1)CNC(CC(=O)c2ccc(cc2)F)C(=O)O JS-1469 c1cc(cc(c1)Cl)N2CCN(CC2)C(CC(=O)c3ccc(cc3)F)C(=O)O JS-1470 c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3cc(cc(c3)Cl)Cl JS-1471 c1cc(ccc1SC2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl)Br JS-1474 c1ccc(cc1)N2CCN(CC2)C3CC(=O)N(C3=O)c4cc(cc(c4)Cl)Cl JS-1475 c1ccc(c(c1)NC(=O)CSc2ccc(cc2)F)Br JS-1476 Cc1ccc(cc1)c2nc3c(cc(cc3Cl)Cl)c(=O)o2 JS-1477 c1cc(ccc1C(=O)CC(C(=O)O)Sc2ccc(cc2)Br)Cl JS-1478 Cc1cc(c2c(c1)c(=O)oc(n2)c3cccc(c3)[N+](=O)[O-])C JS-1479 CCOc1ccc(cc1)c2nnc(n2c3ccccc3)S JS-147C c1ccc(c(c1)c2nc3c(cc(cc3Cl)Cl)c(=O)o2)Cl JS-1480 c1cc(ccc1c2nc3c(cc(cc3Cl)Cl)c(=O)o2)F JS-1481 c1cc(ccc1NC(=O)CSc2ccc(cc2)F)F JS-1482 c1cc(ccc1F)SCC(=O)Nc2ccc(c(c2)Cl)Cl JS-1483 c1cc(ccc1F)SCC(=O)Nc2c(c(c(c(c2F)F)F)F)F JS-1484 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CSc2ccc(cc2)F JS-1485 c1cc(cc(c1)[N+](=O)[O-])NCC(=O)N/N=C/c2ccc(cc2)F JS-1486 c1cc(cc(c1)[N+](=O)[O-])NCC(=O)N/N=C/c2ccc(cc2)OCc3ccc(cc3Cl)Cl JS-1487 c1cc(sc1)/C=N/NC(=O)CNc2ccc(cc2)F JS-1488 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)NCCc2ccc(cc2)Cl JS-1489 CCCCn1c(nnc1S)COc2ccc(cc2)Cl JS-148C CS(=O)(=O)Oc1ccc(cc1)/C=N/c2ccc(cc2)Cl JS-1490 c1cc(c(cc1C=C(C#N)C#N)[N+](=O)[O-])SC2CCCCC2 JS-1491 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C=C(C#N)C#N JS-1492 CCOC(=O)C1=C(NC(=S)NC1c2ccc(cc2)OC)C JS-1493 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)OC)C JS-1495 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)F)C JS-1496 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2)Br)C JS-1497 Cc1ccoc1C(=O)N/N=C/c2ccc(c(c2)[N+](=O)[O-])SC3CCCCC3 JS-1499 c1ccc(cc1)n2c(nnc2S)c3cccs3 JS-149C c1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)Nc4ccc(c(c4)Cl)F JS-1500 c1cc(ccc1COc2ccc(cc2)C=C(C#N)C#N)F JS-1501 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)Cl)OC(=O)c3ccc(cc3)[N+](=O)[O-] JS-1502 c1ccc2c(c1)n(c(=S)s2)CN3CCN(CC3)c4ccc(c(c4)Cl)Cl JS-1504 CCn1c(=O)c2ccccc2nc1SCC(=O)c3ccc(cc3)OCc4ccc(c(c4)Cl)Cl JS-1505 c1ccc(cc1)Sc2ccc(cc2C=C(C#N)C#N)[N+](=O)[O-] JS-1506 Cc1cccc(c1C)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1507 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)Cl)F)Cl JS-1508 Cc1cccc(c1C)NC(=O)CSc2ccc(cc2)Cl JS-1509 c1ccc(c(c1)NC(=O)CCl)F JS-150C Cn1c(nnc1SCC(=O)Nc2cccc(c2)Cl)C(F)(F)F JS-1510 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl JS-1511 c1cc(cc(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F)C(F)(F)F JS-1512 Cc1cc(ccc1Br)NC(=O)CSc2ccc(cc2)Cl JS-1513 CCCCc1ccc(cc1)NC(=O)CSc2ccccn2 JS-1514 Cn1c(nnc1SCC(=O)Nc2cccc(c2)C(F)(F)F)C(F)(F)F JS-1515 c1cc(cc(c1)Cl)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1516 Cn1c(nnc1SCC(=O)Nc2ccc(c(c2)Cl)F)C(F)(F)F JS-1517 Cn1c(nnc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl)C(F)(F)F JS-1518 Cc1cccc(c1C)NC(=O)CSc2nnc(n2C)C(F)(F)F JS-1519 c1ccc(cc1)c2nnc(n2c3ccc(cc3)F)S JS-151C Cc1cc(ccc1Br)NC(=O)CSc2nnc(n2C)C(F)(F)F JS-1520 Cc1cccc(c1C)NC(=O)CSc2nncn2C JS-1523 c1ccc(cc1)c2nc3ccccc3c(=O)n2/N=C/c4ccccc4O JS-1524 CC(C)Cc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3cccc(c3)Cl JS-1525 CC(C)Cc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)F JS-1526 CC(C)Cc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccccc3 JS-1527 Cc1cccc(c1C)NC(=O)CSc2nnnn2c3ccccc3 JS-1529 c1cc(c(cc1NC(=N)NC(=N)N)Cl)F.Cl JS-152C c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3cccc(c3)C(F)(F)F JS-1530 c1ccc2c(c1)nc(s2)SCC(=O)Nc3cccc(c3)C(F)(F)F JS-1531 c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F JS-1532 c1cc(ccc1/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)F)Cl JS-1534 c1ccc2c(c1)c(c[nH]2)CCNC(=O)/C=C/c3ccc(cc3)Cl JS-1535 c1cc(ccc1/C=C/C(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl)Cl JS-1536 COc1ccc(cc1)CNC2=C(C(=O)c3ccccc3C2=O)Cl JS-1538 c1cc(cc(c1)Cl)N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)Cl JS-1539 c1cc(cc(c1)Cl)c2nnc(n2c3ccc(cc3Cl)Cl)S JS-153C c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCc3ccc(cc3)Cl JS-1540 c1ccc(cc1)/C=C/c2nc3ccccc3c(=O)o2 JS-1541 Cc1ccc(cc1N2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl)Cl JS-1542 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)N3CCN(CC3)c4ccc(c(c4)Cl)Cl JS-1544 c1ccc2c(c1)c(=O)n(c(n2)c3cccs3)N JS-1547 CC(C)Cn1c(nnc1S)c2ccccc2 JS-154C Cn1c(nnc1SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F JS-1550 c1ccc(cc1)/C=C/c2nc3ccccc3c(=O)n2N JS-1551 c1cc(ccc1CCNC(CC(=O)c2ccc(cc2)Br)C(=O)O)Cl JS-1554 CCOC(=O)C1=C(NC(=O)NC1c2ccc3c(c2)OCO3)C JS-1555 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2)Cl)C JS-1556 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2)[N+](=O)[O-])C JS-1557 c1ccc(cc1)n2c(nnc2S)CCCOc3ccc(cc3Cl)Cl JS-155C CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)OCc3ccc(cc3)F)C JS-1560 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)CC(C)C)C JS-1561 c1ccc(cc1)c2nnc(o2)SCC(=O)Nc3ccc(c(c3)Cl)F JS-1562 c1ccc(cc1)c2nnc(o2)SCC(=O)Nc3cccc(c3)C(F)(F)F JS-1563 CC(C)(C)c1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)/N=C/c3ccc4c(c3)OCO4 JS-1564 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/N=C/c3ccc4c(c3)OCO4)C JS-1565 c1ccc(cc1)CCc2nc3ccccc3c(=O)n2c4cc(cc(c4)Cl)Cl JS-1566 c1cc(ccc1/N=C/c2ccc3c(c2)OCO3)OS(=O)(=O)c4ccc(cc4)F JS-1568 c1cc(ccc1/N=C/c2ccc3c(c2)OCO3)OS(=O)(=O)c4ccc(cc4)Cl JS-1569 c1ccc(cc1)Cn2c(nnc2S)CCCOc3ccc(cc3Cl)Cl JS-156C CC(C)c1ccc(cc1)NC(=O)CSc2ccc(cc2)F JS-1570 CC(C)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl JS-1571 CC(C)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Br JS-1572 Cc1cccc(c1C)NC(=O)CSc2nccn2C JS-1573 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/N=C/c3cccc(c3)C(F)(F)F)C JS-1576 CC(C)c1ccc(cc1)NC(=O)CSc2ccccn2 JS-1577 CC(C)c1ccc(cc1)NC(=O)CSc2nccn2C JS-1578 CC(C)c1ccc(cc1)NC(=O)CSc2nnnn2c3ccccc3 JS-1579 c1cc(c(cc1NC(=O)CNCCO)Cl)F JS-1580 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CNCCO JS-1581 CC(C)c1ccc(cc1)NC(=O)CSc2nncn2C JS-1582 CC(C)c1ccc(cc1)NC(=O)CSc2nnnn2C JS-1583 CC(C)c1ccc(cc1)NC(=O)CSc2ccc(cn2)C(F)(F)F JS-1584 CN1CCN(CC1)CC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl JS-1585 CC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1586 CCOc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl JS-1587 CCOc1ccc(cc1)/C=C/C(=O)NCCc2ccc(cc2)Cl JS-1588 CCOc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccccc3 JS-1589 c1cc(ccc1Nc2nc([nH]n2)N)Cl JS-158C CC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1590 Cc1cc(c2c(c1)c(=O)oc(n2)c3cccc(c3)C(F)(F)F)C JS-1591 CCn1c(=O)c2ccccc2nc1SCC(=O)c3ccc(c(c3)Cl)Cl JS-1593 Cc1cc(ccc1Br)NC(=O)CSc2nc3ccccc3c(=O)n2c4ccccc4 JS-1594 c1cc(sc1)/C=N/c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl JS-1595 Cc1ccc(c(c1)C)/C=C/C(=O)NC(c2ccccc2)c3ccccc3 JS-1596 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)/N=C/c3cccs3)C JS-1597 c1cc(sc1)/C=N/c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)F JS-1598 c1cc(sc1)/C=N/c2ccc(cc2)OS(=O)(=O)c3cc(ccc3Cl)Cl JS-1599 COc1ccc(c(c1OC)Cl)C#N JS-159C Cc1ccc(c(c1)C)/C=C/C(=O)Nc2ccc(cc2)I JS-1600 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)F JS-1601 Cc1ccc(c(c1)C)/C=C/C(=O)NCCc2c[nH]c3c2cccc3 JS-1602 Cc1ccc(cc1Br)NC(=O)/C=C/c2cc(c(c(c2)OC)OC)OC JS-1603 COc1cc(cc(c1OC)OC)/C=C/C(=O)Nc2ccc(c(c2)Cl)F JS-1604 COc1cc(cc(c1OC)OC)/C=C/C(=O)Nc2cc(cc(c2)Cl)Cl JS-1605 Cc1cc(ccc1Br)NC(=O)/C=C/c2ccc(c(c2OC)OC)OC JS-1606 CSc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)C/C=C/c3ccccc3 JS-1607 CSc1ccc(cc1)/C=C/C(=O)NCCc2c[nH]c3c2cccc3 JS-1608 CSc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)I JS-1609 Cc1ccc(cc1C)NC(=N)NC(=N)NN.Cl JS-160C CSc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)Cl)F JS-1610 c1ccc(cc1)/C=C/CN2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl JS-1611 c1ccc2c(c1)nnn2CNc3ccc(c(c3)Cl)Cl JS-1612 c1cc(ccc1/C=C/C(=O)Nc2ccc(cc2F)Br)Cl JS-1613 c1ccc(cc1)/C=C/CN2CCN(CC2)Cn3c4ccccc4nn3 JS-1614 COc1ccc(c(c1OC)OC)/C=C/C(=O)Nc2ccc(cc2)I JS-1615 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3ccc(cc3)Cl JS-1616 c1cc(c(cc1F)F)NC(=N)NC(=N)N.Cl JS-161C COc1cc(cc(c1O)CNc2cc(ccc2C(F)(F)F)Cl)Br JS-1620 CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2F)F JS-1621 CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)F)F JS-1622 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)F)F JS-1623 COc1cc(cc(c1O)CNc2ccc(cc2)C(F)(F)F)Br JS-1624 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F JS-1625 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2F)Br JS-1626 COc1cc(cc(c1O)CNc2ccc(c(c2)[N+](=O)[O-])Cl)Br JS-1628 Cc1ccc(cc1I)NC(=O)/C=C/c2ccc(cc2)CC(C)C JS-1629 C#CCSc1ccccc1C(=O)O JS-162C COc1cc(cc(c1O)CNc2ccc(cc2F)F)Br JS-1630 Cc1ccc(cc1NC(=O)/C=C/c2ccc(cc2)CC(C)C)F JS-1631 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)I JS-1632 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2cc(c(cc2F)F)F JS-1633 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2F)F)F JS-1634 CC(C)Cc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)C/C=C/c3ccccc3 JS-1637 COc1c(cc(cc1Cl)C(=O)OC)Cl JS-163C CC(C)Cc1ccc(cc1)/C=C/C(=O)NC(c2ccccc2)c3ccccc3 JS-1645 CC(C)Cc1ccc(cc1)/C=C/C(=O)N2CCCC2 JS-1646 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCCc2c[nH]c3c2cccc3 JS-1648 COc1cc(cc(c1O)CNc2ccc(c(c2)[N+](=O)[O-])F)Br JS-1649 CC(C)Cc1ccc(cc1)/C=C/C(=O)NC2CC2 JS-1650 CC(C)Cc1ccc(cc1)/C=C/C(=O)NC(C)c2ccccc2 JS-1651 CC(C)Cc1ccc(cc1)/C=C/C(=O)N2CCCCC2 JS-1652 CC(C)Cc1ccc(cc1)/C=C/C(=O)N2CCOCC2 JS-1653 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCc2ccccc2 JS-1654 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCc2ccco2 JS-1655 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCc2cccs2 JS-1656 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)Cl JS-1657 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)OC JS-1658 c1cc(oc1)CSc2ccc(cc2C=O)[N+](=O)[O-] JS-165C COc1cc(cc(c1O)CNc2ccc3c(c2)OCCO3)Br JS-1661 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)/C=C/c3ccc(cc3)Cl JS-1663 c1ccc(cc1)/C=C/CN2CCN(CC2)CC(=O)Nc3ccc(cc3)I JS-1664 c1ccc(cc1)/C=C/CN2CCN(CC2)CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl JS-1665 c1ccc(cc1)/C=C/CN2CCN(CC2)CC(=O)Nc3ccc(cc3F)F JS-1667 Cc1cc(cc(c1)NC(=O)CN2CCN(CC2)C/C=C/c3ccccc3)C JS-1668 c1ccc(cc1)/C=C/CN2CCN(CC2)C3CC(=O)N(C3=O)c4ccc(cc4)Br JS-1669 c1cc(oc1)CSc2ccc(cc2[N+](=O)[O-])C=O JS-166C c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)I)F JS-1670 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)C4CCCCC4)F JS-1671 CC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccc3F JS-1672 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3cccc(c3)[N+](=O)[O-])F JS-1673 c1ccc(c(c1)C#N)NC(=O)CN2CCN(CC2)c3ccccc3F JS-1674 Cc1cc(cc(c1)NC(=O)CN2CCN(CC2)c3ccccc3)C JS-1675 c1cc(ccc1c2ncc(s2)c3ccc(s3)Br)Cl JS-1676 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3F)F)F JS-1677 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)F)F JS-1678 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)F JS-1679 c1cc(ccc1F)Sc2ccc(cc2C=O)[N+](=O)[O-] JS-167C c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl JS-1680 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3c(c(c(c(c3F)F)F)F)F JS-1681 c1ccc(cc1)/C=C/CN2CCN(CC2)C3CC(=O)N(C3=O)c4ccc(cc4F)F JS-1682 c1ccc(cc1)CN2CCC(CC2)NC3=C(C(=O)c4ccccc4C3=O)Cl JS-1683 COc1ccc(c(c1OC)OC)C2CC(=NN2c3ccc(c(c3)Cl)Cl)c4ccc(cc4)F JS-1685 Cc1ccc(cc1C)NC(=O)/C=C/c2ccc(c(c2OC)OC)OC JS-1686 COc1ccc(c(c1OC)OC)/C=C/C(=O)Nc2ccc(c(c2)Cl)F JS-1687 Cc1ccc(c(c1)NC(=O)/C=C/c2ccc(c(c2OC)OC)OC)OC JS-1688 COc1ccc(c(c1OC)OC)/C=C/C(=O)Nc2ccc(cc2)CC#N JS-1689 c1cc(c(cc1C=O)[N+](=O)[O-])SC2CCCCC2 JS-168C c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F JS-1690 Cc1ccnc(c1)NCc2cc(cc(c2O)OC)Br JS-1691 COc1ccc(c(c1OC)OC)/C=C/C(=O)Nc2ccc(c(c2)Cl)I JS-1692 COc1ccc(c(c1)OC)NC(=O)/C=C/c2ccc(c(c2OC)OC)OC JS-1693 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cccc(c3)C(F)(F)F JS-1694 Cc1cc(ccc1Br)NCc2cc(cc(c2O)OC)Br JS-1695 Cc1cc(ccc1Cl)c2cnc(s2)c3ccc(cc3)Cl JS-1696 COc1ccc(cc1NCc2cc(cc(c2O)OC)Br)Cl JS-1699 c1cc(ccc1CSc2ccc(cc2C=O)[N+](=O)[O-])Cl JS-169C Cc1ccc(cc1F)NCc2cc(cc(c2O)OC)Br JS-1700 COc1cc(cc(c1O)CNc2ccc(c(c2)Cl)F)Br JS-1701 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)C(C)C JS-1702 COc1ccc(c(c1)OC)NCc2cc(cc(c2O)OC)Br JS-1703 COc1cc(cc(c1O)CNc2ccc(c(c2)Cl)Cl)Br JS-1704 CC(C)Cc1ccc(cc1)/C=C/C(=O)NC2CCCCC2 JS-1705 Cc1ccc(cc1C)NCc2cc(cc(c2O)OC)Br JS-1706 Cc1cc(no1)NCc2cc(cc(c2O)OC)Br JS-1707 COc1cc(cc(c1O)CNc2cc(cc(c2)Cl)Cl)Br JS-1708 CCOc1ccc(cc1)NCc2cc(cc(c2O)OC)Br JS-1709 COc1cc(cc(c1O)CNc2ccc(cc2)Br)Br JS-1710 COc1cc(cc(c1O)CNc2ccc(cc2)I)Br JS-1711 CC(C)Cc1ccc(cc1)/C=C/C(=O)NCc2cccc3c2cccc3 JS-1712 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)OC(F)(F)F JS-1713 Cc1c(cco1)C(=O)N/N=C/C=C/c2ccc(cc2)N(C)C JS-1716 Cc1ccc(cc1)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-1717 Cc1ccc(c(c1)C)/C=C/c2cccc[n+]2C.[I-] JS-1718 CC(C)(C)c1ccc(cc1)/C=C/c2cccc[n+]2C.[I-] JS-1719 COc1ccc(c(c1)OC)NC(=O)/C=C/c2cccc(c2)Br JS-1720 CC1(SCCS1)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl JS-1722 c1ccc(cc1)/C=C/CN2CCN(CC2)CCC(=O)c3ccc(cc3)Cl JS-1723 c1ccc(cc1)N2CCN(CC2)CCC(=O)c3ccc(cc3)Cl JS-1724 Cn1c(nnn1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl JS-1725 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl)F JS-1726 c1ccc2c(c1)cccc2CNCC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl JS-1727 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl JS-1728 c1ccc(cc1)C(c2ccccc2)NCC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl JS-1729 c1cc(c(cc1COc2ccc(cc2[N+](=O)[O-])/C=C/C(=O)O)Cl)Cl JS-172C Cc1cc(ccc1NC(=O)CSc2ccc(cc2)Br)Br JS-1730 Cc1cc(ccc1NC(=O)CSc2nnnn2C)Br JS-1733 Cc1cc(ccc1NC(=O)CSc2nnnn2c3ccccc3)Br JS-1734 Cc1cc(ccc1NC(=O)CSc2nnc(s2)C)Br JS-1735 Cc1cc(ccc1NC(=O)CN2CCN(CC2)c3cccc(c3)Cl)Br JS-1736 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3cc(ccc3Cl)C(F)(F)F)F JS-1737 c1ccc2c(c1)cccc2CNCC(=O)Nc3cc(ccc3Cl)C(F)(F)F JS-1738 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3cc(ccc3Cl)C(F)(F)F JS-1739 c1cc(cc(c1)Cl)NC(=O)CSc2ccc(cc2)Br JS-1740 c1cc(cc(c1)Cl)NC(=O)CSc2ccc(cc2)F JS-1741 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)C4CCCCC4 JS-1742 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCCO4 JS-1744 c1ccc(c(c1)CNc2ccc(c(c2)[N+](=O)[O-])F)O JS-1745 CC(C)c1ccc(cc1)NCc2ccccc2O JS-1746 c1ccc(c(c1)CNc2ccc(cc2)C3CCCCC3)O JS-1747 Cc1ccc(cc1F)NCc2ccccc2O JS-1748 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl)Cl JS-1749 c1cc(c(cc1[N+](=O)[O-])C=O)N2CCCC2 JS-174C c1cc(ccc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl)Br JS-1750 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)I JS-1751 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl JS-1752 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cc(cc(c3)Cl)Cl JS-1753 c1ccc(c(c1)CNc2c(c(c(c(c2F)F)F)F)F)O JS-1754 c1ccc(c(c1)CNc2ccc3c(c2)OCCO3)O JS-1755 c1ccc(cc1)/C=C/CN2CCN(CC2)CC(=O)Nc3ccc(cc3)C4CCCCC4 JS-1756 c1ccc(c(c1)CNc2ccc(c(c2)F)F)O JS-1757 c1ccc(c(c1)CNc2ccc(c(c2)Cl)Cl)O JS-1758 c1ccc(c(c1)CNc2ccc(c(c2)Cl)F)O JS-1759 CCCCn1c(n[nH]c1=O)c2ccccc2 JS-175C c1ccc(c(c1)CNc2nnc(s2)SCc3ccc(cc3)F)O JS-1760 c1ccc(c(c1)/C=N/c2ccc(cc2)SCc3ccc(cc3)F)O JS-1761 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3ccc(cc3F)F)F JS-1762 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCCO4)F JS-1763 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cccc(c3)Cl JS-1764 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)F JS-1765 c1ccc(c(c1)CNc2cc(ccc2Br)Br)O JS-1767 CC(C)c1ccc(cc1)NC(=O)C(=S)NCc2ccccc2 JS-1768 COc1cc(cc(c1OC)OC)/C=C/C(=O)Nc2ccc(cc2F)F JS-1769 COc1ccc(cc1)CNC(=O)/C=C/c2cc(c(c(c2)OC)OC)OC JS-1770 COc1cc(cc(c1OC)OC)/C=C/C(=O)N2CCN(CC2)c3cccc(c3)Cl JS-1771 Cc1ccc(cc1NC(=O)/C=C/c2cc(c(c(c2)OC)OC)OC)F JS-1772 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc3c(c2)OCCO3 JS-1773 COc1cc(cc(c1OC)OC)/C=C/C(=O)N2CCN(CC2)Cc3ccccc3 JS-1774 c1cc(ccc1SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F)Cl JS-1775 Cc1cc(nc(n1)SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F)C JS-1776 c1cc(ccc1F)SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F JS-1777 c1cc(ccc1CSc2nc(nc(n2)SCc3ccc(cc3)F)SCc4ccc(cc4)F)F JS-1779 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)N JS-177C Cc1ccc(cc1NC(=O)CSc2nnc(n2C)C(F)(F)F)F JS-1780 Cc1ccc(cc1NC(=O)CSc2ccc(cc2)Br)F JS-1781 c1ccc(c(c1)CNc2ccc(cc2F)F)O JS-1782 Cn1c(nnn1)SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F JS-1783 Cc1ccc(cc1NC(=O)CSc2nc(cc(n2)C)C)F JS-1784 CCCCCC[n+]1ccccc1/C=C/c2ccc(c(c2OC)OC)OC.[I-] JS-1785 Cc1ccc2c(c1)c(=O)n(c(n2)c3ccc(cc3)Cl)N JS-1787 CCC(C)n1c(=O)c2ccccc2[nH]c1=S JS-1788 C[n+]1ccccc1/C=C/c2ccc(cc2)SC.[I-] JS-1789 c1cc(ccc1N)SCC(=O)Nc2ccc(cc2)OC(F)(F)F JS-178C COc1cc2c(cc1OC)nc(oc2=O)c3ccc(cc3)Cl JS-1790 CCCCCC[n+]1ccccc1/C=C/c2ccc(cc2)SC.[I-] JS-1791 CSc1ccc(cc1)/C=N/NC(=O)CSc2ccc(cc2)Cl JS-1792 c1ccc2c(c1)cccc2CNCC(=O)Nc3cccc(c3Cl)Cl JS-1793 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cccc(c3Cl)Cl JS-1794 CC(C)(C)c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)OC)c4ccc(cc4)SC JS-1797 c1ccc(cc1)/C=C/CN2CCN(CC2)CC(=O)Nc3cccc(c3Cl)Cl JS-1798 Cc1cc(nc(n1)SCC(=O)Nc2cccc(c2Cl)Cl)C JS-1799 c1cc(c(c(c1)Cl)Cl)NC(=O)CSc2ccc(cn2)C(F)(F)F JS-1800 c1cc(c(c(c1)Cl)Cl)NC(=O)CNCc2ccc(cc2)Cl JS-1801 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)F JS-1802 CCCCc1ccc(cc1)NC(=O)CSc2nnnn2c3ccccc3 JS-1803 CCCCc1ccc(cc1)NC(=O)CSc2ncccn2 JS-1804 CCCCc1ccc(cc1)NC(=O)CSc2nc(cc(n2)C)C JS-1805 CCCCc1ccc(cc1)NC(=O)CSc2nnc(s2)C JS-1806 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)Br JS-1807 COc1ccc(cc1)C(=O)CC(c2ccc(cc2)SC)Sc3ccc(cc3)Cl JS-1808 COc1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)Sc3ccc(cc3)F JS-1809 CCCCc1ccc(cc1)NC(=O)CN2CCN(CC2)Cc3ccccc3 JS-1810 Cc1ccc(cc1NC(=O)CN2CCN(CC2)Cc3ccccc3)F JS-1811 Cn1c(nnn1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F JS-1813 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)Cl)Cl)Br JS-1814 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCO4 JS-1815 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)F JS-1816 Cc1cc(nc(n1)SCC(=O)Nc2cccc(c2)Cl)C JS-1817 Cc1cc(nc(n1)SCC(=O)Nc2cc(c(cc2F)F)F)C JS-1818 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccccc3C#N JS-1819 CCOc1ccc(cc1)NC(=O)CN2CCCc3c2cccc3 JS-1820 CCOc1ccccc1NC(=O)CN2CCN(CC2)Cc3ccccc3 JS-1821 c1ccc(cc1)N2C(CC(=N2)C3CC3)c4ccc(cc4)Cl JS-1822 Cc1cc(nc(n1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C JS-1823 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)Cl)F JS-1824 c1cc(c(cc1NC(=O)CSCCSCC(=O)Nc2ccc(c(c2)Cl)Cl)Cl)Cl JS-1825 Cn1ccnc1SCC(=O)Nc2ccc(c(c2)Cl)Cl JS-1826 c1cc(ccc1NC(=O)CN2CCN(CC2)c3ccc(cc3)F)Br JS-1827 c1cc(ccc1NC(=O)CN2CCOCC2)Br JS-1828 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccc(cc3)Br JS-1829 c1cc(ccc1N)SCC(=O)Nc2cc(ccc2F)F JS-182C c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3)Br JS-1830 c1ccc2c(c1)cccc2CNCC(=O)Nc3ccc(cc3)Br JS-1831 COc1ccc(cc1)N/C(=N/C#N)/SC JS-1832 Cc1ccnc(c1)NCc2cc(ccc2O)Br JS-1835 c1cc(cc(c1)Cl)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1836 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3)F JS-1837 c1cc(cc(c1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl)C(F)(F)F JS-1838 CCOc1ccc(cc1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1839 CCOc1ccc(cc1)/C=C/C(=O)O JS-183C Cn1ccnc1SCC(=O)Nc2cc(ccc2F)F JS-1840 c1ccnc(c1)SCC(=O)Nc2cc(ccc2F)F JS-1841 Cc1cc(nc(n1)SCC(=O)Nc2cc(ccc2F)F)C JS-1842 Cc1ccc(cc1NC(=O)CN2CCN(CC2)c3cccc(c3)Cl)F JS-1843 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F JS-1844 Cc1ccc(cc1NC(=O)CN2CCN(CC2)c3ccc(cc3)F)F JS-1845 c1cc(ccc1NC(=O)CN2CCN(CC2)c3ccc(cc3)F)F JS-1846 c1ccc(c(c1)C#N)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1847 COc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1848 CCOc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1849 Cc1ccc(c(c1)C)/C=C/C(=O)O JS-184C c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3cc(c(cc3F)F)F JS-1850 CCc1ccc(cc1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-1851 Cc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl)OC JS-1852 c1cc(c(cc1F)NC(=O)CSc2ccc(cn2)C(F)(F)F)F JS-1853 Cc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)F)F JS-1854 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)OC(F)(F)F JS-1855 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3)OC(F)(F)F JS-1856 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)F)F)F JS-1857 c1cc(cc(c1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)F)F)C(F)(F)F JS-1858 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)F)F JS-1859 c1ccc2c(c1)cccc2CNCC(=O)Nc3ccc(c(c3)F)F JS-1860 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3cccc(c3Cl)Cl JS-1861 c1cc(ccc1NC(=O)CN2CCN(CC2)c3ccc(cc3)F)OC(F)(F)F JS-1862 CCCCc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1863 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)SCc3ccc(cc3Cl)Cl JS-1864 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3cc(ccc3F)F JS-1865 c1cc(ccc1CC#N)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1866 Cc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1867 c1cc(c(c(c1)Cl)Cl)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-1868 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CCCOc3ccc(cc3Cl)Cl JS-1869 c1cc(ccc1/C=C/C(=O)O)C#N JS-186C COc1ccc(cc1NC(=O)CCCOc2ccc(cc2Cl)Cl)Cl JS-1870 c1cc(ccc1CNC(=O)CCCOc2ccc(cc2Cl)Cl)Cl JS-1871 COc1ccc(cc1)CNC(=O)CCCOc2ccc(cc2Cl)Cl JS-1872 Cc1ccc(cc1C)NC(=O)CCCOc2ccc(cc2Cl)Cl JS-1873 c1cc(ccc1NC(=O)CCCOc2ccc(cc2Cl)Cl)F JS-1874 c1cc(ccc1NC(=O)CCCOc2ccc(cc2Cl)Cl)Cl JS-1875 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CCCOc2ccc(cc2Cl)Cl JS-1876 c1cc(c(cc1Cl)Cl)OCCCC(=O)Nc2cc(cc(c2)Cl)Cl JS-1877 Cn1c(nnn1)SCC(=O)Nc2ccc(cc2)OC(F)(F)F JS-1878 c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3ccc(cc3)OC(F)(F)F JS-1879 Cn1c(nnn1)SCC(=O)Nc2ccc(cc2)SCc3ccc(cc3Cl)Cl JS-1880 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)Cl JS-1881 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)F)F JS-1882 Cc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccccn3)OC JS-1883 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)OC(F)(F)F JS-1884 CC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccn3 JS-1885 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)SCc4ccc(c(c4Cl)Cl)Cl JS-1886 COc1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)Sc3ccc(cc3)Br JS-1888 c1cc(ccc1C(CC(=O)C2CC2)Sc3ccc(cc3)Cl)Cl JS-1889 c1cc(c(cc1[N+](=O)[O-])Cl)C#N JS-188C c1ccc(c(c1)C#N)NC(=O)CN2CCN(CC2)c3ccccn3 JS-1890 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3cccc(c3Cl)Cl JS-1891 COc1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)SCCSC(CC(=O)c3ccc(cc3)OC)c4ccc(cc4)Cl JS-1892 c1ccc2c(c1)cccc2/C=C\C(=O)N3CCN(CC3)c4cccc(c4)Cl JS-1893 c1ccc2c(c1)cccc2/C=C\C(=O)NCCN3CCOCC3 JS-1894 COc1ccc(c(c1)OC)NC(=O)/C=C\c2cccc3c2cccc3 JS-1895 c1ccc2c(c1)cccc2/C=C\C(=O)Nc3cc(cc(c3)Cl)Cl JS-1896 c1ccc(cc1)Oc2ccc(cc2)NC(=O)/C=C\c3cccc4c3cccc4 JS-1897 c1ccc2c(c1)cccc2/C=C\C(=O)NCc3ccc(cc3)F JS-1898 Cc1ccc(cc1C)NC(=O)/C=C\c2cccc3c2cccc3 JS-1899 COc1ccc(cc1)CNc2cccc(c2)[N+](=O)[O-] JS-189C c1ccc2c(c1)cccc2/C=C\C(=O)Nc3ccc(cc3F)F JS-1900 Cc1cc(ccc1NC(=O)/C=C\c2cccc3c2cccc3)Br JS-1901 CC(C)c1ccc(cc1)C2CC(=NN2C(=S)N)c3ccc(cc3)Br JS-1902 Cc1c(c(c(c(c1C)C)CSc2nc3ccccc3c(=O)n2CC(C)C)C)C JS-1903 Cc1cccc(c1NC(=O)CN2CCN(CC2)c3cccc(c3)Cl)C(C)C JS-1904 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3)SCc4ccc(cc4Cl)Cl JS-1905 Cc1cccc(c1)CSc2nc3ccccc3c(=O)n2c4ccccc4 JS-1906 CCC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccn3 JS-1907 CCCOc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccccn3 JS-1909 c1cc(cc(c1)[N+](=O)[O-])NCc2ccc3c(c2)OCO3 JS-190C Cc1ccc(cc1NC(=O)CN2CCN(CC2)c3ccccn3)F JS-1910 CNC(=S)NNC(=O)Cc1ccc(c(c1)OC)OC JS-1911 CCCOc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3cccc(c3)Cl JS-1912 CCCOc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)F JS-1913 CCCOc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)Cl JS-1914 CCCOc1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)F JS-1915 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCc4ccc(cc4)Cl JS-1916 C#CCSc1nc2ccccc2c(=O)n1c3ccccc3 JS-1917 CC(C)Cn1c(=O)c2ccccc2nc1SCc3ccc(cc3Cl)Cl JS-1918 c1cc(ccc1F)SCC(=O)Nc2ccc(c(c2)F)F JS-1919 c1cc(c(cc1Br)C#N)N JS-191C c1cc(ccc1NC(=O)CSc2ccc(cc2)F)OC(F)(F)F JS-1920 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)Br)c4ccc(cc4)Cl JS-1922 Cn1cnnc1SCC(=O)Nc2ccc(c(c2)F)F JS-1923 COc1ccc(cc1)/C=C/2\C(=O)/C(=C\c3ccc(cc3)OC)/CN(C2)Cc4ccccc4 JS-1924 c1ccc(cc1)N2C(CC(=N2)c3ccc4ccccc4c3)c5cccc(c5)Cl JS-1925 c1ccc(c(c1)N2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])OCc4ccc(c(c4)Cl)Cl)/SC2=S)Cl JS-1926 Cc1cccc(c1)/C=C/C(=O)Nc2ccc(cc2F)F JS-1927 Cc1cccc(c1)/C=C/C(=O)NCc2ccc(cc2)F JS-1928 c1cc(c(cc1Br)F)N2C(=O)C=CC2=O JS-192C Cc1cccc(c1)/C=C/C(=O)Nc2ccc(c(c2F)F)F JS-1930 Cc1cccc(c1)/C=C/C(=O)Nc2ccc(c(c2)Cl)F JS-1931 Cc1cccc(c1)/C=C/C(=O)N2CCN(CC2)c3ccccc3F JS-1932 Cc1cccc(c1)/C=C/C(=O)Nc2ccc(c(c2)F)F JS-1933 Cc1cccc(c1)/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)F JS-1934 Cc1cccc(c1)/C=C/C(=O)Nc2ccc(c(c2)F)C JS-1935 C#CCSc1nnc(s1)NC(=O)c2ccc(cc2)F JS-1936 Cc1cccc(c1)/C=C/C(=O)Nc2cc(ccc2C)F JS-1937 Cc1cccc(c1)/C=C/C(=O)Nc2ccc(cc2F)Br JS-1938 COc1ccc(c(c1OC)OC)/C=C/C(=O)N2CCN(CC2)c3cccc(c3)Cl JS-1939 c1cc(ccc1NC(=S)N)F JS-193C COc1ccc(c(c1OC)OC)/C=C/C(=O)N2CCN(CC2)c3ccccn3 JS-1940 COc1ccc(c(c1OC)OC)/C=C/C(=O)NCc2ccc(cc2)Cl JS-1941 COc1ccc(cc1)CNC(=O)/C=C/c2ccc(c(c2OC)OC)OC JS-1942 c1cc(cc(c1)Br)/C=C/C(=O)N2CCN(CC2)c3cccc(c3)Cl JS-1943 c1cc(cc(c1)Br)/C=C/C(=O)Nc2ccc(cc2F)F JS-1944 c1cc(cc(c1)Br)/C=C/C(=O)NCc2ccc(cc2)F JS-1945 c1ccnc(c1)N2CCN(CC2)C(=O)/C=C/c3cccc(c3)Br JS-1946 COc1ccc(c(c1OC)OC)/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)F JS-1947 c1cc(cc(c1)Br)/C=C/C(=O)NCc2ccc(cc2)Cl JS-1948 C[n+]1ccccc1/C=C/c2ccc(cc2)c3ccccc3.[I-] JS-1949 c1cc(c(cc1Cl)Cl)NC(=S)N JS-194C c1cc(cc(c1)[N+](=O)[O-])/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)F JS-1951 c1cc(ccc1N2C(=O)/C(=C\c3ccc4c(c3)OCO4)/SC2=S)F JS-1952 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)F)F JS-1953 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)Cl JS-1954 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)Br JS-1955 c1cc(ccc1SCC(=O)Nc2cc(ccc2F)F)Br JS-1956 c1cc(ccc1N2C(=O)/C(=C\c3cc4c(cc3Br)OCO4)/SC2=S)F JS-1957 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(cc2)Cl JS-1958 Cc1cc(ccc1NC(=O)CN2CCN(CC2)c3ccccn3)Br JS-1959 c1cc(ccc1NC(=O)CSc2ccc(cc2)Br)Cl JS-1960 c1cc(ccc1NC(=O)CSc2ccc(cc2)Br)Br JS-1961 c1cc(c(cc1F)F)NC(=S)NN JS-1962 COc1ccc(cc1/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)F)Br JS-1963 c1cc(ccc1/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)Cl)OCc4ccc(c(c4)Cl)Cl JS-1964 c1ccc(cc1)CN2C/C(=C\c3sccc3)/C(=O)/C(=C/c4sccc4)/C2 JS-1965 CSc1ccc(cc1)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)F JS-1966 COc1cc(cc(c1O)CNc2ccc(cc2)F)I JS-1967 c1cc(ccc1N2C(=O)/C(=C\c3ccc4c(c3)OCCO4)/SC2=S)F JS-1968 c1ccc(cc1)CNCC(=O)Nc2ccc(cc2)Cl JS-1969 c1ccc2c(c1)cccc2/C=C/C(=O)O JS-196C CN1C/C(=C\c2cc(ccc2)Cl)/C(=O)/C(=C/c3cc(ccc3)Cl)/C1 JS-1970 CC(c1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccc(cc3)C(C)(C)C)/CN(C2)C)(C)C JS-1971 CN1C/C(=C\c2c(c(c(cc2)OC)OC)OC)/C(=O)/C(=C/c3c(c(c(cc3)OC)OC)OC)/C1 JS-1972 c1cc(cc(c1)Cl)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)F JS-1973 c1ccc(cc1)CNCC(=O)Nc2ccc(c(c2)Cl)Cl JS-1974 CCc1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccc(cc3)CC)/CN(C2)C JS-1975 CCc1ccc(cc1)/C=C\2/C(/C(=C/c3ccc(cc3)CC)/CN(C2)C)O JS-1976 c1cc(c(cc1F)NC(=O)CCC(=O)O)F JS-1977 Cc1ccc(cc1NC(=O)CCC(=O)O)F JS-1978 Cc1cc(ccc1NC(=O)CCC(=O)O)F JS-1979 c1cc(ccc1NC(=O)CCl)SCc2ccc(cc2Cl)Cl JS-197C Cc1cc(c(cc1)/C=C\2/C(=O)/C(=C/c3c(cc(cc3)C)C)/CN(C2)C)C JS-1980 CN1C/C(=C\c2ccc(cc2)SC)/C(=O)/C(=C/c3ccc(cc3)SC)/C1 JS-1981 CN1C/C(=C\c2ccc(cc2)F)/C(=O)/C(=C/c3ccc(cc3)F)/C1 JS-1982 Cc1ccc(cc1F)NC(=O)CCC(=O)O JS-1983 c1cc(c(cc1Br)F)NC(=O)CCC(=O)O JS-1984 Cc1ccc(cc1)NC(=O)C(=S)NCc2ccccc2 JS-1985 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(c(c2)F)F JS-1986 c1ccc2c(c1)CCCN2CC(=O)Nc3ccc(c(c3)Cl)F JS-1988 c1cc(c(cc1NC(=O)CCC(=O)O)F)F JS-1989 Cc1ccc(cc1)NC(=O)CCl JS-198C Cc1ccc(c(c1)NC(=O)CSc2ccc(cc2)F)OC JS-1990 Cc1ccc(c(c1)NC(=O)CSc2ccc(cc2)Br)OC JS-1991 c1ccc(cc1)CNC(=O)C(=O)Nc2ccc(c(c2)F)F JS-1992 Cc1ccc(cc1)NC(=O)C(=O)NCc2ccccc2 JS-1993 c1cc(c(cc1Cl)Cl)CSc2nnc(s2)N JS-1994 c1cc(c(cc1CSc2nnc(s2)N)Cl)Cl JS-1995 CCC(C)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Sc3ccc(cc3)SCC(=O)Nc4ccc(cc4)C(C)CC JS-1997 Cc1c(c(c(c(c1C)C)CSc2nnc(s2)N)C)C JS-1998 CN(C)/C=N/c1ccc(cc1C#N)[N+](=O)[O-] JS-199C c1cc(cc(c1)Cl)NC(=O)CSc2ccc(cc2)Sc3ccc(cc3)SCC(=O)Nc4cccc(c4)Cl JS-2000 c1cc(ccc1NC(=O)CSc2ccc(cc2)Sc3ccc(cc3)SCC(=O)Nc4ccc(cc4)OC(F)(F)F)OC(F)(F)F JS-2001 c1cc(ccc1NC(=O)CSc2nnc(s2)N)Cl JS-2002 c1cc(ccc1NC(=O)CSc2nnc(s2)N)OC(F)(F)F JS-2003 c1cc(c(cc1NC(=O)CSc2nnc(s2)N)F)F JS-2004 c1cc(cc(c1)Br)/C=C/C(=O)N2CCN(CC2)c3ccc(cc3)F JS-2005 c1ccc2c(c1)cccc2CNCC(=O)Nc3ccccc3[N+](=O)[O-] JS-2006 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccccc3[N+](=O)[O-] JS-2007 c1cc(cc(c1)Br)/C=C/C(=O)Nc2cccc(c2)I JS-2008 CN1C/C(=C\c2c3c(ccc2)cccc3)/C(=O)/C(=C/c4c5c(ccc4)cccc5)/C1 JS-2009 c1cc(ccc1F)Sc2ccc(cc2[N+](=O)[O-])C=O JS-200C c1ccc(cc1)Oc2ccc(cc2)NC(=O)CSc3ccc(cc3)Cl JS-2010 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)Oc4ccccc4 JS-2011 Cn1cnnc1SCC(=O)Nc2ccc(cc2)Oc3ccccc3 JS-2012 c1cnc(nc1)SCC(=O)Nc2ccc(cc2)Br JS-2013 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)Br JS-2014 CN1CCN(CC1)CC(=O)Nc2ccc(cc2)Oc3ccccc3 JS-2015 c1cc(ccc1C(=O)CSc2ccc(cc2)Cl)OCc3ccc(c(c3)Cl)Cl JS-2016 Cn1c(nnn1)SCC(=O)Nc2ccc(cc2)Oc3ccccc3 JS-2017 COc1ccc(c2c1cccc2)/C=C/C(=O)N3CCN(CC3)c4cccc(c4)Cl JS-2018 COc1ccc(c2c1cccc2)/C=C/C(=O)N3CCN(CC3)Cc4ccccc4 JS-2019 COc1ccc(c2c1cccc2)/C=C/C(=O)N3CCN(CC3)c4ccccn4 JS-2020 c1ccc2c(c1)CCCN2CC(=O)Nc3ccc(cc3)Br JS-2021 c1cc(c(c(c1)Cl)Cl)NC(=O)CSc2ccc(cc2)Sc3ccc(cc3)SCC(=O)Nc4cccc(c4Cl)Cl JS-2022 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)Cl)F)Sc3ccc(cc3)SCC(=O)Nc4ccc(c(c4)Cl)F JS-2023 COc1ccc(cc1)N2CCN(CC2)C(=O)/C=C/c3ccc(c4c3cccc4)OC JS-2024 COc1ccc(c2c1cccc2)/C=C/C(=O)NCc3ccc(cc3)F JS-2025 c1ccc(c(c1)NC(=O)CNCc2ccc(cc2)F)[N+](=O)[O-] JS-2026 COc1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)Oc4ccccc4 JS-2027 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CN3CCN(CC3)c4cccc(c4)Cl JS-2028 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)F)F)Sc3ccc(cc3)SCC(=O)Nc4ccc(c(c4)F)F JS-2029 Cc1cccc(c1C)NC(=O)CCl JS-202C c1ccc2c(c1)CCCN2CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl JS-2030 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CN3CCN(CC3)c4ccc(cc4)F JS-2031 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CN3CCN(CC3)c4ccccn4 JS-2032 Cn1c(nnc1SCC(=O)Nc2ccccc2[N+](=O)[O-])C(F)(F)F JS-2033 c1ccc2c(c1)CCCN2CC(=O)Nc3ccccc3[N+](=O)[O-] JS-2034 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)Cl)Cl)Sc3ccc(cc3)SCC(=O)Nc4ccc(c(c4)Cl)Cl JS-2035 Cc1cccc(c1)SCC(=O)Nc2ccc(c(c2)Cl)F JS-2036 Cc1cccc(c1)SCC(=O)Nc2cccc(c2Cl)Cl JS-2037 c1cc(ccc1CNCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl)F JS-2038 c1cc(ccc1N)SCC(=O)Nc2ccc(cc2)Br JS-2039 c1ccc(c(c1)/C=N/c2ccc(cc2)SCC(=O)Nc3ccc(c(c3)Cl)F)O JS-2040 COc1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)OC(F)(F)F JS-2042 c1cc(ccc1NC(=O)CSc2ccc(cc2)Cl)OC(F)(F)F JS-2043 c1ccc(c(c1)CNc2ccc(cc2)OC(F)(F)F)O JS-2044 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl)Br JS-2045 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccccn3)Br JS-2046 COc1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccccc3Br JS-2047 Cc1ccc(c(c1)C)N2CCN(CC2)CC(=O)Nc3ccccc3Br JS-2048 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccccc3Br JS-2049 COC(=O)c1ccccc1N2C(=O)CCC2=O JS-204C c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])Br JS-2050 Cn1ccnc1SCC(=O)Nc2ccccc2Br JS-2051 CN(C)/C=N/c1nnc(s1)SCc2ccc(cc2)Cl JS-2052 Cc1cc(ccc1Br)NC(=O)CSc2ccccn2 JS-2053 c1ccc(c(c1)NC(=O)CSc2ccc(cc2)Br)Br JS-2054 Cn1c(nnc1SCC(=O)Nc2ccccc2Br)C(F)(F)F JS-2055 Cc1cc(ccc1Br)NC(=O)CSc2ccc(cc2)Br JS-2056 Cc1cc(ccc1Br)NC(=O)CSc2ccc(cc2)F JS-2057 Cc1ccc(cc1)SCC(=O)Nc2ccc(c(c2)C)Br JS-2058 Cc1cc(ccc1Br)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] JS-2059 c1cc(cc(c1)Cl)N2CCN(CC2)CCC(=O)c3ccc(cc3)Br JS-205C Cc1ccc(c(c1)NC(=O)CSc2ccc(cc2)NCc3ccccc3O)OC JS-2060 Cc1cc(ccc1Br)NC(=O)CSc2nnnn2C JS-2061 Cc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])OC JS-2062 Cc1ccc(cc1NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])F JS-2063 c1ccc(c(c1)/C=N/c2ccc(cc2)SCC(=O)Nc3ccc(c(c3)Cl)Cl)O JS-2064 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CN3CCN(CC3)c4ccc(cc4)[N+](=O)[O-] JS-2065 c1cc(cc(c1)Cl)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] JS-2066 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl)[N+](=O)[O-] JS-2067 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])[N+](=O)[O-] JS-2068 c1cc(c(c(c1)Cl)Cl)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] JS-2069 c1cc(ccc1Nc2c3cc(ccc3ncn2)Br)F JS-2070 c1cc(ccc1CNc2c3cc(ccc3ncn2)Br)Cl JS-2071 c1cc(cc(c1)[N+](=O)[O-])Nc2c3cc(ccc3ncn2)Br JS-2072 COc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] JS-2073 Cc1cc(ccc1Br)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2074 Cc1ccc(c(c1)C)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)C)Br JS-2075 Cc1cc(ccc1Br)NC(=O)CN2CCN(CC2)c3ccccn3 JS-2076 c1cc(cc(c1)[N+](=O)[O-])N2C(=O)CCC2=O JS-2077 COc1ccc(c(c1)OC)N2C(=O)CCC2=O JS-2078 CCC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] JS-2079 CC(C)(C)OC(=O)N1CCN(CC1)CCC(=O)c2ccc3ccccc3c2 JS-207c c1cc(c(cc1N2C(=O)CCC2=O)Cl)F JS-2080 Cc1ccc(cc1C#N)N2C(=O)CCC2=O JS-2081 c1cc(ccc1CC#N)N2C(=O)CCC2=O JS-2082 c1ccc(cc1)/C=C/CN2CCN(CC2)CC(=O)Nc3ccccc3Br JS-2083 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(c(c3)Cl)Cl)Br JS-2084 COc1ccc(cc1N2C(=O)CCC2=O)Cl JS-2085 CCOC(=O)c1ccc(cc1)N2C(=O)CCC2=O JS-2086 c1cc(c(cc1N2C(=O)CCC2=O)[N+](=O)[O-])Cl JS-2087 c1ccc(c(c1)C(=O)O)N2C(=O)CCC2=O JS-2088 c1cc(ccc1CC(=O)CSc2ccc(cc2)N)Cl JS-2089 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)F JS-208C Cn1ccnc1SCC(=O)Nc2ccc(cc2)Cl JS-2090 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CSc2ccc(cc2)N JS-2091 c1cc(ccc1NC(=S)Nc2ccc(cc2)Cl)SCC(=O)Nc3ccc(cc3)Cl JS-2092 c1ccnc(c1)SCC(=O)Nc2cc(ccc2Br)Br JS-2093 c1cc(ccc1NC(=O)CN2CCN(CC2)c3ccc(cc3)F)Cl JS-2094 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2095 Cc1ccc(cc1NC(=O)/C=C/c2ccc3c(c2)OCCO3)F JS-2096 c1cc(ccc1NC(=O)/C=C/c2ccc3c(c2)OCCO3)OC(F)(F)F JS-2097 Cc1ccc(cc1F)NC(=O)/C=C/c2ccc3c(c2)OCCO3 JS-2098 c1cc(ccc1N2CCN(CC2)C(=O)/C=C/c3ccc4c(c3)OCCO4)F JS-2099 CCOc1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S JS-209C c1cc(ccc1NC(=O)/C=C/c2ccc3c(c2)OCCO3)F JS-2100 c1cc(ccc1CNC(=O)/C=C/c2ccc3c(c2)OCCO3)F JS-2101 c1cc2c(cc1/C=C/C(=O)Nc3ccc(c(c3)Cl)F)OCCO2 JS-2102 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3cc(ccc3F)F)F JS-2103 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3cc(cc(c3)Cl)F)F JS-2104 Cc1cc(cc(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F)C JS-2105 c1cc(ccc1C2CCCCC2)NC(=O)CN3CCN(CC3)c4ccc(cc4)F JS-2106 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3cc(ccc3Cl)C(F)(F)F)F JS-2107 Cc1ccc(c(c1)Br)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2108 c1cc(c(cc1Nc2c3cc(ccc3ncn2)Br)[N+](=O)[O-])F JS-2109 c1cc(ccc1N)SCc2ccc(c(c2)Cl)Cl JS-210C c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccc(cc3)OC(F)(F)F JS-2111 Cc1ccc(c(c1)C)N2CCN(CC2)CC(=O)Nc3ccc(cc3)OC(F)(F)F JS-2112 COc1ccc(c(c1)OC)NC(=O)/C=C/c2ccc(cc2)OC(F)(F)F JS-2113 Cc1cc(ccc1F)NC(=O)/C=C/c2ccc(cc2)OC(F)(F)F JS-2114 c1ccc(cc1)Oc2ccc(cc2)NC(=O)/C=C/c3ccc(cc3)OC(F)(F)F JS-2115 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)Nc4ccc(cc4)OC(F)(F)F JS-2116 c1cc(ccc1/C=C/C(=O)Nc2ccc(c(c2)Cl)F)OC(F)(F)F JS-2117 Cc1cc(ccc1Br)NC(=O)/C=C/c2ccc(cc2)OC(F)(F)F JS-2118 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OC(F)(F)F JS-2119 c1cc(ccc1OCC(=O)NN)Cl JS-211C c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3cc(ccc3F)F JS-2120 c1cc(ccc1/C=C/C(=O)Nc2ccc(cc2)Cl)OC(F)(F)F JS-2121 CCn1c(=O)c2ccccc2nc1SCc3ccc(cc3)F JS-2122 c1cc2c(cc1/C=C/C(=O)Nc3ccc(cc3F)F)OCCO2 JS-2124 CCn1c(=O)c2ccccc2nc1SCc3c(c(c(c(c3C)C)C)C)C JS-2125 CC(C)c1ccc(cc1)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)Cl JS-2126 c1cc(ccc1N2C(=O)/C(=C\c3ccc4c(c3)OCCO4)/SC2=S)Cl JS-2127 c1cc(ccc1NC(=O)CSCCCCCCSCC(=O)Nc2ccc(cc2)OC(F)(F)F)OC(F)(F)F JS-2128 c1cc(cc(c1)Cl)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)Cl JS-2129 c1ccc(cc1)Cn2c(=O)c3ccccc3[nH]c2=S JS-212C CC(C)(C)c1ccc(cc1)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)Cl JS-2130 c1cc(cc(c1)[N+](=O)[O-])/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)Cl JS-2131 c1cc(c(cc1F)NC(=O)CSCCCCCCSCC(=O)Nc2cc(ccc2F)F)F JS-2132 c1cc(c(c(c1)Cl)Cl)NC(=O)CSCCCCCCSCC(=O)Nc2cccc(c2Cl)Cl JS-2134 c1cc(ccc1NC(=O)CSCCCCCCSCC(=O)Nc2ccc(cc2)Cl)Cl JS-2135 CN1C/C(=C\c2ccc(cc2)OCc3ccc(cc3)F)/C(=O)/C(=C/c4ccc(cc4)OCc5ccc(cc5)F)/C1 JS-2136 CN1C/C(=C\c2cc(ccc2)[N+](=O)[O-])/C(=O)/C(=C/c3cc(ccc3)[N+](=O)[O-])/C1 JS-2138 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)Nc3ccc(cc3)OC(F)(F)F JS-2139 c1cc(ccc1CSc2ccc(cc2)N)Cl JS-213C c1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)Nc4cc(ccc4F)F JS-2140 CCn1c(=O)c2ccccc2nc1SCC(=O)Nc3ccc(cc3)OC(F)(F)F JS-2141 c1c(ccc(c1)Cl)/C=C\2/C(=O)/C(=C/c3ccc(cc3)Cl)/CC2 JS-2143 CCOc1ccc(cc1)/C=C\2/C(/C(=C/c3ccc(cc3)OCC)/CN(C2)Cc4ccccc4)O JS-2144 c1c(ccc(c1)Cl)/C=C\2/C(=O)/C(=C/c3ccc(cc3)Cl)/CCCC2 JS-2145 c1cc2c(cc1[N+](=O)[O-])c(ncn2)Nc3ccc(cc3F)F JS-2146 CC(c1ccc(cc1)/C=C\2/C(/C(=C/c3ccc(cc3)C(C)C)/CN(C2)Cc4ccccc4)O)C JS-2147 c1cc(ccc1CNc2c3cc(ccc3ncn2)[N+](=O)[O-])Cl JS-2148 CC(C)(C)c1ccc(cc1)Nc2c3cc(ccc3ncn2)[N+](=O)[O-] JS-2149 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3cc(ccc3Br)Br)F JS-2150 c1cc(ccc1CNC(=S)C(=O)Nc2cc(ccc2F)F)Cl JS-2151 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3cc(ccc3Br)Br JS-2152 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)Nc4ccccc4Br JS-2153 CCOc1ccc(cc1)Nc2c3cc(ccc3ncn2)[N+](=O)[O-] JS-2154 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])F)Cl JS-2155 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])F JS-2156 Cc1ccc(cc1C)NC(=O)/C=C/c2ccc(cc2)c3ccccc3 JS-2157 CC(C)(C)c1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)c3ccccc3 JS-2158 Cn1cnnc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])F JS-2159 c1ccc(cc1)N2CCN(CC2)c3ccc(cc3C=O)[N+](=O)[O-] JS-215C c1ccc(cc1)c2ccc(cc2)/C=C/C(=O)NCc3ccc(cc3)Cl JS-2160 c1ccc(cc1)c2ccc(cc2)/C=C/C(=O)Nc3ccc(c(c3)F)F JS-2161 c1cc(sc1)/C=N/c2ccc(cc2)SCc3ccc(cc3)F JS-2162 c1cnc(nc1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])F JS-2163 c1ccc(cc1)c2ccc(cc2)/C=C/C(=O)Nc3ccc4c(c3)OCCO4 JS-2164 c1cc2c(cc1Nc3c4cc(ccc4ncn3)[N+](=O)[O-])OCCO2 JS-2165 COc1ccc(c(c1)OC)Nc2c3cc(ccc3ncn2)[N+](=O)[O-] JS-2166 COc1ccc(cc1Nc2c3cc(ccc3ncn2)[N+](=O)[O-])Cl JS-2167 c1cc(cc(c1)Nc2c3cc(ccc3ncn2)[N+](=O)[O-])C(F)(F)F JS-2168 c1cc(ccc1CSc2ccc(cc2)N3C(=O)CCC3=O)F JS-2169 c1ccc(cc1)CC(=S)C(=O)Nc2ccc(c(c2)Cl)Cl JS-216C CCCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)C)C JS-2170 CCCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2OC)OC JS-2171 CCCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)C)Br JS-2172 CCCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)Oc3ccccc3 JS-2173 CCCOc1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)F)C JS-2174 c1ccc(cc1)CN2CCC(CC2)NCC(=O)Nc3ccc(cc3)Cl JS-2176 CCCOc1ccc(cc1)/C=C/C(=O)Nc2cc(ccc2OC)Cl JS-2177 COc1ccc(cc1)N2CCN(CC2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-2178 c1cc(sc1)/C=N/c2ccc(cc2)SCc3ccc(c(c3)Cl)Cl JS-2179 c1cc(c(cc1NC(=O)CN2CCCC2)[N+](=O)[O-])F JS-217C Cc1cc(ccc1NC(=O)/C=C/c2ccc3c(c2)OCO3)F JS-2180 c1ccc(cc1)Oc2ccc(cc2)Nc3c4cc(ccc4ncn3)[N+](=O)[O-] JS-2181 c1cc(ccc1CNC(=O)/C=C/c2ccc3c(c2)OCO3)F JS-2182 Cc1ccc(cc1C)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-2183 Cc1ccc(c(c1)F)NC(=O)/C=C/c2ccc3c(c2)OCO3 JS-2184 c1ccnc(c1)N2CCN(CC2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-2185 c1cc(ccc1N2CCN(CC2)C(=O)/C=C/c3ccc4c(c3)OCO4)F JS-2186 c1cc(cc(c1)Cl)N2CCN(CC2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-2187 c1ccc(cc1)CN2C(=O)/C(=C\c3cc(ccc3Sc4ccc(cc4)Cl)[N+](=O)[O-])/SC2=S JS-2188 c1ccc(c(c1)N2C(=O)/C(=C\c3cc(ccc3Sc4ccc(cc4)Cl)[N+](=O)[O-])/SC2=S)Cl JS-2189 c1ccc2c(c1)c(=O)oc(n2)c3cccs3 JS-218C c1cc(ccc1NC(=O)CSc2ccc(cc2)Cl)N3CCOCC3 JS-2191 c1cc(c(cc1[N+](=O)[O-])/C=C/2\C(=O)NC(=S)S2)SC3CCCCC3 JS-2192 Cc1ccc(cc1)Sc2ccc(cc2/C=C/3\C(=O)NC(=S)S3)[N+](=O)[O-] JS-2193 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3)N4CCOCC4 JS-2194 c1cc(c(cc1[N+](=O)[O-])/C=C/2\C(=O)NC(=S)S2)N3CCCCC3 JS-2195 CCN1C(=O)/C(=C\c2cc(ccc2Sc3ccccc3)[N+](=O)[O-])/SC1=S JS-2196 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=C/3\C(=O)NC(=S)S3)Br JS-2197 c1cc(ccc1CSc2ccc(cc2)NC(=O)CN3CCOCC3)F JS-2199 c1ccc2c(c1)c(=O)oc(n2)c3ccc(cc3)F JS-219C c1ccc(cc1)N2CCN(CC2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-2200 c1cc(ccc1C(=O)CCSc2ccc(cc2)F)Cl JS-2201 c1cc(c(cc1/C=C/2\C(=O)NC(=S)S2)[N+](=O)[O-])N3CCCC3 JS-2203 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/c3ccc4c(c3)OCO4 JS-2204 Cn1cnnc1SCC(=O)Nc2ccc(cc2)N3CCOCC3 JS-2205 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=C/3\C(=O)NC(=S)S3)Cl JS-2206 c1ccc(cc1)CN2CCC(CC2)NC(=O)/C=C/c3cccc(c3)Br JS-2207 c1cc(cc(c1)Br)/C=C/C(=O)Sc2ccc(cc2)Cl JS-2209 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCO JS-220C c1cc(ccc1C(=O)CCSCCSCCC(=O)c2ccc(cc2)Cl)Cl JS-2210 COc1ccc(c(c1OC)OC)/C=C/C(=O)Sc2ccc(cc2)Br JS-2211 COc1ccc(cc1)NCCC(=O)c2ccc(cc2)Cl JS-2212 COc1ccc(cc1)NCCC(c2ccc(cc2)Cl)O JS-2213 COc1ccc(c2c1cccc2)/C=C/C(=O)Sc3ccc(cc3)F JS-2215 Cc1ccc(cc1)SC(=O)/C=C/c2ccc(c3c2cccc3)OC JS-2216 Cc1cc(ccc1Br)NCc2cccc(c2O)OC JS-2218 c1cc(ccc1C(CCSc2ccc(cc2)Cl)O)Cl JS-2219 COc1cccc(c1O)CNc2ccc(cc2F)F JS-2220 c1ccc2cc(ccc2c1)C(=O)CCSc3ccc(cc3)Cl JS-2221 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(c(c3)Cl)Cl JS-2222 COc1cccc(c1O)CNc2ccc(c(c2)F)F JS-2223 c1ccc2c(c1)CCC(C2=O)CSc3ccc(cc3)Br JS-2224 Cc1ccc(nc1)NCc2cccc(c2O)OC JS-2228 c1cc(sc1)C(=O)CCNc2ccc(cc2)Cl JS-2229 COc1ccc(c(c1)OC)NCCC(=O)c2ccc3ccccc3c2 JS-2230 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3ccc4ccccc4c3 JS-2231 c1cc(sc1)C(=O)CCNc2ccc(cc2)I JS-2232 Cc1ccc(nc1)NCCC(=O)c2ccc3ccccc3c2 JS-2233 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3cccs3 JS-2235 c1ccc(cc1)Oc2ccc(cc2)NCCC(c3ccc4ccccc4c3)O JS-2236 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3ccc(cc3)Cl JS-2237 Cc1cc(ccc1NCc2cccc(c2O)OC)Br JS-2238 c1cc(sc1)C(=O)CCNc2ccc(c(c2)F)Cl JS-2239 COc1cc(ccc1NCCC(=O)c2cccs2)Cl JS-2240 Cc1ccc(cc1C)NCCC(=O)c2cccs2 JS-2241 c1cc(sc1)C(=O)CCNc2ccc(cc2)C3CCCCC3 JS-2242 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(c(c3)F)Cl JS-2243 CCOc1ccc(cc1)NCCC(=O)c2ccc(cc2)F JS-2244 CC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)OC JS-2245 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(cc3)C(F)(F)F JS-2247 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3ccco3 JS-2248 CCc1ccc(cc1)NCCC(=O)c2ccc(cc2)F JS-2250 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)OC JS-2251 c1cc(c(cc1C(=O)CCNc2ccc3c(c2)OCO3)Cl)Cl JS-2252 COc1ccc(cc1OC)C(=O)CCSc2ccc(cc2)Br JS-2253 CC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2254 CC(C)c1ccc(cc1)NCCC(=O)c2ccc(c(c2)OC)OC JS-2255 c1cc(cc(c1)[N+](=O)[O-])NCCC(=O)c2ccc(cc2)Cl JS-2256 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(cc3)C(F)(F)F JS-2257 c1cc(cc(c1)[N+](=O)[O-])NCCC(=O)c2ccc3c(c2)OCO3 JS-2258 Cc1ccc(cc1)SCCC(=O)c2ccc(c(c2)OC)OC JS-2259 Cc1cccnc1NCc2cccc(c2O)OC JS-2260 CC(C)c1ccc(cc1)NCCC(=O)c2cccc(c2)Br JS-2261 c1cc(sc1)C(=O)CCNc2ccc(c(c2)[N+](=O)[O-])Cl JS-2263 COc1ccc(cc1NCCC(=O)c2ccc(cc2)[N+](=O)[O-])Cl JS-2264 CCOc1ccc(cc1)NCCC(=O)c2cccc(c2)Br JS-2265 CCOc1ccc(cc1)C(=O)CCNc2ccc(c(c2)Cl)Cl JS-2266 CCOc1ccc(cc1)NCCC(=O)c2ccc(c(c2)Cl)Cl JS-2267 c1cc(ccc1C2CCCCC2)C(=O)CCNc3ccc(c(c3)Cl)Cl JS-2268 CCOc1ccc(cc1)NCCC(=O)c2ccc3c(c2)OCO3 JS-2269 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc3c(c2)OCO3 JS-2270 CCOc1ccc(cc1)NCCC(=O)c2ccc(cc2)C3CCCCC3 JS-2271 c1cc(ccc1NCCC(=O)c2ccc3c(c2)OCO3)I JS-2272 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2cccc(c2)[N+](=O)[O-] JS-2273 COc1ccc(cc1NCCC(=O)c2ccc(cc2)c3ccccc3)Cl JS-2274 c1cc(cc(c1)Br)C(=O)CCNc2ccc(c(c2)Cl)Cl JS-2275 c1ccc2c(c1)CCC(C2=O)CSc3ccc(cc3)Cl JS-2276 c1cc(c(cc1NC(=O)CSc2c(c(c(c(c2F)F)F)F)F)Cl)F JS-2277 c1cc(ccc1C(=O)CCNc2ccc(c(c2)Cl)F)F JS-2278 c1cc(ccc1NC(=O)CSc2c(c(c(c(c2F)F)F)F)F)OC(F)(F)F JS-2279 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3ccc(cc3)F JS-2280 COc1ccc(cc1)C(=O)CCNc2ccc(c(c2)Cl)F JS-2281 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3ccc4c(c3)OCO4 JS-2282 c1cc2c(cc1C(=O)CCNc3ccc(c(c3)Cl)F)OCO2 JS-2283 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)Oc3ccccc3 JS-2284 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2286 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)Br JS-2287 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)Cl JS-2288 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)F JS-2289 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc3c(c2)OCO3 JS-2290 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)C JS-2291 CCC(C)c1ccc(cc1)NCCC(=O)c2ccc3ccccc3c2 JS-2292 CCC(C)c1ccc(cc1)NCCC(=O)c2cccs2 JS-2294 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(cc3)Cl JS-2295 c1cc(ccc1C(=O)CCNc2ccc(cc2)Cl)Br JS-2296 c1cc(ccc1C(=O)CCNc2ccc(cc2)Cl)Cl JS-2297 c1cc(ccc1C(=O)CCNc2ccc(cc2)Cl)F JS-2298 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)Cl JS-2299 c1cc(ccc1NCCC(=O)c2ccc3c(c2)OCO3)Cl JS-2300 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)Cl JS-2301 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(cc3)Cl JS-2302 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(cc2)Cl JS-2303 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(c(c3)Cl)F JS-2304 c1cc(ccc1C(=O)CCNc2ccc(c(c2)Cl)F)Br JS-2305 c1cc(ccc1C(=O)CCNc2ccc(c(c2)Cl)F)Cl JS-2306 Cc1ccc(cc1)C(=O)CCNc2ccc(c(c2)Cl)F JS-2307 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(c(c2)Cl)F JS-2309 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(c(c3)[N+](=O)[O-])Cl JS-2310 c1cc(ccc1C(=O)CCNc2ccc(c(c2)[N+](=O)[O-])Cl)Br JS-2311 c1cc(c(cc1Nc2c3cc(ccc3ncn2)[N+](=O)[O-])Cl)F JS-2312 c1cc(c(cc1Nc2c3cc(ccc3ncn2)[N+](=O)[O-])F)F JS-2313 c1cc(ccc1SCCC(=O)c2ccc(c(c2)Cl)Cl)Br JS-2315 Cc1ccc(cc1)C(=O)CCSc2ccc(cc2)C JS-2316 Cc1ccc(cc1)SCCC(=O)c2ccc3ccccc3c2 JS-2317 CCOc1ccc(cc1)C(=O)CCSc2ccc(cc2)Br JS-2318 Cc1ccc(cc1)SCCC(=O)c2ccc(cc2)c3ccccc3 JS-2319 c1cc(ccc1C(=O)CCSc2ccc(cc2)Br)O JS-2320 C[NH+](C)CCC(=O)c1ccc(cc1)O.[Cl-] JS-2321 c1cc(ccc1C(=O)CCNc2cc(ccc2F)F)Br JS-2322 c1cc(ccc1C(=O)CCNc2ccc(cc2F)F)Br JS-2323 Cc1ccc(cc1F)NCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2325 Cc1ccc(cc1)C(=O)CCNc2ccc(c(c2)F)C JS-2326 Cc1ccc(cc1F)NCCC(=O)c2ccc3ccccc3c2 JS-2327 Cc1ccc(cc1F)NCCC(=O)c2cccs2 JS-2329 Cc1ccc(cc1F)NCCC(=O)c2ccc(cc2)OC JS-2330 c1cc(ccc1C(=O)CCNc2ccc(cc2Cl)Cl)Br JS-2331 Cc1ccc(cc1)SCCC(=O)c2cccs2 JS-2332 Cc1ccc(cc1)SCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2333 Cc1ccc(cc1)SCCC(=O)c2ccc(cc2)F JS-2334 Cc1ccc(cc1F)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2335 c1cc(ccc1C(=O)CCNc2ccc(c(c2)[N+](=O)[O-])Cl)Cl JS-2336 c1cc(ccc1C(=O)CCNc2ccc(c(c2)[N+](=O)[O-])Cl)F JS-2337 COc1ccc(cc1)C(=O)CCNc2ccc(c(c2)[N+](=O)[O-])Cl JS-2338 c1cc2c(cc1C(=O)CCNc3ccc(c(c3)[N+](=O)[O-])Cl)OCO2 JS-2339 Cc1ccc(cc1)C(=O)CCNc2ccc(c(c2)[N+](=O)[O-])Cl JS-2340 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(c(c3)[N+](=O)[O-])Cl JS-2341 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(c(c2)[N+](=O)[O-])Cl JS-2342 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(cc3)C4CCCCC4 JS-2343 c1cc(ccc1C2CCCCC2)NCCC(=O)c3ccc(cc3)Br JS-2344 c1cc(ccc1C2CCCCC2)NCCC(=O)c3ccc(cc3)Cl JS-2345 c1cc(ccc1C2CCCCC2)NCCC(=O)c3ccc(cc3)F JS-2346 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)C3CCCCC3 JS-2347 c1cc(ccc1C2CCCCC2)NCCC(=O)c3ccc4c(c3)OCO4 JS-2348 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)C3CCCCC3 JS-2349 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(cc3)C4CCCCC4 JS-2350 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(cc2)C3CCCCC3 JS-2351 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(c(c3)Cl)Cl JS-2352 c1cc(ccc1C(=O)CCNc2ccc(c(c2)Cl)Cl)Br JS-2353 c1cc(ccc1C(=O)CCNc2ccc(c(c2)Cl)Cl)Cl JS-2354 c1cc(ccc1C(=O)CCNc2ccc(c(c2)Cl)Cl)F JS-2355 COc1ccc(cc1)C(=O)CCNc2ccc(c(c2)Cl)Cl JS-2356 c1cc2c(cc1C(=O)CCNc3ccc(c(c3)Cl)Cl)OCO2 JS-2357 Cc1ccc(cc1)C(=O)CCNc2ccc(c(c2)Cl)Cl JS-2358 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(c(c2)Cl)Cl JS-2359 c1cc(sc1)C(=O)CCNc2ccc(c(c2)Cl)Cl JS-2360 COc1ccc(c(c1)OC)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2361 Cc1ccc(cc1F)NCCC(=O)c2ccc3c(c2)OCO3 JS-2362 Cc1ccc(cc1)SCCC(=O)c2ccc(cc2)Br JS-2363 Cc1ccc(cc1)C(=O)CCSc2ccc(cc2)Sc3ccc(cc3)SCCC(=O)c4ccc(cc4)C JS-2364 c1cc(ccc1C(=O)CCSc2ccc(cc2)Sc3ccc(cc3)SCCC(=O)c4ccc(cc4)Br)Br JS-2365 c1cc(oc1)C(=O)CCSc2ccc(cc2)Cl JS-2367 COc1ccc(cc1)C(=O)CCSCCSCCC(=O)c2ccc(cc2)OC JS-2368 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCSc2ccc(cc2)Cl JS-2370 c1cc(ccc1C(=O)CCSc2ccc(cc2)Cl)Br JS-2371 COc1ccc(cc1)C(=O)CCSc2ccc(cc2)Cl JS-2372 Cc1ccc(cc1)C(=O)CCSc2ccc(cc2)Cl JS-2373 COc1ccc(cc1)C2=NN(CC2)c3ccccc3 JS-2375 c1cc(c2c(c1)OCO2)C(=O)CCSc3ccc(cc3)Cl JS-2376 c1ccc(cc1)c2ccc(cc2)C(=O)CCSc3ccc(cc3)Cl JS-2377 Cc1ccc(cc1)C(=O)CCSCCSCCC(=O)c2ccc(cc2)C JS-2378 c1cc(sc1)C(=O)CCSCCSCCC(=O)c2cccs2 JS-2379 c1cc(ccc1C(=O)CCSCCSCCC(=O)c2ccc(cc2)F)F JS-2381 c1ccc2cc(ccc2c1)C(=O)CCSCCSCCC(=O)c3ccc4ccccc4c3 JS-2382 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCSCCSCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2383 CSc1ccc(cc1)/C=C/C(=O)NCc2ccc(cc2)F JS-2384 c1ccc(cc1)n2c(=O)c3ccccc3nc2SCc4cccc5c4cccc5 JS-2385 COc1ccc(c(c1)OC)NCCC(=O)c2ccc(cc2)Br JS-2386 COc1ccc(c(c1)OC)NCCC(=O)c2ccc(cc2)Cl JS-2387 COc1ccc(c(c1)OC)NCCC(=O)c2ccc(cc2)F JS-2388 COc1ccc(cc1)C(=O)CCNc2ccc(cc2OC)OC JS-2389 COc1ccc(c(c1)OC)NCCC(=O)c2ccc3c(c2)OCO3 JS-2390 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2OC)OC JS-2391 COc1ccc(c(c1)OC)NCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2392 Cc1ccc(cc1C)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2394 Cc1ccc(cc1C)NCCC(=O)c2ccc(cc2)Br JS-2395 Cc1ccc(cc1C)NCCC(=O)c2ccc(cc2)Cl JS-2396 Cc1ccc(cc1C)NCCC(=O)c2ccc(cc2)F JS-2397 Cc1ccc(cc1C)NCCC(=O)c2ccc(cc2)OC JS-2398 Cc1ccc(cc1C)NCCC(=O)c2ccc3c(c2)OCO3 JS-2399 Cc1ccc(cc1)C(=O)CCNc2ccc(c(c2)C)C JS-2400 Cc1ccc(cc1C)NCCC(=O)c2ccc3ccccc3c2 JS-2401 Cc1ccc(cc1C)NCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2402 CCOc1ccc(cc1)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2403 CCOc1ccc(cc1)NCCC(=O)c2ccc(cc2)Br JS-2404 CCOc1ccc(cc1)NCCC(=O)c2ccc(cc2)Cl JS-2405 CCOc1ccc(cc1)NCCC(=O)c2ccc(cc2)OC JS-2406 CCOc1ccc(cc1)NCCC(=O)c2ccc(cc2)C JS-2407 CCOc1ccc(cc1)NCCC(=O)c2ccc3ccccc3c2 JS-2408 CCOc1ccc(cc1)NCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2409 CCOc1ccc(cc1)NCCC(=O)c2cccs2 JS-2410 CCc1ccc(cc1)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2411 Cc1cc(ccc1Br)NC(=O)/C=C/c2ccc(cc2)SC JS-2412 CSc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)F JS-2413 CSc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)Cl JS-2414 CSc1ccc(cc1)/C=C/C(=O)Nc2cccc(c2)[N+](=O)[O-] JS-2415 COc1ccc(c(c1)OC)CNCC(=O)Nc2ccc(cc2)Cl JS-2416 Cc1ccc(cc1F)NCCC(=O)c2ccc(cc2)Cl JS-2417 CCOc1ccc(cc1)C(=O)CCNc2ccc(cc2)OCC JS-2418 c1ccc(cc1)c2ccc(cc2)C(=O)CCSc3c(c(c(c(c3F)F)F)F)F JS-2419 CCOc1ccc(cc1)NCCC(c2ccc(cc2)F)O JS-2421 c1cc(ccc1C(=O)CCSc2c(c(c(c(c2F)F)F)F)F)Br JS-2422 COc1ccc(cc1)NCCC(=O)c2ccc(c(c2)OC)OC JS-2423 c1ccc(cc1)Oc2ccc(cc2)NC(=O)/C=C/c3cccc(c3)Oc4ccccc4 JS-2424 Cc1ccc(cc1C)NC(=O)/C=C/c2cccc(c2)Oc3ccccc3 JS-2425 COc1ccc(c(c1)OC)NC(=O)/C=C/c2cccc(c2)Oc3ccccc3 JS-2426 Cc1cc(ccc1Br)NC(=O)/C=C/c2cccc(c2)Oc3ccccc3 JS-2427 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3ccc(cc3F)F JS-2428 COc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2429 Cc1ccc(cc1F)NCCC(c2ccc3ccccc3c2)O JS-2430 c1cc(cc(c1)Cl)N2CCN(CC2)CC(=O)Nc3ccc(cc3F)F JS-2431 COc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)OC JS-2432 Cc1ccc(cc1C)NCCC(=O)c2ccc(c(c2)Cl)Cl JS-2433 CCc1ccc(cc1)NCCC(=O)c2ccc(c(c2)Cl)Cl JS-2434 CC(C)(C)c1ccc(cc1)NCCC(=O)c2ccc(c(c2)Cl)Cl JS-2435 CCc1ccc(cc1)NCCC(=O)c2ccc(cc2)Br JS-2436 CCc1ccc(cc1)NCCC(=O)c2ccc(cc2)Cl JS-2437 CCc1ccc(cc1)NCCC(=O)c2ccc(cc2)OC JS-2438 CCc1ccc(cc1)NCCC(=O)c2ccc3c(c2)OCO3 JS-2439 CCc1ccc(cc1)NCCC(=O)c2ccc(cc2)C JS-2440 CCc1ccc(cc1)NCCC(=O)c2ccc3ccccc3c2 JS-2441 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(cc3)F JS-2444 c1cc(ccc1C(=O)CCNc2ccc(cc2)F)Br JS-2445 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)F JS-2446 c1cc(ccc1NCCC(=O)c2ccc3c(c2)OCO3)F JS-2447 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)F JS-2448 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(cc3)F JS-2449 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(cc2)F JS-2450 c1cc(sc1)C(=O)CCNc2ccc(cc2)F JS-2451 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(cc3)I JS-2452 c1cc(ccc1C(=O)CCNc2ccc(cc2)I)Br JS-2453 c1cc(ccc1C(=O)CCNc2ccc(cc2)I)Cl JS-2454 c1cc(ccc1C(=O)CCNc2ccc(cc2)I)F JS-2455 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)I JS-2456 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)I JS-2457 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(cc3)I JS-2458 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(cc2)I JS-2459 COc1ccc(cc1NCCC(=O)c2ccc(cc2)Br)Cl JS-2460 COc1ccc(cc1NCCC(=O)c2ccc(cc2)Cl)Cl JS-2461 Cc1cc(ccc1Br)NCCC(=O)c2ccc(c(c2)Cl)Cl JS-2462 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3ccc(c(c3)Cl)Cl JS-2463 c1cc(c(cc1F)F)NC(=O)CSc2c(c(c(c(c2F)F)F)F)F JS-2464 c1ccc(cc1)N2CCN(CC2)CCC(=O)c3ccc4c(c3)OCO4 JS-2465 c1ccc(cc1)c2ccc(cc2)C(=O)CCN3CCN(CC3)c4ccccc4 JS-2467 c1ccc(cc1)N2CCN(CC2)CCC(=O)c3ccc(cc3)Br JS-2468 c1cc(ccc1C(=O)CCSc2c(c(c(c(c2F)F)F)F)F)Cl JS-2469 c1ccc(cc1)c2ccc(cc2)C(=O)CCN3CCN(CC3)c4ccc(cc4)O JS-2470 COc1ccc(cc1NCCC(c2ccc(cc2)F)O)Cl JS-2471 c1cc(ccc1C(=O)CCN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])Cl JS-2472 c1cc(ccc1N2CCN(CC2)CCC(=O)c3ccc4c(c3)OCO4)[N+](=O)[O-] JS-2473 c1cc(sc1)C(=O)CCN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] JS-2474 c1cc(ccc1N2CCN(CC2)CCC(=O)c3ccc4c(c3)OCO4)F JS-2475 COc1ccc(cc1)N2CCN(CC2)CCC(=O)c3ccc4ccccc4c3 JS-2476 COc1ccc(cc1)N2CCN(CC2)CCC(=O)c3ccc4c(c3)OCO4 JS-2477 COc1ccc(cc1)C(=O)CCN2CCN(CC2)c3ccc(cc3)OC JS-2479 COc1ccc(cc1)N2CCN(CC2)CCC(c3ccc4ccccc4c3)O JS-2480 COc1ccc(cc1)N2CCN(CC2)CCC(=O)c3ccc(cc3)c4ccccc4 JS-2481 Cc1ccc(cc1Cl)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2483 COc1ccc(cc1NCCC(=O)c2ccc(cc2)F)Cl JS-2486 COc1ccc(cc1)C(=O)CCNc2cc(ccc2OC)Cl JS-2487 COc1ccc(cc1NCCC(=O)c2ccc3c(c2)OCO3)Cl JS-2488 Cc1ccc(cc1)C(=O)CCNc2cc(ccc2OC)Cl JS-2489 COc1ccc(cc1NCCC(=O)c2ccc3ccccc3c2)Cl JS-2490 COc1ccc(cc1)NCCC(=O)c2ccc(cc2)c3ccccc3 JS-2491 COc1ccc(cc1)NCCC(=O)c2ccc(cc2)F JS-2493 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)OC JS-2494 COc1ccc(cc1)NCCC(=O)c2ccc3c(c2)OCO3 JS-2495 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)OC JS-2496 COc1ccc(cc1)NCCC(=O)c2ccc3ccccc3c2 JS-2497 COc1ccc(cc1)NCCC(=O)c2cccs2 JS-2499 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc4c(c3)OCO4 JS-2500 c1cc(ccc1C(=O)CCNc2ccc3c(c2)OCO3)Cl JS-2502 c1cc(ccc1C(=O)CCNc2ccc3c(c2)OCO3)F JS-2503 COc1ccc(cc1)C(=O)CCNc2ccc3c(c2)OCO3 JS-2504 Cc1ccc(cc1)C(=O)CCNc2ccc3c(c2)OCO3 JS-2506 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc4c(c3)OCO4 JS-2507 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3cccc(c3)[N+](=O)[O-] JS-2509 c1cc(cc(c1)[N+](=O)[O-])NCCC(=O)c2ccc(cc2)Br JS-2510 c1cc(cc(c1)[N+](=O)[O-])NCCC(=O)c2ccc(cc2)F JS-2511 COc1ccc(cc1)NCC2CCc3ccccc3C2=O JS-2512 Cc1ccc(cc1Cl)NC(=O)CN2CCN(CC2)Cc3ccccc3 JS-2513 Cc1ccc(c(c1)C)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)C JS-2514 Cc1ccc(cc1Cl)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2515 Cc1ccc(cc1Cl)NC(=O)CN2CCN(CC2)c3ccccn3 JS-2516 Cc1ccc(cc1Cl)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-2517 Cc1ccc(cc1Cl)NC(=O)CSc2ccc(cc2)Cl JS-2518 Cc1ccc(cc1Cl)NCCC(=O)c2ccc(cc2)F JS-2519 Cc1ccc(cc1Cl)NCCC(=O)c2ccc(cc2)Cl JS-2520 Cc1ccc(cc1Cl)NCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2521 Cc1ccc(cc1Cl)NCCC(=O)c2ccc3c(c2)OCO3 JS-2522 Cc1ccc(cc1Cl)NCCC(=O)c2ccc(cc2)OC JS-2523 Cc1ccc(cc1Cl)NCCC(=O)c2ccc(cc2)Br JS-2524 Cc1ccc(cc1Cl)NCCC(=O)c2cccs2 JS-2525 Cc1ccc(cc1)C(=O)CCNc2ccc(c(c2)Cl)C JS-2526 Cc1ccc(cc1Cl)NC(=O)CSc2nncn2C JS-2527 Cc1ccc(cc1Cl)NCCC(=O)c2ccc3ccccc3c2 JS-2528 Cc1ccc(cc1Cl)NC(=O)CSCc2c(c(c(c(c2C)C)C)C)C JS-2529 Cc1ccc(cc1Cl)NC(=O)CSc2nccn2C JS-2530 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)F)Cl JS-2531 CCOc1ccc(cc1)C(=O)CCS(=O)(=O)c2ccc(cc2)Br JS-2534 Cc1ccc(cc1)C(=O)CCSc2ccc(cc2)Br JS-2535 COc1ccc(cc1)C(=O)CCNc2cccc(c2)[N+](=O)[O-] JS-2536 Cc1ccc(cc1)C(=O)CCNc2cccc(c2)[N+](=O)[O-] JS-2537 c1ccc2cc(ccc2c1)C(=O)CCNc3cccc(c3)[N+](=O)[O-] JS-2538 c1cc(cc(c1)[N+](=O)[O-])NCCC(=O)c2cccs2 JS-2539 c1ccc(cc1)c2ccc(cc2)C(=O)CCNc3ccc(cc3)Oc4ccccc4 JS-2540 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3ccc(cc3)Br JS-2541 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)Oc3ccccc3 JS-2542 c1ccc(cc1)Oc2ccc(cc2)NCCC(=O)c3cccc(c3)[N+](=O)[O-] JS-2543 CC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)Br JS-2544 CC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)Cl JS-2545 CC(C)c1ccc(cc1)NCCC(=O)c2ccc(cc2)F JS-2546 CC(C)c1ccc(cc1)NCCC(=O)c2ccc3c(c2)OCO3 JS-2547 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)C(C)C JS-2548 CC(C)c1ccc(cc1)NCCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2549 CC(C)c1ccc(cc1)NCCC(=O)c2cccs2 JS-2550 c1cc(ccc1C(=O)CCNc2ccc(cc2)C(F)(F)F)Br JS-2551 c1cc(ccc1C(=O)CCNc2ccc(cc2)C(F)(F)F)Cl JS-2552 c1cc(ccc1C(=O)CCNc2ccc(cc2)C(F)(F)F)F JS-2553 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)C(F)(F)F JS-2554 c1cc(ccc1C(F)(F)F)NCCC(=O)c2ccc3c(c2)OCO3 JS-2555 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)C(F)(F)F JS-2556 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(cc2)C(F)(F)F JS-2558 c1cc(sc1)C(=O)CCNc2ccc(cc2)C(F)(F)F JS-2559 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc(cc2)c3ccccc3 JS-2560 COc1ccc(cc1)NCCC(=O)c2ccco2 JS-2561 Cc1ccc(cc1)C(=O)CCNc2ccc3c(c2)OCCO3 JS-2562 Cc1ccc(cc1)C(=O)CCS(=O)(=O)c2ccc(cc2)Br JS-2563 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc(c(c2)OC)OC JS-2564 c1cc(ccc1C(=O)CCNc2ccc3c(c2)OCCO3)Cl JS-2565 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc4c(c3)OCCO4 JS-2566 c1cc(ccc1C(=O)CCNc2ccc3c(c2)OCCO3)F JS-2567 c1cc(ccc1SCCC(=O)c2ccc3c(c2)OCO3)Br JS-2568 C[n+]1ccc(c2c1cccc2)/C=C\c3ccc(cc3)OC.[I-] JS-2569 COc1ccc(c(c1)NC(=O)CSc2ccccn2)OC JS-2570 c1ccc2cc(ccc2c1)C(=O)CCSc3ccc(cc3)F JS-2571 Cc1ccc(cc1)C(=O)CCSc2ccc(cc2)F JS-2572 COc1ccc(cc1)C(=O)CCNc2ccc3c(c2)OCCO3 JS-2573 c1cc(ccc1C(=O)CCNc2ccc3c(c2)OCCO3)Br JS-2574 c1cc(sc1)C(=O)CCSc2ccc(cc2)F JS-2575 c1cc(ccc1C(=O)CCSc2ccc(cc2)F)F JS-2576 COc1ccc(cc1)C(=O)CCSc2ccc(cc2)F JS-2577 c1cc(ccc1S(=O)(=O)CCC(=O)c2ccc(c(c2)Cl)Cl)Br JS-2578 c1cc(ccc1S(=O)(=O)CCC(=O)c2ccc3c(c2)OCO3)Br JS-2579 Cc1ccc(cc1)C(=O)CCS(=O)(=O)c2ccc(cc2)Cl JS-2580 COc1ccc(c(c1)NC(=O)CSc2ccc(cc2)Cl)OC JS-2581 Cc1ccc(cc1)C(=O)CCS(=O)(=O)c2ccc(cc2)F JS-2582 c1cc(sc1)c2n[nH]c(=S)n2c3ccc(c(c3)Cl)F JS-2584 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)F)F JS-2585 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc(cc2)Br JS-2586 c1ccc2cc(ccc2c1)C(=O)CCS(=O)(=O)c3ccc(cc3)F JS-2587 COc1ccc(cc1)C(=O)CCS(=O)(=O)c2ccc(cc2)F JS-2588 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc(cc2)OC JS-2589 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)Cl)Br JS-2590 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)Cl)Cl JS-2591 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc(cc2)F JS-2592 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2cccc(c2)[N+](=O)[O-] JS-2593 COc1cccc(c1O)CNc2ccc(c(c2)Cl)F JS-2594 Cc1c(c(c(c(c1C)C)CSCCC(=O)c2ccc(cc2)Cl)C)C JS-2596 COc1ccc(cc1NCCC(=O)c2ccc3ccccc3c2)[N+](=O)[O-] JS-2597 c1cc(ccc1CSc2ccc(cc2)NS(=O)(=O)c3ccc(cc3)F)F JS-2600 Cc1ccc(cc1Cl)NCCC(=O)c2ccc(c(c2)Cl)Cl JS-2602 COc1cc(c(cc1Cl)OC)NCCC(=O)c2ccc3ccccc3c2 JS-2603 c1cc(ccc1CNC(=O)CSc2ccc(cc2)Cl)F JS-2605 COc1ccc(cc1)CNC(=O)CSc2ccc(cc2)Cl JS-2606 c1ccnc(c1)SCC(=O)NCc2ccc(cc2)F JS-2607 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccccc3)OC JS-2608 c1ccc(cc1)CNC(=O)CN2CCN(CC2)c3ccccc3 JS-2609 c1ccc(cc1)N2CCN(CC2)CC(=O)NCc3ccc(cc3)F JS-2610 COc1ccc(cc1)CNC(=O)CN2CCN(CC2)c3ccccc3 JS-2612 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)OC(F)(F)F JS-2614 Cc1ccc(cc1C)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2615 Cc1ccc(cc1C)NC(=O)CSc2nnc(n2c3ccccc3)c4cccc(c4)Cl JS-2617 c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)F)c4cccc(c4)Cl JS-2618 c1ccc(cc1)c2ccc(cc2)C(=O)CCSc3ccc(cc3)F JS-2619 c1ccc(cc1)c2ccc(cc2)C(=O)CCSc3ccc(cc3)Br JS-2620 c1ccc(cc1)CC(=O)NNC(=S)NCc2ccccc2 JS-2622 Cc1c(c(c(c(c1C)C)CSCCC(=O)c2ccc(cc2)c3ccccc3)C)C JS-2623 c1cc(ccc1C(=O)CCSc2ccc(cc2)F)Br JS-2624 c1cc(ccc1C(=O)CCSc2ccc(cc2)Br)Br JS-2625 Cc1c(c(c(c(c1C)C)CSCCC(=O)c2ccc(cc2)Br)C)C JS-2626 c1cc(ccc1C(=O)CCSc2ccc(cc2)Br)F JS-2627 c1cc(ccc1C(=O)CCSc2c(c(c(c(c2F)F)F)F)F)F JS-2629 Cc1c(c(c(c(c1C)C)CSCCC(=O)c2ccc(cc2)F)C)C JS-2630 COc1ccc(cc1)C(=O)CCSc2ccc(cc2)Br JS-2631 Cc1c(c(c(c(c1C)C)CSCCC(=O)Cc2ccc(cc2)OC)C)C JS-2633 Cc1ccc(cc1)SCCC(=O)c2ccc3c(c2)OCO3 JS-2634 c1cc2c(cc1C(=O)CCSc3c(c(c(c(c3F)F)F)F)F)OCO2 JS-2635 Cc1c(c(c(c(c1C)C)CSCCC(=O)c2ccc3c(c2)OCO3)C)C JS-2636 c1ccc2cc(ccc2c1)C(=O)CCSc3ccc(cc3)Br JS-2637 c1ccc2cc(ccc2c1)C(=O)CCSc3c(c(c(c(c3F)F)F)F)F JS-2638 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCSc2ccc(cc2)Br JS-2640 Cc1cccc(c1)c2nnc(n2C)S JS-2645 c1ccc(cc1)n2c(nnc2SCC(=O)c3ccc(cc3)Cl)c4cccc(c4)Cl JS-2646 Cc1ccc(cc1Cl)NC(=O)CSc2nc(cc(n2)C)C JS-2647 Cc1cc(nc(n1)SCC(=O)Nc2cc(ccc2OC)OC)C JS-2648 Cc1cc(nc(n1)SCC(=O)NCc2ccccc2)C JS-2649 Cc1cccc(c1)c2nnc(n2C)SCC(=O)NCc3ccc(cc3)F JS-2650 Cc1cccc(c1)c2nnc(n2C)SCC(=O)Nc3ccc(c(c3)Cl)C JS-2651 Cc1cccc(c1)c2nnc(n2C)SCC(=O)Nc3ccc(c(c3)F)F JS-2652 Cc1ccc(cc1C)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2653 Cc1ccc(cc1C)NC(=O)CSc2nnnn2C JS-2654 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F)OC JS-2655 Cc1cccc(c1)c2nnc(n2C)SCC(=O)Nc3c(c(c(c(c3F)F)F)F)F JS-2656 Cn1c(nnn1)SCC(=O)Nc2ccc(c(c2)F)F JS-2657 COc1ccc(cc1OC)CC(=O)NNC(=S)Nc2ccc(c(c2)Cl)F JS-2658 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])F)F JS-2659 Cn1c(nnn1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])F JS-2660 c1cc(ccc1SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])F)Br JS-2661 c1cc(ccc1CNC(=O)CN2CCN(CC2)c3ccc(cc3)F)F JS-2662 COc1ccc(cc1OC)CC(=O)NNC(=S)Nc2ccc(cc2)Cl JS-2663 c1ccc(cc1)CNC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2664 Cc1ccc(cc1C)NC(=O)CSc2nc(cc(n2)C)C JS-2665 COc1ccc(cc1)NC(=O)CN2CCCc3c2cccc3 JS-2666 COc1ccc(cc1NC(=O)CSc2ccc(cc2)Cl)[N+](=O)[O-] JS-2668 CCOc1ccc(cc1)NC(=S)NNC(=O)Cc2ccccc2 JS-2669 COc1ccc(cc1OC)C(=O)CCSc2ccc(cc2)F JS-2670 COc1ccc(cc1OC)C(=O)CCSc2ccc(cc2)Cl JS-2671 Cc1c(c(c(c(c1C)C)CSCCC(=O)c2ccc(c(c2)OC)OC)C)C JS-2673 c1cc(ccc1F)SCCC(=O)c2ccc(c(c2)Cl)Cl JS-2674 c1cc(ccc1SCCC(=O)c2ccc(c(c2)Cl)Cl)Cl JS-2675 Cc1ccc(cc1)SCCC(=O)c2ccc(c(c2)Cl)Cl JS-2676 c1cc(c(cc1C(=O)CCSc2c(c(c(c(c2F)F)F)F)F)Cl)Cl JS-2677 Cc1cc(nc(n1)SCC(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl)C JS-2695 Cn1c(nnc1SCC(=O)Nc2ccc(c(c2)F)F)c3ccc(cc3)Cl JS-2696 COc1ccc(cc1)CNC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2697 COc1ccc(cc1)CNC(=O)CSc2ccc(cc2)Br JS-2698 COc1ccc(cc1NC(=O)CN2CCOCC2)[N+](=O)[O-] JS-2699 COc1ccc(cc1NC(=O)CN2CCN(CC2)c3ccc(cc3)F)[N+](=O)[O-] JS-2700 Cn1cnnc1SCC(=O)Nc2cc(ccc2OC)[N+](=O)[O-] JS-2701 c1cc(ccc1SC2CC(=O)N(C2=O)c3ccc(c(c3)[N+](=O)[O-])F)Cl JS-2702 COc1ccc(cc1NC(=O)CNCc2ccccc2)[N+](=O)[O-] JS-2703 CCc1ccc(cc1)C(=O)CCNc2ccc(cc2)OC JS-2704 CCc1ccc(cc1)C(=O)CCSc2ccc(cc2)Br JS-2705 COc1ccc(cc1N2C(=O)CC(C2=O)Sc3ccc(cc3)Br)[N+](=O)[O-] JS-2706 Cn1c(nnn1)SCC(=O)Nc2cc(ccc2OC)[N+](=O)[O-] JS-2707 c1cc(ccc1C(F)(F)F)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2708 CN1CCN(CC1)CC(=O)Nc2cc(ccc2OC)[N+](=O)[O-] JS-2709 Cc1cccc(c1)c2nnc(n2C)SCc3ccc(cc3)F JS-2710 Cc1cccc(c1)c2nnc(n2C)SCC(=O)Nc3ccc(c(c3)[N+](=O)[O-])F JS-2711 Cc1cccc(c1)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)C(F)(F)F JS-2712 Cc1cccc(c1)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)Br JS-2713 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)C(F)(F)F JS-2714 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)C(F)(F)F JS-2715 c1cc(ccc1C(F)(F)F)NC(=O)CSc2ccc(cc2)Cl JS-2716 Cc1cc(nc(n1)SCC(=O)Nc2ccc(cc2)C(F)(F)F)C JS-2718 CCn1c(nnc1SCC(=O)Nc2ccc(c(c2)F)F)c3ccccc3 JS-2720 c1ccc(cc1)c2nnc(n2c3ccccc3)SCc4ccc(cc4)F JS-2723 CCn1c(nnc1SCC(=O)Nc2cc(ccc2F)F)c3ccccc3 JS-2724 Cc1ccc(cc1C)NC(=O)CSc2nnc(n2c3ccccc3)c4ccccc4 JS-2728 CC(C)Cn1c(nnc1S)c2ccc(cc2)Cl JS-2731 c1cc(sc1)C(=O)CCNc2ccc(cc2)Br JS-2732 c1ccc(cc1)c2nnc(n2c3ccccc3)SCc4ccc(c(c4)Cl)Cl JS-2733 CCCCn1c(nnc1SCC(=O)Nc2ccc(c(c2)F)F)c3ccccc3 JS-2734 Cc1ccc(cc1)SC(CC(=O)c2ccc(cc2)Br)C(=O)O JS-2735 Cc1ccc(cc1)C(=O)CC(C(=O)O)SCc2c(c(c(c(c2C)C)C)C)C JS-2736 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2c3ccc(cc3)F)c4cccc(c4)Cl JS-2737 c1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)Nc4ccc(c(c4)F)F JS-2739 CCOc1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cc2)Br JS-2740 CCCCc1ccc(cc1)NC(=O)CSc2nnc(n2CC)c3ccccc3 JS-2741 CCn1c(nnc1SCC(=O)Nc2ccc(cc2)C(C)C)c3cccc(c3)Cl JS-2742 CCOc1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)Nc4ccc(c(c4)C)C JS-2744 Cc1ccc(cc1C)NC(=O)CSc2nnc(n2c3ccccc3)c4cccs4 JS-2745 c1cc(ccc1C(=O)CCNc2ccc(cc2)Br)Cl JS-2746 Cc1ccc(c(c1)NC(=O)CSc2nnc(n2c3ccccc3)Cc4ccccc4)OC JS-2747 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)Br JS-2748 c1ccc(cc1)Cc2nnc(n2c3ccccc3)SCC(=O)Nc4ccc(c(c4)F)F JS-2749 c1cc(ccc1NCCC(=O)c2ccc3c(c2)OCO3)Br JS-2750 COc1ccc(cc1)C(=O)CCNc2ccc(c(c2F)F)F JS-2751 c1cc(ccc1C(=O)CCNc2ccc(c(c2F)F)F)Br JS-2754 c1ccc2cc(ccc2c1)C(=O)CCNc3ccc(c(c3F)F)F JS-2755 CCC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2Cc3ccccc3)Cc4ccccc4 JS-2756 Cc1ccc(cc1)C(=O)CCNc2ccc(c(c2F)F)F JS-2757 CCCCc1ccc(cc1)NC(=O)CSc2nnc(n2CCCC)COc3ccc(cc3)Cl JS-2758 COc1ccc(cc1)CNC(=O)CSc2nnc(n2c3ccccc3)c4cccs4 JS-2760 c1cc(ccc1C(=O)CCNc2ccc(c(c2F)F)F)Cl JS-2761 CCOc1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)NCc4ccc(cc4)OC JS-2762 c1cc(sc1)C(=O)CCNc2ccc(c(c2F)F)F JS-2763 CSc1nnc(n1c2ccccc2)c3ccccc3 JS-2765 CCOc1ccc(cc1)c2nnc(n2c3ccccc3)SC JS-2766 COc1cc(c(cc1Cl)OC)NCCC(=O)c2cccs2 JS-2767 COc1cc(c(cc1Cl)OC)NCCC(=O)c2ccc(cc2)Cl JS-2768 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCNc2ccc(c(c2F)F)F JS-2769 CCn1c(nnc1SC)c2ccc(cc2)F JS-2771 Cc1c(c(c(c(c1C)C)CS(=O)(=O)CCC(=O)c2ccc(cc2)Cl)C)C JS-2772 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)Br)F JS-2773 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)Cl)F JS-2774 Cc1c(c(c(c(c1C)C)CS(=O)(=O)CCC(=O)c2ccc(cc2)F)C)C JS-2776 COc1ccc(cc1)C(=O)CCS(=O)(=O)c2ccc(cc2)Cl JS-2777 CCOc1ccc(cc1)c2nnc(n2c3ccccc3)SCc4ccc(c(c4)Cl)Cl JS-2778 Cc1c(c(c(c(c1C)C)CS(=O)(=O)CCC(=O)c2ccc(cc2)OC)C)C JS-2779 c1cc(ccc1S(=O)(=O)CCC(=O)c2ccc3c(c2)OCO3)Cl JS-2781 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc3c(c2)OCO3 JS-2782 Cn1c(nnn1)SCC(=O)Nc2cc(c(cc2F)F)F JS-2783 Cn1cnnc1SCC(=O)Nc2cc(c(cc2F)F)F JS-2785 c1ccc2cc(ccc2c1)C(=O)CCS(=O)(=O)c3ccc(cc3)Br JS-2786 c1ccc2cc(ccc2c1)C(=O)CCS(=O)(=O)c3ccc(cc3)Cl JS-2787 CSc1nnc(n1c2ccc(cc2)F)Cc3ccccc3 JS-2788 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCS(=O)(=O)c2ccc(cc2)Br JS-2792 c1cc(cc(c1)[N+](=O)[O-])C(=O)CCS(=O)(=O)c2ccc(cc2)Cl JS-2793 COc1ccc(cc1)C(=O)CCNc2cc(c(cc2OC)Cl)OC JS-2794 c1ccc(cc1)c2ccc(cc2)C(=O)CCS(=O)(=O)c3ccc(cc3)F JS-2795 c1ccc(cc1)c2ccc(cc2)C(=O)CCS(=O)(=O)c3ccc(cc3)Br JS-2796 c1ccc(cc1)c2ccc(cc2)C(=O)CCS(=O)(=O)c3ccc(cc3)Cl JS-2797 Cc1c(c(c(c(c1C)C)CS(=O)(=O)CCC(=O)c2ccc(cc2)c3ccccc3)C)C JS-2798 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)F)Br JS-2799 c1cc(ccc1C(=O)CCS(=O)(=O)c2ccc(cc2)Br)Br JS-2800 c1cc(ccc1C(=O)CCS(=O)(=O)c2c(c(c(c(c2F)F)F)F)F)Br JS-2801 COc1cc(c(cc1Cl)OC)NC(=O)CN2CCOCC2 JS-2803 COc1cc(c(cc1Cl)OC)NC(=O)CSc2ccccn2 JS-2804 COc1cc(c(cc1Cl)OC)NC(=O)CN2CCN(CC2)c3cccc(c3)Cl JS-2805 COc1cc(c(cc1Cl)OC)NC(=O)CN2CCN(CC2)Cc3ccccc3 JS-2806 c1cc(ccc1SCC(=O)Nc2cc(c(cc2F)F)F)Cl JS-2807 c1cc(ccc1F)SCCC(=O)c2ccc3c(c2)OCO3 JS-2808 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cc(c(cc3F)F)F JS-2809 Cn1c(nnc1SC)c2ccc(cc2)Cl JS-2810 c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3cc(c(cc3F)F)F JS-2811 c1ccnc(c1)SCC(=O)Nc2cc(c(cc2F)F)F JS-2812 c1cc(ccc1C(=O)CCSc2ccc(cc2)Sc3ccc(cc3)SCCC(=O)c4ccc(cc4)F)F JS-2813 c1cc(ccc1SCC(=O)Nc2cc(c(cc2F)F)F)Sc3ccc(cc3)SCC(=O)Nc4cc(c(cc4F)F)F JS-2815 c1ccc(cc1)n2c(nnc2S)CSc3ccc(cc3)Cl JS-2816 CCCCc1ccc(cc1)NC(=O)CN2CCCc3c2cccc3 JS-2817 COc1ccc(cc1NCCC(=O)c2ccc(cc2)c3ccccc3)[N+](=O)[O-] JS-2818 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)Sc3ccc(cc3)SCC(=O)Nc4ccc(cc4)CCCC JS-2819 COc1ccc(cc1OC)C(=O)CCS(=O)(=O)c2ccc(cc2)F JS-2822 COc1ccc(cc1OC)C(=O)CCS(=O)(=O)c2ccc(cc2)Cl JS-2824 c1cc(sc1)C(=O)CCSc2ccc(cc2)Sc3ccc(cc3)SCCC(=O)c4cccs4 JS-2825 c1cc(ccc1S(=O)(=O)CCC(=O)c2ccc(c(c2)Cl)Cl)Cl JS-2828 Cc1ccc(cc1)S(=O)(=O)CCC(=O)c2ccc(c(c2)Cl)Cl JS-2829 CCCCc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2832 COc1ccc(cc1)C(=O)CCSc2ccc(cc2)Sc3ccc(cc3)SCCC(=O)c4ccc(cc4)OC JS-2833 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cc(ccc3F)F JS-2834 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)C(F)(F)F JS-2835 c1cc(ccc1N2CCN(CC2)CC(=O)Nc3cc(c(cc3F)F)F)F JS-2836 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)F)F JS-2838 c1cc(ccc1SCCC(=O)c2ccc3c(c2)OCO3)Sc4ccc(cc4)SCCC(=O)c5ccc6c(c5)OCO6 JS-2840 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cc(ccc3Br)Br JS-2841 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)Cl)Cl JS-2846 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)Br JS-2847 c1cc(c(cc1NCc2cc(ccc2O)Br)[N+](=O)[O-])F JS-2848 c1ccc(cc1)Cc2nnc(n2c3ccccc3)SCC(=O)Nc4ccc(c(c4)Cl)Cl JS-2850 CCCCc1ccc(cc1)NC(=O)CSc2nnc(n2c3ccccc3)Cc4ccccc4 JS-2851 c1cc(c(cc1Br)CNc2ccc(c(c2F)F)F)O JS-2852 c1cc(c(cc1NCc2cc(ccc2O)Br)F)F JS-2853 c1cc(ccc1NCc2cc(ccc2O)Br)OC(F)(F)F JS-2854 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(c(c3)[N+](=O)[O-])F JS-2855 Cc1cc(ccc1NCc2cc(ccc2O)Br)F JS-2858 c1cc(c(cc1Br)CNc2cc(c(cc2F)F)F)O JS-2859 c1cc(c(cc1NCc2cc(ccc2O)Br)Cl)F JS-2860 c1ccc(cc1)CC(=O)N/N=C/c2cccs2 JS-2861 c1ccc(cc1)CC(=O)N/N=C/c2ccc(cc2)OC(F)(F)F JS-2862 COc1ccc(cc1NCc2cc(ccc2O)Br)[N+](=O)[O-] JS-2864 c1cc(ccc1NCc2cc(ccc2O)Cl)OC(F)(F)F JS-2865 CCCCn1c(nnc1SCC(=O)Nc2cc(ccc2OC)C)c3ccccc3 JS-2866 CCCCc1ccc(cc1)NC(=O)CSc2nnc(n2CCCC)c3ccccc3 JS-2867 c1cc(c(cc1NCc2cc(ccc2O)Cl)Cl)F JS-2868 c1cc(ccc1/C=N/NC(=O)COc2ccc(cc2)Cl)OC(F)(F)F JS-2869 COc1cc(cc(c1OC)OC)/C=N/NC(=O)Cc2ccccc2 JS-2870 Cc1ccc(cc1NCc2cc(ccc2O)Br)F JS-2871 CCCCn1c(nnc1SCC(=O)Nc2ccc(c(c2)Cl)Cl)c3ccccc3 JS-2872 Cc1ccc(cc1C)NCc2cc(ccc2O)Cl JS-2873 Cc1ccnc(c1)NCc2cc(ccc2O)Cl JS-2874 Cc1cc(ccc1Br)NCc2cc(ccc2O)Cl JS-2877 COc1ccc(cc1)NCc2cc(ccc2O)Cl JS-2878 Cc1cc(no1)NCc2cccc(c2O)OC JS-2879 COc1ccc(cc1)NCc2cccc(c2O)OC JS-2880 COc1ccc(cc1)NCc2cc(ccc2O)Br JS-2881 c1cc(cc(c1)[N+](=O)[O-])NCc2cc(ccc2O)Cl JS-2882 Cc1cc(no1)NCc2ccc(cc2O)OC JS-2883 Cc1cc(no1)NCc2cc(cc(c2O)OC)I JS-2884 CC(C)c1ccc(cc1)NCc2cc(cc(c2O)OC)I JS-2886 CC(C)c1ccc(cc1)NCc2cc(cc(c2O)OC)Br JS-2887 CC(C)c1ccc(cc1)NCc2cc(ccc2O)Br JS-2888 c1ccc(cc1)Oc2ccc(cc2)NCc3cc(ccc3O)Br JS-2889 CC(C)c1ccc(cc1)NCc2ccc(cc2O)OC JS-2890 COc1cc(cc(c1O)CNc2ccc(cc2)Oc3ccccc3)Br JS-2891 c1ccc(cc1)n2c(nnc2SCC(=O)Nc3ccc(cc3)F)CCCOc4ccc(cc4Cl)Cl JS-2894 COc1ccc(c(c1)O)CNc2ccc(cc2)Oc3ccccc3 JS-2895 CCCCc1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl JS-2898 CC(C)c1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl JS-2901 CCC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2902 c1ccc(cc1)N2CCN(CC2)C3=C(C(=O)c4ccccc4C3=O)Cl JS-2904 CC(C)c1ccc(cc1)N(Cc2cc(ccc2OC)Br)C(=S)Nc3ccccc3 JS-2905 Cc1ccc(cc1Cl)NC2=C(C(=O)c3ccccc3C2=O)Cl JS-2907 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Nc3ccc(cc3)OC(F)(F)F JS-2908 c1cc(ccc1NCSc2ccc(cc2)Cl)Cl JS-2909 COc1cc(cc(c1O)CNc2ccc(cc2)C3CCCCC3)Br JS-2910 COc1cc(cc(c1O)CNc2ccc(cc2)C3CCCCC3)I JS-2911 Cc1ccc(cc1C)NC(=O)CSc2ccc(cc2)N JS-2912 COc1ccc(c(c1)O)CNc2ccc(cc2)C3CCCCC3 JS-2913 COc1ccc(cc1)NC(=O)CSc2ccc(cc2)N JS-2914 COc1ccc(c(c1)NC(=O)CSc2ccc(cc2)N)OC JS-2915 Cc1ccc(cc1C)NC(=O)CSc2ccc(cc2)/N=C/c3ccccc3O JS-2916 Cc1ccc(cc1C)NC(=O)CSc2ccc(cc2)NC(=S)Nc3ccccc3 JS-2917 COc1ccc(cc1)NC(=O)CSc2ccc(cc2)NC(=S)Nc3ccc(cc3)F JS-2919 CCOc1ccc(cc1)NC(=S)Nc2ccc(cc2)SCC(=O)Nc3ccc(cc3)OC JS-2920 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)NCCC(=O)c3ccc4ccccc4c3 JS-2922 c1cc(ccc1NC(=O)CSc2nnc(s2)N)F JS-2926 c1cc(ccc1N)SCC(=O)Nc2ccc(cc2)Cl JS-2927 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)NCc3ccccc3O JS-2928 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)N3C(=O)CCC3=O JS-2929 Cc1ccc(cc1)NC(=O)CSc2ccccc2N JS-2930 c1ccc(c(c1)CNc2ccc(cc2)SCC(=O)Nc3cccc(c3)[N+](=O)[O-])O JS-2931 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)SCc4ccc(cc4Cl)Cl JS-2932 CCc1ccc(cc1)NC(=O)CSc2nnc(n2c3ccc(cc3)F)Cc4ccccc4 JS-2933 CCCCc1ccc(cc1)NC(=O)CSc2ccc(cc2)N3C(=O)c4ccccc4C3=O JS-2934 CCCCc1ccc(cc1)NC(=O)CSc2ccccc2N JS-2935 Cc1cccc(c1C)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2936 Cc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2937 Cc1ccc(cc1)NC(=O)CSc2ccccc2NCc3ccccc3O JS-2938 CCc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccccc3 JS-2939 Cc1ccc(cc1)NC(=O)CSc2nnc(n2c3ccccc3)Cc4ccccc4 JS-2940 CCCCc1ccc(cc1)NC(=O)CSc2ccccc2/N=C/c3ccccc3O JS-2941 Cc1ccc(cc1C)NCCC(=O)c2ccc(c(c2)OC)OC JS-2942 COc1ccc(cc1OC)C(=O)CCNc2ccc(c(c2)Cl)F JS-2943 CCCCc1ccc(cc1)NC(=O)CSc2ccccc2NC(=S)Nc3ccccc3 JS-2944 COc1ccc(cc1OC)C(=O)CCNc2ccc(cc2F)F JS-2945 CCc1ccc(cc1)NC(=O)CSc2nnc(n2Cc3ccccc3)Cc4ccccc4 JS-2946 c1ccc(c(c1)/C=N/c2ccc(cc2)SCC(=O)Nc3ccc(cc3)OC(F)(F)F)O JS-2947 CCOc1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)Nc4cc(ccc4C)F JS-2948 Cc1ccc(cc1NC(=O)CN2CCN(CC2)c3ccccc3)F JS-2949 COc1ccc(cc1)NC(=O)CSc2ccc(cc2)NCc3ccccc3O JS-2950 Cc1ccc(cc1NC(=O)CSc2nnc(s2)N)F JS-2951 CCOc1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)NCc4ccccc4 JS-2952 c1ccc(c(c1)CNc2ccc(cc2)SCC(=O)Nc3ccc(cc3)OC(F)(F)F)O JS-2953 c1ccc(c(c1)CNc2ccc(cc2)n3cncn3)O JS-2954 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)SCc3ccc(c(c3)Cl)Cl JS-2955 c1cc(c(c(c1)Cl)Cl)NC(=O)CSc2nnc(s2)N JS-2957 Cc1ccc(cc1)C(=O)CCNc2ccc(cc2)N3CCOCC3 JS-2958 COc1ccc(cc1)C(=O)CCNc2ccc(cc2)n3cncn3 JS-2959 c1ccc(c(c1)/C=N/c2ccc(cc2)SCC(=O)Nc3ccc(cc3)Br)O JS-2960 Cc1ccc(cc1NC(=O)CSc2nnc(n2c3ccccc3)c4ccccc4)F JS-2961 c1ccc(cc1)CNC(=O)CSc2nnc(n2c3ccccc3)c4ccccc4 JS-2962 Cc1ccc(cc1Cl)NC(=O)CSc2nnc(s2)N JS-2963 Cc1ccc(cc1)NC(=O)CSc2nnc(s2)N JS-2964 c1cc(ccc1C(F)(F)F)NC(=O)CSc2nnc(s2)N JS-2965 Cc1cc(ccc1NC(=O)CN2CCN(CC2)c3ccccc3)Br JS-2966 CCc1ccc(cc1)NC(=O)CSc2nnc(n2C)c3ccc(cc3)Cl JS-2967 CCCCc1ccc(cc1)NC(=O)CSc2ccccc2NCCC(=O)c3ccc4ccccc4c3 JS-2968 CCc1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cc3)F JS-2969 c1ccc(c(c1)CNc2ccc(cc2)SCc3ccc(cc3Cl)Cl)O JS-2970 Cc1ccc(cc1)NC(=O)CSc2ccc(cc2)F JS-2971 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)n3cncn3 JS-2972 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)N4CCOCC4 JS-2973 COc1ccc(cc1NC(=O)CSc2ccccn2)[N+](=O)[O-] JS-2974 c1cc(ccc1NC(=O)CSc2ccc(cc2)Cl)n3cncn3 JS-2975 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)n4cncn4 JS-2976 c1cc(ccc1/N=C/c2ccc3c(c2)OCO3)O JS-2977 c1cc(ccc1C(=O)/C=C/c2ccc(c(c2)Cl)Cl)O JS-2979 CC(C)(C)C(=O)Nc1ccccc1C(=O)O JS-2981 c1cc(ccc1C(=O)/C=C/C(=O)O)F JS-2982 CCc1ccc(cc1)NC(=O)CCl JS-2985 CCOc1ccc(cc1)NC(=O)CCl JS-2986 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)O)F JS-2988 c1cc(ccc1CC#N)NC(=O)CCl JS-2994 c1ccc2c(c1)cccc2/C=C\C(=O)c3ccc(cc3)O JS-2995 c1cc(ccc1COc2ccc(cc2)C=O)[N+](=O)[O-] JS-2997 CN(C)CCC(=O)c1ccc2ccccc2c1.Cl JS-2998 CN(C)CCC(=O)c1ccco1.Cl JS-3000 CC(CN(C)C)C(=O)c1ccccc1.Cl JS-3001 Cc1cccc(c1CC(=O)CCl)C(C)C JS-3002 CN(C)CCC(=O)c1cccs1.Cl JS-3003 c1ccc(cc1)OCC(=O)Nc2ccccc2C(=O)O JS-3004 c1cc(ccc1/C=N/c2ccc(cc2)Cl)O JS-3005 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)Cl)O JS-3006 CN(C)CCC(=O)c1ccc(cc1)F.Cl JS-3007 Cc1ccc(cc1C)C(=O)CCN(C)C.Cl JS-3008 c1cc(ccc1NC(=O)CCl)I JS-3009 c1cc2c(cc1/C=C/C(=O)O)OCO2 JS-3011 c1ccc(cc1)c2nc3ccccc3c(=O)o2 JS-3012 CCOc1ccc(cc1)/C=N/O JS-3014 COc1ccc(cc1/C=N/O)Br JS-3015 c1cc(c(cc1O)[N+](=O)[O-])C=O JS-3016 CCCCc1ccc(cc1)NC(=O)CCl JS-3018 COc1ccc(c(c1)OC)/C=C/Oc2ccc(cc2)O JS-3020 c1cc2c(cc1/C=N/O)OCO2 JS-3021 c1ccc(cc1)CN(Cc2ccccc2)C(=O)CCC(=O)O JS-3022 Cc1cccc(c1)ONN JS-3023 COc1ccccc1/C=N/O JS-3024 COc1cc(c(cc1OC)Br)C=O JS-3025 c1cc(ccc1/C=N/c2ccc(c(c2)[N+](=O)[O-])F)O JS-3026 c1ccc2c(c1)c(=O)oc(n2)c3ccc(cc3)[N+](=O)[O-] JS-3027 c1ccc(c(c1)C#N)NC(=O)OCCl JS-3028 COc1ccc(c(c1)NC(=O)CCl)OC JS-3029 CN(C)CCC(=O)c1cccc(c1)[N+](=O)[O-].Cl JS-3030 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)F)O JS-3031 c1ccc(cc1)CCC(=O)Nc2ccccc2C(=O)O JS-3032 c1ccc(cc1)C(=O)NC2C3CCC(C3)C2C(=O)O JS-3033 c1cc(ccc1/C=N/c2ccc(cc2)C(F)(F)F)O JS-3034 CN(C)CCC(=O)c1ccc(cc1)OCc2ccc(c(c2)Cl)Cl.Cl JS-3035 COc1ccc(c(c1)OC)NC2=C(C(=O)c3ccccc3C2=O)Cl JS-3038 c1cc(cnc1)CNc2ccc3c(c2)OCO3 JS-3040 CN(C)CCC(=O)c1ccc(cc1)c2ccccc2.Cl JS-3042 c1cc[n+](cc1)Cc2ccc(cc2)F.[I-] JS-3043 c1cc(c(cc1Cl)Cl)NC(=N)NC(=N)N JS-3044 c1cc(ccc1C(=O)CSc2ccc(cc2)Cl)Br JS-3046 CC(C)(C)c1ccc(cc1)c2nc3ccccc3c(=O)o2 JS-3048 c1ccc(c(c1)/C=N/c2ccc(cc2)S)O JS-3051 CN(C)/C=N/c1ccc(cc1C#N)Br JS-3052 c1ccc(cc1)Cc2nnc(n2Cc3ccccc3)SCC(=O)Nc4ccc(cc4)N5CCOCC5 JS-3053 c1cc(c(cc1F)F)NC(=O)CN2CCCCC2 JS-3054 c1cc(ccc1COc2ccc(cc2[N+](=O)[O-])C=O)Cl JS-3055 c1ccc2c(c1)C(=O)N(C2=O)CCCOc3ccc(cc3)/C(=N/O)/N KA-0206 c1ccc2c(c1)C(=O)N(C2=O)CCOc3ccc(cc3)C=O KA-0238 c1ccc2c(c1)C(=O)N(C2=O)CCCOc3ccc(cc3)C#N KA-0239 Cc1ccc(cc1)C(=O)CSC#N KA-0700 c1ccc(c(c1)C(=O)CSC#N)F KA-0701 c1cc(ccc1C(=O)CSC#N)F KA-0703 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSC#N KA-0704 c1cc(c(cc1Cl)Cl)C(=O)CSC#N KA-0706 c1cc(cc(c1)Cl)C(=O)CSC#N KA-0708 c1ccc2cc(ccc2c1)C(=O)CSC#N KA-0709 c1csc(c1Cl)C(=O)CSC#N KA-0710 c1csc(c1Br)C(=O)CSC#N KA-0711 c1cc(ncc1[N+](=O)[O-])c2ccsc2 KA-0712 c1cc(cc(c1)Cl)CSCCN.Cl KA-0714 c1cc(ccc1CSCCN)F.Cl KA-0717 c1ccc(cc1)C2NCCS2 KA-0718 CCOC(=O)c1csc(n1)c2ccc(c(c2)F)C(F)(F)F KA-0720 c1cc(c(cc1c2nc(cs2)CC(=O)O)F)C(F)(F)F KA-0721 Cc1cccc(c1)CSCCN.Cl KA-0722 CC(C)(C)c1ccc(cc1)C2NCCS2 KA-0723 c1cc(cc(c1)S(=O)(=O)N2CCCC2)C(=O)O KA-0724 c1cc(cc(c1)S(=O)(=O)N2CCCCC2)C(=O)O KA-0725 c1cc(c(cc1c2nc(cs2)C(=O)O)F)C(F)(F)F KA-0726 c1ccc(cc1)COc2ccc(cc2)C3NCCS3 KA-0727 CCc1ccc(cc1)C2NCCS2 KA-0728 COC(=O)c1cc(c(=O)n(c1)Cc2ccc(cc2)C(F)(F)F)Cl KA-0730 c1cc(ccc1Cn2cc(cc(c2=O)Cl)C(=O)O)C(F)(F)F KA-0731 c1cc(c(cc1Br)F)C2NCCS2 KA-0733 CN(C)c1ccc(cc1)C2NCCS2 KA-0734 c1cc(cc(c1)S(=O)(=O)N2CCSCC2)C(=O)O KA-0735 c1cc2c(cc1I)OCCCO2 KA-0736 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cccc(c2)C(=O)O KA-0737 CCOc1ccc(cc1)C2NCCS2 KA-0738 CCCCCCCc1ccc(cc1)C2NCCS2 KA-0739 CCOC(=O)/C(=N\O)/n1ccnc1 KA-0740 CC(=O)Nc1ccc(cc1)C2NCCS2 KA-0741 COc1ccc(cc1)C2NCCS2 KA-0742 c1cc(ccc1C2NCCS2)OC(F)(F)F KA-0743 COC(=O)c1cc(cn(c1=O)Cc2ccc(cc2)C(F)(F)F)I KA-0745 CCOC(=O)/C(=N\O)/N1CCN(CC1)c2ccccc2 KA-0746 CCOC(=O)/C(=N\O)/NCc1ccccc1 KA-0747 c1cc(cc(c1)F)NC(=O)CCl KA-0748 c1cc(ccc1C2NCCS2)C(F)(F)F KA-0749 c1cc(ccc1C2NCCS2)F KA-0750 CCOC(=O)C1CCc2c(c3cc(ccc3[nH]2)OC)C1 KA-0801 Cc1ccc(cc1N2CCNC2=O)C(=O)OC KA-0805 c1cc(c(c(c1)F)/C=N/O)F KA-0811 CCOC(=O)C1CCc2c(c3cccc(c3[nH]2)Cl)C1 KA-0813 c1ccc(cc1)CN2CCN(CC2)CCOc3ccc(cc3)CO KA-0814 c1cc(ccc1C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl KA-0815 CC(C)(C)OC(=O)N1CCC(CC1)N2CCNCC2 KA-0818 c1cc(c(c(c1)F)/C(=N/O)/Cl)F KA-0819 COC(=O)c1ccc(cc1)OCCN2CCNCC2.Cl KA-0820 c1ccc(c(c1)/C=N/O)C(F)(F)F KA-0821 c1cc(c(c(c1)F)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)F KA-0822 c1ccc(c(c1)/C(=N/O)/Cl)C(F)(F)F KA-0823 COC(=O)c1coc2c1C(=O)CCC2 KA-0826 c1ccc(c(c1)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F KA-0827 CC(N1C[C@H]2C(=O)[C@@H](C1)CN(C2)C(C)C)C KA-0830 CCCCN1CCC(=O)CC1 KA-0838 CC(=O)C1=Cc2cccc(c2OC1)OC KA-0839 c1ccc(cc1)NC(=O)c2cc(cc(n2)C(=O)Oc3ccccc3)C(F)(F)F KA-0843 CCCCN1CC2CN(CC(C1)C2=O)CCCC KA-0846 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)NN KA-0848 c1ccc(cc1)CNC(=O)c2cc(cc(n2)C(=O)Oc3ccccc3)C(F)(F)F KA-0849 CCCCN1CC2CC(C1)CN(C2)CCCC KA-0852 c1ccc(c(c1)C2=NOC(C2)CNc3c(cc(cn3)C(F)(F)F)Cl)Cl KA-0856 c1cnc(nc1C(F)(F)F)N2CCC(=O)CC2 KA-0858 c1ccc(cc1)C(=O)N2CCc3c(cnc(n3)N)C2 KA-0859 CSc1ccc(cc1)N2CCCS2(=O)=O KA-0860 c1c2c(sc1C(=O)Cl)CCC2 KA-0862 CCCC(C)NC(=O)c1cn2cc(ccc2n1)Cl KA-0900 CCOC(=O)c1cc2cc(ccc2n1C(=O)OC(C)(C)C)Br KA-0920 CCOC(=O)c1cc2cc(ccc2n1C)Br KA-0922 CC(CS(=O)(=O)c1cccc(c1)C(F)(F)F)(c2ccc(cc2)Cl)O KA-0924 COC(=O)c1ccc2c(c1)sc(n2)N KA-0925 c1cc2c(cc1[N+](=O)[O-])sc(n2)Br KA-0928 COC(=O)c1ccc(c(c1)I)Cl KA-5035 c1cc(ccc1C2=CSC3=NCCN23)Br.Br KB-0203 CCOC(=O)[C@H]1CCCN(C1)C(=O)c2ccc(cc2Cl)N3CCC(CC3)C(F)(F)F KB-0701 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)Cl)OCCN3CCC(CC3)C(F)(F)F KB-0708 c1ccc(c(c1)C(=O)/C=C/c2ccc(cc2)OCCN3CCC(CC3)C(F)(F)F)Cl KB-0709 c1cc(ccc1/C=C\C(=O)O)OCCN2CCC(CC2)C(F)(F)F KB-0713 Cn1ccnc1CCl KB-0715 Cn1c(cnc1CO)Br KB-0716 c1cc(cc(c1)C=O)CCN2CCC(CC2)C(F)(F)F KB-0717 c1ccc2c(c1)c(n[nH]2)N3C(=O)c4ccccc4C3=O KB-0720 c1c(sc(n1)N2CCC(CC2)C(F)(F)F)C=O KB-0721 CN(C)c1ccc(cc1C=O)[N+](=O)[O-] KB-0723 COC(=O)c1cccc(c1)CN2CCC(CC2)C(F)(F)F KB-0727 c1cc(ccc1c2csc(n2)N3CCC(CC3)C(=O)O)Br KB-0729 Cc1cc(ccc1S)F KB-0733 Cc1ccc(cc1S)Cl KB-0734 c1cc(c(cc1S)F)N KB-0736 Cn1c(cnc1C=O)Br KB-0739 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)CCO KB-0742 CN(CCO)S(=O)(=O)c1ccccc1 KB-0743 COC(=O)c1ccc(cc1)OCCN2CCC(CC2)C(F)(F)F KB-0745 CNc1nc2ccccc2o1 KB-0749 CNc1nc2ccccc2s1 KB-0751 CN(C)c1c(cccn1)C=O KB-0752 c1ccc(cc1)COC(=O)N2CCN(CC2)c3cnn(c(=O)c3Cl)CC(=O)O KB-0801 CC(C)(C)OC(=O)NS(=O)(=O)N1CCN(CC1)C(=O)OCc2ccccc2 KB-0802 CCOC(=O)Cn1c(=O)cc(cn1)N2CCNCC2 KB-0803 c1ccc(cc1)CN2CCCCNS2(=O)=O KB-0804 c1ccc(cc1)Cn2cc(cn2)[N+](=O)[O-] KB-0807 CCCCCCn1cc(cn1)[N+](=O)[O-] KB-0809 CCOC(=O)C1CCN(CC1)c2cc(=O)[nH]nc2 KB-0810 CCOC(=O)C1CCN(CC1)S(=O)(=O)NC(=O)OC(C)(C)C KB-0815 CCOC(=O)c1c(nc(nn1)c2c(cc(cn2)C(F)(F)F)Cl)Cl KB-5006 c1cc(ncc1C(F)(F)F)n2cc(cn2)S(=O)(=O)NCc3c(cc(cn3)C(F)(F)F)Cl KC-0005 CC(C)(C(=O)NCc1c(cc(cn1)C(F)(F)F)Cl)n2cncn2 KC-0016 c1cc(ccc1C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl)Cl KC-0027 c1cc(c(c(c1)F)C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl)F KC-0029 c1cc2ccn(c2nc1)CC(=O)NCc3c(cc(cn3)C(F)(F)F)Cl KC-0032 c1ccc(cc1)C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl KC-0033 Cc1ccc(cc1)C(=O)NCCSc2c(cc(cn2)C(F)(F)F)Cl KC-0035 Cc1cn(c(=O)[nH]c1=O)CC(=O)NCc2c(cc(cn2)C(F)(F)F)Cl KC-0040 c1cc(c(c(c1)Cl)c2nc(c3n2cc(cc3Cl)C(F)(F)F)[C@H]4N(CCS4)C(=O)Nc5ccc(cc5)Cl)Cl KC-0044 CC(=O)N1CCS[C@H]1c2c3c(cc(cn3c(n2)c4c(cccc4Cl)Cl)C(F)(F)F)Cl KC-0048 CCCNC(=O)N1CCS[C@H]1c2c3c(cc(cn3c(n2)c4c(cccc4Cl)Cl)C(F)(F)F)Cl KC-0049 c1cc(c(c(c1)Cl)c2nc(c3n2cc(cc3Cl)C(F)(F)F)[C@H]4N(CCS4)C(=O)c5ccc(cc5)Cl)Cl KC-0065 COC(=O)N1CCS[C@H]1c2c3c(cc(cn3c(n2)c4c(cccc4Cl)Cl)C(F)(F)F)Cl KC-0072 c1ccc(cc1)n2c(=O)c3cc(ccc3[nH]c2=O)Br KC-0082 Cc1c(c(=O)[nH]c(=O)n1CC(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)C#N KC-0084 CCNC(=O)Nc1ccc(cc1C(=O)OC)Br KC-0089 c1c(cnc(c1Cl)N2CCC[C@H]2C(=O)O)C(F)(F)F KC-0096 c1ccc(cc1)CN(C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)c4ccc(cc4)Cl KC-0207 c1ccc(cc1)CN(C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)c4ccccc4Cl KC-0208 c1cc2c(cc1c3cc([nH]n3)N)OCO2 KC-0209 CN(C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)c3ccc(cc3)Cl KC-0213 CN(C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)c3ccccc3Cl KC-0214 CN(C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)C3CC3 KC-0216 Cc1c(c(c(c(n1)O)C#N)C(F)(F)F)Cl KC-0700 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])n2c(c(cn2)C#N)N KC-0701 c1ccc(cc1)CNc2c3cn[nH]c3ncn2 KC-0702 c1ccc(cc1)CNc2c(c(ncn2)Cl)CO KC-0703 CC1C(=O)N(c2cc(ccc2O1)C(=O)OC)C KC-0704 c1cc2c(cc1[N+](=O)[O-])cc(o2)C(=O)NN KC-0707 COC(=O)c1c(c2cc(c(nc2s1)c3ccccn3)Br)N KC-0708 CC1C(=O)N(c2cc(ccc2O1)C(=O)O)C KC-0709 Cc1c(c(c(c(n1)O)C#N)C(F)(F)F)Br KC-0712 c1cc(c(c(c1)F)N)C(=O)O KC-0713 CC(C)(C)OC(=O)N1CCC(CC1)I KC-0717 Cc1c(c(c(c(n1)Cl)C#N)C(F)(F)F)Br KC-0719 CC(C)(C)OC(=O)Nc1ccc2c(c1)cc(o2)C=O KC-0721 c1ccnc(c1)c2ccc3c(n[nH]c3n2)N KC-0722 c1cc(nnc1I)I KC-0724 COC(=O)c1ccc(cc1C(F)(F)F)F KC-0725 COC(=O)c1c(c2ccc(nc2s1)c3ccccn3)N KC-0727 CCOC(=O)CNC1CCN(CC1)C(=O)OC(C)(C)C KC-0732 CC(C)(C)OC(=O)N1CCC(CC1)Nc2ccc(cc2)[N+](=O)[O-] KC-0737 c1cnc(nc1C#N)Cl KC-0738 CC(C)(C)/C(=N/O)/N KC-0740 c1cc(c(cc1[N+](=O)[O-])CBr)N2CCOCC2 KC-0741 CC(C)(CCC(=O)O)C(=O)OC KC-0742 COC(=O)C(c1cccc(c1)Br)N.Cl KC-0743 CC(C)(C)OC(=O)N1CCN(CC1)c2nccc(n2)C#N KC-0746 c1c(cnc(c1Cl)OC2CCNCC2)C(F)(F)F KC-0747 CC(C)(C)OC(=O)N1CCN(CC1)c2nccc(n2)/C(=N/O)/N KC-0748 Cc1nc2cc(cc(c2o1)Br)OC KC-0749 COc1cc2c(c(c1)Br)oc(n2)CCl KC-0750 c1cnc(cc1/C(=N\O)/N)Cl KC-0753 c1cc(ccc1[N+](=O)[O-])OC2CCNCC2.Cl KC-0754 c1cc(c(c(c1)Br)F)CO KC-0757 CC(C)(C)OC(=O)N1CCC(CC1)Nc2c(cc(cn2)C(F)(F)F)Cl KC-0758 c1cc(c(c(c1)Br)F)CCl KC-0761 COc1cc2c(c(c1)Br)OCC(=O)N2 KC-0763 Cn1c2c(ccc(n2)c3ccccn3)c(n1)N KC-0767 c1cnc(cc1C(=N)NN)Cl KC-0768 c1c(cnc2c1c(c[nH]2)C=O)C(F)(F)F KC-0769 COc1ccc(c(c1)OCc2ccccc2)CO KD-0008 Cn1cc(c(c1)C(F)(F)F)c2nnc(n2c3ccc(cc3)Cl)S KD-0020 c1cc(c(cc1C#N)N=O)N=O KD-0023 COc1cnc(cc1O)C=O KD-0031 COc1cnc(c(c1O)I)CO KD-0032 c1c(c(cc2c1sc(n2)CC#N)C(F)(F)F)C#N KD-0034 c1ccc(cc1)CNc2c(cc(cn2)I)C(=O)O KD-0044 CCOC(=O)c1cc(cnc1NCc2ccccc2)I KD-0057 c1c(c(cc(c1N)Br)[N+](=O)[O-])C(F)(F)F KD-0061 CC(C)(C)OC(=O)Nc1cc(c(cc1I)C#N)C(F)(F)F KD-0064 Cc1nc2cc(c(cc2s1)C#N)C(F)(F)F KD-0066 c1ccc(cc1)COc2c(cc(nc2Cl)CCl)I KD-0068 c1ccc(cc1)COc2c[nH]c(c(c2=O)I)CO KD-0073 c1ccc(cc1)COc2ccc(cc2C(=O)NN)[N+](=O)[O-] KD-0074 c1cc(nc(c1O)I)I KD-0076 c1ccnc(c1)CNS(=O)(=O)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl KD-0086 c1c(c(cc(c1N)I)Br)C(F)(F)F KD-0087 Cn1cc(c(c1)C(F)(F)F)c2nnc(n2c3ccc(cc3)Cl)SC KD-0089 c1cc(ccc1CNS(=O)(=O)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl)Cl KD-0092 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl KD-0093 c1c(cnc(c1Cl)n2cc(cn2)S(=O)(=O)N3CCC(CC3)C(F)(F)F)C(F)(F)F KD-0096 CC(=O)N1CCN(CC1)S(=O)(=O)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl KD-0097 COc1c(c(ccn1)N)Cl KD-0200 C=CCc1c(ccc2c1C(=O)CC2)O KD-0202 c1cc2c(c(c1)Cl)[nH]nc2N KD-0203 c1c(c[nH]c1C(=O)C(Cl)(Cl)Cl)[N+](=O)[O-] KD-0208 COC(=O)c1c(c(nc(n1)Cl)Cl)C(F)(F)F KD-0210 COC(=O)c1c(c(nc(n1)Cl)Cl)I KD-0214 CC1(CC1)Nc2cc(nc(n2)N)Cl KD-0215 COc1c(c(ccn1)N)I KD-0216 COc1c(cccn1)CCl KD-0217 COC(=O)c1cc(c[nH]1)[N+](=O)[O-] KD-0219 c1c(c[nH]c1C(=O)NN)[N+](=O)[O-] KD-0222 c1cnc(c(c1N)Cl)Cl KD-0223 CC1(CC1)Nc2cc(nc(n2)N)N3CC[C@H](C3)NC KD-0225 c1c(cnc(c1Cl)n2cc(cn2)S(=O)(=O)Cl)C(F)(F)F KD-0230 COc1c2cc[nH]c2ccn1 KD-0232 c1c(c[nH]c1C(=O)O)[N+](=O)[O-] KD-0233 c1c(n[nH]c1C(F)(F)F)C(=O)O KD-0237 c1c[nH]c2c1c(cnc2Cl)Br KD-0240 CC(C)(C)OC(=O)c1c(ccs1)CBr KD-0280 CN(C)/C=C/C(=O)c1cccnc1Cl KD-0700 COC(=O)c1ccc(c(n1)N)N KD-0703 c1cc2c(cc1F)cc(s2)C(=O)Cl KD-0704 c1cc2c(cc1F)cc(s2)C(=O)N KD-0705 CNc1c(ccc(c1C#N)Cl)[N+](=O)[O-] KD-0706 c1cc2c(cc1F)cc(s2)C#N KD-0707 CC(=O)n1c2ccc(cc2c(n1)Cl)N KD-0711 COC(=O)c1ccc2c(c1)NCCS2 KD-0712 c1cc(nc(c1C(F)(F)F)Cl)N2CCNCC2 KD-0713 c1cc2c([nH][nH]c2=O)nc1 KD-0714 COC(=O)c1cnc(c(c1O)[N+](=O)[O-])O KD-0715 c1ccc2c(c1)c(nc(n2)C(F)(F)F)N3CCNCC3 KD-0717 c1ccc2c(c1)c(nc(n2)C(F)(F)F)N3CCCNCC3 KD-0718 CNc1c(cc(c(n1)OC)C(=O)OC)Br KD-0719 c1cc(cc2c1cc(s2)C(=O)Cl)Br KD-0720 c1cc(c(nc1)Cl)c2ccncn2 KD-0721 c1cc(c2c(c1)[nH]nn2)N KD-0722 c1cc(cc2c1cc(s2)C(=O)N)Br KD-0724 COC(=O)c1cnc(c(c1Cl)[N+](=O)[O-])Cl KD-0725 c1cc(c2c(c1[N+](=O)[O-])[nH]nc2N)Cl KD-0726 CNc1c(cc(c(n1)OC)C(=O)O)Br KD-0727 c1cc(cc2c1cc(s2)C#N)Br KD-0728 CNc1ccc(cc1N)C(=O)OC KD-0729 Cc1c(c([nH]n1)N)C#N KD-0730 Cn1c2ccc(cc2[nH]c1=O)C(=O)OC KD-0732 Cn1cnc2c1ccc(c2)C(=O)OC KD-0733 c1cc(nc(c1CO)Br)C(F)(F)F KD-0734 C1Cc2c(nc(nc2O)S)C1 KD-0735 COc1ccc(cc1)C(=O)c2cc3cc(ccc3o2)Cl KD-0736 COC(=O)c1cnc(c(c1O)Br)O KD-0737 COc1cc(ncc1C(=O)O)Cl KD-0738 Cc1c2cc(c(=O)[nH]c2ccn1)Br KD-0739 c1cc2c(cc(c(=O)[nH]2)Br)c(c1)O KD-0740 c1cc(ccc1CO)c2ccc(cc2)C(F)(F)F KD-0742 CCOC(=O)c1cn(c(=O)cc1O)C KD-0744 CCOC(=O)c1cnc(c(c1O)Br)O KD-0745 COC(=O)c1cnc(c(c1O)I)O KD-0748 COc1ccc(cc1)/C(=C\C(=O)O)/c2cc3cc(ccc3o2)Cl KD-0749 CCOC(=O)c1cnc(c(c1Cl)Br)Cl KD-0750 C1COCc2c1c(c(s2)N)C(=O)N KD-0751 COC(=O)c1c2c(sc1N)COCC2 KD-0754 CNc1nccc(n1)c2cccnc2Cl KD-0755 c1c(c(cc(c1N)N)Cl)C(F)(F)F KD-0756 Cn1cnc2c1ccc(c2)C(=O)NN KD-0757 Cc1nc2cc(ccc2n1C)C(=O)OC KD-0758 c1ccc(cc1)C(=O)c2c3c(sc2N)COCC3 KD-0763 Cn1cnc2c1ccc(c2)C(=O)O KD-0764 c1cc(c(cc1O)C#N)F KD-0765 Cc1c2cc(c(nc2ccn1)Cl)Br KD-0767 Cc1c(c(n(n1)C)N)C#N KD-0769 CCOC(=O)c1cc(cnc1Oc2ccccc2)C(F)(F)F KD-0770 c1c(c(cc(c1Br)[N+](=O)[O-])Cl)C(F)(F)F KD-0771 c1c(c(c2c(c1Cl)CCNC2)Cl)[N+](=O)[O-] KE-0008 c1cncc2c1c(cc(c2N)[N+](=O)[O-])Cl KE-0009 c1cc(ccc1S(=O)(=O)N2C(=O)/C(=C/c3c(cc(cn3)C(F)(F)F)Cl)/NC2=O)Cl KE-0024 c1ccc2c(c1)ccn2C3CCN(CC3)Cc4ccccn4 KE-0034 CCOC(=O)C(=NNc1ccc(cc1)OC)Cl KE-0041 c1ccc(cc1)COC(=O)c2c(ccc(c2F)N)F KE-0045 COC(=O)C(=O)c1cn(c2c1cccc2)C3CCN(CC3)Cc4ccccn4 KE-0050 c1cc(c(cc1[N+](=O)[O-])C(F)(F)F)C(F)(F)F KE-0208 c1cc(c(cc1Br)Br)[N+](=O)[O-] KE-0211 CCOC(=O)CSc1nnc(s1)NC(=O)CCl KE-0212 c1cc(cc(c1)C(F)(F)F)c2cc3c(cccc3O)nc2Cl KE-0218 c1cc(cc(c1)C(F)(F)F)c2cc3c(cccc3O)nc2N4CCCC4 KE-0223 CC(=O)NC1CCc2c(sc(n2)N)C1 KE-0229 COc1ccc(cc1)CNc2ccc(cc2[N+](=O)[O-])C(=O)OC KE-0299 CCc1c(=O)[nH]c2ccccc2n1 KE-0700 CCOC(=O)c1cnc(cc1NC)Cl KE-0701 COC(=O)Cc1ccccc1F KE-0702 CC(C)(C)OC(=O)N1CCN(CC1)CC2CO2 KE-0704 c1ccc(cc1)N2CC(OC2=O)CBr KE-0706 c1ccc(c(c1)CC(=O)NN)F KE-0707 CCc1c(nc2ccccc2n1)Cl KE-0709 c1cc(nc(c1[N+](=O)[O-])N2CCCCCC2)Cl KE-0711 CC(C)(C)OC(=O)N1CCN(CC1)CC2CN(C(=O)O2)c3ccccc3 KE-0716 COc1ccccc1CC(=O)NN KE-0718 COc1cccc(c1)CC(=O)OC KE-0721 COC(=O)Cc1cccc(c1)F KE-0722 c1ccc(c(c1)CC(=O)NN)Cl KE-0723 c1cc(cc(c1)F)CC(=O)NN KE-0725 C=C1CCC(CC1)C(=O)O KE-0726 c1cc(c(cc1F)F)CC(=O)NN KE-0727 COC(=O)Cc1cccc(c1)C(F)(F)F KE-0732 COc1cccc(c1)CC(=O)NN KE-0733 c1cc(cc(c1)C(F)(F)F)CC(=O)NN KE-0734 c1c(cnc(c1Cl)N2CCC3(CC2)NC(=O)CS3)C(F)(F)F KE-0735 COc1ccc(cc1)N2CC(OC2=O)CBr KE-0736 CC(C)(CC(=O)O)CN.Cl KE-0737 COC(=O)Cc1ccc2c(c1)OCO2 KE-0750 c1cc(ccc1N2CC(OC2=O)CBr)F KE-0757 c1cc2c(cc1CC(=O)NN)OCO2 KE-0758 COc1ccc(cc1)CC(=O)NN KE-0779 c1cc(ccc1CC(=O)NN)Cl KE-0780 CC(C)(C)OC(=O)N1CCN(CC1)CC2CN(C(=O)O2)c3ccc(cc3)OC KE-0799 CC(=O)Nc1ccc(c(c1)Cl)OC KE-0835 CC(=O)Nc1cc(c(cc1[N+](=O)[O-])OC)Cl KE-0840 CC(C)(C)OC(=O)NC1CCN(C1)CC2CN(C(=O)O2)c3ccccc3 KE-0869 c1c(cnc(c1Br)Cl)C(=O)N KE-0871 COc1cc(c(cc1Cl)N)[N+](=O)[O-] KE-5001 c1c2c(cc(c1Br)Br)nc([nH]2)Cl KE-5002 COc1cc(c(cc1Cl)n2cccc2)[N+](=O)[O-] KE-5003 Cc1c(=O)n(c2ccc(cc2n1)C(=O)O)C KE-5004 c1cc(ccc1CN2CCCC2)C(=O)O.Cl KF-0002 c1c(cnc(c1Cl)NCCc2cn(cn2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F KF-0007 c1cc(c(cc1Cl)F)N2CC3(CCNCC3)OC2=O KF-0010 Cc1c(ccc(c1C(=O)O)Br)OC KF-0014 COc1cc2c(cc1O)ncnc2Nc3ccc(cc3F)Br KF-0017 C[C@@H]1CN(C[C@@H](O1)C)Cc2cc(=O)oc3c2ccc(c3)O KF-0021 CCOC(=O)Cc1c(cc(cn1)C(F)(F)F)Cl KF-0029 Cc1c(ccc(c1C(=O)OC)Br)OC KF-0031 c1cc2c(cc(=O)oc2cc1O)CN3CCOCC3 KF-0034 c1ccc2c(c1)cc(c(=O)o2)c3c(cc(cn3)C(F)(F)F)Cl KF-0040 c1cc(ccc1N2CC3(CCNCC3)OC2=O)F KF-0044 c1cc2c(cc1Cl)cc(c(=O)o2)c3c(cc(cn3)C(F)(F)F)Cl KF-0054 c1cc2c(cc(=O)oc2cc1O)CN3CCCC3 KF-0058 CC(C)NC(=O)C1(CC1)c2c(cc(cn2)C(F)(F)F)Cl KF-0064 Cc1cc(c(cc1OC)C(=O)O)Br KF-0071 c1cc(ccc1NC(=O)C2(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl KF-0074 c1cc(ccc1NNC(=O)C2(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl KF-0076 Cc1cc(c(cc1OC)C(=O)OC)Br KF-0079 c1ccc(cc1)CNC(=O)C2(CC2)c3c(cc(cn3)C(F)(F)F)Cl KF-0082 CN(Cc1ccccc1)C(=O)C2(CC2)c3c(cc(cn3)C(F)(F)F)Cl KF-0083 CC(C)(C)OC(=O)C1CCC(CC1)COc2cc3c(cc2OC)c(ncn3)Nc4ccc(cc4F)Br KF-0099 CC(C)(C)OC(=O)N1CCC2(CC1)CC2C#N KF-0200 c1ccc(cc1)CN2CCC(=CC#N)CC2 KF-0234 c1cc(c(cc1Br)C=O)[N+](=O)[O-] KF-0237 c1ccc(cc1)CN2CCC(CC2)CC#N KF-0239 CC(C)(C)OC(=O)N1CCC(=O)C(C1)C(=O)C(F)(F)F KF-0702 c1c2cc(c(nc2ncc1Cl)N3CCCCC3)C#N KF-0705 CCOC(=O)C1(CC1)S(=O)(=O)C KF-0706 CNc1c(cc2cc(cnc2n1)Cl)C#N KF-0707 CN(C)C(=O)c1ccc[nH]1 KF-0708 c1cc(c2c(c1[N+](=O)[O-])[nH]nc2Br)F KF-0711 Cc1c(cc(c(n1)OC)Br)C(=O)C KF-0712 CC(C)(C)OC(=O)N1CCc2c(c(n[nH]2)C(F)(F)F)C1 KF-0716 c1cnc2c(c1C(F)(F)F)c(n[nH]2)N KF-0720 CN(C)c1c(cc2cc(cnc2n1)Cl)C#N KF-0721 CNCc1ccccc1O KF-0722 CCOC(=O)/C(=C/N(C)C)/S(=O)(=O)C KF-0723 c1ccn2c(c1)nccc2=O KF-0724 COC(=O)c1c(c2cc3cc(cnc3nc2s1)Cl)N KF-0732 c1nc(c(s1)C=O)Cl KF-0733 CS(=O)(=O)c1ccc(c(n1)Br)N KF-0735 CC(C)(C)n1c2c(c(ncn2)N)c(n1)Br KF-0737 CS(=O)(=O)c1c(cccn1)C=O KF-0738 COc1c(cc(cc1I)Br)CO KF-0739 c1c2cc(c(nc2ncc1I)N)C#N KF-0742 CC(C)(C)c1ccnc(n1)N KF-0744 CS(=O)(=O)c1ccc(cc1C#N)C=O KF-0747 c1c(cnc(c1Cl)C(=O)O)C(=O)N KF-0748 c1ccc2c(c1)CC=C2C(=O)O KG-0002 CC(C)(C)OC(=O)N1CC2CNCC2C1 KG-0017 Cc1ccc(cc1)CN2CCC(=CC2)C(=O)OC KG-0024 CC(C)(C)OC(=O)N1CC2CN(CC2C1)C(=O)c3ccc(o3)Cl KG-0027 c1cc(c(cc1CC(=NO)C(=O)O)Br)O KG-0028 c1ccc(cc1)[P+](CC(F)(F)F)(c2ccccc2)c3ccccc3.C(F)(F)(F)S(=O)(=O)[O-] KG-0036 CC#CCn1c2c(nc1Br)n(c(=O)n(c2=O)Cc3nc(c4ccccc4n3)C)C KG-0209 COc1cc(ncc1CO)Cl KG-0700 c1ccc(c(c1)n2cccc2CO)F KG-0701 Cc1c(cc(c(=O)[nH]1)Cl)C(=O)C KG-0702 Cc1c(cc(c(=O)[nH]1)I)C(=O)C KG-0703 COC(=O)c1ccc(c(c1)F)N(Cc2ccccc2O)c3c(cc(cn3)C(F)(F)F)Cl KG-0704 c1c(ncc(c1Cl)/C=N/N=C/c2c(cc(nc2)Cl)Cl)Cl KG-0708 CCOC(=O)c1c(c(ccn1)c2ccccc2)C#N KG-0709 c1ccc(cc1)c2ccnc(c2C#N)C(=O)O KG-0710 COc1cc(ncc1C=O)Cl KG-0711 CCOC(=O)c1ccc(cn1)CN2CCN(CC2)C KG-0712 Cc1c(cc(c(n1)Cl)I)C(=O)C KG-0713 CCOC(=O)c1cc(c(cn1)C(F)(F)F)Cl KG-0715 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cncc2Br)[N+](=O)[O-] KG-0716 CCOC(=O)c1ccc(nc1Cl)Cl KG-0717 c1c(c(cnc1C(=O)O)C(F)(F)F)Cl KG-0719 COc1cc(cc(c1)OC)/C=C/c2ccc(cc2)[N+](=O)[O-] KH-0004 c1cc(ncc1c2ncc3n2cc(cc3Cl)C(F)(F)F)Cl KH-0025 Cc1c(cc(n1C)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)N3CCOCC3 KH-0072 CCOC(=O)c1cc(=O)c2cc(cc(c2o1)N)Br KH-0080 CN(c1ccccc1)c2ncc3n2cc(cc3Cl)C(F)(F)F KH-0211 CNc1ccc(cc1[N+](=O)[O-])C(=O)N KH-0701 COC(=O)C(c1ccc(cc1)O)N KH-0702 COc1ccc(cc1)/C=C(\CC(=O)O)/C(=O)OC KH-0704 c1cc(c(cc1C(=O)N)N)N KH-0709 CNc1ccc(cc1N)C(=O)N KH-0710 c1cc(c(cc1CCl)[N+](=O)[O-])[N+](=O)[O-] KH-0711 CCCCc1[nH]c2cc(ccc2n1)C(=O)OC KH-0712 c1cc(c(cc1CO)N)N KH-0713 Cc1cc(cnc1Cl)CO KH-0720 c1cc2cnc(cc2cc1Br)Cl KH-0723 Cc1cc(cnc1Cl)C(=O)O KH-0724 CCOC(=O)c1ccc(cn1)F KK-0202 CCOC(=O)C=C1CC2CCC(C1)N2C(=O)OCC KK-0209 CC(=O)N[C@@H](Cc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl)C(=O)OC KK-0701 CC(=O)NC(Cc1c(ccc(c1F)F)F)C(=O)OC KK-0702 CC(=O)NC(Cc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl)C(=O)OC KK-0703 Cc1cc(cc(c1/C=C(/C(=O)OC)\N)C)OC(=O)C KK-0705 c1c(c(cnc1C(F)(F)F)C(=O)O)Cl KK-0707 Cc1cc(cc(c1CC(C(=O)OC)NC(=O)C)C)O KK-0709 CCOC(=O)C(Cc1ccc(cc1)N)N2C(=O)c3ccccc3C2=O KK-0712 C1C(CNC(=O)N1)O KK-0713 COC(=O)C1(CCCCC1)N KL-0010 Cc1ccc(cc1)S(=O)(=O)O.c1ccc(cc1)C2(CCNCC2)C(=O)O KL-0021 CC(c1cc(cc(c1)/c/2c\3/nc(/c(c/4\[nH]/c(c(\c5n/c(c(\c6[nH]c2cc6)/c7cc(cc(c7)C(C)(C)C)C(C)(C)C)/C=C5)/c8cc(cc(c8)C(C)(C)C)C(C)(C)C)/cc4)/c9cc(cc(c9)C(C)(C)C)C(C)(C)C)C=C3)C(C)(C)C)(C)C KL-0022 CC(=O)Nc1cc(c(cc1NC(=O)C)Cl)N(=O)=O KM-0007 Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2N)Cl)N(=O)=O KM-0008 Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2NS(=O)(=O)c3ccc(cc3)C)Cl)N(=O)=O KM-0010 c1c(c(cnc1Cl)CCl)Cl KM-0018 c1c(c(cnc1Cl)CBr)Cl KM-0022 c1[nH]c2c(n1)c(nc(n2)Cl)Cl KS-1014 COc1ccccc1OCCN.Cl KS-1024 c1ccc(cc1)Oc2ccc(cc2CC(=O)O)Cl LA-0005 CN(c1ccsc1C(=O)OC)C(=O)c2ccc(cc2)Br LA-0208 Cc1cn(c(=O)[nH]c1=O)CC=C LA-0209 c1ccc(cc1)CN2C(C(CCC2=O)C(=O)O)c3ccc4c(c3)OCO4 LA-0213 CC(C)(C)c1ccc(cc1)C2C(CCC(=O)N2Cc3ccccc3)C(=O)O LA-0218 CC(C)(C)OC(=O)C[C@@H](C(=O)N[C@@H](Cc1ccccc1)C(=O)N)NC(=O)OCC2c3ccccc3-c4c2cccc4 LA-0225 CS(=O)(=O)OCCCOS(=O)(=O)C LA-0600 c1cc(ccc1C2NCCS2)OCCCF LA-0700 COC(=O)c1cc2ccc(cc2s1)Br LA-0701 c1cc(ccc1C2NCCS2)OCCBr LA-0703 c1cc(sc1C=O)N2CCSCC2 LA-0704 c1cc(ccc1Cn2cc(cc(c2=O)C(=O)O)I)C(F)(F)F LA-0708 COc1ccc2cc[nH]c2c1 LA-0711 CCCCCCN1CCC(=O)CC1 LA-0800 C1CCC(CC1)N2CCC(=O)CC2 LA-0801 c1ccc(cc1)CNC(=O)c2cc(cc(n2)C(=O)OCc3ccccn3)C(F)(F)F LA-0805 CC(C)(C)C(=O)Nc1cccc(n1)N LA-0807 Cn1cccc(c1=S)C(=O)NN LA-0811 C1CC1N2CCC(=O)CC2 LA-0813 CC(C)CCN1CCC(=O)CC1 LA-0814 CCNC(=O)c1cc(cc(n1)C(=O)OCc2ccccc2)C(F)(F)F LA-0818 CCNC(=O)c1cc(cc(n1)C(=O)OCc2ccccn2)C(F)(F)F LA-0819 c1ccc(cc1)CNC(=O)c2cc(cc(n2)C(=O)OCc3ccccc3)C(F)(F)F LA-0826 c1ccc(cc1)COCCN LA-0829 c1cc(c2c(c1)oc(n2)CCl)[N+](=O)[O-] LA-0846 c1cc2c(cc1Br)c(c([nH]2)C(=O)O)Br LA-0921 c1cc2c(cc1Br)c(c([nH]2)NN)Br LA-0922 c1cc2c(cc1Br)cc([nH]2)C=O LA-0923 c1cc(ccc1C(=O)NNCc2c(cc(cn2)C(F)(F)F)Cl)Cl LB-0016 c1ccc(cc1)C(=O)NNCc2c(cc(cn2)C(F)(F)F)Cl LB-0033 c1cc(c(c(c1)Cl)C(=O)NNCc2c(cc(cn2)C(F)(F)F)Cl)Cl LB-0040 COc1ccc(cc1)C(=O)NNCc2c(cc(cn2)C(F)(F)F)Cl LB-0041 c1cc(ccc1NC(=O)c2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl LB-0045 c1ccc(cc1)c2ccccc2NC(=O)c3ccnc(n3)c4c(cc(cn4)C(F)(F)F)Cl LB-0046 c1cc(ccc1CNC(=O)c2cc(c(nc2)Cl)I)F LB-0200 CC(C)c1nc2ccc(cc2c(=O)o1)Br LB-0201 c1cc(ccc1C2=C(SC3=NCCN23)Br)Br.Br LB-0208 c1ccc(cc1)CN2CC3CCCC(=O)C3C2 LB-0216 c1c(c(c(c(c1[N+](=O)[O-])F)F)F)C(=O)O LB-0607 CS(=O)(=O)c1c(nc(s1)N)c2ccc(cc2)Br LB-0701 c1cc(ncc1CO)C(F)(F)F LB-0702 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cc(cn2)Br)C(=O)OC LB-0703 COc1ccc(cc1)NC(c2cccs2)C(=O)O LB-0704 COC(=O)CC(c1ccc2c(c1)OCO2)N.Cl LB-0706 c1cc(ccc1c2c(sc(n2)N)Br)Br.Br LB-0710 c1c(c[nH]c1C=O)C(=O)CN2CCC(CC2)C(F)(F)F LB-0712 CN(C)S(=O)(=O)c1cccc(c1)C(=O)O LB-0714 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cc(cn2)C(=O)OC)Br LB-0715 CNS(=O)(=O)c1cccc(c1)C(=O)O LB-0716 c1cc(ncc1C=O)C(F)(F)F LB-0717 c1cc(c(cc1CO)N)F LB-0721 COC(=O)c1c(c2ccc(cc2s1)Br)N LB-0725 CS(=O)(=O)N1CCC(CC1)C(=O)Cl LB-0726 COC(=O)CN1CCC(CC1)C(F)(F)F LB-0730 c1c(cnc(c1CCl)Cl)Br LB-0731 c1cc(ccc1c2cc([nH]n2)N)F LB-0732 COc1c(cc(cn1)Br)C(=O)OC LB-0733 COc1cc(ccc1[N+](=O)[O-])F LB-0734 CN(C)c1ccc(cc1[N+](=O)[O-])C=O LB-0735 c1cc(ncc1CCl)C(F)(F)F LB-0736 c1cc(ccc1c2c(sc(n2)N)Br)F.Br LB-0737 CC(C)(C)OC(=O)N(Cc1ccccc1)S(=O)(=O)N2CCCC(C2)C(=O)O LB-0801 CC(C)(C)OC(=O)NS(=O)(=O)Nc1cccc(c1)C#N LB-0803 CC(C)(C)OC(=O)NS(=O)(=O)Nc1nccs1 LB-0804 CC(C)(C)OC(=O)NS(=O)(=O)Nc1cccnc1 LB-0805 CC(C)(C)OC(=O)NS(=O)(=O)Nc1ccc(cc1)C(=O)OC LB-0806 C#CCN1CCC(CC1)C(F)(F)F LB-0807 CC(C)(C)OC(=O)N(CCBr)S(=O)(=O)N1CCN(CC1)C(=O)OCc2ccccc2 LB-0809 c1ccc(cc1)CN2CCNS2(=O)=O LB-0810 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2ccc(s2)Br LB-0811 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2cc(cnc2)Br LB-0812 c1cnccc1C2NCCS2 LB-0815 c1cc(sc1C(=O)N2CCNCC2)Br LB-0816 c1ccc2c(c1)c(ncn2)NN LB-0817 c1c(cnc(c1Cl)Cn2cc(cn2)N)C(F)(F)F LB-5002 c1cc(ccc1NC(=O)Nc2cnn(c2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl LB-5004 CCNC(=O)Nc1cnn(c1)Cc2c(cc(cn2)C(F)(F)F)Cl LB-5007 c1cc(ccc1C(=O)Nc2cnn(c2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl LB-5017 c1ccc(c(c1)C(=O)Nc2cnn(c2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl LB-5018 CCC(=O)Nc1cnn(c1)Cc2c(cc(cn2)C(F)(F)F)Cl LB-5019 c1c(cnc(c1Cl)Cn2cc(cn2)NC(=O)C(F)(F)F)C(F)(F)F LB-5021 c1ccc(c(c1)S(=O)(=O)Nc2cnn(c2)Cc3c(cc(cn3)C(F)(F)F)Cl)Cl LB-5025 CCS(=O)(=O)Nc1cnn(c1)Cc2c(cc(cn2)C(F)(F)F)Cl LB-5029 c1c(cnc(c1Cl)Cn2cc(cn2)NS(=O)(=O)C(F)(F)F)C(F)(F)F LB-5031 CCn1c(=O)c2cc(ccc2[nH]c1=O)Br LC-0006 CS(=O)(=O)N1CCS[C@H]1c2c3c(cc(cn3c(n2)c4c(cccc4Cl)Cl)C(F)(F)F)Cl LC-0017 CNS(=O)(=O)NCc1c(cc(cn1)C(F)(F)F)Cl LC-0043 CC(C(=O)N)Oc1cccc(c1)OC LC-0072 c1cc(ccc1CNS(=O)(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl LC-0084 c1cc(c(c(c1)Cl)CNS(=O)(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl LC-0094 CCOC(=O)CCCCN1CC(=O)C2CCCN2C1=O LC-0097 C1CC2C(=O)NC(=O)N2C1 LC-0098 CNS(=O)(=O)N(Cc1cc(cc(c1)Cl)Cl)Cc2c(cc(cn2)C(F)(F)F)Cl LC-0107 c1cc(ccc1C(=O)CNS(=O)(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl LC-0108 CCOC(=O)c1cc2ccccc2o1 LC-0201 CC(C)NC(=O)N(C)C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl LC-0207 CN(C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccc(cc3)Cl LC-0208 CC(C)C(=O)N(C)C1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl LC-0210 CSc1nccc(n1)/C(=N/O)/C(=O)c2ccc(c(c2)Cl)Cl LC-0215 COC(=O)c1cc(ccc1F)[N+](=O)[O-] LC-0701 CN(C)C(=O)c1cc(c[nH]1)I LC-0702 CN1CCN(CC1)c2ccc(cc2C(=O)OC)[N+](=O)[O-] LC-0703 CC1C(=O)Nc2cc(cc(c2O1)Br)OC LC-0708 c1cnc(nc1C#N)N2CCNCC2 LC-0711 c1cc(ccc1c2nc(on2)CCl)Br LC-0712 CN1CCN(CC1)c2ccc(cc2C(=O)OC)N LC-0713 CC(C)(C)OC(=O)N1CCC(CC1)Oc2cc(ccn2)C#N LC-0714 Cc1[nH]c(nn1)N LC-0715 CNc1ccc(cc1N)[N+](=O)[O-] LC-0716 CN1CCN(CC1)c2ccc(cc2CO)N LC-0718 CC(C)(C)OC(=O)N1CCCCC1C=O LC-0719 COC(=O)c1ccc(cc1Br)N2CCOCC2 LC-0720 c1ccc(cc1)CN2CCCC(C2)C(=O)O.Cl LC-0722 c1ccc(cc1)COc2ccc(cc2Br)C=O LC-0725 c1cc([nH]c(=O)c1C#N)C2CC2 LC-0726 CCOC(=O)c1cn2cc(nc2s1)c3ccccc3.Br LC-0727 c1ccnc(c1)c2ccc(c(=O)[nH]2)C(=O)O LC-0732 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(c(c2)C(=O)OC)[N+](=O)[O-] LC-0733 c1cc(c(cc1N)CO)N2CCOCC2 LC-0736 c1c(c(=O)[nH]c(c1Br)C2CC2)C#N LC-0738 Cn1c(=O)n2c(n1)ccc(n2)Cl LC-0746 c1ccc(cc1)COc2ccc(cc2Br)CO LC-0748 Cn1cnc2c1ccc(c2)[N+](=O)[O-] LC-0749 CCc1nc2cc(cc(c2o1)Br)OC LC-0752 c1ccc(cc1)COc2ccc(cc2Br)/C=C/C(=O)O LC-0755 CCc1nc2cc(ccc2n1C)[N+](=O)[O-] LC-0757 c1ccc(cc1)c2cn3cc(sc3n2)C(=O)O.Cl LC-0761 CN(C)c1ccc(cc1N)[N+](=O)[O-] LC-0762 c1cc(ccc1COc2ccc(cc2Br)C=O)F LC-0763 COc1cc(ccn1)C(=O)OC LC-0768 COC(=O)c1cc(ccc1[N+](=O)[O-])Cl LC-0770 COc1cc(ccn1)C(=O)NN LC-0771 CC1CN(CC(O1)C)c2ccc(c(c2)OC)[N+](=O)[O-] LC-0776 c1ccc(cc1)COc2ccc(nc2Cl)CO LD-0003 c1ccc(cc1)COc2ccc(nc2Cl)C=O LD-0010 c1c[nH]c2c1cc(c(c2)C(F)(F)F)Br LD-0012 c1ccc(cc1)COc2ccc(nc2Br)C=O LD-0016 c1cc(ccc1S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3cnn(c3)c4c(cc(cn4)C(F)(F)F)Cl)Cl LD-0018 c1cc(ccc1NC(=O)N2CCN(CC2)S(=O)(=O)c3cnn(c3)c4c(cc(cn4)C(F)(F)F)Cl)Cl LD-0019 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])c2n[nH]nn2 LD-0021 CC(C)NC(=O)N1CCN(CC1)S(=O)(=O)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl LD-0022 CS(=O)(=O)N1CCN(CC1)S(=O)(=O)c2cnn(c2)c3c(cc(cn3)C(F)(F)F)Cl LD-0023 COC(=O)c1cc(cc(c1O)I)Br LD-0027 COC(=O)c1c2ccc(cc2cc(c1O)Br)Br LD-0032 COc1ccc(nc1Br)CO LD-0033 COc1ccc(nc1Br)C=O LD-0041 COc1c(cc2cc(ccc2c1C(=O)OC)Br)Br LD-0047 c1ccc(cc1)COc2c(cc(nc2Br)CO)I LD-0048 COc1ccc(nc1I)I LD-0049 c1cc(c(cc1[N+](=O)[O-])C(F)(F)F)c2n[nH]nn2 LD-0050 C[Si](C)(C)C#Cc1cccc2c1C(=O)C(=O)N2 LD-0051 c1cc(ccc1NC(=O)c2c(cnc(c2Cl)Cl)C(F)(F)F)Cl LD-0058 c1cc(ccc1CNC(=O)c2c(cnc(c2Cl)Cl)C(F)(F)F)Cl LD-0059 C#Cc1cccc2c1C(=O)C(=O)N2 LD-0064 c1c(c(cc(c1N)Br)Br)C(F)(F)F LD-0065 c1c(c(cc(c1N)Br)Cl)C(F)(F)F LD-0070 c1cc(ccc1NC(=O)c2c(cnc(c2Cl)N)C(F)(F)F)Cl LD-0077 c1ccc(cc1)COc2c[nH]c(c(c2=O)Br)CO LD-0080 CN1CCN(CC1)C(=O)c2c(cnc(c2Cl)N)C(F)(F)F LD-0082 c1cc(c(cc1c2n[nH]nn2)C(F)(F)F)[N+](=O)[O-] LD-0084 c1ccc(cc1)c2nc(cc(n2)O)C(=O)O LD-0088 c1cc2c(cc1Br)CC(=O)N2 LD-0089 c1cc2c(c(c1)I)/C(=N/N)/C(=O)N2 LD-0093 COc1ccccc1CCNC(=O)C(F)(F)F LD-0094 c1cc2c(cc1Br)C3(CCCCC3)C(=O)N2 LD-0097 COc1c(cc(cc1[N+](=O)[O-])[N+](=O)[O-])CCNC(=O)C(F)(F)F LD-0098 c1c(cnc(c1C(F)(F)F)CN)Cl.Cl LD-0099 COc1c(cc(cn1)Br)[N+](=O)[O-] LD-0202 c1c(c(cnc1Cl)I)N LD-0208 c1cnc(c(c1N)I)Cl LD-0209 COc1c(cc(cn1)Br)N LD-0211 CCOC(=O)c1c(c([nH]n1)C(F)(F)F)Br LD-0212 COc1c2c(cc[nH]2)c(cn1)Br LD-0213 COC(=O)c1cc(c[nH]1)N.Cl LD-0220 c1c(c[nH]c1CO)[N+](=O)[O-] LD-0226 c1(c(n[nH]c1C(F)(F)F)C(=O)O)Br LD-0231 COC(=O)c1cc(c[nH]1)Cl LD-0232 COC(=O)c1cc(ccn1)N LD-0238 COC(=O)c1cc(c([nH]1)Cl)Cl LD-0244 C1CNCCC1N2CCS(=O)(=O)CC2 LD-0249 c1c(c(c(c(n1)Cl)Cl)N)C(F)(F)F LD-0250 c1cc(ccc1c2cc(c(nc2)N)[N+](=O)[O-])F LD-0251 c1cnc(c(c1C(F)(F)F)Cl)Cl LD-0253 C[Si](C)(C)C#Cc1cnc(cc1N)Cl LD-0284 c1cc(nc(c1C=O)Br)C(F)(F)F LD-0700 Cc1c(c2nc(cc(n2n1)O)C(F)(F)F)C#N LD-0702 CC(C)(C)OC(=O)N1CCC(CC1)(CN(Cc2ccccc2)Cc3ccccc3)O LD-0704 c1c(c(cc(c1Br)N)Cl)C(F)(F)F LD-0705 c1c(cnc(c1Cl)Cl)C(=O)N LD-0707 CCOC(=O)c1cc(cnc1C#N)C(F)(F)F LD-0708 Cc1c(c(n(n1)C)N)C(=O)N LD-0709 Cc1c(c2nccc(n2n1)N)C#N LD-0710 Cn1c2c(ccc(c2c(n1)N)Cl)[N+](=O)[O-] LD-0711 c1ccc(cc1)CN(Cc2ccccc2)CC3(CCNCC3)O LD-0712 c1cc(c(cc1Br)O)C(=O)NO LD-0716 c1cc2c(nc1)NCCO2 LD-0717 c1cc(c(cc1[N+](=O)[O-])CO)F LD-0719 Cc1c(c([nH]n1)N)C(=O)N.OS(=O)(=O)O LD-0721 c1cc2c(cc1Br)onc2O LD-0722 Cc1c2c(=O)[nH]cnc2n(n1)C LD-0723 CNc1ccc(cc1C(=O)OC)[N+](=O)[O-] LD-0724 c1ccc(cc1)c2nc3cc(c(cc3n2O)Cl)C(F)(F)F LD-0725 Cc1c2c([nH]c(=O)[nH]c2=O)n(n1)C LD-0727 c1c(c(c(c(n1)Cl)[N+](=O)[O-])Cl)C(=O)O LD-0728 COc1cc(cc(c1N)Br)C(=O)OC LD-0730 c1c(c(cnc1Cl)C(=O)N)Cl LD-0731 CCOC(=O)c1cnc(c(c1Cl)N)Cl LD-0733 CCOC(=O)c1cnc(c(c1N)[N+](=O)[O-])Cl LD-0734 COc1cc(ccc1I)C(=O)OC LD-0737 Cc1c2c(ncnc2Cl)n(n1)C LD-0738 c1c(c(cnc1Cl)C#N)Cl LD-0739 CCOC(=O)c1cn(c(=O)cc1Cl)C LD-0740 c1cnc(c(c1C(=O)N)Cl)Cl LD-0744 c1cnc(c(c1CO)Cl)Cl LD-0745 COC(=O)c1cnc(cc1NN)Cl LD-0747 c1cnc(c(c1C#N)Cl)Cl LD-0748 COc1cc(ccc1I)C(=O)O LD-0749 c1c(c(cnc1Cl)CO)Cl LD-0751 c1cc(c(cc1Cl)Cl)c2c(c[nH]n2)c3c(cc(cn3)C(F)(F)F)Cl LE-0006 Cc1cc(c(cc1F)[N+](=O)[O-])OC LE-0017 CCCS(=O)(=O)Nc1ccc(c(c1F)C(=O)OCc2ccccc2)F LE-0019 CCCS(=O)(=O)Nc1ccc(c(c1F)C(=O)O)F LE-0024 c1cc(ccc1NC(=O)NCCc2c(cc(cn2)C(F)(F)F)Cl)Cl LE-0026 COc1cccc(c1)C(=O)NCCc2c(cc(cn2)C(F)(F)F)Cl LE-0030 CCCC(=O)OCCCCO LE-0059 c1c(cnc(c1Cl)CCNS(=O)(=O)C(F)(F)F)C(F)(F)F LE-0061 CCOC(=O)C(c1cc(c(cc1[N+](=O)[O-])F)C)C(=O)OCC LE-0063 CCOC(=O)C1CCN(CC1)c2cc(c(cc2[N+](=O)[O-])F)C.Cl LE-0064 COC(=O)NCCc1c(cc(cn1)C(F)(F)F)Cl LE-0068 CN(C)C(=O)NCCc1c(cc(cn1)C(F)(F)F)Cl LE-0069 CCNC(=O)NCCc1c(cc(cn1)C(F)(F)F)Cl LE-0070 Cc1cc(c(cc1F)[N+](=O)[O-])N(C)CC(=O)O LE-0083 c1c(cnc(c1Cl)CCNC(=O)C(F)(F)F)C(F)(F)F LE-0087 Cc1cc(c(cc1F)[N+](=O)[O-])CC(=O)O LE-0090 CCCC(=O)OCCCCO[N+](=O)[O-] LE-0092 COc1cc2c(cc1Cl)-n3cccc3C4(N2)CCNCC4.Cl LE-0704 COc1cc(cc(c1OC)OC)CC(=O)OC LE-0705 c1cscc1C=C(C#N)C(=O)O LE-0709 c1c(csc1C=C(C#N)C(=O)O)Br LE-0710 CNc1cc(ncc1CO)Cl LE-0711 Cn1c2ccccc2nc1CCl LE-0712 COc1cc(cc(c1OC)OC)CC(=O)NN LE-0713 CCOC(=O)c1cnc(c(c1NC)[N+](=O)[O-])Cl LE-0714 c1cc(oc1)C=C(C#N)C(=O)O LE-0716 c1cc(ccc1Cc2nnc(o2)O)Cl LE-0717 COc1cc(cc(c1OC)OC)c2nnc(o2)O LE-0720 c1cc(c(cc1Cl)Cl)c2nnc(o2)O LE-0721 Cc1ccc(cc1)c2nnc(o2)O LE-0722 c1ccc(cc1)c2nnc(o2)O LE-0723 c1cc(c(cc1F)F)Cc2nnc(o2)O LE-0729 CCOC(=O)c1cnc([nH]c1=O)c2ncccn2 LE-0730 Cc1nc(c(c(n1)Cl)Cl)Cl LE-0732 CC(C)(C)OC(=O)N1CCN(CC1)CC2CN(C(=O)O2)c3ccc(cc3)F LE-0733 c1cc2c(cc(=O)oc2cc1O)CN3CCC(CC3)CO LF-0001 Cc1ccc(cc1C)NCC2(CCN(CC2)C(=O)OCc3ccccc3)O LF-0002 CS(=O)(=O)N1CCN(CC1)C(=O)c2cc3cc(cnc3[nH]2)C(F)(F)F LF-0006 c1ccc(cc1)COC(=O)N2CCC(CC2)(CNc3ccc(cc3Cl)Cl)O LF-0010 Cc1cc(c(cc1OC)C(=O)OC)C#N LF-0018 CC(C)(C(=O)N(C)c1ccc(cc1)Cl)Nc2c(cc(cn2)C(F)(F)F)Cl LF-0020 Cc1ccc(cc1C)N2CC3(CCN(CC3)C(=O)OCc4ccccc4)OC2=O LF-0021 Cc1ccc(cc1C)NCC2(CCNCC2)O LF-0022 C[C@H]1CNCCN1Cc2cc(=O)oc3c2ccc(c3)O.O.Cl.Cl.Cl LF-0024 COc1cc(ccc1F)C(=O)OC LF-0029 COc1cc(c(cc1F)Br)C(=O)OC LF-0032 Cc1c(ccc(c1C(=O)OC)C#N)OC LF-0033 c1cc(c(cc1Cl)Cl)NCC2(CCNCC2)O LF-0035 c1ccc(cc1)COC(=O)N2CCC3(CC2)CN(C(=O)O3)c4ccc(cc4Cl)Cl LF-0038 Cc1ccc(cc1C)N2CC3(CCNCC3)OC2=O LF-0043 c1ccc(c(c1)S(=O)(=O)NC(=N)c2c(cc(cn2)C(F)(F)F)Cl)Cl LF-0051 c1cc(c(c(c1)F)S(=O)(=O)NC(=N)c2c(cc(cn2)C(F)(F)F)Cl)F LF-0053 c1cc(cc(c1)S(=O)(=O)NC(=N)c2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] LF-0054 COc1ccc(cc1OC)NCC2(CCN(CC2)C(=O)OCc3ccccc3)O LF-0061 c1cc(c(cc1Cl)Cl)N2CC3(CCNCC3)OC2=O.Cl LF-0067 c1c(cnc(c1Cl)CN\2CCN/C2=C\[N+](=O)[O-])C(F)(F)F LF-0072 CC(C)(C)OC(=O)N1CCCc2c1c[nH]n2 LF-0076 Cc1cc2c(cc1OC)C(=O)NC2 LF-0088 c1cc(sc1S(=O)(=O)NC(=N)c2c(cc(cn2)C(F)(F)F)Cl)Cl LF-0091 c1cc(ccc1C(=O)NC(=S)Nc2ccc(cn2)C(F)(F)F)Cl LF-0095 c1c(c(cc(c1O)F)Br)C(=O)O LF-0096 c1cc(ccc1C(=O)Nc2nc3c(s2)cc(cn3)C(F)(F)F)Cl LF-0101 c1ccc2c(c1)ncc(n2)Br LF-0206 Cc1c(sc(n1)C=O)Br LF-0216 c1c(cc(cc1C#N)F)C=O LF-0225 Cn1c(cnc1Br)C(=O)OC LF-0227 CN(C(=O)c1cc(cc(c1)I)[N+](=O)[O-])OC LF-0228 C1CNC[C@@H]1O LF-0500 c1ccc(cc1)C2CCNC2.Cl LF-0502 C1CCN(C1)C(=N)N.I LF-0503 C1CC2CNCC2C1.Cl LF-0504 C1CNCC1NC(=O)C(F)(F)F.Cl LF-0505 CCN1CCCC1CN LF-0506 CNC1CCN(C1)Cc2ccccc2 LF-0507 C1CCN(C1)CCCN LF-0508 c1ccc(cc1)CC2CCNCC2 LF-0509 c1ccc(cc1)CN2CCC(CC2)N LF-0510 c1ccc(cc1)C2(CCNCC2)C#N.Cl LF-0511 c1ccc(cc1)C2CCNCC2 LF-0512 C1CNCCC1N LF-0513 CC1CCCCN1CCCN LF-0514 C1CC2(C1)CCNCC2.Cl LF-0515 CNC1CCN(CC1)C LF-0516 CN1CCC(CC1)N LF-0517 c1ccc(cc1)CC2(CCNCC2)O LF-0518 CCC1CCCCN1 LF-0519 C1CNCCC1C(F)(F)F.Cl LF-0520 C1CC(CNC1)O.Cl LF-0521 C1CNCCC1C#N LF-0522 C1CCN(CC1)CCCN LF-0523 C1CNCCC1N2CCOCC2 LF-0524 C1CCN(C1)C2CCNCC2 LF-0525 c1cc(ccc1C(=O)C2CCNCC2)F.Cl LF-0526 CC(C)(C)OC(=O)N1CCCCC1 LF-0527 C1CC(CNC1)(F)F.Cl LF-0528 CN1CCCCC1CCCl.Cl LF-0529 C1CCN(CC1)C(=S)N LF-0530 CN1CCC(CC1)O LF-0531 C1CNCCC1O LF-0532 c1ccc(cc1)CN2CCC(CC2)O LF-0533 CN1CCCC(C1)O LF-0534 c1ccc(cc1)CN2CCCC(C2)O LF-0535 C1CC(CNC1)CO LF-0536 C1CNCCC1CCO LF-0537 C1CCN(CC1)CCO LF-0538 CN1CCN(CC1)CCCN LF-0539 C1CCC(C1)N2CCNCC2 LF-0540 COc1ccc(cc1)CN2CCNCC2 LF-0541 c1cnccc1CN2CCNCC2 LF-0542 C1CCC(CC1)N2CCNCC2 LF-0543 c1cc(ccc1N2CCNCC2)F.Cl.Cl LF-0544 c1cc(ccc1N2CCNCC2)Cl.Cl.Cl LF-0545 c1ccc2c(c1)cccc2N3CCNCC3.Cl LF-0546 COc1ccccc1N2CCNCC2 LF-0547 c1ccc(cc1)CN2CCNCC2 LF-0548 c1ccc(cc1)N2CCNCC2 LF-0549 Cc1ccc(c(c1)N2CCNCC2)C LF-0550 COc1cccc(c1)N2CCNCC2.Cl.Cl LF-0551 COc1ccccc1N2CCNCC2.Cl LF-0552 C1CN(CCN1)CCO LF-0553 c1cc(cc(c1)N2CCNCC2)C(F)(F)F.Cl LF-0554 C1CNCCNC1 LF-0555 C1CN(CCN1)CCN LF-0556 CC(=O)N1CCNCC1 LF-0557 Cc1cccc(c1C)N2CCNCC2.Cl LF-0558 CCOc1ccccc1N2CCNCC2.Cl LF-0559 Cc1ccccc1N2CCNCC2.Cl.Cl LF-0560 C1CNCCN1 LF-0561 Cc1cccc(c1)N2CCNCC2C LF-0562 c1cc(c(cc1F)F)N2CCNCC2 LF-0564 CN1CCN(CC1)CCN LF-0565 c1ccc(c(c1)N2CCNCC2)Cl.Cl LF-0566 COc1ccc(cc1)N2CCNCC2 LF-0567 c1cc(cc(c1)Cl)N2CCNCC2.Cl LF-0568 c1ccnc(c1)N2CCNCC2 LF-0569 c1cc(ncc1C(F)(F)F)N2CCNCC2 LF-0571 c1cc(c(cc1N2CCNCC2)Cl)Cl LF-0572 c1cc(c(cc1Cl)Cl)N2CCNCC2.Cl.Cl LF-0573 Cn1c(ccn1)c2ccc(cc2)[N+](=O)[O-] LF-0700 c1cc(c2nccc(=O)n2c1)C=O LF-0701 CC(C)(C)OC(=O)N1CCc2c(cnc(n2)OC)C1 LF-0702 COc1c(cc(cc1I)Br)C=O LF-0705 COC(=O)COc1ccc(cc1C(=O)OC)Br LF-0707 c1c[nH]c2ccncc2c1=O LF-0708 Cn1c(ccn1)c2cccnc2 LF-0711 c1cncc2c1nccc2Cl LF-0713 Cc1cc(ccc1F)S LF-0716 c1c[nH]c2nccn2c1=O LF-0719 CC(=O)c1cc([nH]c1[N+](=O)[O-])C(=O)C(Cl)(Cl)Cl LF-0721 CC(C)(C)c1ccc(c(=O)[nH]1)C#N LF-0724 c1cc(c(cc1n2cncn2)Cl)CO LF-0731 c1ccc(cc1)CN2CCN(CC2)c3cccc(n3)Cl LF-0733 CCOC(=O)c1c(c2cccnc2n1C)N LF-0734 CCOC(=O)c1ccnc2c1cc[nH]2 LF-0736 c1c[nH]c2c1c(ccn2)C(=O)O LF-0737 CC(C)(C)OC(=O)N1CCN(CC1)c2cccc(n2)Cl LF-0738 CCOC(=CC(=O)C(F)(F)F)OCC LF-0739 COC(=O)c1cc(ccc1O)c2ccccc2 LG-0016 COC(=O)c1cc(cc(c1O)Br)c2ccccc2 LG-0018 Cc1ccc(cc1)c2c(noc2C)C LG-0042 c1ccc(c(c1)Oc2ccnc(n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl LG-0087 c1cc(ccc1CNC(=O)CCCCCN2CCNCC2)C#N.Cl.Cl LG-0202 Cc1c2cc(c(=O)[nH]c2ccn1)I LG-0700 COC(=O)c1cc(c(nc1)N)I LG-0703 CCOC(=O)c1cc(ccc1O)Br LG-0705 COC(=O)c1cc2c(o1)cccc2Cl LG-0706 Cc1c(c(nc(n1)OC)N)C#N LG-0709 Cc1cc(cc(c1NC(=O)C)N)F LG-0710 Cc1c(cc(c(n1)OC)I)C(=O)C LG-0711 Cc1c2c(n[nH]1)NC(=O)CC23CCCCC3 LG-0713 Cc1cc(n(n1)C(=O)OC(C)(C)C)N LG-0714 Cc1cc2nc(cc(n2n1)O)C LG-0715 CNc1c(cc(cn1)Br)C(=O)OC LG-0716 CNc1c(cc(cn1)C(=O)OC)Br LG-0717 Cc1c2cc(c(nc2ccn1)Cl)I LG-0719 c1cc(c(cc1CO)I)F LG-0720 COC(=O)c1cc(cc(c1O)I)C#N LG-0722 COC(=O)c1cc2cccc(c2o1)Br LG-0723 COC(=O)c1cc2c(cc1[N+](=O)[O-])[nH]c(=O)[nH]2 LG-0724 CCOC1c2cccnc2C(=O)O1 LG-0727 c1cc(c(cc1CCl)I)F LG-0730 COC(=O)c1cc2cc(ccc2o1)C(F)(F)F LG-0731 Cc1c(c(nc(n1)SC)N)C#N LG-0732 CCOc1cccc2c1oc(c2)C(=O)OC LG-0738 COC(=O)c1cc2ccc(cc2o1)Cl LG-0740 COC(=O)c1cc(cc(c1O)NC(=O)CCl)Br LG-0741 CCc1ccc2c(c1)cc(o2)C(=O)C LG-0743 COc1c(cc(cn1)I)C(=O)O LG-0744 COC(=O)c1cc2cccc(c2o1)C(F)(F)F LG-0745 Cc1c2cc(c(nc2ccn1)OC)I LG-0747 c1cc(cc2c1cc([nH]2)C(=O)N)Br LG-0748 Cc1ccccc1COc2ccc(cc2)C#N LH-0271 Cc1cc(cnc1O)C(=O)OC LH-0700 Cc1cc(cnc1Cl)C(F)F LH-0701 Cc1cc(cnc1Cl)C(=O)OC LH-0703 Cc1cc(cnc1Cl)C(=O)N LH-0705 CCOC(=O)c1ccc2c(c1)[nH]c(n2)O LH-0706 CCOC(=O)c1ccc2c(c1)[nH]c(=O)c(=O)[nH]2 LH-0707 Cc1cc(cnc1Cl)C(=O)C LH-0708 Cc1cc(cnc1N(C)C)C=O LH-0709 Cc1cc(cnc1S(=O)(=O)C)C=O LH-0715 Cc1cc(cnc1OC)C(=O)OC LH-0717 CCOC(=O)c1ccc2c(c1)nc([nH]2)C(F)(F)F LH-0721 CCC(=O)Nc1cc(ccc1NC)C(=O)OC LH-0722 CCc1nc2cc(ccc2n1C)C(=O)OC LH-0723 Cc1cc(cnc1O)C=O LH-0725 COc1cc(c(cc1[N+](=O)[O-])OC)C=O LH-0732 c1[nH]nc(n1)CCN.Cl.Cl LK-0023 c1ccc(cc1)[C@H]2CCCCN2 LS-1000 c1ccc(cc1)[C@@H]2CCCCN2 LS-1001 C[C@H]1CCCCN1.Cl LS-1003 c1ccc(cc1)C[C@H]2CCCCN2 LS-1004 c1ccc(cc1)C[C@@H]2CCCCN2 LS-1005 CC[C@@H]1CCCCN1.Cl LS-1006 CC[C@H]1CCCCN1.Cl LS-1007 CC(C)(C)OC(=O)NC[C@H]1CCCCN1 LS-1008 CC(C)(C)OC(=O)NC[C@@H]1CCCCN1 LS-1009 CC(C)(C)OC(=O)N1CCCC[C@@H]1CO LS-1012 CC(C)(C)OC(=O)N1CCCC[C@H]1CO LS-1013 c1ccnc(c1)[C@@H]2CCCCN2 LS-1025 CC(C)(C)OC(=O)NC[C@H]1CCCNC1 LS-1026 CC(C)(C)OC(=O)NC[C@@H]1CCCNC1 LS-1027 CC(C)(C)OC(=O)N(C)[C@@H]1CCCNC1 LS-1028 CC(C)(C)OC(=O)N1CCCC[C@H]1CN LS-1031 CC(C)(C)OC(=O)N1CCC[C@@H](C1)CC(=O)O LS-1032 CC(C)(C)OC(=O)N1CCC[C@H](C1)C=O LS-1033 CC(C)(C)OC(=O)N1CCC[C@@H](C1)C=O LS-1034 c1ccc(cc1)C[C@@H](C(=O)N)NC(=O)[C@H](CC(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 MA-0200 CCOC(=O)/C(=N\O)/N1CCCCC1 MA-0700 c1ccc(c(c1)c2nc(cs2)C(=O)O)Cl MA-0703 c1cc(cc(c1)F)c2nc(cs2)C(=O)O MA-0704 COc1cccc(c1)c2nc(cs2)C(=O)O MA-0705 COc1ccc(cc1OC)c2nc(cs2)C(=O)O MA-0706 COc1ccc(cc1)Nc2nc(cs2)C(=O)O.Br MA-0707 c1cc(ccc1Nc2nc(cs2)C(=O)O)Cl MA-0708 CC(=O)Nc1nc(cs1)C(=O)O MA-0709 c1c(c(cnc1Cl)C(=O)O)Cl MA-0710 c1ccc(c(c1)CO)NS(=O)(=O)c2ccc(cc2)I MA-0711 c1ccc(cc1)C(=O)CNc2ccc(cc2)Br MA-0712 c1cc(ccc1c2coc(c2C#N)N)[N+](=O)[O-] MA-0713 c1ccc(cc1)C(=O)CNc2cccc(c2)C(F)(F)F MA-0714 c1ccc(cc1)C(=O)CNc2ccc(cc2)Cl MA-0715 c1ccc(cc1)N2CCN(CC2)c3nc(cs3)C(=O)O MA-0717 c1cc(c(nc1C#N)Br)N MA-0719 c1c(nc(s1)N2CCCCC2)C(=O)O MA-0720 c1cc(ccc1Sc2cnc(s2)N)Br MA-0722 c1ccc(c(c1)CO)NS(=O)(=O)c2ccc(cc2)Cl MA-0724 CCOC(=O)c1c(con1)C(=O)c2ccc(cc2)OC MA-0725 CN1CCN(CC1)c2ccc(cc2)C(=O)OC MA-0726 c1cc(ncc1C(=O)N)C(F)(F)F MA-0809 c1ccc(cc1)COCCN2CCC(=O)CC2 MA-0811 c1ccc(cc1)CNC(=O)c2cc(cc(n2)C(=O)Nc3ccccc3)C(F)(F)F MA-0812 CCNC(=O)c1cc(cc(n1)C(=O)Nc2ccccc2)C(F)(F)F MA-0817 CCOC(=O)c1cc(cnc1O)S(=O)(=O)O MA-0820 c1ccc(cc1)NC(=O)c2cc(cc(n2)C(=O)NCc3ccccn3)C(F)(F)F MA-0821 COc1ccc2c(c1)[nH]cc2C=O MA-0823 CN(C)/C=C(\C#N)/c1ccc(nc1)Cl MA-0825 CCNC(=O)c1cc(cc(n1)C(=O)NCc2ccccc2)C(F)(F)F MA-0826 c1ccc(cc1)CNC(=O)c2cc(cc(n2)C(=O)NCc3ccccc3)C(F)(F)F MA-0827 c1ccc(cc1)CNC(=O)c2cc(cc(n2)C(=O)NCc3ccccn3)C(F)(F)F MA-0828 c1cc(n2ccnc2c1)N MA-0831 CC1CCCN(C1)CC#N MA-0832 C=CCN1CCC(=O)CC1 MA-0834 CCNC(=O)c1cc(cc(n1)C(=O)NCc2ccccn2)C(F)(F)F MA-0836 c1cc(ccc1N)Oc2ncc(cn2)Br MA-0840 Cn1cc(c2c1cc(cc2)OC)C=O MA-0841 c1cc(cc(c1)Oc2ncc(cn2)Br)C=O MA-0842 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2Br)F MA-0845 C[C@@H]1C[C@@H](C(=O)OC1=O)C MA-0846 C=CCCNCc1ccccc1 MA-0848 c1cc(c(cc1F)Br)NC(=S)N MA-0849 c1cc(ccc1C=O)Oc2ncc(cn2)Br MA-0853 c1c(sc(n1)Cl)CN2CCCN(CC2)Cc3cnc(s3)Cl MA-0857 c1ccc(cc1)CN2CC[C@@H]3C[C@H]2C(=O)O3 MA-0859 Cc1c2c(cccc2O)[nH]n1 MA-0860 CC(=O)Nc1nc2c(cccc2s1)Oc3cc(ncn3)Cl MB-0046 C[C@H](c1ccc(cc1)F)N2CCN(CC2)c3cc(ncn3)Oc4cccc5c4nc(s5)NC(=O)C MB-0047 c1ccc(cc1)COC(=O)NC(c2cccc(c2)Cl)S(=O)(=O)c3ccccc3 MB-0053 c1cc(ccc1C2=C(SC3=NCCN23)C=O)Br MB-0206 c1ccc(cc1)CN2CC3CCC(C3C2)N MB-0216 CC(C#N)c1ccc(cc1)[N+](=O)[O-] MB-0700 CC(C#N)c1ccc(cc1)N MB-0701 Cc1nc(cc(n1)Cl)N2CCOCC2 MB-0702 Cc1nc(cc(n1)Cl)N2CCCC2 MB-0703 Cc1nc(cc(n1)Cl)N2CCCCC2 MB-0705 Cc1nc(cc(n1)Cl)N2CCN(CC2)Cc3ccccc3 MB-0706 Cc1nc(cc(n1)Cl)N2CCC(CC2)O MB-0707 COc1cc(ccc1[N+](=O)[O-])N2CCC(CC2)O MB-0708 Cc1nc(cc(n1)Cl)N2CCN(CC2)C MB-0709 Cc1nc(cc(n1)Cl)N2CCN(CC2)C(=O)OC(C)(C)C MB-0710 Cc1nc(cc(n1)Cl)NC MB-0714 Cc1nc(cc(n1)Cl)O MB-0715 c1cc(ccc1S(=O)(=O)N2CCN(CC2)CCO)Cl MB-0716 c1cc(ccc1S(=O)(=O)N2CCN(CC2)CCO)I MB-0717 Cn1c2c(cn1)c(ncn2)N MB-0718 c1c(nc(nc1Cl)N)N2CCN(CC2)CCO MB-0720 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CCO MB-0722 c1cc(ccc1F)S(=O)(=O)N2CCN(CC2)CCO MB-0723 Cc1nc(cc(n1)Cl)N2CCC(CC2)C(=O)O MB-0725 c1cc(c(nc1)N2CCN(CC2)CCO)[N+](=O)[O-] MB-0726 COc1cc(ccc1[N+](=O)[O-])N2CCC(=O)CC2 MB-0727 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(c(c2)OC)[N+](=O)[O-] MB-0728 COC(=O)c1cc(ncc1Cl)Cl MB-0729 COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CCO MB-0730 CCOC(=O)c1cc(ncc1Cl)Cl MB-0731 CCCCc1[nH]c2cc(c(cc2n1)Cl)Cl MB-0732 c1ccc2c(c1)nc(s2)N3CCN(CC3)CCO MB-0733 CCc1nc2c(cccc2o1)[N+](=O)[O-] MB-0735 CCOC(=O)C1CCN(CC1)c2ccc(c(c2)OC)[N+](=O)[O-] MB-0736 COc1cc(ccc1[N+](=O)[O-])N2CCC(CC2)C(=O)O MB-0737 c1cc(c(nc1)N2CCN(CC2)CCO)C#N MB-0738 CCOC(=O)C(=O)N1CCC(CC1)C(F)(F)F MB-0800 Cc1ccc(cc1)C2NCCS2 MB-0801 c1c(c(cnc1Cl)Br)I MB-0802 c1ccc(c(c1)C#N)OCC(=O)O MB-0803 CCOC(=O)C1CCCN(C1)S(=O)(=O)N(CCBr)C(=O)OC(C)(C)C MB-0806 c1c(cncc1Br)C(=O)N2CCNCC2 MB-0809 c1cc(c(cc1[N+](=O)[O-])C=O)N2CCOCC2 MB-0810 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2C=O)[N+](=O)[O-] MB-0811 CN1CCN(CC1)c2ccc(cc2C=O)[N+](=O)[O-] MB-0815 CC1(CC(=O)NC1)C MB-0820 CC(C)(C)OC(=O)N1CCSC1C(=O)O MB-0821 COC(=O)c1cc([nH]n1)[N+](=O)[O-] MB-0822 COC(=O)c1c(c([nH]n1)[N+](=O)[O-])Br MB-0824 CN1CCN(CC1)c2ccc(cc2CO)[N+](=O)[O-] MB-0829 C1CCc2c(c3c(o2)nc(nc3Cl)CCl)C1 MB-5002 COC(=O)c1cc(c(c(c1Nc2ccc(cc2Cl)Br)F)F)[N+](=O)[O-] MB-5003 CCOC(=S)SCc1nc2c(c3c(o2)CCCC3)c(n1)Cl MB-5007 c1cnc(cc1Cl)CO MB-5013 c1ccc(c(c1)C=O)c2ccccc2Cl MC-0021 c1cc(c(c(c1)Cl)CN(Cc2c(cc(cn2)C(F)(F)F)Cl)S(=O)(=O)NCC(=O)c3ccc(cc3)Cl)Cl MC-0048 c1cc2c(cc1Cl)oc(n2)CSc3c(cc(cn3)C(F)(F)F)Cl MC-0057 COC(=O)Cc1ccc2c(c1)oc(n2)CSc3c(cc(cn3)C(F)(F)F)Cl MC-0058 COC(=O)c1ccc2c(c1)oc(n2)CSc3c(cc(cn3)C(F)(F)F)Cl MC-0059 c1cc(ccc1c2nc(on2)CSc3c(cc(cn3)C(F)(F)F)Cl)Cl MC-0063 c1ccc2c(c1)CN(C2)C(=O)[C@@H]3CCCN3c4c(cc(cn4)C(F)(F)F)Cl MC-0205 CN1CC(=O)N(C1=O)CCCCC(=O)NN MC-0206 c1c(cnc(c1Cl)N2CCC[C@H]2C(=O)N3CCCC3)C(F)(F)F MC-0207 c1cc(c(cc1Cl)Cl)N2CCN(CC2)C(=O)[C@@H]3CCCN3c4c(cc(cn4)C(F)(F)F)Cl MC-0212 CC(C)(C)OC(=O)N1CCCCN1C(=O)c2ccc(cc2)[N+](=O)[O-] MC-0700 CC(C)(C)OC(=O)N1CCCCN1C(=O)c2ccc(cc2)N MC-0701 c1cc(ccc1C(=O)N2CCCCN2)[N+](=O)[O-] MC-0703 CCOC(=O)c1c(cccn1)Cl MC-0709 COc1cnc(nc1O)c2ccncc2 MC-0711 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(c(c2)C(=O)O)N MC-0713 CC(C)(c1cc(nc(c1)Cl)OC)O MC-0715 c1cc2c(cc1C(F)(F)F)cc(s2)CO MC-0716 c1c(c(=O)[nH]c(c1Cl)C2CC2)C#N MC-0720 c1cc(ccc1C(=O)N2CCCCN2)N MC-0722 CC1CN(CC(O1)C)c2ccc(c(c2)OC)N MC-0723 CCn1c(=O)c2cc(ccc2[nH]c1=O)N3CCN(CC3)C(=O)OC(C)(C)C MC-0725 COc1cnc(nc1Cl)c2ccncc2 MC-0731 CC(=O)c1cccc2c1oc(n2)CCl MC-0732 COC(=O)c1cc(cnc1Cl)F MC-0746 c1cc([nH]c(=O)c1C(=O)O)C2CC2 MC-0747 CCCNC(=O)Nc1ccc(cc1C(=O)OC)Br MC-0748 CCCn1c(=O)c2cc(ccc2[nH]c1=O)Br MC-0749 CC(C)(C)OC(=O)N1CCN(CC1)CC(c2ccccc2)C(=O)O MC-0752 CCCn1c(=O)c2cc(ccc2[nH]c1=O)N3CCN(CC3)C(=O)OC(C)(C)C MC-0755 CC(C)n1c(=O)c2cc(ccc2[nH]c1=O)N3CCN(CC3)C(=O)OC(C)(C)C MC-0756 CCOC(=O)c1cn2cc(ccc2n1)[N+](=O)[O-] MC-0770 CC(C)(C)OC(=O)N1CCCN1C(=O)c2ccc(cc2)[N+](=O)[O-] MC-0773 c1cc(nc(c1C#N)Cl)C2CC2 MC-0779 CC(C)(C)OC(=O)N1CCCN1C(=O)c2ccc(cc2)N MC-0782 c1cc(cc2c1cc(s2)CO)Br MC-0783 c1cc2ncc(n2cc1[N+](=O)[O-])Br MC-0786 c1cc(ccc1C(=O)N2CCCN2)[N+](=O)[O-] MC-0788 c1cc(ccc1C(=O)N2CCCN2)N MC-0796 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCc3c(cc(cn3)C(F)(F)F)Cl MD-0003 c1ccc2c(c1)C(=O)N(C2=O)CC#Cc3cc(cnc3N)C(F)(F)F MD-0008 c1c(cnc(c1Cl)CC(=O)NNC(=O)CCCl)C(F)(F)F MD-0009 COC(=O)c1cc(cc(c1O)[N+](=O)[O-])Br MD-0013 Cc1ccc(c(c1)C#C)N MD-0015 COc1c(cc(cc1I)Br)C(=O)OC MD-0023 c1c(cc(c(c1CCNC(=O)C(F)(F)F)O)[N+](=O)[O-])[N+](=O)[O-] MD-0027 c1c(cc(c(c1[N+](=O)[O-])N)I)C(F)(F)F MD-0030 COC(=O)c1cc(cc(c1O)N)Br MD-0032 Cc1c(c(=O)c(c[nH]1)I)OCc2ccccc2 MD-0033 c1cc2c(c(c1)I)CC(=O)N2 MD-0034 c1cc2nc(cn2c(c1)F)C=O MD-0035 c1c(cc(c(c1CCNC(=O)C(F)(F)F)Br)[N+](=O)[O-])[N+](=O)[O-] MD-0036 CC(=O)Nc1cc(c(cc1[N+](=O)[O-])Br)C(F)(F)F MD-0041 c1cc2c(cc1Br)c(c([nH]2)Cl)C=O MD-0047 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(c(c2)C(=O)O)[N+](=O)[O-] MD-0048 c1ccc(cc1)c2nc(cc(n2)Cl)C(=O)Cl MD-0052 c1cc(c(c(c1)Cl)C(=O)NCc2c(cc(cn2)Cl)C(F)(F)F)Cl MD-0053 COc1c(cc(cc1I)Br)C(=O)O MD-0055 c1ccc(cc1)COc2ccc(c(c2)C=O)OCc3ccccc3 MD-0059 c1c(c(cc(c1N)[N+](=O)[O-])Br)C(F)(F)F MD-0064 CC(=O)Nc1cc(c(cc1N)Br)C(F)(F)F MD-0065 c1c(c(cc(c1N)N)Br)C(F)(F)F MD-0073 CS(=O)(=O)NCc1c(cc(cn1)Cl)C(F)(F)F MD-0088 c1cc2c(c(c1)I)c(c([nH]2)Cl)C=O MD-0090 CNC(=O)c1cc(ccc1[N+](=O)[O-])N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MD-0094 CN(C)c1c(c2c([nH]1)cccc2I)C=O MD-0099 c1c[nH]cc1C(=O)C(F)(F)F MD-0200 c1c(c(c(c(n1)Cl)Cl)C(=O)Cl)C(F)(F)F MD-0205 COC(=O)c1ccc(cc1)c2cc(c(nc2)N)[N+](=O)[O-] MD-0208 c1cc2c(c3c1CCC3=O)CCO2 MD-0210 CC(C)(C)OC(=O)N1CCN(CC1)c2c(ccc(n2)c3ccccc3)C#N MD-0212 c1ccc(cc1)C/C(=N\O)/c2ccccc2 MD-0215 c1csc2c1CNCC2.Cl MD-0219 c1c(c(c(c(n1)Cl)Cl)C(=O)N)C(F)(F)F MD-0223 c1c(c(c(c(n1)Cl)Cl)C#N)C(F)(F)F MD-0225 c1ccc(cc1)c2ccc(c(n2)N3CCNCC3)C#N MD-0238 c1ccc(cc1)c2ccc(c(n2)Cl)/C(=N/O)/N MD-0239 c1ccc(cc1)c2ccc(c(n2)Cl)c3nc(on3)C(F)(F)F MD-0243 C1CNCC2=CC(=O)SC21.Cl MD-0244 CC(C)c1ccc(c(n1)Cl)/C(=N/O)/N MD-0250 Cc1nc(no1)c2ccc(nc2Cl)c3ccccc3 MD-0253 CC(C)c1ccc(c(n1)Cl)c2nc(on2)C(F)(F)F MD-0254 COC(=O)c1cc(cnc1F)Br MD-0701 CC(C)C(=O)/C=C/N(C)C MD-0703 CNc1ccc(cc1CO)[N+](=O)[O-] MD-0704 c1cnc(c(c1CCl)Cl)Cl MD-0705 CCOC(=O)c1cn(nc1C)C MD-0706 Cc1c(scn1)CO MD-0707 Cc1c2c([nH]n1)ncnc2O MD-0709 COc1c(c(ccn1)I)C=O MD-0710 CCOC(=O)c1c(cc(cn1)Cl)C(F)(F)F MD-0712 CC(C)c1ccc(c(=O)[nH]1)C#N MD-0713 c1c(cnc(c1C(F)(F)F)C(=O)O)Cl MD-0714 c1c2c(cc(c1Cl)[N+](=O)[O-])OCC(=O)N2 MD-0715 CCS(=O)(=O)c1ccc2c(c1)NCCO2 MD-0716 c1cc2c(cc1F)OCCN2 MD-0717 COc1cc(ccc1NC=O)C(=O)OC MD-0723 CC(C)c1ccc(c(n1)Cl)C#N MD-0726 CCOC(=O)c1cccc(n1)C(=O)C MD-0727 c1c2c(cc(c1Cl)[N+](=O)[O-])OCCN2 MD-0729 CC1(OCCO1)c2cccc(n2)C(=O)O MD-0730 Cc1ccc2c(c1)NCCO2 MD-0731 c1c2c(n[nH]1)CCNC2.Cl.Cl MD-0732 CCOC(=O)c1c(cc(cn1)C(=O)O)Cl MD-0733 CCS(=O)(=O)c1ccc2c(c1)N(CCO2)C(=O)CCl MD-0738 CCOC(=O)c1c(c(ccn1)C(F)(F)F)Cl MD-0739 c1cnc(c(c1C(F)(F)F)Cl)C(=O)O MD-0740 CC(=O)c1cccc(n1)C(=O)O MD-0741 CCOC(=O)c1c(cccn1)C=O MD-0742 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCC(CC2)C(=O)O ME-0001 c1c(cnc(c1Cl)CCNC(=O)CI)C(F)(F)F ME-0038 C(CCO[N+](=O)[O-])CO ME-0046 Cn1ccc2c1ccc(c2)[N+](=O)[O-] ME-0069 c1cc(c(c(c1)Cl)C(Nc2c(cc(cn2)C(F)(F)F)Cl)SCC(=O)O)Cl ME-0094 CCCS(=O)(=O)Nc1ccc(c(c1F)C(=O)c2c[nH]c3c2cc(cn3)c4ccc(cc4)Cl)F ME-0096 Cc1ccncc1NC(=O)OC ME-0097 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCNCC2.Cl ME-0103 c1ccc(cc1)c2cc(c3ccccc3n2)C(=O)Cl.Cl ME-0104 C[C@H]1CCNC[C@H]1NC(=O)OC ME-0136 Cc1cc2c(cc1F)NC(=O)CN2C ME-0148 c1c(cn2c(nnc2c1Cl)CO)C(F)(F)F ME-0149 c1c[nH]c2c1cnc(c2)Cl ME-0200 CC(C)COc1ccc(cc1)CC(=O)O ME-0228 CC(C)COc1ccc(cc1)CCO ME-0231 CC(C)COc1ccc(cc1)CC(=O)NN ME-0232 CCOC(=O)c1ccnc(c1)N ME-0233 c1cnc(cc1C(=O)NN)N ME-0241 CCOC(=O)c1ccn2ccnc2c1 ME-0243 C#Cc1cnc(cc1N)Cl ME-0247 c1[nH]nc(n1)C(F)(F)F ME-0700 CCOC(=O)c1cnc(nc1)c2ccccc2 ME-0702 c1cc(c(cc1[N+](=O)[O-])O)NC(=O)C(F)(F)F ME-0703 c1c(cnc(c1N)N2CCCCCC2)Br ME-0704 COc1c(cc(cn1)C(=O)N)Br ME-0705 c1ccc(cc1)c2nc(cc(n2)Cl)CO ME-0706 c1cc(nc(c1N)N2CCNCC2)Cl ME-0708 CC(C)(C)OC(=O)NC1CCCN(C1)CC2CN(C(=O)O2)c3ccc(cc3)F ME-0709 c1c(c(cc2c1[nH]c(n2)C(F)(F)F)Cl)C(F)(F)F ME-0710 CCOC(=O)c1cnc(nc1Cl)c2ncccn2 ME-0711 c1cnc(nc1)c2nc(cc(n2)O)C(=O)O ME-0715 CNc1cc(ncc1C=O)Cl ME-0718 CCOC(=O)c1cn2cc(ccc2n1)I.Cl ME-0719 CNc1ccc(cc1[N+](=O)[O-])C=O ME-0721 CN(C(=O)c1cccnc1Cl)OC ME-0722 c1cc2c(c(c1)I)c(nc(n2)N)N ME-0724 c1cnc(nc1)c2ncc(cn2)C(=O)O ME-0726 Cn1c2ccc(cc2nc1N)[N+](=O)[O-].Br ME-0727 Cn1c2ccc(cc2[nH]c(=O)c1=O)[N+](=O)[O-] ME-0728 c1ccc(cc1)C2=CC(=O)NCCN2 MF-0009 COc1ccc(cc1OC)NCC2(CCNCC2)O MF-0010 Cc1cc2c(cc1O)C(=O)NC2 MF-0011 COc1ccc(cc1OC)N2CC3(CCN(CC3)C(=O)OCc4ccccc4)OC2=O MF-0016 Cc1cc2c(c(c1O)Cl)C(=O)NC2 MF-0019 CCOC(=O)/C=C(/NCCN/C(=C/C(=O)OCC)/c1cc(cc(c1)C(F)(F)F)C(F)(F)F)\c2cc(cc(c2)C(F)(F)F)C(F)(F)F MF-0020 CCc1cn(nn1)c2ccc(c(c2)F)N MF-0021 COc1cc(c(cc1F)[N+](=O)[O-])C(=O)OC MF-0023 c1cc(cc2c1cc(c(=O)o2)c3c(cc(cn3)C(F)(F)F)Cl)O MF-0025 c1cc2cc(c(=O)oc2c(c1)Cl)c3c(cc(cn3)C(F)(F)F)Cl MF-0026 c1ccc(cc1)C2CC(=O)NCCN2 MF-0027 COc1cc(c(cc1F)C#N)C(=O)OC MF-0028 c1c(cnc2c1c(c[nH]2)Cl)C(F)(F)F MF-0033 c1cc(ncc1C(F)(F)F)NC(=S)N MF-0034 c1c(cnc2c1sc(n2)N)C(F)(F)F.Br MF-0035 c1cc(ccc1C(=O)O)I MF-0039 COc1ccc2cc(c(=O)oc2c1)c3c(cc(cn3)C(F)(F)F)Cl MF-0041 Cc1c(cccc1OC)C(=O)O MF-0044 Cc1ccc(cc1OC)C(=O)O MF-0045 COc1cc(ccc1F)C(=O)O MF-0046 Cc1c(ccc2c1C(=O)NC2)OC MF-0047 c1c(cnc(c1Cl)NCC(CO)O)C(F)(F)F MF-0049 CC1(OC(=O)C(=CNc2cc(c(cc2I)C#N)C(F)(F)F)C(=O)O1)C MF-0051 CC(C)(C)OC(=O)N1CCNC(=O)CC1c2ccccc2 MF-0053 COc1cc(c(cc1F)N)C(=O)OC MF-0054 COc1ccc(cc1OC)N2CC3(CCNCC3)OC2=O MF-0059 CCc1cn(nn1)c2cc(ccc2C)N MF-0064 Cc1cn(nn1)c2ccc(c(c2)F)N MF-0065 Cc1c(ccc2c1C(=O)NC2)O MF-0066 COC(=O)c1cc(c(cc1Br)F)O MF-0069 CC(=O)Oc1ccc2cc(c(=O)oc2c1)c3c(cc(cn3)C(F)(F)F)Cl MF-0073 CCNC(=O)Oc1ccc2cc(c(=O)oc2c1)c3c(cc(cn3)C(F)(F)F)Cl MF-0074 CCc1cn(nn1)c2ccccc2 MF-0081 c1(nnc(s1)Br)N MF-0084 Cc1c(=O)[nH]c2ccccc2n1 MF-0223 Cc1c(nc2ccccc2n1)Cl MF-0225 Cc1cc(cc(n1)N2CCNCC2)Cl MF-0701 CC(C)(C)OC(=O)N1CCCC1CC(=O)O MF-0703 CCOC(=O)c1cccc(n1)N2CCN(CC2)Cc3ccccc3 MF-0705 c1c([nH]nc1N)C(F)(F)F MF-0707 c1c2c([nH]n1)ncnc2Cl MF-0708 c1c2c([nH]n1)nc(nc2Cl)N MF-0709 CCOC(=O)c1cc2c(s1)nc(nc2Cl)N MF-0711 C(c1c(nc(nc1Cl)N)Cl)O MF-0712 CNc1ncc(c(n1)C(=O)OC)Br MF-0713 CCOC(=O)c1cccc(n1)N2CCN(CC2)C(=O)OC(C)(C)C MF-0714 c1c(cnc(c1F)C#N)C(F)(F)F MF-0715 CC(C)(C)OC(=O)NCC(=O)c1ccc(cc1)Br MF-0718 CCOC(=O)c1c(c2c(cc(nc2n1C)C)C(F)(F)F)N MF-0719 c1cc2c(cc1Cl)c(n[nH]2)I MF-0720 c1c(c(nc(n1)N2CCOCC2)C(=O)O)Br MF-0722 c1c(cnc(c1F)C(=O)N)C(F)(F)F MF-0723 c1c(cnc(c1Br)Br)Br MF-0724 C(c1c(nc(nc1Cl)N)Cl)Cl MF-0727 CCOC(=O)c1cnc(c(c1O)I)O MF-0730 c1nc2c(c(n1)Cl)c(n[nH]2)Br MF-0733 c1cc(ccc1C#N)c2c(ccs2)C=O MF-0734 c1ccc2c(c1)[nH]c(n2)n3cccn3 MF-0735 CCOC(=O)c1cn(c(=O)c(c1Cl)Cl)C MF-0737 Cc1c2c(cc(cn2nn1)C(F)(F)F)Cl MG-0004 c1ccc(cc1)[P+](CCCCCC(=O)O)(c2ccccc2)c3ccccc3.[Br-] MG-0025 CC(C)/C=C\CCCCC(=O)O MG-0051 Cc1c(cnn1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)Nc3ccccc3 MG-0094 Cc1c(cnn1c2c(cc(cn2)C(F)(F)F)Cl)C(=O)NC MG-0101 CC(C(=O)Nc1ccccc1)Cl MG-0201 COc1ccc(cc1)n2c(nnc2S)c3ccccc3OC MG-0203 c1ccc(cc1)S(=O)c2cc3cccc(c3nc2)N MG-0222 Cc1c(c([nH]n1)N)c2ccc(c(c2)OC)OC MG-0225 Cc1cc(nc(n1)NC(=O)NS(=O)(=O)c2ccccc2C(=O)OCC(=O)CCl)C MG-0226 c1ccc2c(c1)c3c([nH]2)c4cc(ccc4[nH]c3=O)Cl MG-0702 CCOC(=O)c1cc2cc(ccc2s1)NS(=O)(=O)C MG-0703 Cc1c2c(ncnc2[nH]n1)N MG-0704 CN1CCN(CC1)c2ccc(cn2)C(=O)OC MG-0705 c1cc(cc2c1cc([nH]2)C#N)Br MG-0706 CS(=O)(=O)Nc1ccc2c(c1)cc(s2)C(=O)O MG-0707 Cn1c(cc2c1cc(cc2)Br)C=O MG-0711 c1c2c(cc(c1Br)O)NC(=O)CC2 MG-0713 CCOC(=O)c1c(ocn1)C(C)(C)C MG-0714 c1cc(c(nc1)C#N)CC#N MG-0715 COC(=O)C(c1ccc(cc1)C(F)(F)F)N MG-0716 Cc1c(ccc(c1C(=O)N)Br)OC MG-0717 CC(C)(C)OC(=O)N[C@H](Cc1cc(c(cc1F)F)F)CC(=O)O MG-0718 Cc1ccc(cc1)S(=O)(=O)O.c1ccc(cc1)COC(=O)[C@@H](Cc2ccc(cc2)F)N MG-0719 Cc1cc(cc(c1C[C@@H](C(=O)O)N)C)O.Cl MG-0720 Cc1cc(cc(c1C[C@@H](C(=O)O)N)C)O MG-0721 Cc1cc(cc(c1C[C@@H](C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4)C)O MG-0722 C[C@H](c1cc(cc(c1)C(F)(F)F)C(F)(F)F)OC2[C@@H](NCCO2)c3ccc(cc3)F.Cl MG-0723 C[C@H](c1cc(cc(c1)C(F)(F)F)C(F)(F)F)O[C@@H]2C(=O)N(CCO2)Cc3ccccc3 MG-0724 c1ccc(cc1)COC(=O)[C@@H]2C[C@@H]3CCC[C@@H]3N2.Cl MG-0725 C[C@@H](c1cccc(c1)O)N(C)C MG-0726 c1c(c(c(c(n1)Cl)Cl)C(F)(F)F)Cl MG-0727 CC(C)(C(=O)N)C(=O)O MH-0703 Cc1cc(cc(c1I)C)OC(=O)C MH-0707 c1cc(c(cc1[N+](=O)[O-])Br)C#N MH-0709 Cc1cc(cc(c1/C=C(/C(=O)OC)\NC(=O)C)C)OC(=O)C MH-0715 CCOC(=O)c1cc(c(nc1)Cl)C MH-0728 c1ccc(cc1)OCC(=O)Nc2ccc(c(c2F)F)F MS-0001 Cc1csc(c1NC(=O)CCl)C(=O)OC MS-0002 Cc1csc(c1NC(=O)Cc2ccccc2)C(=O)OC MS-0003 CCOC(=O)c1ccccc1NC(=O)c2cccc(c2)Br MS-0004 c1cc(ccc1CC(C(=O)O)NC(=O)CCl)F MS-0005 c1ccc2c(c1)c(=O)oc(n2)c3cccc(c3)Br MS-0006 Cc1ccccc1C(=O)Nc2cccc(c2Cl)F MS-0007 CC1CN(CC(O1)C)c2ccc(cc2)NC(=O)CCl MS-0010 Cc1csc(c1NC(=O)c2ccc(cc2Cl)Cl)C(=O)OC MS-0012 CC1CN(CC(O1)C)c2ccc(cc2)NS(=O)(=O)C MS-0013 c1ccc(c(c1)C(=O)O)NC(=O)c2cccc(c2)Br MS-0014 CC1CN(CC(O1)C)C(=O)c2cccc(c2)C(F)(F)F MS-0018 CC1CN(CC(O1)C)S(=O)(=O)c2ccccc2Cl MS-0019 CC1CN(CC(O1)C)C(=O)c2c(cccc2Cl)Cl MS-0020 Cc1cc(ccc1F)NC(=S)NC MS-0021 Cc1ccc(c(c1)NC(=S)NC)F MS-0022 CNC(=S)Nc1c(cccc1F)F MS-0023 CC(=O)Nc1ccccc1F MS-0024 c1ccc(c(c1)C(=O)N2CC(C2)C(=O)O)F MS-0025 c1cc(cc(c1)Br)C(=O)N2CC(C2)C(=O)O MS-0027 c1ccc(c(c1)C(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)O)F MS-0028 Cc1csc(c1NS(=O)(=O)c2cccc(c2)Cl)C(=O)OC MS-0031 Cn\1ccs/c1=N/C(=S)NC(=O)c2ccc(cc2)Cl MS-0032 CC(C)(C)c1nnc(s1)N MS-0033 CC(C=C)ON1C(=O)c2ccccc2C1=O MS-0036 Cc1ccc(c(c1)NC(=O)C)F MS-0037 Cc1ccc(c(c1)NC(=O)NC)F MS-0038 CNC(=O)Nc1ccccc1F MS-0039 Cc1cc(ccc1F)/N=C/c2ccccc2F MS-0040 c1cc(c(c(c1)Cl)C(=O)NN2CCOCC2)Cl MS-0041 c1cc(c(cc1Cl)S(=O)(=O)NN2CCOCC2)Cl MS-0042 c1ccc(c(c1)C(=O)Nc2ccc(cc2)F)F MS-0043 Cc1cc(ccc1F)NC(=O)c2ccccc2F MS-0044 c1ccc(c(c1)C(=O)Nc2ccc(cc2Cl)F)F MS-0045 Cc1cc(ccc1F)NC(=O)NC MS-0046 Cc1cc(ccc1NC(=O)c2ccccc2F)F MS-0047 CNC(=O)Nc1ccc(cc1Cl)F MS-0048 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)CCl MS-0049 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)/C=C/c3ccccc3 MS-0050 CC(=O)c1ccc(cc1)Oc2nc(on2)c3ccccc3F MS-0052 CC(C)(C)N(C(=O)COc1ccccc1)NC(=O)COc2ccccc2 MS-0053 CC(C)(CO)NC(=O)c1ccncc1 MS-0054 CCCCNC(=O)Nc1ccc(c2c1OC(C2)(C)C)C MS-0055 c1cc2c(cc1Cl)n(c(=O)o2)C/C=C/CCl MS-0056 Cc1cc(nc(n1)NC(=O)COc2ccccc2)C MS-0057 CCC1(CCC(O1)(C)C)COCc2ccccc2F MS-0062 CCOP(=O)(NCCc1ccc(c(c1)OC)OC)OCC MS-0063 Cc1c2ccccc2c(=O)on1 MS-0064 COc1ccc(cc1OC)CCNC(=O)/C=C/C(=O)O MS-0065 c1ccc(c(c1)NC(=O)NC2CC2)F MS-0069 C/C=C/C(=O)NCCOc1ccc(cc1Cl)Cl MS-0070 CN(CO)C(=O)/C=C/c1ccccc1 MS-0072 CC(C)(C)c1nnc(s1)NC(=O)NC MS-0073 c1ccc(cc1)C(c2ccccc2)N3CC(C3)C(=O)O MS-0076 CCOC(=O)c1c(=O)cc(n(n1)c2ccc(cc2)Cl)C MS-0077 c1ccc2c(c1)c(=O)oc(n2)c3ccc(cc3)Cl MS-0078 Cc1ccc(c(c1)NC(=O)c2ccccc2F)C(=O)O MS-0083 CC(C)(C)c1nnc(s1)NC(=O)c2cccc(c2)Br MS-0085 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)Nc3ccccc3C(F)(F)F MS-0087 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)Nc3ccc(cc3)Br MS-0088 Cc1ccc(c2c1CC(O2)(C)C)NC(=S)Nc3ccccc3 MS-0089 Cc1ccc(c2c1CC(O2)(C)C)N MS-0090 c1ccc(c(c1)C(=O)Nc2ccccc2C(=O)O)C(F)(F)F MS-0092 c1ccc(c(c1)C(=O)O)NC(=O)c2ccc(cc2)Cl MS-0093 Cc1cccc(c1)C(=O)Nc2ccccc2C(=O)O MS-0094 c1cc(cc(c1)Br)C(=O)Nc2cc(ccc2C(=O)O)Cl MS-0095 Cc1cc(ccc1C(C)C)N2C(=O)Cc3ccccc3C2=O MS-0103 CC(C)(C)c1csc(n1)NS(=O)(=O)c2cccc(c2)Cl MS-0104 CC(C)(C)c1nnc(s1)NC(=O)NS(=O)(=O)c2ccccc2 MS-0105 c1cc2cnccc2c(c1)/N=C/c3ccc(cc3)OC(F)(F)F MS-0109 c1cc2cnccc2c(c1)/N=C/c3ccc(cc3)C(F)(F)F MS-0110 c1ccc(c(c1)/C=N/c2cccc3c2ccnc3)F MS-0112 Cc1ccc(c2c1CC(O2)(C)C)Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] MS-0113 c1cc(ccc1C(=O)NCCCn2ccnc2)Cl MS-0117 c1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl MS-0119 c1cc(ccc1C(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl)[N+](=O)[O-] MS-0121 c1cc(ccc1C(=O)NCCCn2ccnc2)[N+](=O)[O-] MS-0122 c1cc(cc(c1)Cl)S(=O)(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl MS-0124 Cc1ccc(c2c1CC(O2)(C)C)/N=C/c3ccc(cc3)F MS-0125 Cc1ccc(c2c1CC(O2)(C)C)/N=C/c3ccccc3F MS-0126 Cc1ccc(c2c1CC(O2)(C)C)/N=C/c3ccc(cc3)OC(F)(F)F MS-0128 Cc1ccc(cc1)S(=O)(=O)NCCCN2CCCC2 MS-0130 c1ccc(c(c1)C(=O)O)NC(=O)c2ccccc2F MS-0137 COC(=O)c1c(ccs1)NC(=O)c2ccc(cc2)Cl MS-0138 Cc1csc(c1NC(=O)/C=C/c2ccccc2)C(=O)OC MS-0139 Cc1csc(c1NC(=O)C(c2ccccc2)Cl)C(=O)OC MS-0140 Cc1ccc2c(c1)c(=O)oc(n2)c3ccccc3F MS-0142 Cc1csc(c1NC(=O)/C=C/c2ccc(cc2)Cl)C(=O)OC MS-0143 CC(=O)Nc1cc(ccc1Nc2ccccc2)C(F)(F)F MS-0144 Cc1csc(c1NC(=O)c2ccccc2F)C(=O)OC MS-0145 Cc1csc(c1N(C(=O)c2ccccc2F)C(=O)c3ccccc3F)C(=O)OC MS-0148 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccsc2C(=O)O MS-0149 c1cc(ccc1C(=O)Nc2ccsc2C(=O)O)Cl MS-0151 Cc1csc(c1NC(=O)c2ccc(cc2)C(C)(C)C)C(=O)O MS-0154 CCOC(=O)c1c2c(sc1NC(=O)c3cccc(c3)Br)CCCC2 MS-0156 c1cc(ccc1NC(=O)[C@H]2C[C@H]2C(=O)O)[N+](=O)[O-] MS-0162 Cc1csc(c1NC(=O)c2ccc(cc2)C(C)(C)C)C(=O)OC MS-0164 c1cc(c(cc1Cl)F)NC(=O)[C@H]2C[C@H]2C(=O)O MS-0166 Cc1cc(ccc1C(C)C)NC(=O)NS(=O)(=O)c2ccccc2 MS-0167 Cc1ccc(c(c1)NC(=O)C2CC2C(=O)O)F MS-0168 COC(=O)c1c(ccs1)NC(=O)c2cccc(c2)C(F)(F)F MS-0169 Cc1cc(cc(n1)C)NC(=O)c2cccc(c2)C(F)(F)F MS-0171 COC(=O)c1c(ccs1)NC(=O)c2ccccc2F MS-0172 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)N MS-0173 c1ccc(c(c1)CCN2CCNCC2)C(F)(F)F MS-0174 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)C(Cl)Cl MS-0175 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccc(cc4Cl)Cl MS-0176 c1ccc(c(c1)N2C(=O)c3ccc(cc3C2=O)Oc4ccc(cc4Cl)C(F)(F)F)F MS-0178 c1cc(c(cc1C(F)(F)F)Cl)Oc2ccc3c(c2)C(=O)OC3=O MS-0186 CCOC(=O)c1c2c(sc1NC(=O)c3ccccc3F)CCCC2 MS-0190 C1C2C1C(NC2)C(=O)O MS-0191 C1C(CN1)C(=O)O MS-0192 CN1/C(=C\c2ccccc2F)/C(=O)NC1=N MS-0194 Cc1cc(ccc1C(C)C)NC(=O)C2CC2C(=O)O MS-0197 c1c(cc(cc1F)F)N2C(=O)C3CC3C2=O MS-0198 c1c(cc(cc1F)F)NC(=O)C2CC2C(=O)O MS-0199 c1cc(c(cc1F)NC(=O)C2CC2C(=O)O)F MS-0200 CN1/C(=C\c2ccc(cc2)OC(F)(F)F)/C(=O)NC1=N MS-0202 c1cc2c(c(c1)Cl)nc(s2)NC(=O)C3CC3C(=O)O MS-0203 CCOC(=O)C1C(=O)CSC(S1)c2ccccc2 MS-0204 c1cc2c(cc1Br)cc(c(=O)o2)P(=O)(O)O MS-0205 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N(c3ccccc3)C(C)C MS-0207 C/C(=N/OC(=O)NC)/c1ccco1 MS-0208 c1c(cc(cc1F)F)/C(=N\O)/Cl MS-0210 Cc1cc(ccc1C(C)C)NC(=O)c2c(onc2c3c(cccc3Cl)F)C MS-0211 CCOC(=O)c1ccccc1NC(=O)c2c(onc2c3ccccc3)C MS-0212 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCc3ccc(cc3)OC MS-0214 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCc3ccc(cc3)F MS-0215 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCOCC3 MS-0216 Cc1c(c(no1)c2ccccc2)c3nc4ccccc4c(=O)o3 MS-0218 COC(=O)CN1CCOCC1 MS-0220 c1cc(c(cc1F)N2C(=O)C3CC3C2=O)F MS-0221 CC(C)c1ccc(cc1)N2C(=O)C3CC3C2=O MS-0223 Cc1cccc(c1)C(=O)Nc2ccc(c(c2)C)N3C(=O)c4ccc(cc4C3=O)Cl MS-0224 c1cc(cc(c1)Oc2cccc(n2)Cl)C(=O)O MS-0225 c1cc(ccc1C(=O)Nc2c(nccn2)C(=O)O)Cl MS-0226 c1cc(cc(c1)Oc2cccc(n2)Cl)C(=O)N3CCOCC3 MS-0227 CC1CN(CC(O1)C)C(=O)c2ccc(cc2)C(F)(F)F MS-0228 Cc1cc(ccc1N2C(=O)c3ccc(cc3C2=O)Cl)NC(=O)c4ccc(cc4)C(F)(F)F MS-0230 CC1CN(CC(O1)C)C(=O)c2ccccc2C(F)(F)F MS-0231 Cc1cc(nc2c1ccc(n2)N)C MS-0232 Cc1cc(ccc1Oc2cccc(c2)C(=O)/C(=C/N(C)C)/C#N)Cl MS-0234 CCNC(=O)CN1CCOCC1 MS-0239 c1cc(cc(c1)Br)C(=O)NCCCn2ccnc2 MS-0240 Cc1cccc(c1)N2C(=O)C3CC3C2=O MS-0242 Cc1ccc(cc1)N2C(=O)C3CC3C2=O MS-0243 c1cc(c(cc1Cl)Cl)NC(=O)NCCCn2ccnc2 MS-0244 c1cc(ccc1C(=O)NCCCn2ccnc2)C(F)(F)F MS-0246 c1ccc(c(c1)S(=O)(=O)NCCCn2ccnc2)Cl MS-0248 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCCCC3 MS-0249 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCCCC3 MS-0250 Cc1ccc(c2c1CC(N2)(C)C)NC(=O)c3ccc(cc3)F MS-0253 c1cc(c(cc1Cl)Cl)NC(=O)NCCN2CCOCC2 MS-0255 Cc1ccc(cc1)CCOc2ccc(cc2)[N+](=O)[O-] MS-0257 CC(C)(C)c1ccc(cc1)CC2CCC[N+](C2)(Cc3ccccc3)Cc4ccc(cc4)Br.[Br-] MS-0259 CC(C)(C)c1ccc(cc1)CC2CCC[N+](C2)(Cc3ccccc3)Cc4ccc(cc4)C(C)(C)C.[Br-] MS-0260 CCNC(=O)c1ccc(cc1)Cl MS-0262 c1ccc(cc1)CC2CCCN(C2)c3ccc(cc3)[N+](=O)[O-] MS-0265 CC(C)(C)c1ccc(cc1)CC2CCCN(C2)Cc3ccccc3 MS-0266 c1cc(ccc1NC(=O)Nc2ccc(cc2)Cl)Cl MS-0270 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl MS-0272 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc(cc3)Cl MS-0275 C/C(=N/OC(=O)Nc1ccc(cc1)Cl)/c2ccco2 MS-0276 CC(C)(C)c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccccc3 MS-0279 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3cccc(c3)Br MS-0280 c1ccc(cc1)C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] MS-0281 c1ccc(cc1)Oc2cccc(c2)/C=N/c3ccc(cc3)N4CCOCC4 MS-0283 CCCOc1ccc(cc1)/C=N/c2ccc(cc2)N3CCOCC3 MS-0284 c1cnc(c(n1)C(=O)O)N MS-0291 CC(c1ccccc1)[NH+]2CC[NH+](CC2)c3ccc(c(c3)Cl)Cl.[Cl-].[Cl-] MS-0292 c1cc(c(cc1N2CCN(CC2)C(=O)C3CC3C(=O)O)Cl)Cl MS-0294 c1cc(ccc1Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])N3CCOCC3 MS-0296 c1ccc(cc1)CN2CCC(CC2)Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] MS-0300 c1ccc(cc1)C2CCN(CC2)CC(=O)c3ccc(cc3)Br MS-0302 c1ccc(cc1)C2CCN(CC2)C(=O)Nc3cccc(c3)F MS-0303 c1cc(ccc1Cc2ccncc2)N MS-0305 Cc1ccc(cc1)CS(=O)(=O)NC(=O)N2CCC(CC2)c3ccccc3 MS-0306 c1cc(ccc1CNc2cnccn2)Cl MS-0307 c1cc(cnc1)CNc2ccc(cc2Cl)Br MS-0308 CCOC(=O)CN1CCC(CC1)c2ccccc2 MS-0309 COC(=O)c1cccc(c1)Oc2cccc(n2)Cl MS-0310 c1cc(ccc1Cc2ccncc2)NC(=O)Nc3ccc(c(c3)Cl)Cl MS-0311 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)Cc3ccncc3 MS-0312 c1ccc(cc1)/C=C/C(=O)N2CCC(CC2)c3ccccc3 MS-0314 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC(=O)O MS-0316 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(Cc2cccnc2)c3ccc(cc3Cl)Br MS-0317 Cc1ccc(cc1)CS(=O)(=O)NC(=O)N(Cc2ccc(cc2)Cl)c3cnccn3 MS-0322 CCOC(=O)c1c2c(sc1NC(=O)NS(=O)(=O)c3ccc(cc3)C)CCCC2 MS-0323 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)c3nc4ccc(cc4s3)C MS-0324 CNC(=O)c1cccc(c1)Oc2cccc(n2)Cl MS-0326 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCC(=O)O MS-0328 Cc1csc(c1NC(=O)C2CCCCC2)C(=O)OC MS-0329 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCCC3 MS-0330 Cc1ccc2cc(sc2c1)c3ccc(cc3)NC(=O)[C@@H]4C[C@@H]4C(=O)O MS-0331 CCCOc1ccc(cc1)/C=C\2/C(=O)NC(=O)S2 MS-0333 c1ccc(cc1)Sc2cccc(c2C#N)Cl MS-0335 c1cc(ccc1/C=C\2/C(=O)NC(=O)S2)F MS-0336 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccc(cc3)Cl)Cl MS-0337 c1cc(ccc1C2=CCN(CC2)c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl MS-0338 c1cc(ccc1CC(=O)N)OCC(CN2CCCCC2)O MS-0339 CC(C)(C)c1ccc(cc1)C(=O)N2CC(C2)C(=O)O MS-0341 c1cc(ccc1CC(=O)N)OCC2CO2 MS-0342 c1ccc2c(c1)c(=O)c3c(s2)cccc3Cl MS-0343 c1ccc(c(c1)NC(=O)C2CC2C(=O)O)F MS-0345 c1cc(ccc1CC(=O)N)OCC(CN2CCOCC2)O MS-0348 c1cc(ccc1CC(=O)N)OCC(CNN2CCOCC2)O MS-0349 c1cc(c(cc1Cl)Cl)C(=O)N2CC3CC3C2C(=O)O MS-0351 c1cc(sc1)C(=O)NCCN2CCOCC2 MS-0352 c1cc(cc(c1)C(F)(F)F)C(=O)N2CC3CC3C2C(=O)O MS-0353 c1cc(ccc1C(=O)N2CC3CC3C2C(=O)O)F MS-0354 c1cc(sc1)C(=O)N2CC3CC3C2C(=O)O MS-0356 c1cc(ccc1C(=O)N2CC3CC3C2C(=O)O)Cl MS-0358 C=CCONC(=O)c1ccc(cc1)F MS-0359 c1cc(c(c(c1)[N+](=O)[O-])N2CCC(=CC2)c3ccc(cc3)Cl)[N+](=O)[O-] MS-0362 CC1CN(CC(O1)C)c2ccc(cc2)Nc3c(cccc3[N+](=O)[O-])[N+](=O)[O-] MS-0363 c1cc(c(c(c1)F)/C=C\2/C(=O)NC(=O)S2)F MS-0365 c1cc(ccc1c2csc(n2)N)Br MS-0371 CCCCCCN1CCC(=CC1)c2ccc(cc2)Cl MS-0377 Cc1cc(ccc1C(C)C)NC2C(=O)NC(=O)S2 MS-0378 c1cc(c(cc1Cl)Cl)OCCNC(=O)CCl MS-0379 Cc1ccccc1C(=O)/N=c\2/n(ccs2)C MS-0381 c1ccc2c(c1)ncc(n2)c3cccs3 MS-0383 Cn\1ccs/c1=N\C(=O)c2ccccc2F MS-0385 c1cc(c(c(c1)Cl)Cl)OCC[NH3+].[Cl-] MS-0388 C[NH+](C)CCOc1ccc(cc1Cl)Cl.[Cl-] MS-0389 c1cnc(nc1)P(=O)(O)O MS-0394 c1cc(ccc1C(CN2CCOCC2)O)F MS-0395 Cc1cc2c(c(c1)Br)nc(oc2=O)C MS-0396 c1cc(ccc1CC#N)NC2C(=O)NC(=O)S2 MS-0398 Cc1cc(ccc1C(C)C)Nc2c(c(ncn2)Nc3ccc(c(c3)C)C(C)C)[N+](=O)[O-] MS-0401 CCOC(=O)C(=O)Nc1nc(c(s1)C)c2ccc(cc2)CCCl MS-0403 c1ccc(c(c1)/C=C/2\C(=O)NC(=O)S2)O MS-0405 c1ccc(cc1)C2CCN(CC2)C3C(=O)NC(=O)S3 MS-0408 c1cc(c(c(c1)Cl)OCCCC(=O)O)Cl MS-0409 CC(C)N(c1ccccc1)c2c(c(ncn2)Cl)[N+](=O)[O-] MS-0410 c1cc(nc(c1[N+](=O)[O-])N2CC(C2)C(=O)O)Cl MS-0412 CC1(C(=O)N(C(=O)N1)CC(=O)c2ccc(cc2)Br)c3ccccc3 MS-0414 CNC(=O)C1CN(C1)c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] MS-0415 CCOC(=O)C1CN(C1)c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] MS-0417 CCOC(=O)Cn1c(nc2ccc(cc2c1=O)Cl)C MS-0418 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)COc4ccc(cc4)F MS-0420 c1cc(ccc1OCC(=O)NCC(=O)O)F MS-0422 CCc1nc2c(cc(cc2Br)C)c(=O)o1 MS-0424 c1ccc2c(c1)C(=O)N(C2=O)OCCBr MS-0425 Cc1cc2c(c(c1)Br)nc(n(c2=O)CC(=O)OC)C(F)(F)F MS-0426 Cc1ccc(c(c1)C(=O)O)NC(=O)c2cccc(c2)Br MS-0430 Cc1ccc2c(c1)c(=O)oc(n2)c3cccc(c3)Br MS-0431 Cc1cc(ccc1C(C)C)NC(=O)COc2ccc(cc2)F MS-0432 CC1CCc2cc(ccc2N1C(=O)c3ccccc3)F MS-0433 Cc1ccc(cc1)Oc2[nH]nnn2 MS-0436 c1cc(c(cc1Cl)Cl)CNc2cnccn2 MS-0437 CCn1ccsc1=[NH2+].[I-] MS-0438 Cc1ccc(cc1)CNc2cnccn2 MS-0439 c1cc(ccc1CNc2cnccn2)F MS-0440 CSc1nc(cc(n1)O)Cc2ccccc2 MS-0442 CCOc1nc(nc(n1)Oc2ccc(cc2)[N+](=O)[O-])OCC MS-0444 c1cc(c(cc1O)F)N2C(=O)C3=C(C2=O)CCCC3 MS-0446 c1ccc(c(c1)/C(=N/O)/Cl)F MS-0447 COc1ccc(cc1OC)CCNC(=O)CI MS-0448 CC(C)(C)c1cccc(c1)Oc2[nH]nnn2 MS-0449 CCc1cccc(c1)Oc2[nH]nnn2 MS-0451 c1cc(c(cc1Cl)NC(=O)C(F)(F)F)C(=O)O MS-0452 Cc1cc(nc(n1)S(=O)(=O)C)C MS-0453 c1ccc(cc1)/N=C\2/N(CCS2)C(=S)Nc3cccc(c3)Cl MS-0456 c1ccc2c(c1)C(=O)N(C2=O)OCCON3C(=O)c4ccccc4C3=O MS-0459 Cc1cc(ccc1C(C)C)NC(=O)C MS-0460 Cn1ccsc1=[NH2+].[I-] MS-0461 C(CO[NH3+])O[NH3+].[Cl-].[Cl-] MS-0462 CC1(OCC(O1)C2C(=C(C(=O)O2)O)OCc3ccc(cc3)Br)C MS-0464 c1ccc2c(c1)C(=O)N(C2=O)OCc3cccc(c3)Br MS-0467 CC1(OCC(O1)C2C(=C(C(=O)O2)OCC(=O)c3ccc(cc3)F)OCC(=O)c4ccc(cc4)F)C MS-0468 CN1/C(=C\c2ccc(cc2)F)/C(=O)NC1=N MS-0471 CCOC(=O)Cc1c2ccccc2c(=O)[nH]n1 MS-0472 c1ccc(c(c1)/C=N/Nc2ccccc2Cl)F MS-0473 c1cc(cc(c1)Br)CO[NH3+].[Cl-] MS-0474 c1cc(ccc1/C=C/2\C(=O)NC(=N)S2)Br MS-0477 CN1/C(=C/c2ccc(cc2)Br)/C(=O)NC1=N MS-0478 c1cc(nc(c1[N+](=O)[O-])N2CCCC2C(=O)O)Cl MS-0480 c1cc(nc(c1[N+](=O)[O-])NCC(=O)O)Cl MS-0481 CC(C(=O)O)Nc1c(ccc(n1)Cl)[N+](=O)[O-] MS-0482 Cc1cc(ccc1C(C)C)n2cnnn2 MS-0483 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3ccc(cc3)C(C)(C)C MS-0484 c1cc(nc(c1[N+](=O)[O-])NCCCC(=O)O)NCCCC(=O)O MS-0486 CCc1nc2ccc(cc2c(=O)n1CC(=O)OC)Br MS-0488 CC(C)(C)c1ccc(cc1)Cn2c(=O)c3ccccc3c(n2)CC(=O)O MS-0489 CCCCC(CN1CCC(CC1)c2ccccc2)O MS-0497 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3ccc(cc3)Cl MS-0504 CCCCC(C[N+]1(CCC(CC1)c2ccccc2)C)O.[I-] MS-0507 c1cc(ccc1C(=O)N)N2C(=O)C3CC3C2=O MS-0508 CCCCC(C[N+]1(CCC(CC1)c2ccccc2)Cc3ccc(cc3)Br)O.[Br-] MS-0510 c1cc(ccc1C(=O)N)NC(=O)C2CC2C(=O)O MS-0512 CCCCCCN1CCN(CC1)c2ccc(cc2)F MS-0514 CCCCCCN1CCN(CC1)c2ccc(cc2)OC MS-0515 CCCCC(CNC1CCN(CC1)Cc2ccccc2)O MS-0516 CCCCCCN1CCN(CC1)c2ccc(cc2)Cl MS-0517 CCCCCCN1CCN(CC1)c2ccccc2Cl MS-0518 c1cc(ccc1NC(=O)CC#N)F MS-0519 c1cc(ccc1/C(=C(\C#N)/C(=O)Nc2ccc(cc2)F)/O)Cl MS-0520 Cc1ccc(c(c1)NC(=O)/C(=C(/c2ccc(cc2)C(F)(F)F)\O)/C#N)F MS-0521 Cc1ccc(c(c1)NC(=O)/C(=C(/c2ccc(cc2)C(C)(C)C)\O)/C#N)F MS-0522 Cc1ccc(c(c1)NC(=O)CC#N)F MS-0523 Cc1ccc(c(c1)NC(=O)/C(=C(/c2ccccc2[N+](=O)[O-])\O)/C#N)F MS-0526 CCOC(=O)C(CCSC)NC(=O)c1c(onc1c2c(cccc2Cl)F)C MS-0527 c1cc(ccc1C(Cn2cncn2)(c3ccc(cc3)Cl)O)F MS-0532 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)O MS-0533 CCCCCCN1CCN(CC1)c2cccc(c2)C(F)(F)F MS-0534 CCCCCCN1CCN(CC1)c2cccc(c2)Cl MS-0535 CCCCCCN1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] MS-0536 Cc1csc(c1NC(=O)c2ccc(cc2)Cl)C(=O)OC MS-0537 Cc1csc(c1NC(=O)c2ccc(cc2Cl)Cl)C(=O)O MS-0538 Cc1csc2c1nc(oc2=O)c3ccc(cc3Cl)Cl MS-0539 CCCCCCN1CCN(CC1)c2ccccc2C MS-0541 c1cc(ccc1C(=O)CN2C(=O)C3CC3C2=O)F MS-0543 c1cc(ccc1C(=O)CN2C(=O)CSC2=O)Br MS-0545 CCCCCCCCN1C(=O)C2CC2C1=O MS-0546 c1ccc(c(c1)CN2C(=O)CSC2=O)Cl MS-0547 c1cc(cc(c1)N2CCN(CC2)C3C(=O)NC(=O)S3)C(F)(F)F MS-0548 CCCCCCCCCN1CCN(CC1)c2ccc(c(c2)Cl)Cl MS-0553 c1cc(ccc1C(=O)Cn2cnc(c2Cl)Cl)F MS-0554 CCCCCCCCN1CCN(CC1)c2ccc(c(c2)Cl)Cl MS-0556 c1cc(ccc1C(Cn2cnc(c2Cl)Cl)(c3ccc(cc3)Cl)O)F MS-0557 c1ccc(cc1)C(=O)Cn2cnc(c2Cl)Cl MS-0558 c1ccc2c(c1)C(=O)N(C2=O)CCCn3cnc(c3Cl)Cl MS-0559 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccccc3OC MS-0560 COC(=O)Cn1c2ccccc2c(=O)oc1=O MS-0562 c1ccc(c(c1)C(=O)N)NCc2ccc(cc2)Cl MS-0563 c1ccc2c(c1)c(=O)oc(=O)n2Cc3ccc(cc3)Cl MS-0565 COC(=O)CSCC(=O)c1ccc(cc1)Br MS-0567 Cc1ccc(c2c1CC(O2)(C)C)C#N MS-0568 Cc1ccc(c2c1CC(O2)(C)C)C(=O)N MS-0570 c1cc(c(cc1CN2CCCSC2=S)Cl)Cl MS-0571 c1nc(c(n1CCN2C(=O)C3CC3C2=O)Cl)Cl MS-0572 CCOC(=O)C(C)N1CCCSC1=S MS-0575 c1ccc2c(c1)c(c(s2)C(=O)N3CCCC3)Cl MS-0580 c1ccc2c(c1)c(c(s2)C(=O)N3CCOCC3)Cl MS-0581 COC(=O)c1c(c2ccccc2s1)Cl MS-0583 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)c3c(cccc3Cl)Cl MS-0585 CCOC(=O)N/N=C(\C)/c1ccc(cc1)Oc2ncccn2 MS-0586 c1ccc(cc1)COc2cccc(c2)/C=C/C(=O)O MS-0590 CC(C)CC(C(=O)O)Nc1c(ccc(n1)Cl)[N+](=O)[O-] MS-0591 CCOC1c2c(ccc(c2OC1(C)C)[N+](=O)[O-])C MS-0592 c1cc2cccc3c2c(c1)C(=O)N3CC(=O)O MS-0594 CCOC1c2c(ccc(c2OC1(C)C)NC(=O)NS(=O)(=O)c3ccc(cc3)C)C MS-0599 c1ccc(cc1)C(=O)CCN2C(=O)C3CC3C2=O MS-0601 c1cc(cc(c1)OCc2ccc(cc2)C(F)(F)F)/C=C/C(=O)O MS-0602 CC1CN(CC(O1)C)C(=O)/C=C/c2cccc(c2)OCc3ccc(cc3)C(F)(F)F MS-0604 Cc1cc(ccc1C(C)C)NC(=S)NC(=O)c2ccc(cc2Cl)Cl MS-0605 Cc1cc(cc(=O)o1)OC(=O)c2conc2c3c(cccc3Cl)Cl MS-0607 Cc1cc(cc(=O)o1)OC(=O)/C=C/c2cccc(c2)OCc3ccc(cc3)C(F)(F)F MS-0608 c1cc(oc1)CNC(=S)NC(=O)c2ccc(cc2Cl)Cl MS-0609 c1cc(cc(c1)OCc2ccc(cc2)C(F)(F)F)/C=C/C(=O)N3CCOCC3 MS-0615 c1ccc(cc1)C2(c3ccccc3NC2=O)O MS-0618 c1cc(c(cc1CNc2cnccn2)Cl)Cl MS-0621 CC(C(=O)OC)ON1C(=O)c2ccccc2C1=O MS-0622 c1cc2c(cc1O)OCC2=O MS-0624 COc1ccc(cc1)CNC(=O)/C=C/c2cccc(c2)OCc3ccc(cc3)C(F)(F)F MS-0626 Cc1ccccc1N2C(=O)C3CC3C2=O MS-0627 c1cc(ccc1N)OCC(=O)O.O MS-0628 CCOC(=O)C(Cc1ccc(cc1)C(F)(F)F)(C(=O)OCC)NC(=O)C MS-0630 c1cc(cc(c1)F)NC(=O)N2CCC(=CC2)c3ccc(cc3)Cl MS-0632 CC(C)(C)c1ccc(cc1)Cn2nc(nn2)Cc3cccc(c3)C(C)(C)C MS-0635 c1cc(ccc1CC(C(=O)O)[NH3+])C(F)(F)F.[Cl-] MS-0636 c1cc(ccc1OC(F)(F)F)S(=O)(=O)NN2CCOCC2 MS-0637 Cc1ccc(c2c1C(C(O2)(C)C)Br)[N+](=O)[O-] MS-0639 Cc1ccc(c2c1C(C(O2)(C)C)N3CCCCC3)[N+](=O)[O-] MS-0641 Cc1ccc(c2c1C(C(O2)(C)C)N3CCCC3)[N+](=O)[O-] MS-0642 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC(=O)OC MS-0644 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(cccc2F)F MS-0647 Cc1ccccc1N2C(=O)c3ccccc3C2=O MS-0649 Cc1cc(c(c(c1)[N+](=O)[O-])NC(C)C(=O)N2CCOCC2)[N+](=O)[O-] MS-0650 CCCCCCC1OCC(O1)C2C(=C(C(=O)O2)O)O MS-0651 Cc1ccc(c2c1C(C(O2)(C)C)N3CC(OC(C3)C)C)[N+](=O)[O-] MS-0653 c1cnc(cn1)NC(=O)CC#N MS-0654 c1cc(ccc1C(F)(F)F)NC(=O)CC#N MS-0655 COCCN/C(=C(\C#N)/C(=O)c1ccc(cc1)Cl)/SC MS-0658 CCOP(=O)(Cc1ccccc1N2C(=O)c3ccccc3C2=O)OCC MS-0659 c1ccc(cc1)OCC(=O)/C(=C(/Nc2ccc(cc2F)F)\O)/C#N MS-0660 c1cc(sc1)C(=O)/C(=C(/Nc2ccc(cc2F)F)\O)/C#N MS-0661 c1cc(cc(c1)Br)C(=O)/C(=C(/Nc2ccc(cc2F)F)\O)/C#N MS-0662 c1ccc(cc1)CCNS(=O)(=O)c2ccccc2[N+](=O)[O-] MS-0664 c1ccc2c(c1)c(c([nH]2)C(=O)O)CC(=O)O MS-0665 c1ccc(cc1)CCCCNS(=O)(=O)c2ccccc2[N+](=O)[O-] MS-0667 c1ccc(cc1)CCCCNS(=O)(=O)c2ccccc2N MS-0668 CCCCOC(=O)CCCc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] MS-0669 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCc2ccc(cc2)Cl MS-0670 c1ccc(cc1)CCNS(=O)(=O)c2ccccc2[NH3+].[Cl-] MS-0672 c1ccc2c(c1)N=NN(S2(=O)=O)Cc3ccc(cc3)Cl MS-0674 c1ccc(cc1)CCCCNS(=O)(=O)c2ccccc2[NH3+].[Cl-] MS-0676 c1ccc(c(c1)N)S(=O)(=O)NCc2ccc(cc2)Cl MS-0679 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCc2ccc(cc2)C(F)(F)F MS-0680 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCc2cccc(c2)Cl MS-0681 c1ccc(c(c1)CNS(=O)(=O)c2ccccc2[N+](=O)[O-])Cl MS-0682 c1cc(ccc1Oc2ccc(cc2Cl)[NH3+])F.[Cl-] MS-0683 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCc2ccc(c(c2)Cl)Cl MS-0684 CC(C)(C)c1ccc(cc1)NS(=O)(=O)c2ccccc2[N+](=O)[O-] MS-0685 CC(C)(C)c1ccc(cc1)N2N=Nc3ccccc3S2(=O)=O MS-0689 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)N(=O)=O MS-0690 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCc2cc(cc(c2)Cl)Cl MS-0692 c1ccc(c(c1)[NH3+])S(=O)(=O)NCc2cc(cc(c2)Cl)Cl.[Cl-] MS-0695 c1ccc(cc1)OCCNS(=O)(=O)c2ccccc2[N+](=O)[O-] MS-0696 c1ccc2c(c1)N=NN(S2(=O)=O)Cc3cc(cc(c3)Cl)Cl MS-0697 c1ccc(c(c1)[NH3+])S(=O)(=O)NCc2ccc(c(c2)Cl)Cl.[Cl-] MS-0698 c1ccc2c(c1)N=NN(S2(=O)=O)Cc3ccc(c(c3)Cl)Cl MS-0700 c1ccc(cc1)OCCNS(=O)(=O)c2ccccc2[NH3+].[Cl-] MS-0702 c1c(cnc(c1C(=O)O)O)[N+](=O)[O-] MS-0703 c1ccc(cc1)COc2ccc(cc2)C[NH3+].[Cl-] MS-0705 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)NC MS-0712 Cc1ccc(c(c1)O)NC(=O)c2ccc(cc2Cl)N MS-0714 CC(C)(C)c1ccc(cc1)CN2N=Nc3ccccc3S2(=O)=O MS-0716 c1ccc(c(c1)CNS(=O)(=O)c2ccccc2[NH3+])Cl.[Cl-] MS-0717 CC(=O)OC1CC2CC1C3C2CC=C3 MS-0719 c1c(cnc(c1[N+](=O)[O-])N2CC(C2)C(=O)O)[N+](=O)[O-] MS-0721 C/C(=N/OC(=O)NC)/c1ccc(cc1OC)OC MS-0722 CC(C)(C)N(C(=O)c1ccccc1)/N=C/c2ccccc2 MS-0723 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)CCCl MS-0725 c1ccc2c(c1)C3(C(=O)N2Cc4ccc(c(c4)Cl)Cl)OCCO3 MS-0730 c1ccc(cc1)C(C#N)C2CCCCC2 MS-0731 C/C(=N/NC(=S)NN)/c1ccccn1 MS-0735 c1ccc(cc1)C(C2CCCCC2)C(=O)N MS-0736 C/C(=N\NC(=S)NNC(=S)Nc1ccccc1Cl)/c2ccccn2 MS-0738 C/C(=N/Nc1nnc(s1)Nc2ccccc2Cl)/c3ccccn3 MS-0741 Cc1ccc(c2c1CC(O2)(C)C)NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-0744 C/C(=N/NC(=S)NNC(=S)Nc1ccc(c(c1)Cl)Cl)/c2ccco2 MS-0747 C/C(=N/Nc1nnc(s1)Nc2ccc(c(c2)Cl)Cl)/c3ccco3 MS-0749 C/C(=N/NC(=S)NNC(=S)Nc1ccccc1Cl)/c2ccco2 MS-0750 c1cc2c(cc1Br)C3(C(=O)N2)OCCO3 MS-0751 CCn1c(cc(=O)cc1c2ccc(cc2)Cl)C MS-0753 Cc1ccc2c(c1)C3(C(=O)N2S(=O)(=O)c4ccc(cc4)F)OCCO3 MS-0755 c1ccc2c(c1)C3(C(=O)N2S(=O)(=O)c4ccc(cc4[N+](=O)[O-])Cl)OCCO3 MS-0756 CC1C(OC2(O1)c3ccccc3NC2=O)C MS-0758 Cc1ccc2c(c1)C3(C(=O)N2)OCCO3 MS-0759 C/C(=N/NC(=S)NNC(=S)Nc1ccccc1F)/c2ccco2 MS-0760 CC1C(OC2(O1)c3ccccc3N(C2=O)S(=O)(=O)c4ccccc4Cl)C MS-0765 C=CCNC(=O)/C=C/c1cccc(c1)OCc2ccc(cc2)C(F)(F)F MS-0766 CC(C)O/C(=N\c1ccc(cc1Cl)Cl)/c2cccnc2 MS-0768 CC1C(OC2(O1)c3ccccc3N(C2=O)C4CCOC4=O)C MS-0773 Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)C(=O)N(c4ccc(cc4O3)C)C MS-0777 c1cc(c(c(c1)Cl)C(=O)C(Cl)Cl)Cl MS-0779 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2C)NC(=O)c4ccc(cc4)OC MS-0780 COc1ccc(cc1)CNc2c(cccn2)C(=O)Nc3cccnc3Cl MS-0782 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2C)NC(=O)c4ccc(cc4)O MS-0785 c1cc(c(nc1)Cl)C(=O)Nc2cccnc2Cl MS-0786 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)C(=O)Nc4ccc(cc4O3)C MS-0787 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NS(=O)(=O)c4ccc(cc4)OC MS-0788 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)c4ccc(cc4)OC MS-0790 Cc1csc(c1NC(=O)COc2c(cccc2Cl)Cl)C(=O)OC MS-0791 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)c4ccc(cc4Cl)Cl MS-0792 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)c4ccc(cc4)O MS-0794 Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)C(=O)Nc4ccc(cc4O3)C MS-0795 COc1ccc(cc1)C(=O)Nc2ccsc2C(=O)OC MS-0797 COC(=O)c1c(ccs1)NC(=O)c2cccc(c2)[N+](=O)[O-] MS-0798 COC(=O)c1c(ccs1)NC(=O)COc2cc(cc(c2)Cl)Cl MS-0799 c1ccc(cc1)CN2c3ccccc3C4(C2=O)SCCS4 MS-0804 c1cc(c(c(c1)Cl)C(=O)Nc2ccsc2C(=O)O)Cl MS-0806 Cc1csc(c1NC(=O)c2ccc(cc2)F)C(=O)OC MS-0808 Cc1csc(c1NC(=O)c2ccc(cc2)OC)C(=O)O MS-0810 Cc1csc(c1NC(=O)c2ccc(cc2)F)C(=O)O MS-0811 Cc1csc(c1NC(=O)c2cccc(c2)[N+](=O)[O-])C(=O)O MS-0812 Cc1csc(c1NC(=O)c2c(cccc2Cl)Cl)C(=O)O MS-0814 c1ccc(cc1)Oc2cccc(c2)C(=O)Nc3ccsc3C(=O)O MS-0815 Cc1cc(ccc1C(C)C)N2CC(=O)N(CC2=O)c3ccc(c(c3)C)C(C)C MS-0817 CN(C)/C=C(\C#N)/C(=O)c1cccc(c1)Oc2ccc(cc2)Br MS-0821 CC(C)(C)c1ccc(cc1)Oc2cccc(c2)C(=O)/C(=C\N(C)C)/C#N MS-0826 CCOc1ccc(cc1)Oc2ccccc2C(=O)/C(=C/N(C)C)/C#N MS-0827 Cc1ccccc1Oc2cccc(c2)C(=O)/C(=C/N(C)C)/C#N MS-0828 CN(C)/C=C(\C#N)/C(=O)c1cccnc1Oc2ccc(cc2F)F MS-0829 CCOc1ccc(cc1)Oc2ccccc2C(=O)OC MS-0831 c1ccc(cc1)Oc2cccc(c2)C#N MS-0832 CN1CC(=O)N(C1=O)c2ccc(cc2Cl)Cl MS-0833 c1cc(cc(c1)Oc2ccc(c(n2)Cl)C(F)(F)F)C(F)(F)F MS-0834 CCOC(=O)c1cccc(c1)Oc2ccc(cc2C)Cl MS-0835 CCOc1cccc(c1)Oc2c(cccn2)C(=O)/C(=C/N(C)C)/C#N MS-0836 CCc1ccc(cc1)Oc2ccc(cc2)C(=O)/C(=C/N(C)C)/C#N MS-0840 c1cc(cc(c1)Oc2ccc(cc2)C(=O)CC#N)C(F)(F)F MS-0841 CN(C)/C=C(\C#N)/C(=O)c1ccc(cn1)Oc2cccc(c2)C(F)(F)F MS-0842 CCc1ccc(cc1)Oc2cccc(c2)C(=O)CC#N MS-0843 c1ccc2c(c1)C(=O)N(S2(=O)=O)C/C=C/CBr MS-0844 CCCCCCCCOc1ccc(c(c1)O)C(=O)c2ccccc2O MS-0849 CNC(=O)N(C)C(=O)Nc1ccccc1F MS-0851 COC(=O)c1ccccc1Oc2ccc(cc2)F MS-0852 COC(=O)c1ccccc1Oc2ccc(cc2)Cl MS-0853 CCOC(=O)c1ccc(cc1)Oc2cccc(c2)Cl MS-0854 c1cc(ccc1Nc2ccc(cc2[N+](=O)[O-])Br)O MS-0856 CC(C)(C)c1ccc(cc1)N/C(=C/[N+](=O)[O-])/SC MS-0858 c1cc[n+](c(c1)C=[N+]([O-])[O-])Cc2ccc(cc2)Cl MS-0859 Cc1cc(c(nc1)Br)C(=O)OC MS-0860 CCOC(=O)C(C)Oc1ccc(cc1)Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F MS-0861 c1ccc2c(c1)C(=O)C(=O)N2C/C=C/CCl MS-0865 CCCCCCCCCCc1ccc(cc1)N/C(=C/[N+](=O)[O-])/SC MS-0866 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)N3CCN(CC3)c4ccc(cc4)F MS-0867 Cc1cccc(c1)C2C(=O)C(=C(CC2(C)C)O)/C(=N/OCC=C)/C MS-0869 Cc1ccccc1Oc2c(cccn2)C(=O)/C(=C/N(C)C)/C#N MS-0870 CCN/C=C(\C#N)/C(=O)C(C)(C)C MS-0872 CC(C)(C)C(=O)/C(=C/N1CCCCC1)/C#N MS-0873 c1cc(cc(c1)Oc2ccc(cc2)Br)C(=O)CC#N MS-0875 CCOC(=O)c1cccc(c1)Oc2ccc(cc2)C(C)(C)C MS-0876 CN(C)/C=C(\C#N)/C(=O)c1cccnc1Oc2cc(cc(c2)Cl)Cl MS-0877 c1ccc(cc1)CNc2cnccn2 MS-0878 CC(C)c1ccc(cc1)N/C(=C/[N+](=O)[O-])/SC MS-0881 CC(C)CN/C(=C/[N+](=O)[O-])/SC MS-0885 CN(C)/C=C(\C#N)/C(=O)c1cccnc1Oc2cccc(c2)F MS-0887 c1cc(cc(c1)Oc2ccc(c(c2)F)C(F)(F)F)C(=O)CC#N MS-0888 CCOC(=O)CNc1ccc(c(c1)Cl)Cl MS-0890 CSc1cc(n[nH]1)c2ccc(cc2)F MS-0893 CN(C)/C=C(\C#N)/C(=O)c1ccccc1Oc2ccc(c(c2)C(F)(F)F)Cl MS-0898 c1ccc(c(c1)C(=O)CC#N)Oc2ccc(cc2)Cl MS-0899 c1ccc(cc1)c2nc(cs2)c3ccc(cc3Cl)Cl MS-0900 CC(C)c1ccc(cc1)Oc2cccc(c2)C(=O)/C(=C/N(C)C)/C#N MS-0901 CCc1ccc(cc1)Oc2ccc(cc2)C(=O)OC MS-0902 CN(C)/C=C(\C#N)/C(=O)c1ccc(cc1)Oc2cccc(c2)Cl MS-0903 CCC(=O)C1=C(C(C(CC1=O)(C)C)c2ccccc2)O MS-0905 CC(C)(C)c1ccc(cc1)Oc2cccc(c2)C(=O)CC#N MS-0906 COC(=O)c1ccccc1Oc2ccc(c(c2)C(F)(F)F)Cl MS-0907 CCOC(=O)c1ccc(cc1)Oc2cccc(c2)C(F)(F)F MS-0909 c1ccc(c(c1)C(=O)CC#N)Oc2ccc(c(c2)C(F)(F)F)Cl MS-0911 CN(C)/C=C(\C#N)/C(=O)c1ccccc1Oc2cccc(c2)F MS-0913 c1cc2c(cc1[N+](=O)[O-])C3(C(=O)N2)OCCO3 MS-0917 CN(C)/C=C(\C#N)/C(=O)c1ccccc1Oc2ccc(c(c2)F)C(F)(F)F MS-0922 C=C(C(=O)Nc1ccc(cc1)Cl)Cl MS-0923 c1ccc2c(c1)C(=O)N(S2(=O)=O)C/C(=C\CCl)/Cl MS-0924 CC1(CC(CC(N1)(C)C)OC(=O)CCCCCCCCC(=O)OC2CC(NC(C2)(C)C)(C)C)C MS-0925 Cc1ccccc1Oc2cccc(c2)C3CCC(=O)CC3=O MS-0928 CC1(C(=O)N(C(=O)N1)CC(=O)N2CCN(CC2)c3ccc(cc3)F)c4ccccc4 MS-0930 c1cc(c(cc1CN2c3ccc(cc3C4(C2=O)OCCO4)[N+](=O)[O-])Cl)Cl MS-0931 Cc1cc(ccc1C(C)C)NC(=O)CCl MS-0932 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)CCl MS-0935 COc1ccc(c(c1)S(=O)(=O)N2CCC(=CC2)c3ccc(cc3)Cl)OC MS-0936 c1cc(ccc1C2=CCN(CC2)S(=O)(=O)c3ccc(cc3Cl)Cl)Cl MS-0937 Cc1ccc(n1c2ccc(cc2)Cl)C MS-0938 Cc1cc(c(n1c2ccc(cc2)Cl)C)C(=O)C(F)(F)F MS-0939 c1ccc(cc1)S(=O)(=O)N2CCC(=CC2)c3ccc(cc3)Cl MS-0940 CCOC(=O)c1ccc(cc1)n2c(cc(c2C)C(=O)C(F)(F)F)C MS-0941 Cc1ccc(n1c2ccc(c(c2)Cl)Cl)C MS-0943 Cc1cc(c(n1c2ccc(cc2)Cl)C)C=O MS-0945 Cc1cc(c(n1c2ccc(cc2)Cl)C)C(=O)C(=O)N(C)C MS-0947 Cc1cc(c(n1c2ccc(cc2)Cl)C)C#N MS-0951 Cc1cc(c(n1c2ccc(c(c2)Cl)Cl)C)C(=O)C(=O)O MS-0952 Cc1cc(c(n1c2ccc(c(c2)Cl)Cl)C)C(=O)C(=O)N(C)C MS-0953 Cc1cc(c(n1c2ccc(cc2)Cl)C)C(=O)C(=O)O MS-0955 c1ccc2c(c1)C(=O)Nc3ccccc3N2 MS-0956 CC(C(=O)O)N(c1ccc(c(c1)Cl)F)C(=O)c2ccccc2 MS-0965 c1cc(c(c(c1)Cl)OCC(=O)N2CCN(CC2)C=O)Cl MS-0969 Cc1cc(c(n1c2ccc(cc2)Cl)C)C(=O)C(=O)Nc3ccc(cc3)C(F)(F)F MS-0970 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)C=O MS-0972 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN(CC3)C=O MS-0973 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F MS-0975 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)CC#N MS-0979 C/C(=N\NC(=S)NN)/c1ccco1 MS-0980 CC(C)(C)c1ccc(cc1)CN2C(=O)CSC2=O MS-0982 Cc1cc(cc(c1)CN2C(=O)CSC2=O)C MS-0983 c1cc(ccc1F)S(=O)(=O)N2CCN(CC2)C=O MS-0984 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)F MS-0985 c1cc(ccc1F)S(=O)(=O)N2CCNCC2 MS-0986 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)C=O)C(F)(F)F MS-0987 Cc1cc(cc(c1)CN2C(=O)/C(=C/c3ccc(cc3)F)/SC2=O)C MS-0988 c1cc(cc(c1)S(=O)(=O)N2CCNCC2)C(F)(F)F MS-0989 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)C(=O)c3c(cccc3Cl)Cl)C(F)(F)F MS-0990 CC(C)(C)c1ccc(cc1)CN2C(=O)/C(=C\c3ccc(cc3)F)/SC2=O MS-0991 Cc1cc(cc(c1)CN2C(=O)/C(=C\c3cccc(c3)C(F)(F)F)/SC2=O)C MS-0992 CC(C)(C)c1ccc(cc1)CN2C(=O)/C(=C\c3cccc(c3)C(F)(F)F)/SC2=O MS-0993 CC(C)COC(=O)C(C)N(c1ccc(c(c1)Cl)F)C(=O)c2ccccc2 MS-0994 c1c(c(cc(c1S(=O)(=O)N2CCCCC2)Cl)Cl)C(=O)O MS-0995 Cc1cc(nc(n1)NC(=O)COc2cc(cc(c2)Cl)Cl)C MS-0996 c1c(c(cc(c1S(=O)(=O)N2CCOCC2)Cl)Cl)C(=O)O MS-0997 CCCCOC(=O)C(C)N(c1ccc(c(c1)Cl)F)C(=O)c2ccccc2 MS-0999 CCCCCOC(=O)C(C)N(c1ccc(c(c1)Cl)F)C(=O)c2ccccc2 MS-1000 c1cc(sc1)c2nnc(n2C3CCCCC3)S MS-10000 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)F)/C(=O)C MS-10001 CC(C)(C)C(=O)/C(=C\Nc1cc(cc(c1)Cl)Cl)/C#N MS-10002 CC(C)(C)C(=O)/C(=C/Nc1ccccc1F)/C#N MS-10003 Cc1cc(ccc1Cl)C(=O)CC2C(=O)CC(CC2=O)(C)C MS-10004 CC(C)(C)c1c2c(nn1C)-c3ccc(cc3C2=O)N MS-10005 CC(C)(C)c1c2c(nn1C)-c3ccc(cc3C2=O)NC(=O)C(F)(F)F MS-10006 CC(C)(C)C(=O)/C(=C\Nc1ccc(cc1Cl)Cl)/C#N MS-10007 CC(C)(C)S(=O)(=O)/C(=C\Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C#N MS-10008 Cc1cc(c2ccccc2n1)N/C=C(\C#N)/S(=O)(=O)C(C)(C)C MS-10009 CC(C)(C)c1c2c(nn1C)-c3ccc(cc3C2=O)NC(=O)C4CC4 MS-10010 Cc1cc(c2ccccc2n1)N/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Cl MS-10011 CC1CC(=CC(=O)C1)Nc2cc(cc(c2)Cl)N MS-10012 CCOC(=O)c1cccc(c1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)C(C)(C)C MS-10013 c1ccc2c(c1)/C(=C/c3ccsc3)/C(=O)N2 MS-10014 c1cc(c(cc1[N+](=O)[O-])C(=O)Nc2ccc(cc2F)F)Cl MS-10015 c1cc2c(cc1NC(=O)c3cc(ccc3Cl)[N+](=O)[O-])OCO2 MS-10016 c1cc(ccc1NC(=O)c2cc(ccc2Cl)[N+](=O)[O-])Br MS-10017 c1cc(c(cc1[N+](=O)[O-])C(=O)Nc2nccs2)Cl MS-10018 CNC(=S)N1CCN(CC1)C/C=C/c2ccccc2 MS-10019 CC(C)(C)c1ccc(cc1)CN2C(=O)/C(=C/c3ccc(cc3)C(C)(C)C)/SC2=O MS-1002 c1ccc(cc1)C(=O)N2CCN(CC2)c3ccccn3 MS-10020 CCCNC(=O)NCCN1CCOCC1 MS-10021 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccccc3 MS-10022 CCOC(=O)c1cccc(c1)NC=C2C(=O)NC(=O)NC2=O MS-10023 CCCn1c(=N)c2c(c(=O)[nH]c(n2)c3cccs3)[nH]c1=O MS-10024 COc1ccccc1c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccccc4 MS-10025 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl MS-10026 c1ccc(cc1)/C=C/CN2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl MS-10027 c1c(cc(cc1[N+](=O)[O-])[N+](=O)[O-])C(=O)N2CCN(CC2)C=O MS-10028 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-] MS-10029 CCC1CCCCN1S(=O)(=O)c2ccccc2[N+](=O)[O-] MS-1003 Cc1cc(no1)NC(=O)c2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-] MS-10030 c1c(cc(cc1[N+](=O)[O-])[N+](=O)[O-])C(=O)NC2CC2 MS-10031 c1c(cc(cc1[N+](=O)[O-])[N+](=O)[O-])C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-10032 c1cc(ccc1CNS(=O)(=O)c2ccc(cc2)Cl)F MS-10033 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3cc(ccc3C)Cl MS-10034 c1ccc(cc1)COc2cccnc2NS(=O)(=O)c3cccs3 MS-10035 Cc1cc(no1)NC(=O)c2ccc(cc2Cl)Cl MS-10036 c1cc(c(cc1Cl)Cl)C(=O)NCCN2CCOCC2 MS-10037 COc1ccc(cn1)NC(=O)c2ccc(cc2Cl)Cl MS-10038 c1ccc(cc1)COc2cccnc2NS(=O)(=O)c3ccccc3 MS-10039 CCC1CCCCN1S(=O)(=O)c2ccccc2N MS-1004 Cc1cc(no1)NC(=O)c2c(cccc2F)F MS-10041 c1ccc(cc1)NC(=O)c2[nH]ccn2 MS-1005 CCN1C(=O)/C(=C/Nc2cccc(c2)C(=O)OCC)/SC1=S MS-10050 CC(C)(C)NC(=O)N1CCN(CC1)C=O MS-10051 CCCCCCNC(=O)N1CCN(CC1)c2cc(ccc2C)Cl MS-10052 Cc1ccc(cc1N2CCN(CC2)C(=O)NC(C)(C)C)Cl MS-10053 Cc1ccc(cc1N2CCN(CC2)C(=O)Nc3ccc(c(c3)C)Br)Cl MS-10054 CCC(C)NC(=O)N1CCN(CC1)Cc2ccccc2 MS-10055 CC(C)(C)NC(=O)N1CCN(CC1)Cc2ccccc2 MS-10056 CCC(C)NC(=O)N1CCN(CC1)c2ccccc2F MS-10057 c1ccc(c(c1)N2CCN(CC2)C(=O)Nc3ccc(cc3Cl)C(F)(F)F)F MS-10058 Cc1cc(ccc1Br)NC(=O)N2CCN(CC2)c3ccccc3F MS-10059 c1ccc(cc1)N2CCN(CC2)C(=O)Nc3ccc(cc3)F MS-10060 Cc1ccc(cc1F)NC(=O)N2CCN(CC2)c3ccccc3 MS-10061 CCOC(=O)N1CCN(CC1)C(=O)c2c(cccc2F)F MS-10062 c1ccc(cc1)CN2CCN(CC2)C(=O)c3c(cccc3F)F MS-10063 CCOC(=O)N1CCN(CC1)C(=O)C2CCCCC2 MS-10064 C1CCC(CC1)C(=O)N2CCN(CC2)C=O MS-10065 c1ccc(cc1)CN2CCN(CC2)C(=O)c3ccc(cc3)F MS-10066 c1ccc(cc1)CN2CCN(CC2)C(=O)c3ccccc3[N+](=O)[O-] MS-10067 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NC2CC2 MS-10068 c1ccc(cc1)CCNS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10069 COc1ccc(cn1)NS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10070 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10071 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NCc2ccncc2 MS-10072 c1ccc(cc1)Oc2ccc(cc2)NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10073 CN(C)CCNS(=O)(=O)c1ccc(cc1[N+](=O)[O-])Cl MS-10074 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NCCN2CCOCC2 MS-10075 c1cc2c(cc1NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl)OCO2 MS-10076 c1ccc(cc1)NS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10077 c1ccc(cc1)CNS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10078 CCOC(=O)c1cccc(c1)NC=C2C(=O)c3ccccc3C2=O MS-10079 c1cc(ccc1NS(=O)(=O)c2cc(c(cc2Cl)Cl)C(=O)O)F MS-1008 c1ccc(c(c1)C(=O)/C(=C/Nc2ncccn2)/C#N)Cl MS-10080 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NC2CCCCC2 MS-10081 c1cc(sc1)CNS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10082 c1ccc(cc1)CCN2C(Nc3ccccc3S2(=O)=O)c4ccc(cc4)Cl MS-10083 COc1ccc(cc1)C2Nc3ccccc3S(=O)(=O)N2CCc4ccccc4 MS-10084 c1ccc(cc1)N2CCN(CC2)C(=O)c3cc4ccccc4[nH]3 MS-10085 c1ccc2c(c1)cc([nH]2)C(=O)N3CCN(CC3)c4ccccc4F MS-10086 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cc4ccccc4[nH]3 MS-10087 c1ccc2c(c1)cc([nH]2)C(=O)N3CCN(CC3)C=O MS-10088 CCOC(=O)N1CCN(CC1)C(=O)c2cc3ccccc3[nH]2 MS-10089 Cc1ccc(cc1N2CCN(CC2)C(=O)c3cc4ccccc4[nH]3)Cl MS-10090 c1ccc2c(c1)cc([nH]2)C(=O)N3CCN(CC3)c4ccccn4 MS-10091 CN1CCN(CC1)C(=O)c2cc3ccccc3[nH]2 MS-10092 c1ccc2c(c1)cc([nH]2)C(=O)N3CCN(CC3)c4ncccn4 MS-10093 c1ccc2c(c1)cc([nH]2)C(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 MS-10094 c1ccc(cc1)Cn2c3ccccc3cc2C(=O)N4CCN(CC4)c5ccccc5F MS-10095 CCOC(=O)N1CCN(CC1)C(=O)c2cc3ccccc3n2Cc4ccccn4 MS-10096 CN1CCN(CC1)C(=O)c2cc3ccccc3n2Cc4ccccc4 MS-10097 CN(C)CCNC(=S)Nc1ccc(cc1)[N+](=O)[O-] MS-10098 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ccccc4 MS-10099 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)C4(CCCC4)c5ccccc5 MS-10100 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)C3(CCCC3)c4ccccc4 MS-10101 c1ccc(cc1)CN2CCN(CC2)C(=O)C3(CCCC3)c4ccccc4 MS-10102 CCOC(=O)N1CCN(CC1)C(=O)C2(CCCC2)c3ccccc3 MS-10103 Cc1ccc(cc1N2CCN(CC2)C(=O)C3(CCCC3)c4ccccc4)Cl MS-10104 CN1CCN(CC1)C(=O)C2(CCCC2)c3ccccc3 MS-10105 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ncccn4 MS-10106 CC(=O)c1cccc(c1)NC(=O)C2(CCCC2)c3ccccc3 MS-10107 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)Nc4ccccc4 MS-10108 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(cc(c3)F)C(F)(F)F MS-10109 c1ccc(cc1)NC(=O)c2nccn2Cc3ccc(cc3)C#N MS-1011 c1ccc(cc1)CCNC(=O)C2(CCCC2)c3ccccc3 MS-10110 C#CCNC(=O)C1(CCCC1)c2ccccc2 MS-10111 Cc1cc(nc(n1)NC(=O)C2(CCCC2)c3ccccc3)C MS-10112 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3C#N MS-10113 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)C3(CCCC3)c4ccccc4 MS-10114 COc1ccc(cn1)NC(=O)C2(CCCC2)c3ccccc3 MS-10115 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)OC(F)(F)F MS-10116 c1ccc(cc1)C2(CCCC2)C(=O)Nc3nccs3 MS-10117 c1ccc(cc1)C2(CCCC2)C(=O)NCc3ccncc3 MS-10118 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)Br MS-10119 CSC(=S)NCc1ccc(cc1)Cl MS-1012 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)Br MS-10120 C=CCNC(=O)C1(CCCC1)c2ccccc2 MS-10121 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3Cl MS-10122 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)Cl MS-10123 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)Cl MS-10124 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3[N+](=O)[O-])Cl MS-10125 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(ccc3F)C(F)(F)F MS-10126 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3Cl)Cl MS-10127 Cc1cccc(c1NC(=O)C2(CCCC2)c3ccccc3)C MS-10128 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(c(c3)Cl)Cl MS-10129 CCOC(=O)C1CN(C1)S(=O)(=O)c2ccccc2 MS-1013 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3F MS-10130 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)F MS-10131 CC(C)c1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10132 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc4c(c3)OCO4 MS-10133 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-10134 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)Oc4ccccc4 MS-10135 CCOc1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10136 c1ccc(cc1)COc2cccnc2NC(=O)C3(CCCC3)c4ccccc4 MS-10137 CS(=O)(=O)c1ccc2c(c1)sc(n2)NC(=O)C3(CCCC3)c4ccccc4 MS-10138 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(ccc3Cl)[N+](=O)[O-] MS-10139 COc1ccc(cc1OC)NC(=O)C2(CCCC2)c3ccccc3 MS-10140 COc1ccc(c(c1)NC(=O)C2(CCCC2)c3ccccc3)OC MS-10141 Cc1ccc(c(c1)C)NC(=O)C2(CCCC2)c3ccccc3 MS-10142 COc1ccc(cc1OC)CCNC(=O)C2(CCCC2)c3ccccc3 MS-10143 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3F)F MS-10144 CN(C)CCNC(=O)C1(CCCC1)c2ccccc2 MS-10145 COc1cc(c(cc1OC)NC(=O)C2(CCCC2)c3ccccc3)C(=O)OC MS-10146 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccncc3 MS-10147 COc1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10148 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3 MS-10149 c1ccc(cc1)NC(=O)c2nccn2Cc3ccc(cc3)F MS-1015 c1ccc(cc1)C2(CCCC2)C(=O)NCc3ccc(cc3)F MS-10150 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)F MS-10151 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3OC(F)(F)F MS-10152 c1ccc(cc1)C2(CCCC2)C(=O)Nc3c(cc(cc3Br)F)F MS-10153 CCOC(=O)c1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10154 CN(C)c1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10155 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3C(F)(F)F)F MS-10156 Cc1cc(no1)NC(=O)C2(CCCC2)c3ccccc3 MS-10157 CSc1[nH]nc(n1)NC(=O)C2(CCCC2)c3ccccc3 MS-10158 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(cc(c3)Cl)Cl MS-10159 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(c(c3)C(F)(F)F)F MS-10160 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3Br MS-10161 COc1ccc(cc1NC(=O)C2(CCCC2)c3ccccc3)[N+](=O)[O-] MS-10162 COC(=O)c1ccccc1NC(=O)C2(CCCC2)c3ccccc3 MS-10163 CC(=O)c1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10164 c1ccc(cc1)C2(CCCC2)C(=O)NCCN3CCOCC3 MS-10165 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl MS-10166 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)C#N MS-10167 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3[N+](=O)[O-] MS-10168 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(ccc3Cl)C(F)(F)F MS-10169 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3O MS-10170 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)O MS-10171 c1ccc(cc1)C2(CCCC2)C(=O)Nc3nc4ccccc4s3 MS-10172 c1ccc(cc1)C2(CCCC2)C(=O)Nc3csnn3 MS-10173 c1ccc(cc1)C2(CCCC2)C(=O)Nc3n[nH]nn3 MS-10174 c1ccc(cc1)C2(CCCC2)C(=O)Nc3[nH]ncn3 MS-10175 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)C(F)(F)F MS-10176 c1ccc(cc1)C2(CCCC2)C(=O)NCc3cccnc3 MS-10177 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cn3)C(F)(F)F MS-10178 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)CC#N MS-10179 CCOC(=O)C1CN(C1)S(=O)(=O)c2ccc(cc2)F MS-1018 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(cc(c3)F)F MS-10180 c1ccc(cc1)CNC(=O)C2(CCCC2)c3ccccc3 MS-10181 CCCCNC(=O)C1(CCCC1)c2ccccc2 MS-10182 COc1ccc(c(c1)[N+](=O)[O-])NC(=O)C2(CCCC2)c3ccccc3 MS-10183 CSc1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10184 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)[N+](=O)[O-] MS-10185 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)[N+](=O)[O-] MS-10186 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3C(F)(F)F MS-10187 c1ccc(cc1)C2(CCCC2)C(=O)NCc3cccc(c3)OC(F)(F)F MS-10188 COc1ccc(cc1OC)CNC(=O)C2(CCCC2)c3ccccc3 MS-10189 CCOC(=O)C1CN(C1)S(=O)(=O)c2ccc(cc2)C MS-1019 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(c(c3)C(F)(F)F)[N+](=O)[O-] MS-10190 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)C(F)(F)F MS-10191 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cn3)[N+](=O)[O-] MS-10192 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ncc(s3)[N+](=O)[O-] MS-10193 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)C#N MS-10194 c1ccc(cc1)C2(CCCC2)C(=O)Nc3c(c[nH]n3)Br MS-10195 Cc1cc(ccc1NC(=O)C2(CCCC2)c3ccccc3)O MS-10196 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(ccc3Br)C(F)(F)F MS-10197 c1ccc(cc1)C2(CCCC2)C(=O)NC3CCCCC3 MS-10198 Cc1cccc(c1NC(=O)C2(CCCC2)c3ccccc3)Cl MS-10199 CCOC(=O)C1CN(C1)S(=O)(=O)c2cc(ccc2OC)OC MS-1020 c1ccc(cc1)C2=N/C(=C\c3cc4c(cc3[N+](=O)[O-])OCO4)/C(=O)O2 MS-10200 c1ccc(cc1)C(CCNC(=O)C2(CCCC2)c3ccccc3)c4ccccc4 MS-10201 c1ccc(cc1)COc2ccc(cc2)NC(=O)C3(CCCC3)c4ccccc4 MS-10202 c1ccc(cc1)C(c2ccccc2)NC(=O)C3(CCCC3)c4ccccc4 MS-10203 c1ccc(cc1)C(=O)c2ccccc2NC(=O)C3(CCCC3)c4ccccc4 MS-10204 c1ccc(cc1)C(=O)c2ccc(cc2)NC(=O)C3(CCCC3)c4ccccc4 MS-10205 c1ccc(cc1)C(=O)c2cccc(c2)NC(=O)C3(CCCC3)c4ccccc4 MS-10206 CC(C)c1cccc(c1NC(=O)C2(CCCC2)c3ccccc3)C(C)C MS-10207 c1ccc(cc1)CN2CCC(CC2)NC(=O)C3(CCCC3)c4ccccc4 MS-10208 c1ccc(cc1)C2(CCCC2)C(=O)Nc3c(cc(cc3Br)C4CCCCC4)Br MS-10209 CC(c1cccc2c1cccc2)NC(=O)C3(CCCC3)c4ccccc4 MS-10210 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3Oc4ccccc4 MS-10211 c1ccc(cc1)C2(CCCC2)C(=O)NCc3cccc4c3cccc4 MS-10212 c1ccc(cc1)C2(CCCC2)C(=O)NC34CC5CC(C3)CC(C5)C4 MS-10213 CCCCc1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10214 CC(C)(C)c1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10215 c1ccc(cc1)CCCCNC(=O)C2(CCCC2)c3ccccc3 MS-10216 CCC(C)c1ccccc1NC(=O)C2(CCCC2)c3ccccc3 MS-10217 c1ccc(cc1)C2(CCCC2)C(=O)NC3CCCc4c3cccc4 MS-10218 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccccc3N4CCOCC4 MS-10219 CSC(=S)NCc1ccc(cc1)F MS-1022 CC(=O)c1cc(c(cc1NC(=O)C2(CCCC2)c3ccccc3)OC)OC MS-10220 CCCOC(=O)c1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10221 Cc1cc(c2ccccc2n1)NC(=O)C3(CCCC3)c4ccccc4 MS-10222 COc1cc(cc(c1OC)OC)NC(=O)C2(CCCC2)c3ccccc3 MS-10223 COc1ccc(cc1)CCNC(=O)C2(CCCC2)c3ccccc3 MS-10224 CCc1cccc(c1NC(=O)C2(CCCC2)c3ccccc3)C MS-10225 c1ccc(cc1)CCCNC(=O)C2(CCCC2)c3ccccc3 MS-10226 Cc1cc(c(c(c1)C)NC(=O)C2(CCCC2)c3ccccc3)C MS-10227 CC(C)c1ccccc1NC(=O)C2(CCCC2)c3ccccc3 MS-10228 CCOC(=O)c1cccc(c1)NC(=O)C2(CCCC2)c3ccccc3 MS-10229 CCCCc1n[nH]c(=S)n1Cc2ccc(cc2)Cl MS-1023 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc4c(c3)CCC4 MS-10230 Cc1cc(no1)NS(=O)(=O)c2cc(c(cc2CC(=O)OC)OC)OC MS-10231 c1ccc(cc1)C2(CCCC2)C(=O)NC3CCCCCCC3 MS-10232 CCOC(=O)N1CCC(CC1)NC(=O)C2(CCCC2)c3ccccc3 MS-10233 COc1ccccc1CNC(=O)C2(CCCC2)c3ccccc3 MS-10234 COc1cccc(c1)CNC(=O)C2(CCCC2)c3ccccc3 MS-10235 COc1ccc(cc1)CNC(=O)C2(CCCC2)c3ccccc3 MS-10236 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3)CCO MS-10237 CC(c1ccccc1)NC(=O)C2(CCCC2)c3ccccc3 MS-10238 Cc1ccc(c(c1)NC(=O)C2(CCCC2)c3ccccc3)C MS-10239 CCc1cc(ccc1NC(=O)C2(CCCC2)c3ccccc3)Br MS-10240 COC(=O)c1cc(ccc1NC(=O)C2(CCCC2)c3ccccc3)Br MS-10241 c1ccc(cc1)C2(CCCC2)C(=O)NCc3cccc(c3)C(F)(F)F MS-10242 c1ccc(cc1)C2(CCCC2)C(=O)NCc3ccccc3C(F)(F)F MS-10243 c1ccc(cc1)C2(CCCC2)C(=O)NCCCN3CCOCC3 MS-10244 c1ccc(cc1)C2(CCCC2)C(=O)NCCN3CCCCC3 MS-10245 c1ccc(cc1)C2(CCCC2)C(=O)NC3CCCCCC3 MS-10246 CC(C)(C)c1cc(no1)NC(=O)C2(CCCC2)c3ccccc3 MS-10247 c1ccc(cc1)C2(CCCC2)C(=O)NCc3ccc(cc3)Br MS-10248 c1ccc(cc1)C2(CCCC2)C(=O)NCc3cccc(c3)Br MS-10249 CCC1CCCCN1C(=O)C[n+]2ccccc2.[Cl-] MS-1025 Cc1ccc(cc1Br)NC(=O)C2(CCCC2)c3ccccc3 MS-10250 COc1ccc(cc1NC(=O)C2(CCCC2)c3ccccc3)Cl MS-10251 Cc1ccc(cc1NC(=O)C2(CCCC2)c3ccccc3)Cl MS-10252 Cc1c(cccc1F)NC(=O)C2(CCCC2)c3ccccc3 MS-10253 Cc1ccc(c(c1)NC(=O)C2(CCCC2)c3ccccc3)F MS-10254 COc1cc(ccc1NC(=O)C2(CCCC2)c3ccccc3)[N+](=O)[O-] MS-10255 Cc1c(cccc1[N+](=O)[O-])NC(=O)C2(CCCC2)c3ccccc3 MS-10256 Cc1cccc(c1NC(=O)C2(CCCC2)c3ccccc3)[N+](=O)[O-] MS-10257 Cc1cc(ccc1[N+](=O)[O-])NC(=O)C2(CCCC2)c3ccccc3 MS-10258 Cc1cc(cc(c1NC(=O)C2(CCCC2)c3ccccc3)Cl)Cl MS-10259 CCOC(=O)C1CN(C1)S(=O)(=O)c2cc(ccc2[N+](=O)[O-])Cl MS-1026 Cc1ccc(c(c1Cl)NC(=O)C2(CCCC2)c3ccccc3)Cl MS-10260 c1ccc(cc1)C2(CCCC2)C(=O)Nc3[nH]c4ccccc4n3 MS-10261 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3C(F)(F)F)Cl MS-10262 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(c(c3)Cl)C#N MS-10263 c1ccc(cc1)C2(CCCC2)C(=O)Nc3nc4ccc(cc4s3)[N+](=O)[O-] MS-10264 Cc1ccnc(c1)NC(=O)C2(CCCC2)c3ccccc3 MS-10265 Cc1cccnc1NC(=O)C2(CCCC2)c3ccccc3 MS-10266 c1ccc(cc1)C2(CCCC2)C(=O)NCc3ccccn3 MS-10267 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(ccc3O)[N+](=O)[O-] MS-10268 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(c(c(c3)Br)O)Br MS-10269 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(c(c(c3)Cl)O)Cl MS-10270 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3Cl)F MS-10271 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3F)Cl MS-10272 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3Cl)[N+](=O)[O-] MS-10273 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(ccc3F)F MS-10274 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(c(c3)F)F MS-10275 c1ccc(cc1)C2(CCCC2)C(=O)Nc3c(cccc3F)F MS-10276 CC(C)CCNC(=O)C1(CCCC1)c2ccccc2 MS-10277 CCC(CC)NC(=O)C1(CCCC1)c2ccccc2 MS-10278 CCCCCNC(=O)C1(CCCC1)c2ccccc2 MS-10279 c1cc(ccc1Cn2c(n[nH]c2=S)C(F)(F)F)F MS-1028 CCCC(C)NC(=O)C1(CCCC1)c2ccccc2 MS-10280 c1ccc(cc1)C2(CCCC2)C(=O)NC3CCCC3 MS-10281 c1ccc(cc1)C2(CCCC2)C(=O)Nc3c(cccn3)[N+](=O)[O-] MS-10282 Cc1cnc(s1)NC(=O)C2(CCCC2)c3ccccc3 MS-10283 Cc1csc(n1)NC(=O)C2(CCCC2)c3ccccc3 MS-10284 c1ccc(cc1)C2(CCCC2)C(=O)NC3=NCCS3 MS-10285 Cc1ccc(cc1)N2CCN(CC2)C(=O)C3(CCCC3)c4ccccc4 MS-10286 Cc1cccc(c1)N2CCN(CC2)C(=O)C3(CCCC3)c4ccccc4 MS-10287 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ccccc4Cl MS-10288 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4cccc(c4)Cl MS-10289 Cc1ccc(cc1)Cn2ccnc2C(=O)Nc3ccccc3 MS-1029 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ccc(cc4)Cl MS-10290 Cc1ccccc1N2CCN(CC2)C(=O)C3(CCCC3)c4ccccc4 MS-10291 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ccc(c(c4)Cl)Cl MS-10292 CCCN1CCN(CC1)C(=O)C2(CCCC2)c3ccccc3 MS-10293 CC(=O)c1cccc(c1)n2c(cc3c2CC(CC3=O)(C)C)c4cccc(c4)Br MS-10294 CC1(Cc2c(cc(n2c3cc(c(c(c3)Cl)O)Cl)c4cccc(c4)Br)C(=O)C1)C MS-10295 CC1(Cc2c(cc(n2c3cccc(c3)Cl)c4cccc(c4)Br)C(=O)C1)C MS-10296 CC1(Cc2c(cc(n2c3cc(cc(c3)F)F)c4cccc(c4)Br)C(=O)C1)C MS-10297 CC(C)c1ccc(cc1)n2c(cc3c2CC(CC3=O)(C)C)c4cccc(c4)Br MS-10298 CC1(Cc2c(cc(n2c3ccc(c(c3)Cl)Cl)c4cccc(c4)Br)C(=O)C1)C MS-10299 Cc1ccc(cc1)CNC(=S)SC MS-1030 CC1(Cc2c(cc(n2c3ccc(c(c3)OC)OC)c4cccc(c4)Br)C(=O)C1)C MS-10300 CC1(Cc2c(cc(n2c3ccc(c(c3)F)F)c4cccc(c4)Br)C(=O)C1)C MS-10301 CC1(Cc2c(cc(n2c3ccc(cc3)C(=O)c4ccccc4)c5cccc(c5)Br)C(=O)C1)C MS-10302 CC1(Cc2c(cc(n2c3ccc(c(c3)[N+](=O)[O-])Cl)c4cccc(c4)Br)C(=O)C1)C MS-10303 CC1(Cc2c(cc(n2c3cccc(c3)[N+](=O)[O-])c4cccc(c4)Br)C(=O)C1)C MS-10304 CC(=O)c1cccc(c1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10305 CCOC(=O)c1cccc(c1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10306 c1ccc(cc1)C2Cc3c(cc(n3c4cccc(c4)Cl)c5ccc(cc5)Br)C(=O)C2 MS-10307 c1ccc(cc1)C2Cc3c(cc(n3c4cc(cc(c4)F)F)c5ccc(cc5)Br)C(=O)C2 MS-10308 c1ccc(cc1)C2Cc3c(cc(n3c4cccc(c4)F)c5ccc(cc5)Br)C(=O)C2 MS-10309 c1ccc(cc1)Cn2c(n[nH]c2=S)C(F)(F)F MS-1031 CC(C)c1ccc(cc1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10310 CCOc1ccc(cc1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10311 CCN(CC)c1ccc(cc1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10312 COc1ccc(cc1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10313 c1ccc(cc1)C2Cc3c(cc(n3c4ccc(c(c4)F)F)c5ccc(cc5)Br)C(=O)C2 MS-10314 c1ccc(cc1)C2Cc3c(cc(n3c4cccc(c4)C(=O)c5ccccc5)c6ccc(cc6)Br)C(=O)C2 MS-10315 c1ccc(cc1)C2Cc3c(cc(n3c4ccc5c(c4)CCC5)c6ccc(cc6)Br)C(=O)C2 MS-10316 c1ccc(cc1)C2Cc3c(cc(n3c4ccc(cc4)CCO)c5ccc(cc5)Br)C(=O)C2 MS-10317 c1ccc(cc1)C2Cc3c(cc(n3c4ccc5c(c4)OCCO5)c6ccc(cc6)Br)C(=O)C2 MS-10318 CSc1ccc(cc1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10319 CC(=O)c1ccc(cc1)n2c(cc3c2CC(CC3=O)c4ccccc4)c5ccc(cc5)Br MS-10320 c1ccc(cc1)C2Cc3c(cc(n3c4cccc(c4)O)c5ccc(cc5)Br)C(=O)C2 MS-10321 Cc1cc2c(n1c3ccc(nc3)OC)CC(CC2=O)C MS-10322 Cc1cc2c(n1c3cc(cc(c3)F)F)CC(CC2=O)C MS-10323 Cc1cc2c(n1c3ccc(c(c3)Cl)Cl)CC(CC2=O)C MS-10324 Cc1cc2c(n1c3cccc(c3)F)CC(CC2=O)C MS-10325 Cc1cc2c(n1c3ccc(cc3)C(C)C)CC(CC2=O)C MS-10326 Cc1cc2c(n1c3ccc4c(c3)OCO4)CC(CC2=O)C MS-10327 Cc1cc2c(n1c3ccc(c(c3)OC)OC)CC(CC2=O)C MS-10328 Cc1cc2c(n1c3ccc(cc3)OC)CC(CC2=O)C MS-10329 Cc1cc2c(n1c3ccc(c(c3)F)F)CC(CC2=O)C MS-10330 Cc1cc2c(n1c3cc(cc(c3)Cl)Cl)CC(CC2=O)C MS-10331 Cc1cc2c(n1c3cccc(c3)[N+](=O)[O-])CC(CC2=O)C MS-10332 Cc1ccc(cc1)c2cc3c(n2c4ccc5c(c4)OCO5)CC(CC3=O)C MS-10333 Cc1ccc(cc1)c2cc3c(n2c4ccc(c(c4)OC)OC)CC(CC3=O)C MS-10334 Cc1ccc(cc1)c2cc3c(n2c4ccc(cc4)OC)CC(CC3=O)C MS-10335 CC1Cc2c(cc(n2c3cccc(c3)C(=O)C)c4ccc(cc4)Br)C(=O)C1 MS-10336 CC1Cc2c(cc(n2c3ccc(nc3)OC)c4ccc(cc4)Br)C(=O)C1 MS-10337 CC1Cc2c(cc(n2c3cccc(c3)Cl)c4ccc(cc4)Br)C(=O)C1 MS-10338 CC1Cc2c(cc(n2c3cc(cc(c3)F)F)c4ccc(cc4)Br)C(=O)C1 MS-10339 CC1Cc2c(cc(n2c3ccc(c(c3)Cl)Cl)c4ccc(cc4)Br)C(=O)C1 MS-10340 CC1Cc2c(cc(n2c3cccc(c3)F)c4ccc(cc4)Br)C(=O)C1 MS-10341 CC1Cc2c(cc(n2c3ccc(cc3)C(C)C)c4ccc(cc4)Br)C(=O)C1 MS-10342 CC1Cc2c(cc(n2c3ccc4c(c3)OCO4)c5ccc(cc5)Br)C(=O)C1 MS-10343 CC1Cc2c(cc(n2c3ccc(c(c3)OC)OC)c4ccc(cc4)Br)C(=O)C1 MS-10344 CC1Cc2c(cc(n2c3ccc(cc3)OC)c4ccc(cc4)Br)C(=O)C1 MS-10345 CC1Cc2c(cc(n2c3ccc(c(c3)F)F)c4ccc(cc4)Br)C(=O)C1 MS-10346 CC1Cc2c(cc(n2c3cc(cc(c3)Cl)Cl)c4ccc(cc4)Br)C(=O)C1 MS-10347 CC1Cc2c(cc(n2c3ccc(c(c3)[N+](=O)[O-])Cl)c4ccc(cc4)Br)C(=O)C1 MS-10348 CC1Cc2c(cc(n2c3cccc(c3)[N+](=O)[O-])c4ccc(cc4)Br)C(=O)C1 MS-10349 c1ccc2c(c1)C(=O)C(=O)N2S(=O)(=O)c3ccc(cc3)F MS-1035 Cc1cc2c(n1c3cccc(c3)C(=O)C)CC(CC2=O)(C)C MS-10350 Cc1cc2c(n1c3ccc(c(c3)Cl)Cl)CC(CC2=O)(C)C MS-10351 Cc1cc2c(n1c3ccc(cc3)C(C)C)CC(CC2=O)(C)C MS-10352 Cc1cc2c(n1c3ccc(cc3)C(=O)c4ccccc4)CC(CC2=O)(C)C MS-10353 Cc1cc2c(n1c3cc(cc(c3)Cl)Cl)CC(CC2=O)(C)C MS-10354 Cc1cc2c(n1c3ccc(cc3)C(=O)C)CC(CC2=O)(C)C MS-10355 Cc1cc2c(n1c3ccc(c(c3)[N+](=O)[O-])Cl)CC(CC2=O)(C)C MS-10356 Cc1cc2c(n1c3ccc(cc3)C#N)CC(CC2=O)(C)C MS-10357 Cc1cc2c(n1c3cccc(c3)[N+](=O)[O-])CC(CC2=O)(C)C MS-10358 c1cc(ccc1C2Nc3cc(c(cc3S(=O)(=O)N2)S(=O)(=O)N)F)Cl MS-10359 C#CCn1c(=O)c2ccccc2[nH]c1=S MS-10360 CCC1Nc2cc(c(cc2S(=O)(=O)N1)S(=O)(=O)N)Cl MS-10361 COC(=O)c1ccccc1NC(=S)NCCc2c[nH]c3c2cccc3 MS-10362 C#CCNC(=S)NC(=O)c1cccs1 MS-10363 c1cc(sc1)C(=O)NC(=S)NNC(=O)c2cccs2 MS-10364 c1ccc2c(c1)c(c[nH]2)CCNC(=S)NC(=O)c3cccs3 MS-10365 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)Nc2ncccn2 MS-10366 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)NCCc2c[nH]c3c2cccc3 MS-10367 c1ccc2cc(ccc2c1)S(=O)(=O)NCc3cccnc3 MS-10368 CN1CCN(CC1)S(=O)(=O)c2ccc3ccccc3c2 MS-10369 CCCCc1n[nH]c(=S)n1Cc2ccc(cc2)F MS-1037 c1ccc(cc1)COc2cccnc2NC(=O)/C=C/c3ccccc3 MS-10370 c1ccc(cc1)COc2cccnc2NS(=O)(=O)c3ccc(cc3)OC(F)(F)F MS-10371 CC1(CC(=C(C(=O)C1)C(c2cccc(c2)Cl)C3=C(CC(CC3=O)(C)C)O)O)C MS-10372 CC1(CC(=C(C(=O)C1)C(c2ccc(cc2)F)C3=C(CC(CC3=O)(C)C)O)O)C MS-10373 CC1(CC(=C(C(=O)C1)C(c2cccnc2)C3=C(CC(CC3=O)(C)C)O)O)C MS-10374 CC1(OC(=O)C(=Cc2ccc(cc2)F)C(=O)O1)C MS-10375 CC1(OC(=O)C(=Cc2ccccc2[N+](=O)[O-])C(=O)O1)C MS-10376 c1ccc(cc1)S(=O)(=O)/C(=C/c2c(cccc2Cl)F)/C#N MS-10377 Cc1ccc(cc1N2CCN(CC2)C(=O)c3ccccc3CC(=O)O)Cl MS-10378 CC(C)c1ccc(cc1)NC(=O)c2ccccc2CC(=O)O MS-10379 CN1CC(=O)Nc2ccccc2C1=O MS-1038 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3c(cccn3)OCc4ccccc4 MS-10380 c1ccc(cc1)COc2cccnc2NC(=O)C3CC3 MS-10381 c1ccc(cc1)COc2cccnc2NC(=O)C(c3ccccc3)c4ccccc4 MS-10382 c1ccc(cc1)COc2cccnc2NC(=O)COc3ccccc3 MS-10383 c1ccc(cc1)COc2cccnc2NC(=O)Cc3cccs3 MS-10384 COCC(=O)Nc1c(cccn1)OCc2ccccc2 MS-10385 CN(C)c1ccc(cc1)C(=O)Nc2c(cccn2)OCc3ccccc3 MS-10386 COc1ccccc1C(=O)Nc2c(cccn2)OCc3ccccc3 MS-10387 c1ccc(cc1)COc2cccnc2NC(=O)/C=C/c3ccccc3Cl MS-10388 c1ccc(cc1)COc2cccnc2NC(=O)COc3ccc(cc3)Cl MS-10389 c1ccc(cc1)COc2cccnc2NC(=O)c3ccc4ccccc4c3 MS-10390 c1ccc(cc1)COc2cccnc2NC(=O)C3CCC3 MS-10391 c1ccc(cc1)COc2cccnc2NC(=O)c3cccc4c3cccc4 MS-10392 c1ccc(cc1)COc2cccnc2NC(=O)C34CC5CC(C3)CC(C5)C4 MS-10393 c1ccc(cc1)COc2cccnc2NC(=O)c3ccc(cc3)c4ccccc4 MS-10394 Cc1cc(ccc1Oc2c(cccn2)C(=O)NCC#C)Cl MS-10395 c1ccc(cc1)COc2cccnc2NS(=O)(=O)c3ccc4ccccc4c3 MS-10396 CC1(C2CCC1(C(=O)C2)S(=O)(=O)Nc3c(cccn3)OCc4ccccc4)C MS-10397 c1ccc(cc1)COc2cccnc2NS(=O)(=O)c3ccc(cc3)Cl MS-10398 COc1ccc(cc1)CNC(=O)Nc2c(cccn2)OCc3ccccc3 MS-10399 CCCCc1n[nH]c(=S)n1Cc2ccc(cc2)C MS-1040 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3c(cccn3)OCc4ccccc4 MS-10400 c1ccc(cc1)COc2cccnc2NC(=O)Nc3cccc(c3)Oc4ccccc4 MS-10401 c1ccc(cc1)COc2cccnc2NC(=O)Nc3ccc4c(c3)-c5ccccc5C4 MS-10402 c1ccc(cc1)COc2cccnc2NC(=O)Nc3ccc(cc3)[N+](=O)[O-] MS-10403 c1ccc(cc1)COc2cccnc2NC(=O)Nc3cccc(c3)Cl MS-10404 c1ccc(cc1)COc2cccnc2NC(=O)NC3CCCCC3 MS-10405 CC(C(=O)N1CCN(CC1)c2ccccc2)Sc3ccc(cc3)Cl MS-10406 c1ccc(cc1)COc2cccnc2NC(=O)Nc3cccc(c3)C#N MS-10407 CC(C(=O)NCC#C)Sc1ccc(cc1)Cl MS-10408 c1ccc(cc1)COc2cccnc2NC(=O)Nc3cccc4c3cccc4 MS-10409 CCOC(=O)/C=C(\C)/c1ccc(cc1)F MS-1041 CC(C(=O)N1CCN(CC1)c2ccccc2F)Sc3ccc(cc3)Cl MS-10410 c1ccc(cc1)CNC(=O)Nc2c(cccn2)OCc3ccccc3 MS-10411 c1ccc(cc1)COc2cccnc2NC(=O)Nc3ccc4c(c3)CCC4 MS-10412 c1ccc(cc1)COc2cccnc2NC(=O)Nc3ccccc3c4ccccc4 MS-10413 c1ccc(cc1)CCCCNS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10414 c1ccc2c(c1)cccc2CNS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10415 c1ccc(cc1)CCCNS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10416 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NC2CCCCCCC2 MS-10417 Cc1cccnc1NS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10418 c1ccc(cc1)COc2cccnc2NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10419 Cc1cc(c(c(c1)C)S(=O)(=O)NCC#C)C MS-10420 Cc1cc(c(c(c1)C)S(=O)(=O)NCCc2c[nH]c3c2cccc3)C MS-10421 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NCCN2CCCCC2 MS-10422 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NC2CCCCCC2 MS-10423 c1ccnc(c1)CNS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10424 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NC2CCCC2 MS-10425 c1ccc(cc1)COc2ccc(cc2)NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10426 c1ccc(cc1)C(c2ccccc2)NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10427 c1ccc(cc1)Oc2ccccc2NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10428 c1ccc2c(c1)CCCC2NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10429 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl)N3CCOCC3 MS-10430 c1cc2c(cc1NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl)CCC2 MS-10431 c1cc2c(cc1NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl)OCCO2 MS-10432 Cc1cc(c(c(c1)C)S(=O)(=O)NCC=C)C MS-10433 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)NCCCN2CCOCC2 MS-10434 c1ccc2c(c1)[nH]c(n2)NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10435 Cc1cc(c(c(c1)C)S(=O)(=O)Nc2cc(on2)C)C MS-10436 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10437 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4[N+](=O)[O-])Cl MS-10438 c1ccc(cc1)/C=C/CN2CCN(CC2)S(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10439 c1ccc2c(c1)C(=O)Nc3ccccc3N2C(=O)COc4cc(cc(c4)Cl)Cl MS-1044 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10440 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-10441 CN1CCN(CC1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl MS-10442 c1cc2c(cc1CN3CCN(CC3)S(=O)(=O)c4ccc(cc4[N+](=O)[O-])Cl)OCO2 MS-10443 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)C(=O)N3CCN(CC3)c4ccccc4OC MS-10444 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)C(=O)N3CCN(CC3)Cc4ccccc4 MS-10445 Cc1ccc(cc1N2CCN(CC2)C(=O)c3cccnc3Oc4ccc(cc4)C(C)(C)C)Cl MS-10446 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)C(=O)NCCc3c[nH]c4c3cccc4 MS-10447 c1ccc(cc1)CN2CCN(CC2)C(=O)C34CC5CC(C3)CC(C5)C4 MS-10448 c1ccc(cc1)CN2C(Nc3ccccc3S2(=O)=O)c4ccc(cc4)Cl MS-10449 CC1CN(CC(O1)C)C(=O)/C=C(/C)\c2ccc(cc2)F MS-1045 COc1ccc(cc1OC)CCNC(=O)C23CC4CC(C2)CC(C4)C3 MS-10450 COC(=O)c1c(ccs1)NC(=O)C23CC4CC(C2)CC(C4)C3 MS-10451 Cc1cc(no1)NC(=O)C23CC4CC(C2)CC(C4)C3 MS-10452 COc1ccc(cc1)C2Nc3ccccc3S(=O)(=O)N2Cc4ccccc4 MS-10453 COC(CNC(=O)C1CCCCC1C(=O)O)OC MS-10454 CC(C)CCNC(=O)C1c2ccccc2C(=O)N(C1c3cccnc3)c4ccc(cc4)OC MS-10455 COc1ccc(cc1)N2C(C(c3ccccc3C2=O)C(=O)NCc4ccncc4)c5cccnc5 MS-10456 COc1ccc(cc1)N2C(C(c3ccccc3C2=O)C(=O)NCc4cccc(c4)C(F)(F)F)c5cccnc5 MS-10457 CC(C)CCNC(=O)C1c2ccccc2C(=O)N(C1c3ccc(cc3)OC)c4ccc(cc4)OC MS-10458 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2c4ccc(cc4)OC)C(=O)NCc5ccncc5 MS-10459 c1cc(ccc1c2n[nH]c(=O)o2)OCc3ccc(cc3Cl)Cl MS-1046 CN(C)c1ccc(cc1)NC(=O)C2c3ccccc3C(=O)N(C2c4ccc(cc4)OC)c5ccc(cc5)OC MS-10460 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2c4ccc(cc4)OC)C(=O)NCc5cccc(c5)C(F)(F)F MS-10461 CC(C)CCNC(=O)C1c2ccccc2C(=O)N(C1c3ccsc3)c4ccc(cc4)OC MS-10462 COc1ccc(cc1)N2C(C(c3ccccc3C2=O)C(=O)NCc4ccncc4)c5ccsc5 MS-10463 CC(=O)/C(=C\Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C(=O)Nc2ccccc2 MS-10464 CN1CCN(CC1)C(=S)NCc2ccccc2 MS-10465 c1ccc(c(c1)N2CCN(CC2)C(=O)c3cccnc3C(=O)O)F MS-10466 CC(C)CCNC(=O)C1c2ccccc2C(=O)N(C1c3cccnc3)c4ccc5c(c4)OCO5 MS-10467 c1ccc2c(c1)C(C(N(C2=O)c3ccc4c(c3)OCO4)c5cccnc5)C(=O)NCc6ccncc6 MS-10468 CC(C)CCNC(=O)C1c2ccccc2C(=O)N(C1c3ccc(cc3)OC)c4ccc5c(c4)OCO5 MS-10469 C/C(=C/C(=O)N1CCC(CC1)c2ccccc2)/c3ccc(cc3)F MS-1047 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2c4ccc5c(c4)OCO5)C(=O)NCc6ccncc6 MS-10470 CN(C)c1ccc(cc1)NC(=O)C2c3ccccc3C(=O)N(C2c4ccc(cc4)OC)c5ccc6c(c5)OCO6 MS-10471 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2c4ccc5c(c4)OCO5)C(=O)NCc6cccc(c6)C(F)(F)F MS-10472 CC(C)CCNC(=O)C1c2ccccc2C(=O)N(C1c3ccsc3)c4ccc5c(c4)OCO5 MS-10473 c1ccc2c(c1)C(C(N(C2=O)c3ccc4c(c3)OCO4)c5ccsc5)C(=O)NCc6ccncc6 MS-10474 c1cc(ccc1NC(=O)Nc2ccc(cc2)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl MS-10475 CC(=O)/C(=C/Nc1cccc(c1)OC(C(F)F)(F)F)/C(=O)Nc2ccccc2 MS-10476 C1CN(CCN1C=O)C(=O)/C=C/C(=O)O MS-10477 C#CCNC(=O)/C=C/C(=O)O MS-10478 COc1ccc(cc1OC)CNC(=O)/C=C/C(=O)O MS-10479 COc1ccc(c(c1)OC)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 MS-10480 COc1ccc(cc1OC)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 MS-10481 CCOc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 MS-10482 CSc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 MS-10483 COc1cc(cc(c1OC)OC)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 MS-10484 c1ccc(cc1)N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4ccccc4 MS-10485 c1ccc(cc1)N2C(=O)C(=Cc3cccs3)C(=O)N(C2=O)c4ccccc4 MS-10486 COc1ccc(cc1Cl)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 MS-10487 COc1ccccc1N2C(=O)C(=Cc3cccs3)C(=O)N(C2=O)c4ccccc4OC MS-10488 COc1ccccc1N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4ccccc4OC MS-10489 c1ccc(cc1)Cn2c(=O)oc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl MS-1049 COc1ccccc1N2C(=O)C(=Cc3ccc(c(c3)OC)OC)C(=O)N(C2=O)c4ccccc4OC MS-10490 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3OC)c4ccccc4OC MS-10491 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3cccc(c3)OC)c4cccc(c4)OC MS-10492 COc1cccc(c1)N2C(=O)C(=Cc3ccc(c(c3)OC)OC)C(=O)N(C2=O)c4cccc(c4)OC MS-10493 COc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3cccc(c3)OC)c4cccc(c4)OC MS-10494 COc1cccc(c1)N2C(=O)C(=Cc3cc(c(c(c3)OC)OC)OC)C(=O)N(C2=O)c4cccc(c4)OC MS-10495 COc1cccc(c1)N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4cccc(c4)OC MS-10496 COc1cccc(c1)N2C(=O)C(=Cc3cccs3)C(=O)N(C2=O)c4cccc(c4)OC MS-10497 COc1ccc(cc1)N2C(=O)C(=Cc3cccs3)C(=O)N(C2=O)c4ccc(cc4)OC MS-10498 COc1ccc(cc1)N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4ccc(cc4)OC MS-10499 c1cc(ccc1Cn2c(=O)oc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl)C(F)(F)F MS-1050 COc1ccc(cc1)N2C(=O)C(=Cc3ccc(cc3)SC)C(=O)N(C2=O)c4ccc(cc4)OC MS-10500 COc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)OC)c4ccc(cc4)OC MS-10501 CCOc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)OC)c4ccc(cc4)OC MS-10502 COc1ccc(cc1)N2C(=O)C(=Cc3ccc(c(c3)OC)OC)C(=O)N(C2=O)c4ccc(cc4)OC MS-10503 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)OC)c4ccc(cc4)OC MS-10504 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)c3ccccn3)C MS-10505 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3Cl)c4ccccc4Cl MS-10506 c1cc(cc(c1)Cl)N2C(=O)C(=Cc3cccs3)C(=O)N(C2=O)c4cccc(c4)Cl MS-10507 c1cc(cc(c1)Cl)N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4cccc(c4)Cl MS-10508 COc1ccc(cc1OC)C=C2C(=O)N(C(=O)N(C2=O)c3cccc(c3)Cl)c4cccc(c4)Cl MS-10509 Cc1ccc(cc1)Cn2c(=O)oc(n2)c3ccc(cc3)OCc4ccc(cc4Cl)Cl MS-1051 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3cccc(c3)Cl)c4cccc(c4)Cl MS-10510 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl MS-10511 COc1ccc(cc1OC)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl MS-10512 CCOc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl MS-10513 COc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl MS-10514 CSc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl MS-10515 c1cc(ccc1N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4ccc(cc4)Cl)Cl MS-10516 c1cc(sc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl MS-10517 Cc1cccc(c1)N2C(=O)C(=Cc3ccc(cc3)N(C)C)C(=O)N(C2=O)c4cccc(c4)C MS-10518 Cc1cccc(c1)N2C(=O)C(=Cc3ccc(cc3OC)OC)C(=O)N(C2=O)c4cccc(c4)C MS-10519 c1cc(ccc1c2nn(c(=O)o2)CCC#N)OCc3ccc(cc3Cl)Cl MS-1052 CCOc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3cccc(c3)C)c4cccc(c4)C MS-10520 Cc1cccc(c1)N2C(=O)C(=Cc3ccc(cc3)OC)C(=O)N(C2=O)c4cccc(c4)C MS-10521 Cc1cccc(c1)N2C(=O)C(=Cc3ccc(cc3)SC)C(=O)N(C2=O)c4cccc(c4)C MS-10522 Cc1cccc(c1)N2C(=O)C(=Cc3cc(c(c(c3)OC)OC)OC)C(=O)N(C2=O)c4cccc(c4)C MS-10523 Cc1cccc(c1)N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4cccc(c4)C MS-10524 Cc1cccc(c1)N2C(=O)C(=Cc3cccs3)C(=O)N(C2=O)c4cccc(c4)C MS-10525 Cc1ccc(cc1)N2C(=O)C(=Cc3ccc(cc3)NC(=O)C)C(=O)N(C2=O)c4ccc(cc4)C MS-10526 Cc1ccc(cc1)N2C(=O)C(=Cc3cccs3)C(=O)N(C2=O)c4ccc(cc4)C MS-10527 Cc1ccc(cc1)N2C(=O)C(=Cc3ccsc3)C(=O)N(C2=O)c4ccc(cc4)C MS-10528 Cc1ccc(cc1)N2C(=O)C(=Cc3ccc(cc3)SC)C(=O)N(C2=O)c4ccc(cc4)C MS-10529 Cc1ccc(cc1)CSc2nnc(n2Cc3ccc(cc3)F)C(F)(F)F MS-1053 Cc1ccc(cc1)N2C(=O)C(=Cc3ccccc3OC)C(=O)N(C2=O)c4ccc(cc4)C MS-10530 Cc1ccc(cc1)N2C(=O)C(=Cc3ccc(cc3)OC)C(=O)N(C2=O)c4ccc(cc4)C MS-10531 CCOc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccc(cc3)C)c4ccc(cc4)C MS-10532 Cc1ccc(cc1)N2C(=O)C(=Cc3ccc(c(c3)OC)OC)C(=O)N(C2=O)c4ccc(cc4)C MS-10533 Cc1ccc(cc1)N2C(=O)C(=Cc3ccc(cc3OC)OC)C(=O)N(C2=O)c4ccc(cc4)C MS-10534 Cc1ccc(cc1)N2C(=O)C(=Cc3ccc(cc3)Cl)C(=O)N(C2=O)c4ccc(cc4)C MS-10535 c1cc(ccc1c2c([nH]nn2)C#N)[N+](=O)[O-] MS-10536 c1cc(ccc1C#N)c2c([nH]nn2)C#N MS-10537 CC(=O)Nc1ccc(cc1)c2c([nH]nn2)C#N MS-10538 Cc1ccc(cc1)NC(=O)Nc2ccc(cc2)C MS-10539 c1cc(ccc1/C=C/C(=O)C(=O)O)Cl MS-1054 CCN1C(=O)/C(=C\Nc2ccc(cc2)OC)/SC1=S MS-10540 Cc1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2)C(=O)OC MS-10542 CCCCNC(=O)N1CCN(CC1)C(=O)OCC MS-10543 CCCCNC(=O)N1CCN(CC1)c2ccccc2F MS-10544 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC3CC3 MS-10545 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCc3ccccc3 MS-10546 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC(OC)OC MS-10547 COc1ccc(c(c1)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)OC MS-10548 COc1ccc(c(c1)S(=O)(=O)N2CCN(CC2)Cc3ccccc3)OC MS-10549 CC(C)(C)c1ccc(cc1)CSc2nnc(n2Cc3ccc(cc3)F)C(F)(F)F MS-1055 COc1ccc(cc1OC)CCNC(=S)NCc2cccnc2 MS-10550 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Cc4cccc5c4cccc5 MS-10551 c1ccc(cc1)CN2CCN(CC2)C(=O)Cc3cccc4c3cccc4 MS-10552 c1ccc2c(c1)cccc2CC(=O)N3CCN(CC3)c4ccccn4 MS-10553 CCOC(=O)N1CCN(CC1)C(=O)Cc2cccc3c2cccc3 MS-10554 CCOc1ccccc1/C=C/C(=O)NCCc2ccc(c(c2)OC)OC MS-10555 C=CCNC(=O)/C=C/c1ccc(c(c1)Cl)Cl MS-10556 c1ccnc(c1)N2CCN(CC2)C(=O)/C=C/c3ccc(c(c3)Cl)Cl MS-10557 Cc1ccc(cc1N2CCN(CC2)C(=O)/C=C/c3ccc(c(c3)Cl)Cl)Cl MS-10558 c1cc(c(cc1/C=C/C(=O)N2CCN(CC2)C=O)Cl)Cl MS-10559 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3cc(c(cc3CC(=O)OC)OC)OC)Cl MS-10560 Cc1cc(no1)NC(=S)NC(=O)/C=C/c2ccccc2 MS-10561 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2F)F MS-10562 Cc1cc(nc(n1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)C MS-10563 CCOC(=O)c1cccc(c1)N/C=C(\C#N)/S(=O)(=O)c2cc(ccc2Cl)Cl MS-10564 Cc1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)c3ccccc3F MS-10565 Cc1ccc(cc1)S(=O)(=O)NCC#C MS-10566 c1c(cc(c(c1F)NC(=O)C2CCCCC2)Br)F MS-10567 COc1cccc(c1)NC(=O)C2CCCCC2 MS-10568 c1ccc(cc1)C(c2ccccc2)C(=O)NCCN3CCOCC3 MS-10569 c1cc(sc1)CC(=O)Nc2cc(ccc2Cl)[N+](=O)[O-] MS-10570 c1ccc(c(c1)NC(=O)Cc2cccs2)Cl MS-10571 c1ccc(cc1)OCC(=O)Nc2cccnc2 MS-10572 Cc1cc(nc(n1)NC(=C2C(=O)c3ccccc3C2=O)C)Cl MS-10574 Cc1ccc2c(c1)CCCN2C(=O)c3ccc(cc3)[N+](=O)[O-] MS-10575 CC1Cc2c(sc(n2)NC=C3C(=O)c4ccccc4C3=O)C(=O)C1 MS-10576 c1cc(ccc1CCNC(=S)NNC(=O)c2ccncc2)Cl MS-10577 Cc1cc(ccc1N/C=C(\C#N)/C(=O)c2ccccc2)O MS-10578 Cc1cccc(c1C(=O)O)N/C=C(/C#N)\C(=O)c2ccccc2 MS-10579 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCN3CCOCC3 MS-10580 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)C MS-10581 COc1cc(c(cc1OC)Br)/C=C/C(=O)O MS-10582 c1cc(c(cc1[N+](=O)[O-])/C=C/C(=O)O)Cl MS-10584 c1cc(c(cc1/C=C/C(=O)O)[N+](=O)[O-])Cl MS-10585 c1cc(c(cc1Cl)Cl)C(=O)N MS-10586 c1cc(c(cc1Br)Br)OCC(=O)O MS-10587 Cc1cccc(c1C)OCC(=O)O MS-10588 Cc1ccc(cc1C)OCC(=O)O MS-10589 c1ccc(c(c1)/C=C/C(=O)O)F MS-10591 c1ccc(cc1)C(=O)/C=C/c2ccccc2O MS-10592 c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)O MS-10593 c1cc(cc(c1)[N+](=O)[O-])NC=O MS-10596 CC(C)(C)c1ccc(cc1)C(=O)/C=C/C(=O)O MS-10597 CC(C)c1ccc(cc1)C(=O)/C=C/C(=O)O MS-10598 c1cc(ccc1C(=O)/C=C/C(=O)O)Br MS-10599 c1ccc(cc1)CN2CC(C2)CO MS-1060 c1cc(ccc1C2CCCCC2)C(=O)/C=C/C(=O)O MS-10600 COc1cc(c(cc1OC)[N+](=O)[O-])C(=O)N MS-10601 c1ccc(cc1)CNC(=O)c2ccccc2 MS-10602 c1cc(c(cc1S(=O)(=O)NCCN2CCOCC2)[N+](=O)[O-])Cl MS-10603 Cc1ccc(c(c1)C)NC(=O)C2CCCCC2 MS-10604 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2C)C MS-10605 c1cc(ccc1NS(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl)F MS-10606 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3ccccc3)Cl MS-10607 c1cc(c(cc1S(=O)(=O)NC2CC2)[N+](=O)[O-])Cl MS-10608 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(c(c3)[N+](=O)[O-])Cl MS-10609 c1ccc(c(c1)C(F)(F)F)n2cn[nH]c2=O MS-1061 CCCCCC(=O)Nc1ccc(nc1)OC MS-10610 CCCNC(=O)NCc1ccncc1 MS-10611 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCN2CCOCC2 MS-10612 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl MS-10613 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl MS-10614 CCCCNC(=O)Nc1cccc(c1)C(=O)C MS-10615 c1ccc(cc1)N2CCN(CC2)C(=S)NC(=O)c3c(cccc3F)F MS-10616 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCCc2ccccc2 MS-10617 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccn3 MS-10618 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)I MS-10619 Cc1ccc2c(c1)CCC[N@]2S(=O)(=O)c3ccc(cc3)I MS-10620 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)I MS-10621 c1ccc(cc1)N2CCN(CC2)C(=S)NC(=O)c3ccc(cc3)I MS-10622 CCOC(=O)N1CCN(CC1)C(=S)NC(=O)c2ccc(cc2)I MS-10623 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)NCCc3ccc(c(c3)OC)OC MS-10625 CCN(c1ccccc1)C(=S)NC(=O)c2ccccc2 MS-10626 CCN(c1ccccc1)C(=S)N MS-10627 c1cc(ccc1NC(=O)N2CCN(CC2)C=O)Cl MS-10628 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)OC(F)(F)F MS-10629 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5)C MS-10630 c1c(cnc(c1Cl)NC(=N)S)C(F)(F)F MS-10631 CCOC(=O)Cc1csc(n1)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-10633 c1ccc(cc1)CC(=O)NC(=S)NC2CC2 MS-10634 c1ccc(cc1)CC(=O)NC(=S)Nc2cccc(c2)OC(F)(F)F MS-10635 c1cc(ccc1OCC(=O)NN)OC(F)(F)F MS-10636 c1ccc(cc1)CCNC(=O)Nc2ccccc2 MS-10637 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)COc3ccc4ccccc4c3Br MS-10638 CC1=C(C(NC(=S)N1)c2cccc(c2)Oc3ccccc3)C(=O)OC MS-10639 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)NCCc3ccc(cc3)Cl MS-10640 CCOC(=O)C(=CNc1cc(nc2c1cccc2)C)C(=O)OCC MS-10641 CC1=C/C(=N\NC(=S)N)/CCC1 MS-10642 C/C(=N\O)/c1cc2c(cc1NC=C3C(=O)c4ccccc4C3=O)OCO2 MS-10643 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2cc(ccc2C)C)/C#N MS-10644 c1ccc2c(c1)C(=O)C(=Cc3ccsc3)C2=O MS-10645 C=CCNC(=S)N/N=C/c1ccsc1 MS-10646 CC1(C(NC(S1)c2ccsc2)C(=O)O)C MS-10647 C=CCS/C(=[NH+]\N=C\c1ccsc1)/N.[Cl-] MS-10648 CC\1=NN(C(=O)/C1=C\c2cc3c(cc2[N+](=O)[O-])OCO3)c4ccccc4 MS-10649 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(C(CCl)Cl)Cl MS-1065 c1cc(ccc1C(F)(F)F)NC(=O)C2CC2C(=O)O MS-10650 c1ccc(cc1)NC(=O)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl MS-10651 COc1ccc(cn1)NC(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl MS-10652 Cc1ccc(cc1)c2c3c(n(n2)c4ccc(cc4)[N+](=O)[O-])-c5ccccc5C3=O MS-10653 c1cc(c(cc1/C=N/C(=C(/C#N)\N)/C#N)O)O MS-10654 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)N=Cc3ccc(c(c3)O)O MS-10655 c1ccnc(c1)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccc(cc4)Cl MS-10656 COc1ccc(cc1)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccc(cc4)Cl MS-10657 Cc1cccc(c1NC(=O)c2ccccc2CC(=O)O)Cl MS-10658 CC(C)CC1Cc2c(sc(n2)NC(=O)c3cccs3)C(=O)C1 MS-10659 c1cc(cc(c1)n2c(nnn2)Cl)C(F)(F)F MS-1066 C=CCNC(=S)NNC(=O)COc1cccc2c1cccc2 MS-10660 c1ccc2c(c1)cccc2OCC(=O)NN=C3c4cc(ccc4NC3=O)Br MS-10661 C=CCNC(=S)N/N=C(\c1cccs1)/C2C(=O)c3ccccc3C2=O MS-10662 c1ccc2c(c1)cccc2OCC(=O)N/N=C/3\c4ccccc4NC3=O MS-10663 CC(C)(C)C1=NN(C(=O)C1=CC=Cc2ccccc2)c3ccccc3 MS-10664 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN(C)C(=S)Nc3ccccc3 MS-10665 c1cc(ccc1S(=O)(=O)c2cc3cc(cc(c3oc2=O)I)I)Cl MS-10666 c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3F MS-10667 Cc1c(c(no1)c2c(cccc2Cl)Cl)C3=NCCc4c3cc(c(c4)OC)OC MS-10668 CCN1C(=O)C(=Cc2ccc(c(c2)[N+](=O)[O-])O)SC1=S MS-10669 CSC(=CC(=O)c1cccc(c1)I)SC MS-1067 CC(C)(C)C\1=NN(C(=O)/C1=C\c2ccc(c(c2)OC)OC)c3ccccc3 MS-10670 c1cc(cc(c1)Br)C(=O)O/N=C(\c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F)/N MS-10671 c1cc(cnc1)C(=O)O/N=C(\c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F)/N MS-10672 c1cc(cc(c1)Cl)C(=O)O/N=C(\c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F)/N MS-10673 COc1ccc(cc1)/C=C/C=C(/C#N)\S(=O)(=O)c2ccc(cc2Cl)Cl MS-10674 Cc1c(c(c(c(c1F)F)NNC(=O)Nc2cccc(c2)C(F)(F)F)F)F MS-10675 Cc1c(c(c(c(c1F)F)N2C(=O)CC(=N2)C(C)(C)C)F)F MS-10676 Cc1c(c(c(c(c1F)F)N2C(=O)C(=CC=Cc3ccc(cc3)OC)C(=N2)C(C)(C)C)F)F MS-10677 CCN1C(=O)C(=Cc2ccco2)SC1=S MS-10678 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-10679 c1ccc(cc1)NC(=S)NCCCNC(=S)Nc2ccccc2 MS-1068 CC1CC(=CC(=O)C1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-10680 c1ccc(cc1)C2CC3=C(C(Nc4ccccc4N3)c5ccc(cc5)F)C(=O)C2 MS-10681 CCN1C(=O)/C(=C\C=C\c2ccccc2)/SC1=S MS-10682 Cc1ccc(c(c1)C)c2csc(n2)Nc3ccccc3 MS-10683 CC(=C1C(=O)c2ccccc2C1=O)NCCN(C)C MS-10684 CC(=C1C(=O)c2ccccc2C1=O)NCc3ccc(c(c3)OC)OC MS-10685 c1cc(ccc1NC(=S)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)OC(F)(F)F MS-10686 c1cc(cnc1)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F MS-10687 c1ccc(cc1)c2csc(n2)NC=C3C(=O)c4ccccc4C3=O MS-10688 c1cc(c(cc1Cl)[N+](=O)[O-])S(=O)(=O)N MS-10689 CCN(CC)CC(=O)Nc1ccc(cc1)/C(=N/NC2=NCCN2)/C MS-1069 CC1(OC(=O)C(=CN2CCNCC2)C(=O)O1)C MS-10690 c1cc(sc1)C(=O)Nc2nc(cs2)c3ccc(cc3)Br MS-10691 CN(C(=S)Nc1ccc(cc1)Cl)N MS-10692 CN(C)c1ccc(cc1)NC(=S)N(C)N MS-10693 Cc1ccc(c2c1CC(O2)(C)C)NC(=S)N(C)N MS-10694 c1cc(ccc1NC(=S)NNC(=O)CSc2c(cc(cn2)C(F)(F)F)Cl)OC(F)(F)F MS-10695 c1ccc(cc1)C2CC(=C(C(=O)C2)I)Nc3ccccc3C(=O)O MS-10696 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)n3c(cc4c3CC(CC4=O)(C)C)C MS-10697 c1ccc(cc1)C2CC3=C(C(Nc4ccccc4N3)c5c[nH]c6c5cccc6)C(=O)C2 MS-10698 c1cc(ccc1Sc2ccc(cc2/C=N/C(=C(/C#N)\N)/C#N)[N+](=O)[O-])Cl MS-10699 C[C@@H]1CCC[C@@H](N1C(=O)NCCCN2CCOCC2)C MS-1070 Cc1cc(ccc1C(C)C)NC(=S)NNC(=O)c2ccncc2 MS-10700 Cc1cc(ccc1C(C)C)n2c(n[nH]c2=S)c3ccncc3 MS-10701 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cn3)Br MS-10702 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C(=O)C3CC3C(=O)O MS-10703 CC(C)(C)C\1=NN(C(=O)/C1=C\c2ccc(cc2Cl)Cl)c3c(cc(cn3)C(F)(F)F)Cl MS-10704 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)Cl)CCCC2 MS-10705 CC1(Cc2c(cc(n2c3ccc(cc3)Sc4ccc(cn4)C(F)(F)F)c5ccc(cc5)Br)C(=O)C1)C MS-10706 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccc(cc3)OC(F)(F)F)CCCC2 MS-10707 CC1(Cc2c(cc(n2c3ccc(cc3)Sc4c(cc(cn4)C(F)(F)F)Cl)c5ccc(cc5)Br)C(=O)C1)C MS-10708 c1cc(ccc1N/C=C(/C#N)\c2[nH]nnn2)Sc3c(cc(cn3)C(F)(F)F)Cl MS-10709 CC(C)(C)C(=O)/C(=C\Nc1ccc(cc1)Sc2c(cc(cn2)C(F)(F)F)Cl)/C#N MS-10710 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Sc3c(cc(cn3)C(F)(F)F)Cl)/[N+](=O)[O-] MS-10711 CCCC1CC(=CC(=O)C1)Nc2ccccc2C#N MS-10712 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3ccccc3C#N MS-10713 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C MS-10714 c1ccc(cc1)Cc2n[nH]c(=S)n2c3ccc(cc3)Sc4c(cc(cn4)C(F)(F)F)Cl MS-10715 c1ccc2c(c1)[nH]c(n2)Sc3c(cc(cn3)C(F)(F)F)Cl MS-10716 c1ccc2c(c1)c3c([nH]2)nc(nn3)Sc4ccc(cn4)[N+](=O)[O-] MS-10717 CN1CCN(CC1)C(=S)Nc2ccc(cc2)OC(F)(F)F MS-10718 CN1CCN(CC1)C(=O)Nc2ccc(c(c2)Cl)Cl MS-10719 c1ccc(cc1)Nc2ccc(cc2N)C(F)(F)F MS-1072 Cc1ccc(cc1)SCCC(=O)NCCc2c[nH]c3c2cccc3 MS-10720 COc1ccc(cc1OC)CNC2=CC(=O)CCC2 MS-10721 COc1ccc(c(c1)NC(=C2C(=O)c3ccccc3C2=O)C#N)OC MS-10722 CCOC(=O)c1c2c(sc1NC=C3C(=O)c4ccccc4C3=O)CCCC2 MS-10723 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=O)c3ccccc3 MS-10724 CC(C)(C)C1=NN(C(=O)C1=Cc2cc3c(cc2[N+](=O)[O-])OCO3)c4ccccc4 MS-10725 CCc1cccc2c1[nH]cc2C3CC(=NNC3=O)c4ccc(cc4)Br MS-10726 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cccc(c3)Oc4ccccc4)C(=O)C1)C MS-10727 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)SC)C(=O)C1)C MS-10728 Cc1c(c(c(c(c1F)F)NNC(=S)Nc2ccccc2)F)F MS-10729 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCc4ccccn4 MS-10730 CC(C)(C)C1=NN(C(=O)C1=Cc2ccc3c(c2)OCO3)c4ccccc4 MS-10731 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3 MS-10732 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3)Cl MS-10733 CCc1cccc2c1[nH]cc2C(CC(=O)c3ccccc3)C(=O)O MS-10734 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCOC MS-10735 CCOc1ccc(cc1)NC(=O)c2c(onc2c3ccccc3Cl)C MS-10736 Cc1c-2c(=O)c3ccccc3c2nc4ccccc4[nH]1 MS-10737 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=C3C(=O)c4ccccc4C3=O)C MS-10738 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-10739 Cc1c2ccccc2[nH]c1c3ccc(cc3)Br MS-1074 c1c(cnc(c1Cl)N2CCCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)C(F)(F)F MS-10740 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-10741 c1c(cc(c(c1Br)O)Br)/C=N/C(=C(/C#N)\N)/C#N MS-10742 Cc1cccc(c1NC(=O)C2CC2C(=O)O)C(=O)O MS-10743 c1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccccc2 MS-10744 CC(C)(C)c1ccc(cc1)S(=O)(=O)NCc2ccncc2 MS-10745 CN(C)c1ccc(cc1)C=C2C(=O)c3ccccc3C2=O MS-10746 c1cc(ccc1OC(F)(F)F)S(=O)(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-10747 CC(=O)Nc1ccc(cc1)/C=C(/C#N)\C(=O)C(C)(C)C MS-10748 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)Sc4ccccn4 MS-10749 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc(c3)C#N MS-10750 Cc1ccc(c(c1)C)NC(=O)C2(CCCCC2)C MS-10751 c1cnccc1CNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-10752 c1ccc(cc1)C(=O)/C(=C/c2cccs2)/C#N MS-10753 COc1ccc(cc1Cl)C=C2C(=O)c3ccccc3C2=O MS-10754 c1c(cnc(c1Cl)N2CCCN(CC2)C(=O)C3CC3C(=O)O)C(F)(F)F MS-10755 c1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-10756 c1cc(cnc1)CNC(=O)Nc2ccc(cc2)C(F)(F)F MS-10757 CC(=C1C(=O)c2ccccc2C1=O)NCc3cccnc3 MS-10758 CCOC(=O)/C(=C\NCc1cccnc1)/C#N MS-10759 c1ccc(c(c1)N)Nc2cccc(c2)C(F)(F)F MS-1076 COc1cc(cc(c1OC)OC)C=C(C#N)C#N MS-10760 CC1(CC2=C(C(Nc3ccccc3N2)c4cc(c(c(c4)Br)O)Br)C(=O)C1)C MS-10761 COc1ccc(cn1)NC(=O)C2CC2 MS-10762 CC(=O)c1ccc(cc1)N/C=C(/C(=O)C)\S(=O)(=O)c2ccccc2 MS-10763 C/C(=N\O)/CS(=O)(=O)c1ccc(cc1)Cl MS-10764 CC(=O)/C(=C/Nc1cc(cc(c1)Cl)Cl)/S(=O)(=O)c2ccc(cc2)Cl MS-10765 COc1cc(cc(c1OC)OC)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4cccc(c4)C(F)(F)F MS-10766 Cc1cc(nc(n1)NC=C2C(=O)c3ccccc3C2=O)C MS-10767 CC(=C1C(=O)c2ccccc2C1=O)NCc3cccs3 MS-10768 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)NCc3cccs3 MS-10769 CCOC(=O)Oc1cc(c(cc1Cl)F)[N+](=O)[O-] MS-1077 c1ccc(cc1)C2=C(c3ccccc3C2=O)NCc4cccs4 MS-10770 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3cc(c(c(c3)Br)Br)Br MS-10771 COc1ccc(cc1)c2csc(n2)Nc3ccccc3Cl MS-10772 CC(=O)Nc1ccc(cc1)c2csc(n2)Nc3cccc4c3cccc4 MS-10773 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3nccs3 MS-10774 c1ccc(cc1)NC(=S)NNC(=O)c2ccc(cc2)O MS-10775 c1ccc(cc1)NC(=S)NNC(=O)Cc2cccc(c2)Cl MS-10776 CCN1C(=O)/C(=C\c2ccc(cc2)N(C)C)/SC1=S MS-10777 CSC(=C(C#N)S(=O)(=O)c1ccc(cc1)Cl)SC MS-10778 Cc1cc(ccc1OCC(=O)NN)Cl MS-10779 c1cc(oc1)C(C#N)Nc2ccc(cc2)C(F)(F)F MS-1078 CC1=C(C(=[NH+]CCN1)C(F)(F)F)Br.[Br-] MS-10780 COC(=O)C(CC(=O)c1ccccc1)c2c[nH]c3c2cccc3 MS-10781 c1cc(ccc1[N+](=O)[O-])OCC(=O)NN MS-10782 CCOc1ccc(cc1)C(=O)CC(c2c[nH]c3c2cccc3)C(=O)O MS-10783 CCOc1ccc(cc1)C(=O)CC(c2c[nH]c3c2cccc3)C(=O)OC MS-10784 c1cc(ccc1NC=C(C#N)C#N)OC(F)(F)F MS-10785 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)OC(F)(F)F)/C#N MS-10786 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)F)/[N+](=O)[O-] MS-10787 CC(C)c1ccc(cc1)C2=NNC(=O)C(C2)c3c[nH]c4c3cccc4 MS-10788 c1cc(ccc1N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccc(cc2)Cl)OC(F)(F)F MS-10789 CC(C)c1ccc(cc1)N/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)C(C)C MS-10791 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3cccc(c3)OC(C(F)F)(F)F)C2=O MS-10792 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2F)/[N+](=O)[O-] MS-10793 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)SC(F)(F)F)/C#N MS-10794 CC(C)(C)C(=O)C(=C1Nc2ccccc2N1)C#N MS-10795 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C(\Nc2ccccc2)/SC)/C#N MS-10796 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C(/Nc2ccc(cc2)Cl)\SC)/C#N MS-10797 CC(C)(C)C(=O)/C(=C/1\Nc2ccccc2S1)/C#N MS-10798 CC(C)(C)C(=O)/C(=C/1\Nc2ccc(cc2N1)[N+](=O)[O-])/C#N MS-10799 c1ccc(cc1)C2CC(=O)C(C(=O)C2)CC(=O)c3ccccc3 MS-10800 c1ccc(c(c1)C(F)(F)F)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-10802 c1cc(ccc1OC(F)(F)F)S(=O)(=O)CC#N MS-10803 c1cc(ccc1OC(F)(F)F)S(=O)(=O)/C(=C\Nc2cc(ccc2F)C(F)(F)F)/C#N MS-10804 c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccccc2F)/[N+](=O)[O-] MS-10805 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-])Cl MS-10806 CC(C)NCCN(C(C)C)S(=O)(=O)c1ccc(cc1)OC(F)(F)F MS-10807 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)F MS-10808 CCOC(=O)C(C)C(=O)c1ccc(cc1)C(=O)C(C)C(=O)OCC MS-1081 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)N3CCOCC3 MS-10810 Cc1ccc2c(c1)N/C(=C(/C#N)\S(=O)(=O)c3ccc(cc3)OC(F)(F)F)/N2 MS-10811 c1cc(ccc1OC(F)(F)F)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-] MS-10812 CC(C)C1CC(=O)C(=CNc2ccc(cc2)OC(F)(F)F)C(=O)C1 MS-10817 Cc1ccc(cc1)C(=O)C2C(=O)c3ccccc3C2=O MS-10819 CC1Cc2c(c(nn2C)c3ccc4c(c3)OCO4)/C(=N\O)/C1 MS-10820 CC(=O)c1ccc(cc1)/N=C(\C)/C2C(=O)c3ccccc3C2=O MS-10821 COc1ccc(cc1OC)c2c\3c([nH]n2)-c4ccccc4/C3=N/OC MS-10822 CC1Cc2c(cc(n2c3cccc(c3)C(F)(F)F)c4cccc(c4)Br)/C(=N\O)/C1 MS-10823 c1cc(ccc1OC(F)(F)F)S(=O)(=O)/C(=C\Nc2cc(ccc2F)C(F)(F)F)/[N+](=O)[O-] MS-10824 CC(C)CC1CC(=O)C(=CNc2ccc(cc2)/C(=N\OC)/C)C(=O)C1 MS-10825 C/C(=N/OC)/c1ccc(cc1)NC(=C2C(=O)c3ccccc3C2=O)C MS-10826 CCCCn1c(cc2c1CC(CC2=O)C)c3ccc(cc3)C MS-10827 Cc1ccc(cc1)c2cc3c(n2CCOC)CC(CC3=O)C MS-10828 CC(=C1C(=O)c2ccccc2C1=O)NCc3ccc(cc3F)F MS-10829 CCOC(=O)c1ccccc1CN2C(=O)c3ccccc3S2(=O)=O MS-1083 c1cc(ccc1CC#N)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Br MS-10830 CSC(=C(C#N)S(=O)(=O)c1ccc(cc1)OC(F)(F)F)SC MS-10831 COc1ccc(cc1OC)CCNC(=O)Cc2nc(on2)C(F)(F)F MS-10832 CCC(CC)(C#C)N/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl MS-10833 CC(C)(C)C(=O)/C(=C\Nc1[nH]cnn1)/C#N MS-10834 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(ccc2Br)C(F)(F)F)/C#N)Cl MS-10835 Cc1cc(no1)N/C=C(/C#N)\C(=O)C(C)(C)C MS-10836 CC(=C1C(=O)c2ccccc2C1=O)Nc3cc(ccc3F)C(F)(F)F MS-10837 CCOc1ccc(cc1)N=C2c3cc(ccc3NC2=O)Br MS-10838 CCC(CC)(C#C)N/C=C(/C#N)\C(=O)C(C)(C)C MS-10839 CCOC(=O)c1c[nH]c2cc(ccc2c1=O)OCc3ccccc3 MS-10840 CC(C)(C)C(=O)/C(=C/NCCOC)/C#N MS-10841 c1cnc(nc1)N/C=C(/[N+](=O)[O-])\S(=O)(=O)c2ccc(cc2)OC(F)(F)F MS-10842 CC(C)(C)c1ccc(cc1)S(=O)(=O)CC#N MS-10843 CC(C)(C)C(=O)C(=C1Oc2ccc(cc2S1)O)C#N MS-10844 Cc1ccc(cc1)c2c3c([nH]n2)-c4ccccc4C3=NO MS-10845 CC(C)(C)C(=O)/C(=C/Nc1cccc(c1)OCc2ccccc2)/C#N MS-10846 CC(C)(C)C(=O)C(=C(Nc1ccccc1Cl)SC)C#N MS-10847 c1ccc2cc(ccc2c1)c3csc([nH+]3)Nc4ccc(cc4)OC(F)(F)F.[Br-] MS-10848 CC(C)c1ccc(cc1)c2cc\3c(nn2)CC(C/C3=N\O)(C)C MS-10849 Cc1cc(no1)NC2=CC(=O)CC(C2)C(C)C MS-10850 CCC1CC(=O)C(=CNc2cc(on2)C)C(=O)C1 MS-10851 CCOC(=O)CC(=O)CC1C(=O)CC(CC1=O)(C)C MS-10852 c1cc(ccc1N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccc(cc2)Br)OC(F)(F)F MS-10853 c1cc(ccc1S(=O)(=O)/C(=C/Nc2ccc(cc2F)F)/[N+](=O)[O-])Br MS-10854 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)F)/C#N MS-10855 Cn1c-2c(c(n1)c3ccc(c(c3)OC)OC)/C(=N\O)/c4c2cccc4 MS-10856 Cc1ccc(cc1)S(=O)(=O)Cc2c(c(=O)n(n2C)c3ccccc3)Br MS-10857 CCOC(=O)CC(=O)CC1C(=O)CC(CC1=O)C MS-10858 CCOC(=O)Cc1cc2c(n1c3ccc(cc3)OC(F)(F)F)CC(CC2=O)C MS-10859 CCOC(=O)Cc1cc\2c(n1c3ccc(cc3)OC(F)(F)F)CC(C/C2=N\OC)C MS-10860 C=CCNC(=S)NNC(=O)Nc1ccc(cc1)OC(F)(F)F MS-10861 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2cccc(c2)OC(C(F)F)(F)F)/[N+](=O)[O-] MS-10862 c1ccc(cc1)Nc2ccc(cc2)NC=C(C#N)C#N MS-10863 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)F)/[N+](=O)[O-] MS-10864 CCO/N=C\1/c2ccccc2-c3c1c(nn3C)C(C)(C)C MS-10865 CC1Cc2c(cc(n2CCC(=O)O)c3ccc(cc3)Br)/C(=N/OC)/C1 MS-10866 Cc1c(c(no1)c2ccccc2)C(=O)NCC#C MS-10867 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)SC(F)(F)F MS-10868 CCOC(=O)Cc1cc2c(n1c3cc(on3)C)CC(CC2=O)C MS-10869 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)Oc3ccccc3)/[N+](=O)[O-] MS-10870 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C(/Nc2ccccc2)\S)/C#N MS-10871 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(ccn2)C(F)(F)F)/[N+](=O)[O-])Br MS-10872 c1ccc(cc1)CCNC(=O)CSc2ccc(cc2)Cl MS-10873 CCOC(=O)/C(=C/NCC#C)/C#N MS-10874 c1ccc2c(c1)c(c[nH]2)CCNC(=O)/C=C/c3cc4c(cc3[N+](=O)[O-])OCO4 MS-10875 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-10876 C#CCN/C=C(\C#N)/S(=O)(=O)c1ccccc1 MS-10877 Cc1ccc(cc1)S(=O)(=O)/C(=C\NCC#C)/C#N MS-10878 c1ccc(c(c1)C(F)(F)F)NN=C(C#N)C#N MS-10879 CCOC(=O)C1C(CN(C1=O)O)c2ccc(cc2)F MS-1088 CSC(=C1C(=O)c2ccccc2C1=O)NCC#C MS-10880 Cc1cc2c(cc1C)NC(=C3C(=O)c4ccccc4C3=O)N2 MS-10881 c1ccc2c(c1)C(=O)C(=C3Nc4cc(c(cc4N3)Cl)Cl)C2=O MS-10882 c1ccc2c(c1)C(=O)C(=C3Nc4ccccc4N3)C2=O MS-10883 c1cnc(cc1C(F)(F)F)NC=C(C#N)C#N MS-10884 CC1(Cc2c(sc(n2)N)/C(=N/OC)/C1)C MS-10885 CC(=O)Nc1nc2c(s1)C(=NOC)CC(C2)(C)C MS-10886 CC(C)(C)c1c\2c(n(n1)C)-c3ccccc3/C2=N\OCC=C MS-10887 CC(C)(C)S(=O)(=O)/C(=C\Nc1cc(ccn1)C(F)(F)F)/C#N MS-10888 c1ccc(c(c1)C(=O)NN)N MS-1089 CCON=C1CC(Cc2c1sc(n2)N)(C)C MS-10890 CCO/N=C\1/CC(Cc2c1sc(n2)NC(=O)C)(C)C MS-10891 c1cc(ccc1CBr)S(=O)(=O)Nc2ccc(cc2)F MS-10892 CC(C(=O)NCCOC)Sc1ccc(cc1)Cl MS-10893 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)Sc4ccccn4)C2=O MS-10894 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)n4cnc(c4Cl)Cl)C2=O MS-10895 C/C(=C\C(=O)c1ccccc1)/N/C(=C(/C#N)\N)/C#N MS-10896 CC1(Cc2c(sc(n2)NC(=O)c3ccc(cc3)Cl)/C(=N/OC)/C1)C MS-10897 c1ccnc(c1)Sc2ccc(cc2)NC=C(C#N)C#N MS-10898 c1ccc2c(c1)C(=O)C(=CNCCN3CCOCC3)C2=O MS-10899 CCOC(=O)C(C(C[N+](=O)[O-])c1ccc(cc1Cl)Cl)C(=O)OCC MS-1090 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)Sc4ccccn4 MS-10900 CC(C)C/C=C/C(=O)NC(Cc1c[nH]c2c1cccc2)C(=O)OC MS-10901 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)C(C(F)(F)F)(C(F)(F)F)O)/C#N MS-10902 C1COCCN1C=C(C#N)C#N MS-10903 CC(C)(C)C(=O)C(=C(NCC#C)NCC#C)C#N MS-10904 Cc1cc2c(n1c3ccc(cc3)C(=O)O)CC(CC2=O)(C)C MS-10905 c1ccc2c(c1)C(=O)C(C2=O)C(=O)/C=C/c3ccc4c(c3)OCO4 MS-10906 CC(=C1C(=O)c2ccccc2C1=O)Nc3cccc(c3)OCc4ccccc4 MS-10907 C#CCNC(=O)c1cccnc1Oc2ccccc2 MS-10908 c1ccc(cc1)Oc2c(cccn2)C(=O)NCCc3c[nH]c4c3cccc4 MS-10909 CCOC(=O)C1C(CN(C1=O)O)c2ccccc2 MS-1091 Cc1cc(no1)NC(=O)c2cccnc2Oc3ccccc3 MS-10910 CC1(Cc2c(sc(n2)NC(=O)c3cccnc3Cl)C(=O)C1)C MS-10911 c1cc(cc(c1)Oc2ccc(cc2)N/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Br)C(F)(F)F MS-10912 c1ccc(cc1)COc2cccc(c2)NC(=O)c3cccnc3Cl MS-10913 c1cc(c(nc1)Cl)C(=O)Nc2ccc(cc2)n3cncn3 MS-10914 c1ccc2c(c1)nc(s2)Sc3ccc(cc3C=C(C#N)C#N)[N+](=O)[O-] MS-10915 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)Oc3cccc(c3)C(F)(F)F)/C#N MS-10916 c1cc(cc(c1)Oc2ccc(cc2)N/C=C(\C#N)/S(=O)(=O)c3ccc(cc3Cl)Cl)C(F)(F)F MS-10917 CC(C)CC1CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)F)C(=O)C1 MS-10918 Cc1cc(no1)NC(=O)c2cccnc2Oc3ccc(cc3)Cl MS-10919 CCOC(=O)CC(=NNC(=O)c1ccccc1N)CC(=O)OCC MS-1092 c1cc2cccnc2c(c1)NC(=O)c3cccnc3Oc4ccc(cc4)Cl MS-10920 c1cc[n+](cc1)c2c(c3ccccc3[nH]2)CCNC(=O)c4ccc(cc4)Cl.[Br-] MS-10921 c1ccc(cc1)NC(=O)NNC(=O)Cc2c[nH]c3c2cccc3 MS-10922 c1ccc2c(c1)c(c[nH]2)CC(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F MS-10923 c1ccc(cc1)CCNC(=O)c2cccnc2Oc3ccccc3 MS-10924 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3cccnc3Oc4ccc(cc4)Cl MS-10925 Cc1ccc(cc1)Sc2c(cccn2)C(=O)NCCc3c[nH]c4c3cccc4 MS-10926 c1ccc2c(c1)/C(=N/C(=C(/C#N)\N)/C#N)/C(=O)N2 MS-10927 c1cc[n+](cc1)c2c(c3ccccc3[nH]2)CCNC(=O)c4ccc(cc4)[N+](=O)[O-].[Br-] MS-10928 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)/C#N MS-10929 CCOC(=O)C(C(C[N+](=O)[O-])c1cccc(c1)Oc2ccccc2)C(=O)OCC MS-1093 c1cc(ccc1Sc2ccc(cn2)NC=C(C#N)C#N)Cl MS-10930 COc1ccc(cn1)NC(=O)CCc2ccccc2Cl MS-10931 Cc1cc(no1)NC(=O)COc2ccc(cc2Cl)Cl MS-10932 Cc1cc(no1)NC(=O)CCc2ccccc2Cl MS-10933 c1cc(ccc1N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Br)Oc3c(cc(cn3)C(F)(F)F)Cl MS-10934 CC(C)CC1CC(=O)C(=CNc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)C(=O)C1 MS-10935 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cn2)C(F)(F)F)/[N+](=O)[O-] MS-10936 Cc1ccc(c2c1CC(O2)(C)C)NC=C(C#N)C#N MS-10937 COc1cc(cc(c1OC)OC)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccc(cc4)Cl MS-10939 c1cc(sc1)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccc(cc4)Cl MS-10940 c1ccc2c(c1)/C(=N/c3ccc(cc3)OC(F)(F)F)/C(=O)N2 MS-10941 c1cc2cccnc2c(c1)Oc3ccc(cn3)C(F)(F)F MS-10942 c1cc(cc(c1)NC(=O)NNC(=O)COc2ccc(cc2)F)C(F)(F)F MS-10943 CCO/N=C\1/CC(Cc2c1sc(n2)NC(=O)c3cccs3)CC(C)C MS-10944 c1c(c(cc(c1O)O)[N+](=O)[O-])/C=N/C(=C(/C#N)\N)/C#N MS-10945 Cc1cc(ccc1OCC(=O)NNC2=CC(=O)CC(C2)(C)C)Cl MS-10946 c1cc(ccc1C(F)(F)F)Oc2ccc(cc2C=O)[N+](=O)[O-] MS-10947 c1cc(ccc1C(F)(F)F)Oc2ccc(cc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] MS-10948 CC(=NNC(=S)N)C1C(=O)c2ccccc2C1=O MS-10949 c1ccc(c(c1)CN2C(=O)c3ccccc3S2(=O)=O)C(=O)O MS-1095 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC2=CC(=O)CC(C2)(C)C MS-10950 CC(C)(C)C(=O)/C(=C\c1ccc(cc1)[N+](=O)[O-])/C#N MS-10951 COc1ccc(cc1OC)CC(=O)NN MS-10952 COc1ccc(cc1OC)CC(=O)NNC(=S)NC2CCCCC2 MS-10953 c1cc(c(cc1Cl)Cl)OCC(=O)NN MS-10954 CC(C)(C)C(=O)/C(=C\Nc1ncccn1)/C#N MS-10955 COc1ccc(cc1OC)/C=C\2/C(=O)NC(=S)S2 MS-10957 c1cc(cnc1)/C=C\2/C(=O)NC(=S)S2 MS-10958 CSC(=C(C#N)C#N)Nc1ccccc1 MS-10959 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NN2CCOCC2 MS-1096 CC(C)(C)C(=O)C(=C(Nc1cccc(c1)C(F)(F)F)O)C#N MS-10960 c1ccc(cc1)N/C(=C(/C#N)\S(=O)(=O)c2ccccc2)/S MS-10961 Cc1ccc(cc1)S(=O)(=O)/C(=C(/Nc2ccccc2)\SC)/C#N MS-10962 c1ccc(cc1)n2c(n[nH]c2=S)COc3cccc(c3Cl)Cl MS-10963 c1ccc(cc1)C(=Nc2nc[nH]n2)C3C(=O)c4ccccc4C3=O MS-10964 CCCCCC(=O)n1c(c2c(n1)-c3ccccc3C2=O)c4ccc(cc4)OC MS-10965 COc1cc(cc(c1OC)OC)C(=O)NN MS-10966 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2c(n(n(c2=O)c3ccccc3)C)C)/C#N MS-10968 c1ccc2c(c1)C(=O)C(C2=O)C(=O)c3cccs3 MS-10969 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3ccccc3[N+](=O)[O-] MS-1097 c1ccc2c(c1)-c3c(c([nH]n3)c4cccs4)C2=O MS-10970 c1ccc2c(c1)C(=O)C(=C(c3cccs3)N)C2=O MS-10971 Cc1ccc(cc1)S(=O)(=O)C(=C(SC)SC)C#N MS-10972 c1ccc(cc1)C(=C2C(=O)c3ccccc3C2=O)N MS-10973 c1cc(cc(c1)NN=C(C#N)C#N)C(F)(F)F MS-10974 c1ccc2c(c1)C(=C(C2=O)C(=O)C3CCCCC3)O MS-10975 CCOC(=O)/C(=C/Nc1ccc(cc1)O)/C(=O)C MS-10976 Cc1ccc(cc1)S(=O)(=O)/C(=C(/Nc2ccccc2)\N3CCN(CC3)c4ccccc4)/C#N MS-10977 c1ccc(cc1)Oc2ccc(cc2)NC=C(C#N)C#N MS-10978 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)O MS-10979 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3ccccc3[NH3+].[Cl-] MS-1098 CNC(=C(C#N)C#N)SC MS-10980 CCOC(=O)C(=CNc1ncc(s1)c2ccc(cc2)Br)C#N MS-10981 CC(C)(C)c1c(c(nc(n1)N)Nc2ccccc2)C#N MS-10982 c1ccc(cc1)C(=Nc2cccc(c2)C(F)(F)F)C3C(=O)c4ccccc4C3=O MS-10983 c1ccc(cc1)C2CC(=O)C(C(=O)C2)CC(=O)c3ccc(cc3)Br MS-10984 c1ccc(cc1)C(=Nc2ccc(cc2)F)C3C(=O)c4ccccc4C3=O MS-10985 CSC(=C(C#N)S(=O)(=O)c1ccc(cc1Cl)Cl)SC MS-10986 Cc1ccc(cc1)S(=O)(=O)/C(=C/NN)/C#N MS-10987 c1cc(ccc1S(=O)(=O)/C(=C/NN)/C#N)Cl MS-10988 c1cc(ccc1OCC(=NO)N)Cl MS-10989 c1ccc(cc1)CN2CCC(CC2)N3N=Nc4ccccc4S3(=O)=O MS-1099 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)Nc2ccccc2 MS-10990 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)NC2CCCCC2 MS-10991 CCc1ccc(cc1)c2csc(n2)N MS-10992 Cc1cc(ccc1N)OCc2ccccc2 MS-10993 COC(=O)/C=C/c1ccc(cc1)OCc2ccccc2 MS-10994 COC(=O)c1ccc(cc1)OCc2ccccc2 MS-10995 Cc1cc([nH]n1)c2ccccc2 MS-10996 COC(=O)CCc1ccc(cc1)[N+](=O)[O-] MS-10997 COc1cccc(c1)c2csc(n2)N MS-10998 COc1ccc(c(c1)c2csc(n2)N)OC MS-10999 CNC(=O)NNC(=O)c1cccc(c1)Br MS-1100 COc1ccc(cc1OC)c2csc(n2)N MS-11000 CC(C)(C)OC(=O)CCc1ccc(cc1)Nc2c(c(c(c(c2F)F)C(F)(F)F)F)F MS-11001 c1ccc(cc1)Oc2ccc(cc2)c3csc(n3)N MS-11002 c1ccc-2c(c1)CCc3c2nc(s3)N MS-11003 Cc1c(nc(s1)N)c2ccc(cc2)Cl MS-11004 c1cc(c(cc1c2csc(n2)N)O)O MS-11005 c1ccc(c(c1)c2csc(n2)N)OC(F)(F)F MS-11006 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2csc(n2)N MS-11007 c1ccc(c(c1)c2csc(n2)N)Br MS-11008 c1ccc(c(c1)c2csc(n2)N)[N+](=O)[O-] MS-11009 CCCN(CCOc1c(cc(cc1Cl)Cl)Cl)C(=O)c2ccccn2 MS-1101 COc1cc(ccc1O)c2csc(n2)N MS-11010 c1ccc2cc(ccc2c1)c3csc(n3)N MS-11011 c1cc(ccc1c2csc(n2)N)C3CCCCC3 MS-11012 c1cc(c(cc1F)O)c2csc(n2)N MS-11013 COc1ccc2cc(ccc2c1)c3csc(n3)N MS-11014 CC1(CCc2c1cc(cc2c3csc(n3)N)C(C)(C)C)C MS-11015 c1cc2c(cc1CN3CCN(CC3)CC(=O)Nc4ccc(cc4F)F)OCO2 MS-11016 c1ccc2c(c1)CCN2CC(=O)Nc3ccc(cc3)F MS-11017 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=O)c4cccs4 MS-11018 CCCNC(=O)Nc1ccc-2c(c1)C(=O)c3c2n(nc3C(C)(C)C)C MS-11019 c1ccc(c(c1)C(=O)CC#N)Oc2cc(cc(c2)Cl)Cl MS-1102 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=O)c4c(cccc4F)F MS-11020 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=S)NC4CCCCC4 MS-11021 c1ccc(cc1)COc2cccnc2NS(=O)(=O)c3ccc(c(c3)[N+](=O)[O-])Cl MS-11022 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)C=O)OC MS-11023 Cc1ccc(cc1)NC(=S)Nc2c(cccn2)OCc3ccccc3 MS-11024 CN1CCN(CC1)CC(=O)Nc2cc(cc(c2)C(=O)OC)C(=O)OC MS-11025 c1cc(ccc1NC(=O)CN2CCN(CC2)Cc3ccc4c(c3)OCO4)SC(F)(F)F MS-11026 CC(C)C(=O)N(Cc1ccc(cc1)OC)c2ccc3c(c2)OCO3 MS-11027 CC(C)c1ccc(cc1)CN(c2ccc3c(c2)OCO3)S(=O)(=O)c4cccs4 MS-11028 CC(=O)Nc1ccc(cc1)S(=O)(=O)N(Cc2ccco2)c3ccc4c(c3)OCO4 MS-11029 Cc1cc(ccc1Oc2cccc(c2)C(=O)CC#N)Cl MS-1103 CC(C)C(=O)N(Cc1ccco1)c2ccc3c(c2)OCO3 MS-11030 CC(=O)Nc1ccc(cc1)S(=O)(=O)N(Cc2cccs2)c3ccc4c(c3)OCO4 MS-11031 c1cc(cnc1)CN(c2ccc3c(c2)OCO3)S(=O)(=O)c4cccs4 MS-11032 Cc1c(sc(n1)Nc2ccc(cc2Cl)Cl)C(=O)C MS-11033 CCOC(=O)c1csc(n1)Nc2cc(ccc2OC)Cl MS-11034 c1cnc(nc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)F MS-11035 CC(C)(C)c1ccc(cc1)c2csc(n2)Nc3ccc(cc3)OC(F)(F)F MS-11036 c1cc(ccc1NC(=O)CN2CCN(CC2)Cc3ccc4c(c3)OCO4)F MS-11037 Cc1ccc(cc1)S(=O)(=O)Cc2csc(n2)Nc3ccc(cc3Cl)Cl MS-11038 Cc1ccc(cc1)S(=O)(=O)Cc2csc(n2)Nc3cc(ccc3OC)Cl MS-11039 Cc1ccc(cc1)S(=O)(=O)Cc2csc(n2)Nc3cccc(c3)C(F)(F)F MS-11040 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=O)Nc4cccc(c4)C(F)(F)F MS-11041 Cc1ccccc1NC(=O)Nc2ccc-3c(c2)C(=O)c4c3n(nc4C(C)(C)C)C MS-11042 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=S)Nc4cc(ccc4OC)Cl MS-11043 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=O)c4cc(ccc4Cl)[N+](=O)[O-] MS-11044 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=O)C(=O)c4c[nH]c5c4cccc5 MS-11045 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NS(=O)(=O)c4ccc5ccccc5c4 MS-11046 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=S)Nc4ccc(cc4)OC MS-11047 Cc1cc(c(c(c1)C)S(=O)(=O)Nc2ccc-3c(c2)C(=O)c4c3n(nc4C(C)(C)C)C)C MS-11048 c1cnc(nc1)N2CCN(CC2)CC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-11049 CCC(=O)C1=C(CCC(C1=O)c2cccc(c2)Oc3ccccc3)O MS-1105 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)Nc4ccc(cc4F)F MS-11050 Cc1ccc(cc1N2CCN(CC2)CC(=O)Nc3ccc(cc3F)F)Cl MS-11051 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3F)F MS-11052 c1cnc(nc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3F)F MS-11053 c1cc(sc1)C2=CC(=NCCN2)C(F)(F)F MS-11054 c1cc(sc1C2=[NH+]CCNC(=C2)C(F)(F)F)[N+](=O)[O-].N(=O)(=O)[O-] MS-11055 c1ccc(cc1)C2c3c(=O)[nH]c(=S)[nH]c3OC(=C2C#N)N MS-11056 c1cc(cc(c1)[N+](=O)[O-])C2c3c(=O)[nH]c(=O)[nH]c3OC(=C2C#N)N MS-11057 Cc1c2c([nH]n1)OC(=C(C2c3ccccc3)C#N)N MS-11058 CC1=NNC(=O)C1C(c2ccccc2)C(C#N)C#N MS-11059 Cn1c(n[nH]c1=O)c2cccc(c2)Br MS-1106 CCOc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)OC(=C2C(=O)OCC)N MS-11060 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cccs3)C(=O)C1)C MS-11061 Cc1ccc(cc1)C(=O)Nc2nc3c(s2)C(=O)CC(C3)(C)C MS-11062 c1cc2cccnc2c(c1)Oc3ccc(cc3[N+](=O)[O-])Cl MS-11063 CC(=NO)c1ccc(cc1)N=C2c3cc(ccc3NC2=O)Br MS-11064 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4cccnc4 MS-11065 c1ccc(cc1)NC(=S)N2CCN(CC2)c3ccc(cn3)C(F)(F)F MS-11066 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F MS-11067 CC1(CC2=C(C(Nc3ccc(cc3N2)C(=O)O)c4ccc5c(c4)OCO5)C(=O)C1)C MS-11068 CC1=NN(C(=O)C1=CC=Cc2ccc(cc2)OC)c3ccccc3 MS-11069 COc1ccc(cc1)C=CC=C2C(=O)c3ccccc3C2=O MS-11070 COc1ccc(cc1)C=CC=NC(=C(C#N)N)C#N MS-11071 CCN1C(=O)C(=CC=Cc2ccc(cc2)OC)SC1=S MS-11072 c1ccc(cc1)/C=C/C=C\2/C(=O)NC(=O)S2 MS-11073 c1ccc(cc1)Oc2c(cccn2)C(=O)O/N=C(/c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)\N MS-11074 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C(=O)c3c[nH]c4c3cccc4 MS-11075 c1cc(cnc1)C(=O)Nc2nc(cs2)c3ccc(cc3)Br MS-11076 Cc1c(nc(s1)NC(=O)c2cccnc2)c3ccc(cc3)Br MS-11077 c1cc(ccc1NC(=S)NNC(=O)c2ccncc2)Cl MS-11078 c1cnccc1C(=O)NNC(=O)C2CC2C(=O)O MS-11079 c1cc(cc(c1)Br)C(=O)NNCCC#N MS-1108 c1cc(ccc1NC(=S)NNC(=O)c2ccncc2)OC(F)(F)F MS-11080 CC1CC(=O)C(C(=O)C1)CC(=O)c2ccc(cc2)Br MS-11081 CC1CC2=NNC(=CC2C(=O)C1)c3ccc(cc3)Br MS-11082 CC1Cc2c(cc(n2c3ccc(cc3)Sc4c(cc(cn4)C(F)(F)F)Cl)c5ccc(cc5)Br)C(=O)C1 MS-11083 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccccc3C#N MS-11084 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3nc(cs3)c4ccccc4 MS-11085 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCCc3c[nH]c4c3cccc4 MS-11086 CCOc1ccc(cc1)/C=C(/C#N)\C(=O)C(C)(C)C MS-11087 CCOc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O MS-11088 Cc1ccc(cc1N2CCN(CC2)C(=O)Nc3cccc(c3)C(F)(F)F)Cl MS-11089 CC(C)N(c1ccccc1)C(=O)c2ccccc2CN3C(=O)c4ccccc4S3(=O)=O MS-1109 CC(C)(C)c1ccc(cc1)c2csc(n2)Nc3cccc4c3cccc4 MS-11090 Cc1cc(no1)NC(=O)c2c(onc2c3ccccc3Cl)C MS-11091 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCCN(CC3)S(=O)(=O)c4ccc5ccccc5c4 MS-11092 c1ccc2c(c1)C(=O)C(=Cc3c(c(c(c(c3F)F)F)F)F)C2=O MS-11093 c1ccc2c(c1)/C(=N/NC(=S)N)/CC2=O MS-11094 CC(C(=O)NNC(=S)Nc1ccccc1)Sc2ccc(cc2)Cl MS-11095 CC(c1n[nH]c(=S)n1c2ccccc2)Sc3ccc(cc3)Cl MS-11096 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)C3CC3)C(F)(F)F MS-11097 c1ccc2c(c1)c(c[nH]2)CC(=O)NNC(=O)Nc3ccc(cc3)Cl MS-11098 Cc1ccc2c(c1)CCCN2C(=O)c3c(onc3c4ccccc4Cl)C MS-11099 CNc1c(c(nc(c1Cl)F)F)Cl MS-1110 Cc1ccc(c(c1)C)OCc2n[nH]c(=S)n2c3ccccc3 MS-11100 Cc1cc(nc(c1)NC=C2C(=O)c3ccccc3C2=O)C MS-11101 Cc1cccc(c1)NC2=C(C(=O)c3c2cccc3)c4ccc5c(c4)OCO5 MS-11102 CCOc1ccc(cc1)N/C=C(\C(=O)OCC)/S(=O)(=O)c2ccc(cc2)C MS-11103 CCOC(=O)c1c2c(sc1NC(=O)c3c(onc3c4ccccc4Cl)C)CCCC2 MS-11104 c1ccc(c(c1)C(=O)NNC(=O)Nc2ccc(cc2)Cl)N MS-11105 Cc1ccc(cc1)S(=O)(=O)CC(=O)N/N=C\2/CCCC(=O)C2 MS-11106 c1ccc(cc1)NC(=S)NNC(=O)CS(=O)(=O)c2ccc(cc2)Cl MS-11107 c1cc(cc(c1)NC(=O)NNC(=O)CS(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F MS-11108 CC(C(=O)Nc1ccc(cc1)C(=O)C)Sc2[nH]c(=O)c3ccccc3n2 MS-11109 Cn1ccnc1C(=O)Nc2ccc(cc2Br)Cl MS-1111 c1ccc2c(c1)/C(=N/NC(=O)COc3cccc(c3)C(F)(F)F)/C(=O)N2 MS-11110 c1ccc(cc1)NC(=O)NNC(=O)COc2cccc(c2)C(F)(F)F MS-11111 CCOC(=O)c1cccc(c1)OCC(=O)NNC(=O)Nc2ccccc2 MS-11112 CC\1=NN(C(=O)/C1=C\c2ccc(cc2)OC)c3ccccc3 MS-11113 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)NC(=O)C)/C#N MS-11114 CC(C)c1ccc(cc1)NS(=O)(=O)CC23CCC(C2(C)C)CC3=O MS-11115 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3cccc(c3)F)C MS-11116 CC(C)(C)C\1=NN(C(=O)/C1=C\c2ccc(cc2)OCc3ccc(cc3)[N+](=O)[O-])c4ccccc4 MS-11117 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC2=NCCS2 MS-11118 c1ccc(c(c1)N2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F)F MS-11119 COc1ccc(cc1OC)CCNC(=O)Oc2ccccc2 MS-1112 CC(C)Cc1ccc(cc1)C2NC(C(S2)(C)C)C(=O)O MS-11120 CC1(C(NC(S1)c2ccc(cc2O)OC)C(=O)O)C MS-11121 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)CC34CCC(C3(C)C)CC4=O)Cl MS-11122 CC(C)Cc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)Nc4ccccc4N2 MS-11123 Cc1cc(nc(n1)C)NS(=O)(=O)c2ccc(cc2)NC=C3C(=O)c4ccccc4C3=O MS-11124 Cc1cc(nc(n1)C)NS(=O)(=O)c2ccc(cc2)NC=C3C(=O)OC(OC3=O)(C)C MS-11125 Cc1cc(nc(n1)C)NS(=O)(=O)c2ccc(cc2)N/C=C(/C(=O)C)\C(=O)Nc3ccccc3 MS-11126 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl MS-11127 Cc1ccc(cc1NC(=O)OC)Oc2ccc(cc2Cl)C(F)(F)F MS-1113 c1cc(c(cc1Cl)C(=O)NN)Cl MS-11130 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCc2cccs2 MS-11134 c1ccc(cc1)COc\2cccn(/c2=N\C(=O)c3cccc4c3cccc4)C(=O)c5cccc6c5cccc6 MS-11135 CC(C)(C)C\1=NN(C(=O)/C1=C\c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)c4ccccc4 MS-11136 C/C(=C\C(=O)Nc1ccccc1)/NCCN2CCOCC2 MS-11137 c1c(cc(c(c1[N+](=O)[O-])N)Br)C(F)(F)F MS-11139 CC(C)(C)N(C(=O)c1ccccc1)NC(=O)c2ccccc2 MS-1114 COc1cccc(c1)NC2=C(C(=O)c3c2cccc3)c4ccc5c(c4)OCO5 MS-11140 c1ccnc(c1)Sc2ccc(cc2)NC(=O)/C=C/C(=O)O MS-11141 CC(C)(C)C1=NN(C(=O)C1=Cc2cccs2)C MS-11142 c1ccc(c(c1)C(=O)N)NS(=O)(=O)c2ccc(cc2)OC(F)(F)F MS-11143 c1cc(ccc1C(=O)O)NC(=O)C2CC2C(=O)O MS-11144 c1cc(sc1)CSc2ccc(cc2/C=N/NC(=S)N)[N+](=O)[O-] MS-11145 c1ccc(cc1)S(=O)(=O)/C(=C/c2cc(ccc2Oc3ccc(cc3)Br)[N+](=O)[O-])/C#N MS-11146 CC(C(=O)O)Oc1ccc(cc1)n2cncn2 MS-11149 c1ccc(cc1)C2=NC(=O)CC(=O)S2 MS-1115 CC(C(=O)NN)Oc1ccc(cc1)n2cncn2 MS-11150 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc(cc2)SC(F)(F)F)CC(=O)OC MS-11151 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc(cc2)C(F)(F)F)CC(=O)OC MS-11152 CCOC(=O)Cc1csc(n1)Nc2cc(cc(c2)Cl)Cl MS-11153 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)F MS-11154 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)Cl MS-11155 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)C MS-11156 CCc1cccc(c1Nc2nc(cs2)CC(=O)OCC)CC MS-11157 CCOC(=O)Cc1csc(n1)Nc2cccc(c2)Cl MS-11158 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)C(F)(F)F MS-11159 CCOC(=O)c1c(nc(s1)Nc2cc(cc(c2)Cl)Cl)C MS-11160 CCOC(=O)c1c(nc(s1)Nc2ccc(cc2)F)C MS-11161 CCOC(=O)c1c(nc(s1)Nc2ccc(cc2)Cl)C MS-11162 CCOC(=O)c1c(nc(s1)Nc2ccccc2F)C MS-11163 CCOC(=O)c1c(nc(s1)Nc2cccc(c2)Cl)C MS-11164 CCOC(=O)c1c(nc(s1)Nc2cc(ccc2Cl)Cl)C MS-11165 CCOC(=O)c1c(nc(s1)NCC=C)C MS-11166 c1c(cc(cc1Cl)Cl)Nc2nc(cs2)CC(=O)O MS-11167 CCOC(=O)c1csc(n1)Nc2cc(cc(c2)Cl)Cl MS-11168 CCOC(=O)c1csc(n1)Nc2ccc(cc2)F MS-11169 CCOC(=O)c1csc(n1)Nc2ccc(cc2)Cl MS-11170 CCOC(=O)c1csc(n1)Nc2ccccc2F MS-11171 CCOC(=O)c1csc(n1)Nc2cccc(c2)Cl MS-11172 CCOC(=O)c1csc(n1)Nc2ccccc2Cl MS-11173 CCOC(=O)c1csc(n1)NCC=C MS-11174 CCOC(=O)c1csc(n1)Nc2ccc(cc2)Br MS-11175 c1cc(ccc1S(=O)(=O)C/C(=N/O)/N)Br MS-11176 c1ccc2c(c1)CCN2C(=S)N MS-11178 CCOC(=O)c1c(nc(s1)Nc2ccccc2)C MS-11179 CCOC(=O)c1csc(n1)Nc2ccccc2 MS-11180 CCOC(=O)c1csc(n1)Nc2ccc(cc2)Oc3ccccc3 MS-11181 CCOC(=O)Cc1csc(n1)Nc2cc(ccc2OC)Cl MS-11182 CCOC(=O)Cc1csc(n1)Nc2ccc(c(c2)Cl)Cl MS-11183 CCOC(=O)Cc1csc(n1)Nc2cccc(c2)C(F)(F)F MS-11184 c1cc(ccc1/C=C/C(=O)O)I MS-11185 c1cc(ccc1/C=N/O)I MS-11186 c1cc(ccc1c2csc(n2)N)C(F)(F)F MS-11187 c1cc(cc(c1)NC(=S)N)C(=O)O MS-11188 CC1(CC(=C(C(=O)C1)I)Nc2ccccc2O)C MS-11189 CCC1CCCCN1C(=O)CN2C(=O)CSC2=O MS-1119 Cc1cccc(c1NC(=S)N)C(C)C MS-11190 COc1cccc(c1Oc2ccc(cn2)C(F)(F)F)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl MS-11191 CCOC(=O)C(c1ccccc1)NC=C2C(=O)c3ccccc3C2=O MS-11192 CC1(CC(=O)C(=CNc2ccc(cc2)S(=O)(=O)C)C(=O)C1)C MS-11193 c1ccc(cc1)C2CC3=C(C(Nc4ccccc4N3)c5ccco5)C(=O)C2 MS-11194 c1ccc(cc1)C2CC(=C(C(=O)C2)C(=O)Nc3ccccc3)Nc4ccccc4 MS-11195 c1ccc(cc1)N2CCN(CC2)C(=O)Nc3cccc(c3)C(F)(F)F MS-11196 c1cc(cc(c1)NC(=O)N2CCN(CC2)C(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F MS-11197 c1cc(c(cc1NC(=O)N2CCN(CC2)C(=O)Nc3ccc(c(c3)Cl)Cl)Cl)Cl MS-11198 CC(=O)c1ccc(cc1)NC2=C(C(=O)CC(C2)(C)C)Cl MS-11199 Cc1ccc(cc1)S(=O)(=O)/C(=C/N2CCN(CC2)c3ccccc3)/C#N MS-11200 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4cccc(c4)C(F)(F)F MS-11202 COc1ccc(cc1OC)CCNC2=C(C(=O)CC(C2)c3ccccc3)C(=O)Nc4cccc(c4)C(F)(F)F MS-11203 COc1ccc(cc1OC)CCNC2=C(C(=O)CC(C2)c3ccccc3)C(=O)Nc4ccccc4 MS-11204 CCOC(=O)C(=CNc1ncccn1)C#N MS-11205 c1c(cc(cc1Cl)Cl)NC=C(C#N)C#N MS-11206 c1ccc(cc1)C(=O)C2=C(c3ccccc3C2=O)Nc4cccc(c4)N MS-11207 Cc1ccc(cc1)NC2=C(C(=O)c3c2cccc3)c4ccc(c(c4)OC)OC MS-11208 Cc1cccc(c1)NC2=C(C(=O)c3c2cccc3)c4ccccc4 MS-11209 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)Nc4cccc(c4)[N+](=O)[O-] MS-11210 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)[N+](=O)[O-] MS-11211 c1ccc2c(c1)C(=O)C(=CNc3cc(cc(c3)Cl)Cl)C2=O MS-11212 Cc1ccc(cc1NC2=CC(=O)CC(C2)c3ccccc3)C(C)C MS-11213 Cc1ccc(cc1NC2=C(C(=O)CC(C2)c3ccccc3)Cl)C(C)C MS-11214 CC1=NN(C(=O)C1C(c2ccc3c(c2)OCO3)N4CCN(CC4)C)c5ccccc5 MS-11215 CCOc1ccc(cc1)NC(=S)NC(=O)c2cccs2 MS-11216 c1ccc(cc1)C2CC3=C(C(Nc4ccccc4N3)c5ccccc5Cl)C(=O)C2 MS-11217 CC(C)(C)C(=O)/C(=C\Nc1ccc(cc1)O)/C#N MS-11218 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)Br MS-11219 c1cc(ccc1S(=O)(=O)Cc2nc(on2)C(F)(F)F)Cl MS-11220 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)C(C)C)/C#N MS-11222 c1ccc(cc1)S(=O)(=O)Cc2nc(on2)C(F)(F)F MS-11223 c1nnc(s1)NC=C(C#N)C#N MS-11224 CCOC(=O)C(=CNc1nc[nH]n1)C(=O)OCC MS-11225 CCOC(=O)C(=CNc1nncs1)C(=O)OCC MS-11226 Cc1cc(ccc1F)c2csc(n2)Nc3ccc(cc3)OC MS-11227 Cc1ccc(cc1NC(=O)C2CC2)C(C)C MS-11228 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(c(c4)Cl)Cl MS-11229 c1ccc(cc1)N2CCN(CC2)C(=O)COc3cccc(c3)C(F)(F)F MS-1123 c1cc(ccc1S(=O)(=O)C/C(=N/OC(=O)C2CC2)/N)Cl MS-11230 COC(=O)/C(=C(\Nc1ccccc1)/SC)/C#N MS-11231 CCOC(=O)C(=Cc1ccc(cc1)OCc2ccc(cc2)[N+](=O)[O-])C#N MS-11232 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)OCc4ccc(cc4)[N+](=O)[O-])C2=O MS-11233 COCCNC1=C/C(=[NH+]\CCOC)/c2c1cccc2.[Cl-] MS-11234 Cc1ccc(cc1)S(=O)(=O)/C(=C/NN(C)C)/C#N MS-11235 CC(C)(C)S(=O)(=O)/C(=C\Nc1ccc(cc1)F)/C#N MS-11236 CC1CC(=O)C(C(=O)C1)(C)CC(=O)c2ccc(cc2)Br MS-11237 CC1(CC(=O)C(C(=O)C1)(C)CC(=O)c2ccc(cc2)Br)C MS-11238 c1cc(c(cc1F)F)NC=C(C#N)C#N MS-11239 c1ccc(cc1)N2CCN(CC2)C(=O)COc3cc(cc(c3)F)F MS-1124 Cc1cc(ccc1Cl)C2=NNC3=C(C2)C(=O)CC(C3)(C)C MS-11240 c1ccc2c(c1)[nH]c(n2)SCC(=O)O MS-11241 c1cnc(nc1)N/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl MS-11242 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)N=Cc3ccc4c(c3)OCO4 MS-11243 c1cc(sc1)c2c([nH]nn2)C#N MS-11244 c1ccc(cc1)C(=O)Nc2c(c3ccccc3[nH]c2=O)C(=O)Nc4ccccc4 MS-11245 Cn1c2ccccc2c3c1nc(nn3)SC MS-11246 CCOc1ccc(cc1)NC2=CC(=O)CC(C2)C MS-11247 Cn1c2ccccc2c3c1nc(nn3)N4CCOCC4 MS-11248 CC(C)(C)C(=O)C(=CNc1ccc(cc1)OC(F)(F)F)C#N MS-11249 CC(C)c1ccc(cc1)OCC(=O)N2CCN(CC2)c3ccccc3 MS-1125 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)OC(F)(F)F)C MS-11250 CC1(CC(=C(C(=O)C1)Cl)Nc2ccc(cc2)OC(F)(F)F)C MS-11251 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccc(cc3)OC(F)(F)F MS-11252 c1cc(ccc1C(F)(F)F)N/C=C(/C#N)\c2[nH]nnn2 MS-11253 c1cc(c(cc1F)F)N/C=C(/C#N)\c2[nH]nnn2 MS-11254 CC1(CC(=CC(=O)C1)Nc2cccc(c2)OC(C(F)F)(F)F)C MS-11255 c1cc(c(cc1NC(=O)N/C(=C(/C#N)\N)/C#N)Cl)Cl MS-11256 c1ccc(cc1)CNC2=CC(=O)CC(C2)c3ccccc3 MS-11258 c1ccc(c(c1)NC=C(C#N)C#N)F MS-11259 CC1(Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N/OC)/C1)C MS-11260 Cn1cc(c2c1cccc2)C(CC(=O)c3ccc(cc3)Br)C(=O)O MS-11261 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)OC(F)(F)F)/C#N MS-11262 Cc1cc(ccc1F)c2cc\3c([nH]2)CC(C/C3=N/OC)(C)C MS-11263 COc1cc(cc(c1OC)OC)/C=c\2/c(=O)n3c(=O)c4ccccc4nc3s2 MS-11264 CC1Cc2c(cc(nn2)c3ccc(cc3)Br)C(=NO)C1 MS-11265 CC1Cc2c(cc(nn2)c3ccc(cc3)Br)C(=NOC)C1 MS-11266 CC1(CC(=O)C(=C(Nc2ccccc2)S)C(=O)C1)C MS-11267 CC1(CC(=O)C(=C(Nc2ccc(cc2)Cl)S)C(=O)C1)C MS-11268 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ncccn2)/C#N MS-11269 CCC(CC)O/C(=N\c1cc(cc(c1)Cl)Cl)/c2cncn2C MS-1127 CC1(Cc2c(c(=O)c3ccccc3[nH]2)C(=O)C1)C MS-11270 c1ccc(cc1)C2Cc3c(c(=O)c4ccccc4[nH]3)C(=O)C2 MS-11271 c1cnc(nc1)N/C=C(\C#N)/C(=O)Nc2ccc(cc2Cl)Cl MS-11272 Cc1ccc(cc1)S(=O)(=O)/C(=C\NCc2ccc(cc2F)F)/C#N MS-11273 CC1=NN(C(=O)C1C(CC(=O)c2ccc(cc2)C(C)C)C(=O)O)c3ccccc3 MS-11274 CC1(CC(=C(C(=O)C1)c2nc3ccccc3s2)O)C MS-11275 CC(C(=O)NN)Oc1ccc(cc1Cl)Cl MS-11276 CC(C(=O)NNC(=O)Nc1cccc(c1)C(F)(F)F)Oc2ccc(cc2Cl)Cl MS-11277 Cc1cc(c2ccccc2n1)N/C=C(/C#N)\c3[nH]nnn3 MS-11278 Cc1cc(c2ccccc2n1)NC=C(C#N)C#N MS-11279 c1ccc(c(c1)C(=O)CC#N)Oc2ccc(cc2)F MS-1128 C#CCSc1nc([nH]n1)c2ccccc2 MS-11281 c1cc(ccc1/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)F MS-11282 CO/N=C/1\CC(Cc2c1cc(nn2)c3ccc(cc3)Br)c4ccccc4 MS-11283 CC1Cc2c(cc(nn2)c3ccccc3)C(=NOC)C1 MS-11284 CC1Cc2c(cc(nn2)c3ccc(cc3)Cl)C(=NOC)C1 MS-11285 CC1(Cc2c(cc(n2c3ccc(cc3)F)c4ccc(cc4)Br)/C(=N/OC)/C1)C MS-11286 CC1CC(=O)C(C(=O)C1)CC(=O)c2cccc(c2)Br MS-11287 CC1(CC(=O)C(=CNc2ccc(cc2)[N+](=O)[O-])C(=O)C1)C MS-11288 CC1(Cc2c(c(nn2C)c3ccc4c(c3)OCO4)/C(=N\O)/C1)C MS-11289 CCOC(=O)c1cc([nH]c1c2ccccc2)c3ccc(c(c3)C)Cl MS-11292 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)N2CCN(CC2)C)/C#N MS-11294 CC1(Cc2c(c(nn2C)c3ccc(cc3)OC)/C(=N\OC)/C1)C MS-11295 CC1Cc2c(cc(nn2)c3ccc(cc3)OC)C(=NOC)C1 MS-11296 c1ccc(cc1)Oc2ccc(cc2)N/C=C(/C#N)\S(=O)(=O)c3ccccc3 MS-11297 COc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O MS-11298 CC1Cc2c(c(nn2C)c3ccc(c(c3)OC)OC)/C(=N/O)/C1 MS-11299 CC1Cc2c(c(nn2C)c3ccc(c(c3)OC)OC)/C(=N/OC)/C1 MS-11300 CC1Cc2c(cc(n2c3ccc(cc3)OC(F)(F)F)c4ccc(cc4)C(C)(C)C)/C(=N/OC)/C1 MS-11301 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)OC(F)(F)F)C2=O MS-11302 C/C(=N\OC)/c1ccc(cc1)n2c(cc\3c2CC(C/C3=N/OC)(C)C)c4ccc(cc4)C(C)(C)C MS-11303 Cn1c(c(c(=O)n1c2ccccc2)Br)CS(=O)(=O)c3ccc(cc3)Cl MS-11304 Cc1cc(nc(n1)N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccc(cc2)OC(F)(F)F)C MS-11305 c1ccc(cc1)Oc2ccc(cc2)N/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Cl MS-11306 CC1CC2=C(CC(=NN2)c3ccc(cc3)c4ccccc4)C(=O)C1 MS-11307 CC1Cc2c(cc(nn2)c3ccc(cc3)c4ccccc4)C(=NOC)C1 MS-11308 Cc1cc(no1)NC2=CC(=O)CC(C2)CC(C)C MS-11309 COC(c1ccccc1)/C(=N/O)/c2ccc(cc2)Cl MS-1131 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3[N+](=O)[O-])C(F)(F)F)C2=O MS-11310 CCOc1ccc(cc1)Nc2[nH+]c(cs2)c3ccccc3.[Cl-] MS-11311 Cc1cc(no1)NC2=C(C(=O)c3c2cccc3)c4ccc(cc4)OC MS-11312 CC\1=NN(C(=O)/C1=C/c2cccc(c2)Oc3ccccc3)c4ccccc4 MS-11313 C#CCSc1nc([nH]n1)c2cccc(c2)Cl MS-11314 Cn1c(c(c(=O)n1c2ccccc2)Br)CSc3ccccn3 MS-11315 Cn1c(c(c(=O)n1c2ccccc2)Br)CSc3ccc(cc3)Cl MS-11316 CC(C)(C)C(=O)/C(=C/Nc1cc(ccc1F)C(F)(F)F)/C#N MS-11317 CC1CC2=C(C(=O)C1)C3(C(=C(O2)N)C#N)C(=O)c4ccccc4C3=O MS-11318 Cc1c(sc([nH+]1)Nc2cccc(c2)C(F)(F)F)C(=O)C.[Cl-] MS-11319 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccc3OC MS-1132 Cc1c(sc(n1)Nc2cccc(c2)C(F)(F)F)C(=NO)C MS-11320 Cc1c(sc(n1)Nc2ccc(cc2)OC)C(=NO)C MS-11321 c1ccc(cc1)/C=C/COc2[nH]nc(n2)c3ccccc3 MS-11322 c1ccc2c(c1)C(=O)c3ccc(cc3C2=O)NC=C(C#N)C#N MS-11323 Cc1c(c(=O)n(n1C)c2ccccc2)Cl MS-11324 COc1cccc(c1OC)c2[nH]nc(n2)SCC=C MS-11325 Cc1cc(ccc1F)c2cc\3c(nn2)CC(C/C3=N\OC)C MS-11326 c1ccc(cc1)Nc2ccc(cc2)N/C=C(\C#N)/c3[nH]nnn3 MS-11327 CC1Cc2c(c3ccccc3[nH]2)C(=O)C1 MS-11328 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccccc3Cl MS-11329 COc1ccc(c(c1)S(=O)(=O)N2CCN(CC2)c3ccccc3OC)OC MS-1133 CC(C)/C=N/NC(=S)N MS-11330 CC1(CC(=CC(=O)C1)NNc2ccccc2)C MS-11331 c1ccc2c(c1)C(=O)c3c(ccc(c3C2=O)O)NC=C(C#N)C#N MS-11332 c1ccc(cc1)/C=C/CO/C(=N/N=C/c2ccccc2)/N MS-11333 c1cc(ccc1C=Nc2c([nH]c(=O)n(c2=N)c3ccc(cc3)OC(F)(F)F)C#N)F MS-11334 Cc1cc(no1)NC(=O)c2c(onc2c3ccccc3)C MS-11335 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccccc3C(=O)N MS-11336 CC1CC(=CC(=O)C1)NCCc2ccc(c(c2)OC)OC MS-11337 COc1nnc(n1c2ccccc2)c3ccc(cc3)Cl MS-11338 CCSC(=NN=Cc1ccccc1)[NH3+].[I-] MS-11339 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(cc3Cl)Cl MS-1134 CCOC(=O)C1=C(OCC1=O)Nc2ccc(cc2)OC(F)(F)F MS-11340 CC(C)(/C(=N\O)/c1ccccc1)n2ccnc2 MS-11341 c1ccc2c(c1)cccc2C3=C(c4ccccc4C3=O)Nc5cccc(c5)F MS-11342 Cc1c(c(=O)n(n1C)c2ccccc2)NC3=C(C(=O)c4c3cccc4)c5cccc6c5cccc6 MS-11343 c1ccc(cc1)N2CC(OC2=O)COc3ccccc3 MS-11344 Cc1cc(c2c(c1)occ(c2=O)C=NC(=C(C#N)N)C#N)C MS-11345 Cc1cc(c2c(c1)occ(c2=O)/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)C(C)(C)C)C MS-11346 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C=Cc3cccc(c3)[N+](=O)[O-] MS-11347 CCOc1ccc(cc1)N/C=C(\C#N)/c2[nH]nnn2 MS-11348 CC(=O)Nc1ccc(cc1)NC=C(C#N)C#N MS-11349 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccccc3 MS-1135 C#CCSc1nc(n(n1)C(=O)c2cccs2)c3ccccc3 MS-11350 CC(C)(C)C(=O)c1ccc2c(c1)c3ccccc3s2 MS-11351 COc1ccccc1c2[nH]nc(n2)SC MS-11352 CC1(CC(=O)C(C(=O)C1)CC=C)C MS-11353 c1ccc2c(c1)c(c[nH]2)C3Nc4ccccc4C(=O)N3 MS-11354 C#CCSc1nc(n(n1)C(=O)c2cccs2)c3ccc(cc3)F MS-11355 c1ccnc(c1)Sc2ccc(cc2C=O)[N+](=O)[O-] MS-11356 c1ccnc(c1)Sc2ccc(cc2/C=N/C(=C(/C#N)\N)/C#N)[N+](=O)[O-] MS-11357 CC(C)C(=O)Nc1ccc(cc1)NC=C(C#N)C#N MS-11358 c1ccc(cc1)C2C(=O)c3ccccc3C24Nc5ccccc5C(=O)N4 MS-11359 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3cc(ccc3[N+](=O)[O-])Cl MS-1136 c1ccc2c(c1)c(ccc2Br)NC=C(C#N)C#N MS-11360 c1ccnc(c1)Sc2cccc(c2C#N)F MS-11361 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CSc3ccc(cc3)Cl MS-11362 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CCl MS-11363 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CSc3ccccn3 MS-11364 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CSC(=[NH2+])N.[Cl-] MS-11365 C#CCSC(=NN=Cc1cccs1)[NH3+].[Cl-] MS-11366 C#CCSc1[nH]c(nn1)c2cccs2 MS-11367 Cc1nccn1Cc2c(c(=O)n(n2C)c3ccccc3)Cl MS-11368 CC1(Cc2c(non2)/C(=N\OC)/C1)C MS-11369 c1cc(ccc1N)n2cnc(c2Cl)Cl MS-11370 c1cc(ccc1NC=C(C#N)C#N)n2cnc(c2Cl)Cl MS-11371 c1cc(ccc1NC=C(C#N)c2[nH]nnn2)n3cnc(c3Cl)Cl MS-11372 C#CCSC(=NN=Cc1ccco1)[NH3+].[Cl-] MS-11373 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccc(cc3)Nc4ccccc4 MS-11374 c1cc(ccc1NC=C(C#N)C#N)n2cncn2 MS-11375 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)n4cncn4)C2=O MS-11376 Cc1cc(c(c(c1)Br)N/C=C(\C#N)/C(=O)C(C)(C)C)C MS-11377 CC(C)(C)C(=O)/C(=C\Nc1ccc(cc1)n2cncn2)/C#N MS-11378 CC1(Cc2c(no[n+]2[O-])C(=O)C1)C MS-11379 c1ccc(c(c1)NC(=O)N2CCN(CC2)c3ccccn3)Br MS-1138 c1ccc(cc1)C2CC(=NO)C(=NO)C(=O)C2 MS-11380 c1ccnc(c1)Sc2ccc(cc2)N/C=C(\C#N)/c3[nH]nnn3 MS-11381 Cc1cc2c(n1c3ccc(cc3)NC(=O)C(F)(F)F)CC(CC2=O)(C)C MS-11382 CC1(C(NC(S1)c2cccs2)C(=O)O)C MS-11383 Cc1cc2c(n1c3ccc(cc3)N)CC(CC2=O)(C)C MS-11384 Cc1cc2c(n1c3ccc(cc3)NC(=S)NC)CC(CC2=O)(C)C MS-11385 Cc1cc2c(n1c3ccc(cc3)NC(=O)Nc4cccc(c4)C(F)(F)F)CC(CC2=O)(C)C MS-11386 Cc1cc2c(n1c3ccc(cc3)N/C=C(/C#N)\C(=O)C(C)(C)C)CC(CC2=O)(C)C MS-11387 Cc1cc2c(n1c3ccc(cc3)NC(=O)Nc4ccc(cc4)OC(F)(F)F)CC(CC2=O)(C)C MS-11388 Cc1ccc(cc1)C(=O)N2c3ccccc3C(=Nc4ccc(cc4)OC)C2=O MS-11389 c1ccc(cc1)C2CC(=C(C(=O)C2)C(=O)Nc3ccc(cc3)OC(F)(F)F)Nc4ccccc4 MS-11390 CC(C)CC1CC(=O)C(=CNc2ccc(cc2)n3cncn3)C(=O)C1 MS-11391 C#CCSc1nnc(n1C(=O)c2cccnc2Cl)c3ccccc3 MS-11392 Cn1c2ccccc2c3c1nc(nn3)Sc4ccc(cc4)[N+](=O)[O-] MS-11393 CCOC(=O)/C(=C/NC(C)(C)C)/C#N MS-11394 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cn2)C(F)(F)F)/C#N MS-11395 c1ccnc(c1)Cn2c(c(nn2)c3ccc4c(c3)OCO4)C#N MS-11396 Cn1c(c(nn1)c2cccc(c2)Oc3ccccc3)C#N MS-11397 CC1(CC(=O)C(C(=O)C1)N=Nc2ccc(cc2)F)C MS-11398 CC1(CC(=C(C(=NO)C1)N=Nc2ccc(cc2)F)O)C MS-11399 c1cc(cc(c1)Oc2ccc(cc2)NC=C(C#N)C#N)C(F)(F)F MS-11400 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccccc2C(=O)N MS-11401 Cc1ccc2cccc(c2n1)Oc3c(cc(cn3)C(F)(F)F)Cl MS-11402 c1cc(ccc1COc2ccc(cc2)/C=N/NC(=S)N)[N+](=O)[O-] MS-11403 c1cc(ccc1NC=C(C#N)C#N)Oc2c(cc(cn2)C(F)(F)F)Cl MS-11404 c1cc(ccc1n2c(=N)c3c(c(=O)[nH]c(n3)c4ccc5c(c4)OCO5)[nH]c2=O)Cl MS-11405 c1cc(ccc1n2c(=N)c(c([nH]c2=O)C#N)N=Cc3ccc4c(c3)OCO4)Cl MS-11406 c1ccc2cc(ccc2c1)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F MS-11407 CC1(OC(=O)C(C(=O)O1)N=Nc2ccc(c(c2)Cl)Cl)C MS-11408 Cc1cc2c(n1c3ccc(cc3)NC(=O)c4cccc(c4)C(F)(F)F)CC(CC2=O)(C)C MS-11409 CC1(Cc2c(sc(n2)NC(=O)c3cccc(c3)C(F)(F)F)C(=O)C1)C MS-11410 CCOC(=O)c1c(nc(s1)NC(=O)c2cccc(c2)C(F)(F)F)C MS-11411 c1cc(ccc1C(=O)Nc2ccc(cc2)SC(F)(F)F)Oc3c(cc(cn3)C(F)(F)F)Cl MS-11412 c1ccc2c(c1)C(=NNC(=O)COc3ccc(cc3)[N+](=O)[O-])C(=O)N2 MS-11413 Cc1cc(ccc1OCC(=O)NN=C2c3ccccc3NC2=O)Cl MS-11414 CC1(CC(=C(C(=O)C1)C(=O)Nc2cccc(c2)C(F)(F)F)NCc3ccccc3)C MS-11415 CC1(CC(=CC(=O)C1)NCCc2ccc(c(c2)OC)OC)C MS-11416 CC1(CC(=C(C(=O)C1)C(=O)Nc2cccc(c2)C(F)(F)F)NCCc3ccc(c(c3)OC)OC)C MS-11417 CC1(CC(=C(C(=O)C1)C(=O)Nc2ccccc2)NCCc3ccc(c(c3)OC)OC)C MS-11418 c1ccc2c(c1)C(=O)C(=CNc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C2=O MS-11419 CNc1nc(cs1)c2ccccc2 MS-1142 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3ccccc3Cl)C2=O MS-11420 CC1=NN(C(=O)C1=Cc2c(cc(cc2OC)OC)OC)c3ccccc3 MS-11421 Cc1ccc(cc1)C(=O)N2c3ccccc3C(=O)C2=O MS-11422 COC(=O)c1c(ccs1)NC=C(C#N)C#N MS-11423 CC(C)(C)C(=O)/C(=C\Nc1cccc(c1)C(F)(F)F)/C#N MS-11424 CC(C)(C)C(=O)C(=CNc1ccc(cc1)[N+](=O)[O-])C#N MS-11425 CCOC(=O)/C(=C/c1ccccc1Cl)/C#N MS-11426 CC\1=NN(C(=O)/C1=C\c2ccc(cc2)Cl)c3ccccc3 MS-11427 CC(C)(C)C(=O)/C(=C/c1ccc(c(c1)OC)OC)/C#N MS-11428 c1ccc(cc1)C(=O)NC(=S)Nc2ncccn2 MS-11429 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)F MS-11431 c1ccc(cc1)C2CC(=O)/C(=C/Nc3ncccn3)/C(=O)C2C#N MS-11432 Cc1cc(ccc1F)c2cc3c([nH]2)CC(CC3=O)(C)C MS-11433 c1ccc(cc1)N2CCN(CC2)C3=CC(=O)CCC3 MS-11434 CC1=CC(=NS(=O)(=O)N1)C MS-11435 CC(C)(C)c1ccc(cc1)c2csc([nH+]2)Nc3ccc(cc3)OC(F)(F)F.[Cl-] MS-11436 c1ccc(cc1)c2c(sc(n2)Nc3ccc(cc3)OC(F)(F)F)c4ccccc4 MS-11437 c1ccc(cc1)c2c(sc(n2)[NH2+]c3ccccn3)c4ccccc4.[Cl-] MS-11438 c1ccc(cc1)NC(=O)Nc2cccc(c2)F MS-11439 c1ccc(cc1)NC(=O)Nc2ccc(cc2)Cl MS-11440 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=S)NC3CC3 MS-11441 c1ccc(cc1)n2c(nnc2S)c3cccc(c3)Cl MS-11444 CCn1c(nnc1S)c2ccc(cc2)F MS-11445 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)[N+](=O)[O-])c3ccccc3 MS-11446 COc1cc(ccc1OCc2ccccc2)C(=O)OC MS-11448 COc1cc(ccc1OCc2ccccc2)C(=O)O MS-11449 CN(CCc1ccccc1)C2CCCCC2 MS-1145 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)[N+](=O)[O-])Cl MS-11451 CC(C)Oc1ccc(cc1)S(=O)(=O)CC#N MS-11452 CC(C)Oc1ccc(cc1)S(=O)(=O)C/C(=N/O)/N MS-11453 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc3c(c2)OCO3)CC(=O)OC MS-11454 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc(cc2)SC(F)(F)F)CC(=O)O MS-11455 COc1cc(c(cc1OC)S(=O)(=O)N2CCSCC2)CC(=O)OC MS-11456 COc1cc(c(cc1OC)S(=O)(=O)N2CCOCC2)CC(=O)O MS-11457 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc(cc2)C(F)(F)F)CC(=O)O MS-11458 CCOC(=O)c1csc(n1)Nc2ccc(cc2)OC MS-11459 CC(C(=O)NN)S(=O)(=O)c1ccccc1 MS-11460 c1ccc(c(c1)NC(=O)N)F MS-11461 COc1cccc(c1)C(=O)NN MS-11462 COc1ccc(cc1O)/C=C/C(=O)O MS-11465 c1cc(sc1)CNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-11466 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C MS-11467 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)S(=O)(=O)Nc4ncccn4)C2=O MS-11468 Cc1cc(nc(n1)NC(=O)/C=C/c2ccccc2)C MS-11469 CN(C/C=C/c1ccccc1)C2CCCCC2 MS-1147 COc1cc(ccc1OCc2ccc(cc2)[N+](=O)[O-])C=C3C(=O)c4ccccc4C3=O MS-11470 COc1ccc(cc1OC)/C=C\2/c3ccccc3NC2=O MS-11471 CC1CC(=CC(=O)C1)Nc2ccccc2I MS-11472 c1ccc(cc1)N(C2CCCCC2)C(=O)CCCCl MS-11473 COc1cccc(c1)CC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5Br MS-11474 c1ccc(cc1)C2=NC(C(=O)N(c3c2cccc3)CC(=O)c4ccccc4F)NC(=O)Cc5cccc(c5)C(F)(F)F MS-11475 c1ccc(cc1)C2=NC(C(=O)N(c3c2cccc3)CC(=O)c4ccccc4C(F)(F)F)NC(=O)Nc5cccc(c5)Cl MS-11476 c1ccc2cc(ccc2c1)/C=C/C(=O)O MS-11477 CC(C)c1ccc(cc1)/C=C/C(=O)OC MS-11478 COC(=O)CSc1c(cc(cn1)C(F)(F)F)Cl MS-11479 c1ccc2c(c1)nnn2N MS-1148 CC1(CC(=O)C(C(=O)C1)CC(=O)c2ccccc2)C MS-11481 c1cc(cc(c1)Br)NC(=O)N MS-11483 c1cc(c(cc1Cl)Cl)C(=O)NN MS-11484 COC(=O)c1cccc(c1)NC(=S)N MS-11492 c1ccc(cc1)C(=O)/C=C/c2ccc(cc2)Cl MS-11493 c1ccc(cc1)C(=O)/C=C/c2ccc(cc2)O MS-11494 COc1c(c(cc(c1)/C=N/N=C/c2cc(c(c(c2)OC)O)OC)OC)O MS-11540 CCc1cccc(c1NC(=S)N)CC MS-11541 Cc1ccc(c(c1)C)NC(=S)N MS-11542 c1cc(cc(c1)O)NC(=S)N MS-11543 c1ccc(cc1)CCNC(=S)N MS-11544 COc1ccc(cc1NC(=S)N)Cl MS-11545 COc1cc(cc(c1C=O)OC)OCc2ccccc2 MS-11547 c1cc(ccc1NC(=S)N)Br MS-11548 Cc1cccc(c1NC(=S)N)C MS-11549 C1CCC(=NNC(=S)N)C1 MS-11550 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)CC(CO)O)N MS-1158 c1ccc2c(c1)c3c([nH]2)CNC(C3)C(=O)O MS-1161 C1CSC(N1)C(=O)O MS-1162 c1ccc(cc1)[C@@H]2N[C@@H](CS2)C(=O)O MS-1164 CCOC(=O)C(=C(Nc1ccccc1F)SCc2ccc(c(c2)Cl)Cl)C(=O)OCC MS-1166 CC1(C(=O)Nc2ccccc2N1)C MS-1167 CCOC(=O)C(=C(Nc1ccccc1F)SCc2ccc(cc2)C(C)(C)C)C(=O)OCC MS-1169 c1ccc(cc1)OP(=O)(CCCCN2C(=O)c3ccccc3C2=O)Oc4ccccc4 MS-1176 COC(=O)C(Cc1c[nH]cn1)N.Cl MS-1179 CC(C)CC(NC(c1ccccc1)c2ccccc2)P(=O)O MS-1180 CC1C(=O)Nc2ccccc2N1C(=O)c3ccc(c(c3)Cl)Cl MS-1182 CCOC(=O)C(=C(Nc1ccccc1F)SCC(=O)c2ccc(cc2)C(F)(F)F)C(=O)OCC MS-1184 CCOC(=O)C(=C(Nc1ccccc1F)SCC(=O)c2ccccc2)C(=O)OCC MS-1185 COc1ccc(c(c1)S(=O)(=O)N2CCN(CC2)c3ncccn3)OC MS-1186 Cc1cc(ccc1F)/N=C\2/NCCS2 MS-1187 c1cc(c(cc1/N=C\2/NCCS2)Cl)Cl.Cl MS-1188 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ncccn3 MS-1189 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ncccn3 MS-1190 c1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-1191 c1cnc(nc1)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] MS-1192 c1cc(c(nc1)N2CCN(CC2)c3ncccn3)[N+](=O)[O-] MS-1193 CC1C(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)C(C)(C)C MS-1196 CC1C(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)F MS-1197 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ncccn3 MS-1198 c1cnc(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)C(F)(F)F MS-1199 CCCCc1ccccc1OCC(=O)Nc2nccs2 MS-1203 COc1ccc(cc1)COc2c(cc(cc2Cl)C(=O)OC)Cl MS-1204 CC(C)(C)c1ccc(cc1)COc2c(cc(cc2Cl)C(=O)OC)Cl MS-1205 Cc1cc(ccc1Oc2ccccc2C(=O)CC#N)Cl MS-1206 CCCCc1ccccc1OCC(=O)N(c2ccccc2)C(C)C MS-1207 Cc1ccc(c(c1)C(=O)Nc2cccnc2Cl)[N+](=O)[O-] MS-1209 c1ccc(cc1)CSC2=NCCCN2.Br MS-1214 c1ccc(cc1)CSC2=NCCCN2S(=O)(=O)c3ccc(cc3)F MS-1215 c1ccc2c(c1)C(=O)N(S2(=O)=O)Cn3ccnc3 MS-1218 c1ccc2c(c1)C(=O)N(S2(=O)=O)Cn3cncn3 MS-1219 C1CN=C2N(C1)C(=O)CS2 MS-1220 c1cc(ccc1CSC2=NCCCN2)Cl.Br MS-1221 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCCN=C2SCc3ccccc3 MS-1222 CC(C)(C)c1ccc(cc1)C(=O)N2CCCN=C2SCc3ccc(cc3)Cl MS-1225 c1cc(ccc1CSC2=NCCCN2C(=O)c3ccc(cc3)C(F)(F)F)Cl MS-1226 c1cc(ccc1/C=c/2\c(=O)n3c(=NCCC3)s2)Cl MS-1228 c1cc2c(cc1/C=c/3\c(=O)n4c(=NCCC4)s3)OCO2 MS-1229 COc1cc(ccc1O)/C=c\2/c(=O)n3c(=NCCC3)s2 MS-1230 c1cc(ccc1/C=c/2\c(=O)n3c(=NCCC3)s2)F MS-1231 C[N+]1=C2N(CCC1)C(=O)CS2.[I-] MS-1232 CCOC(=O)C[N+]1=C2N(CCC1)C(=O)CS2.[Br-] MS-1234 c1cc(sc1)/C=c/2\c(=O)n3c(=NCCC3)s2 MS-1235 COC(=O)c1ccccc1NC(=O)NCc2cccnc2 MS-1236 COC(=O)c1ccccc1NC(=O)NCc2ccc(cc2)F MS-1239 CC(C)N(c1ccccc1)C(=O)Nc2ccccc2C(=O)OC MS-1240 COC(=O)c1ccccc1NC(=O)Nc2nccs2 MS-1241 COC(=O)c1ccccc1NC(=O)Oc2ccc(cc2)F MS-1242 CCOC(=O)CSc1[nH]c2ccc(cc2n1)C.Br MS-1243 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)c3cccnc3Cl MS-1244 CCOC1c2c(ccc(c2OC1(C)C)NC(=O)Nc3ccc(cc3)Cl)C MS-1246 CCOC1c2c(ccc(c2OC1(C)C)NC(=O)Nc3ccccc3)C MS-1247 CC(C)c1ccc(cc1)OC(=O)Nc2ccccc2C(=O)OC MS-1249 c1cc(c(nc1)Cl)C(=O)Nc2nccs2 MS-1250 Cc1cc(nc(n1)NC(=O)c2cccnc2Cl)C MS-1251 Cc1ccc2c(c1)nc([nH]2)SCc3ccccc3 MS-1253 CC(=O)CSCC(=O)OC MS-1254 Cc1ccc2c(c1)nc([nH]2)SCC(=O)N3CCOCC3 MS-1255 Cc1ccc2c(c1)nc([nH]2)SCC(=O)N3CCCCC3 MS-1256 COc1ccc(cc1)N2CC(CC2=O)C(=O)OC MS-1257 COc1ccc(cc1)N2CC(CC2=O)C(=O)O MS-1258 Cc1cc(ccc1C(C)C)N2CC(CC2=O)C(=O)O MS-1259 Cc1cc(ccc1C(C)C)NCC(CC(=O)O)C(=O)O MS-1260 Cc1cc(ccc1C(C)C)N2CC(CC2=O)C(=O)Nc3ccc(cc3)C(F)(F)F MS-1261 Cc1cc(ccc1C(C)C)N2CC(CC2=O)C(=O)Nc3ccc(cc3)C(C)(C)C MS-1262 Cc1cc(ccc1F)NC(=O)C2CC(=O)N(C2)c3ccc(c(c3)C)C(C)C MS-1263 COc1ccc(cc1)N2CC(CC2=O)COS(=O)(=O)C MS-1267 CCc1ccc(cc1)OCCOS(=O)(=O)C MS-1269 C/C(=N/Nc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/CSCC(=O)OC MS-1270 COC(=O)c1ccc(cc1)OCC(F)(F)F MS-1272 c1cc(ccc1C(=O)O)OCC(F)(F)F MS-1273 Cc1ccc(cc1)Oc2ccc(cc2)C(=O)OC MS-1274 Cc1cc(ccc1C(C)C)N2CC(CC2=O)C(=O)Nc3nccs3 MS-1275 Cc1cc(ccc1C(C)C)N2CC(CC2=O)C(=O)NCc3cccnc3 MS-1276 Cc1ccc(cc1)Oc2ccc(cc2)C(=O)NCc3ccncc3 MS-1279 Cc1ccc(cc1)Oc2ccc(cc2)C(=O)NCc3cccs3 MS-1280 c1cc(ccc1C(=O)NCc2ccncc2)OCC(F)(F)F MS-1281 CCOC(CNC(=O)c1ccc(cc1)OCC(F)(F)F)OCC MS-1282 CCOC(=O)CNC(=O)c1ccc(cc1)OCC(F)(F)F MS-1283 c1cc(ccc1C(=O)NCC#N)OCC(F)(F)F MS-1284 c1cc(sc1)CNC(=O)c2ccc(cc2)OCC(F)(F)F MS-1285 c1cc(ccc1C(=O)NCCN2CCOCC2)OCC(F)(F)F MS-1287 c1cc(ccc1C(=O)NCCCn2ccnc2)OCC(F)(F)F MS-1288 CCOC(=O)C(=Cc1cccc(c1)Oc2ccccc2)C(=O)OCC MS-1289 Cc1ccc2c(c1)nc([nH]2)SCC(=O)NCC=C MS-1293 c1ccc(cc1)c2c3ccccc3c(=O)[nH]n2 MS-1294 CCc1ccc(s1)C(=O)c2ccccc2C(=O)O MS-1295 Cc1ccc2c(c1)nc([nH]2)SCC(=O)NCc3ccc(cc3)Cl MS-1296 CCOC(=O)Cn1c(=O)c2ccccc2c(n1)c3ccccc3 MS-1297 Cc1ccc(cc1)CNC(=O)CSc2[nH]c3ccc(cc3n2)C MS-1298 CCOC(=O)C(C)n1c(=O)c2ccccc2c(n1)c3ccccc3 MS-1299 Cc1ccc2c(c1)nc([nH]2)SCC(=O)NCc3cccc(c3)OC MS-1301 Cc1ccc2c(c1)nc([nH]2)SCC(=O)NCc3ccc(cc3)F MS-1302 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)CC(=O)O MS-1305 Cc1cc(ccc1C(C)C)NC2=C(C(=O)c3ccccc3C2=O)Cl MS-1306 c1ccc2c(c1)C(=O)c3c4ccc(cc4oc3C2=O)O MS-1308 Cc1cc(ccc1C(C)C)N(C2=C(C(=O)c3ccccc3C2=O)N4CCOCC4)C(=O)C MS-1310 Cc1cc(ccc1C(C)C)N(C2=C(C(=O)c3ccccc3C2=O)N4CCCCC4)C(=O)C MS-1311 Cc1cc(ccc1C(C)C)N(C2=C(C(=O)c3ccccc3C2=O)N4CC(OC(C4)C)C)C(=O)C MS-1312 CC(=C)CN1C(=O)C2C=CC=CC2C(=N1)c3ccccc3 MS-1315 Cc1cc(ccc1C(C)C)N(C2=C(C(=O)c3ccccc3C2=O)N4CCCC4)C(=O)C MS-1316 c1ccc(cc1)C2=NN(C(=O)C3C2C=CC=C3)Cc4ccc(cc4)F MS-1317 CC(c1ccccc1Cl)C(=O)NC MS-1318 CC(C(=O)O)N(c1ccc(cc1)F)C(=O)c2ccccc2 MS-1320 c1ccc(cc1)C(=O)NC2CCCCO2 MS-1322 Cc1cc(cc(c1)Oc2[nH]nnn2)C MS-1323 CCC(C)c1ccc(cc1)Oc2cccc(c2)C(=O)OCC MS-1324 CCOC(=O)Cn1c(=O)c2ccccc2c(n1)c3ccc(cc3)OC MS-1325 C1CCOC(C1)ON2C(=O)CCC2=O MS-1326 CC(C)(C)N(c1ccccc1)NC(=O)c2ccccc2 MS-1327 CCOC(=O)c1cccc(c1)Oc2ccc(cc2)SC MS-1328 C#CC(=O)Nc1ccccc1 MS-1329 c1cc(ccc1C#N)C2CCC(=O)CC2=O MS-1330 CCCC(=O)C1=C(CCC(C1=O)c2cccc(c2)Oc3ccccc3)O MS-1331 C=CCN(CC=C)C1=NS(=O)(=O)c2c1cccc2 MS-1332 C=CCOc1cccc(c1)OCC=C MS-1333 CCOC(=O)CC(=O)Nc1nc(cc(n1)C)C MS-1335 CNC(=S)NNC(=O)c1ccccc1F MS-1336 c1cc2c(cc1C(F)(F)F)ncc(n2)Cl MS-1337 Cn1c(n[nH]c1=S)c2ccccc2F MS-1338 Cn1c(nnc1SCc2ccc(cc2)F)c3ccccc3F MS-1341 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)CC(=O)NCc4ccc(cc4)Cl MS-1342 Cc1ccc(cc1)CNC(=O)Cn2c(=O)c3ccccc3c(n2)c4ccccc4 MS-1343 c1ccc(cc1)CNC(=O)Cn2c(=O)c3ccccc3c(n2)c4ccccc4 MS-1344 Cc1ccc(cc1)CSc2nnc(n2C)c3ccccc3F MS-1345 Cn1c(nnc1SCC(=O)O)c2ccccc2F MS-1346 CNC(=S)NNC(=O)c1cccc(c1)C(F)(F)F MS-1348 Cn1c(n[nH]c1=S)c2cccc(c2)C(F)(F)F MS-1349 c1cc(c(nc1)Cl)C(=O)Nc2cc(ccc2O)Cl MS-1350 c1cc(c(nc1)Sc2ccc(cc2)Cl)C(=O)O MS-1351 Cc1ccc(cc1)Oc2c3ccccc3c(nn2)c4ccccc4 MS-1354 c1ccc(cc1)c2c3ccccc3c(nn2)Oc4cccc(c4)C(F)(F)F MS-1356 c1cc(cnc1)CNC(=O)c2cccnc2Sc3ccc(cc3)Cl MS-1357 c1ccc(cc1)C2CCN(CC2)Cc3ccc(cc3)Cl MS-1358 Cc1ccc2c(c1)nc([nH]2)SCC(=O)NCc3ccc(cc3)OC MS-1359 Cc1ccc(cc1)CSc2nnc(n2C)c3cccc(c3)C(F)(F)F MS-1360 CC[NH+](CC)CC.c1cc(c(c(c1)F)C(=S)[S-])F MS-1361 CCOC(=O)C(CC(=O)N1CCN(CC1)c2cccc(c2)C(F)(F)F)C(=O)OCC MS-1362 COc1ccc(cc1)CNC(=O)c2cccnc2Sc3ccc(cc3)Cl MS-1364 c1cc(c(c(c1)F)n2c(csc2=S)CCl)F MS-1365 c1cc(c(c(c1)F)n2c(csc2=S)CN3CCOCC3)F MS-1366 c1cc(c(c(c1)F)n2c(csc2=S)CN3CCCCC3)F MS-1368 CC1CN(CC(O1)C)Cc2csc(=S)n2c3c(cccc3F)F MS-1369 c1cc(c(c(c1)F)n2c(csc2=S)CN3CCCC3)F MS-1370 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCc3cccnc3 MS-1371 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCCn3ccnc3 MS-1372 CC[NH+](CC)CC.c1cc(c(c(c1NC(=S)[S-])F)F)F MS-1374 Cc1ccc(cc1)OCc2csc(=S)n2c3c(cccc3F)F MS-1375 c1cc(c(c(c1)F)n2c(csc2=S)COc3ccc(cc3)Cl)F MS-1378 Cc1ccc(c(c1)OCc2csc(=S)n2c3c(cccc3F)F)Cl MS-1379 c1cc(cc(c1)OCc2csc(=S)n2c3c(cccc3F)F)C(F)(F)F MS-1380 c1cc(cc(c1)F)OCc2csc(=S)n2c3c(cccc3F)F MS-1381 c1ccc(cc1)CNCc2csc(=S)n2c3c(cccc3F)F MS-1382 CCOC(=O)Cc1c2ccccc2[nH]c1C(=O)O MS-1385 CC1(c2cc(ccc2C(=O)O1)Oc3ccc(cc3Cl)C(F)(F)F)C MS-1387 CC(C)(C)C(=O)/C(=C/N1CCCC1)/C#N MS-1388 Cc1ccc(s1)CNc2cnccn2 MS-1389 CC(=O)Oc1ccc(cc1)Nc2cccc(c2C#N)Cl MS-1390 c1ccc(c(c1)NC(=O)c2cccnc2)Cl MS-1393 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(Cc2ccc(s2)C)c3cnccn3 MS-1395 c1ccc(cc1)c2csc3c2ccc(c3)Cl MS-1397 c1cc(ccc1c2c(c(on2)N)C#N)Br MS-1398 c1ccc(cc1)c2nc(cc(n2)Oc3cccc(c3)C(F)(F)F)Oc4cccc(c4)C(F)(F)F MS-1399 CSc1nnc(nn1)SC MS-1400 c1c(cc(c(c1Cl)n2c(cc(n2)C#N)N)Cl)C(F)(F)F MS-1402 Cc1c(c(=O)n2n1c(c(c2=O)Cl)C)Cl MS-1404 Cc1c(c(=O)n2n1c(=O)c(c2C)Cl)Cl MS-1405 Cc1c(c(n(n1)C)Oc2cccc(c2)Cl)C#N MS-1406 Cc1c(c(n(n1)C)Oc2ccc(cc2)Cl)C#N MS-1407 Cc1c(c(n(n1)C)Oc2cccc(c2)C(F)(F)F)C#N MS-1408 C(=N/O)\c1c(nc(s1)Cl)Cl MS-1409 c1cc(cc(c1)Cl)NC(=O)CS MS-1412 C1CCN/C(=N/C#N)/C1 MS-1413 C1C/C(=N\C#N)/NC1 MS-1414 c1cc(cc(c1)Oc2cccc(n2)C(=O)O)C(F)(F)F MS-1415 COC(=O)c1cccc(n1)Oc2cccc(c2)C(F)(F)F MS-1416 c1cc(ccc1C(=O)Nc2nc(c(s2)C#N)Cl)Br MS-1418 c1cc(cc(c1)Br)C(=O)Nc2nc(c(s2)C#N)Cl MS-1419 c1cc(c(cc1C(=O)Nc2nc(c(s2)C#N)Cl)Cl)Cl MS-1420 c1cc(c(cc1C(=O)Nc2nc(c(s2)C#N)Cl)F)F MS-1421 CC1C(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)OC(=O)C MS-1422 c1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(c(ns2)Cl)C#N MS-1423 c1cc(ccc1c2c(c(on2)NC(=O)c3ccc(cc3)Cl)C#N)Br MS-1425 c1cc(ccc1Oc2ccc(cn2)C=O)F MS-1426 c1cc(ccc1C(=O)Nc2ccc(nc2)Cl)F MS-1427 c1cc(ncc1/C=C/2\C(=O)NC(=O)S2)Cl MS-1428 c1cc(ccc1Oc2ccc(cn2)/C=C/3\C(=O)NC(=O)S3)F MS-1429 c1ccc2c(c1)[nH]c(n2)/N=C/c3cccs3 MS-1431 CSc1nc2ccccc2s1 MS-1432 C[n+]1ccc(cc1)CNC(=O)c2cccc(c2)Oc3ccccc3.[I-] MS-1435 CCCCNC(=O)Oc1ccc(cc1)C(=O)N2c3ccccc3NC(=O)C2C MS-1436 CC1C(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)OC(=O)NC MS-1437 CC1C(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)O MS-1438 CN1C(=O)/C(=C\c2ccc(cc2)Br)/SC1=O MS-1440 CSc1nnc(nn1)NCc2cccnc2 MS-1442 c1cc(ccc1CO/N=C/c2ccc(nc2)Oc3ccc(cc3)F)Br MS-1446 Cc1ccccc1CO/N=C/c2ccc(nc2)Oc3ccc(cc3)F MS-1447 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)OC4C=CC(O4)n5ccc(=O)[nH]c5=O MS-1452 c1cc(cc(c1)Oc2cccc(n2)C(=O)N)C(F)(F)F MS-1454 c1cc(cc(c1)Br)C(=O)Nc2ccc(nc2)Cl MS-1458 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(nc2)Cl MS-1459 c1cc(ccc1C(=O)Nc2ccc(nc2)Cl)C(F)(F)F MS-1461 CC(C)(C)Nc1ccccc1 MS-1462 CSC1=NC(=O)/C(=C/c2ccc(cc2)F)/S1 MS-1463 c1cc(ccc1/C=C/2\C(=O)N=C(S2)S)F MS-1464 CC(C)(C)N(c1ccccc1)S(=O)(=O)c2ccc(cc2)C(F)(F)F MS-1465 CC(C)(C)N(c1ccccc1)S(=O)(=O)c2ccc(cc2Cl)Cl MS-1466 CN(C)C1=NC(=O)/C(=C\c2ccc(cc2)F)/S1 MS-1467 c1cc2c(cc1/C=C/3\C(=O)N=C(S3)S)OCO2 MS-1469 CNC(=O)Oc1cc(on1)CCl MS-1470 CCCCNC(=O)Oc1cc(on1)CCl MS-1471 c1cc(cc(c1)Cl)NC(=O)Oc2cc(on2)CCl MS-1472 c1cc(c(cc1NC(=O)Oc2cc(on2)CCl)Cl)Cl MS-1473 CC(=O)Oc1ccc(cc1)/C=C\2/C(=O)N=C(S2)S MS-1475 CN(C)C1=NC(=O)/C(=C\c2ccc3c(c2)OCO3)/S1 MS-1476 c1cc(ccc1/C=C\2/C(=O)N=C(S2)S)O MS-1478 COc1cc(c(cc1Br)OC)CC(=O)O MS-1479 CC(C)(C)N(c1ccccc1)NS(=O)(=O)c2ccc(cc2)F MS-1480 COc1cc(c(cc1Br)O)C(=O)CCl MS-1481 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCN3CCCCC3 MS-1482 c1cc(cc(c1)OCc2ccc(cc2)C(F)(F)F)/C=C/C(=O)N3CCC(CC3)c4cccc(c4)C(F)(F)F MS-1485 c1cc(nc(c1[N+](=O)[O-])N2CC(CC2C(=O)O)O)Cl MS-1488 Cc1cc(ccc1C(C)C)NS(=O)(=O)N(C)C MS-1490 CCOC(=O)CSC1=NC(=O)/C(=C\c2ccc(cc2)OC(=O)C)/S1 MS-1491 CN(C)S(=O)(=O)Nc1cc(ccc1F)F MS-1493 CN(C)S(=O)(=O)Nc1ccc(cc1F)F MS-1494 CN(C)S(=O)(=O)Nc1cc(cc(c1)F)F MS-1495 C=CCNC1=NC(=O)/C(=C\c2ccc3c(c2)OCO3)/S1 MS-1496 CC(=O)Nc1cc(ccc1OC)OC MS-1499 CN(C)S(=O)(=O)Nc1c(cccc1F)F MS-1500 COC(=O)c1cccn1C(=O)c2ccc(cc2)Cl MS-1501 COC(=O)c1cccn1S(=O)(=O)c2ccc(cc2)F MS-1502 c1cc(cc(c1)Oc2cc(nc(n2)N)Oc3cccc(c3)C(F)(F)F)C(F)(F)F MS-1503 CC(C)(C)c1ccc(cc1)Oc2cc(nc(n2)N)Oc3ccc(cc3)C(C)(C)C MS-1504 c1cc(ccc1Oc2cc(nc(n2)N)Oc3ccc(cc3)F)F MS-1505 c1cc(ccc1Oc2cc(nc(n2)N)Oc3ccc(cc3)Br)Br MS-1506 c1cc(n(c1)S(=O)(=O)c2ccc(cc2)F)C(=O)O MS-1507 CC(C)(C)c1ccc(cc1)Oc2cc(nc(n2)NS(=O)(=O)c3ccc(cc3)F)Oc4ccc(cc4)C(C)(C)C MS-1508 CCOC(=O)c1ccc(cc1)Oc2ccc(cn2)C(F)(F)F MS-1510 c1cc(ccc1C(=O)O)Oc2ccc(cn2)C(F)(F)F MS-1511 CC(C)(C)c1ccc(cc1)Oc2cc(nc(n2)NS(=O)(=O)c3ccc(cc3)OC)Oc4ccc(cc4)C(C)(C)C MS-1512 CCCCN(c1ccccc1)S(=O)(=O)N(C)C MS-1515 c1cc(c(cc1Br)Br)NC(=O)CCl MS-1516 c1ccc(cc1)N2CCN(CC2)C(=O)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F MS-1517 COc1ccc(cc1)N2CCN(CC2)C(=O)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F MS-1518 Cc1ccccc1N2CCN(CC2)C(=O)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F MS-1519 c1cc(ccc1C(=O)N2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])Oc4ccc(cn4)C(F)(F)F MS-1520 c1cc(c(cc1Br)Br)NC(=O)CN2CCOCC2 MS-1521 c1cc(c(cc1Br)Br)NC(=O)CN2CCN(CC2)C=O MS-1522 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCN3CCOCC3 MS-1523 CCN(CC)Cc1cc(ccc1O)NC(=O)C MS-1527 c1cc(c(nc1)NCc2ccc(cc2)F)[N+](=O)[O-] MS-1528 c1cc(ccc1/C=C\2/NC(CS2)C(=O)O)Br MS-1529 Cc1cccc(c1)C2(CCCC2)C#N MS-1533 c1cc(c(nc1)NCc2ccc(cc2)F)N MS-1535 c1cc(ncc1/C=C/2\C(=O)NC(=S)S2)Cl MS-1536 c1ccc(c(c1)/C=C/2\C(=O)NC(=S)S2)F MS-1537 CSC1=NC(=O)/C(=C\c2ccccc2F)/S1 MS-1538 COC(=O)c1cccn1CC#N MS-1539 COC(=O)C1N2C(CS1)C(=O)N(C2=S)c3ccccc3Br MS-1546 COc1ccc(cc1)N2CCN(CC2)CC(=O)N3C(CSC3C(=O)OC)C(=O)OC MS-1548 COC(=O)C1CSC(N1C(=O)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-])C(=O)OC MS-1549 CC1CN(CC(O1)C)CC(=O)N2C(CSC2C(=O)OC)C(=O)OC MS-1550 CCOC(=O)c1c2c(sc1NC(=O)COc3ccc(cc3)F)CCCC2 MS-1552 CC(C)(C)c1nnc(s1)NC(=O)COc2ccc(cc2)F MS-1553 Cc1nc(cc(n1)Cl)Cl MS-1554 c1cc(=O)oc2c1cc(cc2)/[N+](=N/C#N)/[O-] MS-1555 c1cc(c(cc1F)F)NC(=O)CC#N MS-1556 COC(=O)c1cccnc1C#N MS-1559 c1cc(sc1C2NC(CS2)C(=O)O)[N+](=O)[O-] MS-1560 C1C(CN1C(=O)CC(=O)O)C(=O)O MS-1561 Cc1ccc(cc1)C(=O)C(n2cncn2)SC(C)(C)C MS-1562 CC1(CC(=O)C(C(=O)C1)/C=N/c2ccccc2)C MS-1564 c1cc(ccc1C2N(C(=O)CS2)c3cnccn3)Cl MS-1565 CN1c2ccc(cc2SCC1=O)F MS-1567 CSc1cc(nn1c2ccc(cc2)F)c3ccc(c(c3)Cl)Cl MS-1568 C/C(=N\OCc1ccc(cc1)[N+](=O)[O-])/c2ccccn2 MS-1570 Cc1cccc(c1)C2(CCCC2)C(=O)O MS-1572 C/C(=N/OCc1ccc(cc1)Br)/c2ccccn2 MS-1573 CCCO/C(=N\c1ccc(cc1Cl)Cl)/c2cncn2C MS-1574 c1cc(sc1)C(C#N)Nc2ccc(c(c2)Cl)F MS-1575 C/C(=N/O)/c1ccccn1 MS-1578 c1ccc(cc1)Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F MS-1579 c1cc(ccc1OCC(=O)NN2C(=O)CSC2=S)F MS-1580 CSC(=CC(=O)c1ccc(cc1Cl)Cl)SC MS-1581 CSC(=CC(=O)c1cccc(c1)Br)SC MS-1582 c1ccc(cc1)OCC(=O)NN2C(=O)CSC2=S MS-1583 CSC(=CC(=O)c1ccccc1Cl)SC MS-1584 CSc1ccccc1c2cc(no2)c3ccccc3 MS-1590 CC(C)(C)c1nnc(s1)NC(=O)COc2cc(cc(c2)Cl)Cl MS-1591 COc1cccc(c1)c2nc3ccccc3s2 MS-1599 c1ccc(c(c1)c2nc3ccccc3s2)Cl MS-1603 c1ccc2c(c1)nc(s2)c3cccc(c3)Cl MS-1604 c1ccc2c(c1)nc(s2)c3ccc(cc3)Cl MS-1605 c1ccc2c(c1)nc(s2)c3cccc(c3)F MS-1606 c1ccc2c(c1)nc(s2)c3cccc(c3)C(F)(F)F MS-1607 C/C(=N\OCc1ccc(cc1)C(F)(F)F)/c2ccccn2 MS-1609 COC(=O)C1N2C(CS1)C(=O)N(C2=O)c3cccc(c3)Cl MS-1615 Cc1cccc(c1NC(=O)N2C(CSC2C(=O)OC)C(=O)OC)C MS-1616 CC(C)(C)c1ccc(cc1)Oc2cc(nc(n2)c3ccccc3)Oc4ccc(cc4)C(C)(C)C MS-1617 COC(=O)C1CSC(N1C(=O)CC#N)C(=O)OC MS-1618 CN1CNC=C1C(=O)Nc2ccc(cc2Cl)Cl MS-1619 COC(=O)C1(CCCC1=O)Cc2ccc(cc2)Cl MS-1620 CC(C)(C)NC(=O)N1C(CSC1C(=O)OC)C(=O)OC MS-1624 CC(C)C(C(=O)O)Nc1c(ccc(n1)Cl)[N+](=O)[O-] MS-1625 CC(C)C(C(=O)O)Nc1c(ccc(n1)N2CCC[C@H]2C(=O)O)[N+](=O)[O-] MS-1628 CC(C)C(C(=O)O)Nc1c(ccc(n1)NC(Cc2ccc(cc2)O)C(=O)O)[N+](=O)[O-] MS-1629 CC(=O)NN1C(=O)CSC1=S MS-1630 COc1cccc(c1)CNc2ccc(c(n2)NCC(=O)O)[N+](=O)[O-] MS-1631 c1cc(ccc1CNc2ccc(c(n2)NCC(=O)O)[N+](=O)[O-])Cl MS-1632 COc1cccc(c1)C(=O)/C(=C(/Nc2ccc(cc2F)F)\O)/C#N MS-1633 c1cc(c(c(c1)Cl)OCC(=O)/C(=C(/Nc2ccc(cc2F)F)\O)/C#N)Cl MS-1634 c1cc(c(c(c1)Cl)OCC(=O)NN2C(=O)CSC2=S)Cl MS-1635 CC(=O)N(C(=O)C)N1C(=O)/C(=C/c2ccc(cc2)Cl)/SC1=S MS-1636 CC(=O)N(C(=O)C)N1C(=O)/C(=C/c2ccc3c(c2)OCO3)/SC1=S MS-1637 CC(=O)N(C(=O)C)N1C(=O)/C(=C/c2cccc(c2)F)/SC1=S MS-1638 c1cc(cc(c1)F)/C=C/2\C(=O)N(C(=S)S2)NC(=O)CCl MS-1640 CC(C)(C)c1nnc(s1)NC(=O)c2ccc(cc2F)F MS-1643 c1c[nH]c2c1cc(cc2Br)Br MS-1644 CC(C1CC1)(C(=O)O)N MS-1645 c1cc(c(c(c1)F)CNc2c(cccn2)[N+](=O)[O-])F MS-1646 c1cc(c(nc1)NCc2ccc(c(c2)F)F)[N+](=O)[O-] MS-1649 c1cc(c(nc1)NCc2ccc(c(c2)Cl)Cl)[N+](=O)[O-] MS-1650 COC(=O)C1N2C(CS1)C(=O)N(CC2=O)Cc3ccc(c(c3)Cl)Cl MS-1652 COC(=O)C1N2C(CS1)C(=O)N(CC2=O)Cc3ccc(cc3)F MS-1654 Cc1cccc(c1)CN2CC(=O)N3C(C2=O)CSC3C(=O)OC MS-1655 Cc1cccc(c1NC(=O)N2C(CSC2C(=O)O)C(=O)O)C MS-1662 c1c(cc(c(c1C(CCl)O)N)Br)Br MS-1663 c1ccc(cc1)CCNC2=C(C(=O)c3ccccc3C2=O)Cl MS-1664 CC(=C)COc1ccc(cc1)F MS-1665 Cc1cc(on1)NC(=O)CCl MS-1667 Cc1cc(on1)NC(=O)CN2CCOCC2 MS-1668 CCC(=O)N(CCc1ccccc1)C2=C(C(=O)c3ccccc3C2=O)Cl MS-1670 CC(=O)N(CCc1ccccc1)C2=C(C(=O)c3ccccc3C2=O)Cl MS-1671 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)/C=C\3/C(=O)NC(=O)S3 MS-1673 Cc1cc(on1)NC(=O)C MS-1674 CC(=O)/N=C\1/NC(=O)/C(=C/c2cccc(c2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)/N1C MS-1678 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)/C=C/C(=O)O MS-1679 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)/C=C\3/C(=O)NC(=S)S3 MS-1680 c1ccc(cc1)COc2c3c(cccc3F)ncn2 MS-1681 COc1cccc(c1)COc2ccsc2C(=O)OC MS-1683 CC(CN1CCOCC1)(COc2ccc(cc2)F)O MS-1685 CC(CN1CCCCC1)(COc2ccc(cc2)F)O MS-1686 CCOC(=O)C(C)Oc1c2c(cccc2F)ncn1 MS-1687 CC(CN1CCCC1)(COc2ccc(cc2)F)O MS-1688 c1ccc2c(c1)c(c[nH]2)C[C@@H](C(=O)O)Nc3c(cccn3)[N+](=O)[O-] MS-1689 COC(=O)c1c(ccs1)OCCBr MS-1690 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C=O MS-1692 COc1cc(nc(n1)S(=O)(=O)C)OC MS-1693 c1cc(cc(c1)OC(F)(F)F)Oc2c(c(ncn2)Oc3cccc(c3)OC(F)(F)F)[N+](=O)[O-] MS-1694 COc1cc(nc(n1)Oc2cccc(c2)C(F)(F)F)OC MS-1695 CCOC(=O)c1ccc(cc1)Oc2nc(cc(n2)OC)OC MS-1696 c1cc(ccc1Oc2c(c(ncn2)Oc3ccc(cc3)F)[N+](=O)[O-])F MS-1697 CC(C)(C)c1ccc(cc1)Oc2c(c(ncn2)Oc3ccc(cc3)C(C)(C)C)[N+](=O)[O-] MS-1698 Cc1ccc(cc1[N+](=O)[O-])Oc2c(c(ncn2)Oc3ccc(c(c3)[N+](=O)[O-])C)[N+](=O)[O-] MS-1699 Cc1ccc(cc1Oc2c(c(ncn2)Oc3cc(ccc3C)C=O)[N+](=O)[O-])C=O MS-1700 COc1cc(nc(n1)Oc2ccc(cc2)C(=O)O)OC MS-1701 CC(=O)Nc1ccc(cc1)Oc2nc(cc(n2)OC)OC MS-1702 CCN(c1ccc(cc1)Oc2nc(cc(n2)OC)OC)C(=O)C MS-1704 CCc1ccc(cc1)Oc2cccc(c2)C=C(C(=O)OCC)C(=O)OCC MS-1706 CCc1ccc(cc1)Oc2cccc(c2)C(C[N+](=O)[O-])C(C(=O)OCC)C(=O)OCC MS-1707 CCc1ccc(cc1)Oc2cccc(c2)C3CN(C(=O)C3C(=O)OCC)O MS-1709 Cc1c(c(on1)C)C(=O)NCCc2ccccc2 MS-1710 Cc1cc(ccc1C(C)C)NS(=O)(=O)c2c(noc2C)C MS-1712 Cc1c(c(on1)C)S(=O)(=O)N(C)Cc2cccnc2 MS-1714 Cc1c(c(on1)C)S(=O)(=O)N2CCN(CC2)c3ccccc3 MS-1716 Cc1cc(ccc1N)Oc2nc(cc(n2)OC)OC MS-1717 Cc1cc(ccc1NS(=O)(=O)c2ccccc2Cl)Oc3nc(cc(n3)OC)OC MS-1718 Cc1cc(ccc1NS(=O)(=O)c2ccccc2C(=O)OC)Oc3nc(cc(n3)OC)OC MS-1719 Cc1cc(ccc1NS(=O)(=O)c2ccc(cc2)C(C)(C)C)Oc3nc(cc(n3)OC)OC MS-1720 CC(C)(C)c1ccc(cc1)c2nc3cc(ccc3c(=O)o2)Cl MS-1722 C/C=C/C(=O)NCCc1ccc(c(c1)OC)OC MS-1723 c1cc(ccc1NC(=O)OC/C=C/CO)Cl MS-1724 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2c(ncnc2Oc3cccc(c3)OC(F)(F)F)Oc4cccc(c4)OC(F)(F)F MS-1729 c1cc(cc(c1)OC(F)(F)F)Oc2c(c(ncn2)Oc3cccc(c3)OC(F)(F)F)N MS-1731 COc1ccc(cc1Oc2nc(cc(n2)OC)OC)/C=N/O MS-1732 COc1ccc(cc1Oc2nc(cc(n2)OC)OC)C=O MS-1733 CCO/N=C/c1ccc(c(c1)Oc2nc(cc(n2)OC)OC)OC MS-1734 COc1ccc(cc1Oc2nc(cc(n2)OC)OC)/C=N/OC MS-1735 CNC(=O)N1CCOC12CCCCC2 MS-1739 CCn1c(c(c(=O)c(c1c2ccc(cc2)Cl)C(=O)OC)Br)C MS-1741 c1cc(ccc1CN(Cc2ccc(cc2)F)c3ncc(cn3)[N+](=O)[O-])F MS-1743 Cc1cc(ccc1C(C)C)Nc2ncc(s2)[N+](=O)[O-] MS-1744 CC(C)(C)c1ccc(cc1)CN(Cc2ccc(cc2)C(C)(C)C)c3ncc(cn3)[N+](=O)[O-] MS-1745 c1cc(cc(c1)Br)CN(Cc2cccc(c2)Br)c3ncc(cn3)[N+](=O)[O-] MS-1746 c1cc(ccc1CN(Cc2ccc(cc2)Cl)c3ncc(cn3)[N+](=O)[O-])Cl MS-1747 c1cc(ccc1CN(Cc2ccc(cc2)C(F)(F)F)c3ncc(cn3)[N+](=O)[O-])C(F)(F)F MS-1748 c1ccc2c(c1)N(c3c(cccn3)C(=O)N2C(=O)CCl)C(=O)CCl MS-1750 Cc1cccc2c1occ2 MS-1751 Cc1ccccc1OCC(OC)OC MS-1755 C1CCC2(CC1)N(CCO2)C(=O)[C@H]3C[C@H]3C(=O)O MS-1756 Cc1ccc(cc1Cl)NC(=O)NC MS-1757 Cc1ccc(cc1Cl)NC(=O)Nc2ccc(c(c2)Cl)C MS-1758 Cc1ccc(cc1)NC(=O)N(C)C MS-1759 CC(=O)Nc1ccccc1N MS-1760 Cc1nc2ccccc2n1C MS-1761 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccnc(n2)SC MS-1764 CSc1nccc(n1)NC(=O)c2cccc(c2)Br MS-1765 CSc1nccc(n1)NC(=O)c2cccc(c2)C(F)(F)F MS-1766 CC1CNC2(O1)CCCC2 MS-1768 CC1CN(C2(O1)CCCC2)C(=O)C3CC3C(=O)O MS-1769 CC(=O)N(C)c1cccc(c1)N MS-1770 CC(C)(C)OC(=O)Nc1ccccc1N MS-1771 CC(C)(C)OC(=O)N(C)N MS-1772 CC(=O)N(C)c1ccccc1N MS-1773 CC(C)(C)OC(=O)N(C)CCN MS-1774 CC(C)(C)OC(=O)Nc1ccccc1[N+](=O)[O-] MS-1775 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCOC34CCCCC4 MS-1776 Cc1ccc(c(c1)C(=O)O)NC(=O)c2ccccc2F MS-1777 c1ccc2c(c1)c(c(c(=O)o2)[N+](=O)[O-])NCCCn3ccnc3 MS-1780 c1ccc(cc1)CCNc2c3ccccc3oc(=O)c2[N+](=O)[O-] MS-1781 c1ccc(cc1)C2CCN(CC2)c3c4ccccc4oc(=O)c3[N+](=O)[O-] MS-1782 c1ccc(cc1)CCCCNc2c3ccccc3oc(=O)c2[N+](=O)[O-] MS-1783 c1ccc2c(c1)c(c(c(=O)o2)[N+](=O)[O-])NCc3cccc(c3)F MS-1784 c1cc(ccc1CN2CCC3(C2=O)CCCC3=O)F MS-1785 c1ccc2c(c1)c(c(c(=O)o2)[N+](=O)[O-])Oc3cccc(c3)F MS-1788 c1ccc2c(c1)c(c(c(=O)o2)[N+](=O)[O-])SCC(=O)Nc3cccc(c3)Cl MS-1789 CCOC(=O)C1(CCCC1=O)CC#N MS-1790 CC(CO)(COCc1ccccc1Br)O MS-1793 c1ccc(cc1)COc2ccc(cc2)C(=O)O MS-1799 Cc1c(scn1)C(=O)Nc2cccc3c2C(CC3(C)C)C MS-1803 CC(=O)Nc1cccc(c1)[N+](=O)[O-] MS-1807 Cn1cccn1 MS-1808 CCOC(=O)c1c(c2ccccc2[nH]1)c3ccc(cc3)F MS-1809 Cc1cccc(c1)S(=O)(=O)Nc2cccc-3c2C(=O)c4c3cccc4 MS-1810 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2cccc-3c2C(=O)c4c3cccc4 MS-1811 C1CSCCC1=NO MS-1812 c1ccc2c(c1)-c3cccc(c3C2=O)NS(=O)(=O)c4ccc(cc4)F MS-1813 c1ccc2c(c1)-c3cccc(c3C2=O)NS(=O)(=O)c4ccc(cc4)Br MS-1814 c1ccc2c(c1)-c3cccc(c3C2=O)NS(=O)(=O)c4ccc(cc4)C(F)(F)F MS-1815 c1ccc2c(c1)-c3cccc(c3C2=O)NC(=O)c4ccccc4Br MS-1816 c1cc(cc(c1)Br)CON=C2CCSCC2 MS-1817 c1cc(cc(c1)F)CON=C2CCSCC2 MS-1818 CC(C)(C)c1ccc(cc1)CON=C2CCSCC2 MS-1819 COc1cccc(c1)CON=C2CCSCC2 MS-1820 c1cc2c(cc1Br)cc(c(=O)o2)C(=O)NCCN3CCOCC3 MS-1821 c1cc2c(cc1Br)cc(c(=O)o2)C(=O)NCCN3CCCCC3 MS-1822 c1ccc(cc1)CCCNC(=O)c2cc3cc(ccc3oc2=O)Br MS-1823 CCOC(=O)CNC(=O)c1cc2cc(ccc2oc1=O)Br MS-1824 COc1ccccc1N2CCN(CC2)C(=O)c3cc4cc(ccc4oc3=O)Br MS-1825 CCOC(=O)c1c(c2ccccc2[nH]1)c3ccc(cc3)C MS-1826 Cc1ccc(cc1)c2c3ccccc3n(c2C(=O)O)Cc4ccc(cc4)Br MS-1827 CC(C)(C)c1ccc(cc1)Oc2c3ccccc3nc(n2)c4ccccc4 MS-1829 c1ccc(cc1)c2nc3ccccc3c(n2)Oc4cccc(c4)OC(F)(F)F MS-1830 CCOC(=O)c1ccc(cc1)Oc2c3ccccc3nc(n2)c4ccccc4 MS-1831 c1ccc(cc1)c2nc3ccccc3c(n2)Oc4cccc(c4)Br MS-1832 c1ccc(cc1)c2nc3ccccc3c(n2)Oc4ccc(cc4)F MS-1833 c1cc-2c(cc1Cl)C(=O)c3c2c(cc(c3)Cl)Cl MS-1834 c1ccc(cc1)NNC(=O)c2cccc(c2)C(F)(F)F MS-1836 CCOC(=O)c1nc2ccccc2c(n1)Cl MS-1837 c1ccc(cc1)c2nc3ccccc3c(n2)NC(=O)c4ccc(cc4)F MS-1838 CSCCC(C(=O)O)Nc1c(ccc(n1)Cl)[N+](=O)[O-] MS-1841 c1cc(nc(c1[N+](=O)[O-])NC(CC(=O)N)C(=O)O)Cl MS-1842 CC(=O)Nc1cccc(c1)CN MS-1843 CN1C(=O)CC(=O)NC1=O MS-1844 c1ccc2c(c1)C(=O)N(C2=O)Cc3cccc(c3)[N+](=O)[O-] MS-1845 Cc1cc(n(n1)C)NC(=O)NC MS-1846 Cc1cc(n(n1)C)NC(=O)Nc2ccc(cc2F)F MS-1847 c1ccc(c(c1)C(=O)NCCO)O MS-1848 Cc1cc(n(n1)C)NC(=O)Nc2cccc(c2)C(F)(F)F MS-1849 Cc1cc(n(n1)C)NC(=O)Nc2ccccc2[N+](=O)[O-] MS-1850 c1ccc2c(c1)C(=O)N(CO2)CCO MS-1851 Cc1cc(n(n1)C)NC(=O)c2ccc(cc2)F MS-1852 c1cc(ccc1S(=O)(=O)N2CCOC23CCCCC3)Br MS-1854 c1cc(cc(c1)F)OCC2NCCS2 MS-1855 Cn1c(=O)cc([nH]c1=O)Nc2ccc(cc2)Cl MS-1856 CCc1ccc(cc1)OCCNCc2ccncc2 MS-1857 CCc1ccc(cc1)OCCNCc2cccnc2 MS-1858 CCOC(=O)c1nc2ccccc2c(n1)NCc3ccccc3C MS-1859 CCOC(=O)c1nc2ccccc2c(n1)NCc3cccc(c3)OC MS-1861 CCOC(=O)c1nc2ccccc2c(n1)NCc3cccc(c3)Cl MS-1862 CCOC(=O)c1nc2ccccc2c(n1)NCc3ccccc3F MS-1863 CC1(CN(N(C1=O)C(=O)c2ccc(cc2)C(C)(C)C)c3ccccc3)C MS-1864 CC1(CN(N(C1=O)C(=O)c2ccc(cc2)F)c3ccccc3)C MS-1865 Cc1ccccc1C(=O)N2C(=O)C(CN2c3ccccc3)(C)C MS-1866 CC1(CN(N(C1=O)C(=O)c2ccc(cc2)C#N)c3ccccc3)C MS-1868 Cn1c(=O)cc([nH]c1=O)Cl MS-1869 Cc1ccc(cc1)S(=O)(=O)N2CCOC23CCCCC3 MS-1871 CCc1ccc(cc1)OCCN2CCN(CC2)C=O MS-1872 Cc1ccc(c(c1)C)OCCOS(=O)(=O)C MS-1873 Cn1c(=O)c(c([nH]c1=O)Cl)[N+](=O)[O-] MS-1874 Cc1ccc(c(c1)C)OCCN2CCN(CC2)C=O MS-1876 CCc1ccc(cc1)OCCn2cccn2 MS-1878 Cc1ccc(c(c1)C)OCCn2cccn2 MS-1879 CC(C)(C)c1nnc(s1)NC(=O)Cc2cccc(c2)F MS-1881 c1c(nc(nc1O)C2CC2)CCl MS-1882 Cc1cc(nc(n1)CCl)O MS-1883 Cc1nc(cc(n1)O)CCl MS-1884 CCCCCCCCCOc1ccc(cc1)CCc2ccc(cc2)OCCCCCCCCC MS-1885 Cc1cc(n(n1)C)NC(=O)COc2ccc(cc2)F MS-1887 CC(=O)Nc1cccc(c1)CNCc2cccc(c2)NC(=O)C MS-1889 CC(=O)Nc1cccc(c1)CN(Cc2cccc(c2)NC(=O)C)S(=O)(=O)c3ccc(cc3)C(C)(C)C MS-1890 CC(=O)Nc1cccc(c1)CN(Cc2cccc(c2)NC(=O)C)S(=O)(=O)c3ccc(cc3)Br MS-1891 Cc1cccc(c1)S(=O)(=O)N(Cc2cccc(c2)NC(=O)C)Cc3cccc(c3)NC(=O)C MS-1892 CC(=O)Nc1cccc(c1)CN(Cc2cccc(c2)NC(=O)C)S(=O)(=O)c3ccccc3C(F)(F)F MS-1893 CCOC(=O)c1nc2ccccc2c(n1)NCC=C MS-1894 CC1(CN(N(C1=O)Cc2ccc(cc2)F)c3ccccc3)C MS-1895 Cc1cc(nc(n1)CN2CCOCC2)O MS-1896 Cc1cc(nc(n1)CN2CC(CC(C2)C)C)O MS-1897 Cc1cc(nc(n1)CN2CCC(CC2)c3ccccc3)O MS-1898 Cc1cc(c(c(c1)[N+](=O)[O-])N2CCC[C@@H]2C(=O)O)[N+](=O)[O-] MS-1899 Cc1cc(c(c(c1)[N+](=O)[O-])N2CC(C[C@@H]2C(=O)O)C)[N+](=O)[O-] MS-1900 Cc1cc(c(c(c1)[N+](=O)[O-])N2CC(C2)C(=O)O)[N+](=O)[O-] MS-1901 Cc1cc(c(c(c1)[N+](=O)[O-])NC2(CCCCC2)C(=O)O)[N+](=O)[O-] MS-1902 c1c(nc(nc1O)C2CC2)CN3CCOCC3 MS-1903 CC1CN(CC(O1)C)Cc2cc(nc(n2)C3CC3)O MS-1904 c1ccc(cc1)C2CCN(CC2)Cc3cc(nc(n3)C4CC4)O MS-1905 c1c(nc(nc1O)C2CC2)CN3CCCCC3 MS-1906 Cc1nc(cc(n1)O)CN2CCOCC2 MS-1907 Cc1nc(cc(n1)O)CN2CCCCC2 MS-1908 Cc1nc(cc(n1)O)CN2CCC(CC2)c3ccccc3 MS-1909 CC(C)c1nc(cc(n1)O)CN2CCCCC2 MS-1910 CC1CN(CC(O1)C)Cc2cc(nc(n2)C(C)C)O MS-1911 CC(C)c1nc(cc(n1)O)CN2CCOCC2 MS-1912 CC1CN(CC(O1)C)CC2COC(O2)(C)C MS-1915 CC1(OCC(O1)CN2CCOCC2)C MS-1916 CC(C)c1nc(cc(n1)O)CCl MS-1918 c1cc(ccc1CCc2ccc(cc2)O)O MS-1919 CC(=O)N1C(=O)C(CN1c2ccccc2)(C)COC(=O)C MS-1921 CC(=O)OCC1(CN(NC1=O)c2ccccc2)C MS-1922 CC(=O)OCC1(CN(N(C1=O)C(=O)c2ccc(cc2)F)c3ccccc3)C MS-1923 c1ccc2c(c1)-c3ccccc3C2C(=O)Nc4ccc(cc4)F MS-1928 c1ccc2c(c1)-c3ccccc3C2C(=O)NCc4ccc(cc4)F MS-1929 c1ccc(cc1)CCNC(=O)C2c3ccccc3-c4c2cccc4 MS-1930 c1ccc(cc1)CCCNC(=O)C2c3ccccc3-c4c2cccc4 MS-1931 CCCCCCCOC(C)C(=O)OC MS-1933 CCCCCCCOC(C)C(=O)O MS-1934 Cc1cc(ccc1C#N)OC MS-1940 c1ccc2c(c1)C(CCO2)OCc3ccc(cc3)F MS-1942 CC(C)(C)c1ccc(cc1)COC2CCOc3c2cccc3 MS-1943 c1ccc2c(c1)C(CCO2)OCc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-1944 COc1cccc(c1)COC2CCOc3c2cccc3 MS-1945 Cc1ccc(c(c1)C)COC2CCOc3c2cccc3 MS-1946 c1cc(ccc1COc2ccnc3c2ccc(c3)C(F)(F)F)F MS-1947 c1cc(ccc1Cn2ccc(=O)c3c2cc(cc3)C(F)(F)F)F MS-1948 CC(C)(C)c1ccc(cc1)COc2ccnc3c2ccc(c3)C(F)(F)F MS-1949 CCOC(=O)NC12CC3CC(C1)CC(C3)C2 MS-1950 CCCCCCCCCOc1ccc(cc1)CCc2ccc(cc2)O MS-1952 CCCCCCCCCOc1ccc(cc1)C(=O)Oc2ccc(cc2)CCc3ccc(cc3)O MS-1953 C=CCO/N=C/c1c[nH]c2c1cc(cc2)Br MS-1957 c1ccc(cc1)CO/N=C/c2c[nH]c3c2cc(cc3)Br MS-1958 CCO/N=C\c1c[nH]c2c1cc(cc2)Br MS-1961 c1cc(cc(c1)N/N=C\c2c[nH]c3c2cc(cc3)Br)C(F)(F)F MS-1963 CC(C)(C)c1ccc(cc1)Cn2c3ccccc3ccc2=O MS-1964 COc1cccc(c1)Cn2c3ccccc3ccc2=O MS-1965 c1ccc2c(c1)ccc(=O)n2Cc3cccc(c3)F MS-1966 Cc1ccc(cc1)S(=O)(=O)N2CC[C@H](C2)O MS-1967 Cc1ccc(cc1)S(=O)(=O)N2CC[C@H](C2)OS(=O)(=O)C MS-1969 c1cc(ccc1CCn2ccnc2)[N+](=O)[O-] MS-1973 c1cc(ccc1CCn2ccnc2)N MS-1974 CCOC(=O)C1=C(C2C=C(C=CC2N=C1)C)OCc3ccc(cc3)Cl MS-1979 CCOC(=O)C1=C(C2C=C(C=CC2N=C1)C)OCc3ccc(cc3)C(F)(F)F MS-1980 CCOC(=O)c1cnc2ccc(cc2c1OCc3cc(cc(c3)F)F)C MS-1981 C1C2C1C(=O)OC2=O MS-1982 CCOC(=O)C1=C(C2C=C(C=CC2N=C1)C)OCC#N MS-1983 CCOC(=O)c1cnc2c(ccc(c2c1O)C)F MS-1984 CCOC(=O)C(=CNc1cc(ccc1F)C)C(=O)OCC MS-1985 CCNc1c(cnc2c1c(ccc2F)C)C(=O)OCC MS-1987 CCOC(=O)c1cnc2c(ccc(c2c1N(C)C)C)F MS-1989 CCOC(=O)c1cnc2c(ccc(c2c1NCC=C)C)F MS-1990 c1cc(cc2c1cc[nH]2)Br MS-1991 c1cc2c(cc[nH]2)c(c1)Br MS-1992 c1cc2cc[nH]c2c(c1)Br MS-1993 c1cc2c(cc1C(=O)O)CCO2 MS-1996 c1cc2c(cc1CO)CCO2 MS-1997 CCOC(=O)c1cnc2c(ccc(c2c1NCCOC)C)F.Cl MS-1998 CCOC(=O)CN1CCN(CC1)C=O MS-1999 C1CN(CCN1CC(=O)N2CCOCC2)C=O MS-2000 CC(=O)C(=C1Nc2ccccc2O1)C(=O)C MS-2003 COC(CNc1cc(=O)oc2c1cccc2)OC MS-2004 c1ccc2c(c1)c3c(cc[nH]3)c(=O)o2 MS-2005 c1cc(ccc1C(=O)CC(C#N)c2ccc3c(c2)OCO3)F MS-2006 C=C(c1ccc(cc1)Cl)c2ccc3c(c2)CCO3 MS-2008 CCOC(=O)/C=C/c1ccc(cc1)O MS-2009 c1cc(ccc1/C=C/CO)O MS-2010 CSC(=S)NCc1cccnc1 MS-2011 c1cc(sc1)CN2CC(CC2=O)C(=O)O MS-2012 CSC(=S)NCc1cccs1 MS-2013 c1cc(sc1)CNC(=S)NN MS-2014 COC(=O)C1CC(=O)N(C1)Cc2cccs2 MS-2015 c1cc(sc1)Cn2c(n[nH]c2=S)C(F)(F)F MS-2016 c1cc(cnc1)Cn2c(n[nH]c2=S)C(F)(F)F MS-2017 c1cc(cnc1)CNC(=S)NN MS-2018 COc1cccc(c1)CSc2nnc(n2Cc3ccc(cc3)F)C(F)(F)F MS-2020 c1cc(ccc1Cn2c(nnc2SCc3ccc(c(c3)C(F)(F)F)F)C(F)(F)F)F MS-2021 c1cc(ccc1Cn2c(nnc2SCc3ccc(c(c3)F)F)C(F)(F)F)F MS-2022 c1cc(ccc1Cn2c(nnc2SCc3ccc(cc3)[N+](=O)[O-])C(F)(F)F)F MS-2023 Cn1c(nnc1SCc2cccc(c2)OC)c3cccs3 MS-2024 Cn1c(nnc1SCc2ccc(cc2)F)c3cccs3 MS-2025 CC(C)(C)c1ccc(cc1)CSc2nnc(n2C)c3cccs3 MS-2026 Cn1c(nnc1SCc2cccc(c2)Br)c3cccs3 MS-2027 Cc1ccccc1CSc2nnc(n2C)c3cccs3 MS-2028 c1ccc(cc1)CC2CCN(CC2)c3ccccc3/C(=N\O)/N MS-2029 COC(=O)C(CC(=O)c1ccc(cc1)F)c2ccc3c(c2)OCO3 MS-2031 CO/N=C/c1c[nH]c2c1cc(cc2)Br MS-2033 CCOC(=O)CSc1nnc(n1Cc2ccc(cc2)F)C(F)(F)F MS-2034 CCOC(=O)C(C)Sc1nnc(n1Cc2ccc(cc2)F)C(F)(F)F MS-2035 CCCc1cc([nH]n1)C(=O)O MS-2036 CCC/N=C/c1ccc(cc1)O MS-2037 CCCNCc1ccc(cc1)O.Cl MS-2038 CCCN(Cc1ccc(cc1)O)C(=O)NC MS-2039 c1cc(sc1)C/N=C/c2ccc(cc2)O MS-2040 c1cc(sc1)CNCc2ccc(cc2)O.Cl MS-2041 CCOC(=O)CSc1nnc(s1)NC(=O)c2ccc(cc2)C(C)(C)C MS-2042 CCOC(=O)CSc1nnc(s1)NC(=O)c2ccc(cc2)F MS-2043 CCOC(=O)CSc1nnc(s1)NC(=O)c2cccc(c2)OC MS-2044 CCOC(=O)CSc1nnc(s1)NC(=O)c2cccc(c2)OC(F)(F)F MS-2045 CCOC(=O)CSc1nnc(s1)N MS-2046 CC(C)(C)c1ccc(cc1)C(=O)Nc2nnc(s2)SCC(=O)O MS-2047 c1cc(ccc1C(=O)Nc2nnc(s2)SCC(=O)O)F MS-2048 COc1cccc(c1)C(=O)Nc2nnc(s2)SCC(=O)O MS-2049 c1cc(cc(c1)OC(F)(F)F)C(=O)Nc2nnc(s2)SCC(=O)O MS-2050 COc1cc(c(cc1Br)OC)C(=O)CN2C(=O)c3ccccc3C2=O MS-2051 CCOC(=O)C(C(C[N+](=O)[O-])c1ccccc1)C(=O)OCC MS-2052 Cc1cc(ccc1C(C)C)N2CC(CC2=O)C(=O)NCc3cccs3 MS-2053 c1ccc(cc1)OCC(=O)Nc2nnc(s2)SCC(=O)O MS-2054 CC(=O)Nc1nnc(s1)SCC(=O)O MS-2055 C(C(=O)Nc1nnc(s1)SCC(=O)O)C(=O)O MS-2056 c1cc2c(cc1C(=O)Nc3nnc(s3)SCC(=O)O)OCO2 MS-2057 Cc1c(c(on1)C)C(=O)Nc2nnc(s2)SCC(=O)O MS-2058 c1cc(ccc1CN2CCN(CC2)CC(=O)N3CCOCC3)F MS-2059 c1cc(ccc1CN2CCN(CC2)CC(=O)N3CCOCC3)Br MS-2060 c1cc(c(c(c1)Br)NC(=O)C(F)(F)F)Br MS-2061 C1CN(CCN1)CC(=O)N2CCOCC2.Cl.Cl MS-2062 c1cc(ccc1CN2CCN(CC2)CC(=O)N3CCOCC3)C(F)(F)F MS-2063 CCOC(=O)CSc1nnc(s1)NC(=O)CN2CCCCC2 MS-2064 C1COCCN1CC(=O)Nc2nnc(s2)SCC(=O)O MS-2065 CCOC(=O)CSc1nnc(s1)NC(=O)CN2CCN(CC2)C=O MS-2066 CCOC(=O)CSc1nnc(s1)NC(=O)CN2CCSCC2 MS-2067 CCOC(=O)CSc1nnc(s1)NC(=O)CN2CCN(CC2)c3ccccc3 MS-2068 Cc1ccc(c(c1)C(=O)NCc2cccs2)NC(=O)C(F)(F)F MS-2070 c1ccc(c(c1)C(=O)NCc2cccs2)NC(=O)C(F)(F)F MS-2071 COC(=O)CCC(=O)Nc1nnc(s1)C(F)(F)F MS-2072 COc1ccc(cc1)CNC(=O)CCC(=O)Nc2nnc(s2)C(F)(F)F MS-2074 C(CC(=O)O)C(=O)Nc1nnc(s1)C(F)(F)F MS-2075 c1cc(sc1)CNC(=O)CCC(=O)Nc2nnc(s2)C(F)(F)F MS-2076 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)F)C(=O)N3CCOCC3 MS-2077 c1cc(ccc1N2CCOCC2)[N+](=O)[O-] MS-2079 c1cc(ccc1C(=O)N2CCOC23CCCCC3)[N+](=O)[O-] MS-2080 COc1ccc(cc1)/N=C\2/N(CCS2)C(=S)Nc3cccc(c3)Cl MS-2083 Cc1ccccc1/N=C\2/N(CCS2)C(=S)Nc3cccc(c3)Cl MS-2084 CSc1ccc(cc1)Oc2cccc(c2)C(=O)CC#N MS-2085 CCCC(=S)/N=c\1/n(c(cs1)CC(=O)OCC)C MS-2087 CC1(C2(CCC1(OC2=O)C(=O)OC\3CCCN/C3=C/[N+](=O)[O-])C)C MS-2088 CC1([C@@H]([C@H]1C(=S)/N=c\2/n(ccs2)C)C=C(Cl)Cl)C MS-2093 Cc1ccccc1NC(=S)NCCO MS-2094 c1ccc(cc1)CCCN\2CCCN/C2=C\[N+](=O)[O-] MS-2095 CCOC(=O)CC1=CN2CCN=C2S1 MS-2098 c1c(cc(c(c1Br)NC(=O)C(F)(F)F)Br)Br MS-2100 CCCc1c(c[nH]n1)[N+](=O)[O-] MS-2101 COc1ccc(cc1)CNc2nc(c(s2)C#N)Cl MS-2102 c1cc(cc(c1)Cl)CNc2nc(c(s2)C#N)Cl MS-2103 Cc1ccc(cc1)CNc2nc(c(s2)C#N)Cl MS-2104 c1ccc(cc1)CNc2nc(c(s2)C#N)Cl MS-2105 c1cc(sc1)CNc2nc(c(s2)C#N)Cl MS-2106 c1ccnc(c1)CNc2nc(c(s2)C#N)Cl MS-2107 C1COCCN1CCNc2nc(c(s2)C#N)Cl MS-2108 c1cc2c(cc1[N+](=O)[O-])c(=O)cc([nH]2)C(=O)O MS-2111 c1cc2c(cc1NC(CCO)CO)OCO2 MS-2113 Cc1cc(c(c(c1)[N+](=O)[O-])NCCCC(=O)O)[N+](=O)[O-] MS-2114 CCCc1c(cn(n1)C(=O)c2ccc(cc2)Cl)[N+](=O)[O-] MS-2115 c1cc(ccc1NC(=O)Nc2ccc(cc2F)F)N3CCOCC3 MS-2117 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)Nc3cc(ccc3Br)Br MS-2120 Cc1cc(c(c(c1)[N+](=O)[O-])NC(c2ccccc2)C(=O)O)[N+](=O)[O-] MS-2121 CC(=O)N(C)c1ccccc1[N+](=O)[O-] MS-2125 CC1CN(CC(O1)C)c2ccc(cc2)NC(=O)CC#N MS-2126 CCOC(=O)CNc1nc(c(s1)C#N)Cl MS-2127 Cc1ccc(cc1)C(=O)Nc2nc(c(s2)C#N)Cl MS-2128 c1cc2c(cc1Nc3nc(c(s3)C#N)Cl)OCO2 MS-2129 COCCNc1nc(c(s1)C#N)Cl MS-2131 CC(CCc1ccccc1)Nc2nc(c(s2)C#N)Cl MS-2132 CC(CNc1nc(c(s1)C#N)Cl)O MS-2133 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc(c3)OC(C)C MS-2134 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCc3ccc4c(c3)OCO4 MS-2135 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3ccncc3 MS-2136 Cc1c(scn1)C(=O)OC(C#N)c2cccc(c2)Oc3ccccc3 MS-2138 Cc1c(scn1)C(=O)OCc2c(c(c(c(c2Cl)Cl)Cl)Cl)Cl MS-2139 CCN(CC)c1ccc(cc1F)C(=O)OCc2c(c(c(c(c2Cl)Cl)Cl)Cl)Cl MS-2140 Cc1c(scn1)C(=O)OC MS-2142 Cc1c(scn1)C(=O)O MS-2143 CS(=O)(=O)c1cccc(n1)Cl MS-2144 c1cc(nc(c1)C#N)C#N MS-2145 CCOCCOc1cccc(c1NS(=O)(=O)C)[N+](=O)[O-] MS-2146 CCOC(=O)c1ccc(c(c1O)C)SC MS-2147 CCOC(=O)c1cc(c(c(c1O)C)SC)Br MS-2148 CCc1c(ccc(c1OC)C(=O)O)S(=O)(=O)C MS-2149 CCOC(=O)c1ccc(c(c1O)C)S(=O)(=O)C MS-2150 CS(=O)(=O)c1ccc(c(c1C(=O)O)O)C(=O)O MS-2151 CCOC(=O)c1cc(c(c(c1O)C)Cl)Br MS-2152 CCc1c(ccc(c1OC)C(=O)OCc2c(c(c(c(c2Cl)Cl)Cl)Cl)Cl)S(=O)(=O)C MS-2153 Cc1cc(n2c(n1)ncn2)C MS-2155 COc1cc(nc(n1)OC(c2ccccc2)C(=O)O)OC MS-2156 CC1CC(c2c1c(ccc2)NC(=O)C3C(C3(Cl)Cl)(C)C)(C)C MS-2158 CC1CC(c2c1c(ccc2)NC(=O)C3C(C3(SC)SC)(C)C)(C)C MS-2159 CC1CC(c2c1c(ccc2)N/C(=C\[N+](=O)[O-])/SC)(C)C MS-2160 CCc1c(ccc(c1OC)C(=O)OC(C#N)c2cccc(c2)Oc3ccccc3)OS(=O)C MS-2161 CS(=O)(=O)c1nc(cc(n1)Oc2cccc(c2)C(F)(F)F)Oc3cccc(c3)C(F)(F)F MS-2162 c1cc(c(cc1Oc2cc(nc(n2)O)Oc3ccc(c(c3)C(F)(F)F)Cl)C(F)(F)F)Cl MS-2163 CSc1nc(cc(n1)Oc2ccc(c(c2)C(F)(F)F)Cl)Oc3ccc(c(c3)C(F)(F)F)Cl MS-2165 c1cc(c(cc1Oc2cc(nc(n2)O)Oc3ccc(c(c3)C(F)(F)F)F)C(F)(F)F)F MS-2166 c1cc(c(cc1Oc2cc(nc(n2)Oc3ccc(c(c3)C(F)(F)F)Cl)Oc4ccc(c(c4)C(F)(F)F)Cl)C(F)(F)F)Cl MS-2167 COC(=O)c1cccnc1Oc2cccc(c2)C(F)(F)F MS-2169 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(C)Cc3cccnc3 MS-2170 c1cnccc1CNC(=O)C2CC2C(=O)O MS-2171 c1cnccc1CN2C(=O)C3CC3C2=O MS-2172 CC(=O)N(C)c1ccccc1NC(=O)CCl MS-2177 Cc1cc(ccc1C(C)C)NC(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C MS-2178 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccccc3OC MS-2180 CCC1(c2cc(ccc2NC1=O)Br)O MS-2183 CCOc1ccc(cc1C(=O)O)S(=O)(=O)NCc2ccc3c(c2)OCO3 MS-2184 CCOc1ccc(cc1C(=O)O)S(=O)(=O)N2CCOCC2 MS-2185 CCOc1ccc(cc1C(=O)O)S(=O)(=O)NCc2cccs2 MS-2187 CCOc1ccc(cc1C(=O)O)S(=O)(=O)N2CCC(CC2)c3ccccc3 MS-2188 CC1(CN(C1=O)c2ccsc2C(=O)O)C MS-2191 CC1(CN(C1=O)c2ccc(cc2)C(=O)O)C MS-2193 Cc1cc(no1)N/C=C/2\C(=O)OC(=N2)c3ccccc3 MS-2194 COc1cc(nc2c1cc(cc2)[N+](=O)[O-])C(=O)O MS-2195 Cc1ccc(c(n1)OCCCC#N)C#N MS-2197 CCCC1C(=O)Nc2ccccc2N1C(=O)c3cccc(c3)C MS-2199 CCCC1C(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)C(C)(C)C MS-2200 CCC1C(=O)Nc2ccccc2N1C(=O)c3cccc(c3)OC(F)(F)F MS-2201 CCC1C(=O)Nc2ccccc2N1C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-2202 CCC1C(=O)Nc2ccccc2N1C(=O)COc3ccccc3 MS-2203 CCC1C(=O)Nc2ccccc2N1C(=O)c3ccc(nc3)Cl MS-2205 CCC1C(=O)Nc2ccccc2N1C(=O)CC(=O)OCC MS-2206 CCCc1cc(n(n1)C)C(=O)O MS-2208 CC1(CN(C1=O)c2ccsc2C(=O)NCc3ccc4c(c3)OCO4)C MS-2210 Cc1ccc(c(c1)NC(=O)c2c(ccs2)N3CC(C3=O)(C)C)F MS-2212 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)c4c(noc4C)C MS-2213 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2)NC(=O)c4ccc5c(c4)OCO5 MS-2214 CCOC(=O)C/C(=C/C(=O)CC(C)C)/O MS-2215 c1cc(ccc1/C=C/2\C(=O)NC(=S)S2)F MS-2217 c1cc2c([nH]c(=O)c(=O)[nH]2)nc1 MS-2219 CCOC(=O)c1cc(n[nH]1)CC(C)C MS-2220 CCN(CC)C1=NC(=O)/C(=C\c2ccc(cc2)F)/S1 MS-2221 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(C(CCl)Br)Br MS-2224 Cc1ccc2c(c1)C(=O)c3ccccc3CO2 MS-2226 CC(C)c1ccc2c(c1)C(=O)c3ccccc3CO2 MS-2227 COc1ccc2c(c1)C(=O)c3ccccc3CO2 MS-2229 CCOC(=O)C1C(=O)Nc2ccccc2S1 MS-2231 CCC1C(=O)Nc2ccccc2N1C(=O)CCl MS-2232 CCOC(=O)C1=C(NC(=O)CC1c2cccc(c2)Oc3ccccc3)C MS-2233 CCOC(=O)C1=C(NC(=O)CC1c2cccc(c2)Oc3cccc(c3)C(F)(F)F)C MS-2234 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2)C#N)C MS-2235 CCOC(=O)C1=C(NC(=O)CC1c2ccc(cc2)OC(F)(F)F)C MS-2236 Cc1ccc(cc1)OCc2ccccc2C(=O)O MS-2237 c1ccc(c(c1)COc2ccc(cc2)C#N)C(=O)O MS-2238 CC(C)c1ccc(cc1)OCc2ccccc2C(=O)O MS-2239 COc1ccc(cc1)OCc2ccccc2C(=O)O MS-2240 c1ccc2c(c1)c(=O)c(co2)/C=C\3/C(=O)NC(=S)S3 MS-2241 CN1C(=O)C(=Cc2coc3ccccc3c2=O)C(=O)N(C1=O)C MS-2242 CN1C(=O)C(C(=O)N(C1=O)C)C(=O)c2ccccc2 MS-2243 CN1C(=O)C(C(=O)N(C1=O)C)C(=O)c2cccc(c2)C(F)(F)F MS-2244 CN1C(=O)C(C(=O)N(C1=O)C)C(=O)c2ccc(cc2)Cl MS-2245 COC(=O)Oc1ccc(cc1Cl)Cl MS-2246 C1CCC(=C(C1)C(=O)O)Cl MS-2247 COC(=O)Oc1cc(c(cc1Cl)F)[N+](=O)[O-] MS-2249 c1ccc(cc1)COC(=O)NO MS-2251 CO/C(=N\c1cccnc1)/c2ccc(cc2)Cl MS-2259 c1ccc(cc1)NC(=O)NS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] MS-2262 Cc1c(c2ccnc(c2[nH]1)Cl)SC MS-2267 CSC(=S)Nc1ccc(cc1)F MS-2272 CCCCCCCCCOc1ccc(cc1)C(=O)Nc2ccc3c(c2)C(=O)Nc4ccc(cc4O3)C MS-2275 c1ccc2c(c1)c(=O)c(co2)/C=C/C(=O)O MS-2277 CN1C(=O)C(=Cc2ccccc2)C(=O)N(C1=O)C MS-2278 CC(=O)Oc1ccccc1C=C2C(=O)N(C(=O)N(C2=O)C)C MS-2279 c1ccc(cc1)SCc2ccccc2C(=O)O MS-2280 CC(=O)Oc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)C)C MS-2281 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2CC#N)[N+](=O)[O-] MS-2282 CNC(=O)c1cccc(c1)N MS-2283 Cc1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(C)O MS-2285 c1ccc2c(c1)NC(=O)C(S2)CO MS-2286 c1ccc2c(c1)COc3ccc(cc3C2=O)O MS-2287 CC(=O)Oc1ccc2c(c1)C(=O)c3ccccc3CO2 MS-2288 CNC(=O)Oc1ccc2c(c1)C(=O)c3ccccc3CO2 MS-2289 c1ccc(cc1)C(=O)Oc2ccc3c(c2)C(=O)c4ccccc4CO3 MS-2290 CNC(=O)OC1c2ccccc2COc3c1cc(cc3)OC MS-2291 Cc1ccc(cc1)S(=O)(=O)NC(=O)OC2c3ccccc3COc4c2cc(cc4)OC MS-2292 CC(=O)NN1C(=O)/C(=C/c2ccc(cc2)C#N)/SC1=S MS-2297 c1cc(ccc1/C=C\2/C(=O)N(C(=S)S2)N3C(=O)C4CC4C3=O)C#N MS-2298 c1ccc2c(c1)C(=O)N(C2=O)CCCCn3ncnn3 MS-2299 c1ccc(cc1)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)C4CC4C3=O MS-2300 CCCCCCCCN1c2ccc(cc2Oc3ccc(cc3C1=O)[N+](=O)[O-])C MS-2302 CN(C)S(=O)(=O)c1ccc(cc1)C#N MS-2303 c1cc(ccc1C#N)S(=O)(=O)N MS-2304 CC(=O)OCC1C(=O)Nc2ccccc2S1 MS-2305 c1ccc2c(c1)C(=O)NCCO2 MS-2306 Cc1ccc(cc1)CN2CCOc3ccccc3C2=O MS-2307 COc1cccc(c1)CN2CCOc3ccccc3C2=O MS-2308 CCOC(=O)C(C)N1CCOc2ccccc2C1=O MS-2309 c1ccc2c(c1)C(=O)N(CCO2)Cc3ccc(cc3)F MS-2310 c1ccc2c(c1)C(=O)N(CCO2)Cc3ccc(cc3)C(F)(F)F MS-2311 c1ccc2c(c1)C(=O)N(CCO2)CC#N MS-2312 Cc1ccc(cc1)S(=O)(=O)NC(=O)OCC2C(=O)Nc3ccccc3S2 MS-2313 c1ccc(cc1)Oc2cccc(c2)/C=C/C(=O)N3CCOCC3 MS-2314 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2Cc4ccc(cc4)F)[N+](=O)[O-] MS-2315 Cc1ccc2c(c1)Oc3ccc(cc3C(=O)N2Cc4ccc(cc4)C(C)(C)C)[N+](=O)[O-] MS-2316 CCOc1ccc(cc1)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)C4CC4C3=O MS-2317 c1ccc(cc1)/C=C\2/C(=O)N(C(=S)S2)N3C(=O)c4ccccc4C3=O MS-2319 CCOc1ccc(cc1C(=O)O)S(=O)(=O)NCc2ccccc2 MS-2321 CC(=O)c1cc(c(=O)oc1/C=C/NCc2cccc(c2)OC)NC(=O)c3ccccc3 MS-2326 COc1cccc(c1O)/C=C(\C#N)/C(=O)Nc2ccc(cc2)C(F)(F)F MS-2327 CCOc1ccc(cc1)/C=C(\C#N)/C(=O)Nc2ccc(cc2)C(F)(F)F MS-2328 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2ccc(cc2)C(F)(F)F)C#N MS-2329 c1cc2c(cc1Cl)n[se]n2 MS-2331 c1cc(c(c2c1n[se]n2)[N+](=O)[O-])Cl MS-2332 c1cc(c(c(c1N)N)[N+](=O)[O-])Cl MS-2335 c1ccc2c(c1)OCC(O2)CO MS-2337 Cc1cccc(c1)NC(=O)C2COc3ccccc3O2 MS-2338 c1ccc2c(c1)OCC(O2)C(=O)Nc3cccc(c3)C(F)(F)F MS-2339 c1ccc2c(c1)OCC(O2)C(=O)Nc3ccc(cc3)F MS-2340 c1cc(c(c2c1[nH]c(=O)c(=O)[nH]2)[N+](=O)[O-])Cl MS-2341 c1ccc(cc1)CNCC2COc3ccccc3O2 MS-2343 c1ccc(cc1)CCNCC2COc3ccccc3O2 MS-2344 c1ccc(cc1)CCCNCC2COc3ccccc3O2 MS-2345 c1ccc(cc1)CCCCNCC2COc3ccccc3O2 MS-2346 CC(=O)OCC1COc2ccccc2O1 MS-2347 Cc1ccc(cc1)S(=O)(=O)OCC2COc3ccccc3O2 MS-2348 COc1cccc(c1O)/C=C\2/C(=O)c3cc(ccc3O2)O MS-2349 Cc1cc(c(n1c2ccc(cc2)[N+](=O)[O-])C)C(=O)C(F)(F)F MS-2351 Cc1ccc(n1c2ccc(cc2)[N+](=O)[O-])C MS-2353 Cc1ccc(n1c2ccc(cc2)NS(=O)(=O)c3ccccc3)C MS-2354 Cc1ccc(n1c2ccc(cc2)NS(=O)(=O)c3ccccc3C(=O)OC)C MS-2355 Cc1ccc(n1c2ccc(cc2)NC(=O)c3ccccc3F)C MS-2356 Cc1cc(c(n1c2ccc(cc2)NC(=O)c3ccccc3F)C)C(=O)C(F)(F)F MS-2357 Cc1cc(c(n1c2ccc(cc2)N)C)C(=O)C(F)(F)F MS-2358 Cc1cc(c(n1c2ccc(cc2)[N+](=O)[O-])C)C(=O)C(=O)N(C)C MS-2359 Cc1ccc(n1c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Br)C MS-2360 Cc1cc(c(n1c2ccc(cc2)[N+](=O)[O-])C)C(=O)C(=O)N(CC=C)CC=C MS-2361 Cc1cc(c(n1c2ccc(cc2)[N+](=O)[O-])C)C(=O)C(=O)NCCOC MS-2362 Cc1cc(c(n1c2ccc(cc2)[N+](=O)[O-])C)C(=O)C(=O)NC(C)C MS-2363 Cc1ccc2c(c1)c(=O)n(c(n2)C(F)(F)F)N3C(=O)C4CC4C3=O MS-2366 c1cc2c(cc1Cl)c(=O)n(c(n2)C(F)(F)F)N MS-2367 CCOC1=C(C(C(=C(N1)C)C(=O)OCC)c2cccc(c2)C)C=O MS-2368 CC(C)c1ccc(cc1)C(CC(=O)c2ccc(cc2)F)C#N MS-2370 CC(C)c1ccc(cc1)C(CC(=O)c2ccc(cc2)F)C(=O)O MS-2371 CCN(CC)C(=O)C(=O)c1cc(n(c1C)c2ccc(cc2)F)C MS-2372 Cc1cc(c(n1c2ccc(cc2)F)C)C(=O)C(=O)NC MS-2373 Cc1ccc(n1c2ccc(cc2)F)C MS-2374 CCCCCCC(=O)C(F)(F)F MS-2375 c1ccc(c(c1)N)Nc2ccc(cc2C(=O)O)[N+](=O)[O-].Cl MS-2376 Cc1cccc(c1)C(=O)N2c3ccccc3NC(=O)CC2C MS-2379 CC1CC(=O)Nc2ccccc2N1C(=O)c3cccc(c3)F MS-2380 CC1CC(=O)Nc2ccccc2N1C(=O)c3cccc(c3)C(F)(F)F MS-2381 CC1CC(=O)Nc2ccccc2N1C(=O)c3cccc(c3)OC MS-2382 CC1CC(=O)Nc2ccccc2N1C(=O)NC MS-2383 CC1CC(=O)Nc2ccccc2N1 MS-2384 CC1=Nc2ccccc2NC(=O)C1 MS-2385 Cc1ccc(cc1)S(=O)(=O)N2c3ccccc3NC(=O)CC2C MS-2386 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)OC MS-2387 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)Br MS-2388 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccccc3 MS-2389 c1ccc2c(c1)Nc3ccc(cc3C(=O)N2)[N+](=O)[O-] MS-2390 CC1CN(C2(O1)CCCCCC2)C(=O)Nc3cccc(c3)Cl MS-2391 CC1CN(C2(O1)CCCCCC2)C(=O)Nc3ccc(cc3)F MS-2392 CC1CN(C2(O1)CCCCCC2)C(=O)Nc3cccc(c3)C(F)(F)F MS-2393 CC1CN(C2(O1)CCCCCC2)C(=O)Nc3ccccc3 MS-2394 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc3c(c2)nns3 MS-2395 c1cc(cc(c1)Cl)NC(=O)Nc2ccc3c(c2)nns3 MS-2396 c1cc2c(cc1NC(=O)Nc3ccc(cc3Cl)Cl)nns2 MS-2398 Cc1cc(c(n1c2nccs2)C)C(=O)C(=O)NC MS-2400 Cc1cc(c(n1c2nccs2)C)C(=O)C(F)(F)F MS-2401 Cc1ccc(n1c2ccc3c(c2)nns3)C MS-2402 Cc1cc(c(n1c2ccc3c(c2)nns3)C)C(=O)C(F)(F)F MS-2403 c1cc2c(cc1OCC#N)OCC2=O MS-2404 c1cc2c(cc1NC(=O)C3CC3C(=O)O)nns2 MS-2405 Cc1cc(c(n1c2ccc3c(c2)nns3)C)C(=O)C(=O)NC MS-2409 c1cc2c(cc1N3C(=O)C4CC4C3=O)nns2 MS-2410 CC1CC(=O)Nc2ccccc2N1C(=O)CN3CCOCC3 MS-2411 CC1CC(=O)Nc2ccccc2N1C(=O)CNCCN3CCOCC3 MS-2412 CC1CC(=O)Nc2ccccc2N1C(=O)CNCc3ccc4c(c3)OCO4 MS-2413 CC1CC(=O)Nc2ccccc2N1C(=O)CNCCc3ccccc3 MS-2414 CC1CC(=O)Nc2ccccc2N1C(=O)CCl MS-2415 CC1CC(=O)Nc2ccccc2N1C(=O)CN3CCN(CC3)c4ccccc4 MS-2416 CC1CC(=O)Nc2ccccc2N1C(=O)CN3CCN(CC3)C=O MS-2418 Cc1cc(c(n1c2ccc3c(c2)nns3)C)C(=O)C(=O)O MS-2419 CC(CNCCN1CCOCC1)(COc2ccc(cc2)Cl)O MS-2420 CC(CO)Nc1ccc(c(c1)Cl)F MS-2422 CC(CO)N(Cc1ccccc1)c2ccc(c(c2)Cl)F MS-2423 CC(C)(C)c1ccc(cc1)NCC(C)(COc2ccc(cc2)Cl)O MS-2424 c1cc2c(cc1O)CCCC2=O MS-2425 c1cc(c(nc1)N2CC(C2)C(=O)O)[N+](=O)[O-] MS-2429 c1cc(c(nc1)N2C[C@H]3C[C@H]3[C@H]2C(=O)O)[N+](=O)[O-] MS-2430 CCN(CC)S(=O)(=O)NC(=O)Nc1c(cnn1c2ccccc2)C#N MS-2432 c1cc(c(nc1)NC(c2cccs2)C(=O)O)[N+](=O)[O-] MS-2433 CN(CCO)c1cnccn1 MS-2434 CN(CCOc1ccc(cc1)/C=C/2\C(=O)NC(=O)S2)c3cnccn3 MS-2437 CC(CNc1cnccn1)O MS-2438 CN1C(=O)C(=Cc2ccc(cc2)OCCN(C)c3cnccn3)C(=O)N(C1=O)C MS-2439 CN(CCOc1ccc(cc1)/C=C/C(=O)O)c2cnccn2 MS-2440 c1cc(ccc1C=O)Oc2cnccn2 MS-2441 c1cc(ccc1/C=C/2\C(=O)NC(=O)S2)Oc3cnccn3 MS-2442 CN1C(=O)C(=Cc2ccc(cc2)Oc3cnccn3)C(=O)N(C1=O)C MS-2443 c1cc(ccc1/C=C/2\C(=O)NC(=S)S2)Oc3cnccn3 MS-2444 CN(CCOc1ccc(cc1)C=O)c2cnccn2 MS-2445 c1cc(ccc1C=O)OCCOc2ccc(cc2)C3CCCCC3 MS-2447 CN1C(=O)C(=Cc2ccc(cc2)OCCOc3ccc(cc3)C4CCCCC4)C(=O)N(C1=O)C MS-2448 c1cc(c(nc1)NCC(=O)O)[N+](=O)[O-] MS-2450 CC(=O)c1ccc(cc1)Oc2cnccn2 MS-2451 CCC(=O)c1ccc(cc1)Oc2cnccn2 MS-2452 c1cc(ccc1C(=O)N2CCOCC2)Oc3cnccn3 MS-2453 CC1CCCCN1C(=O)c2ccc(cc2)Oc3cnccn3 MS-2454 c1cc(cc(c1)Oc2cnccn2)N MS-2455 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccc(c2)Oc3cnccn3 MS-2456 c1cc(cc(c1)NC(=O)Nc2cccc(c2)Oc3cnccn3)C(F)(F)F MS-2457 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)Oc3cnccn3 MS-2458 COC(=O)c1ccccc1S(=O)(=O)Nc2cccc(c2)Oc3cnccn3 MS-2459 c1cc(cc(c1)Oc2cnccn2)NS(=O)(=O)c3ccc(cc3)OC(F)(F)F MS-2460 c1cc(cc(c1)Oc2cnccn2)NS(=O)(=O)c3ccc(cc3)F MS-2461 c1cc(cc(c1)Oc2cnccn2)NC(=O)CCl MS-2462 c1cc(cc(c1)Oc2cnccn2)NC(=O)CN3CCOCC3 MS-2463 c1cc(cc(c1)Oc2cnccn2)NC(=O)CN3CCCCC3 MS-2464 C=CCN(CC=C)CC(=O)Nc1cccc(c1)Oc2cnccn2 MS-2465 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc(c2)Oc3cnccn3 MS-2466 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccc(c2)Oc3cnccn3 MS-2467 CC(c1ccc(cc1)Oc2cnccn2)O MS-2468 C/C(=N/O)/c1ccc(cc1)Oc2cnccn2 MS-2469 CCO/N=C(/C)\c1ccc(cc1)Oc2cnccn2 MS-2470 C/C(=N/OCC=C)/c1ccc(cc1)Oc2cnccn2 MS-2471 c1cc(c(cc1Cl)[N+](=O)[O-])NCC(=O)O MS-2472 c1cc(c(cc1F)F)/C=C/2\C(=O)NC(=O)S2 MS-2473 c1ccc2c(c1)N=Cc3cc(ccc3O2)[N+](=O)[O-] MS-2474 c1ccc2c(c1)NCc3cc(ccc3O2)[N+](=O)[O-] MS-2475 Cc1ccc(cc1)S(=O)(=O)N2Cc3cc(ccc3Oc4c2cccc4)[N+](=O)[O-] MS-2476 c1ccc2c(c1)N(Cc3cc(ccc3O2)[N+](=O)[O-])S(=O)(=O)c4ccc(cc4)Br MS-2477 c1ccc2c(c1)N(Cc3cc(ccc3O2)[N+](=O)[O-])S(=O)(=O)c4ccccc4Cl MS-2478 COC(=O)c1ccccc1S(=O)(=O)N2Cc3cc(ccc3Oc4c2cccc4)[N+](=O)[O-] MS-2479 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2Cc3cc(ccc3Oc4c2cccc4)[N+](=O)[O-] MS-2480 c1ccc2c(c1)N(Cc3cc(ccc3O2)[N+](=O)[O-])C(=O)Nc4cccc(c4)C(F)(F)F MS-2481 CC(=O)N1Cc2cc(ccc2Oc3c1cccc3)[N+](=O)[O-] MS-2482 CC(=O)N1Cc2cc(ccc2Oc3c1cccc3)N MS-2483 Cc1ccc(cc1)C(=O)c2cccc3c2NCc4cc(ccc4O3)[N+](=O)[O-] MS-2484 c1ccc2c(c1)N(Cc3cc(ccc3O2)[N+](=O)[O-])C(=O)c4cccc(c4)OC(F)(F)F MS-2485 CC(=O)N1Cc2cc(ccc2Oc3c1cccc3)NS(=O)(=O)c4ccc(cc4)Br MS-2486 CC(=O)N1Cc2cc(ccc2Oc3c1cccc3)NS(=O)(=O)c4ccccc4Cl MS-2487 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)CN(c4ccccc4O3)C(=O)C MS-2488 CC1(COCN1C(=O)c2ccc(cc2)Cl)C MS-2491 CC1(COCN1S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])C MS-2492 CC1(COCN1S(=O)(=O)c2ccccc2C(F)(F)F)C MS-2493 Cc1ccc(cc1)S(=O)(=O)N2COCC2(C)C MS-2495 CCN(CC)CC(=O)N1c2ccccc2CCc3c1cccc3 MS-2496 CC1(COCN1C(=O)c2ccc(c(c2)Cl)Cl)C MS-2497 CC1(COCN1Cc2ccc(cc2)[N+](=O)[O-])C MS-2498 CC1(COCN1C(=O)c2ccc(cc2)C#N)C MS-2499 CC1(COCN1Cc2ccccc2F)C MS-2500 CC1(COCN1Cc2ccc(cc2)C(F)(F)F)C MS-2501 CC1(COCN1Cc2ccccc2)C MS-2502 CCOC(=O)COc1cnc2ccccc2n1 MS-2503 c1ccc2c(c1)ncc(n2)OCC(=O)O MS-2504 CCc1ccc(cc1)OCCN2CC(OC2)(C)C MS-2506 C=CCN(CC=C)CC(=O)N1c2ccccc2CCc3c1cccc3 MS-2507 c1ccc2c(c1)CCc3ccccc3N2C(=O)CN4CCOCC4 MS-2508 c1ccc2c(c1)CCc3ccccc3N2C(=O)NS(=O)(=O)N4CCOCC4 MS-2510 c1ccc2c(c1)CCc3ccccc3N2C(=O)NS(=O)(=O)N4CCCCC4 MS-2511 Cc1csc(c1n2cccc2)C(=O)O MS-2512 c1ccc2c(c1)C=Nc3ccccc3O2 MS-2513 Cc1ccc(c2c1CC(O2)(C)C)Nc3cnccn3 MS-2514 Cc1ccc(cc1)C(=O)N(Cc2ccc(cc2)Cl)c3cnccn3 MS-2515 CC(C)(C)N(C(=O)c1ccccc1[N+](=O)[O-])N MS-2516 CC(C)(C)N(C(=O)c1ccccc1N)N MS-2517 c1cc(ncc1[N+](=O)[O-])NCC(=O)O MS-2518 c1cc(ncc1[N+](=O)[O-])NC2(CCCC2)C(=O)O MS-2519 c1ccc2c(c1)ncc(n2)OCCO MS-2520 c1cc(ncc1[N+](=O)[O-])NCCC(=O)O MS-2521 C1CCCC(CCC1)NC(=O)C2CC2C(=O)O MS-2522 CC(C(=O)O)Nc1ccc(cn1)[N+](=O)[O-] MS-2523 CN(CCC#N)c1ccc(cc1)[N+](=O)[O-] MS-2524 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2nc(nc(n2)OC)C MS-2525 c1ccc(cc1)COC(=O)N2CCCC2/C=C/CN3CCCC3 MS-2526 CCN(CC)C/C=C/C1CCCN1C(=O)OCc2ccccc2 MS-2527 c1ccc(cc1)COC(=O)N2CCCC2/C=C/CN3CCOCC3 MS-2528 CC1CN(CC(O1)C)C/C=C/C2CCCN2C(=O)OCc3ccccc3 MS-2529 CN1CCCC1/C=C/COc2ccc(cc2)F MS-2531 Cc1cc(c(c(c1)[N+](=O)[O-])NCCC(=O)O)[N+](=O)[O-] MS-2533 c1ccc(cc1)COC(=O)N2CCCC2/C=C/COc3ccc(c(c3)Cl)Cl MS-2534 CN1CCCC1/C=C/COc2ccc(c(c2)Cl)Cl MS-2535 c1ccc(cc1)COC(=O)N2CCCC2/C=C/COc3ccccc3 MS-2536 CN1CCCC1/C=C/COc2ccccc2 MS-2537 Cc1cc(c(c(c1)[N+](=O)[O-])N2CCOCC2)[N+](=O)[O-] MS-2538 c1ccc(cc1)COC(=O)N2CCCC2/C=C/Cn3ccnc3 MS-2539 CN1CCCC1/C=C/CN2CCOCC2 MS-2540 Cc1cc(c(c(c1)[N+](=O)[O-])N2CC(OC(C2)C)C)[N+](=O)[O-] MS-2541 Cc1cc(c(c(c1)[N+](=O)[O-])N2CCCC2)[N+](=O)[O-] MS-2542 c1ccc(cc1)/C=N/NC(=O)CCCO MS-2543 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2nnc(s2)C MS-2545 COC(=O)/C=C/c1ccc(cc1)n2ccnc2 MS-2546 c1cc(ccc1/C=N/c2ccc(cc2)F)n3ccnc3 MS-2547 c1cc(ccc1CNc2ccc(cc2)F)n3ccnc3 MS-2548 CCC(C)Nc1c(cc(cc1[N+](=O)[O-])C)[N+](=O)[O-] MS-2549 CCCCNc1c(cc(cc1[N+](=O)[O-])C)[N+](=O)[O-] MS-2550 Cc1ccc(cc1)CNC(=S)Nc2ccc(cc2)Br MS-2551 CC(C)(C)N1C(=O)c2ccccc2NC(=O)N1 MS-2552 Cc1ccccc1CN2C(=O)Nc3ccccc3C(=O)N2C(C)(C)C MS-2553 CC(C)(C)N1C(=O)c2ccccc2NC(=O)N1Cc3ccc(cc3)Br MS-2554 CC(C)(C)N1C(=O)c2ccccc2NC(=O)N1Cc3ccccc3 MS-2555 CC(C)(C)N1C(=O)c2ccccc2NC(=O)N1Cc3cccc(c3)OC MS-2556 Cc1ccc(cc1)CN/C(=N/c2ccc(cc2)Br)/SC MS-2557 Cc1cc(ccc1Br)/N=C/c2ccc(cc2)n3cncn3 MS-2559 Cc1cc(ccc1Br)NCc2ccc(cc2)n3cncn3 MS-2560 COC(=O)/C=C/c1ccc(cc1)n2cncn2 MS-2561 Cc1cc(ccc1O)C=C2C(=O)N(C(=O)N(C2=O)C)C MS-2562 CN1C(=O)C(=Cc2ccccc2OCC(=O)O)C(=O)N(C1=O)C MS-2563 Cc1ccc(c(c1)NC(C#N)c2ccc(cc2)n3cncn3)F MS-2566 Cc1cc(ccc1Br)/N=C/c2ccc(cc2)n3ccnc3 MS-2567 Cc1cc(ccc1Br)NC(C#N)c2ccc(cc2)n3ccnc3 MS-2568 Cc1cccc(c1)NC(C#N)c2ccc(cc2)n3ccnc3 MS-2569 Cc1cccc(c1)NCc2ccc(cc2)n3ccnc3 MS-2570 Cc1cccc(c1)/N=C/c2ccc(cc2)n3ccnc3 MS-2571 CC1C(=O)Nc2ccccc2O1 MS-2573 CCCC1(OCCO1)CC(=O)NC2CCOC2=O MS-2574 CCCC(=O)CC(=O)NC1CCOC1=O MS-2575 CC1(CC2=C(C(=O)C1)C(C(=C(O2)N)C#N)(C)C(O)OC)C MS-2576 COc1ccccc1CNC2=C(C(=O)c3ccccc3C2=O)Cl MS-2577 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCc3ccc(c(c3)Cl)Cl MS-2578 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCc3ccc(cc3)F MS-2579 CC(=O)N(Cc1ccc(cc1)F)C2=C(C(=O)c3ccccc3C2=O)Cl MS-2580 CC(=O)N(Cc1ccc(c(c1)Cl)Cl)C2=C(C(=O)c3ccccc3C2=O)Cl MS-2581 CCOC(=O)C(=Cc1ccc(cc1)n2cncn2)C(=O)OCC MS-2582 CCOC(=O)C(C(C[N+](=O)[O-])c1ccc(cc1)n2cncn2)C(=O)OCC MS-2583 CC(=O)N(Cc1ccc(cc1)F)C2=C(C(=O)c3ccccc3C2=O)NCc4ccccc4 MS-2584 COc1cccc(c1CC2C(=O)NC(=O)S2)OC MS-2585 c1ccc(cc1)Oc2cccc(c2)CC3C(=O)NC(=O)S3 MS-2586 CN1C(=O)/C(=C/c2cccc(c2)Oc3ccccc3)/SC1=O MS-2588 c1ccc2c(c1)CN(c3ccccc3O2)C(=O)CCl MS-2589 CC1(CC2=C(C(=O)C1)C3(CC(=O)OC3O2)C)C MS-2590 CC1(c2c(c3ccccc3oc2=O)OC(=C1C#N)N)C(OC)OC MS-2591 C[C@@]12CC(=O)N(C1OC3=C2C(=O)CC(C3)(C)C)C4CC4 MS-2592 CC12CC(=O)OC1Oc3c2c(=O)oc4c3cccc4 MS-2593 CC12CC(=NC1NC(=O)C2)c3ccccc3O MS-2594 CC12CC(NC1NC(=O)C2)c3ccccc3O MS-2595 CC(=O)N(Cc1ccc(c(c1)Cl)Cl)C2=C(C(=O)c3ccccc3C2=O)NC MS-2596 CCN1C(=O)/C(=C\c2cccc(c2)Oc3ccccc3)/SC1=O MS-2597 CC(=O)N(Cc1ccc(cc1)F)C2=C(C(=O)c3ccccc3C2=O)NCCc4ccccc4 MS-2598 CC(C)NC1=C(C(=O)c2ccccc2C1=O)N(Cc3ccc(c(c3)Cl)Cl)C(=O)C MS-2599 CC(=O)N(Cc1ccccc1OC)C2=C(C(=O)c3ccccc3C2=O)NC MS-2602 CC(C)NC1=C(C(=O)c2ccccc2C1=O)Cl MS-2603 CCOC(=O)C(=Cc1ccc(cc1)n2ccnc2)C(=O)OCC MS-2604 c1cc(ccc1/C=C\2/NC(CS2)C(=O)O)n3ccnc3 MS-2605 CCC(=O)N(C1=C(C(=O)c2ccccc2C1=O)NC)C(C)C MS-2607 c1ccc2c(c1)C(=O)N(C2=O)c3ccc(cc3)/C=C/4\NC(CS4)C(=O)O MS-2608 CC(=O)N1C(C[C@]2(C1NC(=O)C2)C)c3ccccc3OC(=O)C MS-2611 C[C@]12CC(N(C1NC(=O)C2)C(=O)c3ccccc3)c4ccccc4OC(=O)c5ccccc5 MS-2612 C[C@]12CC(N(C1NC(=O)C2)C(=O)c3cccc(c3)C(F)(F)F)c4ccccc4OC(=O)c5cccc(c5)C(F)(F)F MS-2613 Cc1cccc(c1)C(=O)N2C(C[C@]3(C2NC(=O)C3)C)c4ccccc4OC(=O)c5cccc(c5)C MS-2615 CCOC(=O)CN1c2ccccc2OC(C1=O)C MS-2616 CC1C(=O)N(c2ccccc2O1)CC(=O)NCc3ccc(cc3)OC MS-2617 CC1C(=O)N(c2ccccc2O1)CC(=O)NCCc3ccc(cc3)OC MS-2618 CCC(=O)N(C1=C(C(=O)c2ccccc2C1=O)NC(C)C)C(C)C MS-2619 CCC(=O)N(C1=C(C(=O)c2ccccc2C1=O)Cl)C(C)C MS-2620 Cc1cc(ccc1C(C)C)NC(C#N)c2ccc(cc2)n3ccnc3 MS-2622 CC1C(=O)N(c2ccccc2O1)Cc3ccc(cc3)F MS-2623 Cc1ccc(c(c1)C)CN2c3ccccc3OC(C2=O)C MS-2624 CC1C(=O)N(c2ccccc2O1)Cc3ccccc3Cl MS-2625 CC1C(=O)N(c2ccccc2O1)Cc3cccc(c3)OC MS-2626 CCN1c2ccc(cc2C(=O)C1=O)Br MS-2627 CC(=O)N1C(C[C@]2(C1NC(=O)C2)C)c3ccccc3O MS-2628 C[C@]12CC(N(C1NC(=O)C2)C(=O)c3cccc(c3)C(F)(F)F)c4ccccc4O MS-2629 c1ccc(cc1)C2(c3cc(ccc3NC2=O)Br)O MS-2631 CCCCN1c2ccc(cc2C(C1=O)(c3ccc(cc3)C)O)Br MS-2632 CCCCN1c2ccc(cc2C(C1=O)(c3ccccc3)O)Br MS-2633 C[C@]12CC(N(C1NC(=O)C2)S(=O)(=O)c3ccccc3)c4ccccc4OS(=O)(=O)c5ccccc5 MS-2635 c1ccc2c(c1)C(=O)C(=O)N2Cc3ccc(cc3)F MS-2636 CC(=O)N1C(C[C@]2(C1NC(=O)C2)C)c3ccccc3OC(=O)c4ccc(nc4)Cl MS-2637 Cc1cc(no1)C(=O)Oc2ccccc2C3C[C@@]4(CC(=O)NC4N3C(=O)C)C MS-2638 CC(=O)N1C(C[C@]2(C1NC(=O)C2)C)c3ccccc3OC(=O)c4conc4c5ccccc5Cl MS-2639 Cc1nc(cs1)CN2CCOCC2 MS-2640 Cc1nc(cs1)CN2CCN(CC2)C=O MS-2641 Cc1nc(cs1)CN2CCCCC2 MS-2642 Cc1c(c(n(n1)C)Cl)/C=C\2/C(=O)NC(=O)S2 MS-2643 Cc1ccc(cc1)S(=O)(=O)NC(=O)NC2(CCCCC2)C#C MS-2644 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCC(F)(F)F MS-2645 Cc1c(c(n(n1)C)Cl)/C=C\2/C(=O)NC(=S)S2 MS-2646 Cc1cc(=O)oc2c1ccc(c2)OS(=O)(=O)C MS-2647 Cc1c(c(n(n1)C)Cl)/C=C/2\C(=O)N=C(S2)SC MS-2648 Cc1c(c(n(n1)C)Cl)/C=C/C(=O)O MS-2649 Cc1c(c(n(n1)C)Cl)/C=C/C(=O)N2CCOCC2 MS-2650 CCOC(=O)C1=C(C(=O)NCC1)O MS-2651 c1ccc(c(c1)N)OCCOc2ccccc2N MS-2652 c1cc(cc(c1)OCCCl)[N+](=O)[O-] MS-2653 c1ccc(c(c1)[N+](=O)[O-])OCCCl MS-2654 CCOC(=O)C(=O)Nc1ccccc1OCCOc2ccccc2NC(=O)C(=O)OCC MS-2655 Cc1ccc(s1)/C=C/C(=O)c2ccc(cc2)F MS-2656 CCN(CC)C(=O)/C=C/c1c(nn(c1Cl)C)C MS-2657 c1cc(sc1)CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)O MS-2658 c1cscc1CC(=O)N2C[C@@H]3C[C@@H]3[C@H]2C(=O)O MS-2659 CCOC(=O)C1=C(C(=O)NCC1)OCc2cccc(c2)Br MS-2660 c1cc(cc(c1)Br)COC2=C(CCNC2=O)C(=O)O MS-2661 CCOC(=O)CNc1ccccc1OCCOc2ccccc2NCC(=O)OCC MS-2662 Cc1ccc(o1)/C=C/C(=O)c2ccc(cc2)F MS-2663 Cc1ccc(o1)C(CC(=O)c2ccc(cc2)F)C#N MS-2664 c1ccc(c(c1)C#N)Sc2ccccc2N MS-2667 c1ccc2c(c1)C(=Nc3ccccc3S2)N MS-2668 Cc1cc(=O)oc2c1ccc(c2)OCc3ccc(cc3)[N+](=O)[O-] MS-2669 c1ccc(cc1)OCC(=O)Nc2ccccc2Sc3ccccc3C#N MS-2670 Cc1csc(c1n2ccc(c2)C(=O)C(=O)N(C)C)C(=O)OC MS-2673 CCN(CC)C(=O)C(=O)c1ccn(c1)c2c(csc2C(=O)OC)C MS-2674 Cc1csc(c1n2ccc(c2)C(=O)C(=O)N(CC=C)CC=C)C(=O)OC MS-2676 c1ccc2c(c1)C(N(C2=O)Cc3cccs3)O MS-2677 c1ccc2c(c1)C(N(C2=O)Cc3cccs3)SCC(=O)O MS-2678 c1ccc2c(c1)C3N(C2=O)Cc4c(ccs4)C(=O)CS3 MS-2679 c1ccc2c(c1)C(=Nc3ccccc3O2)N MS-2680 CCOC(=O)C1=C(C(=O)N(CC1)Cc2ccccc2)O MS-2682 c1ccc(cc1)OCC(=O)Nc2ccccc2Sc3cccc(c3C#N)F MS-2683 c1ccc(c(c1)N)Sc2cccc(c2C#N)F MS-2685 c1cc(c(cc1COC2=C(CCNC2=O)C(=O)O)F)F MS-2687 CCOC(=O)C1=C(C(=O)N(CC1)Cc2ccc(cc2)C(C)(C)C)O MS-2688 CCOC(=O)C1=C(C(=O)NCC1)OCc2ccc(cc2)C(C)(C)C MS-2689 c1ccc(cc1)COC2=C(CCNC2=O)C(=O)O MS-2690 c1cc(ccc1COC2=C(CCNC2=O)C(=O)O)[N+](=O)[O-] MS-2692 c1ccc2c(c1)C3N(C2=O)Cc4c(ccs4)C(CS3)O MS-2693 CC(=O)OC1c2ccccc2C(=O)N1Cc3cccs3 MS-2694 c1ccc(cc1)C(=O)OC2c3ccccc3C(=O)N2Cc4cccs4 MS-2695 CC(C)(C)NC(=O)OC1c2ccccc2C(=O)N1Cc3cccs3 MS-2696 c1ccc(cc1)CCn2c(c(c3c(c2=O)cccn3)C#N)N MS-2697 COc1ccc(cc1)CNC(=O)CSC2c3ccccc3C(=O)N2Cc4cccs4 MS-2698 c1ccc2c(c1)C(N(C2=O)Cc3cccs3)SCC(=O)NCc4ccc(cc4)Cl MS-2699 c1cc(cc(c1)OCCOC(=O)c2ccc(cc2)F)NC(=O)c3ccc(cc3)F MS-2704 c1ccc2c(c1)CCN2C(=O)C3CC3C(=O)O MS-2705 CCOC(=O)C(C(=O)N1CCc2c1cccc2)C(=O)OCC MS-2707 CCCNC1C(=C(CCN1)C(=O)OCC)O MS-2708 CCOC(=O)C1=C(C(NCC1)NCCOC)O MS-2709 c1cc(ccc1N)OCCn2cncn2 MS-2710 c1cc(ccc1[N+](=O)[O-])OCCn2cncn2 MS-2711 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)OCCn3cncn3 MS-2712 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)OCCn3cncn3 MS-2713 c1cc(ccc1NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)OCCn3cncn3 MS-2714 c1ccc(cc1)/C=C\2/C(=O)c3ccsc3CN4C(S2)c5ccccc5C4=O MS-2715 c1ccc2c(c1)C3N(C2=O)Cc4c(ccs4)C(=O)/C(=C/c5cccc(c5)F)/S3 MS-2716 c1ccc2c(c1)C3N(C2=O)Cc4c(ccs4)C(=O)/C(=C/c5cccc(c5)Oc6cccc(c6)C(F)(F)F)/S3 MS-2717 c1ccc2c(c1)C3N(C2=O)Cc4c(ccs4)C(=O)/C(=C/c5cccc(c5)Oc6ccc(cc6)Cl)/S3 MS-2718 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCc3c2cccc3 MS-2719 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccccc3)CCCC2 MS-2720 CO/N=C/1\CSC2c3ccccc3C(=O)N2Cc4c1ccs4 MS-2722 CCO/N=C\1/CSC2c3ccccc3C(=O)N2Cc4c1ccs4 MS-2723 c1ccc(cc1)CO/N=C\2/CSC3c4ccccc4C(=O)N3Cc5c2ccs5 MS-2724 c1cc(ccc1/C=C\2/C(=O)NC(=O)S2)n3cncn3 MS-2725 CN1C(=O)/C(=C/c2ccc(cc2)n3cncn3)/SC1=O MS-2726 c1ccc(cc1)N/N=C/2\CSC3c4ccccc4C(=O)N3Cc5c2ccs5 MS-2727 CC(=O)OC1CSC2c3ccccc3C(=O)N2Cc4c1ccs4 MS-2728 CC(C)(C)NC(=O)OC1CSC2c3ccccc3C(=O)N2Cc4c1ccs4 MS-2729 c1cc(ccc1CC2C(=O)NC(=O)S2)n3cncn3 MS-2730 c1cnn(c1)c2ccc(cc2)CC3C(=O)NC(=O)S3 MS-2732 CC(C)(C)c1ccc(cc1)/C=C\2/C(=O)NC(=O)S2 MS-2734 c1cc(ccc1C=C(C(=O)Nc2ccc(cc2)C(F)(F)F)C(=O)Nc3ccc(cc3)C(F)(F)F)Cl MS-2736 c1cc(ccc1C(F)(F)F)NC(=O)C(=Cc2ccc3c(c2)OCO3)C(=O)Nc4ccc(cc4)C(F)(F)F MS-2737 Cc1ccc(c2c1CC(O2)(C)C)NC(=S)Nc3ccc(c(c3)Cl)Cl MS-2738 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(c3c2OC(C3)(C)C)C MS-2739 c1ccc(cc1)C=C(C(=O)Nc2ccc(cc2)C(F)(F)F)C(=O)Nc3ccc(cc3)C(F)(F)F MS-2740 Cc1ccc(c2c1CC(O2)(C)C)n3c(ccc3C)C MS-2742 Cc1ccc(cc1)CN2C(=O)CSC2=O MS-2743 Cc1ccc(c2c1CC(O2)(C)C)n3c(cc(c3C)C(=O)C(F)(F)F)C MS-2744 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)Nc3c(cccc3Cl)Cl MS-2745 Cc1ccc(cc1)CN2C(=O)/C(=C/c3ccc(cc3)F)/SC2=O MS-2746 Cc1ccc(cc1)CN2C(=O)/C(=C\c3ccc4c(c3)OCO4)/SC2=O MS-2747 c1cc2c(cc1C(=O)Cn3cncn3)CCO2 MS-2748 c1cc2c(cc1c3csc(n3)N)CCO2 MS-2749 CC(=O)Nc1nc(cs1)c2ccc3c(c2)CCO3 MS-2750 C#CC1(CCCCC1)NC(=O)Nc2cccc(c2)C(F)(F)F MS-2751 C#CC1(CCCCC1)NC(=O)Nc2ccc(cc2)Cl MS-2752 C#CC1(CCCCC1)NC(=O)Nc2cccc(c2)Cl MS-2753 C#CC1(CCCCC1)NC(=O)Nc2ccc(cc2)F MS-2754 C#CC1(CCCCC1)NC(=O)Nc2ccc(cc2F)F MS-2755 c1ccc2c(c1)CN3C(c4ccccc4C3=O)SCC2=O MS-2756 c1ccc(cc1)N2C(c3ccccc3C2=O)SCC(=O)O MS-2757 c1ccc(cc1)/C=C\2/C(=O)c3ccccc3CN4C(S2)c5ccccc5C4=O MS-2758 c1ccc(cc1)CN2C(c3ccccc3C2=O)SCC(=O)O MS-2759 c1ccc2c(c1)CN3C(c4ccccc4C3=O)S/C(=C\c5ccc(cc5)Cl)/C2=O MS-2760 Cc1cc(no1)NC(=O)CSC2c3ccccc3C(=O)N2Cc4ccccc4 MS-2761 c1ccc(cc1)CN2C(c3ccccc3C2=O)O MS-2763 CC(=O)OC1c2ccccc2C(=O)N1Cc3ccccc3 MS-2764 CCOC(=O)c1ccc(cc1)n2c(c(c3c(c2=O)cccn3)C#N)N MS-2765 CC(=O)OC1c2ccccc2C(=O)N1c3ccccc3 MS-2766 c1ccc(cc1)CN2C(c3ccccc3C2=O)SCC(=O)Nc4nccs4 MS-2767 c1ccc2c(c1)CN3C(c4ccccc4C3=O)S/C(=C\c5ccc(cc5)C#N)/C2=O MS-2768 C#CC1(CCCCC1)NS(=O)(=O)c2ccc(cc2)F MS-2769 C#CC1(CCCCC1)NS(=O)(=O)c2ccccc2C(F)(F)F MS-2770 C#CC1(CCCCC1)NS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] MS-2771 Cc1ccc(cc1)S(=O)(=O)NC2(CCCCC2)C#C MS-2772 C#CC1(CCCCC1)NS(=O)(=O)c2ccccc2 MS-2773 CN(C)C(=O)CSC1c2ccccc2C(=O)N1c3ccccc3 MS-2774 CCN(CC)C(=O)CSC1c2ccccc2C(=O)N1c3ccccc3 MS-2775 c1ccc(cc1)N2C(c3ccccc3C2=O)SCC(=O)N4CCOCC4 MS-2776 CC(C)(C)NC(=O)NC1(CCCCC1)C#C MS-2778 CN(C)C(=O)NC1(CCCCC1)C#C MS-2779 CN(C)C(=C(C#N)C#N)SC MS-2780 CSC(=C(C#N)C#N)NCc1cccnc1 MS-2781 CC(C)NC(=O)NC1(CCCCC1)C#C MS-2782 CCCCNC(=O)NC1(CCCCC1)C#C MS-2783 c1ccc(cc1)/C=C/CN2CCN(CC2)Cc3ccc(cc3)F MS-2784 C#CC1(CCCCC1)NC(=O)c2cccc(n2)Cl MS-2785 c1ccc(cc1)/C=C/CN2CCN(CC2)Cc3ccc(cc3)Br MS-2786 c1ccc2c(c1)CN3C(c4ccccc4C3=O)SCC2O MS-2787 CC(=O)O/C/1=C/SC2c3ccccc3C(=O)N2Cc4c1cccc4 MS-2789 c1ccc(cc1)CN2C(c3ccccc3C2=O)SCC(=O)N4CCOCC4 MS-2792 C[N+]1(CC[N+](CC1)(C)Cc2ccc(cc2)C(F)(F)F)C/C=C/c3ccccc3.[I-].[I-] MS-2793 C[N+]1(CC[N+](CC1)(C)Cc2ccc(cc2)Br)C/C=C/c3ccccc3.[I-].[I-] MS-2795 c1ccc(cc1)/C=C/CN2CCN(CC2)Cc3ccc(cc3)C(F)(F)F MS-2796 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)c3ccc(cc3)Cl MS-2798 C#CC1(CCCCC1)NC(=O)[C@H]2C[C@H]2C(=O)O MS-2799 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCSC(C)(C)C MS-2800 CC(C)(C)SCCNC(=O)[C@H]1C[C@H]1C(=O)O MS-2802 CC(C)(C)SCCNC1=C(C(=O)c2ccccc2C1=O)Cl MS-2803 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)c3ccc(cc3)F MS-2804 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)C/C=C/c3ccccc3 MS-2805 CC(C)(C)SCCNC(=O)Nc1cccc(c1)C(F)(F)F MS-2806 Cc1ccc(cc1)Nc2ccccc2N.Cl MS-2807 c1cc2cn[nH]c2cc1NC(=O)CN3CCOCC3 MS-2808 Cc1ccc(cc1)S(=O)(=O)NCCSC(C)(C)C MS-2809 CC(C)(C)SCCNS(=O)(=O)c1ccc(cc1)F MS-2810 c1cc2cn[nH]c2cc1NC(=O)CN3CCCCC3 MS-2811 CC(C)(C)SCCNS(=O)(=O)c1ccc(cc1)Cl MS-2812 CC(C)(C)SCCNS(=O)(=O)c1ccc(cc1)[N+](=O)[O-] MS-2813 CN(C)CC(=O)Nc1ccc2cn[nH]c2c1 MS-2814 Cc1ccc(n1c2ccc3cn[nH]c3c2)C MS-2815 Cc1cc(c(n1c2ccc3cn[nH]c3c2)C)C(=O)C(=O)O MS-2816 Cc1ccc(cc1)n2c(c(cn2)C#N)N(Cc3ccc(cc3)C(C)(C)C)Cc4ccc(cc4)C(C)(C)C MS-2817 COC(=O)c1c(ccs1)OCc2ccc(cc2)Br MS-2818 COC(=O)COc1ccsc1C(=O)OC MS-2819 COc1ccsc1C(=O)NCCN2CCOCC2 MS-2821 COc1ccsc1C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 MS-2822 COc1ccsc1C(=O)N2CCN(CC2)c3cccc(c3)C(F)(F)F MS-2823 COc1ccsc1C(=O)NCC(OC)OC MS-2824 COc1ccsc1C(=O)N2CC3CC3C2C(=O)OC MS-2825 CCOC(=O)C(C)Oc1ccsc1C(=O)OC MS-2826 CC(C(=O)N(C)C)Oc1ccsc1C(=O)N(C)C MS-2827 COC(=O)c1c(c2cccnc2s1)NC(=O)NS(=O)(=O)c3ccccc3 MS-2828 Cc1ccc(cc1)S(=O)(=O)Nc2ccsc2C#N MS-2830 c1ccc2c(c1)c(=O)n(nn2)Cc3cccnc3 MS-2831 c1ccc2c(c1)c(=O)n(nn2)CCN3CCOCC3 MS-2832 c1ccc2c(c1)c(=O)n(nn2)Cc3ccncc3 MS-2833 c1ccc2c(c1)c(=O)n(nn2)Cc3ccccn3 MS-2834 COC(=O)Cn1c(=O)c2ccccc2nn1 MS-2835 c1ccc2c(c1)c(=O)n(nn2)CCCBr MS-2836 c1ccc2c(c1)c(=O)n(nn2)CCO MS-2837 c1cc(sc1)C(=O)NNC(=O)c2cccs2 MS-2838 CS/C(=C(/C#N)\C(=O)c1ccc(cc1)Cl)/N2CCN(CC2)Cc3ccc4c(c3)OCO4 MS-2840 CS/C(=C(/C#N)\C(=O)c1ccc(cc1)Cl)/NCCN2CCOCC2 MS-2841 COC(CN/C(=C(\C#N)/C(=O)c1ccc(cc1)Cl)/SC)OC MS-2842 CS/C(=C(/C#N)\C(=O)c1ccc(cc1)Cl)/NCc2cccnc2 MS-2843 CS/C(=C(/C#N)\C(=O)c1ccc(cc1)Cl)/NCc2ccncc2 MS-2844 Cc1ccc(cc1)n2c(c(cn2)C#N)N(Cc3ccc(c(c3)F)F)Cc4ccc(c(c4)F)F MS-2845 CC(C)(C)c1ccc(cc1)COc2c3c(cccc3F)ncn2 MS-2846 c1cc2c(c(c1)F)c(ncn2)OCc3ccc(cc3)F MS-2847 CC(=O)Oc1c2c(cccc2F)ncn1 MS-2848 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)c3cc(c(s3)Br)Br MS-2849 c1cc(cc(c1)N2CCN(CC2)C(=O)c3cc(c(s3)Br)Br)C(F)(F)F MS-2850 c1ccc2c(c1)C3N(C2=O)c4ccccc4C(=O)CS3 MS-2851 CC(=O)OC(c1c(cccc1F)F)C(=O)O MS-2852 CC(=O)OC(c1c(cccc1F)F)C(=O)NCCN2CCOCC2 MS-2853 CC(=O)OC(c1c(cccc1F)F)C(=O)NCc2ccc(cc2)OC MS-2854 CC(=O)OC(c1c(cccc1F)F)C(=O)Nc2nncs2 MS-2855 CC(=O)OC(c1c(cccc1F)F)C(=O)N2CCOCC2 MS-2856 C1COCCN1CCNc2c(c(ns2)Cl)C#N MS-2857 c1ccc(cc1)CCNc2c(c(ns2)Cl)C#N MS-2858 COc1ccc(cc1)CCNc2c(c(ns2)Cl)C#N MS-2859 CN(CCC#N)c1c(c(ns1)Cl)C#N MS-2860 CC(C)(C)c1ccc(cc1)Cn2cc(nc2)[N+](=O)[O-] MS-2861 c1ccc2c(c1)c(=O)n(nn2)Cc3ccc4c(c3)OCO4 MS-2863 c1ccc2c(c1)c(=O)n(nn2)CCCOc3ccc(cc3)F MS-2864 c1ccc2c(c1)c(=O)n(nn2)CCCOc3cc(cc(c3)Cl)Cl MS-2865 c1cc(ccc1C(=O)Cn2c3c(sc2=N)CCCC3)Cl.Br MS-2866 c1ccc(cc1)C(=O)Cn2c3c(sc2=N)CCCC3.Br MS-2869 c1ccc(cc1)c2cn3c4c(sc3n2)CCCC4 MS-2870 c1cc(sc1)C(=O)N/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)Cl MS-2872 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/NC(=O)c5ccsc5)Cl MS-2873 c1cscc1C(=O)NN MS-2874 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)CO)Cl MS-2875 c1ccc(cc1)C(=O)Nc2c(c(ns2)Cl)C#N MS-2877 Cc1cccc(c1)C(=O)Nc2c(c(ns2)Cl)C#N MS-2878 c1ccc(c(c1)C(=O)Nc2c(c(ns2)Cl)C#N)F MS-2879 c1ccc(cc1)c2c(n3c4c(sc3n2)CCCC4)C(=O)C(F)(F)F MS-2881 COC(=O)c1ccc(c(c1)F)n2cncn2 MS-2883 c1cc(ccc1C(=O)Cn2c3c(sc2=N)CCCC3)F MS-2884 c1cc(ccc1c2cn3c4c(sc3n2)CCCC4)F MS-2886 CSc1nc[nH]n1 MS-2889 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)C=O)F MS-2890 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)CO)F MS-2894 c1cc(sc1)C(=O)N/N=C/c2c(nc3n2c4c(s3)CCCC4)c5ccc(cc5)F MS-2895 c1cc(ccc1c2c(n3c4c(sc3n2)CCCC4)/C=N/O)F MS-2896 c1cc(ccc1c2cn3c4c(sc3n2)CCCC4)[N+](=O)[O-] MS-2897 CC(=O)Nc1ccc(cc1)c2cn3c4c(sc3n2)CCCC4 MS-2898 c1cc(ccc1c2cn3c4c(sc3n2)CCCCC4)Cl MS-2901 c1cc(ccc1c2cn3c4c(sc3n2)CCCC4)N MS-2902 COC(=O)c1ccc(nc1)n2c3c(cn2)CCCC3 MS-2903 C1CCc2c(sc(n2)N)CC1 MS-2904 c1[nH]nc(n1)Cl MS-2906 COC(=O)c1ccc(c(c1)F)n2cnc(n2)Cl MS-2907 CC(C)C(=O)Nc1ccc(cc1)c2cn3c4c(sc3n2)CCCC4 MS-2908 Cc1nc[nH]n1 MS-2909 Cc1ncn(n1)c2ccc(cn2)C(=O)OC MS-2910 COC(=O)c1cc(c(c(c1)F)n2cncn2)F MS-2911 c1ccc(cc1)c2cn3c4c(sc3n2)CCCCC4 MS-2912 COC(=O)c1ccc(nc1)n2cnc(n2)c3ccccc3 MS-2914 Cc1ncn(n1)c2ccc(cc2F)C(=O)OC MS-2915 Cc1ccc(n1c2cnccn2)C MS-2919 Cc1cc(c(n1c2cnccn2)C)C(=O)C(F)(F)F MS-2920 Cc1cc(c(n1c2cnccn2)C)C=O MS-2921 CCCCNC(=O)N1CCN(CC1)C(=O)NCCCC MS-2922 Cc1cc(c(n1c2cnccn2)C)C(=O)C(=O)O MS-2923 Cc1cc(c(n1c2cnccn2)C)/C=N/NC(=O)c3ccsc3 MS-2924 Cc1cc(c(n1c2cnccn2)C)/C=N/NC(=O)c3cccs3 MS-2925 Cc1cc(c(n1c2cnccn2)C)/C=C\3/C(=O)NC(=O)S3 MS-2926 c1cc(sc1)C(=O)N/N=C/c2ccc(cc2)n3ccnc3 MS-2928 Cc1ccc(cc1)C(c2ccc(cc2)n3ccnc3)O MS-2929 c1cc(ccc1C(c2ccc(cc2)Cl)O)n3ccnc3 MS-2931 CCCCCCOc1cccc(c1)O MS-2932 CN(C1CCCC1)C(=O)Nc2cccc(c2)Cl MS-2933 CC(C)N(c1ccccc1)c2c(c(ncn2)NCCC(=O)O)[N+](=O)[O-] MS-2934 c1cc(c(cc1Cl)Cl)OCCCN.Cl MS-2936 c1cc(c(c(c1)Cl)OCCCN)Cl.Cl MS-2937 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(c2ccccc2)C(C)C MS-2938 COc1cc(ccc1O)/C=N/NC(=O)c2cccs2 MS-2940 CC(C)N(c1ccccc1)c2c(c(ncn2)NC(CCS(=O)(=O)C)C(=O)O)[N+](=O)[O-] MS-2942 CC(C)N(c1ccccc1)c2c(c(ncn2)NC(Cc3ccccc3)C(=O)O)[N+](=O)[O-] MS-2943 Cc1cccc(c1)C(=O)Nc2c(c3c(s2)CCCC3)C#N MS-2945 c1ccc(cc1)c2nc([nH]n2)S MS-2946 Cc1nc([nH]n1)S MS-2947 CCOC(=O)CN1C(=O)Nc2ccccc2C(=O)N1C(C)(C)C MS-2948 CC(C)(C)N1C(=O)c2ccccc2NC(=O)N1CC#N MS-2949 Cc1cccc(c1)C(=O)Nc2ccccc2C(=O)N(C(C)(C)C)NC(=O)c3cccc(c3)C MS-2950 CC(C)(C)N(C(=O)c1ccccc1N)NC(=O)c2cccc(c2)OC MS-2951 CC(C)(C)N(C(=O)c1ccccc1NC(=O)c2cccs2)NC(=O)c3cccs3 MS-2952 CCCCNC(=O)NN(C(=O)c1ccccc1N)C(C)(C)C MS-2953 CC(C)(C)OC(=O)NCCCOc1ccc(c(c1)O)C(=O)OC MS-2954 CC(C)(C)N(C(=O)c1ccccc1N)NC(=O)Nc2ccccc2 MS-2955 CC(C)(C)N(C(=O)c1ccccc1NC(=O)c2cccc(c2)C(F)(F)F)NC(=O)Nc3ccccc3 MS-2956 CCOCCN1C(=O)Nc2ccccc2C(=O)N1C(C)(C)C MS-2957 Cc1cccc(c1)C(=O)Nc2ccccc2C(=O)N(C(C)(C)C)NC(=O)Nc3ccccc3 MS-2958 Cc1c(c(on1)C)C(=O)Nc2ccccc2C(=O)N(C(C)(C)C)NC(=O)Nc3ccccc3 MS-2959 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2C(=O)N(C(C)(C)C)NC(=O)Nc3ccccc3 MS-2960 CC(C)(C)N1C(=O)c2ccccc2NC(=O)N1CCCN3C(=O)c4ccccc4C3=O MS-2961 CN(C)S(=O)(=O)c1ccc(cc1)CN.Cl MS-2963 CC(C)N(c1ccccc1)c2c(c(ncn2)Nc3ccccc3)[N+](=O)[O-] MS-2964 CN(C1CCCC1)C(=O)Nc2ccc(cc2Cl)Cl MS-2965 c1ccc2c(c1)c(c(s2)Cl)CC(=O)O MS-2967 c1cc(sc1)C(=O)NNCCC#N MS-2968 c1cc(sc1)c2nn(c(=S)o2)CCC#N MS-2970 c1cc(sc1)c2n[nH]c(=S)o2 MS-2971 c1cc(sc1)c2nn(c(=O)o2)CCC#N MS-2972 c1cc(cc(c1)OCc2ccc(cc2)F)C(=O)NN MS-2973 COC(=O)c1cccc(c1)OCc2ccc(cc2)F MS-2974 c1cc(cc(c1)OCc2ccc(cc2)F)c3n[nH]c(=S)o3 MS-2975 c1cc(ccc1COc2ccc(cc2)c3n[nH]c(=O)o3)F MS-2976 c1ccc(cc1)CNc2c(c(ncn2)Cl)[N+](=O)[O-] MS-2977 CC(C)NC(=O)NNC(=O)c1cccc(c1)OCc2ccc(cc2)F MS-2978 c1ccc(cc1)CCNc2c(c(ncn2)NCCc3ccccc3)[N+](=O)[O-] MS-2979 CC(C)(C)NC(=S)NCc1ccco1 MS-2980 Cc1cc(ccc1C(C)C)NC(=O)N(C)C MS-2981 CC(C)(C)NC(=S)NCc1cccnc1 MS-2982 c1cc(cnc1)CNC(=S)N MS-2983 c1ccc(cc1)Nc2c(ccc(n2)Cl)[N+](=O)[O-] MS-2984 CC(C)(C)NC(=S)NCc1ccncc1 MS-2985 c1ccc(cc1)c2csc(n2)NCc3cccnc3 MS-2986 c1cc(cnc1)CNc2nc(cs2)c3ccc(cc3)Cl MS-2987 CC(C)(C)n\1c(cs/c1=N\Cc2ccncc2)c3ccccc3 MS-2988 CC(C)(C)n\1c(cs/c1=N\Cc2ccncc2)c3ccc(cc3)Cl MS-2989 CC(C)N(C1CCCCC1)C(=O)Nc2cccc(c2)Cl MS-2991 CC(C)N(C1CCCCC1)C(=O)Nc2ccc(cc2)Cl MS-2992 CC(C)N(C1CCCCC1)C(=O)Nc2cccc(c2)C(F)(F)F MS-2993 CCc1[nH]c(=O)c2ccccc2n1 MS-2994 CC(c1[nH]c(=O)c2ccccc2n1)Br MS-2995 CC(c1[nH]c(=O)c2ccccc2n1)N3CCOCC3 MS-2996 CC(c1[nH]c(=O)c2ccccc2n1)N3CCCCC3 MS-2997 CC(c1[nH]c(=O)c2ccccc2n1)N3CCN(CC3)C MS-2998 CC(c1[nH]c(=O)c2ccccc2n1)NCc3ccccc3 MS-2999 CC(c1[nH]c(=O)c2ccccc2n1)NCc3ccc(cc3)Cl MS-3000 CC(c1[nH]c(=O)c2ccccc2n1)NCCc3ccccc3 MS-3001 c1ccnc(c1)CNC(=O)Nc2ccc(cc2F)F MS-3002 CC(C)(C)n\1c(cs/c1=N\Cc2cc[n+](cc2)C)c3ccccc3.[I-] MS-3003 CC(C)(C)n\1c(cs/c1=N\Cc2cccnc2)c3ccccc3 MS-3004 CC(C)(C)n\1c(cs/c1=N\Cc2cccnc2)c3ccc(cc3)Cl MS-3005 CC(C)N(C1CCCCC1)C(=O)Nc2ccc(cc2F)F MS-3006 CC(C)(C)n\1c(cs/c1=N\Cc2ccco2)c3ccc(cc3)Cl MS-3007 CC(C)(C)n\1c(cs/c1=N\Cc2cccnc2)c3ccc(cc3)OC MS-3009 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCc3ccccn3 MS-3010 CC(C)(C)n\1c(cs/c1=N\Cc2ccco2)c3ccc(cc3)OC MS-3011 CC(C)(C)n\1c(cs/c1=N\Cc2ccco2)c3ccccc3 MS-3012 CC(C)(C)n\1c(cs/c1=N\Cc2ccc(cc2)Cl)c3ccc(cc3)OC MS-3013 CC(C)(C)n\1c(cs/c1=N\Cc2ccc(cc2)Cl)c3ccc(cc3)F MS-3014 CC(C)(C)n\1c(cs/c1=N\Cc2ccc(cc2)Cl)c3ccccc3 MS-3015 CC(C)(C)n\1c(cs/c1=N\Cc2ccc(cc2)Cl)c3ccc(cc3)Cl MS-3016 COc1ccc(cc1)c2csc(n2)NCc3ccc(cc3)Cl MS-3018 CCOC(=O)c1ccccc1N(C)S(=O)(=O)C MS-3020 CN1c2ccccc2C(=O)CS1(=O)=O MS-3021 c1c(cc(c(c1Br)O)Br)CC(C(=O)O)N MS-3024 CN(c1ccsc1C(=O)OC)S(=O)(=O)C MS-3025 CN1c2ccsc2C(=O)CS1(=O)=O MS-3028 CCc1nc2ccccc2c(=O)n1CC(=O)OCC MS-3029 CCCCCNC(C)c1[nH]c(=O)c2ccccc2n1 MS-3030 CCOC(=O)Cn1c(=O)c2ccccc2nc1C(C)Br MS-3032 CCCCCN(C(C)c1[nH]c(=O)c2ccccc2n1)C(=O)CCl MS-3033 CCOC(=O)Cn1c(=O)c2ccccc2nc1C(C)N3CCOCC3 MS-3034 CCCCCN(C(C)c1[nH]c(=O)c2ccccc2n1)C(=O)C MS-3035 CCCCCN1C(c2nc3ccccc3c(=O)n2CC1=O)C MS-3036 c1ccc(cc1)C2=NCC(=O)Nc3c2cccc3 MS-3038 CN(C)N1C(=O)CCC1=O MS-3040 c1ccc2c(c1)C(=O)CS(=O)(=O)N2Cc3ccc(c(c3)F)F MS-3041 CCOC(=O)c1ccccc1N(Cc2ccc(c(c2)F)F)S(=O)(=O)C MS-3042 CC(=O)NC1=NN(C(=O)C1)c2ccccc2 MS-3045 Cc1ccc(cc1)CN2c3ccccc3C(=NCC2=O)c4ccccc4 MS-3046 c1ccc(cc1)NC(=O)N2CCCCC2 MS-3047 CN1c2ccsc2C(=C(S1(=O)=O)C(=O)NCc3ccccc3)O MS-3048 c1ccc(cc1)C2=NCC(=O)N(c3c2cccc3)Cc4ccc(cc4)C(F)(F)F MS-3049 c1cc(c(c(c1)F)C(=O)NCC(=O)O)F MS-3050 C/C(=C\1/C(=O)OC(=N1)c2c(cccc2F)F)/N(C)C MS-3051 C/C(=C\1/C(=O)OC(=N1)c2ccccc2)/N(C)C MS-3052 C/C(=C\1/C(=O)OC(=N1)c2ccc(cc2)Cl)/N(C)C MS-3053 c1ccc(cc1)C2=NCC(=O)N(c3c2cccc3)Cc4ccc(cc4)[N+](=O)[O-] MS-3055 c1ccc(cc1)C2=NCC(=O)N(c3c2cccc3)Cc4cccc(c4)Br MS-3056 CN(C)/C(=C/1\C(=O)OC(=N1)c2ccccc2)/CBr MS-3057 CN(C)/C(=C\1/C(=O)OC(=N1)c2ccccc2)/CN3CCCCC3 MS-3058 CN(C)/C(=C\1/C(=O)OC(=N1)c2ccccc2)/CN3CCOCC3 MS-3059 Cc1ccn2c(c1)ncc2/C(=C/3\C(=O)OC(=N3)c4ccccc4)/N(C)C MS-3060 CN(C)/C(=C\1/C(=O)OC(=N1)c2ccccc2)/CN3CCN(CC3)C=O MS-3061 CC(C)(C)c1ccc(cc1)CN2c3ccccc3C(=NCC2=O)c4ccccc4 MS-3062 CN1CCN(CC1)C/C(=C/2\C(=O)OC(=N2)c3ccccc3)/N(C)C MS-3063 CN(C)/C(=C/1\C(=O)OC(=N1)c2ccccc2)/Cn3cncn3 MS-3064 CN(C)/C(=C\1/C(=O)OC(=N1)c2ccccc2)/COc3ccc(cc3Cl)Cl MS-3065 CN(C)/C(=C/1\C(=O)OC(=N1)c2c(cccc2F)F)/Cn3cncn3 MS-3066 c1cc(cc(c1)O)NC(=O)C2C[C@@H]2C(=O)O MS-3069 c1cc(ccc1N2C(=O)CCC2=O)O MS-3070 CCc1nc2ccccc2c(=O)n1CCCN3C(=O)c4ccccc4C3=O MS-3071 CC(c1nc2ccccc2c(=O)n1CCCN3C(=O)c4ccccc4C3=O)Br MS-3073 COC(=O)c1ccc(nc1)N2CCOCC2 MS-3074 c1ccc2c(c1)c(=O)c(co2)N3CCOCC3 MS-3076 CC(C)NC(=O)c1ccc(nc1)N2CCOCC2 MS-3077 c1ccnc(c1)CNC(=O)c2ccc(nc2)N3CCOCC3 MS-3078 c1ccc2c(c1)c(=O)c(co2)N3CCCCC3 MS-3079 Cc1cc(ccc1F)NC(=C(C#N)C#N)SC MS-3084 Cc1cc(ccc1F)Nc2c(c([nH]n2)N)C#N MS-3085 Cc1cc(ccc1F)Nc2c(c([nH]n2)/N=C/N(C)C)C#N MS-3088 Cc1cccc(c1)S(=O)(=O)Nc2c(c(n[nH]2)Nc3ccc(c(c3)C)F)C#N MS-3089 Cc1cc(ccc1F)Nc2c(c([nH]n2)NS(=O)(=O)c3ccc(cc3)F)C#N MS-3090 Cc1cc(ccc1F)Nc2c(c(n(n2)C)N)C#N MS-3091 Cc1cc(ccc1F)Nc2c(c(nn2C)N)C#N MS-3092 Cc1cc(n(n1)C)NC(=O)NCc2ccccc2 MS-3094 c1ccc2c(c1)C(=O)NC3(N2)CCCC3 MS-3098 CCN1C(=O)c2ccccc2NC13CCCC3 MS-3099 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2ccccn2 MS-3105 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2cccnc2 MS-3106 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2ccncc2 MS-3107 Cc1cccc(c1NC(=O)NC(=N)NC)C MS-3109 c1cc(ccc1CC(=O)N)OCCN MS-3111 CC(C)(C)OC(=O)NCCOc1ccc(cc1)CC(=O)N MS-3113 c1ccc(cc1)COC2CCCN(C2)C(=O)C(F)(F)F MS-3114 c1cc(ccc1c2cc(c(o2)N)C#N)Cl MS-3117 c1cc(oc1)CN2[C@H](CCC2=O)C(=O)O MS-3118 c1ccc2c(c1)nc(c(n2)N3CCOCC3)N4CCOCC4 MS-3119 c1ccc2c(c1)nc(c(n2)N3CCCCC3)N4CCCCC4 MS-3120 c1ccn(c1)c2c(cc(o2)c3ccc(cc3)Cl)O MS-3121 c1cc(oc1)CNC(CCC(=O)O)C(=O)O MS-3122 CC(c1ccccc1)NC(=O)C2CCC(=O)N2Cc3ccco3 MS-3123 CN(Cc1ccccc1)C(=O)[C@H]2CCC(=O)N2Cc3ccco3 MS-3124 Cc1ccc(cc1)CNC(=O)[C@@H]2CCC(=O)N2Cc3ccco3 MS-3125 c1ccc2c(c1)C(N(C2=O)COc3cccc(c3)F)O MS-3126 c1ccc2c(c1)C(N(C2=O)COc3ccc(cc3Cl)Cl)O MS-3127 C[n+]1cccc(c1)CNC2=C(C(=O)c3ccccc3C2=O)Cl.[I-] MS-3128 c1ccc2c(c1)C3c4cc(cc(c4OCN3C2=O)Cl)Cl MS-3129 CCOC(=O)COC1c2ccccc2C(=O)N1COc3cccc(c3)F MS-3130 c1ccc2c(c1)C(=O)N(C2=O)Cn3ccnc3 MS-3132 c1ccc(cc1)CCNc2c(cccn2)[N+](=O)[O-] MS-3135 c1ccc(cc1)n2c(c(c(n2)CC#N)C#N)n3cccc3 MS-3138 CN(C)C(=O)C(=O)c1cccn1c2cccc(c2C#N)Cl MS-3139 CC(C)N(C)C(=O)C(=O)c1cccn1c2cccc(c2C#N)Cl MS-3140 CCN(CC)C(=O)C(=O)c1cccn1c2cccc(c2C#N)Cl MS-3141 c1ccn(c1)c2cccc(c2C#N)Cl MS-3142 c1ccn(c1)c2c(cc(o2)c3ccc(cc3)Cl)C/N=C\c4cccc(c4)F MS-3144 c1ccc(cc1)CC2[C@H](CCC2=O)C(=O)O MS-3146 c1coc2c1C(=O)C3CCC(=O)N3C2 MS-3148 CSc1c(nc2ccccc2n1)SC MS-3149 CC(c1ccccc1)NC(=O)[C@H]2CCC(=O)N2Cc3ccccc3 MS-3150 Cc1cccc(c1NC(=O)N/C(=N/C(=S)Nc2ccccc2)/NC)C MS-3152 c1c(cc(c(c1[N+](=O)[O-])O)Cl)F MS-3153 CC(C)(C)c1ccc(cc1)CSc2nc3cc(cc(c3o2)Cl)F MS-3154 c1cc(ccc1CSc2nc3cc(cc(c3o2)Cl)F)C(F)(F)F MS-3155 CN1CCN(CC1)c2nc3ccccc3o2 MS-3156 c1ccc2c(c1)nc(o2)S MS-3157 c1ccc(cc1)CCNc2c(cccn2)NC(=O)c3cccnc3Cl MS-3158 COCCNc1c(cccn1)[N+](=O)[O-] MS-3159 CCCc1[nH]c(=O)c2ccccc2n1 MS-3160 CCCc1nc2ccccc2c(=O)n1CC(=O)c3ccccc3 MS-3161 CCCc1nc2ccccc2c(=O)n1CC(=O)c3ccc(cc3)OC MS-3162 CC(C)c1[nH]c(=O)c2ccccc2n1 MS-3163 CCCc1nc2ccccc2c(=O)n1CC(=O)c3ccc(cc3)F MS-3164 c1ccn(c1)c2cccc(c2CN)Cl MS-3166 c1ccc(cc1)NC(=O)NCc2c(cccc2Cl)n3cccc3 MS-3167 CCCCNC(=O)NCc1c(cccc1Cl)n2cccc2 MS-3170 c1ccn(c1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F MS-3172 c1ccn(c1)c2ccc(cc2N)C(F)(F)F MS-3173 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(ccc2n3cccc3)C(F)(F)F MS-3175 Cc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2n3cccc3)C(F)(F)F MS-3176 c1ccc(cc1)S(=O)(=O)Nc2cc(ccc2n3cccc3)C(F)(F)F MS-3178 c1ccc2c(c1)c(=O)[nH]c(n2)CN3CCOCC3 MS-3180 c1cc(c(nc1)Cl)C(=O)Nc2nncs2 MS-3181 CN1CCN(CC1)Cc2[nH]c(=O)c3ccccc3n2 MS-3182 c1ccc(c(c1)C(=O)N)NC(=O)CN2CCOCC2 MS-3183 CC1CCCCN1CC(=O)Nc2ccccc2C(=O)N MS-3184 CC1CCCCN1Cc2[nH]c(=O)c3ccccc3n2 MS-3185 c1ccc(cc1)OCc2[nH]c(=O)c3ccccc3n2 MS-3187 CC1CN(CC(O1)C)Cc2[nH]c(=O)c3ccccc3n2 MS-3188 c1ccc(cc1)OCC(=O)Nc2ccccc2C(=O)N MS-3189 CCCCOc1ccc(cc1)C(=O)Nc2nncs2 MS-3190 c1cc(ccc1C(=O)Nc2nncs2)F MS-3192 CC(C)(C)c1nnc(s1)NC(=O)c2cccnc2Cl MS-3193 CC(C)(C)c1nnc(s1)NC(=O)c2cccnc2 MS-3194 CC(C)(C)c1nnc(s1)NC(=O)c2ccc(nc2)Cl MS-3195 CC(C)(C)c1nnc(s1)NC(=O)c2ccc(nc2Cl)Cl MS-3196 c1ccc(cc1)CC2CCN(CC2)CC(=O)Nc3ccccc3C(=O)N MS-3197 c1ccc(cc1)CN2CCN(CC2)Cc3[nH]c(=O)c4ccccc4n3 MS-3198 c1ccc(cc1)CC2CCN(CC2)Cc3[nH]c(=O)c4ccccc4n3 MS-3199 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccccc3C(=O)N MS-3200 c1cc(nc(c1C(=O)NCCN2CCCCC2)Cl)Cl MS-3201 c1ccc(c(c1)C(=O)N)NC(=O)CNCc2cccnc2 MS-3202 c1ccc2c(c1)c(=O)[nH]c(n2)CNCc3cccnc3 MS-3203 c1ccc(c(c1)CNCc2[nH]c(=O)c3ccccc3n2)Cl MS-3205 CCc1ccc(cc1)NCc2[nH]c(=O)c3ccccc3n2 MS-3206 c1ccc(c(c1)C(=O)N)NC(=O)CNCc2ccco2 MS-3207 c1ccn(c1)c2ccc(cc2)C#N MS-3208 CCN(CC)C(=O)C(=O)c1cccn1c2ccc(cc2)C#N MS-3209 c1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)n3cccc3 MS-3211 c1ccn(c1)c2ccc(cc2NC(=O)CCl)C(F)(F)F MS-3212 CCN(CC)CC(c1cccn1c2ccc(cc2)CN)O MS-3213 c1ccn(c1)c2ccc(cc2NC(=O)CN3CCCCC3)C(F)(F)F MS-3214 CCN(CC)CC(c1cccn1c2ccc(cc2)CNC(=O)NC(C)C)O MS-3216 c1ccc(c(c1)CN)n2cccc2 MS-3218 c1ccn(c1)c2ccc(cc2NC(=O)CN3CCOCC3)C(F)(F)F MS-3220 CCN(CC)C(=O)C(=O)c1cccn1c2ccccc2C#N MS-3224 CN(C)C(=O)C(=O)c1cccn1c2ccccc2C#N MS-3225 c1cc(nc(c1C(=O)NCCN2CCOCC2)Cl)Cl MS-3226 CC(C)N(C(C)C)C(=O)C(=O)c1cccn1c2ccccc2C#N MS-3227 c1cc(ccc1SC2C(=O)NC(=O)S2)Cl MS-3228 c1ccc(c(c1)C(=O)N)NC(=O)CSc2ccc(cc2)Cl MS-3232 c1ccc2c(c1)c(=O)[nH]c(n2)CSc3ccc(cc3)Cl MS-3233 Cn\1ccs/c1=N\S(=O)(=O)c2ccc(cc2)Br MS-3234 Cc1ccc(cc1)S(=O)(=O)/N=c\2/n(ccs2)C MS-3235 CC(C)(C)c1ccc(cc1)Cn2c(nc3ccccc3c2=O)CSc4ccc(cc4)Cl MS-3237 CCCC(C(=O)O)Nc1ccccc1[N+](=O)[O-] MS-3238 CCCC1C(=O)Nc2ccccc2N1S(=O)(=O)c3ccccc3 MS-3239 CCCC1C(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)F MS-3240 c1ccc2c(c1)c(=O)[nH]c(n2)CS(=O)(=O)c3ccc(cc3)Cl MS-3241 c1ccc(c(c1)N)NC2CCCCC2 MS-3242 c1ccc(cc1)Cn2c(nc3ccccc3c2=O)CSc4ccc(cc4)Cl MS-3243 CCOC(=O)CSc1[nH]nc(n1)NS(=O)(=O)c2cccc(c2)C MS-3245 CCOC(=O)CSc1[nH]nc(n1)NS(=O)(=O)c2ccccc2C(F)(F)F MS-3246 CCOC(=O)CSc1[nH]nc(n1)NC(=O)c2cccc(c2)C MS-3247 CCOC(=O)CSc1[nH]nc(n1)NC(=O)c2ccc(cc2)F MS-3248 CCOC(=O)CSc1[nH]nc(n1)NC(=O)c2cccc(c2)C(F)(F)F MS-3249 CCOC(=O)CSc1[nH]nc(n1)NC(=O)c2ccccc2 MS-3250 CCOC(=O)CSc1[nH]nc(n1)NC(=O)NC(C)C MS-3251 CCCCNC(=O)Nc1nc([nH]n1)SCC(=O)OCC MS-3252 CCOC(=O)CSc1[nH]nc(n1)N MS-3253 CCOC(=O)CSc1[nH]nc(n1)NC(=O)C MS-3254 CCC(=O)Nc1nc([nH]n1)SCC(=O)OCC MS-3255 CCOC(=O)CSc1nnc(s1)NC(=O)NC(C)C MS-3256 Cc1cccc(c1)S(=O)(=O)Nc2nc([nH]n2)SCc3ccccc3C MS-3257 Cc1ccccc1CSc2[nH]nc(n2)NS(=O)(=O)c3ccccc3 MS-3258 Cc1ccccc1CSc2[nH]nc(n2)NC(=O)c3cccs3 MS-3260 Cc1ccccc1CSc2[nH]nc(n2)NC(=O)c3ccc(nc3)Cl MS-3261 Cc1ccccc1CSc2[nH]nc(n2)N MS-3263 CCCC1C(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3Cl)Cl MS-3264 CC(C)(C)c1ccc(cc1)S(=O)(=O)/N=c\2/n(ccs2)C MS-3265 CC(C)c1cc(c(c(c1)C(C)C)S(=O)(=O)/N=c\2/n(ccs2)C)C(C)C MS-3266 Cn\1ccs/c1=N\S(=O)(=O)c2ccc(cc2)F MS-3267 CC(C)c1ccc(cc1)COc2ccc(cc2)C(=O)N3CCOCC3 MS-3268 CC(C)c1ccc(cc1)COc2ccc(cc2)C(=O)O MS-3269 Cn\1ccs/c1=N/C(=O)C2CC2C(=O)O MS-3270 Cn\1ccs/c1=N\C(=O)Nc2ccccc2 MS-3271 Cc1ccc(cc1)S(=O)(=O)NC(=O)/N=c\2/n(ccs2)C MS-3272 CC(C)c1ccc(cc1)COc2cccc(c2)C(=O)N3CC(OC3)(C)C MS-3273 Cn\1ccs/c1=N\C(=O)Nc2cccc(c2)C(F)(F)F MS-3274 Cn\1ccs/c1=N\C(=O)Nc2cccc(c2)Cl MS-3275 CC(C)C12CCC(O1)(C(C2)OC(=O)Nc3cccc(c3)Cl)C MS-3276 COc1ccc(cc1)C(=O)Cn2cn[n+](c2)CC(=O)c3ccc(cc3)OC.[Br-] MS-3277 CC(C)C12CCC(O1)(C(C2)OCc3ccccc3)C MS-3278 c1ccc(cc1)C(=O)Cn2cnc(n2)N MS-3279 CC(C)c1ccc(cc1)COc2ccc(cc2)C(=O)NCc3cccnc3 MS-3280 CC1(COCN1C(=O)/C(=C/c2ccc(cc2)OC)/C#N)C MS-3281 COc1ccc(cc1)/C=C(\C#N)/C(=O)N2CCOCC2 MS-3282 COc1ccc(cc1)/C=C(/C#N)\C(=O)O MS-3283 COc1ccc(cc1)/C=C(\C#N)/C(=O)NCc2cccnc2 MS-3284 COc1ccc(cc1)/C=C(\C#N)/C(=O)NCC(=O)O MS-3285 CCN(CC)C(=O)/C(=C/c1ccc(cc1)OC)/C#N MS-3286 COc1ccc(cc1)/C=C(\C#N)/C(=O)NCc2ccco2 MS-3287 c1ccc(cc1)Nc2nnc(s2)SCc3ccc(cc3)C#N MS-3288 C=CCNc1n[nH]c(=S)s1 MS-3289 CC(C)(C)c1ccc(cc1)CSc2nnc(s2)Nc3ccccc3 MS-3290 c1ccc(cc1)Nc2nnc(s2)SCc3ccc(c(c3)Cl)Cl MS-3291 c1ccc(cc1)Nc2nnc(s2)SCc3ccc(cc3)F MS-3292 C=CCN(c1n[nH]c(=S)s1)C(=O)NCc2ccccc2 MS-3294 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(c2ccccc2)c3n[nH]c(=S)s3 MS-3296 c1ccc(cc1)Nc2nnc(s2)SCC#N MS-3299 CCOC(=O)CSc1nnc(s1)Nc2ccccc2 MS-3300 C=CCNc1nnc(s1)SCC(=O)O MS-3301 CCOC(=O)CSc1nnc(s1)NC(=O)NCCOc2ccc(cc2)Cl MS-3302 CC(c1ccccc1)NC(=O)CC#N MS-3303 CC(c1ccccc1)NC(=O)/C(=C/c2ccccc2F)/C#N MS-3304 c1ccc(cc1)CNC(=O)/C(=C\c2ccccc2F)/C#N MS-3305 CC(=O)Oc1cccc(c1)/C=C(\C#N)/C(=O)NCc2ccc(cc2Cl)Cl MS-3306 c1ccc(cc1)CNC(=O)/C(=C/c2cccc(c2)Cl)/C#N MS-3307 c1ccc(cc1)CNC(=O)/C(=C/c2ccc(cc2)Br)/C#N MS-3309 CCCCNC(=O)Nc1nnc(s1)SCC(=O)OCC MS-3310 CCOC(=O)CSc1nnc(s1)NC(=O)OCc2cc3ccccc3o2 MS-3311 c1ccn(c1)c2cccc(c2N)C(F)(F)F MS-3312 CCOC(=O)CSc1nnc(s1)N(C(=O)OCc2ccc(cc2)F)C(=O)OCc3ccc(cc3)F MS-3313 CC(CN1C(SCC1=O)c2cccc(c2)C(F)(F)F)O MS-3314 CCOC(=O)CSc1nnc(s1)NC(=O)Nc2ccccc2 MS-3316 CCOC(=O)CSc1nnc(s1)NC(=O)NC2CCCCC2 MS-3317 CCOC(=O)CSc1nnc(s1)NC(=O)OCc2ccc(cc2)F MS-3318 c1ccc(cc1)CN2C(SCC2=O)c3cccc(c3)C(F)(F)F MS-3319 c1cc(cc(c1)C(F)(F)F)C2N(C(=O)CS2)Cc3ccc(cc3)Cl MS-3320 CCOC(=O)/C=C\1/CSc2ccccc2N1 MS-3321 c1ccc(cc1)CN2C(SCC2=O)c3cccc(c3)O MS-3322 CCCCNC(=O)Oc1cccc(c1)C2N(C(=O)CS2)Cc3ccccc3 MS-3323 c1ccc(cc1)CN2C(SCC2=O)c3cccc(c3)OC(=O)Nc4ccccc4 MS-3324 Cc1cccc(c1)n2c(c(cn2)C#N)n3cccc3 MS-3334 c1ccn(c1)c2cccc(c2C#N)F MS-3335 Cc1cccc(c1)n2c(c(cn2)CN)n3cccc3 MS-3336 c1ccn(c1)c2cc(ccc2C#N)Cl MS-3340 c1ccc(c(c1)N)n2ccnc2 MS-3342 c1ccc(c(c1)NC(=O)Nc2cccc(c2)C(F)(F)F)n3ccnc3 MS-3344 c1ccc(c(c1)NC(=O)Nc2cccc(c2)Cl)n3ccnc3 MS-3345 c1ccc(cc1)NC(=O)Nc2ccccc2n3ccnc3 MS-3346 Cc1cccc(c1NC(=O)Nc2ccccc2n3ccnc3)C MS-3347 CCOC(=O)Nc1ccccc1C(=O)C(C#N)c2ccccc2 MS-3351 CCOc1nc2ccccc2c(=O)o1 MS-3353 CC(C(=O)O)Sc1cnccn1 MS-3354 CCC(C)O/C(=N/c1cccnc1)/c2ccc(cc2Cl)Cl MS-3361 CC(C)(C)C(=O)N(Cc1ccc(cc1)Cl)c2cnccn2 MS-3362 CCOC(=O)C(C)Sc1cnccn1 MS-3363 CCc1ccc(cc1)/N=C/c2ccc(cc2)Oc3cnccn3 MS-3364 Cc1cc(c(n1c2ccc(cc2)Cl)C)/C=N/c3ccccc3F MS-3365 Cc1cc(c(n1c2ccc(cc2)Cl)C)/C=N/c3cccc(c3)Cl MS-3366 CCc1ccc(cc1)/N=C/c2cc(n(c2C)c3ccc(cc3)Cl)C MS-3367 c1ccc2c(c1)cc(o2)/C=C\3/C(=O)NC(=O)S3 MS-3368 Cc1cc(c(n1c2ccc(cc2)Cl)C)/C=N/NC(=O)c3ccsc3 MS-3369 Cc1cccc(c1NC(=O)Nc2ccc3c(c2)nns3)C MS-3370 c1ccc2c(c1)cc(o2)CC3C(=O)NC(=O)S3 MS-3371 CC(C)(C)c1cccc(c1)Oc2nnnn2Cc3ccc(c(c3)Cl)Cl MS-3372 CC(=O)N(Cc1ccc(cc1)Cl)c2cnccn2 MS-3373 Cc1ccc(cc1)CN(c2cnccn2)C(=O)C(F)(F)F MS-3374 c1cc(ccc1CN(c2cnccn2)C(=O)C(F)(F)F)Cl MS-3375 CC(C)NC(=O)Nc1ccc2c(c1)nns2 MS-3376 CCc1ccc(cc1)NCc2ccc(cc2)Oc3cnccn3 MS-3377 c1cc(ccc1CC#N)/N=C/c2ccc(cc2)Oc3cnccn3 MS-3378 Cc1cc(c(cc1N(=O)=O)Cl)C(C#N)c2ccc(cc2)Cl MS-3379 c1ccc(cc1)NC(=O)NCc2ccccc2n3cccc3 MS-3380 c1ccc(c(c1)CNC(=O)c2ccc(cc2)OC(F)(F)F)n3cccc3 MS-3381 CCCc1ccc(cc1)C(=O)NCc2ccccc2n3cccc3 MS-3382 c1ccc(c(c1)CNC(=O)c2cccc(c2)C(F)(F)F)n3cccc3 MS-3383 c1ccc(c(c1)CNC(=O)NCc2ccccc2n3cccc3)n4cccc4 MS-3384 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)CN3CCOCC3 MS-3385 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)CN3CCCCC3 MS-3386 Cc1ccc(c2c1CC(O2)(C)C)NC(=O)CN3CCCC3 MS-3387 C1CS/C(=N\C#N)/N1 MS-3389 C1CS/C(=C/[N+](=O)[O-])/N1 MS-3390 C1CN/C(=N\C#N)/SC1 MS-3391 C1CCN/C(=N\S(=O)(=O)C(F)(F)F)/C1 MS-3392 C1CN(/C(=C/[N+](=O)[O-])/N1)C/C=C/Cl MS-3393 C1C/C(=N\S(=O)(=O)C(F)(F)F)/NC1 MS-3394 CN(Cc1ccc(nc1)Cl)C/C(=C\2/NCCCS2)/[N+](=O)[O-] MS-3395 c1c(cc(nc1Cl)Cl)[N+](=O)[O-] MS-3396 C1C/C(=C\[N+](=O)[O-])/NC1 MS-3397 CN/C(=C/[N+](=O)[O-])/NCc1ccc(nc1)Cl MS-3398 c1cc(ncc1CN\2CCN/C2=C/[N+](=O)[O-])Cl MS-3399 CCc1c(c(ncn1)NCc2conc2c3ccc(cc3)C(C)(C)C)Cl MS-3400 C/C(=N/C#N)/NCCNc1ccc(nc1)Cl MS-3402 c1ccc(cc1)Oc2ccc(cc2)C(=O)NCc3ccncc3 MS-3403 c1ccc(cc1)Oc2ccc(cc2)C(=O)N3CC4CC4C3C(=O)O MS-3404 c1ccc(cc1)Oc2ccc(cc2)C(=O)N3CC(C3)C(=O)O MS-3405 Cc1ccc(c2c1CC(O2)(C)C)NS(=O)(=O)c3ccccc3 MS-3406 Cc1cccc(c1)S(=O)(=O)Nc2ccc(c3c2OC(C3)(C)C)C MS-3407 Cc1ccc(c2c1CC(O2)(C)C)NS(=O)(=O)c3ccccc3Cl MS-3408 CCc1ccc(cc1)CNc2ccc(c3c2OC(C3)(C)C)C MS-3409 Cc1ccc(c2c1CC(O2)(C)C)/N=C/c3ccc(cc3)C#N MS-3411 Cc1cccc(c1C#N)n2cccc2 MS-3412 Cc1cccc(c1CN)n2cccc2 MS-3413 Cc1ccc(c2c1CC(O2)(C)C)NCc3ccc(cc3)C#N MS-3414 c1cc(ccc1CNc2cnccn2)C#N MS-3416 Cc1ccc(c2c1CC(O2)(C)C)N(Cc3cccc(c3)Oc4cccc(c4)C(F)(F)F)C(=O)C MS-3420 CC(C)N(c1ccccc1)C(=O)c2ccc(cc2)Oc3ccccc3 MS-3421 CC(C)(C)C(C(Cc1ccccc1Cl)n2cncn2)O MS-3422 c1cc(c(c(c1)Cl)C#N)n2ccnc2 MS-3423 c1cc(c(c(c1)Cl)CN)n2ccnc2 MS-3425 COC(=O)c1cccn1c2cccc(c2C#N)Cl MS-3426 CCc1ccc(cc1)/C=N/Cc2c(cccc2Cl)n3cccc3 MS-3427 c1cc(c(c(c1)Cl)C#N)n2cncn2 MS-3430 Cc1cccc(c1NC(=O)NCc2c(cccc2Cl)n3cncn3)C MS-3431 c1ccc(cc1)S(=O)(=O)NCc2c(cccc2Cl)n3cncn3 MS-3432 c1cc(cc(c1)NC(=O)NCc2c(cccc2Cl)n3cncn3)C(F)(F)F MS-3434 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2c(cccc2Cl)n3ccnc3 MS-3435 Cc1cn(c2c1cccc2)c3cccc(c3C#N)Cl MS-3438 CCCCNC(=O)NCc1c(cccc1Cl)n2cc(c3c2cccc3)C MS-3439 Cc1cccc(c1NC(=O)NCc2c(cccc2Cl)n3cc(c4c3cccc4)C)C MS-3440 c1cc(cc(c1)C(F)(F)F)C(=O)NC(=O)NCc2c(cccc2Cl)n3ccnc3 MS-3441 c1cc(c(c(c1)Cl)CN)n2cccc2CO MS-3442 Cc1cn(c2c1cccc2)c3cccc(c3CN)Cl MS-3444 c1ccc2c(c1)ccn2c3cccc(c3C#N)Cl MS-3445 CC(C)C12CCC(O1)(C(C2)Oc3cccc(c3CN)Cl)C MS-3446 Cc1cccc(c1NC(=O)NCc2c(cccc2Cl)n3ccc4c3cccc4)C MS-3447 CC(C)(C)C(=O)C(Cc1ccccc1Cl)n2cncn2 MS-3448 CC(C)(C)C(=O)C(Cc1ccccc1)n2cncn2 MS-3449 c1cc(c(c(c1)F)n2cccc2C#N)F MS-3452 COc1cccc(c1C#N)n2cccc2 MS-3455 c1ccn(c1)c2c(cccc2Cl)C#N MS-3456 CCC(=O)NCc1c(cccc1Cl)n2cccc2 MS-3457 c1ccn(c1)c2cccc(c2CNC(=O)CCl)Cl MS-3459 CC(C)C12CCC(O1)(C(C2)OCc3ccccc3Cl)C MS-3463 CC1(OCC(O1)C2C(=C(C(=O)O2)O)OCC(=O)c3ccc(cc3)OC)C MS-3464 CC(C)C12CCC(O1)(C(C2)Oc3cccc(c3C#N)Cl)C MS-3466 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2c(cccc2Cl)OC3CC4(CCC3(O4)C)C(C)C MS-3467 CC(C)C12CCC(O1)(C(C2)Oc3cccc(c3CNS(=O)(=O)c4ccccc4)Cl)C MS-3468 CC(C)C12CCC(O1)(C(C2)Oc3cccc(c3CNC(=S)NCC=C)Cl)C MS-3469 c1ccn(c1)c2c(cccc2Cl)CNC(=O)C3CCCCC3 MS-3472 c1ccc(cc1)OCC(=O)NCc2c(cccc2Cl)n3cccc3 MS-3474 CC(=CC(=O)NCc1c(cccc1Cl)n2cccc2)C MS-3475 CC(C)C12CCC(O1)(C(C2)Oc3cccc(c3CNS(=O)(=O)c4ccc(cc4)Br)Cl)C MS-3478 CC(C)C12CCC(O1)(C(C2)Oc3cccc(c3CNS(=O)(=O)c4ccc(cc4)F)Cl)C MS-3479 CC(C)C12CCC(O1)(C(C2)Oc3cccc(c3CNC(=O)C4CC4C(=O)O)Cl)C MS-3481 c1ccc2c(c1)C(CCO2)Oc3cccc(c3C#N)Cl MS-3482 c1cc(ccc1C#N)Oc2cnccn2 MS-3483 c1ccc(c(c1)N)Sc2cnccn2 MS-3484 Cc1ccc(cc1)C(=O)N2CC(C2)C(=O)O MS-3485 c1ccc(cc1)NC(=O)Nc2ccccc2Sc3cnccn3 MS-3489 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccccc2Sc3cnccn3 MS-3490 c1ccc(cc1)S(=O)(=O)Nc2ccccc2Sc3cnccn3 MS-3491 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccccc2Sc3cnccn3 MS-3493 C=CCNC(=S)NCc1c(cccc1Cl)OC2CCOc3c2cccc3 MS-3494 Cc1ccc(cc1)S(=O)(=O)NC(=O)OC2CC3(CCC2(O3)C)C(C)C MS-3496 Cc1ccc(cc1)S(=O)(=O)N(Cc2ccccc2Cl)C(=O)OC3CC4(CCC3(O4)C)C(C)C MS-3497 Cc1ccc(cc1)S(=O)(=O)N(Cc2ccc(cc2)C#N)C(=O)OC3CC4(CCC3(O4)C)C(C)C MS-3498 Cc1ccc(cc1)S(=O)(=O)N(Cc2ccccc2)C(=O)OC3CC4(CCC3(O4)C)C(C)C MS-3499 CC(C)C12CCC(O1)(C(C2)OC(=O)Nc3ccccc3)C MS-3500 Cc1ccc(cc1)S(=O)(=O)NC(=O)OC2CCOc3c2cccc3 MS-3501 COc1ccccc1CCNC(=O)c2cccc(c2)F MS-3502 COc1cc(ccc1Oc2cnccn2)C=O MS-3503 c1cnc(cn1)Sc2nnc(s2)N MS-3504 CCC(=O)NCc1c(cccc1Cl)n2cc(c3c2cccc3)C MS-3505 COc1cc(ccc1Oc2cnccn2)/C=N/O MS-3506 COc1cc(ccc1Oc2cnccn2)/C=C\3/C(=O)NC(=O)S3 MS-3507 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2nnc(s2)Sc3cnccn3 MS-3511 COc1cccc(c1CNC(=O)c2ccc(cc2)C#N)n3cccc3 MS-3516 CN(C)C(=O)C(=O)c1cccn1c2cccc(c2C#N)OC MS-3517 c1cc([nH]c1)/C=C/2\C(=O)NC(=O)S2 MS-3518 CCCCCC1C(C/C(=C\c2ccc(cc2)Br)/C1=O)CC(=O)O MS-3519 CC(=O)OC1CC2CC1C3C2CC4C3O4 MS-3520 Cc1ccc(cc1)S(=O)(=O)NC(=O)OC2CC3CC2C4C3CC=C4 MS-3521 CCN(CC)C(=O)C(=O)c1cccn1c2cccc(c2C#N)OC MS-3523 CCN(C)C(=O)C(=O)c1cccn1c2cccc(c2C#N)OC MS-3524 CSc1cccc(c1C#N)n2cccc2 MS-3525 c1ccc2c(c1)C(=O)N(C2=O)CCOc3cccc(c3C#N)n4cccc4 MS-3526 c1ccn(c1)c2cccc(c2C#N)n3cccc3 MS-3527 c1ccn(c1)c2cccc(c2CN)n3cccc3 MS-3528 CCN(CC)C(=O)C(=O)c1cccn1c2cccc(c2C#N)n3cccc3C(=O)C(=O)N(CC)CC MS-3529 CSc1cccc(c1CN)n2cccc2 MS-3530 c1cc(ccc1CCC(=O)O)F MS-3533 c1ccc(c(c1)CCC(=O)O)F MS-3534 Cc1c(sc[n+]1Cc2ccccc2)CCO.[Cl-] MS-3535 CCOC(C)C(=O)Nc1c2c([nH]cn2)ncn1 MS-3537 CN(C)CCOc1cc(cc(c1)Cl)Cl MS-3540 C[N+](C)(C)CCOc1cc(cc(c1)Cl)Cl.[I-] MS-3541 CCN(CC)C(=O)C(=O)c1cccn1c2c(cccc2Cl)C#N MS-3543 CCc1ccc(cc1)C(=O)NCc2c(cccc2n3cccc3)n4cccc4 MS-3544 c1ccn(c1)c2cccc(c2CNC(=O)c3ccc(c(c3)Cl)Cl)n4cccc4 MS-3545 Cc1cc(cc(c1)OCCN(CCOC)Cc2ccc(cc2)Cl)C MS-3547 Cc1cc(cc(c1)OCC(=O)N(CCOC)Cc2ccc(cc2)Cl)C MS-3548 c1cc([nH]c1)/C=C/2\C(=O)NC(=S)S2 MS-3549 CC(=O)Nc1nnc(s1)Sc2cnccn2 MS-3550 CCOC(=O)COc1cccc(c1)CCNC(=O)c2ccccc2 MS-3552 COc1cccc(c1)C(=O)N2CC3CC3C2C(=O)O MS-3554 COc1cccc(c1)CCNC(=O)c2ccc(cc2)C#N MS-3555 CC(C)Oc1cccc(c1)CCN MS-3556 c1cc(cc(c1)OC2CCCC2)CCN MS-3557 c1ccc(cc1)COc2cccc(c2)CCN MS-3558 c1cc(c(cc1F)F)NC(=O)c2cc(cnc2)Br MS-3560 COC(=O)c1cccc(n1)Cl MS-3561 c1cc(cc(c1)Oc2cccc(n2)C(=O)Nc3cc(cc(c3)F)F)C(F)(F)F MS-3562 c1cc(nc(c1)Cl)C(=O)Nc2cc(cc(c2)F)F MS-3563 c1cc(cc(c1)Oc2cccc(n2)C(=O)Nc3ccc(cc3F)F)C(F)(F)F MS-3564 c1cc(cc(c1)Oc2cc(ccn2)C(=O)Nc3ccc(cc3F)F)C(F)(F)F MS-3565 c1cc(cc(c1)Oc2c(cccn2)C(=O)Nc3ccc(cc3F)F)C(F)(F)F MS-3566 CCN(CC)C(=O)/C(=C\c1ccc2c(c1)OCO2)/C#N MS-3567 c1cc2c(cc1/C=C(/C#N)\C(=O)N3CCOCC3)OCO2 MS-3568 Cc1ccc(c(c1)C)COC2CC(SC3C2C=C(C=C3)Cl)C MS-3569 CC(C)(C)OC(=O)N1CC(C1)C(=O)O MS-3571 Cc1cc(n2cc(nc2n1)c3ccc(cc3)Cl)O MS-3573 CCOC(=O)COc1cc(nc2n1cc(n2)c3ccc(cc3)Cl)C MS-3578 Cc1cc(cc(=O)[nH]1)O MS-3580 Cc1cc(c(c(=O)[nH]1)[N+](=O)[O-])O MS-3581 CCOC(=O)COc1cc(nc2n1cc(n2)c3ccccc3)C MS-3582 Cc1cc(n2cc(nc2n1)c3ccccc3)OCC(=O)O MS-3583 Cc1cc(on1)NC(=O)c2ccc(cc2)C#N MS-3584 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(no2)C MS-3585 CC1CC(C2C=C(C=CC2S1)Cl)OCc3ccc(cc3)C(C)(C)C MS-3586 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(nn2C)C MS-3587 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(cc(cn2)C(F)(F)F)C(F)(F)F MS-3588 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(cc(cn2)Cl)C(F)(F)F MS-3589 c1ccn(c1)c2c(cccn2)C#N MS-3590 CC1CC(C2C=C(C=CC2S1)Cl)O MS-3591 CC1CC(C2C=C(C=CC2S1)Cl)OC(=O)Nc3ccccc3 MS-3592 CC1CC(C2C=C(C=CC2S1)Cl)OC(=O)Nc3cccc(c3)C(F)(F)F MS-3593 CC1CC(C2C=C(C=CC2S1)Cl)OCc3cccc(c3)OC MS-3594 c1ccc(cc1)CCNc2cnccn2 MS-3596 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(CCc2ccccc2)c3cnccn3 MS-3597 c1ccc(cc1)CC(C(=O)O)NC(=O)COc2ccc(c(c2)Cl)Cl MS-3598 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)CC#N MS-3600 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(nc(n2)C)C MS-3601 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(on2)C MS-3602 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2nnc(s2)C3CC3 MS-3603 CCCNC(=O)Nc1nnc(s1)C2CC2 MS-3604 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2c3ccccc3C(=O)NC2(C)C MS-3605 CC1(Nc2ccccc2C(=O)N1)C MS-3606 Cc1cc2c(cc(c(=O)o2)C(=O)CC(=O)C)c(=O)o1 MS-3607 CC1=CC(=O)/C(=C/NNc2ccccc2)/C(=O)O1 MS-3608 CC1=CC(=O)/C(=C/NNc2ccccc2Cl)/C(=O)O1 MS-3609 CC1=CC(=O)/C(=C/NNc2ccc(cc2)F)/C(=O)O1 MS-3610 CC1(Nc2ccccc2C(=O)N1Cc3ccc(c(c3)Cl)Cl)C MS-3611 Cc1ccc(cc1)S(=O)(=O)N2CC3CC3C2C(=O)O MS-3612 c1cc(ccc1S(=O)(=O)N2CC3CC3C2C(=O)O)Br MS-3613 c1cc(ccc1F)S(=O)(=O)N2CC3CC3C2C(=O)O MS-3614 Cc1ccc(cc1)S(=O)(=O)NCCOc2ccc(cc2Cl)Cl MS-3615 c1cc(ccc1F)S(=O)(=O)NCCOc2ccc(cc2Cl)Cl MS-3616 c1cc(ccc1F)S(=O)(=O)N2CC(C2)C(=O)O MS-3617 Cc1ccc(cc1)S(=O)(=O)N2CC3CC3C2C(=O)Nc4ccc(cc4)Cl MS-3618 c1c(c(cc(c1S(=O)(=O)N2CC3CC3C2C(=O)O)Cl)Cl)C(=O)O MS-3619 Cc1ccc(cc1)S(=O)(=O)N2CC3CC3C2C(=O)Nc4ccc(cc4)F MS-3620 Cc1ccc(c(c1)Oc2cnccn2)C(C)C MS-3621 CCOC(=O)CSc1[nH]c(=O)c2ccccc2n1 MS-3625 c1cc(ncc1C(=O)O)NN MS-3627 Cc1cc(ccc1C(C)C)NC(=O)/C=N/O MS-3629 CC(=O)NCc1c(cccc1Cl)n2cccc2 MS-3631 CCOC(=O)c1cc([nH]n1)c2ccc(cc2)Cl MS-3645 c1ccn(c1)c2cccc(c2CNC(=O)c3ccc(c(c3)F)C(F)(F)F)Cl MS-3646 Cc1cc(c(cc1C)O)C2(c3ccccc3NC2=O)O MS-3650 c1ccc2c(c1)ccn2S(=O)(=O)c3ccc(cc3)Br MS-3651 Cc1cc(c(cc1C)O)C2(c3ccc(cc3NC2=O)Br)O MS-3652 CC(C)c1ccc(c(c1)O)C2(c3ccccc3NC2=O)O MS-3653 CC(C)c1ccc(c(c1)O)C2(c3ccc(cc3NC2=O)Br)O MS-3654 c1ccc2c(c1)C(C(=O)N2)(c3ccccc3O)O MS-3655 c1ccc(c(c1)C2(c3ccc(cc3NC2=O)Br)O)O MS-3656 Cc1cc(ccc1F)C2(c3ccccc3NC2=O)O MS-3657 Cc1cc2c(cc1F)C(C(=O)N2)(c3ccc(cc3O)C(C)C)O MS-3659 c1cnccc1N2CCNC2=O MS-3660 CCO/N=C/C(=O)Nc1ccc(cc1F)F MS-3661 c1cc(c(cc1F)F)NC(=O)/C=N/OCC#N MS-3662 c1ccc(cc1)CO/N=C/C(=O)Nc2ccc(cc2F)F MS-3663 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(cc(cn2)C(F)(F)F)Cl MS-3664 Cc1cc(ccc1C(C)C)N2CCNC2=O MS-3665 c1ccc2c(c1)c(c3c(n2)CCC3)Cl MS-3666 Cc1ccc(c2c1CC(O2)(C)C)[N+](=O)[O-] MS-3667 CCCc1ccccc1OCC(=O)O MS-3669 CC(CNC1=C(C(=O)c2ccccc2C1=O)Cl)O MS-3671 c1cc(cnc1)CC(C(Cc2ccc(cc2)Br)c3cc(cc(c3)Cl)Cl)O MS-3672 CC1(C(C1(C)C)C(=O)OC(C#N)c2cccc(c2)Oc3ccccc3)C MS-3673 C1CNC(=C[N+](=O)[O-])N1 MS-3675 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C=O MS-3676 c1cc(c(cc1Cl)Cl)OC(CC(=O)O)C(=O)O MS-3679 C1C2C1C(=O)NC2=O MS-3680 c1cc(ccc1NC(=O)CCl)F MS-3681 c1ccc(cc1)COC(=O)N2CCCC2/C=C/CO MS-3682 CC(C(=O)O)Oc1cc(ccc1[N+](=O)[O-])Oc2ccc(cc2Cl)C(F)(F)F MS-3683 CCNC(=O)Cc1cccc2c1cccc2 MS-3685 Cc1cc(c(c(c1)[N+](=O)[O-])Cl)[N+](=O)[O-] MS-3686 COC(c1ccc(c(c1)Cl)Cl)C(=O)O MS-3687 CC(C(c1ccc(cc1)F)C(=O)c2ccccc2)C(=O)O MS-3688 CC(C)Cc1cc(n(n1)C)[N+](=O)[O-] MS-3689 CC(C)Cc1cc(n(n1)C)C(=O)O MS-3690 CC1C2CCN(CC2(CCC1O)C)Cc3ccccc3 MS-3691 c1ccc(c(c1)Nc2ccc(cc2)O)[N+](=O)[O-] MS-3693 CC1=NNC(=O)C1 MS-3694 CSC1=NCCN1.I MS-3695 C1CCC(=C(C#N)C#N)CC1 MS-3697 Cc1cccc(c1NC(=O)N/C(=N/C(=O)Nc2c(cccc2C)C)/NC)C MS-3699 CC(=O)Oc1c(cc(cc1I)C(=O)O)I MS-3701 c1ccn(c1)c2cccc(c2CNC(=O)c3ccc(cc3F)F)Cl MS-3703 c1[nH]nc(n1)Br MS-3704 COc1ccc(cc1)/C=C/C(=O)OC MS-3707 c1cc(cc(c1)OCCO)[N+](=O)[O-] MS-3708 CC1c2c(c3ccccc3[nH]2)CCN1 MS-3709 COC(=O)c1cc(cnc1)Br MS-3710 CCN1CCN(CC1)S(=O)(=O)c2cc(c(nc2)OCC)C(=O)O MS-3711 c1ccc(cc1)C(c2ccccc2)N3CC(C3)C#N MS-3712 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3Cl)Cl)/C(=O)O2 MS-3714 CCC(C(=O)O)Oc1ccc(cc1C)Cl MS-3715 c1cc(c(cc1Cl)OCCN)Cl.Cl MS-3716 Cc1cc(ccc1C(C)C)N.Cl MS-5000 CCOC(=O)C(CCSC)NC(=O)C MS-5001 CCOC(=O)C(C)N(c1ccc(c(c1)Cl)F)C(=O)c2ccccc2 MS-5002 c1ccc(cc1)CN2C(=O)C3CC3C2=O MS-5003 CC1(C(C1(C)C)C(=O)O)C MS-5005 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])CCCC(=O)O MS-5007 CC(C(=O)OCCOC)Oc1cc(ccc1[N+](=O)[O-])Oc2ccc(cc2Cl)C(F)(F)F MS-5008 c1cc(ccc1[N+](=O)[O-])OCCCl MS-5009 Cc1cc(c(c(c1)[N+](=O)[O-])NC(C)C(=O)O)[N+](=O)[O-] MS-5011 Cc1cc(ccc1C(C)(C)C)NC(=O)NC MS-5013 CC(C)Cc1c(c(n(n1)C)C(=O)N)[N+](=O)[O-] MS-5014 CCCc1c[nH]c(c1[N+](=O)[O-])C(=O)O MS-5015 CNC1=C(C(=O)c2ccccc2C1=O)Cl MS-5016 c1ccc(cc1)c2c3c(nn2C(=O)c4cccs4)-c5ccccc5C3=O MS-6000 c1ccc(cc1)C2CC3=C(C(Nc4ccccc4N3)c5cccnc5)C(=O)C2 MS-6001 COc1ccc(cc1OC)CCNC2=C(C(=O)c3c2cccc3)c4ccccc4 MS-6002 CC(=C1C(=O)c2ccccc2C1=O)Nc3nc[nH]n3 MS-6003 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=C3C(=O)c4ccccc4C3=O)C#N MS-6004 c1ccc(cc1)n2c(=O)nc(s2)NC(=O)c3ccc(cc3)Cl MS-6005 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)Nc3ccc(cc3)OC(F)(F)F MS-6006 c1ccc(cc1)COc2ccc(cc2)C(=O)NNC(=O)Nc3cccc(c3)C(F)(F)F MS-6007 COc1ccc(cn1)NC2=C(C(=O)c3c2cccc3)c4ccccc4 MS-6008 Cn1cc(c2c1cccc2)C3CC(=NNC3=O)c4ccc(cc4)Br MS-6009 CC(C)CC1CC(=CC(=O)C1)NCC#C MS-6010 CC(C)CC1CC(=O)C(=CNc2cccc(c2)OC(C(F)F)(F)F)C(=O)C1 MS-6011 COc1ccc(cc1)C(N2CCN(CC2)c3ccccc3)Sc4ccccc4 MS-6012 CC(=O)Nc1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl MS-6013 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3cccc(c3)C(F)(F)F MS-6014 c1ccc2c(c1)C(=O)C(=CNc3cccc4c3nccc4)C2=O MS-6015 CC1(CC2=C(C(=O)C1)C3(C(=C(O2)N)C#N)C(=O)c4ccccc4C3=O)C MS-6016 c1cc(ccc1OC(F)(F)F)S(=O)(=O)C/C(=N\O)/N MS-6017 Cn1cc(c2c1cccc2)C3CC(=NNC3=O)c4ccc(cc4)C5CCCCC5 MS-6018 CC1(Cc2c(sc(n2)NC(=O)c3ccc(cc3)OC)C(=O)C1)C MS-6019 COc1ccc(cc1)Nc2[nH+]c(cs2)c3ccc(cc3)c4ccccc4.[Br-] MS-6020 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccccc2 MS-6021 c1cc2c(cc1F)c3c([nH]2)CCCC3 MS-6022 c1ccc2c(c1)c(c[nH]2)CC(=O)NNC(=S)NC3CCCCC3 MS-6023 CC(C)(C)C(=O)/C(=C/c1cc(ccc1Sc2nc3ccccc3s2)[N+](=O)[O-])/C#N MS-6024 c1cc(ccc1NC2=C(C(=O)CCC2)Cl)[N+](=O)[O-] MS-6025 CC1(CC(=C(C(=O)C1)Cl)N2CCN(CC2)c3ccccc3)C MS-6026 c1ccc2c(c1)c(=O)c(=NNC(=O)COc3ccccc3Cl)c2=O MS-6027 Cc1cc(ccc1OCC(=O)NN=c2c(=O)c3ccccc3c2=O)Cl MS-6028 Cc1c(c(=O)n(n1C)c2ccccc2)NC3=CC(=O)CC(C3)c4ccccc4 MS-6029 CCOC(=O)/C(=C/N1CCN(CC1)c2ccccc2)/C#N MS-6030 Cc1c(c(=O)n(n1C)c2ccccc2)NC3=CC(=O)CC(C3)(C)C MS-6031 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4cc(cc(c4)Cl)Cl MS-6032 c1cc(cnc1)/C=N/C(=C(/C#N)\N)/C#N MS-6033 CSC(=C(C#N)S(=O)(=O)c1ccccc1)SC MS-6034 CC(=C1C(=O)c2ccccc2C1=O)Nc3cc(cc(c3)Cl)Cl MS-6035 CC1(CC(=CC(=O)C1)NCCOC)C MS-6036 CC(C)(C)CC(C)(C)NC=C(C#N)C#N MS-6037 CC(C)(C)C(=O)/C(=C\NCCc1ccc(c(c1)OC)OC)/C#N MS-6038 COc1cc2c(cc1OC)C(=NCC2)COc3ccc(cc3Cl)Cl MS-6039 CC(C)c1ccc(cc1)/C=C/C(=O)NC(Cc2c[nH]c3c2cccc3)C(=O)OC MS-6040 c1ccc(cc1)n2c(nnc2S)CSc3[nH]c4ccccc4n3 MS-6041 c1cc(cnc1)c2c([nH]nn2)C#N MS-6042 c1cc(cc(c1)Cl)/C=N/c2c([nH]c(=O)n(c2=N)c3cccc(c3)C(F)(F)F)C#N MS-6043 COc1ccc(cn1)NC(=C2C(=O)c3ccccc3C2=O)C#N MS-6044 CC1(CC2=C(CC(=NN2)c3ccc(cc3)Br)C(=O)C1)C MS-6045 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)n3cnc(c3Cl)Cl)C MS-6046 COc1ccc(cc1)c2c3c(nn2C(=O)c4ccccc4)-c5ccccc5C3=O MS-6047 c1ccc(cc1)C(=Nc2ccc(cc2)Oc3ccccc3)C4C(=O)c5ccccc5C4=O MS-6048 c1cc(cc(c1)NC=CC=[NH+]c2cccc(c2)C(F)(F)F)C(F)(F)F.[Cl-] MS-6049 c1ccc(cc1)NC(=O)NNC(=O)COc2cccc3c2cccc3 MS-6050 C=CCNC(=S)NN=C1c2cc(ccc2NC1=O)Br MS-6051 COc1cccc2c1oc(=O)c(c2)C(=C(C#N)C#N)N MS-6052 c1c(cc(c(c1O)C=NC(=C(C#N)N)C#N)I)I MS-6053 c1ccc2c(c1)C(=O)C(=CNc3ccc(cn3)Br)C2=O MS-6054 CCN1C(=O)C(=Cc2cccc(c2)Oc3ccccc3)SC1=S MS-6055 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)Nc3ccc(cc3)OC(F)(F)F MS-6056 c1cc(cc(c1)OC(C(F)F)(F)F)NC=C(C#N)c2[nH]nnn2 MS-6057 c1ccc2c(c1)C(=O)NC(N2)c3cc4c(cc3[N+](=O)[O-])OCO4 MS-6058 Cc1cc(c2cc(c(=O)oc2c1)C=C(C#N)C(=O)C(C)(C)C)C MS-6059 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C=Cc3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl MS-6060 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccccc3Cl MS-6061 c1ccc2c(c1)c(c[nH]2)/C=C\3/C(=O)NC(=S)N3 MS-6062 Cn1c(c(c(=O)n1c2ccccc2)Cl)CSC(=[NH2+])N.[Br-] MS-6063 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3)[N+](=O)[O-] MS-6064 CC(=O)Nc1ccc(cc1)OCC(=O)NCCc2c[nH]c3c2cccc3 MS-6065 Cc1cc(c2c(c1)C(=NNC(=S)N)C(=O)N2)C MS-6066 C=CCn1c(nnc1S)CSc2[nH]c3ccccc3n2 MS-6067 CC1(Cc2c(sc(n2)NC(=O)c3cccnc3Oc4ccccc4)C(=O)C1)C MS-6068 c1ccc(cc1)n2c(n[nH]c2=S)Cc3c[nH]c4c3cccc4 MS-6070 Cc1ccc(cc1)S(=O)(=O)CC(=O)NN=C2c3ccccc3NC2=O MS-6071 Cc1cc(ccc1Oc2c(cccn2)C(=O)NCCc3c[nH]c4c3cccc4)Cl MS-6072 CC1CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)C(C)C)C(=O)C1 MS-6073 c1c(cc(cc1C(F)(F)F)NC=CC=[NH+]c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F.[Cl-] MS-6074 Cc1c(c2c(o1)CC(CC2=O)(C)C)C(=O)C MS-6075 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C MS-6076 Cc1cc(nc(n1)NC=C(C#N)C#N)Cl MS-6077 CC1(CC(=C(C(=O)C1)I)Nc2cccc(c2)[N+](=O)[O-])C MS-6078 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCc3ccc(c(c3)OC)OC MS-6079 Cn1c(c(c(=O)n1c2ccccc2)Br)Cn3cnc(c3Cl)Cl MS-6080 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc(cc(c3)Cl)Cl MS-6081 CCCCNC1=CC(=[NH+]CCCC)c2c1cccc2.[Cl-] MS-6082 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-6083 COc1ccc(cc1OC)CCNC(=O)c2cccs2 MS-6084 CCOc1ccc(cc1)N2C(=O)CSC23c4ccccc4NC3=O MS-6085 CC1(CC2=C(C(Nc3cc(ccc3N2)Cl)c4c[nH]c5c4cccc5)C(=O)C1)C MS-6086 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)Nc3cccc(c3)C(F)(F)F MS-6087 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)F MS-6088 CCOP(=O)(Cc1c(c(=O)n(n1C)c2ccccc2)Br)OCC MS-6089 CCN1C(=O)/C(=C/c2c[nH]c3c2cccc3)/SC1=S MS-6090 c1ccc2c(c1)c(c[nH]2)CCNC(=O)COc3ccc(cc3Cl)Cl MS-6091 c1cc(ccc1c2csc(n2)NC(=O)CCl)Br MS-6092 CC(=O)Nc1nc2c(s1)C(=O)CC(C2)(C)C MS-6093 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3cc(ccc3OC)OC MS-6094 Cn1c(c(c(=O)n1c2ccccc2)Br)COCC(F)(F)F MS-6095 c1cc(c(nc1)Cl)C(=O)Nc2ccc(cc2)n3cnc(c3Cl)Cl MS-6096 CC1(Cc2cccc(c2O1)Oc3ccc(cn3)[N+](=O)[O-])C MS-6097 CC(C)(C)C1=NN(C(=O)C1=Cc2cc(cc(c2O)I)I)c3ccc(cc3)[N+](=O)[O-] MS-6099 c1ccc(cc1)Oc2cccc(c2)C=C3C(=O)Nc4ccccc4S3 MS-6100 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4ccc(cc4)C(C)C MS-6101 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)SC)C(=O)C1)C MS-6102 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4ccccn4 MS-6103 Cc1cccc(c1C)OCC(=O)N2CCN(CC2)c3ccccc3F MS-6104 Cc1cc(no1)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C MS-6105 c1cc(ncc1C(F)(F)F)n2cnc(c2Cl)Cl MS-6106 CC1(CC2=C(C(Nc3ccc(cc3N2)Cl)c4ccc(c(c4)[N+](=O)[O-])Cl)C(=O)C1)C MS-6107 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc(ccc3Cl)C(F)(F)F MS-6108 CC(C)C(=O)n1c-2c(c(n1)c3ccc(cc3)OC)C(=O)c4c2cccc4 MS-6109 c1ccc(c(c1)C(=O)O)NC2=C(C(=O)CCC2)I MS-6110 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc(ccc3OC)OC MS-6112 Cc1cc(ccc1OCC(=O)NNC(=S)Nc2ccc(cc2)Cl)Cl MS-6113 CC1CC(=CC(=O)C1)Nc2ccc(cc2)NC(=S)Nc3ccccc3 MS-6114 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)Nc2ccc(cc2)Cl MS-6115 C1CC(=C(C(=O)C1)I)NCCNC2=C(C(=O)CCC2)I MS-6116 CC1(CC(=CC(=O)C1)Nc2cccc3c2nccc3)C MS-6117 CCC1CC(=O)C(=CNc2cccc3c2nccc3)C(=O)C1 MS-6118 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cccc4c3nccc4 MS-6119 Cn1c(c(c(=O)n1c2ccccc2)Br)CSC(=NN=Cc3ccc(cc3)OC)[NH3+].[Br-] MS-6120 CC1(CC(=O)C(=CNc2ccc3c(c2)OCO3)C(=O)C1)C MS-6121 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cccc4c3nccc4 MS-6122 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)Oc4ccc5ccccc5c4 MS-6123 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-6124 CC(C(=O)NCCc1ccc(c(c1)OC)OC)Cl MS-6125 CC1(Cc2c(sc(n2)NC(=O)c3cccnc3)C(=O)C1)C MS-6126 COc1cccc(c1Oc2c(cc(cn2)C(F)(F)F)Cl)C=O MS-6127 c1ccc(c(c1)N2CCN(CC2)C(=O)Nc3cccc(c3)C(F)(F)F)F MS-6128 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)n4cnc(c4Cl)Cl MS-6129 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3cccc4c3nccc4 MS-6130 CC1=NNC2=C(C1)C(=O)CC(C2)(C)C MS-6131 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)N=Cc3ccc(cc3)F MS-6132 Cc1c(sc(n1)Nc2ccc(cc2Cl)Cl)C(=NO)C MS-6133 Cc1ccc(cc1)S(=O)(=O)C(=Cc2cc3c(cc2[N+](=O)[O-])OCO3)C#N MS-6134 Cc1cc(nc(n1)NC=C(C#N)c2[nH]nnn2)C MS-6136 CC(C(=O)NNC(=S)Nc1ccc(cc1)Cl)Oc2ccc(cc2Cl)Cl MS-6137 Cc1cc(no1)NC(=C2C(=O)c3ccccc3C2=O)C MS-6138 CC(C)CC1CC(=CC(=O)C1)Nc2[nH]nnn2 MS-6139 CC(=C1C(=O)c2ccccc2C1=O)NCCc3ccc(c(c3)OC)OC MS-6140 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(nc3)OC MS-6141 c1ccc(cc1)COc2ccc(cc2)c3nnc(n3c4ccccc4)S MS-6142 c1cc(cc(c1)Oc2cccc(c2C#N)F)C(F)(F)F MS-6143 CC(C)C/C=C/C(=O)Nc1ccccc1C(=O)N MS-6144 c1ccc(cc1)Oc2ccc(cc2)N/C=C(\C#N)/c3[nH]nnn3 MS-6145 c1ccc2c(c1)C(=NNC(=O)CS(=O)(=O)c3ccc(cc3)Cl)C(=O)N2 MS-6146 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4cccc(c4)OC(C(F)F)(F)F MS-6147 COc1cc(cc(c1OC)OC)C=Nc2c([nH]c(=O)n(c2=N)c3ccccc3)C#N MS-6148 Cc1cc(no1)NC(=O)C(=O)c2c[nH]c3c2cccc3 MS-6149 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(c(c4)[N+](=O)[O-])Cl)C(=O)C1)C MS-6150 CC1(CC2=C(C(Nc3cc(ccc3N2)Cl)c4ccccc4O)C(=O)C1)C MS-6151 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc5c(c4)OCO5 MS-6152 CCON=C1CC(Cc2c1sc(n2)NC(=O)c3ccc(cc3)Cl)(C)C MS-6153 c1ccc2c(c1)c(c[nH]2)CCNC(=O)Cn3cnc(c3Cl)Cl MS-6154 c1ccc(c(c1)N2CCN(CC2)C3=CC(=O)CCC3)F MS-6155 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3ccc(cc3F)F MS-6156 CC(C)CC1CC2=C(C(Nc3ccccc3N2)c4cccc(c4)Oc5ccccc5)C(=O)C1 MS-6157 CC(C(=O)O)Sc1nc2c(c3ccccc3[nH]2)nn1 MS-6158 Cc1c(c(c(c(c1F)F)NNC(=S)Nc2ccc(cc2)Cl)F)F MS-6159 Cc1cc(ccc1C(C)C)NC(=O)C(=O)c2c[nH]c3c2cccc3 MS-6160 Cc1cc(ccc1C(C)C)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C MS-6161 COc1ccc(cc1)C=CC=C(C#N)C#N MS-6162 CC(C)(C)C(=O)C(=CC=Cc1ccc(cc1)OC)C#N MS-6163 c1cc(ncc1C(F)(F)F)N2CCN(CC2)c3ccc(cn3)C(F)(F)F MS-6164 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-6165 c1ccc(cc1)NC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-6166 CC1(CC(=C(C(=O)C1)I)Nc2cccc(c2)OC(C(F)F)(F)F)C MS-6167 CCC(CC)(C#C)N/C=C(/C#N)\C(=O)OCC MS-6168 c1cc2c(cc1C=Nc3ccc(cc3N)C(=O)O)OCO2 MS-6169 COc1ccc(cc1OC)CCNC(=O)c2ccccc2[N+](=O)[O-] MS-6170 CC(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl MS-6171 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC(=O)O MS-6172 c1ccc(c(c1)C(=O)Nc2[nH]nnn2)[N+](=O)[O-] MS-6173 c1cc(ccc1NC2=CC(=[NH+]c3ccc(cc3)Cl)CCC2)Cl.[Cl-] MS-6174 CC1=CC(=NS(=O)(=O)N1)C(F)(F)F MS-6175 Cc1ccc(cc1)S(=O)(=O)NNC2=CC(=O)CCC2 MS-6176 CC(C)(C)c1c2c(nn1C)-c3ccccc3C2=O MS-6177 CC1(CC(=C(C(=O)C1)C(=O)Nc2ccccc2)NCc3ccccc3)C MS-6178 CC(C)(C)c1c2c(nn1c3ccccc3)-c4ccccc4C2=O MS-6179 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccc(cc3)F MS-6180 Cc1ccc2cccc(c2n1)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F MS-6181 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C(F)(F)F MS-6182 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)N3CCN(CC3)c4ccccc4F MS-6183 c1ccc(cc1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-6184 c1cc(ccc1NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl MS-6185 COc1ccc(cc1)C=CC=NNC(=S)N MS-6186 CCOC(=O)C(CC(=O)c1ccc(cc1)Br)C(=O)c2ccccc2 MS-6187 Cc1cc(nc(n1)NC=C2C(=O)CC(CC2=O)c3ccccc3)Cl MS-6188 CCOc1ccc(cc1)C(=O)CC(C2C(=NN(C2=O)c3ccccc3)C)C(=O)O MS-6189 CC1=NN(C(=O)C1C(CC(=O)c2ccc(cc2)Br)C(=O)O)c3ccccc3 MS-6190 CC(C)c1ccc(cc1)C=C2C(=O)c3ccccc3C2=O MS-6191 CC(C)(C)C1=NN(C(=O)C1C(CC(=O)c2ccc(cc2)Br)C(=O)O)c3ccccc3 MS-6192 CC1CC(=O)C(=CNc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)C(=O)C1 MS-6193 CC1(OC(=O)C(=CNc2cc(ccc2OC)OC)C(=O)O1)C MS-6194 c1cc(ccc1NC=C2C(=O)CCCC2=O)Oc3c(cc(cn3)C(F)(F)F)Cl MS-6195 CC1(OC(=O)C(=CNC2CCCCC2)C(=O)O1)C MS-6196 CC1(CC2=C(C(Nc3cc(ccc3N2)Cl)c4ccc(cc4)N(C)C)C(=O)C1)C MS-6197 c1cc(ccc1N2C(=O)CSC23c4cc(ccc4NC3=O)Br)Cl MS-6198 Cc1cc(ccc1OC/C(=N\O)/N)Cl MS-6199 c1ccc(cc1)COc2ccc(cc2)C(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F MS-6200 CCOC(=O)C(=C(Nc1ccccc1)SC)C#N MS-6201 COc1ccc(cc1OC)CCNC(=O)CC#N MS-6202 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CCCCl MS-6203 CC1Cc2c(c(nn2C)c3ccc(cc3)OC)C(=O)C1 MS-6204 CC(C)(C)c1ccc(cc1)C2=NNC(=O)C(C2)c3c[nH]c4c3cccc4 MS-6205 CC(C)c1ccc(cc1)C(=O)CC(c2c[nH]c3c2cccc3)C(=O)O MS-6206 CC1(Cc2c(sc(n2)N)C(=O)C1)C MS-6207 c1ccc2c(c1)[nH]c(n2)SCC(=O)NNC(=S)NC3CCCCC3 MS-6208 CC1(OC(=O)C(=CNc2ccc(cc2[N+](=O)[O-])OC)C(=O)O1)C MS-6209 COc1ccc(cc1)C=CC=C2C(=O)NC(=S)N2 MS-6210 CC1(CC2=C(C(Nc3ccccc3N2)c4ccccn4)C(=O)C1)C MS-6211 c1ccc(cc1)C(=O)CC(c2c[nH]c3c2cccc3)C(=O)O MS-6212 Cc1ccc(cc1)S(=O)(=O)NNC2=CC(=O)CC(C2)(C)C MS-6213 Cc1cc(ccc1OCC(=O)NN=C2c3ccccc3N(C2=O)CN4CCOCC4)Cl MS-6214 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)NC=C3C(=O)c4ccccc4C3=O MS-6215 c1ccnc(c1)Sc2ccc(cc2)[N+](=O)[O-] MS-6217 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)NC=C3C(=O)CC(CC3=O)c4ccccc4 MS-6218 c1ccc2c(c1)c(ccc2Br)NC(=O)C(=O)c3c[nH]c4c3cccc4 MS-6219 CC(C)C1C2=C(CC(CC2=O)(C)C)Nc3ccccc3N1 MS-6220 CCC1C2=C(CC(CC2=O)(C)C)Nc3ccccc3N1 MS-6221 CC1(CC2=C(C(Nc3ccccc3N2)c4ccccc4[N+](=O)[O-])C(=O)C1)C MS-6222 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3)F MS-6223 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=S)NC2CCCCC2 MS-6224 CC1C2=C(CC(CC2=O)(C)C)Nc3ccc(cc3N1)Cl MS-6225 COc1ccc(cc1)NC2=C(C(=O)CCC2)Cl MS-6226 CC1(OC(=O)C(=CNc2ccc(cc2)Oc3ccccc3)C(=O)O1)C MS-6227 CCOc1ccc(cc1)NC2=C(C(=O)CC(C2)C)Cl MS-6228 c1ccc(cc1)NC(=S)N2CCN(CC2)C(=S)Nc3ccccc3 MS-6229 CC(C)(C)C1=NN(C2(C1C(=O)c3c2cccc3)O)C(=O)N MS-6230 CCOc1ccc(cc1)N2C(=O)CSC23c4cc(ccc4NC3=O)Br MS-6231 c1cc(ccc1S(=O)(=O)C(=Cc2cc3c(cc2[N+](=O)[O-])OCO3)C#N)Cl MS-6232 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccccc3[N+](=O)[O-] MS-6233 CC(=C1C(=O)c2ccccc2C1=O)N3CCN(CC3)c4ccccc4 MS-6234 c1cc(ccc1c2csc(n2)N)[N+](=O)[O-] MS-6235 Cc1ccc(c(c1)C)c2csc(n2)N MS-6236 CC(=C1C(=O)c2ccccc2C1=O)NCCCNC(=C3C(=O)c4ccccc4C3=O)C MS-6237 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc5ccccc5c4)C(=O)C1)C MS-6238 Cc1cccc(c1)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F MS-6239 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C=O MS-6240 COc1ccc(cc1OC)CNC(=O)c2ccccc2[N+](=O)[O-] MS-6241 CC1(OC(=O)C(=CNc2nc(cs2)c3ccccc3)C(=O)O1)C MS-6242 c1cc(cc(c1)Br)c2csc(n2)N MS-6243 CC(C)(C)C(=O)C(=CNc1nc(cs1)c2ccccc2)C#N MS-6244 CC1(CC(=CC(=O)C1)Nc2cccnc2N)C MS-6245 CC1(OC(=O)C(=CNc2nc(cs2)c3cccc(c3)Br)C(=O)O1)C MS-6246 CC(C)(C)c1c2c(n[nH]1)-c3ccc(cc3C2=O)[N+](=O)[O-] MS-6247 CC1CC(=CC(=O)C1)N2CCN(CC2)c3ccccc3 MS-6248 Cc1ccc(cc1)S(=O)(=O)C(=CC=Cc2ccccc2)C#N MS-6249 c1ccc(cc1)S(=O)(=O)C(=Cc2c[nH]c3c2cccc3)C#N MS-6250 Cc1cc(no1)NC=C2C(=O)c3ccccc3C2=O MS-6251 Cc1cc(ccc1OCC(=O)NNC(=S)Nc2ccccc2)Cl MS-6252 CC1(CC(=CC(=O)C1)Nc2nc[nH]n2)C MS-6253 CC(C)(C)C(=NO)Cn1cnc(c1Cl)Cl MS-6254 CC1(CC2=C(C(Nc3ccc(cc3N2)C(=O)O)c4c(cccc4Cl)F)C(=O)C1)C MS-6255 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC(=O)Nc4ccc(cc4F)F MS-6256 CCCC1C2=C(CC(CC2=O)(C)C)Nc3ccccc3N1 MS-6257 Cc1ccc(cc1)c2csc(n2)NC=C3C(=O)OC(OC3=O)(C)C MS-6258 Cc1cc(ccc1F)c2csc(n2)NC(=O)c3cccnc3 MS-6259 c1cc(cnc1)C(=O)Nc2nc(cs2)c3ccc(c(c3)Cl)Cl MS-6260 Cc1ccc(cc1)c2csc(n2)N MS-6261 Cc1ccc(cc1)c2csc(n2)NC(=O)c3cccnc3 MS-6262 Cc1ccc(cc1)c2csc(n2)NC(=O)c3ccc(cc3)C MS-6263 Cc1cc(ccc1F)c2csc(n2)NC=C3C(=O)OC(OC3=O)(C)C MS-6264 Cc1c(nc(s1)N)c2ccc(cc2)Br MS-6265 c1c(cnc(c1Cl)SC(=S)N2CCCC2)C(F)(F)F MS-6266 Cc1cc(ccc1C(C)C)NC(=S)N(C)N MS-6267 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccccc3C(=O)O MS-6268 CC1(CC(=CC(=O)C1)Nc2ccccc2C(=O)O)C MS-6269 CN(C)c1ccc(cc1)NC=C(C#N)c2[nH]nnn2 MS-6270 CC1(CC(=CC(=O)C1)NC2CCCCC2)C MS-6271 CC(C)(C)C(=O)CS(=O)(=O)c1ccc(cc1)Cl MS-6272 c1cc(ccc1COc2ccc(cc2)C=C(C#N)C#N)[N+](=O)[O-] MS-6273 COc1ccc(cc1)/C=C/2\C(=O)Nc3ccccc3S2 MS-6274 CCOc1ccc(cc1)C2=NNC(=O)C(C2)c3cn(c4c3cccc4)C MS-6275 COc1ccc(cc1OC)CCNC(=O)COc2ccc(cc2Cl)Cl MS-6276 CCOc1ccc(cc1)C2=NNC(=O)C(C2)c3c[nH]c4c3cccc4 MS-6278 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)OC(F)(F)F)C2=O MS-6279 C#CCSC(=NN=Cc1ccc(cc1)F)[NH3+].[Cl-] MS-6280 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)NC3=CC(=O)CC(C3)(C)C)C MS-6281 C=CCNC(=S)NNC(=O)CSc1[nH]c2ccccc2n1 MS-6282 CC(C)(C)c1c2c(no1)-c3ccccc3C2=O MS-6283 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)Cl MS-6284 CSc1ccc(cc1)C2C3=C(CC(CC3=O)c4ccccc4)Nc5ccccc5N2 MS-6285 CC(C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Cl MS-6286 c1ccc2c(c1)c(c[nH]2)CCNC(=S)Nc3ccc(cc3)OC(F)(F)F MS-6287 CC(=NO)c1ccc(cc1)NC=C2C(=O)c3ccccc3C2=O MS-6288 CC(C)c1ccc(cc1)S(=O)(=O)C/C(=N/O)/N MS-6289 c1ccc2c(c1)-c3c(c([nH]n3)C4CCCCC4)C2=NN MS-6290 c1ccc(cc1)S(=O)(=O)C2(CC2)C#N MS-6291 COc1ccc(cc1)C=C2Cc3ccccc3C2=O MS-6292 c1ccc(cc1)C2CC(=C(C(=O)C2)Br)Nc3ccccc3C(=O)O MS-6293 CC1(CC(=CC(=O)C1)NCc2ccccc2)C MS-6294 CC1(CC(=C(C(=O)C1)I)Nc2ccccc2C(=O)O)C MS-6295 c1cc(ccc1NC2=CC(=O)CCC2)OC(F)(F)F MS-6296 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3ccc(cc3)OC(F)(F)F MS-6297 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(nc3)OC MS-6298 CC1(CC2=C(C(Nc3ccccc3N2)c4c[nH]c5c4cccc5)C(=O)C1)C MS-6299 COc1ccc(cc1)C=C2Cc3cc(c(cc3C2=O)OC)OC MS-6300 CC1(CC(=CC(=O)C1)Nc2ccccc2)C MS-6301 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)[N+](=O)[O-])C2=O MS-6302 CC(C)(C)C(=O)C(=Cc1ccc(cc1)OC)C#N MS-6303 Cc1c(sc(n1)Nc2ccccc2Cl)C(=NO)C MS-6304 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(c(c2)C)Cl MS-6305 CC1(CC(=CC(=O)C1)Nc2cccc(c2)[N+](=O)[O-])C MS-6306 c1ccc(cc1)Oc2cccc(c2)COC(=O)CC#N MS-6307 COc1ccc(cc1)N2C(C(C2=O)Oc3ccc(cc3Cl)Cl)c4ccc5c(c4)OCO5 MS-6308 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C=Cc3cc(ccc3Cl)[N+](=O)[O-] MS-6309 CC(=NO)c1ccc(cc1)NC=C2C(=O)OC(OC2=O)(C)C MS-6310 c1cc2cccnc2c(c1)NC=C(C#N)C#N MS-6311 CC(C)/C=C/c1nc2c(cc(cc2Cl)Cl)c(=O)o1 MS-6312 c1ccc2c(c1)C(=O)NC(N2)c3cccs3 MS-6313 c1ccc2c(c1)C(=O)NC(N2)c3ccc(cc3)OCc4ccc(cc4)[N+](=O)[O-] MS-6314 Cc1cccc(c1NC=C(C#N)c2[nH]nnn2)Cl MS-6315 c1ccc2c(c1)C(=O)NC(N2)c3cccnc3 MS-6317 c1ccc2c(c1)C(=O)C(=Cc3cc(ccc3Cl)[N+](=O)[O-])C2=O MS-6318 CC(C)(C)C1=NN(C(=O)C1=CC=Cc2ccc(cc2)[N+](=O)[O-])c3ccccc3 MS-6319 c1ccc(c(c1)C(=O)n2cnc(n2)N)[N+](=O)[O-] MS-6320 CC1Cc2c(sc(n2)NC(=O)C)C(=O)C1 MS-6321 CC1Cc2c(sc(n2)N)C(=O)C1 MS-6322 CC(C)(C)C(=O)C(=Cc1cc(c(cc1[N+](=O)[O-])OC)OC)C#N MS-6323 Cn1c(c(c(=O)n1c2ccccc2)Cl)COc3cccc(c3)C(F)(F)F MS-6324 CC(C)(C)C(=O)NCCc1ccccc1 MS-6325 CC(C)(C)C(=O)C(=Cc1ccccc1[N+](=O)[O-])C#N MS-6326 c1ccc(cc1)NC(=O)NNC(=O)CSc2[nH]c3ccccc3n2 MS-6327 c1ccc2cc(ccc2c1)Oc3ccc(cc3)NC=C(C#N)C#N MS-6328 CC(C)(C)c1c2c(n(n1)c3ccc(cc3)[N+](=O)[O-])-c4ccccc4C2=O MS-6329 c1ccc2c(c1)C(=O)C(=CNc3ccc4c(c3)OCO4)C2=O MS-6330 c1cc2cccnc2c(c1)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F MS-6331 c1ccc(c(c1)C=C2C(=O)c3ccccc3C2=O)[N+](=O)[O-] MS-6332 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)Nc3ccc(cc3)Cl MS-6333 c1ccc(cc1)C2CC(=O)C(C(=O)C2)C(=O)Nc3cccc(c3)C(F)(F)F MS-6334 c1c(cnc(c1Cl)N2CCN(CC2)C(=S)NC3CCCCC3)C(F)(F)F MS-6335 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4cccc(c4)C(=O)O MS-6336 c1cnccc1C(=O)NNC(=S)NC2CCCCC2 MS-6337 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCN(C)C MS-6338 CC1(CC2=C(C(Nc3ccccc3N2)c4cc(c(c(c4)OC)O)OC)C(=O)C1)C MS-6339 COc1ccc(cc1OC)Cc2n[nH]c(=S)n2c3ccccc3 MS-6340 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)I)C2=O MS-6341 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)F)C2=O MS-6342 COc1ccc(cc1)C(=O)C2C(=O)c3ccccc3C2=O MS-6343 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)CC#N)C2=O MS-6344 c1ccc2c(c1)C(=O)C(=CNc3cc(ccc3F)C(F)(F)F)C2=O MS-6345 CC(C)C=CC(=O)NCCc1c[nH]c2c1cccc2 MS-6346 CCC(CC)(C#C)NC=C(C#N)C#N MS-6347 CC(C)(C)C(=O)/C(=C/C=C/c1ccccc1)/C#N MS-6348 CC1CC(=CC(=O)C1)Nc2ccccc2C(F)(F)F MS-6349 CC(C)(C)C(=O)C(=C1C(=O)c2ccccc2C1=O)C#N MS-6350 c1c(c(cc2c1OCO2)[N+](=O)[O-])C=NC(=C(C#N)N)C#N MS-6351 CCOC(=O)c1c(nc(s1)NC(=O)C(F)(F)F)C MS-6352 c1cc2cccnc2c(c1)NS(=O)(=O)c3ccc(cc3)Cl MS-6353 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CCSc3ccc(cc3)Cl MS-6354 c1ccc(cc1)S(=O)(=O)C(=Cc2cccnc2)C#N MS-6355 CCOC(=O)C(=CNc1ccc(cc1)C(=O)C)C#N MS-6356 CC1(Cc2c(sc(n2)NC(=O)COc3ccc(cc3Cl)Cl)C(=O)C1)C MS-6357 CC(C)(C(=O)c1ccccc1)n2cncn2 MS-6358 COc1ccc(cc1)n2cc(nc2S)c3ccc(cc3)[N+](=O)[O-] MS-6359 CC(=C1C(=O)c2ccccc2C1=O)NNC(=O)c3ccccc3 MS-6360 CC(=C1C(=O)c2ccccc2C1=O)NNC(=O)Cc3ccc(c(c3)OC)OC MS-6361 CC(C)(C)C1=NN(C(=O)C1=Cc2cccs2)c3ccccc3 MS-6362 CC1(Cc2c(cc(nn2)c3ccc(cc3)Br)C(=NO)C1)C MS-6363 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)N=Cc3ccc(cc3Cl)Cl MS-6364 c1ccc(c(c1)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccc(cc4)Cl)[N+](=O)[O-] MS-6365 Cc1cc(c2ccccc2n1)NC(=C3C(=O)c4ccccc4C3=O)C MS-6366 C#CCn1cnc(c1Cl)Cl MS-6367 CC(C)c1c2c([nH]n1)-c3ccccc3C2=O MS-6368 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)Cl MS-6369 CC1(Cc2cccc(c2O1)Oc3c(cc(cn3)C(F)(F)F)Cl)C MS-6370 CC1(Cc2c(c(nn2C)c3ccc(c(c3)OC)OC)C(=O)C1)C MS-6371 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)OC(F)(F)F MS-6372 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCc3c[nH]c4c3cccc4 MS-6373 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)n4cncn4 MS-6374 Cc1ccc(cc1)c2csc(n2)NC(=O)c3c(onc3c4ccccc4Cl)C MS-6375 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4cc(c(c(c4)OC)O)OC MS-6376 c1cc(ccc1NC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl MS-6377 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3c(onc3c4ccccc4Cl)C MS-6378 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-6379 CC1(CC(=C(C(=O)C1)I)Nc2ccc(cc2)OC(F)(F)F)C MS-6380 c1ccc2c(c1)C(=O)C(=Cc3cc4c(cc3[N+](=O)[O-])OCO4)C2=O MS-6381 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccccc3Br MS-6382 Cc1c(c(no1)c2ccccc2)C(=O)NCCc3c[nH]c4c3cccc4 MS-6383 CC(C)(C)C(=O)C(=Cc1ccc(cc1)F)C#N MS-6384 c1ccc(cc1)NC(=S)Nc2ccc(cc2)NC3=CC(=O)CCC3 MS-6385 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)N(C)C)/C#N MS-6387 c1cc(ccc1NC=C(C#N)C#N)F MS-6388 c1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccc3 MS-6389 c1ccc(cc1)Oc2ccc(cc2)N=C3c4ccccc4NC3=O MS-6390 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3cccc(c3)C(F)(F)F MS-6391 c1ccc2c(c1)C(=NNC(=O)COc3ccc(cc3)F)C(=O)N2 MS-6393 CC1(CC(=CC(=O)C1)N2CCN(CC2)CCO)C MS-6394 c1ccc2c(c1)C(=O)C(=CNc3ncccn3)C2=O MS-6395 CC1(CC(=CC(=O)C1)Nc2cc(cc(c2)Cl)NC(=O)Nc3cccc(c3)C(F)(F)F)C MS-6396 COc1cc(ccc1O)C=C(C#N)C#N MS-6397 Cn1c(c(c(=O)n1c2ccccc2)Br)CBr MS-6398 c1cc(ccc1C=C(C#N)C#N)N2CCCCC2 MS-6399 c1ccc(c(c1)C(=O)N)NC=C(C#N)C#N MS-6400 CC(=Nc1cccc(c1)OC(C(F)F)(F)F)C2C(=O)c3ccccc3C2=O MS-6401 CC1(CC(=NO)C(=NO)C(=O)C1)C MS-6402 CC(C)(C)C(=O)C(=C(Nc1ccccc1)S)C#N MS-6403 CC(C)(C)C(=O)C(=C(Nc1ccccc1)O)C#N MS-6404 c1ccc(cc1)NC(=S)NNC(=O)COc2cccc(c2Cl)Cl MS-6405 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])n2cnc(c2Cl)Cl MS-6406 CCN1C(=O)C(=Cc2cc(ccc2Cl)[N+](=O)[O-])SC1=S MS-6407 c1ccc(cc1)C=CC(=O)NCCc2c[nH]c3c2cccc3 MS-6408 Cc1cc(ccc1OCc2c(c(=O)n(n2C)c3ccccc3)Br)Cl MS-6409 c1ccc(c(c1)C(=O)O)NC=C(C#N)C#N MS-6410 CC(C)(C)c1ccc(cc1)C(=O)CC(c2c[nH]c3c2cccc3)C(=O)O MS-6411 CC1(CC(=O)C(=CNc2ccc(cn2)Br)C(=O)C1)C MS-6412 c1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccc3F MS-6413 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4ccccc4F MS-6414 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4cccc(c4)OC(F)(F)F MS-6415 c1ccc(cc1)CSc2[nH]c(=O)c3ccccc3n2 MS-6416 CCCC1CC(=O)CC(=O)C1 MS-6417 CC1(CC(=O)C(=CNc2ccsc2C(=O)OC)C(=O)C1)C MS-6418 COc1ccc(cn1)NC(=O)c2ccccc2CC(=O)O MS-6419 c1ccc2c(c1)nc(s2)SCC(=O)NNC(=O)Nc3ccc(cc3)Cl MS-6420 CC(C)(C)C(=O)C(=Cc1ccc(c(c1)[N+](=O)[O-])Cl)C#N MS-6421 c1ccc2c(c1)nc(s2)SCC(=O)NN MS-6422 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccccc2C#N MS-6423 CC(=O)c1ccc(cc1)NC=C2C(=O)OC(OC2=O)(C)C MS-6424 CC(C)(C)C(=O)C(=Cc1ccc2c(c1)OCO2)C#N MS-6425 CCOC(=O)C(=CNc1cccc(c1)C(F)(F)F)C#N MS-6426 c1cc(ccc1NC2=CC(=O)CCC2)F MS-6427 c1cc(ccc1NC2=CC(=O)CCC2)[N+](=O)[O-] MS-6428 CC1CC(=CC(=O)C1)Nc2ccc(cc2)C(=O)C MS-6429 CC1(CC(=CC(=O)C1)Nc2ccccc2O)C MS-6430 c1cc(cc(c1)NC=C(C#N)C#N)C(F)(F)F MS-6431 CC(=O)c1ccc(cc1)NC2=CC(=O)CC(C2)c3ccccc3 MS-6432 Cc1cc(=O)n([nH]1)C(=S)N MS-6433 c1ccc(cc1)N2CCN(CC2)C=C(C#N)C#N MS-6434 c1cc(oc1)C=NC(=C(C#N)N)C#N MS-6435 Cc1cc(ccc1OCC(=O)NNC(=S)NC2CCCCC2)Cl MS-6436 Cc1c(c(no1)c2ccccc2)C(=O)Nc3[nH]cnn3 MS-6437 c1cc(ccc1C=NC(=C(C#N)N)C#N)OCC(=O)O MS-6438 c1ccc(c(c1)C=NC(=C(C#N)N)C#N)[N+](=O)[O-] MS-6439 Cc1cc(ccc1Oc2cccc(c2C#N)F)Cl MS-6440 c1ccc2c(c1)C(=NNC(=O)c3ccccc3Cl)C(=O)N2 MS-6441 COc1cccc(c1O)C=NC(=C(C#N)N)C#N MS-6442 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)N=Cc3cccs3 MS-6443 c1cc(cc(c1)Cl)C=NC(=C(C#N)N)C#N MS-6444 c1cc(ccc1n2c(=N)c3c(c(=O)[nH]c(n3)c4cc5c(cc4[N+](=O)[O-])OCO5)[nH]c2=O)Cl MS-6445 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccccn3 MS-6446 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccco3 MS-6447 CC(C)(C)C(=O)Cn1cnc(c1Cl)Cl MS-6448 c1ccc(c(c1)OCC(=O)NN=C2c3cc(ccc3NC2=O)Br)Cl MS-6449 c1cc(cc(c1)NC(=O)NNC(=O)COc2ccc(cc2)[N+](=O)[O-])C(F)(F)F MS-6450 c1cc(ccc1OCC(=O)NNC(=S)NC2CCCCC2)F MS-6451 Cc1c(c(=O)n(n1C)c2ccccc2)NC=C(C#N)C(=O)C(C)(C)C MS-6452 c1ccc2c(c1)cc(c(=O)o2)C(=C(C#N)C#N)N MS-6453 COc1ccc(cc1OC)c2c3c([nH]n2)-c4ccccc4C3=O MS-6454 c1ccc(cc1)NC(=S)NNC(=O)COc2cccc3c2cccc3 MS-6455 c1ccc(cc1)NC(=S)NNC(=O)Cc2c[nH]c3c2cccc3 MS-6456 c1cc(ccc1N=C2c3cc(ccc3NC2=O)Br)OC(F)(F)F MS-6457 CC(C)(C)c1c2c([nH]n1)-c3ccccc3C2=NOC MS-6458 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)C(=O)O MS-6459 COc1cc(c(cc1OC)[N+](=O)[O-])C=NNC(=S)N MS-6460 CCOC(=O)C1=C(OCC1=O)Nc2ccc(c(c2)Cl)Cl MS-6461 CC1(CC(=CC(=O)C1)Nc2ccccc2C#N)C MS-6462 CC1(OC(=O)C(=CNc2ccsc2C(=O)OC)C(=O)O1)C MS-6463 CC1(OC(=O)C(=CNc2ccccc2C#N)C(=O)O1)C MS-6464 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccccc3C#N MS-6465 CCCCCC(=O)Nc1nc(cs1)c2ccc(cc2)Br MS-6466 CCCCCC(=O)Nc1nc(cs1)c2ccccc2 MS-6467 CC1(CC(=C(C(=O)C1)Br)Nc2ccc(cc2)OC(F)(F)F)C MS-6468 CN(C)c1ccc(cc1)/C=C\2/C(=O)NC(=S)S2 MS-6469 c1ccc(cc1)C2CC(=O)C(=CNc3ccccc3)C(=O)C2 MS-6470 COc1ccc(cc1)/N=C\2/c3ccccc3NC2=O MS-6471 CC1(OC(=O)C(=CNCCc2ccc(c(c2)OC)OC)C(=O)O1)C MS-6472 CCOC(=O)C(=Cc1ccco1)C#N MS-6473 COc1ccc(cc1)NC2=CC(=O)CCC2 MS-6474 c1ccc(c(c1)NC2=CC(=O)CCC2)F MS-6475 CC1CC(=CC(=O)C1)Nc2ccc(cc2)N MS-6476 Cc1c(sc(n1)Nc2ccccc2Cl)C(=O)C MS-6477 CN1CCN(CC1)C(=S)Nc2ccccc2 MS-6478 Cc1cc(ccc1OCC(=O)NN=C2c3cc(ccc3NC2=O)Br)Cl MS-6479 CC1CC(=CC(=O)C1)Nc2ccccc2NC(=O)C(C)C MS-6480 c1cc(ccc1[N+](=O)[O-])OCC(=O)NN=C2c3cc(ccc3NC2=O)Br MS-6481 c1ccc(cc1)C=CC=C(C#N)S(=O)(=O)c2ccccc2 MS-6482 c1ccc2c(c1)C(=C(C2=O)c3[nH]c4cc(ccc4n3)Cl)O MS-6483 CCOC(=O)C(C#N)C1(C(=O)c2ccccc2C1=O)O MS-6484 Cc1ccc2cccc(c2n1)Oc3ccc(cc3)[N+](=O)[O-] MS-6485 CN1c2ccccc2/C(=N/NC(=S)N)/C1=O MS-6486 Cn1c2ccccc2c3c1nc(nn3)S MS-6487 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)N MS-6488 c1cc(c(cc1Cl)Cl)OCC(=O)Nc2nc[nH]n2 MS-6489 c1cc(ccc1c2c([nH]nn2)C#N)OC(F)(F)F MS-6490 c1ccc(cc1)C2=C(c3ccccc3C2=O)N MS-6491 c1ccc(cc1)Oc2cccc(c2)c3c([nH]nn3)C#N MS-6492 COc1cccc(c1OC)C=NN=C([NH3+])SCC=C.[Br-] MS-6493 CC(=O)c1cc(ccc1OC)NC(=O)C MS-6494 c1ccc(cc1)C=CC=NNC(=S)N MS-6495 CC(C)(C)C1=NN(C(=O)C1=Cc2cccc(c2O)OC)c3ccccc3 MS-6496 CCN1C(=O)C(=Cc2cccc(c2O)OC)SC1=S MS-6497 c1cc(oc1)C2NC(CS2)C(=O)O MS-6498 COc1ccc(c(c1)NC=C2C(=O)c3ccccc3C2=O)OC MS-6499 COc1ccc(cc1OC)CCNC2=CC(=O)CC(C2)c3ccccc3 MS-6500 CC(=C1C(=O)c2ccccc2C1=O)NNC(=O)Cc3ccccc3 MS-6501 CC(=C1C(=O)c2ccccc2C1=O)NNC(=O)c3ccncc3 MS-6502 Cc1cc(ccc1C(C)C)NC(=C2C(=O)c3ccccc3C2=O)C MS-6503 c1cc(ccc1NC(=S)N2CCN(CC2)C(=S)Nc3ccc(cc3)OC(F)(F)F)OC(F)(F)F MS-6504 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CCCl MS-6505 CC(=C1C(=O)c2ccccc2C1=O)NNC(=O)c3cc(c(c(c3)OC)OC)OC MS-6506 COc1ccc(cc1OC)C(=O)C=Cc2cccs2 MS-6507 CC(C(=O)O)Sc1ccc(cc1)Cl MS-6508 c1ccc(cc1)Oc2ccc(cc2)C(=O)C=Cc3cccs3 MS-6509 COc1ccc(cc1OC)C(=O)C=Cc2ccc(cc2)Cl MS-6510 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(cc3)CBr MS-6511 CCOc1ccc(cc1)Nc2nc(cs2)c3ccc(c(c3)C)F MS-6512 c1ccc(cc1)NC2=C(C(=O)CCC2)Br MS-6513 Cc1c(sc(n1)N)C(=O)C MS-6514 C1CC(=CC(=O)C1)NCCNC2=CC(=O)CCC2 MS-6515 c1ccc2c(c1)C(=O)C(C2=O)C=Nc3cccc(c3)C(F)(F)F MS-6516 CC1(CC(=O)C(=CNc2cccc(c2)[N+](=O)[O-])C(=O)C1)C MS-6517 CC1(CC(=C(C(=O)C1)Br)Nc2ccc(cc2)Cl)C MS-6519 c1ccc(cc1)C(=C2C(=O)c3ccccc3C2=O)NNc4ccccc4 MS-6520 c1ccc(cc1)CNC2=CC(=O)CCC2 MS-6521 CCOC(=O)C(=CNc1cccc(c1)OCc2ccccc2)C#N MS-6522 CC(=C1C(=O)c2ccccc2C1=O)Nc3cc(ccc3Cl)C(F)(F)F MS-6523 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4cccc(c4)Cl MS-6524 Cc1c(sc(n1)Nc2ccccc2)C(=O)C MS-6525 c1ccc(cc1)Nc2nc(cs2)c3ccc(cc3)Br MS-6526 c1ccc(cc1)c2c3c(n[nH]2)-c4ccccc4C3=O MS-6527 c1ccc2c(c1)/C(=N/c3ccc(cc3)Cl)/C(=O)N2 MS-6528 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)Br MS-6530 c1ccc2c(c1)/C(=N/c3cccc(c3)Cl)/C(=O)N2 MS-6531 c1cc(cc(c1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3ccc(cc3)F)C(F)(F)F MS-6532 c1ccc2c(c1)NC(=O)/C(=C\c3ccc(cc3)OC(F)(F)F)/S2 MS-6533 Cn1c(c(c(=O)n1c2ccccc2)Br)CO MS-6534 c1cc(ccc1OC(F)(F)F)S(=O)(=O)Cc2nc(on2)C(F)(F)F MS-6535 CCOc1ccc(cc1)C(=O)CC(c2cn(c3c2cccc3)C)C(=O)O MS-6536 Cn1c(c(c(=O)n1c2ccccc2)Br)CSC(=S)N3CCCC3 MS-6537 c1ccc(cc1)C(=C2C(=O)c3ccccc3C2=O)Nc4ccc(cc4)OC(F)(F)F MS-6538 CCOP(=O)(Cc1c(c(=O)n(n1C)c2ccccc2)Cl)OCC MS-6539 c1ccc2c(c1)c(c[nH]2)CCNC(=O)COc3ccc(cc3)Br MS-6540 CCN(CC)C(=S)SCc1c(c(=O)n(n1C)c2ccccc2)Br MS-6541 CCOC(=O)c1cccc(c1)OCc2c(c(=O)n(n2C)c3ccccc3)Br MS-6542 Cc1cc(c2cc(c(=O)oc2c1)C=C3C(=O)c4ccccc4C3=O)C MS-6543 Cc1ccc(cc1)C(=O)NCCc2c[nH]c3c2cccc3 MS-6544 c1cc(cc(c1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3ccco3)C(F)(F)F MS-6545 CC(C)(C(=O)c1ccc(cc1)Br)n2cncn2 MS-6546 COc1cc(cc(c1OC)OC)C2NC(CS2)C(=O)O MS-6547 COc1cccc(c1O)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccc(cc4)Cl MS-6548 CC(C)c1ccc(cc1)C(=O)C(C)(C)n2cncn2 MS-6550 CC(C)(C)c1ccc(cc1)c2csc(n2)Nc3ccccc3 MS-6551 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)n4cnc(c4Cl)Cl MS-6552 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCc3c[nH]c4c3cccc4 MS-6553 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)Sc4ccccn4 MS-6554 CC1(CC2=C(C(Nc3cc(ccc3N2)Cl)c4ccco4)C(=O)C1)C MS-6555 CC1(CC2=C(C(Nc3cc(ccc3N2)Cl)c4ccccc4F)C(=O)C1)C MS-6556 Cc1ccc(cc1)c2c3c(n(n2)c4ccccc4)-c5ccccc5C3=O MS-6557 c1ccc(cc1)S(=O)(=O)C/C(=N/O)/N MS-6558 Cc1ccc(cc1)S(=O)(=O)C/C(=N/OC(=O)c2cccs2)/N MS-6560 COc1ccc(cc1)/C(=N\N)/C2C(=O)c3ccccc3C2=O MS-6561 Cc1ccc(cc1)C(=O)Nc2nc3c(s2)C(=O)CC(C3)C MS-6563 c1ccc2c(c1)c(c[nH]2)C(CC(=O)c3ccc(cc3)Br)C(=O)O MS-6564 CC(=O)Nc1ccc(cc1)NC2=CC(=O)CCC2 MS-6565 CC(C)(C)c1c2c(nn1C)-c3ccc(cc3C2=O)[N+](=O)[O-] MS-6566 CCOc1ccc(cc1)NC=C2C(=O)c3ccccc3C2=O MS-6567 c1ccc(c(c1)NN=C(C#N)C#N)F MS-6568 CC1(CC(=C(C(=O)C1)Br)Nc2ccc(cc2)N(C)C)C MS-6569 c1ccc(cc1)C2CC(=CC(=O)C2)N3CCN(CC3)c4ccccc4 MS-6570 c1cc(cc(c1)OC(C(F)F)(F)F)NC=C(C#N)C#N MS-6571 c1cc(cc(c1)NC(=O)N/C(=C(/C#N)\N)/C#N)C(F)(F)F MS-6572 c1ccc(cc1)N/C=C(\C#N)/c2[nH]nnn2 MS-6573 CC(C)c1ccc(cc1)S(=O)(=O)Cc2nc(on2)C(F)(F)F MS-6574 c1ccc2c(c1)C(=O)C(=CNc3cc(ccc3Cl)C(F)(F)F)C2=O MS-6575 Cc1cc(no1)NC=C2C(=O)CC(CC2=O)CC(C)C MS-6576 COc1cc(cc(c1OC)OC)C(=O)N/N=C\2/c3ccccc3NC2=O MS-6577 CC(C)CC1CC(=CC(=O)C1)Nc2ccc(cc2)Cl MS-6578 c1ccc2c(c1)c(=O)oc(n2)/C=C/c3cccc(c3)[N+](=O)[O-] MS-6579 CC1(CC(=O)C(C(=O)C1)/N=N/c2ccccc2)C MS-6580 CC(C)(C)c1ccc(cc1)C2=NNC(=O)C(C2)c3cn(c4c3cccc4)C MS-6581 C#CCNC=C(C#N)C#N MS-6582 c1cc(ccc1S(=O)(=O)C2(CC2)C#N)Cl MS-6583 COc1ccc(cn1)NC(=O)COc2ccc(cc2Cl)Cl MS-6584 COC(=O)CNC(=O)/C=C/c1cccc(c1)[N+](=O)[O-] MS-6585 CC1(CC(=O)C(=CNc2ccc(cc2)Oc3ccc4ccccc4c3)C(=O)C1)C MS-6586 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)Nc3cccc(c3)OC(C(F)F)(F)F MS-6587 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F MS-6588 c1cc(c(c(c1)Cl)c2c([nH]nn2)C#N)Cl MS-6589 COc1ccc(cc1OC)NC(=O)c2ccccc2[N+](=O)[O-] MS-6590 CCOC(=O)/C(=C/1\c2ccccc2NC1=O)/C#N MS-6591 c1cc(ccc1N/C=C(/C#N)\c2[nH]nnn2)OC(F)(F)F MS-6592 CC1(C(NC(S1)c2ccccc2O)C(=O)O)C MS-6593 CC(C)(C)C(=O)/C(=C\Nc1nc(cs1)c2ccc(cc2)Br)/C#N MS-6594 c1cc(sc1)/C=N/C(=C(/C#N)\N)/C#N MS-6595 COc1ccc(cn1)NC=C2C(=O)c3ccccc3C2=O MS-6596 c1ccc(cc1)NC(=O)NNC(=O)c2ccc(cc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F MS-6597 CCO/N=C(\C)/c1ccccc1OCc2c(c(=O)n(n2C)c3ccccc3)Br MS-6598 c1ccnc(c1)/C=N/C(=C(/C#N)\N)/C#N MS-6599 CC(C)(C)c1c2c(nn1C(=O)c3ccc(cc3)Cl)-c4ccccc4C2=O MS-6600 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCC(=O)OC MS-6601 c1ccc(cc1)N(/C=C/C=[N+](c2ccccc2)c3ccccc3)c4ccccc4.[Cl-] MS-6602 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)N(C)C)c3ccccc3 MS-6603 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC#N MS-6604 CC(C)(C)C(=O)/C(=C\N1CCN(CC1)c2ccccc2)/C#N MS-6605 COc1ccc(cc1)C(=C2C(=O)c3ccccc3C2=O)NCCc4ccc(c(c4)OC)OC MS-6606 CC1(CC(=C(C(=O)C1)I)Nc2ccc(cc2)C(=O)O)C MS-6607 C=CCNC(=S)NNC(=O)COc1ccc(cc1)[N+](=O)[O-] MS-6608 Cc1ccc(c(c1)C)N/C=C/C=[NH+]/c2ccc(cc2C)C.[Cl-] MS-6609 c1cc(ccc1NN=C(C#N)C#N)F MS-6610 CC1(CC(=C(C(=O)C1)Cl)Nc2ccc(cc2)Cl)C MS-6611 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)OC(F)(F)F)/C#N MS-6612 CC(=O)c1ccc(cc1)NC=C2C(=O)c3ccccc3C2=O MS-6613 CS/C(=N\N=C\c1ccc2c(c1)OCO2)/[NH3+].[I-] MS-6614 COc1ccccc1/C=N/N=C(/[NH2+]CC=C)\SC.[I-] MS-6615 c1cc(c(cc1F)F)N/C=C/C=[NH+]/c2ccc(cc2F)F.[Cl-] MS-6616 CC1(CC2=C(C(Nc3cc(ccc3N2)Cl)c4c(cccc4Cl)F)C(=O)C1)C MS-6617 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)SC(F)(F)F MS-6618 Cc1ccc2cccc(c2n1)Oc3ccc(cc3[N+](=O)[O-])Cl MS-6619 c1cc(ccc1C2NC(CS2)C(=O)O)OC(F)(F)F MS-6620 Cc1cc(ccc1F)c2csc(n2)NC=C3C(=O)c4ccccc4C3=O MS-6621 c1ccc(cc1)NC2=CC(=O)CCC2 MS-6622 CC(C)CC(=O)C1C(=O)c2ccccc2C1=O MS-6623 c1ccc(c(c1)Nc2nc(cs2)c3ccc(cc3)Br)Cl MS-6624 c1ccc2c(c1)/C(=N/Nc3ccc(cc3)[N+](=O)[O-])/C(=O)N2 MS-6625 c1ccc2c(c1)/C(=N/N)/C(=O)N2 MS-6626 Cc1c(sc(n1)c2cccnc2)C(=O)C MS-6627 c1cc(cnc1)c2nc(cs2)c3ccc(cc3)Br MS-6628 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccc(cc3)N MS-6629 c1ccc(cc1)NC(=S)NNC(=S)Nc2ccccc2 MS-6630 c1ccc(cc1)CNC2=C(C(=O)CCC2)I MS-6631 c1ccc(cc1)Nc2ccc(cc2)/N=C\3/c4ccccc4NC3=O MS-6632 CC1(OC(=O)C(=CNCCc2ccccc2)C(=O)O1)C MS-6633 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=O)Nc2ccccc2 MS-6634 CC1CC(=O)C(=CNc2ccc(cc2)C(=O)C)C(=O)C1 MS-6635 CS(=O)(=O)NNC(=O)COc1ccc(cc1Cl)Cl MS-6636 Cc1ccc(cc1)S(=O)(=O)NNC(=O)COc2ccc(cc2Cl)Cl MS-6637 CC(=O)Nc1ccc(cc1)NC=C2C(=O)OC(OC2=O)(C)C MS-6638 CC1CC(=O)C(=CNc2ccccc2)C(=O)C1 MS-6639 c1ccc(cc1)NC(=S)NN=C2c3ccccc3NC2=O MS-6640 c1ccc(cc1)NC2=C(C(=O)c3c2cccc3)Br MS-6641 c1cc(ccc1NC2=C(C(=O)CCC2)Cl)F MS-6642 CC1CC(=C(C(=O)C1)Cl)Nc2ccc(cc2)C(=O)C MS-6643 CC(=O)c1ccc(cc1)NC2=C(C(=O)CC(C2)(C)C)Br MS-6644 CC(C)(C)c1c2c(n[nH]1)-c3ccccc3C2=O MS-6645 CC1(CC(=CC(=O)C1)Nc2ccc(cc2N)Cl)C MS-6646 CC(=O)Nc1ccc(cc1)NC2=C(C(=O)CCC2)Br MS-6647 Cc1ccc(cc1)S(=O)(=O)CC(=O)N MS-6648 Cc1cc(ccc1OCc2n[nH]c(=S)n2c3ccccc3)Cl MS-6649 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)O)/C#N MS-6650 CC1(CC(=CC(=O)C1)N2CCN(CC2)c3ccccc3)C MS-6651 c1ccc(cc1)C2CC(=C(C(=O)C2)Cl)Nc3ccc(cc3)I MS-6652 Cc1c(c(=O)n(n1C)c2ccccc2)NC=C(C#N)C#N MS-6653 Cc1ccc(cc1)S(=O)(=O)CC(=O)C(C)(C)C MS-6654 c1ccc(cc1)N2C(=O)CSC2=C(C#N)C#N MS-6655 COC(=O)/C(=C/1\N(C(=O)CS1)c2ccccc2)/C#N MS-6656 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)[N+](=O)[O-] MS-6657 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4cccc(c4)[N+](=O)[O-] MS-6658 CC(C)c1ccc(cc1)NC(=C2C(=O)c3ccccc3C2=O)C MS-6659 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)N MS-6661 CC(C)c1ccc(cc1)NC2=C(C(=O)c3c2cccc3)c4ccc(c(c4)OC)OC MS-6662 CC(C)c1ccc(cc1)NC2=C(C(=O)c3c2cccc3)c4ccccc4 MS-6663 Cc1ccc(cc1)S(=O)(=O)/C(=C(/NC)\SC)/C#N MS-6664 c1cc(c(cc1Cl)Cl)S(=O)(=O)CC#N MS-6665 c1c(cc(cc1C(F)(F)F)NC(=C(C#N)C#N)C#N)C(F)(F)F MS-6666 CCO/C=C(\C(=O)C)/S(=O)(=O)c1ccc(cc1)Cl MS-6667 CC1(CC(=CC(=O)C1)Nc2[nH]nnn2)C MS-6668 CC(C)(C)C(=O)/C(=C/c1ccc(c(c1)OC)O)/C#N MS-6669 CC(C)(C)C(=O)/C(=C/c1cccc(c1)Oc2ccccc2)/C#N MS-6670 CSC(=C1C(=O)c2ccccc2C1=O)SC MS-6671 CC1CC(=CC(=O)C1)NNc2ccccc2 MS-6672 Cc1cc(no1)NC2=C(C(=O)c3c2cccc3)c4ccccc4 MS-6673 COc1ccc(cn1)N/C=C(/C#N)\c2[nH]nnn2 MS-6674 c1ccc2c(c1)C(=O)c3c(ccc(c3C2=O)NC=C(C#N)C#N)N MS-6675 c1ccc2c(c1)c(c[nH]2)C3CC(=NNC3=O)c4ccc(cc4)Br MS-6676 c1ccc(cc1)Oc2cccc(c2)C=C3C(=O)c4ccccc4C3=O MS-6677 c1cc(ccc1[N+](=O)[O-])OCC(=O)NNC(=S)NC2CCCCC2 MS-6678 c1ccc(c(c1)C(=O)N)NC(=C(C#N)C#N)C#N MS-6679 COc1cc(cc(c1OC)OC)/C=N/C(=C(/C#N)\N)/C#N MS-6680 c1cc(c(cc1/C=C/c2nc3c(cc(cc3Cl)Cl)c(=O)o2)[N+](=O)[O-])Cl MS-6681 c1ccc(cc1)C#CC(=O)Nc2ccccc2C(=O)N MS-6682 c1ccc(c(c1)C(=O)N)NC(=O)/C=C/c2cccc(c2)[N+](=O)[O-] MS-6683 c1ccc(c(c1)C(=O)N)NC(=O)/C=C/c2cc(ccc2Sc3ccccn3)[N+](=O)[O-] MS-6684 CC(C)(C)C(=O)/C(=C/NCCC(=O)O)/C#N MS-6685 CC(C)(C)c1ccc(cc1)S(=O)(=O)C/C(=N/O)/N MS-6686 CC(C)(C)c1ccc(cc1)S(=O)(=O)C/C(=N/OC(=O)c2cccs2)/N MS-6687 c1cc(sc1)C(=O)Nc2ccc(cc2)NC=C(C#N)C#N MS-6688 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3Cl)Cl MS-6689 Cc1ccc2cccc(c2n1)Oc3ccc(cc3)NC=C(C#N)C#N MS-6690 COCC(=O)NCCc1c[nH]c2c1cccc2 MS-6691 CC1(CC(=O)C(=CNc2ccc(cc2OC)[N+](=O)[O-])C(=O)C1)C MS-6692 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)Nc3ccc(cc3)F MS-6693 c1cc(cc(c1)Oc2ccc(cc2)N)C(F)(F)F MS-6694 Cn1cc(c2c1cccc2)C(CC(=O)c3ccc(cc3)C4CCCCC4)C(=O)O MS-6695 c1ccc2cc(ccc2c1)Oc3ccc(cc3N)C(F)(F)F MS-6696 c1cc(cc(c1)C(F)(F)F)c2c([nH]nn2)C#N MS-6697 c1cc2c(cc1c3c([nH]nn3)C#N)OCO2 MS-6698 CC1(Cc2c(c(nn2C)c3ccc(c(c3)OC)OC)/C(=N\O)/C1)C MS-6699 c1ccc2c(c1)c(c[nH]2)CCNC(=O)/C=C/c3ccc(c(c3)[N+](=O)[O-])Cl MS-6700 CN(C)N=C(c1ccc(cc1)OC)C2C(=O)c3ccccc3C2=O MS-6701 Cc1cc(nc(n1)NC(=C2C(=O)c3ccccc3C2=O)C)C MS-6702 CC1(C(NC(S1)c2ccc3c(c2)OCO3)C(=O)O)C MS-6703 c1cc(ccc1[N+](=O)[O-])Oc2c(cc(cn2)C(F)(F)F)Cl MS-6704 Cn1c2c(c(n1)c3ccc(c(c3)OC)OC)C(=O)CCC2 MS-6705 COc1ccc(cc1OC)C2NC(CS2)C(=O)O MS-6706 c1cc(c(cc1Cl)Cl)/C=N/C(=C(/C#N)\N)/C#N MS-6707 c1ccc(cc1)C2CC3=NNC(=CC3C(=O)C2)c4ccc(cc4)Br MS-6708 CC(C)(C)C(=O)/C(=C\c1ccc(c(c1)[N+](=O)[O-])O)/C#N MS-6709 Cc1ccc2c(c1)NC(=C3C(=O)c4ccccc4C3=O)N2 MS-6710 C/C(=N/OC)/c1ccccc1OCc2c(c(=O)n(n2C)c3ccccc3)Br MS-6711 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)OC(F)(F)F MS-6712 c1cc(ccc1S(=O)(=O)C/C(=N/O)/N)Cl MS-6713 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] MS-6714 CC1(OC(=O)C(=CNc2cc(ccc2Oc3ccc4ccccc4c3)C(F)(F)F)C(=O)O1)C MS-6715 CC1(OC(=O)C(=CNc2ccc(nc2)OC)C(=O)O1)C MS-6716 Cn1cc(c2c1cccc2)/C=N/C(=C(/C#N)\N)/C#N MS-6717 c1cc(ccc1n2cnc(c2Cl)Cl)[N+](=O)[O-] MS-6718 c1ccc2c(c1)C(=O)c3cccc(c3C2=O)NC=C(C#N)C#N MS-6719 CCC1CC(=O)C(=CNc2ccc(cc2)OC(F)(F)F)C(=O)C1 MS-6720 c1ccc(cc1)N/C=C/C=[NH+]/c2ccccc2.[Cl-] MS-6721 CC1(Cc2cccc(c2O1)Oc3ccc(cc3)[N+](=O)[O-])C MS-6722 Cc1ccc(c(c1)[N+](=O)[O-])NC=C(C#N)C#N MS-6723 CC1(C(NC(S1)c2ccc(cc2)Br)C(=O)O)C MS-6724 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)Nc3ccc(cc3)SC(F)(F)F MS-6725 COc1ccc(cc1)c2c3c(n(n2)c4ccccc4)-c5ccccc5C3=O MS-6726 c1cc(ccc1/C=N/C(=C(/C#N)\N)/C#N)Cl MS-6727 CC(=O)c1cccc(c1)NC(=O)Nc2ccccc2 MS-6728 CC(C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)S(=O)(=O)c2ccc(cc2)Cl MS-6729 c1cc2c(cc1/C=N/C(=C(/C#N)\N)/C#N)OCO2 MS-6730 CC(C(=O)N/N=C\1/c2cc(ccc2NC1=O)Br)Oc3ccc(cc3Cl)Cl MS-6731 c1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2)[N+](=O)[O-] MS-6732 c1ccc(cc1)C(=O)NNC(=O)Nc2cccc(c2)C(F)(F)F MS-6733 COc1ccc(cc1OC)CCNC(=C2C(=O)c3ccccc3C2=O)c4ccccc4 MS-6734 Cc1cc(ccc1OCC(=O)N/N=C(/C)\C2C(=O)c3ccccc3C2=O)Cl MS-6736 c1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2Cl)Cl MS-6737 c1ccc2c(c1)[nH]c(n2)SCC(=O)NN MS-6738 c1ccnc(c1)NC(=O)c2ccc(cc2)[N+](=O)[O-] MS-6739 c1cc(cc(c1)NC(=O)c2ccc(cc2)[N+](=O)[O-])C(F)(F)F MS-6740 c1cc(ccc1C(=O)Nc2ccc(cc2F)F)[N+](=O)[O-] MS-6741 c1ccc2c(c1)c(c[nH]2)C=C(C#N)C#N MS-6742 C=CCNC(=S)NNC(=O)Nc1ccc(cc1)Cl MS-6744 c1cc(ccc1C(=O)Nc2ccc(cc2F)F)N MS-6745 c1cc(ccc1C(=O)Nc2ccc(cc2)Cl)N MS-6746 c1cc(cc(c1)NC(=O)c2ccc(cc2)N)C(F)(F)F MS-6747 Cc1ccc2cccc(c2n1)Oc3ccc(cn3)C(F)(F)F MS-6748 CC(=C1C(=O)c2ccccc2C1=O)NCC=C MS-6749 CC(C)(C)C(=O)/C(=C\NC(C)(C)C)/C#N MS-6750 c1cc(ccc1SCC#N)Cl MS-6751 COC(=O)CSc1cccc(c1C#N)F MS-6753 c1cc(c(cc1Cl)S(=O)(=O)CC#N)Cl MS-6755 c1ccc(c(c1)C(=O)O)NC(=O)/C=C/C(=O)O MS-6756 c1cc(cc(c1)NC(=O)/C=C/C(=O)O)C(=O)O MS-6757 c1cc(ccc1C(=O)O)NC(=O)/C=C/C(=O)O MS-6758 Cc1ccc(cc1)Sc2ccc(cc2/C=N/C(=C(/C#N)\N)/C#N)[N+](=O)[O-] MS-6759 CN(C)c1ccc(cc1)NC=C(C#N)C#N MS-6760 c1ccc(cc1)NC=C(C#N)C#N MS-6761 CC(C)CC1CC(=O)C(=CNc2ccc(cc2)C(=O)C)C(=O)C1 MS-6762 c1cc(c(c(c1)Cl)Cl)OCC(=O)NNC(=S)NC2CCCCC2 MS-6763 CC(C)(C)C1=NN(C(=O)C1=Cc2ccc(cc2)N(C)C)C MS-6764 CC(C)(C)C\1=NN(C(=O)/C1=C/c2cccc(c2)Oc3ccccc3)c4ccc(cc4)[N+](=O)[O-] MS-6765 c1cc(ccc1Oc2ccc(cc2/C=N/NC(=S)N)[N+](=O)[O-])Br MS-6766 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)NC(=S)Nc3ccccc3)C MS-6767 c1ccc(cc1)NC(=S)NNC(=O)c2ccccc2N MS-6768 Cc1ccc(c(c1)C)OCC(=O)NNC(=S)Nc2ccccc2 MS-6769 Cc1ccc(c(c1)C)OCC(=O)NNC(=O)Nc2ccccc2 MS-6770 Cc1ccc(c(c1)C)OCC(=O)NNC(=S)NCC=C MS-6771 c1cc(ccc1N/C=C/C=[NH+]/c2ccc(cc2)Br)Br.[Cl-] MS-6772 Cc1ccc(cc1C)OCC(=O)NCCc2ccc(c(c2)OC)OC MS-6773 COc1ccc(c(c1)[N+](=O)[O-])N/C=C/C=[NH+]/c2ccc(cc2[N+](=O)[O-])OC.[Cl-] MS-6774 CC1CC(=CC(=O)C1)Nc2ccc(cc2)NC(=O)Nc3ccccc3 MS-6775 CC(=O)c1ccc(cc1)NC2=C(C(=O)CC(C2)(C)C)I MS-6776 c1cc(cc(c1)OC(C(F)F)(F)F)NC(=O)CCl MS-6777 CC(C)c1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)Nc4ccccc4N2 MS-6778 CC(C)CC1CC(=O)C(=CNc2cc(cc(c2)Cl)Cl)C(=O)C1 MS-6779 Cc1cccc(c1C)OCC(=O)Nc2ccc(cc2)OC(F)(F)F MS-6780 Cc1cccc(c1C)OCC(=O)Nc2cc(ccc2OC)OC MS-6781 c1cc(c(c(c1)Cl)Cl)OCC(=O)NNC(=S)Nc2ccc(cc2)Cl MS-6782 c1cc2c(cc1Br)/C(=N/NC(=S)N)/C(=O)N2 MS-6783 CC1(CC(=C(C(=O)C1)I)Nc2cccc3c2nccc3)C MS-6784 c1ccc2c(c1)c3c([nH]2)nc(nn3)Sc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-] MS-6785 Cc1csc(c1NC=C2C(=O)c3ccccc3C2=O)C(=O)OC MS-6786 COc1ccc(cc1OC)CCNC(=O)c2cccnc2Oc3ccc(cc3)Cl MS-6787 CC(C(=O)Nc1ccc(cc1)OC(F)(F)F)Cl MS-6788 Cc1ccc(c(c1)C)Oc2c(cccn2)C(=O)O MS-6789 Cc1cc(nc(n1)N/C=C(\C#N)/C(=O)OCc2cccc(c2)Oc3ccccc3)C MS-6791 CC1Cc2c(cc(nn2)c3ccc(cc3Cl)Cl)/C(=N\OC)/C1 MS-6792 c1ccc2c(c1)C(=O)C(=CNc3cc(ccc3[N+](=O)[O-])C(F)(F)F)C2=O MS-6793 CCC1(Nc2ccccc2C(=O)N1)C MS-6794 c1ccc2c(c1)C(=O)C(C2=O)C(=O)C3CC3 MS-6795 CC(C)(C)C1CCC2(CC1)Nc3ccccc3C(=O)N2 MS-6796 CNC(=C(C#N)C#N)S MS-6797 c1cc(sc1)C(=O)Nc2ccc(cc2)[N+](=O)[O-] MS-6798 COc1ccc(cc1c2csc(n2)Nc3ccccc3)O MS-6799 COc1ccc(cc1OC)CCNC(=O)c2ccc(cc2)[N+](=O)[O-] MS-6800 COc1ccc(cc1OC)C(=O)C2C(=O)c3ccccc3C2=O MS-6801 c1cc(ccc1C(=O)Nc2ccc(cn2)C(F)(F)F)[N+](=O)[O-] MS-6802 c1ccc(cc1)C(=O)NNC(=S)Nc2ccccc2 MS-6803 c1ccnc(c1)Sc2ccc(cc2)NC3=CC(=O)CCC3 MS-6804 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] MS-6805 Cc1c(c(c(c(c1F)F)NNC(=O)Nc2ccc(c(c2)Cl)Cl)F)F MS-6806 c1ccc(c(c1)C(=O)N)NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])Cl MS-6807 c1cc(c(cc1c2csc(n2)[NH3+])Cl)Cl.[Br-] MS-6808 CC1(CC2=C(C(Nc3ccc(cc3N2)C(=O)O)c4c[nH]c5c4cccc5)C(=O)C1)C MS-6809 COc1cc(ccc1O)C2NC(CS2)C(=O)O MS-6810 CN(C)c1ccc(cc1)C2NC(CS2)C(=O)O MS-6811 c1ccc(cc1)C2CC(=C(C(=O)C2)Cl)Nc3ccccc3C(=O)O MS-6812 CCCC(=O)Nc1ccccc1C(=O)OC MS-6813 COc1ccc(cc1)c2c(n[nH]n2)C#N MS-6814 c1ccc(c(c1)CC(=O)O)C(=O)Nc2ccc(cc2F)F MS-6815 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3cccs3 MS-6816 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCc3ccccc3 MS-6817 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(C)(C)C#C MS-6818 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCc3ccc(c(c3)OC)OC MS-6819 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3ccccc3 MS-6820 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)/C(=N/OC(=O)c4c(onc4c5ccccc5Cl)C)/C MS-6821 CC(=C1C(=O)c2ccccc2C1=O)NCCc3c[nH]c4c3cccc4 MS-6822 CCc1cccc2c1[nH]cc2C(CC(=O)c3ccc(cc3)Br)C(=O)O MS-6823 COc1ccc(cc1OC)CNC2=C(C(=O)CCC2)I MS-6824 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3nc[nH]n3 MS-6825 c1cc(sc1)C2=NS(=O)(=O)NC(=C2)C(F)(F)F MS-6826 c1cc(cc(c1)NC2=CC(=O)CCC2)C(F)(F)F MS-6827 c1cc(cc(c1)NC2=C(C(=O)CCC2)Cl)C(F)(F)F MS-6829 c1ccc(c(c1)C(=O)O)NC2=C(C(=O)CCC2)Cl MS-6830 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)NCC=C MS-6831 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2c3ccccc3 MS-6832 C1CC(=CC(=O)C1)N2CCOCC2 MS-6833 CC(C)(C)C1=NOC2(C1C(=O)c3c2cccc3)O MS-6834 CC(C)(C)C(=N)C1C(=O)c2ccccc2C1=O MS-6835 c1ccc(cc1)C2=NCCNC(=C2)C(F)(F)F MS-6836 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)C(=O)O)C MS-6837 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)N(C)C)C MS-6838 CC(=O)c1ccc(cc1)NC=C2C(=O)CC(CC2=O)(C)C MS-6839 COC(=O)/C(=C(/Nc1cccc(c1)C(F)(F)F)\O)/C#N MS-6840 CS/C(=C(\C#N)/S(=O)(=O)c1ccccc1)/Nc2ccccc2 MS-6841 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cn3)Br MS-6842 C/C(=N\NC(=O)COc1cccc2c1cccc2)/C3C(=O)c4ccccc4C3=O MS-6843 Cn1c2ccccc2c3c1nc(nn3)SCc4ccccc4 MS-6844 CCOc1ccc(cc1)C=C(C#N)C#N MS-6845 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cc2)OC(F)(F)F)/[N+](=O)[O-] MS-6846 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-] MS-6847 c1ccc(cc1)N2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccccc3 MS-6848 CS/C(=C(/C#N)\S(=O)(=O)c1ccccc1)/Nc2cccc(c2)Cl MS-6849 CCC(CC)(C#C)N/C=C(/[N+](=O)[O-])\S(=O)(=O)c1ccc(cc1)Br MS-6850 c1ccc(cc1)N/C(=C(/C#N)\S(=O)(=O)c2ccccc2)/O MS-6851 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2cc(nc3c2cccc3)C)/C#N MS-6852 CC(C)C(=O)C1C(=O)c2ccccc2C1=O MS-6853 CCOc1ccc(cc1)C2C(=C(OC3=C2C(=O)CC(C3)(C)C)N)C#N MS-6854 Cc1ccc(cc1)S(=O)(=O)/C(=C(/Nc2ccccc2)\O)/C#N MS-6855 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ncccn2)/C#N MS-6856 Cc1cc(c2ccccc2n1)N/C=C(\C#N)/S(=O)(=O)c3ccccc3 MS-6857 Cc1ccc(cc1)S(=O)(=O)/C(=C(/Nc2ccccc2)\S)/C#N MS-6858 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2cc(cc(c2)Cl)Cl)/C#N MS-6859 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl MS-6860 c1ccc(cc1)N\2C(=O)CS/C2=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl MS-6861 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)F MS-6862 CN/C(=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl)/SC MS-6863 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cc2)OC(F)(F)F)/C#N MS-6864 c1cc(ccc1C2C(=C(OC3=C2C(=O)CCC3)N)C#N)OC(F)(F)F MS-6865 c1cc(ccc1N/C=C(\[N+](=O)[O-])/S(=O)(=O)c2ccc(cc2)Cl)SC(F)(F)F MS-6866 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(c(c3)OC)OC)C(=O)C1)C MS-6867 COc1ccc(cc1OC)C2C(=C(OC3=C2C(=O)CCC3)N)C#N MS-6868 Cc1cccc(c1)C(=O)NCCc2c[nH]c3c2cccc3 MS-6869 c1ccc(cc1)Oc2cccc(c2)C=C(C#N)C#N MS-6870 CC1(CC2=C(C(C(=C(O2)N)C#N)c3c[nH]c4c3cccc4)C(=O)C1)C MS-6871 CSc1ccc(cc1)C=C(C#N)C#N MS-6872 c1ccc(cc1)NC(=S)N2CCCN(CC2)C(=S)Nc3ccccc3 MS-6873 CC1CN(C(CN1C(=S)Nc2ccccc2)C)C(=S)Nc3ccccc3 MS-6874 CC1CN(C(CN1C(=O)Nc2ccc(cc2)Cl)C)C(=O)Nc3ccc(cc3)Cl MS-6875 CC1CN(C(CN1C(=O)Nc2ccccc2)C)C(=O)Nc3ccccc3 MS-6876 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)C(C)C MS-6877 COc1ccc(cc1OC)CCNC(=O)c2ccc(cc2)Cl MS-6878 c1ccc2c(c1)C(=O)c3cccc(c3C2=O)N/C=C(/C#N)\S(=O)(=O)c4ccc(cc4)Cl MS-6879 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(ccc2Cl)C(F)(F)F)/C#N)Cl MS-6880 c1ccc(cc1)S(=O)(=O)/C(=C(\Nc2cccc(c2)C(F)(F)F)/O)/C#N MS-6881 CC(C)c1ccc(cc1)S(=O)(=O)CC#N MS-6882 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3)Cl MS-6883 CC1CC2=C(C(C(=C(O2)N)C#N)c3ccc4c(c3)OCO4)C(=O)C1 MS-6884 CC1CC2=C(C(C(=C(O2)N)C#N)c3cccs3)C(=O)C1 MS-6885 CC1CC2=C(C(C(=C(O2)N)C#N)c3ccc4ccccc4c3)C(=O)C1 MS-6886 c1ccc(cc1)NC(=O)N2CCCN(CC2)C(=O)Nc3ccccc3 MS-6887 CC1(CC(=O)C(C(=O)C1)CC(=O)c2ccc(cc2)Br)C MS-6888 c1ccc2cc(ccc2c1)C=C(C#N)C#N MS-6889 c1ccc2cc(ccc2c1)C3C(=C(OC4=C3C(=O)CCC4)N)C#N MS-6890 c1cc(ccc1NC(=O)N2CCCN(CC2)C(=O)Nc3ccc(cc3)Cl)Cl MS-6891 CC(=O)c1ccc(cc1)NC=C2C(=O)CC(CC2=O)c3ccccc3 MS-6892 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)C(F)(F)F MS-6893 c1cc(ccc1c2csc([nH+]2)N)F.[Br-] MS-6894 CCOC(=O)/C(=C/NCCc1ccccc1)/C#N MS-6895 CC1(CC(=O)C(C(=O)C1)C(=S)Nc2cccc(c2)C(F)(F)F)C MS-6896 CC1(CC(=C(C(=O)C1)I)NCc2ccccc2)C MS-6897 Cc1c(sc([nH+]1)Nc2ccccn2)C(=O)C.[Cl-] MS-6898 Cc1ccc(cc1)NC2=C(C(=O)c3c2cccc3)c4ccccc4 MS-6899 c1ccc2c(c1)C(=O)C(=CNc3c(cc(cn3)C(F)(F)F)Cl)C2=O MS-6900 c1ccc2c(c1)C(=O)C(C2=O)c3ccncc3 MS-6901 CC1(CC(=CC(=O)C1)Nc2ccccc2F)C MS-6903 CC(=O)c1ccc(cc1)N/C=C(\C#N)/C(=O)C(C)(C)C MS-6904 Cc1c(sc([nH+]1)Nc2ncccn2)C(=O)C.[Cl-] MS-6905 CC(C)(C)C(=O)/C(=C\Nc1ccc(cc1F)F)/C#N MS-6906 CC(C)(C)C(=O)/C(=C\Nc1ccc(cc1)OC)/C#N MS-6907 CC(C)(C)C(=O)/C(=C\Nc1ccccc1C(F)(F)F)/C#N MS-6908 CC(C)(C)C(=O)/C(=C/Nc1cccc2c1nccc2)/C#N MS-6909 CCOC(=O)/C(=C/c1c(cc(cc1OC)OC)OC)/C#N MS-6910 c1ccc(c(c1)Nc2nc(cs2)c3ccc(cc3)F)Cl MS-6911 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(cc(c2)Cl)Cl)/C#N)Cl MS-6912 CC(C)(C)C(=O)/C(=C/Nc1ccc(cc1)Oc2ccccc2)/C#N MS-6913 c1ccc(cc1)Oc2ccc(cc2)N3C(=O)CSC34c5ccccc5NC4=O MS-6914 CCOc1ccc(cc1)/N=C\2/c3ccccc3NC2=O MS-6915 CCOC(=O)c1c(nc(s1)Nc2ccccc2Cl)C MS-6916 c1ccc(cc1)C(=O)NCCc2c[nH]c3c2cccc3 MS-6917 CC1(OC(=O)C(=CNc2ccc3c(c2)OCO3)C(=O)O1)C MS-6918 CC1(OC(=O)C(=CN(c2ccccc2)c3ccccc3)C(=O)O1)C MS-6919 COc1cc2c(cc1OC)nc-3c(c2c4ccc5ccccc5c4)C(=O)c6c3cccc6 MS-6920 c1ccc2cc(ccc2c1)S(=O)(=O)NCCc3c[nH]c4c3cccc4 MS-6921 Cc1ccc(c(c1)C)NC(=O)c2c(onc2c3ccccc3Cl)C MS-6922 c1cc(cc(c1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F MS-6923 c1cc(ccc1C(F)(F)F)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-6924 CC(C)(C)S(=O)(=O)/C(=C/Nc1ccc(cc1)C(F)(F)F)/C#N MS-6925 c1cc(ccc1S(=O)(=O)/C(=C\Nc2cc(ccc2F)C(F)(F)F)/C#N)Cl MS-6926 CC(C)(C)S(=O)(=O)/C(=C\Nc1cccc(c1)C(F)(F)F)/C#N MS-6927 c1cc(cc(c1)F)N/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl MS-6928 COc1ccc(cn1)NS(=O)(=O)c2ccc3ccccc3c2 MS-6929 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc4c(c3)OCO4 MS-6930 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)F)C2=O MS-6931 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc4ccccc4c3 MS-6932 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc(c3)Br MS-6933 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(C)(C)CC(C)(C)C MS-6934 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)C(=O)C MS-6935 c1ccc2c(c1)/C(=N/c3cccc(c3)Br)/C(=O)N2 MS-6936 c1ccc2c(c1)cccc2Nc3[nH+]c(cs3)c4ccc(cc4)Cl.[Cl-] MS-6937 CSc1ccc(cc1)/C=N/C(=C(/C#N)\N)/C#N MS-6939 CC(C)(C)C(=O)/C(=C/c1ccc2ccccc2c1)/C#N MS-6940 CCCCCCCCNC(=O)c1c(onc1c2ccccc2Cl)C MS-6941 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F MS-6942 c1ccc2c(c1)C(=O)C(=CN3CCN(CC3)c4ccccc4F)C2=O MS-6943 CC(=C1C(=O)c2ccccc2C1=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-6944 CC1Cc2c(cc(n2c3ccc(cc3)OC(F)(F)F)c4ccc(cc4)Br)C(=O)C1 MS-6945 Cc1cc2c(n1c3ccc(c(c3)C(F)(F)F)F)CC(CC2=O)(C)C MS-6946 c1cc(ccc1C(F)(F)F)Oc2ccc(cc2/C=N/C(=C(/C#N)\N)/C#N)[N+](=O)[O-] MS-6947 COc1ccc(cc1OC)CCNC(=O)CSc2c(cc(cn2)C(F)(F)F)Cl MS-6948 COC(=O)c1c(c2cc(ccc2s1)[N+](=O)[O-])/N=N/C(C#N)C#N MS-6949 CC1(CC(=O)C(=CNc2ccc(cc2)SC)C(=O)C1)C MS-6950 c1c(cnc(c1Cl)SC(=[NH2+])N)C(F)(F)F.[Cl-] MS-6951 CC(C)(C)C(=O)/C(=C\N1CCN(CC1)c2ccccc2F)/C#N MS-6952 c1ccc(c(c1)N2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)F MS-6953 c1ccc(c(c1)N2CCN(CC2)C=C(C#N)C#N)F MS-6954 CC1(CC(=O)C(=CNc2cc(c(cc2OC)Br)OC)C(=O)C1)C MS-6955 CC1(Cc2c(cc(n2c3cccc(c3)C(=O)O)c4ccc(cc4)Br)C(=O)C1)C MS-6956 Cc1cc2c(n1c3cccc(c3)C(=O)O)CC(CC2=O)(C)C MS-6957 CC1(Cc2c(cc(n2c3ccc(cc3)C(=O)O)c4ccc(cc4)Br)C(=O)C1)C MS-6958 CC1(Cc2c(cc(n2c3ccc(nc3)OC)c4ccc(cc4)Br)/C(=N\OC)/C1)C MS-6959 CC1(Cc2c(cc(n2c3ccc(nc3)OC)c4ccc(cc4)Br)/C(=N/OCC=C)/C1)C MS-6960 c1ccc(cc1)N2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl MS-6961 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl MS-6962 c1ccc2c(c1)C(=O)C(C2=O)C(=O)/C=C/c3ccc(cc3)Br MS-6963 CC1(OC(=O)C(=CNc2cc(c(cc2OC)Br)OC)C(=O)O1)C MS-6964 c1cc(c(c(c1)Cl)C/C(=N\O)/N)Cl MS-6965 Cc1ccc(c(c1)[O-])C(=O)O.Cc1ccc(c(c1)[O-])C(=O)O.[Cu+2] MS-6966 c1ccc(c(c1)C/C(=N\O)/N)[N+](=O)[O-] MS-6967 c1cc(ccc1OCC(=O)NN)Br MS-6968 c1cc(ccc1NC(=O)NNC(=O)COc2ccc(cc2)Br)Cl MS-6969 c1ccc(c(c1)/C=C/C=N/C(=C(/C#N)\N)/C#N)[N+](=O)[O-] MS-6970 c1cc(c(cc1Cl)/C=N/C(=C(/C#N)\N)/C#N)O MS-6971 CC(=O)Nc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O MS-6972 CC(=C1C(=O)c2ccccc2C1=O)NCc3ccncc3 MS-6973 c1cc(ccc1C/C(=N\O)/N)Br MS-6975 CC(C)(C)C(=O)/C(=C\c1cccc(c1)Br)/C#N MS-6976 CC(C)(C)C(=O)/C(=C\c1ccc(cc1)C(=O)O)/C#N MS-6977 c1cc(ccc1/C=N/C(=C(/C#N)\N)/C#N)C(=O)O MS-6978 CC(=O)Nc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)Nc4ccccc4N2 MS-6979 CC1(CC2=C(C(Nc3ccccc3N2)c4cccc(c4)Br)C(=O)C1)C MS-6980 CC(=O)Nc1ccc(cc1)/C=C(\C#N)/C(=O)c2ccccc2 MS-6981 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)C(=O)O)C(=O)C1)C MS-6982 CN(C)c1ccc(cc1)/C=N/C(=C(/C#N)\N)/C#N MS-6983 COc1ccc(cc1)OCC(=O)NNC(=S)Nc2ccccc2 MS-6984 COc1ccc(cn1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-6986 COc1ccc(cc1)OCC(=O)NN MS-6987 CC(C)(C)c1c\2c(n(n1)C)-c3ccccc3/C2=N\O MS-6988 CO/N=C\1/c2ccccc2-c3c1c(n[nH]3)C4CC4 MS-6989 COc1ccc(c(c1)S(=O)(=O)Nc2ccccc2C(=O)N)OC MS-6990 CC1(Cc2c(cc(n2c3ccc(cc3)F)c4ccc(cc4)Br)C(=O)C1)C MS-6991 Cc1cc2c(n1c3ccc(cc3)F)CC(CC2=O)(C)C MS-6992 c1cc(ccc1S(=O)(=O)/C(=C\Nc2ccc(cc2C(F)(F)F)F)/C#N)Cl MS-6993 c1cc(cc(c1)Br)C(=O)Cn2cnc(c2Cl)Cl MS-6994 Cc1ccc(c(c1)C)NC(=C2C(=O)c3ccccc3C2=O)C MS-6995 COc1ccc(cc1)OCC(=O)NNC(=O)Nc2ccc(cc2)Cl MS-6996 COc1ccc(cc1)OCC(=O)NNC(=O)NC2CCCCC2 MS-6997 COc1ccc(cc1)OCc2n[nH]c(=S)n2c3ccccc3 MS-6998 COc1ccc(cc1)OCC(=O)N/N=C\2/c3ccccc3NC2=O MS-6999 c1ccc(c(c1)/C=C/C=C2C(=O)c3ccccc3C2=O)[N+](=O)[O-] MS-7000 c1ccc(cc1)C2c3c(=O)[nH]c(=O)[nH]c3OC(=C2C#N)N MS-7001 Cc1c2c([nH]n1)OC(=C(C2c3ccc(cc3)Br)C#N)N MS-7002 Cc1c2c([nH]n1)OC(=C(C2c3ccc(cc3)Cl)C#N)N MS-7003 Cc1c2c([nH]n1)OC(=C(C2c3ccccc3OC)C#N)N MS-7004 Cc1c2c([nH]n1)OC(=C(C2c3ccccc3F)C#N)N MS-7005 Cc1c2c([nH]n1)OC(=C(C2c3ccc(cc3)F)C#N)N MS-7006 Cc1c2c([nH]n1)OC(=C(C2c3cccc(c3)[N+](=O)[O-])C#N)N MS-7007 Cc1c2c([nH]n1)OC(=C(C2c3ccc(cc3)[N+](=O)[O-])C#N)N MS-7008 CCOC(=O)C1=C(OC2=C(C1c3ccccc3F)C(=O)CC(C2)(C)C)N MS-7009 CC1(CC2=C(C(C(=C(O2)N)C(=O)OC)c3cccc(c3)[N+](=O)[O-])C(=O)C1)C MS-7010 CC1(CC2=C(C(C(=C(O2)N)C(=O)OC)c3ccc(cc3)Br)C(=O)C1)C MS-7011 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)Cl)C(=O)C1)C MS-7012 CCCCOc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)OC(=C2C(=O)OCC)N MS-7013 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cccc(c3)F)C(=O)C1)C MS-7015 Cc1c2c([nH]n1)OC(=C(C2c3cccs3)C#N)N MS-7016 CCc1ccc(cc1)OCC(=O)NN MS-7017 CN(C)c1cccc(c1)OCC(=O)NNC(=S)Nc2ccccc2 MS-7018 CN(C)c1cccc(c1)OCC(=O)NN MS-7019 CC1(CC(=CC(=O)C1)Nc2ccc(cc2NC(=S)Nc3ccccc3)Cl)C MS-7020 COC(=O)c1ccc(cc1)C=C2C(=O)c3ccccc3C2=O MS-7021 c1cc(cc(c1)NC=C(C#N)C#N)C#N MS-7022 CCc1ccc(cc1)OCC(=O)N/N=C/2\c3ccccc3NC2=O MS-7023 CC(C(=O)N/N=C/1\c2ccccc2NC1=O)Oc3ccc(cc3Cl)Cl MS-7024 CCc1ccc(cc1)OCC(=O)N/N=C\2/c3ccccc3N(C2=O)C MS-7025 COC(=O)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F MS-7026 CCc1ccc(cc1)OCC(=O)NNC(=S)NC2CCCCC2 MS-7027 CC(C)(C)C(=O)/C(=C\c1cccc(c1Cl)Cl)/C#N MS-7028 CC(C(=O)N/N=C\1/c2ccccc2N(C1=O)C)Oc3ccc(cc3Cl)Cl MS-7029 CN1c2ccccc2/C(=N/NC(=O)c3ccncc3)/C1=O MS-7030 CCN1C(=O)/C(=C/c2ccc(cc2)C(=O)O)/SC1=S MS-7031 CCc1ccc(cc1)OCC(=O)NNC(=S)Nc2ccccc2 MS-7032 CC(=O)c1ccc(cc1)NC2=C(C(=O)c3c2cccc3)c4ccccc4 MS-7033 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-])Br MS-7034 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)NCc3ccncc3 MS-7035 COc1cc2c(cc1OC)C(=NCC2)c3cccnc3Oc4ccc(cc4)Cl MS-7036 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc4ccccc4c3 MS-7037 Cn1c(c(c(=O)n1c2ccccc2)Cl)COc3cccc(c3)Cl MS-7038 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2cccc3c2nccc3)/C#N MS-7039 CC1(Cc2c(cc(n2c3ccc(nc3)OC)c4ccc(cc4)Br)C(=O)C1)C MS-7040 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3OC)C=O MS-7041 CN(c1ccc(cn1)C(F)(F)F)NC2=CC(=O)CCC2 MS-7042 CN1c2ccccc2/C(=N/NC(=S)NCC=C)/C1=O MS-7043 COc1ccc(cc1Br)C=C(C#N)C#N MS-7044 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4cc(c(c(c4)Br)O)Br MS-7045 CC(=O)Nc1cccc(c1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F MS-7046 c1cc(c(c(c1)Cl)Cl)C=C(C#N)C#N MS-7047 CC(=O)Nc1ccc(cc1)/C=N/C(=C(/C#N)\N)/C#N MS-7048 c1c(cc(c(c1I)O)I)/C=N/C(=C(/C#N)\N)/C#N MS-7049 c1ccc2cc(ccc2c1)/C=N/C(=C(/C#N)\N)/C#N MS-7050 c1ccc2c(c1)cccc2Nc3[nH+]c(cs3)c4ccc(cc4)F.[Br-] MS-7051 CCOC(=O)c1c([nH+]c(s1)Nc2cccc3c2cccc3)C.[Cl-] MS-7052 CCOC(=O)/C(=C\Nc1ccc(cc1C)C)/C#N MS-7053 CCOC(=O)/C(=C/Nc1ccc(cc1)OC(F)(F)F)/C#N MS-7054 CCOC(=O)/C(=C\Nc1cccc(c1)OC(C(F)F)(F)F)/C#N MS-7055 CC(C)(C)c1ccc(cc1)C(=O)NCCc2ccc(c(c2)OC)OC MS-7056 CCOC(=O)/C(=C/Nc1c(cccc1Cl)C)/C#N MS-7057 c1ccc2c(c1)C(=O)C(C2=O)C(=O)/C=C/c3cccs3 MS-7058 Cc1ccc(cc1)S(=O)(=O)N2C3(c4ccccc4C(=O)C3C(=N2)C(C)(C)C)O MS-7059 CC(C)(C)C(=O)/C(=C/Nc1ccc(cc1C(F)(F)F)F)/C#N MS-7060 c1ccc(cc1)NC(=S)NNC(=O)COc2ccc3ccccc3c2Br MS-7061 COc1ccc(cc1Br)C=C2C(=O)c3ccccc3C2=O MS-7062 COc1ccccc1N2CCN(CC2)Cc3ccc(cc3)F MS-7063 c1ccc(cc1)NC(=S)NNC(=O)CC#N MS-7064 CC(C(=O)NN)Sc1ccc(cc1)Cl MS-7065 CCOC(=O)C1=C(OC2=C(C1c3cccnc3)C(=O)CC(C2)C)N MS-7066 c1ccc(cc1)C(=O)N/N=C\2/CC(=O)c3c2cccc3 MS-7067 c1ccc(cc1)NC(=S)N/N=C/2\CC(=O)c3c2cccc3 MS-7068 COc1ccc(cc1Br)/C=C\2/C(=O)NC(=O)S2 MS-7069 CCN1C(=O)/C(=C/c2ccc(c(c2)Br)OC)/SC1=S MS-7070 CCOC(=O)/C(=C/Nc1cccc(c1)F)/C#N MS-7071 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)C(=O)OC)/C#N MS-7072 c1ccc2c(c1)C(=O)C(=Cc3cc(ccc3O)O)C2=O MS-7073 c1ccc(cc1)C(=O)/C(=C\c2ccc(cc2)[N+](=O)[O-])/C#N MS-7074 CC(C)(C)c1cc(=O)n([nH]1)C(=S)N MS-7075 COc1cc(cc(c1OC)OC)/C=C(/C#N)\C(=O)c2ccccc2 MS-7076 CC(C)(C)c1c2c(n(n1)C(=O)CCCCl)-c3ccccc3C2=O MS-7077 c1ccc(cc1)CCNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-7078 c1ccc2c(c1)C(=O)C(=Cc3c(cccc3Cl)F)C2=O MS-7079 c1ccc(cc1)C2CC3=C(C(Nc4ccccc4N3)c5cccc(c5)[N+](=O)[O-])C(=O)C2 MS-7080 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C(C(C(F)(F)F)(F)F)(F)F MS-7081 c1cc(oc1)C(=O)N2CCN(CC2)C(=S)NC3CCCCC3 MS-7082 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4cccc(c4O)O MS-7083 CC(C)(C)C(=O)/C(=C/c1cccc(c1)[N+](=O)[O-])/C#N MS-7085 CC1(C/C(=N\NC(=O)c2ccncc2)/CC(=O)C1)C MS-7086 c1cc(sc1)C(=O)NC2CCSC2=O MS-7087 c1ccc2c(c1)c(c[nH]2)CCNC(=O)C3CC3 MS-7088 c1ccc(c(c1)C(=O)N)NC(=O)/C=C/c2cc(ccc2Cl)[N+](=O)[O-] MS-7089 CC(=O)C/C(=N\NC(=S)N)/c1ccccc1 MS-7090 CC(C(=O)NNC1=CC(=O)CCC1)Oc2ccc(cc2Cl)Cl MS-7091 CC(=O)c1ccc(cc1)NC(=O)C2CC2 MS-7092 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)C(F)(F)F MS-7093 c1ccc2c(c1)c(c[nH]2)CCNC(=O)/C=C/c3ccc(cc3)Br MS-7094 c1ccc2c(c1)cccc2CC(=O)NCc3ccncc3 MS-7095 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCCc2c[nH]c3c2cccc3 MS-7096 c1cc(ccc1NC(=O)C(C(C(F)(F)F)(F)F)(F)F)F MS-7097 c1cc(c(cc1C(F)(F)F)NC(=O)C(C(C(F)(F)F)(F)F)(F)F)F MS-7098 CCOC(=O)COc1ccc2cc(ccc2c1)Br MS-7099 c1ccc2c(c1)ccc(c2Br)OCC#N MS-7100 c1ccc2c(c1)ccc(c2Br)OC/C(=N/O)/N MS-7101 c1ccc2c(c1)C(=O)C(=Cc3cccc(c3)C(F)(F)F)C2=O MS-7102 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=S)N MS-7103 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)C3CC3 MS-7104 CN(c1ccc(cc1)O)C(=O)c2cccs2 MS-7105 COc1ccc(cc1)OC/C(=N/O)/N MS-7106 c1ccc2c(c1)cccc2OCC#N MS-7107 c1ccc2cc(ccc2c1)OCC#N MS-7108 c1ccc2c(c1)cccc2OC/C(=N\O)/N MS-7109 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)c3ccco3 MS-7110 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4c(cccc4Cl)Cl MS-7111 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)c3cccs3 MS-7112 c1ccc(cc1)NC(=O)N2CCN(CC2)C(=O)c3ccco3 MS-7113 c1ccc2cc(ccc2c1)OC/C(=N/O)/N MS-7114 CCOC(=O)/C(=C\Nc1cc(nc2c1cccc2)C)/C#N MS-7115 c1cc(ccc1S(=O)(=O)CC(=O)NN)Cl MS-7116 COc1ccc(cc1)N2C(=O)CCSC23c4ccccc4NC3=O MS-7117 c1cc(ccc1S(=O)(=O)C[N+](=O)[O-])Br MS-7118 Cn1c(c(c(=O)n1c2ccccc2)Br)Cn3cnc(c3C#N)C#N MS-7119 COc1cc(c(cc1OC)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC(=O)OC MS-7120 CC1(CC2=C(C(Nc3ccccc3N2)c4cc(ccc4Sc5ccccn5)[N+](=O)[O-])C(=O)C1)C MS-7121 c1ccc2c(c1)nc(s2)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl MS-7122 c1cc(c(nc1)Cl)C(=O)Nc2ccc(cc2)SC(F)(F)F MS-7123 COc1ccc(cc1)/C=C/C=C(\C#N)/S(=O)(=O)c2ccccc2 MS-7124 CC1(OC(=O)C(=CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)C(=O)O1)C MS-7125 Cc1cc(ccc1C(C)C)n2c(nn(c2=S)C)C(F)(F)F MS-7126 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)n3c(cc4c3CC(CC4=O)(C)C)c5ccc(cc5)Br MS-7127 C=C1Cn2c(=O)c3c(ccs3)nc2S1 MS-7128 CCOC(=O)CC1=Nn2c(nnc2SC1)c3ccccc3 MS-7129 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C\2/c3ccccc3NC2=O MS-7130 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=C(\C#N)/C(=O)c2ccccc2 MS-7131 c1ccc2c(c1)C(=O)C(=CNc3cccc(c3)C(=O)O)C2=O MS-7132 c1ccc2c(c1)C(=O)C(=CNc3ccccc3C(=O)O)C2=O MS-7133 Cc1ccc(c(c1)C(=O)O)NC=C2C(=O)c3ccccc3C2=O MS-7134 Cc1ccc(c(c1)C(=O)O)NC=C2C(=O)OC(OC2=O)(C)C MS-7135 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C=C2C(=O)c3ccccc3C2=O MS-7136 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=N/NC(=S)N MS-7137 c1cc(c(c(c1)Cl)/C=N/NC(=S)N)F MS-7138 Cc1ccc(cc1)Sc2c(cccn2)C(=O)NN(C)c3c(cc(cn3)C(F)(F)F)Cl MS-7139 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(c(c2)Cl)Cl)/C(=O)C MS-7140 CC(=C1C(=O)c2ccccc2C1=O)N3CCN(CC3)C(=O)c4ccco4 MS-7141 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2c(cc(cn2)C(F)(F)F)Cl)/[N+](=O)[O-] MS-7142 CC(=O)CS(=O)(=O)c1ccc(cc1)Cl MS-7143 COC(=O)c1c(c2cc(ccc2s1)[N+](=O)[O-])N MS-7144 CCCCCCCCCCCCCCCCCCNS(=O)(=O)c1ccc(cc1)C MS-7145 COc1cccc(c1Oc2c(cc(cn2)C(F)(F)F)Cl)/C=C(\C#N)/S(=O)(=O)c3ccccc3 MS-7146 COc1cccc(c1Oc2c(cc(cn2)C(F)(F)F)Cl)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl MS-7147 Cc1cc2c(n1c3ccc(cc3)NC(=O)C)CC(CC2=O)(C)C MS-7148 CC1(Cc2cccc(c2O1)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)C MS-7149 c1cc(cnc1)C(=O)Nc2ccc(cc2)C(F)(F)F MS-7150 c1ccc(cc1)NC(=S)NNC(=O)COc2ccc3cc(ccc3c2)Br MS-7151 CS(=O)(=O)c1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)OC(F)(F)F MS-7152 c1cc(ccc1/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl)Oc3ccc(cn3)C(F)(F)F MS-7153 c1cc(ccc1Sc2ccc(cc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-])Cl MS-7154 c1ccc(cc1)S(=O)(=O)/C(=C/c2cc(ccc2Sc3ccc(cc3)Cl)[N+](=O)[O-])/C#N MS-7155 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2cc(ccc2Sc3ccc(cc3)Cl)[N+](=O)[O-])/C#N MS-7156 c1cc(ccc1C(F)(F)F)Oc2ccc(cc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)OC(F)(F)F)[N+](=O)[O-] MS-7157 COc1ccc(c(c1)S(=O)(=O)NCCc2c[nH]c3c2cccc3)OC MS-7158 C/C(=N/O)/c1ccc(cc1)NC(=O)/C=C/C(=O)O MS-7159 c1ccc(c(c1)Nc2nc(cs2)c3cccc(c3)[N+](=O)[O-])Cl MS-7160 Cc1c(sc(n1)Nc2cc(ccc2OC)Cl)C(=O)C MS-7161 Cc1cc(ccc1Cl)c2csc(n2)Nc3cc(ccc3OC)Cl MS-7162 CCOc1ccc(cc1)NC=C2C(=O)NC(=O)NC2=O MS-7163 COc1ccc(c(c1)NC=C2C(=O)NC(=O)NC2=O)OC MS-7164 COc1ccc(cc1Nc2nc(cs2)c3ccc(cc3)F)Cl MS-7165 c1ccc(c(c1)C(=O)O)NC=C2C(=O)NC(=O)NC2=O MS-7166 Cc1ccc2c(c1)CCCN2S(=O)(=O)c3ccc(cc3)C(C)(C)C MS-7167 COc1ccc(cc1Nc2nc(cs2)c3ccc(cc3)Br)Cl MS-7168 c1ccc(cc1)NC(=S)NNC(=O)c2cccs2 MS-7169 c1ccc2c(c1)/C(=N/NC(=O)c3cccs3)/C(=O)N2 MS-7170 c1ccc(cc1)n2c(n[nH]c2=S)c3cccs3 MS-7171 c1ccc(cc1)NC(=O)NNC(=O)c2cccs2 MS-7172 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCc2c[nH]c3c2cccc3)C)C MS-7173 c1cc(sc1)C(=O)NNC(=O)Nc2ccc(cc2)Cl MS-7174 Cc1ccc2c(c1)CCCN2C(=S)Nc3ccccc3 MS-7175 COc1cccc(c1O)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4cccc(c4)C(F)(F)F MS-7176 Cc1ccc2c(c1)CCCN2C(=O)Nc3ccc(cc3)Cl MS-7177 Cc1cc(ccc1Cl)c2csc(n2)Nc3cccnc3 MS-7178 COc1ccc(cc1Nc2nc(cs2)c3ccc4ccccc4c3)Cl MS-7179 Cc1ccc2c(c1)CCCN2C(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-] MS-7180 Cc1ccc(c(c1)OCC(=O)NN)Cl MS-7181 Cc1ccc(c(c1)OCc2n[nH]c(=S)n2c3ccccc3)Cl MS-7182 Cc1cc(ccc1C(C)C)NC(=S)NNc2c(c(c(c(c2F)F)C)F)F MS-7183 c1cc(ccc1OCC(=O)NN)I MS-7184 c1ccc(cc1)n2c(n[nH]c2=S)COc3ccc4cc(ccc4c3)Br MS-7185 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)I MS-7186 Cc1ccc2c(c1)CCCN2C(=O)c3cccnc3 MS-7187 c1ccnc(c1)Sc2ccc(cc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Br)[N+](=O)[O-] MS-7188 Cc1cc(c2ccccc2n1)NC=C3C(=O)c4ccccc4C3=O MS-7189 CS(=O)(=O)c1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-7190 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F)/C#N MS-7191 c1cc(c(c(c1)Cl)Cl)OCC(=O)NN MS-7192 CC1Cc2c(c(nn2C)c3ccc(c(c3)OC)OC)C(=O)C1 MS-7193 CC1(CC(=CC(=O)C1)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C MS-7194 CC1(CC2=C(C(Nc3c(cccn3)N2)c4ccc5c(c4)OCO5)C(=O)C1)C MS-7195 CC1(CC2=C(C(Nc3c(cccn3)N2)c4c(cccc4Cl)F)C(=O)C1)C MS-7196 c1ccc(cc1)C2CC(=CC(=O)C2)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-7197 c1cc2cccnc2c(c1)N/C=C(\C#N)/c3[nH]nnn3 MS-7198 CC(=C1C(=O)c2ccccc2C1=O)NCCN3CCOCC3 MS-7199 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)C(=O)N MS-7200 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3cc(ccc3Cl)Cl MS-7201 CC(C)(C)C(=O)/C(=C/NCCc1c[nH]c2c1cccc2)/C#N MS-7202 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)CC#N MS-7203 CC(C)(C)c1c(c[nH]n1)C#N MS-7204 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3cccc(c3)OC(C(F)F)(F)F MS-7205 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)C(C(F)(F)F)(C(F)(F)F)O)C2=O MS-7206 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3cccc(c3)OC(F)(F)F MS-7207 c1ccc(cc1)COc2cccc(c2)NC=C3C(=O)c4ccccc4C3=O MS-7208 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)C(=O)N)C2=O MS-7209 c1ccc(cc1)N(C=C2C(=O)c3ccccc3C2=O)c4ccccc4 MS-7210 COc1cc(ccc1NC=C2C(=O)c3ccccc3C2=O)[N+](=O)[O-] MS-7211 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)N3CCN(CC3)C(=O)c4ccco4 MS-7212 c1ccc(cc1)COc2cccc(c2)NC(=O)C(=O)c3c[nH]c4c3cccc4 MS-7213 COc1cc(cc(c1O)OC)C=C2C(=O)c3ccccc3C2=O MS-7214 Cc1ccc2c(c1)CCCN2C(=S)Nc3ccc(cc3)Cl MS-7215 CC1(OC(=O)C(=CNc2ccc(cc2)C(=O)N)C(=O)O1)C MS-7216 c1ccc2c(c1)C(=O)C(=Cc3cc(ccc3O)Cl)C2=O MS-7217 COc1ccc(cc1OC)CCNC2=C/C(=[NH+]/CCc3ccc(c(c3)OC)OC)/c4c2cccc4.[Cl-] MS-7218 Cc1ccc(c(c1)N)NC2=CC(=O)CC(C2)(C)C MS-7219 CN(C)c1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccccc2 MS-7220 Cc1c(sc(n1)c2cccnc2)/C(=N\O)/C MS-7221 CCOc1ccc(cc1)Nc2[nH+]c(c(s2)C(=O)C)C.[Cl-] MS-7222 Cn1c(c(c(=O)n1c2ccccc2)Br)CSC(=[NH2+])N.[Br-] MS-7223 COc1ccc(cc1OC)CCNC(=O)C(=O)c2c[nH]c3c2cccc3 MS-7224 c1ccc2cc(ccc2c1)OCC(=O)N MS-7225 c1ccc(cc1)CCNc2nc(cs2)c3ccc(cc3)[N+](=O)[O-] MS-7226 COc1ccc(cc1OC)CCNC(=O)c2cccnc2Cl MS-7227 c1ccc2c(c1)C(=O)C(=CNCc3ccc(cc3)C(=O)O)C2=O MS-7228 c1ccc(cc1)n2c(n[nH]c2=S)CSc3nc4c(c5ccccc5[nH]4)nn3 MS-7229 c1ccc(cc1)S(=O)(=O)/C(=C/c2cccc(c2)OC(F)(F)F)/C#N MS-7230 c1ccc(cc1)C2/C(=N/Cc3ccc(cc3)C(=O)O)/c4ccccc4C2=O MS-7231 CNC(=O)c1ccccc1NC=C2C(=O)c3ccccc3C2=O MS-7232 Cc1cc(ccc1Cl)c2csc(n2)NCCc3ccccc3 MS-7233 CCCCNS(=O)(=O)c1ccccc1 MS-7234 c1ccc(cc1)NC(=O)NNC(=O)c2ccccc2N MS-7235 COc1ccc(cc1)c2csc(n2)Nc3cccc4c3cccc4 MS-7236 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)C(=O)O MS-7237 CCOC(=O)/C(=C/Nc1ccc2c(c1)OCO2)/C#N MS-7238 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3cccc(c3)Oc4ccccc4 MS-7239 c1ccc(cc1)Oc2cccc(c2)C(=O)NCCc3c[nH]c4c3cccc4 MS-7240 c1ccc(cc1)Oc2cccc(c2)C(=O)NCc3cccs3 MS-7241 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc4c(c3)OCO4 MS-7242 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCc3cccs3 MS-7243 c1ccc\2c(c1)C(=C/C2=[NH+]\Cc3cccs3)NCc4cccs4.[Cl-] MS-7244 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3cc(c(c(c3)I)I)I MS-7245 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccc4c(c3)OCO4 MS-7246 CC(=C1C(=O)c2ccccc2C1=O)N3CCN(CC3)c4ccc(cc4)F MS-7247 CCOC(=O)/C(=C/N1CCN(CC1)c2ccc(cc2)F)/C#N MS-7248 c1ccc2c(c1)/C(=N/c3ccc4c(c3)OCO4)/C(=O)N2 MS-7249 Cc1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccc3c(c2)OCO3 MS-7251 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2cccnc2)/C#N MS-7252 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)Br MS-7253 CCC(=O)Nc1cc(ccc1Cl)NC2=CC(=[OH+])CC(C2)C.[Cl-] MS-7254 CC(C)C(=O)NC(=S)Nc1cccc(c1)C(F)(F)F MS-7255 c1ccc(cc1)CNS(=O)(=O)c2ccccc2 MS-7256 CC(C(=O)Nc1ccc(cc1)C(=O)C)Cl MS-7257 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=S)Nc2ccccc2 MS-7258 Cc1ccc(cc1)S(=O)(=O)CC(=O)NN MS-7259 CC(=O)Nc1ccc(cc1)c2csc(n2)Nc3cccnc3 MS-7260 c1ccnc(c1)NC(=O)c2cccc(c2)[N+](=O)[O-] MS-7261 c1ccc(cc1)NC(=S)NNC(=O)C(=O)NNC(=S)Nc2ccccc2 MS-7262 CCOC(=O)c1c2c(sc1NC(=O)c3ccc(cc3)[N+](=O)[O-])CCCC2 MS-7263 CCOC(=O)c1c2c(sc1NC=C3C(=O)OC(OC3=O)(C)C)CCCC2 MS-7264 c1cc(ccc1c2csc(n2)NC(=S)N)[N+](=O)[O-] MS-7265 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3cccnc3Nc4cccc(c4)C(F)(F)F MS-7266 c1cc(cc(c1)F)C=C(C#N)C#N MS-7267 COC(=O)/C(=C\c1ccc(cc1)Br)/C#N MS-7269 Cc1cc(ccc1Cl)C2=NNC3=C(C2)C(=O)CC(C3)C MS-7270 CCOc1ccc2c(c1)sc(n2)NC=C3C(=O)OC(OC3=O)(C)C MS-7271 c1ccc2c(c1)C(=O)C(=CNc3ncc(s3)[N+](=O)[O-])C2=O MS-7273 CC1(OC(=O)C(=CNc2ncc(s2)[N+](=O)[O-])C(=O)O1)C MS-7274 CC1(Cc2cccc(c2O1)OCC(=O)N)C MS-7275 CC1(Cc2cccc(c2O1)OCC(=O)NN)C MS-7276 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)N MS-7277 Cn1c2c(c(n1)c3ccc(c(c3)OC)OC)C(=O)CC(C2)c4ccccc4 MS-7278 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)NC=C(C#N)C#N MS-7280 c1ccc(cc1)NC(=S)NNC(=O)CC(=O)NNC(=S)Nc2ccccc2 MS-7281 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccc(cc3N)Cl MS-7282 CCOC(=O)c1cc([nH]c1c2ccccc2)c3ccc(cc3)Br MS-7283 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2cccnc2 MS-7284 CC(C)(C)OC(=O)CCc1ccc(cc1)[N+](=O)[O-] MS-7285 CCOc1ccc(cc1)NC=C2C(=O)OC(OC2=O)(C)C MS-7286 c1ccc2c(c1)/C(=N/NC(=O)COc3ccc(cc3Cl)Cl)/C(=O)N2 MS-7287 c1ccc2c(c1)/C(=N/NC(=O)COc3ccccc3Cl)/C(=O)N2 MS-7288 c1ccnc(c1)Sc2ccc(cc2)NC(=O)c3cccnc3Cl MS-7289 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=O)Nc3ccccc3)C MS-7290 CN(C)c1ccc(cc1)/C=C\2/Cc3cc(c(cc3C2=O)OC)OC MS-7291 Cc1ccc2c(c1)CCCN2C(=O)c3ccc(cc3Cl)Cl MS-7292 c1ccc2cc(ccc2c1)S(=O)(=O)Nc3ccc(cc3)n4cnc(c4Cl)Cl MS-7293 CCOc1ccc(cc1)NC(=O)c2ccccc2CC(=O)O MS-7294 c1ccc(cc1)Oc2cccc(c2)/C=N/C(=C(/C#N)\N)/C#N MS-7295 c1ccc(c(c1)/C=N/c2ccccc2O)O MS-7296 c1ccc(cc1)n2c(n[nH]c2=S)Cc3n[nH]c(=S)n3c4ccccc4 MS-7297 CCOc1ccc2c(c1)sc(n2)N/C=C(\C#N)/C(=O)C(C)(C)C MS-7298 CC(=O)Nc1ccc(cc1)SCC#N MS-7299 CCOc1ccc2c(c1)sc(n2)NC(=O)c3c(onc3c4ccccc4Cl)C MS-7300 c1ccc(cc1)S(=O)(=O)/C(=C\N)/C#N MS-7301 CC1(C(NC(S1)c2cccnc2)C(=O)O)C MS-7302 CC1(Cc2c(sc(n2)NC(=O)c3ccc(cc3)Cl)C(=O)C1)C MS-7303 c1cc(ccc1S(=O)(=O)CC(=O)N)Cl MS-7304 Cc1cc(nc(n1)N)Sc2ccccn2 MS-7305 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2nc(cc(n2)C)C)/C#N MS-7306 Cc1c(c(ccc1OCC(=O)N)Cl)C MS-7307 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2nc(cc(n2)Cl)C)/C#N MS-7308 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)OCO3 MS-7309 c1cc(ccc1OCC(=O)N)F MS-7310 c1ccc2c(c1)cccc2OCC(=O)N MS-7311 CC(=O)Nc1ccc(cc1)OCC(=O)N MS-7312 c1ccc(cc1)C(=O)/C=C/c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl MS-7313 c1ccc(cc1)C(=O)/C=C/c2ccccc2Oc3c(cc(cn3)C(F)(F)F)Cl MS-7314 c1ccc(cc1)Oc2ccc(cc2)NS(=O)(=O)c3cccc4c3nccc4 MS-7315 COc1cccc(c1)C(=O)NNC(=S)Nc2ccccc2 MS-7316 COc1cccc(c1)c2n[nH]c(=S)n2c3ccccc3 MS-7317 Cc1cc(nc(n1)N)Oc2ccc(cc2)OC MS-7318 c1ccc2c(c1)C(=O)C(=CNc3cc(ccc3Cl)C(=O)O)C2=O MS-7319 CC1=NN(C(=O)C1C(CC(=O)c2ccc(cc2)Cl)C(=O)O)c3ccccc3 MS-7320 CC(=O)NCc1ccc(cc1)F MS-7321 Cc1cc(nc(n1)[NH3+])N2CCN(CC2)c3ccccc3.[Cl-] MS-7322 c1cc(cc(c1)Cl)CC(=O)NN MS-7323 CC(=O)Nc1ccc(cc1)c2csc(n2)Nc3ccc(cc3)C#N MS-7324 CC1CN(C(CN1C=C2C(=O)c3ccccc3C2=O)C)C=C4C(=O)c5ccccc5C4=O MS-7325 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)F MS-7326 CCOC(=O)/C(=C\NCc1ccc(cc1)F)/C#N MS-7327 Cc1c(c(c(c(c1C)C)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)F)C)C MS-7328 CC(C)(C)c1ccc(cc1)C(=O)CC(c2cn(c3c2cccc3)C)C(=O)O MS-7329 c1ccc2c(c1)/C(=N/NC(=O)Cc3cccc(c3)Cl)/C(=O)N2 MS-7330 c1ccc(cc1)n2c(n[nH]c2=S)Cc3cccc(c3)Cl MS-7332 COc1ccc(cc1OC)CNC(=O)/C=C/c2ccccc2 MS-7333 Cc1cc(nc(n1)NC=C2C(=O)c3ccccc3C2=O)Sc4ccccn4 MS-7334 CCN(CC)C(=S)Sc1cc(nc(n1)N)C MS-7335 c1ccc(cc1)/C=C/C(=O)Nc2cccc(c2)C(=O)N MS-7336 c1ccc2c(c1)c(=O)[nH]c(n2)SCc3ccc(cc3)[N+](=O)[O-] MS-7337 Cc1cc(nc(n1)N)N2CCN(CC2)c3ccc(cc3)F MS-7338 CCC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)I MS-7339 CCCCCCCCC/C=C/CC(CC(=O)Nc1ccc(cc1)C(C)C)C(=O)O MS-7340 Cc1ccc2c(c1)CCCN2C=C3C(=O)c4ccccc4C3=O MS-7341 COC(=O)c1ccc(cc1)OCC(=O)NN MS-7342 COC(=O)c1ccc(cc1)OCC(=O)NNC2=CC(=O)CCC2 MS-7343 CC1(Cc2c(sc(n2)NC=C3C(=O)c4ccccc4C3=O)C(=O)C1)C MS-7344 c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl MS-7345 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)N3CCOCC3)O MS-7346 COC(=O)c1ccc(cc1)OCC(=O)N/N=C\2/c3ccccc3NC2=O MS-7347 Cc1cc(ccc1N/C=C(\C#N)/C(=O)C(C)(C)C)O MS-7348 Cc1cc(ccc1NC2=C(C(=O)c3c2cccc3)c4ccccc4)O MS-7349 CCCCCCCCC/C=C/CC(CC(=O)Nc1ccc(cc1)Oc2ccccc2)C(=O)O MS-7350 CCCCCCCCC/C=C/CC(CC(=O)Nc1ccccc1C#N)C(=O)O MS-7351 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccccc3F MS-7352 CCOC(=O)C(=CNc1cccc2c1nccc2)C(=O)OCC MS-7353 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cc(ccc2Sc3ccccn3)[N+](=O)[O-])c4ccccc4 MS-7354 COC(=O)c1ccc(cc1)OCC(=O)NNC(=S)Nc2ccc(cc2)Cl MS-7355 c1ccc(cc1)C(=O)/C(=C/Nc2cccc3c2nccc3)/C#N MS-7356 c1cc(cc(c1)[N+](=O)[O-])N/C=C/C=[NH+]/c2cccc(c2)[N+](=O)[O-].[Cl-] MS-7357 c1ccc2cc(ccc2c1)C3=CC(=NCCN3)C(F)(F)F MS-7358 CC(C)(C)c1ccc(cc1)S(=O)(=O)CC(=O)NN MS-7359 c1cc(ccc1C(=O)O)OCc2n[nH]c(=S)n2c3ccc(cc3)Cl MS-7360 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc4c(c3)OCO4 MS-7361 CC1(CC(=O)C(=CNc2ccc(cc2)Cl)C(=O)C1)C MS-7362 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)N3CCCCC3)/C#N MS-7363 CN(C)c1ccc(cc1)C=C(C#N)C#N MS-7365 Cc1ccc(cc1N2CCN(CC2)C(=O)Nc3ccccc3)Cl MS-7366 Cc1ccc(cc1N2CCN(CC2)C(=S)Nc3ccccc3)Cl MS-7367 c1cc(ccc1NC(=S)Nc2ccc3c(c2)OCO3)Sc4c(cc(cn4)C(F)(F)F)Cl MS-7368 Cc1ccc(cc1N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl)Cl MS-7369 Cc1ccc(cc1N2CCN(CC2)C(=S)Nc3ccc(cc3)C(C)C)Cl MS-7370 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F MS-7371 CSc1ccc(cc1)/C=C(/C#N)\S(=O)(=O)c2ccccc2 MS-7372 CSc1ccc(cc1)/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl MS-7373 CS(=O)(=O)c1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccccc2 MS-7374 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl MS-7375 CCOc1ccc(cc1)/C=C(/C#N)\S(=O)(=O)c2ccccc2 MS-7376 Cc1cc2c(n1c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)CC(CC2=O)(C)C MS-7377 Cc1cc2c(n1c3ccc(cc3)C(=O)Nc4ccc(cc4F)F)CC(CC2=O)(C)C MS-7378 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)C2CC2C(=O)O MS-7379 CCC1(C(=C)SC(=N1)Nc2ccc(cc2)OC(F)(F)F)CC MS-7380 c1ccc2c(c1)C/C(=C/c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F)/C2=O MS-7381 CCN(/C=C(\C#N)/C(=O)C(C)(C)C)c1ccccc1 MS-7382 CN(C)c1ccc(cc1)/C=C(\C#N)/C(=O)c2ccccc2 MS-7383 CCOC(=O)C(=CNc1cc(ccc1OC)OC)C(=O)OCC MS-7384 c1ccc(cc1)n2c(n[nH]c2=S)CSc3c(cc(cn3)C(F)(F)F)Cl MS-7385 c1c(cc(cc1C(F)(F)F)NC(=O)C2CC2C(=O)O)C(F)(F)F MS-7386 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)c4ccccc4F MS-7387 COc1cc(c(cc1OC)S(=O)(=O)Nc2cc(ccc2F)C(F)(F)F)CC(=O)OC MS-7388 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)Oc4ccccc4 MS-7389 c1ccc(cc1)Oc2cccc(c2)/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Cl MS-7390 c1ccc(c(c1)C(=O)O)NC(=O)C2CC2C(=O)O MS-7391 CCOC(=O)C(=CNc1ccc(cc1)C(C(F)(F)F)(C(F)(F)F)O)C(=O)OCC MS-7392 Cc1cc2c(n1Cc3ccc(c(c3)OC)OC)CC(CC2=O)(C)C MS-7393 CC1(CC2=C(C(Nc3ccccc3N2)c4c(cccc4Cl)Cl)C(=O)C1)C MS-7394 CC(=O)Nc1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-7395 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-7396 c1ccnc(c1)Sc2ccc(cc2)N/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Cl MS-7397 CC(=C1C(=O)c2ccccc2C1=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-7398 c1c(cc(c2c1c(=O)c(co2)/C=N/C(=C(/C#N)\N)/C#N)Cl)Cl MS-7399 CS(=O)(=O)N1CCCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl MS-7400 c1cc(c(cc1Cl)[N+](=O)[O-])NC=C(C#N)C#N MS-7401 c1cc2c(cc1NC=C(C#N)C#N)OCO2 MS-7402 CC(C)(C)C(=O)/C(=C\c1coc2c(c1=O)cc(cc2Cl)Cl)/C#N MS-7403 c1ccc(cc1)c2c(nc3c(n2)cccn3)c4ccccc4 MS-7404 c1ccc(cc1)/C=C/C(=O)NC2=NCCS2 MS-7405 CN(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccccc3 MS-7406 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)N(C)C)/C#N MS-7407 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(cc4)OC(F)(F)F)C(=O)C1)C MS-7408 c1cc(cc(c1)Oc2ccc(cc2)[N+](=O)[O-])C(F)(F)F MS-7409 COC(=O)c1ccc(cc1)OCC(=O)NNC(=S)Nc2ccccc2 MS-7410 c1ccc(cc1)n2c(n[nH]c2=S)COc3ccc(cc3)C(=O)O MS-7411 COC(=O)c1ccc(cc1)OCC(=O)NNC(=S)Nc2ccc(cc2)OC(F)(F)F MS-7412 CN(C(=S)Nc1ccc(cc1)OC(F)(F)F)N MS-7414 c1cc(ccc1N=C=S)Sc2c(cc(cn2)C(F)(F)F)Cl MS-7415 COc1cc(c(cc1OC)S(=O)(=O)Nc2cccc(c2)C(F)(F)F)CC(=O)OC MS-7416 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2cccc(c2)Oc3ccccc3)/C#N MS-7417 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3ccc(cc3F)F)C MS-7418 CC(=O)c1cc2c(cc1NC(=O)CCl)OCO2 MS-7419 COc1ccc(cc1)Nc2nc(cs2)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl MS-7420 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cc(ccc2Sc3ccc(cc3)Cl)[N+](=O)[O-])c4ccccc4 MS-7421 c1cc(c(cc1C(F)(F)F)NC(=O)C2CC2C(=O)O)F MS-7422 CC(C)(C)S(=O)(=O)/C(=C\c1ccc(cc1)O)/C#N MS-7423 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3cccc(c3)Br)C MS-7424 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)CC34CCC(C3(C)C)CC4=O MS-7425 c1cc(ccc1NC(=O)c2ccc(nc2Cl)Cl)Sc3c(cc(cn3)C(F)(F)F)Cl MS-7426 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)/C=C/c4ccccc4 MS-7428 c1cc(c(nc1)Cl)C(=O)Nc2ccc(cc2)Sc3c(cc(cn3)C(F)(F)F)Cl MS-7429 COc1cc(c(cc1OC)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)OC MS-7430 CC1(OC(=O)C(=CNc2ccc(cc2)Sc3c(cc(cn3)C(F)(F)F)Cl)C(=O)O1)C MS-7431 c1cc(ccc1NC=C(C#N)C#N)Sc2c(cc(cn2)C(F)(F)F)Cl MS-7432 CC(C(=O)NNC(=S)Nc1ccc(cc1)OC(F)(F)F)Oc2ccc(cc2Cl)Cl MS-7433 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3cccc(c3)OCc4ccccc4 MS-7434 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-7435 CC(=O)/C(=C/Nc1ccc(cc1)Cl)/S(=O)(=O)c2ccc(cc2)Cl MS-7436 CC(=O)/C(=C/Nc1ccc(cc1)F)/S(=O)(=O)c2ccc(cc2)Cl MS-7437 COc1ccc(cc1)N2C(C(C2=O)OC)c3ccc4c(c3)OCO4 MS-7438 c1ccc2c(c1)cc([nH]2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-7439 CC(C(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)Cl MS-7440 CC(C(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl)Sc3ccc(cc3)Cl MS-7441 c1c(cnc(c1Cl)Cl)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-7442 CCOC(=O)CCNC(=O)NNC(=O)COc1ccc(cc1)F MS-7443 CCOC(=O)CCNC(=O)Nc1cc(ccc1OC)OC MS-7444 CC(=O)Nc1ccc(cc1)C2NC(C(S2)(C)C)C(=O)O MS-7445 c1ccc(cc1)c2cc(n[nH]2)C(F)(F)F MS-7446 c1ccc2cc(ccc2c1)c3cc(n[nH]3)C(F)(F)F MS-7447 Cc1cc(n(n1)C(=O)c2ccc(cc2)Cl)c3ccccc3 MS-7448 c1ccc(cc1)c2c(c(n[nH]2)C(F)(F)F)Br MS-7449 c1ccc2c(c1)cccc2Nc3[nH+]c(cs3)c4ccc(c(c4)O)O.[Cl-] MS-7450 c1cc(cc(c1)Nc2[nH+]c(cs2)c3ccc(c(c3)O)O)C(F)(F)F.[Cl-] MS-7451 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)NCCc3ccc(c(c3)OC)OC)C MS-7452 c1cc(ccc1/C=N/c2c([nH]c(=O)n(c2=N)c3ccc(cc3)Cl)C#N)F MS-7453 c1ccc(cc1)/C=C/C=N/C(=C(/C#N)\N)/C#N MS-7454 c1ccc(cc1)/C=C/C=N/c2c([nH]c(=O)n(c2=N)c3cccc(c3)C(F)(F)F)C#N MS-7456 c1ccc(cc1)/C=C/C=N/c2c([nH]c(=O)n(c2=N)c3ccc(cc3)OC(F)(F)F)C#N MS-7457 c1cc(cc(c1)C(F)(F)F)/C=N/C(=C(/C#N)\N)/C#N MS-7458 CCOC(=O)CCNC(=S)N1CCN(CC1)c2ccccc2F MS-7459 c1ccc(c(c1)N2CCN(CC2)C(=O)N3CCOCC3)F MS-7460 c1ccc2c(c1)CCN2C=C3C(=O)c4ccccc4C3=O MS-7462 CCOC(=O)CCNC(=S)NNC(=O)c1ccncc1 MS-7463 Cc1ccc(cc1)S(=O)(=O)N/N=C\2/c3ccccc3N(C2=O)C MS-7464 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)C(=O)c4ccco4 MS-7465 c1ccc2cc(ccc2c1)S(=O)(=O)Nc3cccc4c3nccc4 MS-7466 Cc1cc(ccc1OCC(=O)N/N=C/2\c3ccccc3N(C2=O)C)Cl MS-7467 CN1c2ccccc2/C(=N/c3ccc(cc3)CC#N)/C1=O MS-7468 c1ccc2c(c1)/C(=N/c3ccc(cc3)CC#N)/C(=O)N2 MS-7469 c1ccc2c(c1)/C(=N/c3ccc(cc3)F)/C(=O)N2 MS-7470 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)C3CC3C(=O)O MS-7471 CC1(CC2=C(C(Nc3ccc(cc3N2)C(=O)OC)c4ccc(c(c4)OC)OC)C(=O)C1)C MS-7473 c1cc(sc1)C(=O)N/N=C/2\c3cc(ccc3NC2=O)I MS-7474 c1cc(sc1)C(=O)N/N=C/2\c3cc(ccc3NC2=O)Cl MS-7475 CC(=O)/C(=C\Nc1ccc(nc1)OC)/C(=O)Nc2ccccc2 MS-7476 CC(=O)/C(=C\Nc1ccc(c(c1)OC)OC)/C(=O)Nc2ccccc2 MS-7477 CC(=O)/C(=C\N1CCc2c1cccc2)/C(=O)Nc3ccccc3 MS-7478 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)NC(=O)C MS-7479 CCc1ccc(cc1)OCc2n[nH]c(=S)n2C MS-7480 CCOC(=O)CCNC(=O)NNC(=O)COc1ccccc1Cl MS-7481 CCOC(=O)C(Cc1ccccc1)NC(=O)NNC(=O)COc2ccc(cc2C)Cl MS-7482 Cc1ccc(cc1)S(=O)(=O)Cc2ccccn2 MS-7483 c1ccc(cc1)n2c(n[nH]c2=S)c3ccccc3Cl MS-7484 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCc2ccncc2 MS-7485 CCOC(=O)CCNC(=O)Nc1ccc(nc1)OC MS-7486 c1cc(cc(c1)OC(C(F)F)(F)F)NC=O MS-7487 COc1cc(cc(c1OC)OC)C(=O)NNC2=CC(=O)CCC2 MS-7488 CN(C)c1ccc(cc1)/C=C\2/C(=NN(C2=O)c3ccccc3)c4ccccc4 MS-7489 CCOC(=O)CCNC(=O)N1CCN(CC1)c2ccccc2F MS-7490 c1ccc(cc1)C\2=NN(C(=O)/C2=C\c3c[nH]c4c3cccc4)c5ccccc5 MS-7491 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)N(C(=S)S2)CC=C MS-7492 COc1ccc(cc1Br)/C=C\2/C(=O)N(C(=S)S2)CC=C MS-7493 C=CCN1C(=O)/C(=C\c2c[nH]c3c2cccc3)/SC1=S MS-7494 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccccc3C(F)(F)F MS-7495 Cc1cc(no1)NS(=O)(=O)c2ccccc2C(F)(F)F MS-7496 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)N2CCN(CC2)c3ccccc3F MS-7497 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCc3c2cccc3 MS-7498 Cc1ccc2c(c1)CCCN2/C=C(/C(=O)C)\C(=O)Nc3ccccc3 MS-7499 Cc1ccsc1C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-7501 CCOC(=O)CNC(=O)NNC(=O)C(C)Oc1ccc(cc1Cl)Cl MS-7502 CC(C)(C)C\1=NN(C(=O)/C1=C\c2ccc(cc2)N(C)C)c3ccccc3 MS-7504 CC(C)Cc1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)OC MS-7505 CCOC(=O)CNC(=O)NNC(=O)COc1ccc(cc1C)Cl MS-7506 c1cscc1/C=N/NC(=S)N MS-7507 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccsc2)/C#N MS-7508 CC(=O)Nc1ccc(cc1)c2csc(n2)Nc3ccc(cc3)Oc4ccccc4 MS-7509 CC(C)(C)C\1=NN(C(=O)/C1=C\c2ccsc2)c3ccccc3 MS-7510 c1ccc(cc1)Oc2ccc(cc2)Nc3nc(cs3)c4ccc(cc4)Br MS-7511 CC(=O)Nc1ccc(cc1)/C=C(\C#N)/S(=O)(=O)C(C)(C)C MS-7512 CC(C)(C)S(=O)(=O)/C(=C\c1ccc(cc1)N(C)C)/C#N MS-7513 COc1ccc(cc1OC)/C=C/C(=O)c2ccsc2 MS-7514 c1cscc1/C=N/C(=C(/C#N)\N)/C#N MS-7515 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3ccsc3 MS-7516 c1cc(cc(c1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3ccsc3)C(F)(F)F MS-7517 c1cc(ccc1n2c(=N)c3c(c(=O)[nH]c(n3)c4ccsc4)[nH]c2=O)Cl MS-7518 CC(=O)Nc1ccc(cc1)c2csc(n2)Nc3ccc(cc3)OC MS-7519 CC(=O)Nc1ccc(cc1)c2csc(n2)Nc3cccc(c3)C(F)(F)F MS-7520 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)C3CC3C(=O)O)C(F)(F)F MS-7521 c1cc(nc(c1C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl MS-7522 c1ccc(cc1)C2CC2C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-7523 c1cc(c(c(c1)Cl)/C=N/C(=C(/C#N)\N)/C#N)F MS-7524 CC(C)(C)C(=O)/C(=C\Nc1cc(ccc1OC)OC)/C#N MS-7525 c1ccc(c(c1)C(=O)O)Sc2ccc(cc2)[N+](=O)[O-] MS-7526 c1cc(c(cc1F)F)NC(=O)/C=C/C(=O)O MS-7527 CC(=O)Nc1ccc(cc1)/C=C\2/C(=NN(C2=O)c3ccccc3)C(C)(C)C MS-7528 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cc(c(c(c2)Br)O)Br)c3ccccc3 MS-7529 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccc3F MS-7530 c1ccc(cc1)n2c(n[nH]c2=S)c3ccc(cc3)O MS-7531 CCOc1ccc(cc1)N/C=C(/C(=O)C)\C(=O)Nc2ccccc2 MS-7532 c1ccc2cc(ccc2c1)/C=C/C(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F MS-7533 CCCCCCCCCCOc1ccc(cc1)/C=N/C(=C(/C#N)\N)/C#N MS-7534 c1ccc(c(c1)[NH2+]c2nc(cs2)c3cccc(c3)Br)Cl.[Br-] MS-7535 CCOC(=O)C/C(=N/Nc1nc2ccccc2s1)/C(F)(F)F MS-7536 CC(C)Cc1ccc(cc1)/C=N/C(=C(/C#N)\N)/C#N MS-7537 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4ncccn4 MS-7538 c1cc(sc1)C(=O)N2CCN(CC2)c3ncccn3 MS-7539 COC(=O)c1c(ccs1)NC(=O)c2cccs2 MS-7540 c1cc(sc1)C(=O)NC2=NCCS2 MS-7541 c1cc(cc(c1)OC(F)(F)F)CNC(=O)c2cccs2 MS-7542 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)c4ncccn4 MS-7543 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ncccn3 MS-7544 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)C(=O)c3ccco3 MS-7545 CC/C(=N/NC(=S)N)/C1C(=NN(C1=O)c2ccccc2)C MS-7546 c1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccccc3F MS-7547 CCOC(=O)/C(=N\OC)/c1csc(n1)NC(=O)/C=C/c2ccccc2 MS-7548 Cc1ccc(cc1N2CCN(CC2)C(=O)/C=C/c3ccccc3)Cl MS-7549 c1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ccccc3 MS-7550 CC(C)Cc1ccc(cc1)/C=N/N=C(\[NH3+])/SCc2ccc(cc2)Br.[Br-] MS-7551 c1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3ncccn3 MS-7552 Cc1csc(c1NC(=S)NC(=O)c2ccccc2)C(=O)OC MS-7553 c1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)C(=O)c3ccco3 MS-7554 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)NC(=O)c3ccccc3 MS-7555 Cc1ccc(cc1N2CCN(CC2)C(=S)NC(=O)c3ccccc3)Cl MS-7556 c1ccc(cc1)C(=O)NC(=S)NCc2ccncc2 MS-7557 c1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)c3ccccc3F MS-7558 Cc1cc(nc(n1)NC(=S)NC(=O)c2ccccc2)C MS-7559 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)Nc2ccsc2C(=O)OC MS-7560 COC(=O)c1c(ccs1)NC(=S)N2CCN(CC2)c3ncccn3 MS-7561 COC(=O)c1c(ccs1)NC(=S)NNC(=O)c2cccs2 MS-7562 CC(=O)Nc1ccc(cc1)OCC(=O)NNC(=S)Nc2ccsc2C(=O)OC MS-7563 c1cc(cc(c1)OC(F)(F)F)CNC(=O)c2cccnc2Cl MS-7564 c1ccc2c(c1)CCN2C(=O)c3ccccc3N MS-7565 Cc1ccc(cc1N2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F)Cl MS-7566 c1ccc(cc1)/C=C/C(=O)N2CCN(CC2)C(=O)c3ccco3 MS-7567 c1ccc(cc1)/C=C/CSC(=[NH2+])N/N=C/c2cccc(c2)OC(F)(F)F.[Br-] MS-7568 c1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl MS-7569 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCN(CC2)c3ncccn3 MS-7570 c1cnc(nc1)N2CCN(CC2)C(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-] MS-7571 c1ccc(cc1)C(=O)NC(=S)NCc2cccc(c2)OC(F)(F)F MS-7572 Cc1cc(ccc1OCC(=O)NNC(=S)NC(=O)c2ccccc2)Cl MS-7573 CC(C(=O)NNC(=S)NC(=O)c1ccccc1)Oc2ccc(cc2Cl)Cl MS-7574 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)NCc3cccc(c3)OC(F)(F)F MS-7575 COc1ccc(cc1OC)CNC(=S)Nc2ccsc2C(=O)OC MS-7576 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)O MS-7577 CC(C)Cc1ccc(cc1)/C=N/NC(=[NH2+])SCc2ccc(cc2)OC(F)(F)F.[Br-] MS-7578 Cc1ccc(cc1N2CCN(CC2)C(=O)c3cccnc3Oc4ccccc4)Cl MS-7579 Cc1ccc(cc1N2CCN(CC2)C(=O)c3cccnc3Cl)Cl MS-7580 c1ccc(cc1)N2CCN(CC2)C(=O)c3cccnc3Oc4ccccc4 MS-7581 c1cc(ccc1C(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)OC(F)(F)F MS-7582 Cc1ccc(cc1N2CCN(CC2)C(=S)Nc3ccsc3C(=O)OC)Cl MS-7583 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)/C(=C/N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)/C#N MS-7584 c1ccc(cc1)C(=O)/C(=C\N2CCN(CC2)c3ccc(cn3)C(F)(F)F)/C#N MS-7585 Cc1cccc(c1C(=O)O)NC(=O)C2CC2C(=O)O MS-7586 c1cc(cc(c1)OC(C(F)F)(F)F)NC(=O)C2CC2C(=O)O MS-7587 Cc1ccsc1C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F MS-7588 c1cc(ccc1NC(=O)CCl)SC(F)(F)F MS-7589 CC(C)Cc1ccc(cc1)/C=N/NC(=S)N MS-7590 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCc4c3cccc4)C MS-7591 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCc4c3cccc4 MS-7592 c1ccc(cc1)Oc2ccc(cc2)NC(=O)C(=O)c3c[nH]c4c3cccc4 MS-7593 Cc1cc(nc(n1)C)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cccs3 MS-7594 CC1(CC2=C(C(Nc3ccccc3N2)c4cccc(c4)Oc5ccccc5)C(=O)C1)C MS-7595 COc1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2Cl)Cl MS-7596 Cc1cc(ccc1OCC(=O)NNC(=S)Nc2ccc(cc2)OC)Cl MS-7597 COc1ccc(cc1)NC(=S)NNC(=O)COc2ccccc2Cl MS-7598 COc1ccc(cc1)NC(=S)NNC(=O)COc2cccc3c2cccc3 MS-7599 Cc1ccc(c(c1)C)OCC(=O)NNC(=S)Nc2ccc(cc2)OC MS-7600 CC(C(=O)NNC(=S)Nc1ccc(cc1)OC)Oc2ccc(cc2Cl)Cl MS-7601 COc1ccc(cc1)NC(=S)NCc2cccnc2 MS-7602 CN1CCN(CC1)C(=S)Nc2ccc(cc2)OC MS-7603 COc1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccc3 MS-7604 COc1ccc(cc1)NC(=S)NCc2cccc(c2)OC(F)(F)F MS-7605 COc1ccc(cc1)NC(=S)NCc2ccc(c(c2)OC)OC MS-7606 COc1ccc(cc1)NC(=S)NCc2ccncc2 MS-7607 COc1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccc3F MS-7608 CCc1ccc(cc1)OCC(=O)NNC(=S)Nc2ccc(cc2)OC MS-7609 COc1ccc(cc1)NC(=S)NNC(=O)COc2cccc(c2Cl)Cl MS-7610 COc1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2)C(=O)OC MS-7611 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)Nc3ccc(cc3)OC MS-7612 COc1ccc(cc1)NC(=S)NCCc2ccc(c(c2)OC)OC MS-7613 CN(C)CCNC(=S)Nc1ccc(cc1)OC MS-7614 COc1ccc(cc1)NC(=S)NNC(=O)c2cc(c(c(c2)OC)OC)OC MS-7615 COc1ccc(cc1)NC(=S)NCCc2c[nH]c3c2cccc3 MS-7616 COc1ccc(cc1)NC(=S)Nc2cccc(c2)OC(C(F)F)(F)F MS-7617 COC(=O)c1c(ccs1)NC(=O)C(C(C(C(=O)O)(F)F)(F)F)(F)F MS-7618 c1cc(cc(c1)OC(C(F)F)(F)F)NC(=O)C(C(C(C(=O)O)(F)F)(F)F)(F)F MS-7619 COc1ccc(cc1)NC(=S)NNC(=O)c2ccccc2 MS-7620 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3)NC(=S)NCC=C MS-7621 CC(C)Cc1ccc(cc1)/C=N/NC(=[NH2+])SCc2ccc(c(c2)F)F.[Br-] MS-7622 c1cc(sc1)/C=N/NC(=[NH2+])SCc2ccc(c(c2)F)F.[Br-] MS-7623 Cc1cc(c2c(c1)occ(c2=O)/C=N/NC(=[NH2+])SC/C=C/c3ccccc3)C.[Br-] MS-7624 Cc1ccc(cc1)S(=O)(=O)/C(=C\c2ccc(c(c2)Br)OC)/C#N MS-7625 CC(C)(C)C1=NN(C(=O)C1)c2nc3ccccc3s2 MS-7626 Cc1ccc(cc1)Sc2c(cccn2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-7627 Cc1cc(no1)N/C=C/C=[NH+]/c2cc(on2)C.[Cl-] MS-7629 c1ccc(cc1)NC(=S)NNC(=O)CSc2c(cc(cn2)C(F)(F)F)Cl MS-7630 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F)C MS-7631 CCc1ccc(cc1)OCC(=O)NNC(=S)NC(=O)c2ccccc2 MS-7632 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3ccsc3C(=O)OC MS-7633 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-7634 Cc1ccc2c(c1)CCCN2C(=O)c3c(onc3c4c(cccc4Cl)F)C MS-7635 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCc3ccc(c(c3)OC)OC MS-7636 c1ccc2c(c1)[nH]c(=O)c(n2)/C=C/c3cccnc3 MS-7637 COc1cc(cc(c1OC)OC)C(=O)O/N=C(\c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F)/N MS-7638 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(\c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)/N MS-7639 Cc1cccc(c1)C(=O)O/N=C(/c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)\N MS-7640 Cn1c(c(c(=O)n1c2ccccc2)Br)Cn3c(c(nn3)c4ccc(cc4)OC)C#N MS-7641 c1cc(ccc1c2[nH]c(=O)on2)Oc3c(cc(cn3)C(F)(F)F)Cl MS-7642 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl MS-7644 c1ccc2c(c1)C(=O)NC(N2)c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl MS-7645 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4ccc(cc4)Oc5c(cc(cn5)C(F)(F)F)Cl)[nH]c2=O MS-7646 c1cc2c(cc1c3c(n(nn3)c4c(cc(cn4)C(F)(F)F)Cl)C#N)OCO2 MS-7647 c1cc(ccc1/C=N/NC(=O)N)Oc2c(cc(cn2)C(F)(F)F)Cl MS-7648 c1cc(ccc1/C=N/NC(=S)N)Oc2c(cc(cn2)C(F)(F)F)Cl MS-7649 c1cc(ccc1/C(=N\O)/N)Oc2c(cc(cn2)C(F)(F)F)Cl MS-7650 c1cc(ccc1c2nc(on2)C(F)(F)F)Oc3c(cc(cn3)C(F)(F)F)Cl MS-7651 CC(C)(C)C(=O)CC(=O)Nc1ccc(cc1F)F MS-7652 c1ccc(c(c1)C(=O)NCCCCNC(=O)c2ccccc2[N+](=O)[O-])[N+](=O)[O-] MS-7653 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)c3ncccn3 MS-7654 Cc1cc(c2c(c1)occ(c2=O)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Br)C MS-7655 Cc1c(c(nc(n1)NC=C2C(=O)c3ccccc3C2=O)C)Br MS-7656 CCCCOc1ccc(cc1)/C=N/c2c([nH]c(=O)n(c2=N)c3ccccc3)C#N MS-7657 CCCCOc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O MS-7658 Cc1ccc(c(c1)C)OCC(=O)NNC(=S)NC(=O)c2ccccc2 MS-7659 c1ccc(cc1)Oc2ccc(cc2)NC(=O)C3CC3C(=O)O MS-7660 CC(C)(C)C(=O)/C(=C\NCc1ccccc1)/C#N MS-7661 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc3c(c2)OCO3)/C#N MS-7662 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2cccc(c2)C(=O)C)/C#N MS-7663 CCN1C(=O)/C(=C/c2coc3cc(cc(c3c2=O)C)C)/SC1=S MS-7665 CCN1C(=O)/C(=C\c2ccc(cc2)NC(=O)C)/SC1=S MS-7666 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C MS-7667 CCCCCC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2nccc(n2)C MS-7668 COc1ccc(c(c1)NC(=O)Cc2ccccc2C(=O)O)OC MS-7669 CCOC(=O)c1c[nH]n(c1=N)c2nc3ccccc3s2 MS-7670 Cc1ccc2c(c1)CCCN2S(=O)(=O)c3cccs3 MS-7671 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)NC(=O)C MS-7672 CC1(CC(=O)C(=CNc2cc(ccc2OC)OC)C(=O)C1)C MS-7673 Cc1cc2c([nH]1)CC(CC2=O)(C)C MS-7674 c1cnc(nc1)NC(=O)c2ccc(cc2)C(F)(F)F MS-7675 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)C(F)(F)F MS-7676 CC(=O)c1cccc(c1)NC=C2C(=O)c3ccccc3C2=O MS-7677 CC(=O)c1cccc(c1)NC(=C2C(=O)c3ccccc3C2=O)C MS-7678 COc1ccc(cc1OC)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4cccc(c4)C(F)(F)F MS-7679 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3)C(F)(F)F MS-7680 Cc1c(c(nc(n1)NC(=O)c2cccs2)C)Br MS-7681 Cc1c(c(nc(n1)NC(=C2C(=O)c3ccccc3C2=O)C)C)Br MS-7682 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3OC)C=C4C(=O)c5ccccc5C4=O MS-7683 COc1ccc(cc1OC)CCNC(=O)c2ccc(cc2)C(F)(F)F MS-7684 Cc1c(c(nc(n1)N/C=C(\C(=O)C)/C(=O)Nc2ccccc2)C)Br MS-7685 Cc1cc(nc(n1)NC(=O)c2ccc(cc2)C(F)(F)F)C MS-7686 Cc1cc(nc(n1)NC(=O)c2cccs2)C MS-7687 c1ccc(cc1)/C=C/C(=O)Nc2ncccn2 MS-7688 CCOC(=O)C/C(=N/NC(=O)Cc1c[nH]c2c1cccc2)/C(F)(F)F MS-7689 Cc1ccc(cc1)S(=O)(=O)/C(=C\c2ccc(cc2)C#N)/C#N MS-7690 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3OC)/C=N/C(=C(/C#N)\N)/C#N MS-7691 c1cc(cnc1)Nc2nc(cs2)c3ccc(cc3)Br MS-7692 c1ccc(cc1)C(=O)/C(=C/c2ccc(c(c2)[N+](=O)[O-])Cl)/C#N MS-7693 c1ccc(cc1)C(=O)/C(=C/C=C/c2ccccc2[N+](=O)[O-])/C#N MS-7694 CCN1C(=O)/C(=C\c2cc(c(c(c2)OC)OC)OC)/SC1=S MS-7695 c1ccc(cc1)NC(=S)NCCN2CCOCC2 MS-7696 CC(C(=O)NNC(=S)Nc1ccccc1)Oc2ccc(cc2Cl)Cl MS-7697 COc1ccc(cc1)c2csc(n2)NC=C3C(=O)c4ccccc4C3=O MS-7698 CC1(OC(=O)C(=CNc2nc(cs2)c3ccc(cc3)OC)C(=O)O1)C MS-7699 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)N MS-7700 c1cc(cnc1)Nc2nc(cs2)c3ccc(c(c3)Cl)Cl MS-7701 C=CCNc1nc(cs1)c2ccc(c(c2)Cl)Cl MS-7702 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=S)Nc2ccc(cc2)Cl MS-7703 c1ccc(cc1)C(=O)NC(=S)NNC(=O)COc2ccc(cc2Cl)Cl MS-7704 c1ccc(cc1)C(=O)NC(=S)NNC(=O)COc2ccc(cc2)F MS-7705 c1ccc(cc1)C(=O)NC(=S)NNC(=O)c2ccncc2 MS-7706 COc1ccc(cc1Br)/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Br MS-7707 CSc1ccc(cc1)/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Br MS-7708 Cc1c(c(n(n1)c2ccccc2)C)/C=N/NC(=S)N MS-7709 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC=C4C(=O)c5ccccc5C4=O MS-7710 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)C(C)C MS-7711 COC(=O)c1c(ccs1)NC(=O)Cc2ccccc2C(=O)O MS-7712 CCCCOc1ccc(cc1)/C=C(/C#N)\C(=O)OC MS-7713 COc1ccc(cn1)NC(=S)NC(=O)c2ccccc2 MS-7714 c1ccc(cc1)NC(=S)Nc2nccs2 MS-7715 c1ccnc(c1)/C=N/NC(=S)N MS-7716 CCOC(=O)C1=C(OC2=C(C1c3ccccc3)C(=O)CC(C2)(C)C)N MS-7717 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3cccc(c3)Oc4ccccc4 MS-7718 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)/C=C/c4ccccc4 MS-7719 c1ccc2c(c1)C/C(=C/c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)/C2=O MS-7720 CC(C(=O)Nc1cc2c(cc1C(=O)C)OCO2)Cl MS-7721 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4c(onc4c5c(cccc5Cl)Cl)C MS-7722 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4c(onc4c5ccccc5Cl)C MS-7723 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)C(C)Cl MS-7724 CC(=O)Nc1ccc(cc1)/C=C\2/C(=O)NC(=S)N2 MS-7725 Cc1cc(nc(n1)N/C=C\2/C(=O)NC(=S)N2)C MS-7726 Cc1cc(c2c(c1)occ(c2=O)/C=C\3/C(=O)NC(=S)N3)C MS-7727 CC(=O)Nc1ccc(cc1)OCC(=O)NNC(=S)Nc2ccc(cc2)OC MS-7728 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)C(F)(F)F)C2=O MS-7729 CC(=O)/C(=C/Nc1cccc(c1)C(F)(F)F)/C(=O)Nc2ccccc2 MS-7730 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2coc3cc(cc(c3c2=O)C)C MS-7731 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4ccc(cc4)[N+](=O)[O-] MS-7732 Cc1ccc2c(c1)nc(s2)c3ccc(cc3)NC(=O)c4cc(cc(c4)[N+](=O)[O-])[N+](=O)[O-] MS-7733 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)cn[nH]3 MS-7734 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc4c(c3)cn[nH]4 MS-7735 COc1cc2c(cc1OC)C(=O)/C(=C\c3ccc(cc3)OC(F)F)/C2 MS-7736 COc1ccc(cc1)/C=C/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-7737 Cc1cc(cc(c1)OC(C)C(=O)NN)C MS-7738 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4cc(cc(c4)[N+](=O)[O-])[N+](=O)[O-] MS-7739 CCS/C(=N\N=C\c1c(cccc1Cl)F)/[NH3+].[Cl-] MS-7740 CSc1ccc(cc1)/C=C\2/Cc3ccccc3C2=O MS-7741 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl MS-7742 Cc1ccc(c(c1)OCC(=O)NNC(=S)Nc2ccccc2)Cl MS-7743 CC(=O)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F MS-7744 CCOC(=O)c1cccc(c1)NC=C2C(=O)CCCC2=O MS-7746 CCOC(=O)c1cccc(c1)NC=C2C(=O)OC(OC2=O)(C)C MS-7747 CC(=O)/C(=C/Nc1ccsc1C(=O)OC)/C(=O)Nc2ccccc2 MS-7749 CC(=O)/C(=C/Nc1ccc(cc1F)F)/C(=O)Nc2ccccc2 MS-7750 CN1c2ccccc2/C(=N/NC(=O)c3cc(c(c(c3)OC)OC)OC)/C1=O MS-7751 CC(=O)/C(=C/Nc1ccc(cc1)C(F)(F)F)/C(=O)Nc2ccccc2 MS-7752 CC(=O)/C(=C/Nc1ccc(c(c1)C(F)(F)F)F)/C(=O)Nc2ccccc2 MS-7753 CC(=O)/C(=C/Nc1ccc(cc1)F)/C(=O)Nc2ccccc2 MS-7754 CC(C)(C)C(=O)/C(=C(\Nc1ccc(c(c1)Cl)Cl)/O)/C#N MS-7755 c1cc(cc(c1)NC(=C(C#N)C#N)C#N)C(F)(F)F MS-7756 CC(C)N(CCN(C(C)C)S(=O)(=O)c1ccc(cc1)OC(F)(F)F)S(=O)(=O)c2ccc(cc2)OC(F)(F)F MS-7757 c1ccc(cc1)C(=O)/C(=C\N2CCN(CC2)c3ccccn3)/C#N MS-7758 c1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)c3ccccn3 MS-7759 Cc1cc(cc(c1)OC(C)C(=O)N/N=C\2/c3cc(ccc3NC2=O)Br)C MS-7760 CCOC(=O)COc1ccc2ccc(=O)oc2c1 MS-7761 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccn3 MS-7762 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4ccccn4 MS-7763 c1ccnc(c1)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl MS-7764 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCN(CC3)c4ccccn4)C MS-7765 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)[N+](=O)[O-] MS-7766 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)c3ccccn3 MS-7767 CN1c2ccccc2/C(=N/NC(=O)c3cccs3)/C1=O MS-7768 CC(=O)/C(=C\Nc1ccc(cc1)OC)/C(=O)Nc2ccccc2 MS-7769 CCN1C(=O)/C(=C\Nc2ccc(cc2)C(F)(F)F)/SC1=S MS-7770 CCN1C(=O)/C(=C\Nc2ccc(c(c2)C(F)(F)F)F)/SC1=S MS-7771 CCN1C(=O)/C(=C\Nc2ccc(cc2)F)/SC1=S MS-7772 CCN1C(=O)/C(=C\Nc2ccc(nc2)OC)/SC1=S MS-7773 CCN1C(=O)/C(=C\Nc2cccc(c2)Cl)/SC1=S MS-7774 Cc1cc(no1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-7775 COc1ccc(cc1OC)CCNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-7776 c1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)F MS-7777 c1cc(oc1)C(=O)N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl MS-7778 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl MS-7779 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)Cl MS-7780 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4cc(c(cc4Cl)Cl)Cl MS-7781 c1ccc(c(c1)C(=O)N)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-7782 c1ccnc(c1)N2CCN(CC2)C(=O)c3cccs3 MS-7783 CC(C)C1=NN(C(=O)C1)c2nc3ccccc3s2 MS-7784 CC\1=NN(C(=O)/C1=C\Nc2ccc(cc2)Oc3ccccc3)c4ccccc4 MS-7785 CC\1=NN(C(=O)/C1=C/Nc2ccsc2C(=O)OC)c3ccccc3 MS-7786 CC\1=NN(C(=O)/C1=C/Nc2ccccc2)c3ccccc3 MS-7787 CC1(C(NC(S1)c2ccccc2)C(=O)O)C MS-7788 Cc1cc(cc(c1)OC(C)C(=O)NC(=O)Nc2ccccc2)C MS-7789 Cc1ccc(cc1N2CCN(CC2)C(=O)N3CCOCC3)Cl MS-7790 c1ccc(c(c1)CC(=O)N/N=C/2\c3cc(ccc3NC2=O)I)Cl MS-7791 c1ccc(cc1)NC(=O)NNC(=O)Cc2ccccc2Cl MS-7792 c1ccc(c(c1)CC(=O)N/N=C/2\c3ccccc3NC2=O)Cl MS-7793 c1ccc(c(c1)CC(=O)NNC(=O)Nc2cccc(c2)C(F)(F)F)Cl MS-7794 Cc1cc(c2c(c1)c3c(n2C)nc(nn3)SC)C MS-7795 Cc1cc2c(n1c3ccc4c(c3)OCO4)CC(CC2=O)(C)C MS-7796 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cccc(c3)C(F)(F)F MS-7797 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCN(CC3)c4cccc(c4)C(F)(F)F)C MS-7798 c1ccc(cc1)NC(=O)N2CCN(CC2)c3cccc(c3)C(F)(F)F MS-7799 c1ccc(cc1)C(=O)/C(=C/N2CCN(CC2)c3cccc(c3)C(F)(F)F)/C#N MS-7800 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4cccc(c4)C(F)(F)F MS-7801 c1cc(cc(c1)N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)C(F)(F)F MS-7802 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3c(cccc3F)F MS-7803 Cc1ccc(cc1N2CCN(CC2)C(=O)c3c(cccc3F)F)Cl MS-7804 c1ccc(c(c1)N2CCN(CC2)C(=O)c3c(cccc3F)F)F MS-7805 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3c(cccc3F)F MS-7806 Cc1cc(nc(n1)NC(=O)c2c(cccc2F)F)C MS-7807 c1cc(c(c(c1)F)C(=O)N2CCN(CC2)C(=O)c3ccco3)F MS-7808 COC(=O)c1ccccc1NC(=O)c2c(cccc2F)F MS-7809 COc1ccc(cc1OC)CCNC(=O)c2c(cccc2F)F MS-7810 CCOc1ccc2c(c1)sc(n2)NC(=O)c3c(cccc3F)F MS-7811 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4c(cccc4F)F MS-7812 c1ccc2c(c1)c(c[nH]2)CCNC(=O)Nc3ccc(cc3)NC(=O)NCCc4c[nH]c5c4cccc5 MS-7814 CN(C)CCNC(=O)Nc1ccc(cc1)NC(=O)NCCN(C)C MS-7815 c1ccc(cc1)CCNC(=O)Nc2ccc(cc2)NC(=O)NCCc3ccccc3 MS-7816 c1ccc(c(c1)C(=O)/C(=C/Nc2ccc3c(c2)OCO3)/C#N)Cl MS-7817 c1ccc(c(c1)C(=O)/C(=C/Nc2ccc(cc2)C(F)(F)F)/C#N)Cl MS-7818 Cc1cc(no1)N/C=C(\C#N)/C(=O)c2ccccc2Cl MS-7819 c1ccc(c(c1)C(=O)/C(=C/Nc2ccc(c(c2)C(F)(F)F)F)/C#N)Cl MS-7820 c1ccc(c(c1)C(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl MS-7821 CC1(OC(=O)C(=CNCc2ccc(cc2)C(=O)O)C(=O)O1)C MS-7822 c1cc(ccc1N)n2cncn2 MS-7823 Cc1cc(c2c(c1)c3c([nH]2)nc(nn3)S)C MS-7824 c1cc(ccc1C(C(F)(F)F)(C(F)(F)F)O)NC=C(C#N)C#N MS-7825 Cc1ccc(cc1)c2csc(n2)NCC=C MS-7826 COc1ccc(cc1OC)CNC(=O)c2ccccc2N MS-7827 Cc1cc(ccc1Cl)c2csc([nH+]2)NCC=C.[Cl-] MS-7828 C=CCNc1nc(cs1)c2ccc(cc2)[N+](=O)[O-] MS-7829 c1ccc(cc1)NC(=S)NNC(=O)Cc2ccccc2Cl MS-7830 c1ccc(cc1)n2c(n[nH]c2=S)Cc3ccccc3Cl MS-7831 c1cc(cnc1)CNC(=O)C2CC2C(=O)O MS-7832 Cn1cc(c2c1cccc2)C(CC(=O)c3ccccc3)C(=O)O MS-7833 Cc1ccc(cc1)C(=O)CC(c2cn(c3c2cccc3)C)C(=O)O MS-7834 CC(=O)Nc1ccc(cc1)c2csc([nH+]2)NCC=C.[Br-] MS-7835 CC(=O)Nc1ccc(cc1)c2csc(n2)NC=C3C(=O)OC(OC3=O)(C)C MS-7836 CCOC(=O)Cc1csc(n1)Nc2ccccc2 MS-7837 CC1(C(NC(S1)c2cccc3c2cccc3)C(=O)O)C MS-7838 c1cc(cnc1)CNC(=O)Nc2ccc(cc2)NC(=O)NCc3cccnc3 MS-7840 Cc1cc(ccc1OCC(=O)NNC(=S)Nc2ccc(cc2)[N+](=O)[O-])Cl MS-7841 c1cc(sc1)C(=O)NNC(=S)Nc2ccc(cc2)[N+](=O)[O-] MS-7842 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)Nc2ccc(cc2)[N+](=O)[O-] MS-7843 CC(C(=O)NNC(=S)Nc1ccc(cc1)[N+](=O)[O-])Oc2ccc(cc2Cl)Cl MS-7844 c1ccc(c(c1)OCC(=O)NNC(=S)Nc2ccc(cc2)[N+](=O)[O-])Cl MS-7845 c1ccc2c(c1)c(c[nH]2)CCNC(=S)Nc3ccc(cc3)[N+](=O)[O-] MS-7846 c1cc(ccc1NC(=S)NCCN2CCOCC2)[N+](=O)[O-] MS-7847 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)Nc3ccc(cc3)[N+](=O)[O-] MS-7848 c1cc(cnc1)CNC(=S)Nc2ccc(cc2)[N+](=O)[O-] MS-7849 C=CCNC(=S)NNC(=S)Nc1ccc(cc1)[N+](=O)[O-] MS-7850 CCc1ccc(cc1)OCC(=O)NNC(=S)Nc2ccc(cc2)[N+](=O)[O-] MS-7851 c1ccc(c(c1)CC(=O)NNC(=S)Nc2ccc(cc2)[N+](=O)[O-])Cl MS-7852 Cc1ccc(c(c1)C)OCC(=O)NNC(=S)Nc2ccc(cc2)[N+](=O)[O-] MS-7853 c1cc(ccc1NC(=S)NNC(=O)c2ccncc2)[N+](=O)[O-] MS-7854 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3cc(c(cc3CC(=O)OC)OC)OC MS-7855 COc1ccccc1N2CCN(CC2)C(=O)c3cccs3 MS-7856 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(cc3)[N+](=O)[O-] MS-7857 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCN(CC3)c4ccccc4OC)C MS-7858 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl MS-7859 COc1ccccc1N2CCN(CC2)C(=O)c3ccc(cc3)[N+](=O)[O-] MS-7860 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)c4ccccc4OC MS-7861 CCCCCCCCC/C=C\CC(CC(=O)Nc1ccc(cc1)Br)C(=O)O MS-7862 Cc1c(sc(n1)Nc2cccc3c2cccc3)C(=O)C MS-7863 Cc1c(c(no1)c2ccccc2)C(=O)NCc3ccc(c(c3)OC)OC MS-7864 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)Nc3ccc(cc3)C(C)C MS-7865 CC(C)c1ccc(cc1)N/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl MS-7866 c1csc2c1[nH]c(=S)n(c2=O)N MS-7867 c1ccc(cc1)C(=O)NC(=S)NCCCCCNC(=S)NC(=O)c2ccccc2 MS-7868 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc(c(c2)C(F)(F)F)F)CC(=O)OC MS-7869 Cc1ccc2c(c1)CCCN2S(=O)(=O)c3cc(c(cc3CC(=O)OC)OC)OC MS-7870 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccccc2C(=O)OC)CC(=O)OC MS-7871 COc1cc(c(cc1OC)S(=O)(=O)N2CCN(CC2)c3ccccc3)CC(=O)OC MS-7872 COc1cc(c(cc1OC)S(=O)(=O)NCCc2c[nH]c3c2cccc3)CC(=O)OC MS-7873 COc1cc(c(cc1OC)S(=O)(=O)N2CCN(CC2)c3ccccc3F)CC(=O)OC MS-7874 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=S)Nc4ccc(cc4)OC(F)(F)F MS-7875 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)OC(F)(F)F MS-7876 c1ccc(cc1)N2CCN(CC2)C(=S)Nc3ccc(cc3)OC(F)(F)F MS-7877 COc1ccc(cc1OC)CNC(=S)Nc2ccc(cc2)OC(F)(F)F MS-7878 c1ccc(c(c1)N2CCN(CC2)C(=S)Nc3ccc(cc3)OC(F)(F)F)F MS-7879 c1cc(sc1)C(=O)NNC(=S)Nc2ccc(cc2)OC(F)(F)F MS-7880 c1cc(sc1)C(=O)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-7881 COc1ccc(cc1OC)CCNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-7882 c1c(cc(cc1C(F)(F)F)NC(=S)NCCN2CCOCC2)C(F)(F)F MS-7883 c1ccc(cc1)N2CCN(CC2)C(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-7884 c1ccc(c(c1)N2CCN(CC2)C(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)F MS-7885 COc1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S MS-7886 CC(=O)Nc1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S MS-7887 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)Cc3cccnc3 MS-7888 COc1ccc(cc1OC)CCn2c(=O)c3ccccc3[nH]c2=S MS-7889 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3F)F MS-7890 COCCn1c(=O)c2ccccc2[nH]c1=S MS-7891 c1ccc(cc1)CCn2c(=O)c3ccccc3[nH]c2=S MS-7892 c1ccc(cc1)CCNC(=S)NC(=O)c2cccs2 MS-7893 COCCNC(=S)NC(=O)c1cccs1 MS-7894 c1cc(cnc1)CNC(=S)NC(=O)c2cccs2 MS-7895 COc1ccc(cc1OC)CCNC(=S)NC(=O)c2cccs2 MS-7896 COc1ccc(cc1)NC(=S)NC(=O)c2cccs2 MS-7897 c1ccc(c(c1)C(=O)NNC(=S)NC(=O)c2cccs2)Cl MS-7898 c1cc(sc1)C(=O)NC(=S)NNC(=O)c2ccc(cc2)O MS-7899 CC(C)(C)C(=O)/C(=C/N1CCN(CC1)C/C=C/c2ccccc2)/C#N MS-7900 Cc1ccc(cc1)S(=O)(=O)/C(=C/N2CCN(CC2)Cc3ccccc3)/C#N MS-7901 c1ccc(cc1)NC(=O)N2CCN(CC2)c3cccc(c3)Cl MS-7902 CC(C)(C)C(=O)/C(=C\N1CCN(CC1)Cc2ccccc2)/C#N MS-7903 c1ccc(cc1)/C=C/C(=O)N2CCN(CC2)c3cccc(c3)Cl MS-7904 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)CCl MS-7905 CCOC(=O)/C(=N\OC)/c1csc(n1)NC(=O)c2ccc(cc2)Cl MS-7906 c1cc(sc1)CNC(=O)CCl MS-7907 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)CSc3nc4c(c5ccccc5[nH]4)nn3 MS-7908 c1cc(sc1)CNS(=O)(=O)c2ccc(cc2)OC(F)(F)F MS-7909 COc1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-7910 CCOC(=O)/C(=C/N1CCN(CC1)c2cccc(c2)C(F)(F)F)/C#N MS-7911 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=S)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F MS-7912 c1cc(sc1)C(=O)NC(=S)Nc2ccc(cc2F)F MS-7913 Cc1cc(no1)NC(=S)NC(=O)c2ccc(cc2)C(C)(C)C MS-7914 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)C MS-7915 CC(C)(C)c1ccc(cc1)C(=O)NCCc2c[nH]c3c2cccc3 MS-7916 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3cccc(c3)C(F)(F)F MS-7917 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 MS-7918 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)Cc3ccccc3 MS-7919 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3cccc(c3)Cl MS-7920 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)C MS-7921 CC(C)(C)c1ccc(cc1)C(=O)NCCOC MS-7922 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccccc3 MS-7923 Cc1ccc(cc1N2CCN(CC2)C(=O)c3ccc(cc3)C(C)(C)C)Cl MS-7924 c1ccc2cc(ccc2c1)S(=O)(=O)Nc3ccccc3C(=O)N MS-7925 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3 MS-7926 c1ccc(cc1)/C=C/CN2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3 MS-7927 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3 MS-7928 COC(=O)CNS(=O)(=O)c1ccc2ccccc2c1 MS-7929 Cc1ccc2c(c1)CCCN2S(=O)(=O)c3ccc4ccccc4c3 MS-7930 C#CCNS(=O)(=O)c1ccc2ccccc2c1 MS-7931 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)c4ccccc4F MS-7932 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3ccccc3 MS-7933 c1ccc(cc1)COc2cccnc2NC(=O)c3cccs3 MS-7934 c1ccc(cc1)COc2cccnc2NC(=S)NC(=O)c3ccc(cc3)Cl MS-7935 Cc1ccc(cc1)C(=O)NC(=S)Nc2c(cccn2)OCc3ccccc3 MS-7936 CC1(CC(=C(C(=O)C1)C(c2ccc(cc2)C(=O)O)C3=C(CC(CC3=O)(C)C)O)O)C MS-7937 CNC(=S)N1CCN(CC1)c2cccc(c2)Cl MS-7938 c1ccc(c(c1)C(=O)N)NS(=O)(=O)c2ccc(cc2)Br MS-7939 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(cc3)Br MS-7940 c1ccc(cc1)c2c(n(c(n2)c3cccc4c3cccc4)c5ccc(cc5)OC(F)(F)F)c6ccccc6 MS-7941 COc1ccc(cc1)c2nc(c(n2c3ccc(cc3)OC(F)(F)F)c4ccccc4)c5ccccc5 MS-7942 COc1cc(cc(c1OC)OC)c2nc(c(n2c3ccc(cc3)OC(F)(F)F)c4ccccc4)c5ccccc5 MS-7943 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)Oc3ccccc3 MS-7944 c1cc(oc1)C(=O)N2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Br MS-7945 c1cc(oc1)C(=O)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Br MS-7946 CC(C)(C)c1ccc(cc1)C2=NCCc3c2cc(c(c3)OC)OC MS-7947 c1ccc(cc1)COc2cccnc2NC(=O)Nc3cccc(c3)C(F)(F)F MS-7948 CC1(CC(=C(C(=O)C1)C(c2ccccc2F)C3=C(CC(CC3=O)(C)C)O)O)C MS-7949 CC(C)c1ccc(cc1)C(C2=C(CC(CC2=O)(C)C)O)C3=C(CC(CC3=O)(C)C)O MS-7950 CC1(CC(=C(C(=O)C1)C(c2cccs2)C3=C(CC(CC3=O)(C)C)O)O)C MS-7951 CC1(OC(=O)C(=Cc2c(cccc2Cl)F)C(=O)O1)C MS-7952 CC1(OC(=O)C(=Cc2ccccc2OC)C(=O)O1)C MS-7953 Cc1ccc(cc1C)/C(=N\O)/c2ccccc2 MS-7954 Cc1ccc(cc1C)/C(=N\OC(=O)c2cccs2)/c3ccccc3 MS-7955 c1ccc(c(c1)CC(=O)O)C(=O)Nc2cccc(c2)Cl MS-7957 c1ccc(c(c1)CC(=O)O)C(=O)Nc2ccc(cc2Cl)Cl MS-7958 c1ccc(c(c1)CC(=O)O)C(=O)Nc2cccc(c2)[N+](=O)[O-] MS-7959 c1ccc(c(c1)CC(=O)O)C(=O)Nc2cccc(c2)Br MS-7960 c1ccc(c(c1)CC(=O)O)C(=O)Nc2ccc(cc2)OC(F)(F)F MS-7961 c1ccc(c(c1)CC(=O)O)C(=O)Nc2ccc3c(c2)OCO3 MS-7962 COc1ccc(cc1)n2c(c(nc2c3ccc(cc3)O)c4ccccc4)c5ccccc5 MS-7963 c1ccc(c(c1)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ncccn3)[N+](=O)[O-] MS-7964 c1cc(sc1)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ncccn3 MS-7965 Cc1ccc(cc1)S(=O)(=O)/C(=C\c2cc(c(c(c2)Br)O)Br)/C#N MS-7966 COc1ccc(cc1)c2nc(c(n2c3ccc(cc3)OC)c4ccccc4)c5ccccc5 MS-7967 Cc1ccc(cc1)S(=O)(=O)CC(=O)N/N=C\2/c3cc(ccc3NC2=O)Br MS-7968 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=S)Nc2ccc(cc2)OC(F)(F)F MS-7969 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=S)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C MS-7970 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)C(=O)O MS-7971 Cc1ccc(cc1)S(=O)(=O)CC(=O)NNC(=S)NC(=O)c2cccs2 MS-7972 c1ccc(cc1)CN2CCN(CC2)/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Br MS-7973 Cc1ccc(cc1N2CCN(CC2)/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Br)Cl MS-7974 CC(C)(C)C(=O)/C(=C\c1ccc(cc1)N2CCCCC2)/C#N MS-7975 Cc1ccc(cc1C)/C(=N\OC(=O)c2c(onc2c3c(cccc3Cl)F)C)/c4ccccc4 MS-7976 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4ccccc4F MS-7977 Cc1cc(ccc1Oc2c(cccn2)C(=O)N3CCN(CC3)c4ccccc4OC)Cl MS-7978 Cc1cc(ccc1Oc2c(cccn2)C(=O)N3CCN(CC3)Cc4ccccc4)Cl MS-7979 Cc1cc(ccc1Oc2c(cccn2)C(=O)N3CCN(CC3)c4ccccc4F)Cl MS-7980 Cc1ccc(cc1N2CCN(CC2)C(=O)c3cccnc3Oc4ccc(cc4C)Cl)Cl MS-7981 Cc1cc(ccc1Oc2c(cccn2)C(=O)Nc3ccc4c(c3)OCO4)Cl MS-7982 CC(C(=O)NCCc1ccccc1)Sc2ccc(cc2)Cl MS-7983 Cc1ccc(cc1N2CCN(CC2)C(=O)C(C)Sc3ccc(cc3)Cl)Cl MS-7984 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)c3ccccc3OC)C MS-7985 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)Cc3ccccc3)C MS-7986 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)c3ccccc3)C MS-7987 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)c3ccccc3F)C MS-7988 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3c(cc(cc3C)C)C)Cl MS-7989 Cc1cc(c(c(c1)C)S(=O)(=O)Nc2ccc(cc2F)F)C MS-7990 Cc1cc(c(c(c1)C)S(=O)(=O)Nc2cccc(c2)Br)C MS-7991 Cc1cc(c(c(c1)C)S(=O)(=O)NCCC(c2ccccc2)c3ccccc3)C MS-7992 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)C MS-7993 Cc1cc(c(c(c1)C)S(=O)(=O)NCC(OC)OC)C MS-7994 Cc1cc(c(c(c1)C)S(=O)(=O)NCCc2ccc(c(c2)OC)OC)C MS-7995 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)C(=O)N3CCN(CC3)c4ccccc4 MS-7996 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccc4c(c3)OCO4 MS-7997 Cc1c(cc(cc1)Cl)N2CCN(CC2)C(=O)C34C[C@H]5C[C@@H](C3)C[C@@H](C4)C5 MS-7998 c1cc(c(cc1)F)N2CCN(CC2)C(=O)C34C[C@H]5C[C@@H](C3)C[C@@H](C4)C5 MS-7999 CC1(OC(=O)C(=CNc2ccc(cc2)S(=O)(=O)Nc3ncccn3)C(=O)O1)C MS-8000 c1cc(ccc1C(=O)NC(=S)N2CCN(CC2)C=O)Cl MS-8001 COc1ccc(cc1OC)CCNC(=O)c2cccnc2C(=O)O MS-8002 CC1(CC(=O)C(=CNc2ccccc2C(=O)N)C(=O)C1)C MS-8003 c1ccc2c(c1)C(=O)C(=CNc3ccc4cn[nH]c4c3)C2=O MS-8004 C#CCNC(=S)Nc1ccc(cc1)[N+](=O)[O-] MS-8005 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccccc3F MS-8006 CC1(C(CCC1(C)C(=O)Nc2cccc(c2)Br)C(=O)O)C MS-8007 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)C3CCCCC3C(=O)O MS-8008 c1ccc(c(c1)N2CCN(CC2)C(=O)C3CCCCC3C(=O)O)F MS-8009 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)C3CCCCC3C(=O)O MS-8010 Cc1cc(no1)NC(=O)C2CCCCC2C(=O)O MS-8011 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)C3CCCCC3C(=O)O MS-8012 c1cc(cnc1)CNC(=O)C2CCCCC2C(=O)O MS-8013 c1ccc(cc1)Oc2ccc(cc2)NC(=O)C3CCCCC3C(=O)O MS-8014 c1cc2c(cc1CN3CCN(CC3)C(=O)C4CCCCC4C(=O)O)OCO2 MS-8015 c1cc(cc(c1)Br)NC(=O)C2CCCCC2C(=O)O MS-8016 CCCCCNC(=S)N1CCN(CC1)Cc2ccccc2 MS-8017 CC(C)NC(=S)N1CCN(CC1)C(=O)c2ccco2 MS-8018 CC(=O)c1ccc(cc1)NC(=O)c2cccnc2C(=O)O MS-8019 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cccnc3C(=O)O MS-8020 c1ccc(cc1)CCNC(=O)c2cccnc2C(=O)O MS-8021 COc1ccc(c(c1)S(=O)(=O)N2CCC(CC2)C(=O)N)OC MS-8022 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCC(CC2)C(=O)N MS-8023 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)Nc3ccc(cc3)Cl MS-8024 c1ccc2c(c1)CCN2C(=O)Nc3ccc(cc3)Cl MS-8025 c1cc(cnc1)CNC(=O)Nc2ccc(cc2)Cl MS-8026 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3c(cccc3Cl)F MS-8027 CCOC(=O)/C(=C/N1CCN(CC1)c2ccc(cn2)C(F)(F)F)/C#N MS-8028 CN(C)c1ccc(cc1)/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl MS-8029 c1ccc(cc1)c2c3=c(c4ccccc4c3=O)[nH]c5ccccc5n2 MS-8030 c1cc(ccc1NC2=CC(=O)CCC2)NC3=CC(=O)CCC3 MS-8031 CC(C)(C)C\1=NN(C(=O)/C1=C\c2ccc(cc2Cl)Cl)c3ccc(cc3)[N+](=O)[O-] MS-8032 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cccs2)c3ccc(cc3)[N+](=O)[O-] MS-8033 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cc(c(c(c2)OC)OC)OC)c3ccc(cc3)[N+](=O)[O-] MS-8034 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cccc3c2cccc3)c4ccccc4 MS-8035 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)Nc3ccccc3)C MS-8036 c1ccc(cc1)CNC(=S)N2CCN(CC2)C/C=C/c3ccccc3 MS-8037 c1ccc(c(c1)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl)F MS-8038 CC1(Cc2cccc(c2O1)OCC(=O)N/N=C\3/c4ccccc4NC3=O)C MS-8039 CC(C)c1ccc(cc1)/N=C\2/c3ccccc3NC2=O MS-8040 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=O)Nc3ccc(c(c3)Cl)Cl)C MS-8041 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=O)Nc3ccc(cc3)Cl)C MS-8042 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=S)Nc3ccc(cc3)OC)C MS-8043 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=S)Nc3cc(ccc3OC)Cl)C MS-8044 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=S)Nc3ccc(cc3)[N+](=O)[O-])C MS-8045 Cc1ccccc1NC(=O)NNC(=O)COc2cccc3c2OC(C3)(C)C MS-8046 CCOC(=O)N1CCN(CC1)C(=S)NCc2ccccc2 MS-8047 c1ccc(c(c1)N2CCN(CC2)C(=O)/C=C/C(=O)O)F MS-8048 c1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)Cl)F MS-8049 c1cc(c(cc1NS(=O)(=O)c2cc(ccc2Cl)Cl)C(F)(F)F)F MS-8050 CSc1nc(nn1S(=O)(=O)c2cc(ccc2Cl)Cl)N MS-8051 Cc1cc(no1)NS(=O)(=O)c2cc(ccc2Cl)Cl MS-8052 c1ccnc(c1)NS(=O)(=O)c2cc(ccc2Cl)Cl MS-8053 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)Cl MS-8054 c1cc(c(cc1Cl)S(=O)(=O)NCCN2CCOCC2)Cl MS-8055 c1ccc(cc1)/C=C/CN2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)Cl MS-8056 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3cc(ccc3Cl)Cl MS-8057 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2cc(ccc2Cl)Cl MS-8058 COC(CNS(=O)(=O)c1cc(ccc1Cl)Cl)OC MS-8059 COc1ccc(cn1)NS(=O)(=O)c2cc(ccc2Cl)Cl MS-8060 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] MS-8061 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)CBr MS-8062 c1ccc(cc1)S(=O)(=O)NCc2cccnc2 MS-8063 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)CSc3[nH]c(=O)c4ccccc4n3 MS-8064 CC(C)(C)C1=NN(C(=O)C1)c2ccc(cc2)[N+](=O)[O-] MS-8065 CCOc1ccc(cc1)NC2=C/C(=[NH+]/c3ccc(cc3)OCC)/c4c2cccc4.[Cl-] MS-8066 c1cc(sc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-8067 c1ccc(cc1)CCNC(=S)Nc2ccc(cc2)[N+](=O)[O-] MS-8068 COc1ccccc1N2CCN(CC2)C(=O)c3c(cccc3F)F MS-8069 c1cc(cc(c1)Br)NC(=O)C23CC4CC(C2)CC(C4)C3 MS-8070 c1ccc(cc1)Oc2ccc(cc2)NC(=O)Nc3ccc(cc3)Cl MS-8071 COC(=O)c1cc(cc(c1)NC(=O)CCC(=O)O)C(=O)OC MS-8072 COC(=O)c1cc(cc(c1)NC(=O)C2CCCCC2C(=O)O)C(=O)OC MS-8073 COC(=O)c1cc(cc(c1)NC(=O)Nc2ccccc2)C(=O)OC MS-8074 Cc1cc(c(c(c1)C)S(=O)(=O)Nc2cc(cc(c2)C(=O)OC)C(=O)OC)C MS-8075 COC(=O)c1cc(cc(c1)NS(=O)(=O)c2ccc3ccccc3c2)C(=O)OC MS-8076 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3cc(cc(c3)C(=O)OC)C(=O)OC)C MS-8077 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(cc(c3)C(=O)OC)C(=O)OC MS-8078 COC(=O)c1cc(cc(c1)NC=C2C(=O)c3ccccc3C2=O)C(=O)OC MS-8079 CCOC(=O)N1CCN(CC1)C(=S)Nc2ccc(cc2)C MS-8080 c1cc(ccc1NC(=S)N2CCN(CC2)C=O)[N+](=O)[O-] MS-8081 CCOC(=O)N1CCN(CC1)C(=S)NC(C)(C)C MS-8082 CC(C)(C)NC(=S)N1CCN(CC1)Cc2ccc3c(c2)OCO3 MS-8083 CC(C)(C)NC(=S)N1CCN(CC1)C(c2ccccc2)c3ccccc3 MS-8084 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)N(C)C MS-8085 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(nc3)OC MS-8086 COc1ccc(cn1)NC(=S)NC(=O)C2CC2 MS-8087 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=S)NC(=O)c4c(cccc4F)F MS-8088 CC1=C(C(NC(=S)N1)c2ccc(cc2)C(C)C)C(=O)OC MS-8089 CC1=C(C(NC(=S)N1)c2ccc(cc2)Cl)C(=O)OC MS-8090 CC1=C(C(NC(=S)N1)c2ccccc2OC)C(=O)OC MS-8091 CC1=C(C(NC(=S)N1)c2ccc(cc2)F)C(=O)OC MS-8092 CC1=C(C(NC(=S)N1)c2ccc(c(c2)OC)OC)C(=O)OC MS-8093 CC1=C(C(NC(=S)N1)c2cccc3c2cccc3)C(=O)OC MS-8094 CC(C)(C)NC(=S)N1CCN(CC1)c2ccccc2F MS-8095 CC(C)(C)NC(=S)NCCc1c[nH]c2c1cccc2 MS-8096 CC(C)(C)NC(=S)NNC(=O)c1ccncc1 MS-8097 Cc1ccc(cc1)NC(=S)NNC(=O)COc2ccccc2Cl MS-8098 Cc1ccc(cc1)n2c(n[nH]c2=S)COc3ccccc3Cl MS-8099 CC1(Cc2c(cc(n2c3ccc(cc3)S)c4ccc(cc4)Br)C(=O)C1)C MS-8100 Cc1cc2c(n1CCC(=O)O)CC(CC2=O)(C)C MS-8102 Cc1ccc(cc1)NC(=S)NNC(=O)COc2cccc3c2OC(C3)(C)C MS-8103 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=S)NC)C MS-8105 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=O)NS(=O)(=O)c3ccccc3)C MS-8106 c1ccc(cc1)CN2CCN(CC2)C(=O)/C=C/C(=O)O MS-8107 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)/C=C/C(=O)O MS-8108 c1ccc(cc1)CNC(=S)N2CCN(CC2)c3ccccn3 MS-8109 Cc1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccn3 MS-8110 CCOC(=O)N1CCN(CC1)C(=S)NC MS-8111 CCCCNC(=O)N1CCN(CC1)Cc2ccccc2 MS-8112 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccccc3C(=O)OC MS-8113 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCc3ccc(c(c3)OC)OC MS-8114 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)OC MS-8115 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3F)F MS-8116 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(ccc3F)C(F)(F)F MS-8117 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3ccc(cc3)Cl MS-8118 Cc1cc(no1)NC(=O)c2ccc(cc2)Cl MS-8119 CS(=O)(=O)c1ccc2c(c1)sc(n2)NC(=O)c3ccc(cc3)Cl MS-8120 c1ccc(cc1)N2CCN(CC2)C(=O)C(=O)c3c[nH]c4c3cccc4 MS-8121 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)N3CCN(CC3)c4ncccn4 MS-8122 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)C(=O)c4c[nH]c5c4cccc5 MS-8123 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)C(=O)c3c[nH]c4c3cccc4 MS-8124 CCOC(=O)N1CCN(CC1)C(=O)C(=O)c2c[nH]c3c2cccc3 MS-8125 c1ccc(cc1)CN2CCN(CC2)C(=O)C(=O)c3c[nH]c4c3cccc4 MS-8126 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)N3CCC(CC3)C(=O)N MS-8127 c1cc(c(c(c1)F)C(=O)NC(=S)N2CCCN(CC2)C(=S)NC(=O)c3c(cccc3F)F)F MS-8128 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=S)NC(=O)c3c(cccc3F)F MS-8129 c1cc(c(c(c1)F)C(=O)NC(=S)N2CCN(CC2)C=O)F MS-8130 c1cc(c(c(c1)F)C(=O)NC(=S)N2CCN(CC2)Cc3ccc4c(c3)OCO4)F MS-8131 c1ccnc(c1)N2CCN(CC2)C(=S)NC(=O)c3c(cccc3F)F MS-8132 c1cc(c(cc1C(F)(F)F)NC(=O)c2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-])Cl MS-8133 Cc1cc2c(n1c3cccc(c3)OC(F)(F)F)CC(CC2=O)(C)C MS-8134 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)C(=O)C MS-8135 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc(c3)OC MS-8136 COc1ccc(c(c1)S(=O)(=O)N2CCN(CC2)c3ccccn3)OC MS-8137 COc1ccc(c(c1)S(=O)(=O)N2CCN(CC2)c3ccccc3F)OC MS-8138 COc1ccc(c(c1)S(=O)(=O)N2CCN(CC2)c3ccccc3)OC MS-8139 c1ccc2c(c1)c(c[nH]2)CCNC(=S)Nc3ccc(cc3)C#N MS-8140 c1cc(ccc1C#N)NC(=S)N2CCN(CC2)Cc3ccc4c(c3)OCO4 MS-8141 c1ccnc(c1)N2CCN(CC2)C(=S)Nc3ccc(cc3)C#N MS-8142 c1ccc(c(c1)N2CCN(CC2)C(=S)Nc3ccc(cc3)C#N)F MS-8143 c1ccc(cc1)N2CCN(CC2)C(=S)Nc3ccc(cc3)C#N MS-8144 c1cc(ccc1C#N)NC(=S)NCCN2CCN(CC2)C(=S)Nc3ccc(cc3)C#N MS-8145 CC(C(=O)NNC(=S)NCc1ccccc1)Oc2ccc(cc2Cl)Cl MS-8146 Cc1ccc(cc1N2CCN(CC2)C(=O)Cc3cccc4c3cccc4)Cl MS-8147 c1ccc(cc1)/C=C/C(=O)NC(=S)NCCN2CCOCC2 MS-8148 COc1cc(c(cc1OC)S(=O)(=O)N2CCN(CC2)c3ccccn3)CC(=O)OC MS-8149 c1ccc(c(c1)C#N)NC2=CC(=O)CCC2 MS-8150 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCCc2ccc(c(c2)OC)OC MS-8151 Cc1ccc2c(c1)CCC[N@]2S(=O)(=O)c3ccc(cc3)NC(=O)C MS-8152 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8153 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccccc3 MS-8154 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccc3 MS-8155 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)Cc3ccccc3 MS-8156 CC(C)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)NC(=O)C MS-8157 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)I MS-8158 c1cc(ccc1S(=O)(=O)NC2CC2)I MS-8159 c1ccc(c(c1)N2CCN(CC2)C(=S)NC(=O)c3ccc(cc3)I)F MS-8160 CC1=C(C(NC(=O)N1)c2cccc(c2)Oc3ccccc3)C(=O)OC MS-8161 CCOC(=O)C1=C(NC(=O)NC1c2cc(c(c(c2)OC)OC)OC)c3ccccc3 MS-8162 c1cnc(nc1)NC(=S)N MS-8163 Cc1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)C#N MS-8164 Cc1ccc(cc1)NC(=S)NNC(=O)C(C)Oc2ccc(cc2Cl)Cl MS-8165 CC1CC(=O)C(C(=O)C1)CC(=O)c2ccc(cc2Cl)Cl MS-8166 c1ccc(cc1)/C=C/C(=O)Nc2ccccc2Br MS-8167 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)N3CCN(CC3)C=O MS-8168 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)C#N MS-8169 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8170 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2)OC(F)(F)F MS-8171 Cc1ccc(c(c1)C)NC(=S)NC(=O)/C=C/c2ccccc2 MS-8172 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2)F MS-8173 CCOC(=O)N1CCN(CC1)C(=O)c2cccc(c2)OC(C(F)F)(F)F MS-8174 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cccc(c3)OC(C(F)F)(F)F MS-8175 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)c3cccc(c3)OC(C(F)F)(F)F MS-8176 c1ccc(c(c1)N2CCN(CC2)C(=O)c3cccc(c3)OC(C(F)F)(F)F)F MS-8177 c1ccc2c(c1)CCN2C(=S)NC(=O)c3ccc(cc3)[N+](=O)[O-] MS-8178 Cc1ccc(cc1)C(=O)NC(=S)Nc2cc(ccc2OC)OC MS-8179 Cc1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)Cl MS-8180 Cc1ccc(cc1)C(=O)NC(=S)Nc2ccc(c(c2)Cl)Cl MS-8181 Cc1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)c3cc(ccc3C)Cl MS-8182 Cc1ccc(cc1)S(=O)(=O)NCC=C MS-8183 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccccc2Br MS-8184 c1cc(c(cc1[N+](=O)[O-])NC(=O)C2CCCCC2)Cl MS-8185 c1ccc(cc1)C(c2ccccc2)C(=O)Nc3cc(ccc3Cl)[N+](=O)[O-] MS-8186 c1ccc(cc1)CC(=O)Nc2cc(ccc2Cl)[N+](=O)[O-] MS-8187 c1cc(c(cc1[N+](=O)[O-])NC(=O)C2CC2)Cl MS-8188 CC(C)C(=O)Nc1c(cc(cc1Br)F)F MS-8189 c1ccc(cc1)C(c2ccccc2)C(=O)Nc3c(cc(cc3Br)F)F MS-8190 c1c(cc(c(c1F)NC(=O)C2CC2)Br)F MS-8191 CC1CC(=O)C(C(=O)C1)CC(=O)c2ccc(cc2)Cl MS-8192 c1cscc1/C=C/2\C(=O)NC(=S)N2 MS-8193 CCN1C(=O)/C(=C\c2ccc(c(c2)OC)OCc3ccc(cc3)[N+](=O)[O-])/SC1=S MS-8194 Cc1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2OC)[N+](=O)[O-] MS-8195 Cc1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2[N+](=O)[O-])Cl MS-8196 COc1cc(c(cc1Br)Br)NC(=O)C2CCCCC2 MS-8197 c1ccc(cc1)C(c2ccccc2)C(=O)Nc3ccccc3Br MS-8198 c1ccc(cc1)C(c2ccccc2)C(=O)N3CCN(CC3)c4ccccn4 MS-8199 c1ccc(cc1)C(c2ccccc2)C(=O)Nc3ccc(cc3F)F MS-8200 COc1ccc(cc1OC)CCNC(=O)C(c2ccccc2)c3ccccc3 MS-8201 c1ccc(cc1)CN2CCN(CC2)C(=O)C(c3ccccc3)c4ccccc4 MS-8202 c1ccc(cc1)C(c2ccccc2)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 MS-8203 c1ccc(cc1)C(c2ccccc2)C(=O)Nc3ccc(cc3)OC(F)(F)F MS-8204 c1cc(sc1)CC(=O)Nc2c(cc(cc2Br)F)F MS-8206 c1cc(sc1)CC(=O)Nc2ccc(cc2F)F MS-8207 c1ccc(c(c1)NC(=O)Cc2cccs2)F MS-8208 c1ccnc(c1)N2CCN(CC2)C(=O)Cc3cccs3 MS-8209 Cc1ccc(cc1N2CCN(CC2)C(=O)Cc3cccs3)Cl MS-8210 c1ccc(cc1)CN2CCN(CC2)C(=O)Cc3cccs3 MS-8211 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Cc4cccs4 MS-8212 COc1cccc(c1)NC(=O)COc2ccccc2 MS-8213 c1ccc(cc1)OCC(=O)Nc2c(cc(cc2Br)F)F MS-8214 c1ccc(cc1)CN2CCN(CC2)C(=O)COc3ccccc3 MS-8215 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)COc4ccccc4 MS-8216 c1ccc(cc1)OCC(=O)N2CCN(CC2)c3ccccc3F MS-8217 c1ccc(cc1)OCC(=O)NCCN2CCN(CC2)C(=O)COc3ccccc3 MS-8218 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)OC(F)(F)F MS-8219 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)Nc3ccc(cc3)OC(F)(F)F MS-8220 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)NC3CC3 MS-8221 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccc(cc4)Cl MS-8222 c1ccc(cc1)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl MS-8223 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccccc4 MS-8224 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)Nc3ccccc3 MS-8225 CC1(CC(=C(C(=O)C1)SC(=NC(=O)c2ccc(cc2)OC)NC(=O)c3ccc(cc3)OC)O)C MS-8226 c1cc(ccc1C(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl MS-8227 c1cc(ccc1c2csc(n2)Nc3ccc(cc3)OC(F)(F)F)Cl MS-8228 c1cc(cc(c1)Br)c2csc(n2)Nc3ccc(cc3)OC(F)(F)F MS-8229 COc1cc(ccc1OCc2ccc(cc2)[N+](=O)[O-])/C=C(/C#N)\C(=O)c3ccccc3 MS-8230 CC(C)(C)S(=O)(=O)/C(=C\c1ccc(c(c1)OC)OCc2ccc(cc2)[N+](=O)[O-])/C#N MS-8231 CC(C)(C)C(=O)/C(=C\c1ccc(c(c1)OC)OCc2ccc(cc2)[N+](=O)[O-])/C#N MS-8232 c1ccc(cc1)/C=C\2/c3ccccc3NC2=O MS-8233 c1ccc(cc1)CNC(=S)NNC(=O)Cc2c[nH]c3c2cccc3 MS-8234 CC1(Cc2c(cc(n2c3ccc(cc3)C(=O)N)c4ccc(cc4)Br)C(=O)C1)C MS-8235 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cccs3 MS-8236 C/C(=C\C(=O)Nc1ccc(cc1)Cl)/N2CCN(CC2)c3ccccc3 MS-8237 c1ccc(cc1)OCC(=O)Nc2ccc(cc2)OC(F)(F)F MS-8238 c1ccc(cc1)OCC(=O)Nc2ccccc2Cl MS-8239 c1ccc(cc1)OCC(=O)Nc2ccc(cc2F)F MS-8240 c1ccc(cc1)OCC(=O)Nc2ccccc2F MS-8241 Cc1ccc(cc1N2CCN(CC2)C(=O)COc3ccccc3)Cl MS-8242 c1ccc(cc1)OCC(=O)NCCN2CCOCC2 MS-8243 c1ccc(cc1)OCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8244 c1ccc(cc1)OCC(=O)Nc2ccccc2I MS-8245 c1ccc(cc1)C(c2ccccc2)C(=O)Nc3ccccc3I MS-8246 c1ccc(cc1)CC(=O)Nc2ccccc2I MS-8247 c1ccc(c(c1)NC(=O)Cc2cccs2)I MS-8248 COc1cc(c(cc1OC)NC(=S)NCc2ccccc2)C(=O)OC MS-8249 COc1cc(c(cc1OC)NC(=O)COc2ccccc2)C(=O)OC MS-8250 CC(C(=O)Nc1ccccc1F)Cl MS-8251 CC(C(=O)Nc1cc(ccc1O)Cl)Cl MS-8252 C/C(=C\C(=O)Nc1ccc(cc1)Cl)/NCCN2CCOCC2 MS-8253 C/C(=C\C(=O)Nc1ccc(cc1)Cl)/N2CCN(CC2)Cc3ccccc3 MS-8254 c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3 MS-8255 COc1ccc(cc1OC)CCNC(=O)Nc2ccccc2 MS-8256 CC(C)N(c1ccccc1)c2ccc(cc2)NC(=S)NC(=O)c3ccccc3 MS-8257 CC(C)N(c1ccccc1)c2ccc(cc2)NC(=S)N MS-8258 c1ccc(cc1)C(=O)NC(=S)NC2CC2 MS-8259 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl MS-8260 COc1ccc(cc1OC)NC(=O)C(=O)c2c[nH]c3c2cccc3 MS-8261 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4ccc5ccccc5c4 MS-8262 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)[N+](=O)[O-])Cl MS-8263 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3ccc(cc3)NC(=O)C)Cl MS-8264 c1ccc2c(c1)C(=O)C(=CNc3cc(ccc3Cl)[N+](=O)[O-])C2=O MS-8265 COc1cccc(c1)NC=C2C(=O)c3ccccc3C2=O MS-8266 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)Oc3ccccc3 MS-8267 Cc1ccc(cc1)S(=O)(=O)/C(=C\Nc2nc(cc(n2)C)C)/C(=O)C MS-8268 Cc1cc(nc(n1)N/C=C(/C(=O)C)\S(=O)(=O)c2ccc(cc2)Cl)C MS-8269 CC(=O)/C(=C/Nc1ncccn1)/S(=O)(=O)c2ccc(cc2)Cl MS-8270 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccccc3N MS-8271 c1ccc(c(c1)N2CCN(CC2)C(=O)c3cccnc3Cl)F MS-8272 c1cc(c(cc1[N+](=O)[O-])C(=O)NCCN2CCOCC2)Cl MS-8273 COC(=O)c1cc(cc(c1)NC(=O)c2cc(ccc2Cl)[N+](=O)[O-])C(=O)OC MS-8274 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3cc(ccc3Cl)[N+](=O)[O-] MS-8275 CNC(=S)N1CCN(CC1)C(c2ccccc2)c3ccccc3 MS-8276 CNC(=S)Nc1nccs1 MS-8277 CNC(=S)N1CCN(CC1)c2ccccc2 MS-8278 CCCNC(=O)NCCc1ccc(c(c1)OC)OC MS-8279 CCCNC(=O)N1CCN(CC1)C(=O)OCC MS-8280 CCCNC(=O)N1CCN(CC1)c2ccccc2 MS-8281 CCCNC(=O)NCC=C MS-8282 CCCNC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F MS-8283 CCCCNC(=O)N1CCN(CC1)c2ccccc2 MS-8284 c1ccc(cc1)CC(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8285 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)NC(=O)Cc3ccccc3 MS-8286 CC(C)N(c1ccccc1)c2ccc(cc2)NC(=S)NC(=O)Cc3ccccc3 MS-8287 CC(C)N(c1ccccc1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)NC(=O)C MS-8288 CC1CC(=CC(=O)C1)Nc2ccccc2Br MS-8289 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cc(ccc2OC)Br)c3ccccc3 MS-8290 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccccn2)/C(=O)C MS-8291 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2ccccc2 MS-8292 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4ccc(cc4)F)[nH]c2=O MS-8293 CCCn1c(=N)c2c(c(=O)[nH]c(n2)c3cccc(c3)Br)[nH]c1=O MS-8294 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4cccc(c4)Oc5ccccc5)[nH]c2=O MS-8295 c1cc(ccc1S(=O)(=O)NCCN2CCOCC2)Cl MS-8296 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc(cc3)Cl MS-8297 C1CCC(C(C1)C(=O)NC2CC2)C(=O)O MS-8298 c1cc(ccc1NC(=O)C2CCCCC2C(=O)O)I MS-8299 c1cc(c(cc1F)F)NC(=O)C2CCCCC2C(=O)O MS-8300 CC1=CC(=O)N(C1=O)c2nccs2 MS-8301 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-] MS-8302 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 MS-8303 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)I MS-8304 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl MS-8305 Cc1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)Br MS-8306 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3ccc(c(c3)[N+](=O)[O-])Cl)Cl MS-8307 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=S)Nc3ccccc3 MS-8308 c1ccc(c(c1)N2CCN(CC2)C(=S)NC3CCCCC3)F MS-8309 Cc1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccc3F MS-8310 CC(C(=O)Nc1cc(ccc1Cl)[N+](=O)[O-])Cl MS-8311 CCCNC(=O)N1CCN(CC1)c2ccccc2F MS-8312 CCCNC(=O)NCCc1c[nH]c2c1cccc2 MS-8313 CCCNC(=O)N1CCN(CC1)Cc2ccccc2 MS-8314 CCCNC(=O)N1CCN(CC1)C/C=C/c2ccccc2 MS-8315 Cc1ccc(cc1)S(=O)(=O)NC(=O)NC2CC2 MS-8316 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(n(n(c2=O)c3ccccc3)C)C MS-8317 c1ccc(c(c1)N2CCN(CC2)S(=O)(=O)c3ccc(c(c3)[N+](=O)[O-])Cl)F MS-8318 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8319 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)Cc3ccccc3 MS-8320 c1cc(ccc1S(=O)(=O)NCCN2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)Cl MS-8321 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Cl MS-8322 CC(C)c1ccc(cc1)/C=C(\C#N)/C(=O)OC MS-8323 COC(=O)/C(=C\c1cccc(c1)Oc2ccccc2)/C#N MS-8324 COC(=O)/C(=C\c1cccc2c1cccc2)/C#N MS-8325 COC(=O)/C(=C\c1c[nH]c2c1cccc2)/C#N MS-8326 CC1(Cc2c(cc(n2CCC(=O)O)c3ccc(cc3)Br)C(=O)C1)C MS-8327 c1ccc(cc1)NC(=S)NNC(=O)CSc2nc3c(c4ccccc4[nH]3)nn2 MS-8328 Cc1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2)OC(F)(F)F MS-8329 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(C)c2cc(ccc2C(=O)c3ccccc3)Cl MS-8330 Cc1ccc(cc1)n2c(n[nH]c2=S)COc3ccc(cc3)OC(F)(F)F MS-8331 COc1ccc(cc1/C=C(/C#N)\S(=O)(=O)c2ccccc2)Br MS-8332 CCCCNC(=O)NCC=C MS-8333 c1ccc(cc1)S(=O)(=O)NCCN2CCOCC2 MS-8334 CC(C)c1ccc(cc1)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4ccccc4 MS-8335 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4c(cccc4Cl)F)[nH]c2=O MS-8336 Cc1cccc(c1)C(=O)Nc2ccc(cc2)I MS-8337 c1c(cc(cc1C(F)(F)F)NC(=O)C2CCCCC2C(=O)O)C(F)(F)F MS-8339 c1ccnc(c1)N2CCN(CC2)C(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-] MS-8340 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)C/C=C/c3ccccc3 MS-8341 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)C=O MS-8342 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccc(c2)F MS-8343 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(nc2)OC MS-8344 Cc1ccc(cc1)C(=O)N2CCN(CC2)C=O MS-8345 Cc1ccc(cc1)C(=O)NCc2ccncc2 MS-8346 Cc1ccc(cc1N2CCN(CC2)CC(=O)N(c3ccccc3)c4ccccc4)Cl MS-8347 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)N(c4ccccc4)c5ccccc5 MS-8348 c1ccc(cc1)N(c2ccccc2)C(=O)CN3CCN(CC3)c4ccccc4F MS-8349 COc1ccc(cc1)C(=O)NCCc2ccccc2 MS-8350 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc(cc3)[N+](=O)[O-] MS-8351 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=S)NC3CCCCC3 MS-8352 CC(C(=O)Nc1ccc(cc1)I)Cl MS-8353 CCCCCC(=O)N1CCN(CC1)C/C=C/c2ccccc2 MS-8354 CCCNC(=O)N1CCN(CC1)c2ccccn2 MS-8355 CCCNC(=O)N1CCN(CC1)C=O MS-8356 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2F)F MS-8357 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)Cl MS-8358 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccc(c2)C(=O)C MS-8359 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCc2ccccc2 MS-8360 CCCCNC(=O)N1CCN(CC1)C(c2ccccc2)c3ccccc3 MS-8361 CCCCNC(=O)N1CCN(CC1)c2ccccn2 MS-8362 CCCCNC(=O)NCCc1ccccc1 MS-8363 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(c(c2)[N+](=O)[O-])Cl MS-8364 COc1cc(ccc1OCc2ccc(cc2)[N+](=O)[O-])/C=C(\C#N)/S(=O)(=O)c3ccccc3 MS-8365 CCCCNC(=O)NCCc1ccc(c(c1)OC)OC MS-8366 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4cccc5c4cccc5)[nH]c2=O MS-8367 c1ccc(cc1)n2c(=N)c3c(c(=O)[nH]c(n3)c4ccco4)[nH]c2=O MS-8368 CCCNC(=O)N/C(=C(/C#N)\N)/C#N MS-8369 c1ccc2c(c1)CCN2C(=O)C(F)(F)F MS-8370 Cc1cccc(c1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8371 Cc1ccc(cc1N2CCN(CC2)C(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-])Cl MS-8372 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)c3cc(ccc3C)Cl MS-8373 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(c(cc2C(=O)OC)OC)OC MS-8374 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)F MS-8375 c1ccc(cc1)CN2CCN(CC2)CC(=O)N(c3ccccc3)c4ccccc4 MS-8376 c1c(cc(c(c1F)NC(=O)/C=C/C(=O)O)Br)F MS-8377 Cc1ccc(cc1N2CCN(CC2)C(=O)c3ccc(cc3Cl)Cl)Cl MS-8378 CN1CCN(CC1)S(=O)(=O)c2ccccc2 MS-8379 c1ccc(cc1)/C=C/CN2CCN(CC2)S(=O)(=O)c3ccccc3 MS-8380 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccccc3 MS-8381 CCOC(=O)N1CCN(CC1)C(=S)Nc2ccccc2 MS-8382 Cc1ccc(cc1N2CCN(CC2)C(=S)NC3CCCCC3)Cl MS-8383 Cc1ccc(cc1)NC(=S)N2CCN(CC2)C/C=C/c3ccccc3 MS-8384 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)c3ccccc3F MS-8385 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccccc2C#N MS-8386 c1ccc(cc1)C(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8387 COC(=O)/C(=C\c1cc2c(cc1[N+](=O)[O-])OCO2)/C#N MS-8388 COC(=O)/C(=C\c1ccsc1)/C#N MS-8389 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)F MS-8390 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F MS-8391 c1cc2c(cc1CN3CCN(CC3)CC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)OCO2 MS-8392 c1ccc2c(c1)CCN2S(=O)(=O)c3cccs3 MS-8393 Cc1ccc(cc1)NC(=S)NNC(=O)COc2cccc(c2Cl)Cl MS-8394 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)Nc3cc(cc(c3)Cl)Cl MS-8395 CN1c2ccccc2C(C1=O)(c3ccccc3)c4ccccc4 MS-8396 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)C(c3ccccc3)c4ccccc4)OC MS-8397 Cc1ccc(cc1N2CCN(CC2)CC(=O)Nc3cc(ccc3OC)OC)Cl MS-8398 Cc1ccc(cc1N2CCN(CC2)CCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl MS-8399 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccccn3)OC MS-8400 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ncccn3)OC MS-8401 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)Nc4ccccc4Br MS-8402 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)Cc3ccc4c(c3)OCO4)OC MS-8403 COC(=O)c1cc(cc(c1)NC(=O)CN2CCN(CC2)c3ccccc3)C(=O)OC MS-8404 COC(=O)c1cc(cc(c1)NC(=O)CN2CCN(CC2)c3ncccn3)C(=O)OC MS-8405 CCOC(=O)N1CCN(CC1)CC(=O)Nc2ccccc2Br MS-8406 c1ccc(cc1)/C=C/CN2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCO4 MS-8407 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCO4 MS-8408 c1ccnc(c1)N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCO4 MS-8409 Cc1ccc(cc1N2CCN(CC2)CC(=O)Nc3ccccc3Br)Cl MS-8410 c1cc2c(cc1CN3CCN(CC3)CC(=O)Nc4ccc5c(c4)OCO5)OCO2 MS-8411 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)Nc3ccc(cc3)OC(F)(F)F MS-8412 CCOC(=O)N1CCN(CC1)CC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-8413 CCOC(=O)N1CCN(CC1)CC(=O)Nc2ccc(cc2F)F MS-8414 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccccc3F)Br MS-8415 COc1ccc(c(c1)NC(=O)CN2CCc3c2cccc3)OC MS-8416 CC(=O)c1cc2c(cc1NC(=O)CN3CCc4c3cccc4)OCO2 MS-8417 c1ccc2c(c1)CCN2CC(=O)Nc3ccc4c(c3)OCO4 MS-8418 COc1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ccccc3F)OC MS-8419 c1ccc(cc1)COc2cccnc2NC(=O)c3ccc(cc3)[N+](=O)[O-] MS-8420 c1ccc(cc1)COc2cccnc2NC(=O)C3CCCCC3 MS-8421 Cc1ccc(cc1)C(=O)Nc2c(cccn2)OCc3ccccc3 MS-8422 CC(=O)c1cc2c(cc1NC(=O)CN3CCN(CC3)c4ccccc4F)OCO2 MS-8423 CC(=O)c1cc2c(cc1NC(=O)CN3CCN(CC3)C(c4ccccc4)c5ccccc5)OCO2 MS-8424 CC(=O)c1cc2c(cc1NC(=O)CN3CCN(CC3)C)OCO2 MS-8425 Cc1ccc(cc1N2CCN(CC2)CC(=O)Nc3cc4c(cc3C(=O)C)OCO4)Cl MS-8426 CC(=O)c1cc2c(cc1NC(=O)CN3CCN(CC3)c4ccccc4)OCO2 MS-8427 c1ccc(c(c1)N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCO4)F MS-8428 CCOC(=O)N1CCN(CC1)CC(=O)Nc2ccc3c(c2)OCO3 MS-8429 Cc1ccc(cc1N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCO4)Cl MS-8430 Cc1c(sc(n1)Nc2ccc(cc2)OC(F)(F)F)C(=O)C MS-8431 Cc1c(sc(n1)NCCc2ccccc2)C(=O)C MS-8432 CCOC(=O)c1c(nc(s1)NCCc2ccccc2)C MS-8434 c1cc(ccc1c2csc(n2)Nc3ccc(cc3)OC(F)(F)F)F MS-8436 c1ccnc(c1)Nc2nc(cs2)c3ccc(cc3)F MS-8437 c1ccc(cc1)CCNc2nc(cs2)c3ccc(cc3)F MS-8438 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3ncccn3)Br MS-8439 c1cc(c(cc1F)F)NC(=O)N2CCN(CC2)C=O MS-8440 Cc1ccc(cc1N2CCN(CC2)C(=O)NC3CCCCC3)Cl MS-8441 CCOC(=O)N1CCN(CC1)C(=O)Nc2ccc-3c(c2)Cc4c3cccc4 MS-8442 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccccc4F MS-8443 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccc(cc4)Br MS-8444 CCOC(=O)N1CCN(CC1)C(=O)Nc2cc(cc(c2)Cl)Cl MS-8445 Cc1ccc(cc1N2CCN(CC2)C(=O)Nc3ccccc3OC)Cl MS-8446 Cc1ccc(cc1N2CCN(CC2)C(=O)NCc3ccccc3)Cl MS-8447 CCOc1ccc(cc1)NC(=O)N2CCN(CC2)c3cc(ccc3C)Cl MS-8448 CCc1ccccc1NC(=O)N2CCN(CC2)c3cc(ccc3C)Cl MS-8449 Cc1ccc(cc1N2CCN(CC2)C(=O)Nc3ccc(cc3)F)Cl MS-8450 CCC(C)NC(=O)N1CCN(CC1)c2cc(ccc2C)Cl MS-8451 c1ccc(cc1)CNC(=O)N2CCN(CC2)Cc3ccccc3 MS-8452 CCc1ccccc1NC(=O)N2CCN(CC2)Cc3ccccc3 MS-8453 CCCCCCNC(=O)N1CCN(CC1)c2ccccc2F MS-8454 COc1ccccc1NC(=O)N2CCN(CC2)c3ccccc3F MS-8455 Cc1ccc(cc1F)NC(=O)N2CCN(CC2)c3ccccc3F MS-8456 CC(C)(C)NC(=O)N1CCN(CC1)c2ccccc2F MS-8457 CCc1ccccc1NC(=O)N2CCN(CC2)c3ccccc3F MS-8458 CCCCCCNC(=O)N1CCN(CC1)c2ccccc2 MS-8459 CCOc1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3 MS-8460 CC(C)(C)NC(=O)N1CCN(CC1)c2ccccc2 MS-8461 CCC(C)NC(=O)N1CCN(CC1)c2ccccc2 MS-8462 CC(C)(C)NC(=O)N1CCN(CC1)C MS-8463 CCOC(=O)N1CCN(CC1)C(=O)NCc2ccccc2 MS-8464 CCOc1ccc(cc1)NC(=O)N2CCN(CC2)C(=O)OCC MS-8465 CCOc1ccccc1NC(=O)N2CCN(CC2)C(=O)OCC MS-8466 CCCCc1ccc(cc1)NC(=O)N2CCN(CC2)C(=O)OCC MS-8467 CCC(C)NC(=O)N1CCN(CC1)C=O MS-8468 Cc1ccc(cc1Cl)NC(=O)N2CCN(CC2)C MS-8469 Cc1ccc(cc1Cl)NC(=O)N2CCN(CC2)Cc3ccccc3 MS-8470 Cc1ccc(cc1Cl)NC(=O)N2CCN(CC2)c3ccccc3 MS-8471 CC(C)(C)c1c2c(no1)-c3ccc(cc3C2=O)[N+](=O)[O-] MS-8472 c1ccc(cc1)/C=C/C(=O)Nc2ccc(cc2)C(=O)N MS-8473 CN(C)c1ccc(cc1)NC(=O)c2cccnc2C(=O)O MS-8474 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4cc5ccccc5[nH]4 MS-8475 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ccccc4F MS-8476 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ccccn4 MS-8477 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 MS-8478 c1ccc(cc1)C2(CCCC2)C(=O)NC3CC3 MS-8479 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cc(ccc3O)Cl MS-8480 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)C(=O)O MS-8481 COC(=O)c1cccc(c1NC(=O)C2(CCCC2)c3ccccc3)C(=O)OC MS-8482 COCCNC(=O)C1(CCCC1)c2ccccc2 MS-8483 c1ccc(cc1)C2(CCCC2)C(=O)Nc3cccc(c3)O MS-8484 CCN(CC)c1ccc(cc1)NC(=O)C2(CCCC2)c3ccccc3 MS-8486 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cn3)Br MS-8487 COc1cc(c(c(c1OC)OC)NC(=O)C2(CCCC2)c3ccccc3)C(=O)OC MS-8488 CC(C)(C)C1CCC(CC1)NC(=O)C2(CCCC2)c3ccccc3 MS-8489 COC(=O)c1ccc(c(c1)NC(=O)C2(CCCC2)c3ccccc3)C(=O)OC MS-8490 Cc1cc(c(c(c1NC(=O)C2(CCCC2)c3ccccc3)C)Br)C MS-8491 CCOC(=O)c1ccccc1NC(=O)C2(CCCC2)c3ccccc3 MS-8492 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc4c(c3)OCCO4 MS-8493 CC1CCCCC1NC(=O)C2(CCCC2)c3ccccc3 MS-8494 Cc1cccc(c1)NC(=O)C2(CCCC2)c3ccccc3 MS-8495 c1ccc(cc1)C2(CCCC2)C(=O)NCc3ccc(cc3F)Br MS-8496 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(c(c3)C(F)(F)F)Cl MS-8497 c1ccc(cc1)C2(CCCC2)C(=O)Nc3ccc(cc3Br)Br MS-8498 CC(C)(CNC(=O)C1(CCCC1)c2ccccc2)CO MS-8499 Cc1ccc(c(c1)N2CCN(CC2)C(=O)C3(CCCC3)c4ccccc4)C MS-8500 c1ccc(cc1)C2(CCCC2)C(=O)N3CCN(CC3)c4ccc(cc4)F MS-8501 Cc1cc2c(n1c3cccc(c3)Cl)CC(CC2=O)C MS-8502 Cc1cc2c(n1c3cc(c(c(c3)Cl)O)Cl)CC(CC2=O)(C)C MS-8503 Cc1cc2c(n1c3cccc(c3)Cl)CC(CC2=O)(C)C MS-8504 Cc1cc2c(n1c3cc(cc(c3)F)F)CC(CC2=O)(C)C MS-8505 Cc1cc2c(n1c3ccc(c(c3)OC)OC)CC(CC2=O)(C)C MS-8506 Cc1cc2c(n1c3ccc(cc3)OC)CC(CC2=O)(C)C MS-8507 Cc1cc2c(n1c3ccc(c(c3)F)F)CC(CC2=O)(C)C MS-8508 c1ccc2c(c1)c(c[nH]2)CCNC(=O)Cc3ccc(cc3)[N+](=O)[O-] MS-8509 c1ccc(c(c1)C(=O)c2ccccn2)N MS-8510 Cc1cc2c(n1c3cccc(c3)C(=O)C)CC(CC2=O)C MS-8511 Cc1cc(ccc1[N+](=O)[O-])n2c(cc3c2CC(CC3=O)C)C MS-8512 Cc1cc2c(n1c3ccc(c(c3)[N+](=O)[O-])Cl)CC(CC2=O)C MS-8513 c1ccc(cc1)COc2cccnc2NC(=O)Nc3ccccc3 MS-8514 c1ccc(cc1)COc2cccnc2NC(=O)Nc3ccccc3Oc4ccccc4 MS-8515 c1ccc(cc1)COc2cccnc2NC(=O)NS(=O)(=O)c3ccccc3 MS-8516 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc(cc3[N+](=O)[O-])Cl MS-8517 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)Br)/C#N MS-8518 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)[N+](=O)[O-])/C#N MS-8519 COCCNS(=O)(=O)c1ccccc1[N+](=O)[O-] MS-8520 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2c4ccc5c(c4)OCO5)C(=O)O MS-8521 c1ccc(c(c1)NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)Cl MS-8522 c1cc(cc(c1)Cl)NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F MS-8523 c1cc(ccc1NC(=S)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)[N+](=O)[O-] MS-8524 Cc1ccc(cc1)NC(=O)NCc2ccccc2Cl MS-8525 c1ccc(c(c1)CNC(=O)Nc2cccc(c2)Cl)Cl MS-8526 c1ccc(c(c1)CNC(=S)Nc2ccc(cc2)[N+](=O)[O-])Cl MS-8527 c1ccc(c(c1)CNC(=S)Nc2ccc(cc2)Cl)Cl MS-8528 c1ccc(c(c1)NC(=O)NNC(=O)c2ccncc2)Cl MS-8529 c1cnccc1C(=O)NNC(=O)NC2CCCCC2 MS-8530 CCc1ccc(cc1)OCC(=O)NNC(=O)NS(=O)(=O)c2ccc(cc2)C MS-8531 CCc1ccc(cc1)OCC(=O)NNC(=O)NS(=O)(=O)c2ccc(cc2)Cl MS-8532 Cc1ccc(cc1)S(=O)(=O)NC(=O)NNC(=O)COc2ccc(cc2)OC(F)(F)F MS-8533 c1ccc(c(c1)CNC(=O)Nc2cccc(c2)C(F)(F)F)Cl MS-8534 Cc1cc(no1)NC(=O)c2cccnc2C(=O)O MS-8535 COCCNC(=O)c1cccnc1C(=O)O MS-8536 c1cc(ccc1c2c([nH]nn2)C#N)Br MS-8537 CC(=O)Nc1ccc(cc1)S(=O)(=O)/N=C\2/N(CCS2)S(=O)(=O)c3ccc(cc3)NC(=O)C MS-8538 c1ccc(cc1)CCNS(=O)(=O)c2ccccc2N MS-8539 CCOC(=O)Nc1ccsc1C=O MS-8540 c1ccc(c(c1)CNC(=O)NC2CCCCC2)Cl MS-8541 Cc1ccccc1NC(=O)N2CCN(CC2)c3ccccn3 MS-8542 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3F MS-8543 CCOC(=O)Nc1c(ccs1)/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)C MS-8544 COc1cc(cc(c1)OC)NC(=O)NNC(=O)c2ccncc2 MS-8545 c1cc(c(cc1NC(=O)NNC(=O)c2ccncc2)Cl)Cl MS-8546 c1ccc2c(c1)c(c[nH]2)CCNC(=O)Nc3ccc(c(c3)Cl)Cl MS-8547 c1ccc2c(c1)c(c[nH]2)CCNC(=O)Nc3cc(ccc3Cl)Cl MS-8548 Cc1ccc(cc1)NC(=O)N2CCCN(CC2)C(=O)Nc3ccc(cc3)C MS-8549 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 MS-8550 c1ccc(c(c1)N2CCN(CC2)C(=S)Nc3ccc(cc3)[N+](=O)[O-])F MS-8551 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)Nc3ccc4c(c3)OCO4 MS-8552 c1cc(oc1)C(=O)N2CCN(CC2)C(=S)Nc3ccc(cc3)Cl MS-8553 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)Nc3ccc(c(c3)Cl)Cl MS-8554 c1cc(ccc1NC(=S)N2CCN(CC2)Cc3ccc4c(c3)OCO4)Cl MS-8555 c1cc2c(cc1CN3CCN(CC3)C(=O)Nc4ccc(c(c4)Cl)Cl)OCO2 MS-8556 CNC(=S)N1CCN(CC1)Cc2ccc3c(c2)OCO3 MS-8557 CCCNC(=O)N1CCCN(CC1)C(=O)NCCC MS-8558 C1CCC(CC1)NC(=O)N2CCCN(CC2)C(=O)NC3CCCCC3 MS-8559 c1ccc(cc1)NC(=O)NCc2ccccn2 MS-8560 c1cc(cnc1)CNC(=S)NC2CCCCC2 MS-8561 c1cnccc1CNC(=O)NC2CCCCC2 MS-8562 c1ccc(cc1)NC(=O)NCc2ccncc2 MS-8563 c1cnccc1CNC(=S)NC2CCCCC2 MS-8564 c1cc(sc1)CC(=O)NNC(=O)NC2CCCCC2 MS-8565 c1ccc(cc1)NC(=O)NNC(=O)Cc2cccs2 MS-8566 c1ccc(cc1)COc2ccc(cc2)C(=O)NNC(=O)NC3CCCCC3 MS-8567 c1ccc(cc1)COc2ccc(cc2)C(=O)NNC(=S)NC3CCCCC3 MS-8568 CCCCc1ccc(cc1)NC(=O)N2CCN(CC2)C=O MS-8569 C1CCC(CC1)NC(=O)N2CCN(CC2)C=O MS-8570 c1ccc(cc1)CNC(=O)N2CCN(CC2)C=O MS-8571 CCOc1ccc(cc1)NC(=O)N2CCN(CC2)C=O MS-8572 CCOC(=O)CNC(=O)N1CCN(CC1)C=O MS-8573 CCc1ccccc1NC(=O)N2CCN(CC2)C=O MS-8574 c1cc(ccc1NC(=O)N2CCN(CC2)C=O)F MS-8575 COc1ccc(cc1)NC(=O)N2CCN(CC2)C=O MS-8576 c1ccc2c(c1)cccc2NC(=O)N3CCN(CC3)C=O MS-8577 CC(C)(C)c1c2c(n(n1)C)-c3ccc(cc3C2=O)NC(=S)Nc4ccc(cc4)[N+](=O)[O-] MS-8578 c1ccc(c(c1)NS(=O)(=O)c2ccccc2[N+](=O)[O-])N3CCOCC3 MS-8579 c1ccc(cc1)NC2=NC(=O)CS2 MS-8580 CC(C)c1ccc(cc1)/C=N/c2ccc3c(c2)OCO3 MS-8581 COc1ccc(cc1)NC(=S)NNC(=O)c2ccccc2N MS-8582 c1ccc2c(c1)nc(s2)Sc3ccc(cc3C=O)[N+](=O)[O-] MS-8584 CC(C(=O)Nc1ccc(cc1)Br)Cl MS-8585 CC(C(=O)Nc1ccc(cc1)Cl)Cl MS-8586 c1ccc2c(c1)C(=O)C(=CNc3ccccc3Br)C2=O MS-8587 c1ccc(cc1)NC(=S)NNC(=O)CCC(=O)NNC(=S)Nc2ccccc2 MS-8588 CCCCNC(=O)Nc1cccc(c1)OC MS-8589 c1ccc2c(c1)c(c(s2)C(=O)Nc3cccc(c3)Br)Cl MS-8590 Cc1ccc(c(c1)NC(=O)c2c(c3ccccc3s2)Cl)C MS-8591 CN(C(=S)Nc1ccccc1)N MS-8592 COc1cc(ccc1OCc2ccc(cc2)[N+](=O)[O-])/C=C\3/c4ccccc4NC3=O MS-8593 c1ccc(cc1)C2Cc3c(c(n[nH]3)Nc4cccc(c4)C(F)(F)F)/C(=N/N)/C2 MS-8594 Cc1ccc(cc1)S(=O)(=O)NC(=O)NNC(=O)Cc2c[nH]c3c2cccc3 MS-8595 COc1ccc(cc1)n2c(nnc2S)Cc3c[nH]c4c3cccc4 MS-8597 Cc1ccc(cc1N2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC(C)C)Cl MS-8598 CC(C)Oc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccn3 MS-8599 Cc1ccccc1n2c(nnc2S)Cc3c[nH]c4c3cccc4 MS-8600 c1ccc(cc1)Cn2c(nnc2S)Cc3c[nH]c4c3cccc4 MS-8601 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4cccc5c4nccc5 MS-8602 CC(C)Oc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 MS-8603 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3cccc4c3nccc4 MS-8604 CC(C)Oc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccc3 MS-8605 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3cccc4c3nccc4 MS-8606 c1ccc(cc1)CNC(=S)NNC(=O)c2cccs2 MS-8607 c1ccc(cc1)Cn2c(nnc2S)c3cccs3 MS-8608 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)n3cncn3 MS-8609 COC(=O)c1c(ccs1)NC(=O)C2(CCCC2)c3ccccc3 MS-8610 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccccc3 MS-8611 CC(C)N(c1ccccc1)c2ccc(cc2)NC(=S)NC(=O)c3ccc(cc3)Cl MS-8612 CC(C)CC1CC(=CC(=O)C1)Nc2ccccc2I MS-8613 CC\1=NN(C(=O)/C1=C/c2ccc(c(c2)OC)OC)c3ccccc3 MS-8614 CCOc1ccc(cc1)/C=C/2\C(=NN(C2=O)c3ccccc3)C MS-8615 CC\1=NN(C(=O)/C1=C/c2cccs2)c3ccccc3 MS-8616 Cc1c(c(n(n1)c2ccccc2)O)C(c3ccc(cc3)[N+](=O)[O-])c4c(nn(c4O)c5ccccc5)C MS-8617 CCOC(=O)c1ccccc1NC(=O)Nc2ccccc2C MS-8620 Cc1ccccc1n2c(=O)c3ccccc3[nH]c2=O MS-8621 CC1(Cc2c(c(n[nH]2)Nc3cccc(c3)C(F)(F)F)/C(=N\N)/C1)C MS-8622 c1ccc(cc1)S(=O)(=O)/C(=C/c2cccc(c2)C(F)(F)F)/C#N MS-8623 CN(C)C(=O)n1c-2c(c(n1)c3cccs3)C(=O)c4c2cccc4 MS-8624 CCOC(=O)Nc1c(ccs1)/C=N/NC(=S)N MS-8625 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccc3c(c2)OCO3)/C#N MS-8626 c1ccc(cc1)CNC(=O)c2ccsc2 MS-8627 CC(c1ccccc1)NC(=O)c2ccsc2 MS-8628 COc1ccc(cc1)NC(=O)c2ccsc2 MS-8630 c1cc(ccc1C(F)(F)F)NC(=O)c2ccsc2 MS-8631 c1cscc1C(=O)N MS-8632 CC(=O)NC(Cc1ccccc1)C(=O)NCc2ccccc2 MS-8633 CC(=O)NC(Cc1ccccc1)C(=O)Nc2ccc(cc2)OC MS-8635 CCC(C)NC(=S)N1CCN(CC1)c2ccccn2 MS-8636 CCC(C)NC(=S)N1CCN(CC1)Cc2ccccc2 MS-8637 CCC(C)NC(=S)N1CCN(CC1)C(c2ccccc2)c3ccccc3 MS-8638 CCC(C)NC(=S)N1CCN(CC1)c2ccccc2 MS-8639 CCC(C)NC(=S)N1CCN(CC1)c2cc(ccc2C)Cl MS-8640 CCC(C)NC(=S)N1CCN(CC1)c2ccc(cc2)F MS-8641 CCC(C)NC(=S)N1CCN(CC1)C(=O)OCC MS-8642 CC1(CC(=C(C(=O)C1)C(=O)Nc2ccccc2)O)C MS-8643 COc1ccc(cc1)NC(=S)N2CCc3c2cccc3 MS-8644 CC1Cc2c(c(cn2CCC(=O)O)c3ccc(cc3)Br)C(=O)C1 MS-8646 Cc1c(c(n(n1)c2ccccc2)O)C(c3ccc(cc3)Cl)c4c(nn(c4O)c5ccccc5)C MS-8647 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccc(c2)OC MS-8648 c1ccc(cc1)n2c(n[nH]c2=O)COc3ccc(cc3)C(=O)O MS-8649 Cc1ccc(cc1)S(=O)(=O)/C(=C\c2c(cccc2Cl)Cl)/C#N MS-8650 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3)Cl)c4ccccc4 MS-8651 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cccc(c3)Cl)c4ccccc4 MS-8653 Cc1ccccc1NC(=S)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8655 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cccc4c3cccc4)c5ccccc5 MS-8657 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3OC)OC)c4ccccc4 MS-8658 Cc1ccc(c(c1)C)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8659 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cc(cc(c3)Cl)Cl)c4ccccc4 MS-8660 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(c(c3)Cl)Cl)c4ccccc4 MS-8661 Cc1ccc(cc1NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)F MS-8662 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cccc(c3)C(F)(F)F)c4ccccc4 MS-8663 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccccc3Cl)c4ccccc4 MS-8664 Cc1cccc(c1C)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8665 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3Cl)Cl)c4ccccc4 MS-8667 Cc1cc(cc(c1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)C MS-8668 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3c(cccc3Cl)Cl)c4ccccc4 MS-8671 Cc1cccc(c1NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)C MS-8672 Cc1ccc(cc1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-8674 CN1c2ccccc2C(=NC(C1=O)NC(=O)NCc3ccc(c(c3)Cl)Cl)c4ccccc4 MS-8675 CCOc1ccc(cc1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8682 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3)SC)c4ccccc4 MS-8683 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(c(c3)F)F)c4ccccc4 MS-8684 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cc(cc(c3)F)F)c4ccccc4 MS-8685 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cccc(c3)SC)c4ccccc4 MS-8687 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3C(F)(F)F)Cl)c4ccccc4 MS-8688 CN1c2ccccc2C(=NC(C1=O)NC(=O)NCC=C)c3ccccc3 MS-8690 CCOC(=O)NC(=O)NC1C(=O)N(c2ccccc2C(=N1)c3ccccc3)C MS-8692 CN1c2ccccc2C(=NC(C1=O)NC(=O)NC3CCCC3)c4ccccc4 MS-8694 CN1c2ccccc2C(=NC(C1=O)NC(=O)NCc3ccc(cc3Cl)Cl)c4ccccc4 MS-8695 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)NC(C)C)c4ccccc4 MS-8696 CCCCCCNC(=O)NC1C(=O)N(c2ccccc2C(=N1)c3ccccc3)CC(=O)c4ccccc4C MS-8697 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)NC4CCCC4)c5ccccc5 MS-8698 CCc1cccc(c1NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)C MS-8702 CCOC(=O)CCNC(=O)NC1C(=O)N(c2ccccc2C(=N1)c3ccccc3)C MS-8704 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cccc(c3)SC(F)(F)F)c4ccccc4 MS-8705 Cc1ccccc1CNC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8706 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(c(c3)Cl)F)c4ccccc4 MS-8708 Cc1ccc(cc1Cl)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8709 CC1=C(C(=O)CC(C1)(C)C)C(c2ccc(cc2)F)C3=C(CC(CC3=O)(C)C)O MS-8711 Cc1cc(nc(n1)NC(=O)c2c(onc2c3c(cccc3Cl)F)C)C MS-8712 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCC=C MS-8713 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCCc3ccc(c(c3)OC)OC MS-8714 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCC#C MS-8715 COc1ccc(cc1)NC(=S)N2CCN(CC2)C(=S)Nc3ccc(cc3)OC MS-8716 COc1ccc(cc1)NC(=S)Nc2ccsc2C(=O)OC MS-8717 COc1ccc(cc1)NC(=S)NNC(=S)Nc2ccccc2 MS-8718 CCOC(=O)c1c2c(sc1NC(=O)C(C(C(C(=O)O)(F)F)(F)F)(F)F)CCCC2 MS-8719 COC(=O)c1ccccc1NC(=O)C(C(C(C(=O)O)(F)F)(F)F)(F)F MS-8720 CC(C)(C)C\1=NN(C(=O)/C1=C\c2c[nH]c3c2cccc3)c4ccccc4 MS-8721 c1ccc(cc1)C(=O)/C(=C/c2c[nH]c3c2cccc3)/C#N MS-8722 c1ccc2c(c1)c(c[nH]2)CC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-8723 Cc1ccsc1C(=O)NCCc2ccc(c(c2)OC)OC MS-8724 CC(C)(C)C1=NN(C(=O)C1=Cc2cc(c(c(c2)OC)O)OC)c3ccccc3 MS-8725 Cc1c(c(no1)c2ccccc2Cl)C(=O)N(C)c3ccc(cc3)O MS-8726 c1cc2cccnc2c(c1)Oc3ccc(cc3C#N)[N+](=O)[O-] MS-8727 CCC(CC)(C#C)NC(=O)c1c(onc1c2c(cccc2Cl)Cl)C MS-8728 c1ccc2c(c1)C(=O)C(=CNc3ccc(cc3)C(=O)O)C2=O MS-8729 Cc1cccc(c1C(=O)O)NC=C2C(=O)c3ccccc3C2=O MS-8730 CC(=O)Nc1ccc(cc1)c2csc(n2)NC(=S)N MS-8731 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCC=C MS-8732 Cc1ccc(cc1C#N)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C MS-8733 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)Nc4cccc(c4)C(=O)O MS-8734 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)C(=NOC(=O)c4c(onc4c5c(cccc5Cl)Cl)C)C MS-8735 c1ccc2c(c1)nc(s2)SCC(=O)NNC(=S)NC3CCCCC3 MS-8736 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc(cc2)Sc3c(cc(cn3)C(F)(F)F)Cl)CC(=O)OC MS-8737 c1cc(ccc1S(=O)(=O)C/C(=N\OC(=O)C(F)(F)F)/N)Cl MS-8738 CC(C(=O)Nc1nc2c(s1)C(=O)CC(C2)c3ccccc3)Sc4ccc(cc4)Cl MS-8739 CC(C)(C)C\1=NN(C(=O)/C1=C\c2cc(c(c(c2)OC)O)OC)c3c(cc(cn3)C(F)(F)F)Cl MS-8740 c1cc(ccc1C(C(F)(F)F)(C(F)(F)F)O)NC(=O)C2CC2C(=O)O MS-8741 c1ccc2c(c1)ccc3c2sc(c3Cl)C(=O)Nc4ccc(cc4)OC(F)(F)F MS-8742 c1ccc2c(c1)ccc3c2sc(c3Cl)C(=O)Nc4ccc(cc4)Sc5c(cc(cn5)C(F)(F)F)Cl MS-8743 CC1=NN(C(=O)C1/C(=N/O)/c2ccccc2)c3ccccc3 MS-8744 CC1=NN(C(=O)C1/C(=N\NC(=S)Nc2ccccc2)/c3ccccc3)c4ccccc4 MS-8745 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)\N MS-8746 CCc1ccc(cc1)OCc2n[nH]c(=S)n2c3ccccc3 MS-8747 c1cc(ccc1NC(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl MS-8748 c1cc(c(cc1NC(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl MS-8749 CN1c2ccccc2/C(=N/NC(=S)Nc3ccccc3)/C1=O MS-8750 CN1c2ccccc2/C(=N/c3cc(cc(c3)Cl)Cl)/C1=O MS-8751 COc1ccc(cc1OC)/C=C/c2c(=O)[nH]c3ccccc3n2 MS-8752 CC(C)(C)c1c2c(n(n1)c3ccc(cn3)C(F)(F)F)-c4ccccc4C2=O MS-8753 c1ccc(cc1)C2=NCCc3c2[nH]c4c3cccc4 MS-8754 CC(C)c1cc(=O)n([nH]1)C(=S)N MS-8755 CC(C)(C)c1c2c(n(n1)C(=O)C3CC3)-c4ccccc4C2=O MS-8756 CC(C)(C)C(=O)/C(=C/c1cccc(c1)C(F)(F)F)/C#N MS-8757 CN(c1ccc(cc1)O)S(=O)(=O)c2ccc3ccccc3c2 MS-8758 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C MS-8759 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(cc3)OC(F)(F)F MS-8760 CN(C)c1ccc(cc1)c2[nH]c(=O)c3c(n2)c(=N)n(c(=O)[nH]3)c4cccc(c4)C(F)(F)F MS-8761 c1ccc2c(c1)c(c[nH]2)CCNC(=O)COc3ccc(cc3)[N+](=O)[O-] MS-8762 c1ccc2c(c1)cccc2Nc3nc(cs3)c4cccc(c4)[N+](=O)[O-] MS-8763 c1ccc(cc1)Nc2nc(cs2)c3cccc(c3)[N+](=O)[O-] MS-8764 CCc1ccc(cc1)c2csc(n2)Nc3cccc4c3cccc4 MS-8765 CCc1ccc(cc1)c2csc(n2)Nc3ccccc3Cl MS-8766 Cc1cc(ccc1Cl)c2csc(n2)Nc3ccncc3 MS-8767 COc1ccc(cc1Nc2nc(cs2)c3cccc(c3)[N+](=O)[O-])Cl MS-8768 Cc1c(nc(s1)Nc2cc(ccc2OC)Cl)/C(=N/O)/C MS-8769 CCOC(=O)c1c(nc(s1)Nc2cc(ccc2OC)Cl)C MS-8770 c1cc(cc(c1)Cl)NC=C2C(=O)NC(=O)NC2=O MS-8771 c1cc(sc1)C(=O)NNC(=O)Nc2ccc(cc2)C(F)(F)F MS-8772 c1ccc2cc(ccc2c1)c3csc(n3)Nc4cccc5c4cccc5 MS-8773 c1ccc2cc(ccc2c1)c3csc(n3)Nc4cccnc4 MS-8774 CCOc1ccc(cc1)NC2=C(C(=O)c3c2cccc3)c4ccc5c(c4)OCO5 MS-8775 COC(=O)CNC(=O)C=Cc1cc2c(cc1[N+](=O)[O-])OCO2 MS-8776 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3)OC(F)(F)F MS-8777 c1cc(ccc1C(F)(F)F)NC(=O)N2CCN(CC2)c3ccc(cc3)F MS-8778 c1cc(ccc1NC(=O)N2CCN(CC2)c3ccc(cc3)F)OC(F)(F)F MS-8779 c1ccc2c(c1)c(=O)[nH]c(n2)SCC(=O)Nc3ccc4c(c3)OCO4 MS-8780 CN(C)c1ccc(cc1)/C=N/O MS-8781 CCOc1ccc2c(c1)sc(n2)NS(=O)(=O)c3ccc(cc3)NC(=O)C MS-8782 COc1cc2c(cc1OC)C(=O)/C(=C/C=C/c3ccccc3)/C2 MS-8783 CC(C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Oc2ccc3ccccc3c2 MS-8784 CC1(Cc2cccc(c2O1)OCC(=O)NC(=O)Nc3ccccc3)C MS-8785 c1cc2cccnc2c(c1)NS(=O)(=O)c3cccc4c3nccc4 MS-8786 CCOC(=O)c1c(oc2c1C(=O)CC(C2)(C)C)C MS-8787 Cc1cc(ccc1Cl)c2csc(n2)Nc3ccc(cc3)C#N MS-8788 CC1(Cc2cccc(c2O1)OCc3ccc(cc3)[N+](=O)[O-])C MS-8789 CSc1[nH]nc(n1)NC(=O)/C=C/c2ccccc2 MS-8790 CC1Cc2c(sc(n2)NC(=O)/C=C/c3ccccc3)C(=O)C1 MS-8791 c1cc(c(cc1NC(=O)Nc2ccc(c(c2)Cl)Cl)Cl)Cl MS-8792 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3)CBr MS-8793 CCOC(=O)Cn1c(c(nn1)c2ccc3c(c2)OCO3)C#N MS-8794 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3)Br MS-8795 c1ccc2c(c1)c(c[nH]2)CCNC(=O)COc3cccc(c3)C(F)(F)F MS-8796 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccccc3[N+](=O)[O-] MS-8797 c1cc2cccnc2c(c1)Oc3c(cc(cn3)C(F)(F)F)Cl MS-8798 Cc1cc(no1)NC(=O)c2ccc(cc2)[N+](=O)[O-] MS-8799 c1cc(c(cc1F)F)/N=C/2\c3cc(ccc3NC2=O)Br MS-8800 CC1CC(=O)C(C(=O)C1)CC(=O)c2ccc(cc2)c3ccccc3 MS-8801 c1ccc(cc1)c2ccc(cc2)c3csc([nH+]3)Nc4ccccc4.[Br-] MS-8802 Cc1nc(=O)[nH]n1c2ccccc2 MS-8803 CC1(Cc2cccc(c2O1)Oc3ccc(cn3)C(F)(F)F)C MS-8804 c1cc(ccc1NC(=O)C2CC2C(=O)O)Br MS-8805 c1cc(ccc1C(=O)N)Oc2ccc(cn2)C(F)(F)F MS-8806 Cc1ccc(c(c1)C)OCC(=O)NNC(=S)NC2CCCCC2 MS-8807 Cc1cccc(c1C)OCC(=O)n2cnc(n2)N MS-8808 CC1(CC2=C(C(Nc3ccccc3N2)c4ccccc4F)C(=O)C1)C MS-8809 CC1(CC(=CC(=O)C1)N2CCN(CC2)c3ccccc3F)C MS-8810 CC1CC2=C(C(Nc3ccccc3N2)c4c(cccc4Cl)F)C(=O)C1 MS-8811 c1cc(ncc1Br)NC=C(C#N)C#N MS-8812 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl MS-8813 Cc1ccc2c(c1)NC(C3=C(N2)CC(CC3=O)(C)C)c4c(cccc4Cl)F MS-8814 CC1(CC2=C(C(Nc3ccc(cc3N2)C(=O)O)c4ccccc4F)C(=O)C1)C MS-8815 Cc1ccc(cc1)C(=Nc2nc[nH]n2)C3C(=O)c4ccccc4C3=O MS-8816 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)OC(F)(F)F MS-8817 c1ccc(cc1)NC(=O)NCCc2c[nH]c3c2cccc3 MS-8818 c1ccc2c(c1)c(c[nH]2)CCNC(=O)Nc3ccc(cc3)Cl MS-8819 CC1(OC(=O)C(=CNc2cccc3c2nccc3)C(=O)O1)C MS-8820 c1cc(cc(c1)Oc2ccc(cc2C=O)[N+](=O)[O-])C(F)(F)F MS-8821 c1cc(cc(c1)Oc2ccc(cc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-])C(F)(F)F MS-8822 Cc1ccc(cc1)S(=O)(=O)CC(=O)CCl MS-8823 COc1cccc(c1)C(=O)O/N=C(\c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F)/N MS-8824 c1cc(cc(c1)Oc2ccc(cc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)OC(F)(F)F)[N+](=O)[O-])C(F)(F)F MS-8825 COc1cccc(c1Oc2c(cc(cn2)C(F)(F)F)Cl)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)OC(F)(F)F MS-8826 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)Nc3ccc(cc3)Cl MS-8827 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3cccc(c3)C(F)(F)F MS-8828 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-8829 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl MS-8830 Cc1ccc(c(c1)C)Oc2c(cccn2)C(=O)Nc3cc(on3)C MS-8831 Cc1ccc(c(c1)C)Oc2c(cccn2)C(=O)Nc3cccc4c3nccc4 MS-8832 Cc1ccc(c(c1)C)Oc2c(cccn2)C(=O)NCCc3ccccc3 MS-8833 CC(C)(C)C(=O)/C(=C\c1cc(ccc1Sc2ccccn2)[N+](=O)[O-])/C#N MS-8834 CC(C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)Sc2[nH]c(=O)c3ccccc3n2 MS-8835 c1c(cc(cc1C(F)(F)F)NC(=O)c2c(c(c(c(c2Cl)Cl)Cl)Cl)C(=O)O)C(F)(F)F MS-8836 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)Nc3ccc(cn3)Br MS-8837 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccc(cc2Cl)Cl MS-8838 COC(=O)c1c(ccs1)NC(=O)C(=O)c2c[nH]c3c2cccc3 MS-8839 CCOC(=O)C(c1ccccc1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl MS-8840 c1cc(c(cc1F)F)NC=C2C(=O)CCCC2=O MS-8841 c1cc(ccc1NC(=S)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)Cl MS-8842 COc1cccc(c1OC)c2nc(no2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F MS-8843 COC(=O)CSc1ccc(c(c1)C#N)[N+](=O)[O-] MS-8844 Cc1c(c(c(c(c1F)F)N2C(=O)C(=CC=Cc3ccc(cc3)OC)C(=N2)C)F)F MS-8845 Cc1ccc2cccc(c2n1)Oc3ccc(c(c3)C#N)[N+](=O)[O-] MS-8846 Cc1ccc(cc1)S(=O)(=O)NNC2=CC(=O)c3c2cccc3 MS-8847 c1cc(ccc1[NH2+]C=CC=Nc2ccc(cc2)OC(F)(F)F)OC(F)(F)F.[Cl-] MS-8848 c1ccc2c(c1)C=CC(=O)C2=CNc3ccc(cc3)OC(F)(F)F MS-8849 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-8850 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2cccc(c2)C(F)(F)F MS-8851 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2cccnc2 MS-8852 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2cccnc2Cl MS-8853 CC(=O)Nc1cccc(c1)OCc2c(c(=O)n(n2C)c3ccccc3)Br MS-8854 COc1cc(c(cc1OC)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)CC(=O)OC MS-8855 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)[N+](=O)[O-] MS-8856 c1ccc(cc1)C2CC3=C(C(Nc4ccccc4N3)c5cccc(c5)OC(F)(F)F)C(=O)C2 MS-8857 Cc1c(nc(s1)NC=C2C(=O)OC(OC2=O)(C)C)c3ccc(cc3)Br MS-8858 Cc1c(nc(s1)NC=C2C(=O)c3ccccc3C2=O)c4ccc(cc4)Br MS-8859 Cc1c(c(c(c(c1F)F)N2C(=O)CC(=N2)C)F)F MS-8860 Cc1cc(c2ccccc2c1C)OC(=O)C MS-8861 CCOC(=O)c1ccc(cc1)OCc2c(c(=O)n(n2C)c3ccccc3)Br MS-8862 Cc1cc(ccc1C(C)C)NC(=O)c2c(onc2c3ccccc3Cl)C MS-8863 c1cc(c(cc1C(=O)/C(=C\Nc2c(cc(cn2)C(F)(F)F)Cl)/C#N)Cl)Cl MS-8864 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccccc3[N+](=O)[O-] MS-8865 CC1(C(=C)SC(=N1)Nc2ccc(cc2)OC(F)(F)F)C MS-8866 CC1(Cc2cccc(c2O1)Oc3ccc(cc3C4C5=C(CC(CC5=O)(C)C)Nc6ccccc6N4)[N+](=O)[O-])C MS-8867 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC(=O)NN MS-8868 CCOC(=O)C1=C(OCC1=O)Nc2ccc(cc2)Cl MS-8869 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3cccc4c3cccc4 MS-8870 CC1(CC2=C(C(Nc3c(cccn3)N2)c4c[nH]c5c4cccc5)C(=O)C1)C MS-8871 Cc1cc(ccc1Oc2c(cccn2)C(=O)O)Cl MS-8872 Cc1cc(ccc1Oc2c(cccn2)C(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F)Cl MS-8873 CCC(CC)(C#C)NC(=O)c1c(onc1c2c(cccc2Cl)F)C MS-8874 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3ccc(cc3)OC(F)(F)F)C MS-8875 c1cc(ccc1N/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl)Sc3c(cc(cn3)C(F)(F)F)Cl MS-8876 CC1(C(=C)SC(=N1)Nc2ccc(cc2)Sc3c(cc(cn3)C(F)(F)F)Cl)C MS-8877 CC1(CC2=C(C(Nc3ccc(cc3N2)C(=O)O)c4cccs4)C(=O)C1)C MS-8878 CC(C(=O)Nc1nc2c(s1)C(=O)CC(C2)(C)C)Sc3ccc(cc3)Cl MS-8879 CC(=C1C(=O)c2ccccc2C1=O)NNc3c(cc(cn3)C(F)(F)F)Cl MS-8880 CN1CCN(CC1)C(=O)Nc2ccc(cc2)Cl MS-8881 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC(=O)NNC(=S)Nc4ccc(cc4)OC(F)(F)F MS-8882 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(nc2)OC)/C#N MS-8883 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCc4n[nH]c(=S)n4c5ccc(cc5)OC(F)(F)F MS-8884 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C(=O)c3ccc(nc3Cl)Cl MS-8885 Cc1ccc(cc1)S(=O)(=O)/C(=C\N2CCN(CC2)c3cc(ccc3C)Cl)/C#N MS-8886 CCOC(=O)/C(=C\N1CCN(CC1)c2cc(ccc2C)Cl)/C#N MS-8887 Cc1ccc(cc1N2CCN(CC2)C(=O)C3CC3C(=O)O)Cl MS-8888 c1ccc2c(c1)C(=O)NC(N2)c3ccc(cc3)OC(F)F MS-8889 Cc1cccc(c1)Oc2ccc(cc2C3C4=C(CC(CC4=O)(C)C)Nc5ccccc5N3)[N+](=O)[O-] MS-8890 COc1ccc(cc1OC)C=C(C#N)C#N MS-8891 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc4ccccc4c3)C(=O)C1)C MS-8892 c1ccc(cc1)C2CC3=C(C(C(=C(O3)N)C#N)c4cccs4)C(=O)C2 MS-8893 CCOc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)OC(=C2C(=O)C(C)(C)C)N MS-8894 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)OC(F)(F)F)C(=O)C1)C MS-8895 CC1CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)OC(F)(F)F)C(=O)C1 MS-8896 CSc1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N MS-8897 CC1(CC2=C(C(Nc3ccccc3N2)c4ccc(c(c4)[N+](=O)[O-])O)C(=O)C1)C MS-8898 c1ccc(cc1)Nc2nc(cs2)c3ccc(cc3)F MS-8899 COc1ccc(cc1)Nc2[nH+]c(cs2)c3ccc(cc3)F.[Br-] MS-8900 c1ccc2cc(ccc2c1)S(=O)(=O)Nc3ccc(cc3)Sc4c(cc(cn4)C(F)(F)F)Cl MS-8901 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C(=O)C(C(C(F)(F)F)(F)F)(F)F MS-8902 c1cc(c(nc1)Cl)C(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-8903 CC1CC(=CC(=O)C1)NN(C)c2ccc(cn2)C(F)(F)F MS-8904 CC(=O)c1ccccc1OCc2c(c(=O)n(n2C)c3ccccc3)Br MS-8905 CN(c1ccc(cn1)C(F)(F)F)NC2=CC(=O)CC(C2)c3ccccc3 MS-8906 c1ccc2c(c1)c(c[nH]2)C(=O)C(=O)N3CCCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl MS-8907 c1ccc2cc(ccc2c1)S(=O)(=O)NCc3ccncc3 MS-8908 Cc1cc(ccc1C(C)C)NC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-8909 CC(C)(C)C1=NN(C(=O)C1C(c2ccc(cc2)C#N)C3C(=NN(C3=O)C)C(C)(C)C)C MS-8910 c1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2)Br MS-8911 Cc1cc(cc(c1Br)C)OCC(=O)NN MS-8912 Cc1cc(cc(c1Br)C)OCC(=O)NNC(=O)Nc2ccc(cc2)C(F)(F)F MS-8913 c1ccc(cc1)n2c(n[nH]c2=S)COc3ccc(cc3)Br MS-8914 Cc1cc(cc(c1Br)C)OCC(=O)NNC(=S)Nc2ccccc2 MS-8915 Cc1cc(cc(c1Br)C)OCc2n[nH]c(=S)n2c3ccccc3 MS-8916 Cc1ccc(cc1)c2csc(n2)Nc3cccc4c3cccc4 MS-8917 c1ccc(cc1)C(=O)/C=C/c2ccc(cc2)[N+](=O)[O-] MS-8921 CCCCCC(=O)n1c(cc(n1)c2ccc3ccccc3c2)C(F)(F)F MS-8922 c1ccc(cc1)n2c(=N)c(c([nH]c2=O)C#N)/N=C/c3cccc(c3)C(F)(F)F MS-8923 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)NCc3ccc(cc3)F)C MS-8924 CCN1C(=O)/C(=C/c2coc3c(c2=O)cc(cc3Cl)Cl)/SC1=S MS-8925 c1ccc(cc1)NC(=S)N/N=C\2/c3cc(ccc3NC2=O)Cl MS-8926 c1cc(ccc1/N=C\2/c3cc(ccc3NC2=O)I)OC(F)(F)F MS-8927 c1cc2c(cc1I)/C(=N/NC(=O)c3ccncc3)/C(=O)N2 MS-8928 CC1(CC2=C(C(Nc3ccc(cc3N2)C(=O)OC)c4cccnc4)C(=O)C1)C MS-8929 CC(=O)/C(=C\Nc1ccc(cc1)OC(F)(F)F)/C(=O)Nc2ccccc2 MS-8930 c1ccnc(c1)C(=O)N2CCN(CC2)c3ncccn3 MS-8931 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccccc3F)N MS-8932 c1cc(cc(c1)OC(F)(F)F)CNC(=O)C2CC2C(=O)O MS-8933 COC(=O)c1c(ccs1)NC(=S)N2CCN(CC2)c3ccccc3F MS-8934 c1ccc(cc1)N2CCN(CC2)C(=O)c3cccnc3Cl MS-8935 CCCCOc1ccc(cc1)/C=N/C(=C(/C#N)\N)/C#N MS-8936 CCCCOc1ccc(cc1)/C=N/c2c([nH]c(=O)n(c2=N)c3ccc(cc3)Cl)C#N MS-8937 c1ccc(cc1)C(=O)/C(=C/c2ccco2)/C#N MS-8938 c1ccc(cc1)C(=O)/C(=C/c2c(cccc2Cl)Cl)/C#N MS-8939 c1ccc2c(c1)C(=O)C(=CNc3nc(cs3)c4cccc(c4)[N+](=O)[O-])C2=O MS-8940 c1ccc(cc1)/C=C/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Br MS-8941 c1ccc(cc1)CS/C(=N\N=C\c2ccccc2O)/[NH3+].[Cl-] MS-8942 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 MS-8943 CC(=O)c1cc2c(cc1N/C=C(/C#N)\S(=O)(=O)c3ccccc3)OCO2 MS-8944 CC(=O)Nc1ccc(cc1)c2csc(n2)NC=C3C(=O)c4ccccc4C3=O MS-8945 c1ccc2cc(ccc2c1)/C=N/O MS-8946 c1cc(c(c(c1)Cl)Cl)/C=N/O MS-8947 c1ccc2c(c1)cc3ccccc3c2/C=N/O MS-8948 COc1cccc(c1OC)/C=N/O MS-8949 COc1ccc(c(c1)OC)/C=N/O MS-8950 c1cc(ccc1/C=N/O)F MS-8951 c1cc(c(cc1/C=N/O)Cl)Cl MS-8952 c1ccc(c(c1)/C=N/O)Br MS-8953 c1cc(cc(c1)Br)/C=N/O MS-8954 c1cc(c(c(c1)Cl)/C=N/O)F MS-8955 CCN(CC)c1ccc(cc1)/C=N/O MS-8956 c1cc(cc(c1)C#N)/C=C/C(=O)O MS-8957 COc1ccc(c(c1OC)OC)/C=C/C(=O)O MS-8958 COc1cccc(c1OC)/C=C/C(=O)O MS-8959 c1ccc(cc1)NC(=S)NNC(=O)c2ccccc2Cl MS-8961 COc1cc(cc(c1O)OC)/C=C/C(=O)O MS-8962 COc1cc(cc(c1OC)OC)/C=C/C(=O)OC MS-8964 CCOC(=O)C(Cc1ccccc1)NC(=O)Nc2ccc(nc2)OC MS-8965 CCCCCCCC(=O)Oc1ccc(cc1)[N+](=O)[O-] MS-8966 COC(=O)c1cccs1 MS-8967 Cc1ccccc1/C=C/C(=O)O MS-8968 Cc1cc(cc2c1NC(=O)C2=O)Cl MS-8969 c1cc(c(cc1F)N)N MS-8972 c1cc(sc1)C(=O)NCc2ccncc2 MS-8973 c1ccc2c(c1)c(c(s2)C(=O)Nc3cccc(c3)I)Cl MS-8974 CC(C)(C)c1ccc(cc1)NC(=O)c2c(c3ccccc3s2)Cl MS-8975 c1cc(ccc1/C=N/O)C#N MS-8977 COc1ccc(cc1)NC(=O)N MS-8978 c1cc(c(cc1C(=O)N)Cl)Cl MS-8979 c1cc(c(cc1/C=C/C(=O)O)Br)O MS-8980 c1cc(c(cc1/C=C/C(=O)O)F)O MS-8981 COc1cc(cc(c1OC)OC)C(=O)N/N=C\2/CC(=O)c3c2cccc3 MS-8983 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3ccccn3)C MS-8984 CCOC(=O)CCNC(=O)Nc1ccc(cn1)Br MS-8985 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)OC(F)(F)F MS-8986 Cc1cc(ccc1Br)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8987 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(c(c3)C(F)(F)F)F)c4ccccc4 MS-8988 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(c(c3)C(F)(F)F)Cl)c4ccccc4 MS-8989 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc4c(c3)CCC4)c5ccccc5 MS-8990 Cc1ccc(cc1F)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8991 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(c(c3)Cl)OC)c4ccccc4 MS-8992 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc4c(c3)OCO4)c5ccccc5 MS-8993 Cc1ccc(cc1[N+](=O)[O-])NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-8994 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(c(c3)[N+](=O)[O-])Cl)c4ccccc4 MS-8995 CCNC(=O)NC1C(=O)N(c2ccccc2C(=N1)c3ccccc3)C MS-8996 CCCCNC(=O)N[C@@H]1C(=O)N(c2ccccc2C(=N1)c3ccccc3)C MS-8997 CC(C)(C)NC(=O)NC1C(=O)N(c2ccccc2C(=N1)c3ccccc3)C MS-8998 CN1c2ccccc2C(=NC(C1=O)NC(=O)NC34CC5CC(C3)CC(C5)C4)c6ccccc6 MS-8999 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)NC3CCCCC3)c4ccccc4 MS-9000 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)NCc3ccccc3)c4ccccc4 MS-9001 CN1c2ccccc2C(=NC(C1=O)NC(=O)NCCc3ccccc3)c4ccccc4 MS-9002 CN1c2ccccc2C(=NC(C1=O)NC(=O)NCc3ccccc3F)c4ccccc4 MS-9003 CN1c2ccccc2C(=NC(C1=O)NC(=O)NCc3cccc(c3)F)c4ccccc4 MS-9004 CCCc1ccccc1NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9005 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccccc4SC)c5ccccc5 MS-9006 CCc1cccc(c1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9007 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cccc(c4)SC)c5ccccc5 MS-9008 Cc1ccccc1C(=O)CN2c3ccccc3C(=N[C@@H](C2=O)NC(=O)Nc4ccc(cc4)[N+](=O)[O-])c5ccccc5 MS-9009 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cc(ccc4Cl)C(F)(F)F)c5ccccc5 MS-9010 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(c(c4)C(F)(F)F)Cl)c5ccccc5 MS-9011 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)NCc4ccccc4)c5ccccc5 MS-9012 CC(C)c1ccccc1NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9013 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccccc3F)c4ccccc4 MS-9014 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccccc3Br)c4ccccc4 MS-9015 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccccc3[N+](=O)[O-])c4ccccc4 MS-9016 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccccc3OC(F)(F)F)c4ccccc4 MS-9017 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccccc3Oc4ccccc4)c5ccccc5 MS-9018 CCc1cccc(c1)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9019 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cccc(c3)[N+](=O)[O-])c4ccccc4 MS-9020 CC(=O)c1cccc(c1)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9021 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cccc(c3)Oc4ccccc4)c5ccccc5 MS-9022 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cccc(c3)F)c4ccccc4 MS-9023 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cccc(c3)C#N)c4ccccc4 MS-9024 CCc1ccc(cc1)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9025 CC(C)c1ccc(cc1)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9026 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3)C#N)c4ccccc4 MS-9027 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3)Br)c4ccccc4 MS-9028 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3)Oc4ccccc4)c5ccccc5 MS-9029 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3)OCc4ccccc4)c5ccccc5 MS-9030 CC(=O)c1ccc(cc1)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9031 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3)[N+](=O)[O-])c4ccccc4 MS-9032 Cc1c(cccc1Cl)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9033 Cc1c(cccc1[N+](=O)[O-])NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9034 CCc1cccc(c1NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)CC MS-9035 Cc1ccc(cc1NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)Cl MS-9036 Cc1ccc(cc1NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)[N+](=O)[O-] MS-9037 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cc(ccc3F)C(F)(F)F)c4ccccc4 MS-9038 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cc(ccc3F)F)c4ccccc4 MS-9039 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cc(ccc3Cl)C(F)(F)F)c4ccccc4 MS-9040 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cc(ccc3[N+](=O)[O-])Cl)c4ccccc4 MS-9041 Cc1ccc(c(c1)NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)OC MS-9042 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cc(ccc3OC)[N+](=O)[O-])c4ccccc4 MS-9043 Cc1cc(ccc1NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)Cl MS-9044 Cc1cc(ccc1NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)[N+](=O)[O-] MS-9045 Cc1cc(ccc1NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)OC MS-9046 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3F)F)c4ccccc4 MS-9047 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3F)Br)c4ccccc4 MS-9048 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3Cl)Br)c4ccccc4 MS-9049 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3C(F)(F)F)F)c4ccccc4 MS-9050 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3C(F)(F)F)Br)c4ccccc4 MS-9051 Cc1ccc(c(c1)[N+](=O)[O-])NC(=O)N[C@@H]2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C MS-9052 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3[N+](=O)[O-])OC)c4ccccc4 MS-9053 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3ccc(cc3OC)[N+](=O)[O-])c4ccccc4 MS-9054 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cc(cc(c3)F)C(F)(F)F)c4ccccc4 MS-9055 CN1c2ccccc2C(=N[C@@H](C1=O)NC(=O)Nc3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-])c4ccccc4 MS-9056 CCOC(=O)Nc1c(ccs1)/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)OC(F)(F)F MS-9057 CCOC(=O)Cc1csc(n1)NC(=S)N MS-9058 CC(C)(C)c1ccc(cc1)S(=O)(=O)CC(=O)N MS-9059 Cc1cc(ccc1C(C)C)NS(=O)(=O)c2cccc3c2nccc3 MS-9060 COc1ccc(cc1OC)CCNS(=O)(=O)c2cccc3c2nccc3 MS-9061 Cc1cc(nc(n1)NC=C2C(=O)OC(OC2=O)(C)C)C MS-9062 CCc1cccc2c1[nH]cc2C(CC(=O)c3ccc(cc3)C(C)(C)C)C(=O)O MS-9063 Cc1cc(nc(n1)N)Oc2cccc3c2OC(C3)(C)C MS-9064 CCC(=C1C(=O)c2ccccc2C1=O)Nc3cccc4c3nccc4 MS-9065 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=N/C(=C(/C#N)\N)/C#N MS-9066 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=N/c2c([nH]c(=O)n(c2=N)c3ccccc3)C#N MS-9067 c1cc(ccc1CNS(=O)(=O)c2cc(ccc2Cl)Cl)F MS-9068 CCN(CC)c1ccc(cc1)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C MS-9069 c1ccc(cc1)Oc2ccc(cc2)Nc3c(c(c(c(c3F)F)C(F)(F)F)F)F MS-9070 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)C(C(F)(F)F)(C(F)(F)F)O MS-9071 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc4c(cc3C(=O)C)OCO4 MS-9072 c1ccc2c(c1)C(=O)C(=Cc3coc4c(c3=O)cc(cc4Cl)Cl)C2=O MS-9073 CC(=C1C(=O)c2ccccc2C1=O)Nc3c(cccn3)N MS-9074 c1c(cc(c2c1c(=O)c(co2)/C=N/NC(=S)N)Cl)Cl MS-9075 COc1ccc(cc1OC)c2[nH]c3cccnc3n2 MS-9076 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3ccc(cc3)N(C)C MS-9077 c1ccc(cc1)Oc2cccc(c2)c3[nH]c(=O)c4c(n3)c(=N)n(c(=O)[nH]4)c5cccc(c5)C(F)(F)F MS-9078 CN(C)c1cccc(c1)OCc2nnc(n2c3ccccc3)S MS-9079 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3cc(cc(c3)Cl)Cl)C MS-9080 CC1(C(NC(S1)c2cccc(c2)Oc3ccccc3)C(=O)O)C MS-9081 CCSc1c(cccn1)C(=O)Nc2ccc(cc2)OC(F)(F)F MS-9082 CCSc1c(cccn1)C(=O)Nc2cccc3c2nccc3 MS-9083 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)Nc2cccc(c2)C(F)(F)F MS-9084 Cc1cc(ccc1Cl)c2csc(n2)Nc3ccc(cc3F)F MS-9085 COc1cccc(c1O)C(=O)[O-].COc1cccc(c1O)C(=O)[O-].[Cu+2] MS-9086 COc1ccccc1/C=N/NC(=[NH2+])SC/C=C/c2ccccc2.[Cl-] MS-9087 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=S)Nc4ccccc4 MS-9088 Cc1cc(ccc1F)c2csc([nH+]2)Nc3ccc(cc3)Oc4ccccc4.[Cl-] MS-9089 c1ccc(cc1)c2c(n(c(n2)c3ccc(cc3)O)c4ccc(cc4)OC(F)(F)F)c5ccccc5 MS-9090 CCOC(=O)COc1ccc2ccccc2c1Br MS-9091 c1ccc2c(c1)ccc(c2Br)OCC(=O)NN MS-9092 CC(=O)c1ccc(cc1)/N=C\2/c3ccccc3N(C2=O)C MS-9093 c1ccc2c(c1)/C(=N/Nc3nc4ccccc4s3)/C(=O)N2 MS-9094 c1cc(cc2c1cc(cc2)Br)OCC(=O)NN MS-9095 Cn1c(c(c(=O)n1c2ccccc2)Br)COc3ccc(cc3)SC(F)(F)F MS-9096 c1cc(cc(c1)Br)/C=N/C(=C(/C#N)\N)/C#N MS-9097 CN(C)c1ccc(cc1)NC=C2C(=O)c3ccccc3C2=O MS-9098 CN(C)c1ccc(cc1)/C=N/c2c([nH]c(=O)n(c2=N)c3ccccc3)C#N MS-9099 Cc1ccc2c(c1)CCCN2C(=S)Nc3ccc(cc3)OC(F)(F)F MS-9100 c1ccc2c(c1)C(=O)C(=CNc3nccs3)C2=O MS-9101 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3ccc(cc3)OC(F)(F)F)C2=O MS-9102 c1ccc(cc1)CNC2=C(C(=O)CC(C2)c3ccccc3)C(=O)Nc4cccc(c4)C(F)(F)F MS-9103 CC(C)(C)C(=O)C(=Cc1c[nH]c2c1cccc2)C#N MS-9104 CC(C)(C)C(=O)C(=CNc1ccc(cc1)SC(F)(F)F)C#N MS-9105 CC1(CC(=O)C(=CNc2cccc(c2)C(F)(F)F)C(=O)C1)C MS-9106 CCOC(=O)/C(=C/c1cccc(c1)Oc2ccccc2)/C#N MS-9107 CC(C)COC(=O)/C(=C\c1cccc(c1)Oc2ccccc2)/C#N MS-9108 CC(C)(C)S(=O)(=O)/C(=C\Nc1ccc(c(c1)C(F)(F)F)F)/C#N MS-9111 CC1(Cc2c(c(nn2C)c3ccc4c(c3)OCO4)C(=O)C1)C MS-9112 COc1ccc(cc1)N2C(C(C2=O)c3cccc4c3cccc4)c5ccc6c(c5)OCO6 MS-9113 CC(C)c1ccc(cc1)S(=O)(=O)/C(=C/c2cccc(c2)Oc3ccccc3)/C#N MS-9114 CC(C)(C)C(=O)/C(=C/1\Nc2ccc(cc2N1)Cl)/C#N MS-9115 CC(C)c1ccc(cc1)S(=O)(=O)C(=C2Nc3ccccc3N2)C#N MS-9116 CC1(CC(=CC(=O)C1)Nc2cccc(c2)NC3=CC(=O)CC(C3)(C)C)C MS-9117 CC1Cc2c(cc(nn2)c3ccc(cc3)Br)C(=O)C1 MS-9118 c1ccnc(c1)N/C=C(/C#N)\C(=O)Nc2ccc(cc2Cl)Cl MS-9119 CC1(Cc2c(cc(n2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)c4ccc(cc4)Br)C(=O)C1)C MS-9120 CC1Cc2c(cc(nn2)c3ccc(cc3)C(C)(C)C)/C(=N/OC)/C1 MS-9121 CCCC1CC2=C(CC(=NN2)c3ccc(cc3)Br)C(=O)C1 MS-9122 CCCC1Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N/OC)/C1 MS-9123 CCCC1Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N/O)/C1 MS-9124 CCC1Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N/OC)/C1 MS-9125 C/C(=N\OC)/c1ccc(cc1)N/C=C(\C#N)/C(=O)C(C)(C)C MS-9126 Cc1cc\2c(n1c3ccc(cc3)F)CC(C/C2=N/OC)C MS-9127 CC(C)C1Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N\OC)/C1 MS-9128 CC(C)C1Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N/O)/C1 MS-9129 CC1(Cc2c(c(nn2C)c3ccc(cc3)OC)C(=O)C1)C MS-9130 Cc1cc(ccc1Cl)c2cc\3c(nn2)CC(C/C3=N/OC)C MS-9131 CC(C)CC1Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N/OC)/C1 MS-9132 CC(C)CC1Cc2c(cc(nn2)c3ccc(cc3)Br)/C(=N/O)/C1 MS-9133 Cc1ccc(cc1)c2cc3c(nn2)CC(CC3=O)C MS-9134 CC1CC2=C(CC(=NN2)c3ccc(cc3Cl)Cl)C(=O)C1 MS-9135 C/C(=N/OC)/c1ccc(cc1)/N=C/C2C(=O)c3ccccc3C2=O MS-9136 c1ccc2c(c1)C(=O)C(=CNCc3ccc(cc3F)F)C2=O MS-9137 Cc1nc(no1)CC(=O)NCCc2ccc(c(c2)OC)OC MS-9138 Cc1cc2c(n1c3ccc(cc3)F)CC(CC2=O)C MS-9139 CC1(Cc2c(c(nn2C)c3ccc4c(c3)OCO4)/C(=N\OC)/C1)C MS-9140 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(cc(c2)F)F)/C#N)Cl MS-9141 CC1Cc2c(cc(nn2)c3ccc(cc3)C(C)C)/C(=N\OC)/C1 MS-9142 COc1ccc(cn1)NC=C(C#N)C#N MS-9143 CC1CC(=O)C(C(=O)C1)CC(=O)c2ccc(cc2)[N+](=O)[O-] MS-9144 CC1Cc2c(cc(n2c3ccc(cc3)C(F)(F)F)c4ccc(cc4)C(C)(C)C)/C(=N/OC)/C1 MS-9145 COc1cc2c(cc1OC)nc-3c(c2c4ccccc4)C(=O)c5c3cccc5 MS-9146 CC1Cc2c(c(nn2C)c3cccc(c3OC)OC)C(=O)C1 MS-9147 CC1Cc2c(c(nn2C)c3cccc(c3OC)OC)/C(=N\OC)/C1 MS-9148 c1cc(ccc1CC#N)NC(=O)C(F)(F)F MS-9149 Cc1cc2c(n1c3cc(on3)C)CC(CC2=O)(C)C MS-9150 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=C(C#N)C#N)C#N MS-9151 c1ccc(cc1)C2Cc3c(sc(n3)N)C(=O)C2 MS-9152 CC(C)C(=O)n1c(c2c(n1)-c3ccccc3C2=O)C(C)(C)C MS-9153 CC(=O)Nc1nc2c(s1)C(=O)CC(C2)c3ccccc3 MS-9154 CC(C)CC1Cc2c(sc(n2)N)C(=O)C1 MS-9155 CCO/N=C/1\CC(Cc2c1cc(nn2)c3ccc(cc3)C)C MS-9156 Cc1c(c(on1)C)C(=O)NCCc2ccc(c(c2)OC)OC MS-9157 Cc1c(c(no1)c2ccccc2)C(=O)NCCc3ccc(c(c3)OC)OC MS-9158 COc1ccc(cn1)NC(=C(C#N)C#N)C#N MS-9159 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(nc3)OC MS-9160 CC(C)c1cc(c(c(c1)C(=O)O)[O-])C(C)C.CC(C)c1cc(c(c(c1)C(=O)O)[O-])C(C)C.[Cu+2] MS-9161 CCO/N=C/1\CC(Cc2c1cc(nn2)c3ccc(cc3Cl)Cl)C MS-9162 c1ccc(cc1)CNC(=C2C(=O)c3ccccc3C2=O)NCc4ccccc4 MS-9164 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3)[N+](=O)[O-] MS-9165 Cc1c(c(no1)c2ccccc2)C3=NCCc4c3[nH]c5c4cccc5 MS-9166 CC[n+]1c(sc2c1cccc2)C.[I-] MS-9167 c1ccc2c(c1)c(c[nH]2)CCNC(=O)/C=C/c3ccc(c(c3)[N+](=O)[O-])Sc4ccccn4 MS-9168 c1ccc2c(c1)c(=O)oc(n2)/C=C/c3cccs3 MS-9169 Cn1cnnc1SCc2c(c(=O)n(n2C)c3ccccc3)Br MS-9170 c1ccc2c(c1)C(=O)C(=Cc3cc(ccc3Sc4ccccn4)[N+](=O)[O-])C2=O MS-9171 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(ccn2)C(F)(F)F)/C#N)Cl MS-9172 c1ccc(cc1)NC(=S)NNC(=O)CSc2[nH]c3ccccc3n2 MS-9173 c1ccc2c(c1)[nH]c(n2)SCC(=O)NNC(=O)Nc3cccc(c3)C(F)(F)F MS-9174 CC(=O)Nc1ccc(cc1)OCc2c(c(=O)n(n2C)c3ccccc3)Br MS-9175 CCO/N=C/1\CC(Cc2c1cc(n2c3ccc(nc3)OC)c4ccc(cc4)Br)(C)C MS-9176 c1ccnc(c1)Sc2ccc(cc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] MS-9177 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)n4cncn4 MS-9178 Cc1cc(c(c(c1)C(=O)O)NC(=O)Nc2ccc(cc2)OC(F)(F)F)C MS-9179 c1cc(ccc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)n3cnc(c3Cl)Cl MS-9180 c1cc(c(cc1Cl)Cl)/C=C/C(=O)O MS-9181 CC1Cc2c(sc(n2)NC(=O)c3cccnc3Oc4ccccc4)C(=O)C1 MS-9183 CC1Cc2c(sc(n2)NC(=O)c3cccnc3Cl)C(=O)C1 MS-9184 CC(C)(C)c1ccc(cc1)S(=O)(=O)/C(=C\Nc2ccc(cn2)C(F)(F)F)/C#N MS-9185 c1cc(ccc1N/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl)Oc3c(cc(cn3)C(F)(F)F)Cl MS-9186 CC1=NN(C(=O)C1=Cc2cc(c(cc2[N+](=O)[O-])OC)OC)c3ccccc3 MS-9187 Cc1ccc2cccc(c2n1)Oc3ccc(cn3)[N+](=O)[O-] MS-9188 CCOC(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl MS-9189 c1cc(ccc1NC(=O)C2CC2C(=O)O)Oc3c(cc(cn3)C(F)(F)F)Cl MS-9190 CC1(CC(=O)C(=CNc2ccc(c(c2)OC)OC)C(=O)C1)C MS-9191 CC1(CC(=O)C(=CNc2ccc(cc2[N+](=O)[O-])OC)C(=O)C1)C MS-9192 CC(C)CC1CC(=O)C(=CNc2ccc(nc2)OC)C(=O)C1 MS-9193 c1ccc2c(c1)cccc2Oc3ccc(cc3NC=C(C#N)C#N)C(F)(F)F MS-9194 CCC1CC(=O)C(=CNc2cc(ccc2Oc3cccc4c3cccc4)C(F)(F)F)C(=O)C1 MS-9195 c1cc(ccc1C(F)(F)F)Oc2ccc(cc2)N MS-9196 CCN(CC)C(=S)Sc1c(cc(cn1)C(F)(F)F)Cl MS-9198 CCOC(=O)c1c2c(sc1NC=C(C#N)C#N)CCCC2 MS-9199 CCOC(=O)c1c2c(sc1N/C=C(/C#N)\C(=O)C(C)(C)C)CCCC2 MS-9200 COc1cc2c(cc1OC)C(=O)/C(=C/c3cccc(c3)Oc4ccccc4)/C2 MS-9201 CC(C)C1CC(=O)C(=CNc2ccc(nc2)OC)C(=O)C1 MS-9202 c1cc(ccc1S(=O)(=O)/C(=C\Nc2ccc(cn2)C(F)(F)F)/[N+](=O)[O-])Cl MS-9203 c1cc(c(cc1Cl)Cl)S(=O)(=O)/C(=C/Nc2ccc(cn2)C(F)(F)F)/C#N MS-9204 c1ccc2c(c1)CC(=Cc3ccc(cc3)OC(F)F)C2=O MS-9205 c1cc(cc(c1)OC(F)(F)F)/C=C/C(=O)O MS-9206 Cc1cc2c(n1c3ccc(cc3)NC(=O)c4ccccc4)CC(CC2=O)(C)C MS-9207 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)OC(F)(F)F)CCCC2 MS-9208 CC1(CC(=O)C(=CNc2ccc(cc2)O)C(=O)C1)C MS-9209 c1ccnc(c1)Sc2c(cc(cn2)C(F)(F)F)Cl MS-9210 CC(C)c1c2c([nH]n1)-c3ccccc3C2=NN MS-9211 c1ccc2c(c1)C(=O)C(=CNc3ccccn3)C2=O MS-9212 CC1(Cc2cccc(c2O1)OCc3c(c(=O)n(n3C)c4ccccc4)Br)C MS-9213 Cc1nc(nn1c2ccccc2)OCc3c(c(=O)n(n3C)c4ccccc4)Br MS-9214 c1cc(c(c(c1)Cl)c2c([nH]nn2)C#N)F MS-9215 COc1cc2c(cc1OC)C(=O)/C(=C\c3ccc(cc3)Oc4c(cc(cn4)C(F)(F)F)Cl)/C2 MS-9216 CC(C)(C)c1c2c(nn1c3ccc(cc3)[N+](=O)[O-])-c4ccc(cc4C2=O)[N+](=O)[O-] MS-9217 c1ccc(cc1)N2CCN(CC2)C(=O)C3CC3C(=O)O MS-9218 COc1ccc(cc1)C(=O)Nc2nc(=O)[nH]s2 MS-9219 Cn1c(=S)n(c(n1)c2ccc(cc2Cl)Cl)c3ccccc3 MS-9220 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)Oc4ccc(cn4)C(F)(F)F)C2=O MS-9221 c1cc(ccc1NC=C2C(=O)CCCC2=O)OC(F)(F)F MS-9222 CCC1CC(=O)C(=CNc2cc(cc(c2)F)F)C(=O)C1 MS-9223 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)Oc4cccc(c4)C(F)(F)F MS-9224 COc1ccc(cc1OC)C2=C(c3ccccc3C2=O)Nc4ccc(cc4)Oc5cccc(c5)C(F)(F)F MS-9225 CSc1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)OC(F)(F)F MS-9226 Cc1ccc(cc1)Sc2ccc(cc2/C=C(/C#N)\S(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] MS-9227 c1ccc(c(c1)C(=O)O/N=C(\c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F)/N)Cl MS-9228 c1cc(cc(c1)OC(F)(F)F)N/C=C(/C#N)\S(=O)(=O)c2ccc(cc2)Cl MS-9229 Cn1c(=S)n(c(n1)c2cccs2)c3ccccc3 MS-9230 CC(=C1C(=O)c2ccccc2C1=O)N3CCN(CC3)c4ccccc4F MS-9231 c1cc(cc(c1)NC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F MS-9233 c1cc(cc(c1)NC(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)C(F)(F)F MS-9234 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)NC=C3C(=O)CC(CC3=O)C MS-9235 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl)CC(=O)OC MS-9237 c1cc(ccc1S(=O)(=O)/C(=C\N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)/C#N)Cl MS-9238 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F MS-9239 CC1(CC2=C(C(Nc3ccccc3N2)c4cc(ccc4Oc5ccc(cc5)C(F)(F)F)[N+](=O)[O-])C(=O)C1)C MS-9240 CC(C)(CCC(=S)N1CCOCC1)c2ccccc2 MS-9241 CCOc1ccc(cc1)Nc2nc(cs2)c3ccc(cc3)Br MS-9242 c1ccc2c(c1)c(=O)c(=NNC(=O)c3ccncc3)c2=O MS-9243 CN(C)C(=S)Nc1ccc(cc1)Sc2c(cc(cn2)C(F)(F)F)Cl MS-9244 Cc1cc(ccc1Oc2c(cccn2)C(=O)NN(C)c3c(cc(cn3)C(F)(F)F)Cl)Cl MS-9245 c1cc(ccc1C#N)Oc2c(c(c(c(n2)F)Cl)N)Cl MS-9246 c1cc(ccc1NC(=S)NNC(=O)CSc2c(cc(cn2)C(F)(F)F)Cl)SC(F)(F)F MS-9247 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C(=O)c3cc(c(nc3)Cl)Cl MS-9249 c1cc(nc(c1C(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl MS-9250 c1cc(ccc1C[N+]23CN4CN(C2)CN(C4)C3)SC(F)(F)F.[Br-] MS-9251 COc1ccc(cc1OC)CNC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-9252 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)C(=O)O)C2=O MS-9253 COc1cc(c(cc1OC)S(=O)(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)CC(=O)OC MS-9254 CCC1(C(=C)SC(=N1)Nc2ccc(cc2)SC(F)(F)F)CC MS-9255 c1ccc2c(c1)ccc3c2sc(c3Cl)C(=O)Nc4ccc(cc4)SC(F)(F)F MS-9256 c1cc(ccc1n2c(n[nH]c2=S)CSc3c(cc(cn3)C(F)(F)F)Cl)SC(F)(F)F MS-9257 Cc1ccnc(n1)NS(=O)(=O)c2ccc(cc2)NC=C3C(=O)CC(CC3=O)(C)C MS-9258 c1cc(ccc1OC(F)(F)F)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl MS-9259 CC1(C2CCC1(/C(=N\O)/C2)CS(=O)(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C MS-9260 CC(C(=O)NNC(=S)NCc1ccc(c(c1)OC)OC)Sc2ccc(cc2)Cl MS-9261 Cc1cc2c(n1c3cccc(c3)C#N)CC(CC2=O)(C)C MS-9262 c1ccc2c(c1)C(=C(C2=O)c3ccc4c(c3)OCO4)Nc5ccc(cc5)Br MS-9263 COc1ccc(cc1OC)CCNC2=C(C(=O)c3c2cccc3)c4ccc5c(c4)OCO5 MS-9264 CCO/N=C/1\CC(Cc2c1cc(nn2)c3ccc(c(c3)C)Cl)(C)C MS-9265 CC(=C1C(=O)c2ccccc2C1=O)Nc3ccc(cc3)C(C(F)(F)F)(C(F)(F)F)O MS-9266 Cc1cc(no1)NC(=O)c2cccnc2Cl MS-9267 CC1(Cc2c(cc(o2)c3ccc(cc3)Br)C(=O)C1)C MS-9268 C/C(=N\C(=C(\C#N)/N)\C#N)/c1ccc(cc1)Oc2ccccc2 MS-9269 CCOC=C1C(=O)c2ccccc2C1=O MS-9270 CC(=C1C(=O)c2ccccc2C1=O)OC MS-9271 Cc1cccc(c1NC=C(C#N)C#N)Cl MS-9272 CC1(CC(=CC(=O)C1)Nc2cccc(c2)C(F)(F)F)C MS-9273 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccccc2Cl MS-9274 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC3=NCCS3 MS-9275 c1cc(c(cc1c2csc([nH+]2)Nc3ccc(cc3F)F)O)O.[Cl-] MS-9276 CC1(CC(=O)C(C(=O)C1)SC(=N)N)C MS-9277 CCC(C)c1ccc(cc1)NC(=O)CSc2nc3ccccc3o2 MS-9278 Cc1cc2c(n1c3ccc(cc3)Oc4ccccc4)CC(CC2=O)(C)C MS-9279 Cc1cc2c(n1c3ccc(cc3)C(=O)N)CC(CC2=O)(C)C MS-9280 Cc1cc(c2c(c1)c(=O)oc(n2)C(C)Sc3ccc(cc3)Cl)C MS-9281 CC1(Cc2cccc(c2O1)OCC(=O)NNC(=S)NC(C)(C)C)C MS-9282 c1ccc2c(c1)C(=O)C(C2=O)/C(=N/N)/C3CC3 MS-9283 Cc1ccc(cc1)n2c(n[nH]c2=S)COc3cccc4c3OC(C4)(C)C MS-9284 c1ccc(cc1)CCNc2nc(=O)c3cccnc3s2 MS-9285 c1ccc(cc1)CN(c2ccccc2Br)C(=O)/C=C/c3ccccc3 MS-9286 CC(C)C(=O)N(C)c1c(cc(cc1Br)F)F MS-9287 Cn1c(nnn1)SCC(=O)Nc2cc(ccc2F)F MS-9288 CNC(=S)NNC(=O)CNc1ccc2c(c1)OCO2 MS-9289 COc1ccc(cc1c2c([nH]nn2)C#N)Br MS-9290 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cc(cc(c3)C(=O)OC)C(=O)OC)c4ccccc4 MS-9296 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4)OC)c5ccccc5 MS-9297 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4Cl)Cl)c5ccccc5 MS-9298 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4OC)OC)c5ccccc5 MS-9299 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4)C(F)(F)F)c5ccccc5 MS-9300 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cccc(c3)C(=O)OC)c4ccccc4 MS-9301 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cc(cc(c4)Cl)Cl)c5ccccc5 MS-9302 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(c(c4)Cl)Cl)c5ccccc5 MS-9303 CCOC(=O)c1ccc(cc1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9304 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cccc(c4)C(=O)OC)c5ccccc5 MS-9305 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4c(cccc4Cl)Cl)c5ccccc5 MS-9306 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cc(cc(c4)C)C)c5ccccc5 MS-9307 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccccc4C(F)(F)F)c5ccccc5 MS-9308 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccccc4OC)c5ccccc5 MS-9309 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Cc4cccc(c4)C(F)(F)F)c5ccccc5 MS-9310 Cc1cc(ccc1NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)Br MS-9311 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)c4ccccc4 MS-9312 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(c(c3)[N+](=O)[O-])F)c4ccccc4 MS-9313 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4Cl)[N+](=O)[O-])c5ccccc5 MS-9314 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4Br)Br)c5ccccc5 MS-9315 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cc(ccc4OC)[N+](=O)[O-])c5ccccc5 MS-9316 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4Cl)Br)c5ccccc5 MS-9317 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4F)F)c5ccccc5 MS-9318 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4C)Br)c5ccccc5 MS-9319 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4)OC(F)(F)F)c5ccccc5 MS-9320 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc-4c(c3)Cc5c4cccc5)c6ccccc6 MS-9321 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3c(cccc3F)C(F)(F)F)c4ccccc4 MS-9322 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc5c(c4)OCO5)c6ccccc6 MS-9323 Cc1ccc(c(c1)[N+](=O)[O-])NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9324 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4[N+](=O)[O-])Cl)c5ccccc5 MS-9325 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4)Oc5ccccc5)c6ccccc6 MS-9326 CCOc1ccc(cc1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9327 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccccc3c4ccccc4)c5ccccc5 MS-9328 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(c(c4)Cl)OC)c5ccccc5 MS-9329 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4)C(=O)C)c5ccccc5 MS-9330 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4)F)c5ccccc5 MS-9331 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccccc4F)c5ccccc5 MS-9332 CCc1ccc(cc1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9333 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4)C(C)C)c5ccccc5 MS-9334 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4C)Cl)c5ccccc5 MS-9335 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cc(cc(c4)F)F)c5ccccc5 MS-9336 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccccc4Br)c5ccccc5 MS-9337 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cccc(c4)C(=O)C)c5ccccc5 MS-9338 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(c(c4)F)C)c5ccccc5 MS-9339 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4c(cccc4Cl)C)c5ccccc5 MS-9340 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cccc(c4C)Cl)c5ccccc5 MS-9341 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4C(F)(F)F)Cl)c5ccccc5 MS-9342 Cc1ccc(c(c1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C)OC MS-9343 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccccc4C(C)C)c5ccccc5 MS-9344 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4C(F)(F)F)Br)c5ccccc5 MS-9345 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cccc(c4C)[N+](=O)[O-])c5ccccc5 MS-9346 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(c(c4)[N+](=O)[O-])C)c5ccccc5 MS-9347 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4c(cccc4F)F)c5ccccc5 MS-9348 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(c(c4)C)Br)c5ccccc5 MS-9349 COc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)OCc4ccccc4)c5ccccc5 MS-9350 c1ccc(cc1)COC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5Br MS-9351 CC1(Cc2c(cc(n2c3ccc(cc3)Cl)c4ccc(cc4)Br)C(=O)C1)C MS-9352 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3ccc(cc3Cl)C(F)(F)F)c4ccccc4 MS-9353 CN1c2ccccc2C(=NC(C1=O)NC(=O)NCc3ccc(cc3)Br)c4ccccc4 MS-9354 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4F)Br)c5ccccc5 MS-9355 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4cc(cc(c4)F)C(F)(F)F)c5ccccc5 MS-9356 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4c(cccc4F)C(F)(F)F)c5ccccc5 MS-9357 CN1c2ccccc2C(=NC(C1=O)NC(=O)Nc3cc(ccc3F)[N+](=O)[O-])c4ccccc4 MS-9358 CCCCc1ccc(cc1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9359 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Oc4ccc(cc4)[N+](=O)[O-])c5ccccc5 MS-9360 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(cc4[N+](=O)[O-])OC)c5ccccc5 MS-9361 CC1(CC2=C(C(Nc3cc(ccc3N2)Cl)c4cccc(c4O)O)C(=O)C1)C MS-9362 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc5c(c4)CCC5)c6ccccc6 MS-9363 CCOC(=O)CCNC(=O)NC1C(=O)N(c2ccccc2C(=N1)c3ccccc3)CC(=O)c4ccccc4C MS-9364 CCOc1ccccc1NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9365 c1ccc(cc1)C2=NC(C(=O)N(c3c2cccc3)CC(=O)c4ccccc4F)NC(=O)Nc5cccc(c5)Cl MS-9366 COc1cccc(c1)NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5F MS-9367 CN1c2ccccc2C(=NC(C1=O)NC(=O)Cc3ccc(cc3)Oc4ccccc4)c5ccccc5 MS-9368 Cc1ccccc1C(=O)CN2c3ccccc3C(=NC(C2=O)NC(=O)Nc4ccc(c(c4)Cl)F)c5ccccc5 MS-9369 c1ccc(cc1)C2=NC(C(=O)N(c3c2cccc3)CC(=O)c4ccccc4[N+](=O)[O-])NC(=O)Cc5cccc(c5)Br MS-9370 Cc1cccc(c1NC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)C)[N+](=O)[O-] MS-9371 Cc1ccccc1CNC(=O)NC2C(=O)N(c3ccccc3C(=N2)c4ccccc4)CC(=O)c5ccccc5C MS-9372 c1cc(cc(c1)NC2=C(C(=O)CCC2)Br)C(F)(F)F MS-9373 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4)C#N MS-9374 Cc1cc(ccc1Br)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9375 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4SC MS-9376 CC(C)c1ccccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9377 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4)OCc5ccccc5 MS-9378 COc1ccc(cc1Cl)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9379 Cc1ccc(cc1F)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9380 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(c(c4)F)F MS-9381 Cc1ccc(cc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)[N+](=O)[O-] MS-9382 Cc1ccc(c(c1)[N+](=O)[O-])NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9383 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc5c(c4)OCO5 MS-9384 Cc1ccc(c(c1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)Cl MS-9385 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc-5c(c4)Cc6c5cccc6 MS-9386 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4c(cccc4F)C(F)(F)F MS-9387 CCc1cccc(c1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)C MS-9388 Cc1ccc(cc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)F MS-9389 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)NCc4ccc(c(c4)Cl)Cl MS-9390 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)NCc4ccc(cc4Cl)Cl MS-9391 CN(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9392 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4C(F)(F)F)F MS-9393 Cc1cc(ccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)Cl MS-9394 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4Cl)Br MS-9395 Cc1cc(ccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)OC MS-9396 CCc1cccc(c1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)CC MS-9397 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cccc(c4)[N+](=O)[O-] MS-9398 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4)OC(F)(F)F MS-9399 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)NCc4ccc(cc4)Br MS-9400 Cc1ccc(c(c1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)OC MS-9401 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(c(c4)[N+](=O)[O-])F MS-9402 Cc1cc(ccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)Br MS-9403 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4Cl)Cl MS-9404 Cc1cccc(c1C)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9405 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cccc(c4)Cl MS-9406 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cc(ccc4F)[N+](=O)[O-] MS-9407 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cccc(c4Cl)Cl MS-9408 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)NC4CCCCC4 MS-9409 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4C(=O)OC MS-9410 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(c(c4)Cl)Cl MS-9411 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4)SC MS-9412 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4F)F MS-9413 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cccc(c4)F MS-9414 Cc1ccc(cc1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9415 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4)Br MS-9416 c1cc(cc(c1)NC2=C(C(=O)CCC2)[N+](=O)[O-])C(F)(F)F MS-9417 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4F MS-9418 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4Br MS-9419 Cc1ccc(cc1[N+](=O)[O-])NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9420 Cc1c(cccc1Cl)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9421 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cccc(c4)C#N MS-9422 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F MS-9423 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4)F MS-9424 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cc(cc(c4)Cl)Cl MS-9425 CCOc1ccc(cc1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9426 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cc(ccc4Cl)Cl MS-9427 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4OC(F)(F)F MS-9428 Cc1cccc(c1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)C(C)(C)C MS-9429 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cccc5c4cccc5 MS-9430 Cc1cc(ccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)[N+](=O)[O-] MS-9431 COc1cccc(c1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9432 CC(=O)c1ccc(cc1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9433 COc1ccccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9434 Cc1cccc(c1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)Cl MS-9435 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)NCC=C MS-9436 COc1ccc(c(c1)OC)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9437 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4Cl MS-9438 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4[N+](=O)[O-])Cl MS-9439 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC)C MS-9440 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4[N+](=O)[O-] MS-9441 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cc(ccc4F)F MS-9442 Cc1ccc(cc1)CNC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9443 c1ccc2c(c1)C(=O)C(C2=O)C=Nc3ccccc3F MS-9444 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccccc4I MS-9445 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4ccc(c(c4)Cl)F MS-9446 COc1cc2c(cc1OC)C(=NCC2)Cc3ccc(cc3)NC(=O)Nc4cccc(c4)I MS-9447 CCOc1ccccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9448 CCc1ccccc1NC(=O)Nc2ccc(cc2)CC3=NCCc4c3cc(c(c4)OC)OC MS-9449 c1ccc(c(c1)NC2=C(C(=O)CCC2)Cl)F MS-9450 COc1ccc(cc1)CNC(=O)C2c3ccccc3C(=O)N(C2c4cccnc4)c5ccc(cc5)OC MS-9451 COc1ccc(cc1)N2C(C(c3ccccc3C2=O)C(=O)NCC(=O)OC)c4cccnc4 MS-9452 COc1ccc(cc1)CNC(=O)C2c3ccccc3C(=O)N(C2c4cccnc4)c5ccc6c(c5)OCO6 MS-9453 COc1ccc(cc1)CNC(=O)C2c3ccccc3C(=O)N(C2c4ccc(cc4)OC)c5ccc6c(c5)OCO6 MS-9454 CCC(=O)n1c(c2c(n1)-c3ccccc3C2=O)C(C)(C)C MS-9455 c1ccc2c(c1)cccc2CNS(=O)(=O)c3ccccc3[N+](=O)[O-] MS-9458 Cc1ccccc1NC(=O)N2CCN(CC2)Cc3ccccc3 MS-9459 c1ccnc(c1)N2CCN(CC2)C(=O)Nc3cc(ccc3F)F MS-9460 Cc1ccccc1NC(=O)NCc2ccccc2OC MS-9461 Cc1ccccc1NC(=O)NCc2ccc(cc2)OC MS-9462 COc1cc(ccc1O)/C=C/2\C(=O)SC(=S)N2 MS-9463 c1cc(c(cc1Cl)c2[nH]nnn2)Cl MS-9465 Cc1cccc(c1C)C(=O)N MS-9466 c1cc(c(c(c1)Cl)c2[nH]nnn2)Cl MS-9467 c1ccc(cc1)CN2CCN(CC2)C(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-9468 COc1ccccc1CNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-9469 c1ccnc(c1)N2CCN(CC2)C(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F MS-9470 c1ccnc(c1)CNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-9471 COc1ccc(cc1)CNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-9472 c1cc(c(c(c1)Cl)Cl)c2[nH]nnn2 MS-9473 CC(C)(C)C(=O)Nc1ccc(cc1)C(F)(F)F MS-9474 COC(=O)c1ccsc1NC(=S)Nc2ccc3c(c2)OCO3 MS-9475 COC(=O)c1ccsc1NC(=S)Nc2cc(ccc2Cl)[N+](=O)[O-] MS-9476 COC(=O)c1ccc(o1)CS(=O)(=O)c2ccc(cc2)Br MS-9477 COC(=O)c1ccc(o1)CS(=O)(=O)c2ccc(cc2)Cl MS-9478 CCOC(=O)c1csc(n1)Nc2cccc(c2)F MS-9479 COc1cc(c(cc1OC)S(=O)(=O)N)CC(=O)OC MS-9480 CCOC(=O)Cc1csc(n1)Nc2ncccn2 MS-9481 Cc1ccc(cc1)S(=O)(=O)C(C)C(=O)NN MS-9482 Cc1cc(cc\2c1NC(=O)/C2=N\NC(=S)N)Cl MS-9483 CCOc1ccccc1/C=C/C(=O)O MS-9484 CCOc1cccc(c1)C(=O)NN MS-9485 COC(=O)c1cc(ccc1[N+](=O)[O-])O MS-9489 c1ccc(cc1)CNC(=O)C(c2ccccc2)c3ccccc3 MS-9491 CC(c1ccccc1)NC(=O)C(c2ccccc2)c3ccccc3 MS-9492 c1ccc(cc1)C(c2ccccc2)C(=O)N3CCOCC3 MS-9493 COc1ccc(cc1)NC(=O)C(c2ccccc2)c3ccccc3 MS-9494 c1ccc(cc1)C(c2ccccc2)C(=O)Nc3ccc(cc3)C(F)(F)F MS-9495 c1ccc(cc1)C(c2ccccc2)C(=O)N MS-9496 c1cc(ccc1C(=O)N)[N+](=O)[O-] MS-9497 c1ccc(cc1)CNC(=O)c2ccc(cc2)[N+](=O)[O-] MS-9498 CC(c1ccccc1)NC(=O)c2ccc(cc2)[N+](=O)[O-] MS-9499 COc1ccc(cc1)NC(=O)c2ccc(cc2)[N+](=O)[O-] MS-9500 c1cc(ccc1C(=O)Nc2ccc(cc2)C(F)(F)F)[N+](=O)[O-] MS-9501 CCOC(=O)Cc1csc(n1)NC(=S)NC(=O)c2ccccc2 MS-9502 c1c(nc(s1)NC(=S)N)CC(=O)O MS-9503 CCOC(=O)Cc1csc(n1)Nc2nc(cs2)CC(=O)OCC MS-9504 c1ccc(c(c1)NC(=S)N)OC(F)(F)F MS-9505 c1cc(ccc1NC(=S)N)Oc2ccc(cn2)C(F)(F)F MS-9507 Cc1cc(nc(n1)NC(=S)N)C MS-9508 Cc1c(c(nc(n1)NC(=S)N)C)Br MS-9509 c1cc(ccc1c2csc(n2)N)N MS-9510 c1cc(ccc1NC(=S)N)Oc2c(cc(cn2)C(F)(F)F)Cl MS-9511 c1cc(ccc1NC(=S)N)Sc2c(cc(cn2)C(F)(F)F)Cl MS-9512 c1cc(cc(c1)Oc2ccc(cc2)NC(=S)N)C(F)(F)F MS-9513 CC(C)(C)c1ccc(cc1)S(=O)(=O)Cc2ccc(o2)C(=O)OC MS-9514 c1cc(ccc1NC(=S)N)Sc2ccc(cc2)Cl MS-9515 COc1cc(c(cc1OC)S(=O)(=O)Nc2ccc3c(c2)OCO3)CC(=O)O MS-9516 COc1ccc(cc1)NS(=O)(=O)c2cc(c(cc2CC(=O)OC)OC)OC MS-9517 COc1ccc(cc1)NS(=O)(=O)c2cc(c(cc2CC(=O)O)OC)OC MS-9518 COc1cc(c(cc1OC)S(=O)(=O)N2CCSCC2)CC(=O)O MS-9519 CC(C)Oc1ccc(cc1)S(=O)(=O)C(C)C(=O)NN MS-9520 COc1ccc(cc1NC(=S)N)C(F)(F)F MS-9521 Cc1ccc(cc1)S(=O)(=O)Cc2ccc(o2)C(=O)OC MS-9522 COC(=O)c1ccc(o1)CS(=O)(=O)c2ccccc2 MS-9523 CN1CCN(CC1)S(=O)(=O)c2cc(c(cc2CC(=O)OC)OC)OC MS-9524 COc1cc(c(cc1OC)S(=O)(=O)N2CCCCC2)CC(=O)OC MS-9525 COc1cc(c(cc1OC)S(=O)(=O)N2CCCCC2)CC(=O)O MS-9526 COc1cc(c(cc1OC)S(=O)(=O)N2CCc3c2cccc3)CC(=O)O MS-9527 COc1cc(c(cc1OC)S(=O)(=O)N2CCc3c2cccc3)CC(=O)OC MS-9528 CC(C)Oc1ccc(cc1)/C=C/C(=O)O MS-9529 CC(C)Oc1cccc(c1)NC(=O)c2ccccc2CC(=O)O MS-9530 c1ccc(cc1)Nc2nc(cs2)CC(=O)O MS-9535 c1cc(ccc1Nc2nc(cs2)CC(=O)O)OC(F)(F)F MS-9536 c1ccc(cc1)Oc2ccc(cc2)Nc3nc(cs3)CC(=O)O MS-9537 c1c(cc(cc1C(F)(F)F)Nc2nc(cs2)CC(=O)O)C(F)(F)F MS-9538 c1cc(ccc1Nc2nc(cs2)CC(=O)O)Br MS-9539 c1cc(ccc1Nc2nc(cs2)CC(=O)O)Cl MS-9540 c1cc(cc(c1)Cl)Nc2nc(cs2)CC(=O)O MS-9541 c1cc(c(cc1Nc2nc(cs2)CC(=O)O)Cl)Cl MS-9542 CCOC(=O)Cc1csc(n1)Nc2cc(ccc2Cl)Cl MS-9543 c1cc(c(cc1Cl)Cl)Nc2nc(cs2)CC(=O)O MS-9544 c1cc(c(c(c1)Cl)Nc2nc(cs2)CC(=O)O)Cl MS-9545 CCc1cccc(c1Nc2nc(cs2)CC(=O)O)CC MS-9546 c1cc(cc(c1)F)Nc2nc(cs2)CC(=O)O MS-9547 Cc1ccc(cc1)Nc2nc(cs2)CC(=O)O MS-9548 COc1ccc(cc1)Nc2nc(cs2)CC(=O)O MS-9549 c1cnc(nc1)Nc2nc(cs2)CC(=O)O MS-9550 c1cc(cc(c1)Nc2nc(cs2)CC(=O)O)C(F)(F)F MS-9551 c1ccc(c(c1)C(F)(F)F)Nc2nc(cs2)CC(=O)O MS-9552 c1cc(ccc1C(F)(F)F)Nc2nc(cs2)CC(=O)O MS-9553 CCOC(=O)Cc1csc(n1)Nc2ccccc2C(F)(F)F MS-9554 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)OC MS-9555 c1cc(ccc1Nc2nc(cs2)CC(=O)O)F MS-9556 CCOC(=O)Cc1csc(n1)Nc2cccc(c2)F MS-9557 c1ccc(c(c1)Nc2nc(cs2)CC(=O)O)F MS-9558 CCOC(=O)Cc1csc(n1)Nc2c(cccc2Cl)Cl MS-9559 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2Cl)Cl MS-9560 c1cc(c(cc1Cl)Nc2nc(cs2)CC(=O)O)Cl MS-9561 COc1ccc(cc1Nc2nc(cs2)CC(=O)O)Cl MS-9562 CCOC(=O)Cc1csc(n1)Nc2ccc(cc2)Br MS-9563 COc1cc(ccc1O)c2n[nH]c(=S)n2c3ccccc3 MS-9564 COc1cc(ccc1OCc2ccccc2)c3n[nH]c(=S)n3c4ccccc4 MS-9565 Cc1ccc(cc1)n2c(n[nH]c2=S)c3ccc(c(c3)OC)O MS-9566 Cc1ccc(cc1)n2c(n[nH]c2=S)c3ccc(c(c3)OC)OCc4ccccc4 MS-9567 Cn1c(n[nH]c1=S)c2ccc(c(c2)OC)O MS-9568 Cn1c(n[nH]c1=S)c2ccc(c(c2)OC)OCc3ccccc3 MS-9569 COc1cc(ccc1O)c2n[nH]c(=S)n2c3ccc(cc3)Cl MS-9570 COc1cc(ccc1OCc2ccccc2)c3n[nH]c(=S)n3c4ccc(cc4)Cl MS-9571 COc1cc(ccc1OCc2ccccc2)c3n[nH]c(=S)n3Cc4ccccc4 MS-9572 COc1cc(ccc1O)c2n[nH]c(=S)n2Cc3ccccc3 MS-9573 COc1cc(ccc1O)c2n[nH]c(=S)n2c3ccc(cc3)C(F)(F)F MS-9574 COc1cc(ccc1OCc2ccccc2)C(=O)NN MS-9575 CCOC(=O)c1c(nc(s1)Nc2ccccc2Br)C MS-9576 CCOC(=O)c1csc(n1)Nc2ccccc2Br MS-9577 CCOC(=O)c1c(nc(s1)Nc2cccc(c2)F)C MS-9578 CCOC(=O)c1csc(n1)Nc2cccc(c2)Br MS-9579 CCOC(=O)c1c(nc(s1)Nc2cccc(c2)Br)C MS-9580 CCOC(=O)c1c(nc(s1)Nc2ccc(cc2)Br)C MS-9581 CCOc1ccc(cc1)Nc2nc(c(s2)C(=O)OCC)C MS-9582 CCOc1ccc(cc1)Nc2nc(cs2)C(=O)OCC MS-9583 CCOC(=O)c1csc(n1)Nc2ccccn2 MS-9584 CCOC(=O)c1c(nc(s1)Nc2ccccn2)C MS-9585 CCOC(=O)c1csc(n1)Nc2cccnc2 MS-9586 CCOC(=O)c1c(nc(s1)Nc2cccnc2)C MS-9587 CCOC(=O)c1csc(n1)NCc2ccccc2 MS-9588 CCOC(=O)c1c(nc(s1)NCc2ccccc2)C MS-9589 CCOC(=O)c1csc(n1)Nc2cccc(c2)OC(F)(F)F MS-9590 CCOC(=O)c1c(nc(s1)Nc2cccc(c2)C(F)(F)F)C MS-9591 CCOC(=O)c1csc(n1)Nc2cccc(c2)C(F)(F)F MS-9592 CCOC(=O)c1csc(n1)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MS-9593 CCOC(=O)c1c(nc(s1)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C MS-9594 CCOC(=O)c1csc(n1)Nc2cc(ccc2Cl)Cl MS-9595 CCOC(=O)c1csc(n1)Nc2ccc(cc2Cl)Cl MS-9596 CCOC(=O)c1c(nc(s1)Nc2ccc(cc2Cl)Cl)C MS-9597 CCOC(=O)c1csc(n1)Nc2ccc(c(c2)OC)OC MS-9598 CCOC(=O)c1c(nc(s1)Nc2ccc(c(c2)OC)OC)C MS-9599 Cc1c(sc(n1)Nc2ccccc2)C(=O)O MS-9600 c1ccc(c(c1)Nc2nc(cs2)C(=O)O)Cl MS-9601 CC1(OC(=O)C(=CNc2ccc(cc2)Nc3ccccc3)C(=O)O1)C MS-9602 Cc1c(sc(n1)Nc2ccccc2Cl)C(=O)O MS-9603 COc1ccc(cc1Nc2nc(cs2)C(=O)O)Cl MS-9604 Cc1c(sc(n1)Nc2cc(ccc2OC)Cl)C(=O)O MS-9605 Cc1c(sc(n1)Nc2ccccc2Br)C(=O)O MS-9606 c1ccc(c(c1)Nc2nc(cs2)C(=O)O)Br MS-9607 Cc1c(sc(n1)Nc2ccccc2F)C(=O)O MS-9608 c1ccc(c(c1)Nc2nc(cs2)C(=O)O)F MS-9609 c1cc(cc(c1)F)Nc2nc(cs2)C(=O)O MS-9610 Cc1c(sc(n1)Nc2cccc(c2)F)C(=O)O MS-9611 c1cc(cc(c1)Br)Nc2nc(cs2)C(=O)O MS-9612 CC1CC(=CC(=O)C1)Nc2ccc(cc2)Nc3ccccc3 MS-9613 Cc1c(sc(n1)Nc2cccc(c2)Br)C(=O)O MS-9614 Cc1c(sc(n1)Nc2cccc(c2)Cl)C(=O)O MS-9615 c1cc(cc(c1)Cl)Nc2nc(cs2)C(=O)O MS-9616 Cc1c(sc(n1)Nc2ccc(cc2)Cl)C(=O)O MS-9617 c1cc(ccc1Nc2nc(cs2)C(=O)O)Br MS-9618 Cc1c(sc(n1)Nc2ccc(cc2)Br)C(=O)O MS-9619 c1cc(ccc1Nc2nc(cs2)C(=O)O)F MS-9620 CCOc1ccc(cc1)Nc2nc(c(s2)C(=O)O)C MS-9621 Cc1c(sc(n1)Nc2ccc(cc2)F)C(=O)O MS-9622 CCOc1ccc(cc1)Nc2nc(cs2)C(=O)O MS-9623 COc1ccc(cc1)Nc2nc(cs2)C(=O)O MS-9624 Cc1c(sc(n1)Nc2ccc(cc2)OC)C(=O)O MS-9625 c1ccc(cc1)Oc2ccc(cc2)Nc3nc(cs3)C(=O)O MS-9626 Cc1c(sc(n1)Nc2ccc(cc2)Oc3ccccc3)C(=O)O MS-9627 c1ccnc(c1)Nc2nc(cs2)C(=O)O MS-9628 Cc1c(sc(n1)Nc2ccccn2)C(=O)O MS-9629 c1cc(cnc1)Nc2nc(cs2)C(=O)O MS-9630 Cc1c(sc(n1)Nc2cccnc2)C(=O)O MS-9631 c1ccc2cc(ccc2c1)Nc3nc(cs3)C(=O)O MS-9632 Cc1c(sc(n1)Nc2ccc3ccccc3c2)C(=O)O MS-9633 Cc1c(sc(n1)NCc2ccccc2)C(=O)O MS-9634 C=CCNc1nc(cs1)C(=O)O MS-9635 Cc1c(sc(n1)NCC=C)C(=O)O MS-9636 c1cc(ccc1Nc2nc(cs2)C(=O)O)OC(F)(F)F MS-9637 Cc1c(sc(n1)Nc2ccc(cc2)OC(F)(F)F)C(=O)O MS-9638 c1cc(cc(c1)OC(F)(F)F)Nc2nc(cs2)C(=O)O MS-9639 Cc1c(sc(n1)Nc2cccc(c2)C(F)(F)F)C(=O)O MS-9640 c1cc(cc(c1)Nc2nc(cs2)C(=O)O)C(F)(F)F MS-9641 c1c(cc(cc1C(F)(F)F)Nc2nc(cs2)C(=O)O)C(F)(F)F MS-9642 Cc1c(sc(n1)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)O MS-9643 Cc1c(sc(n1)Nc2cc(cc(c2)Cl)Cl)C(=O)O MS-9644 c1c(cc(cc1Cl)Cl)Nc2nc(cs2)C(=O)O MS-9645 Cc1c(sc(n1)Nc2cc(ccc2Cl)Cl)C(=O)O MS-9646 c1cc(c(cc1Cl)Nc2nc(cs2)C(=O)O)Cl MS-9647 c1cc(c(cc1Cl)Cl)Nc2nc(cs2)C(=O)O MS-9648 Cc1c(sc(n1)Nc2ccc(cc2Cl)Cl)C(=O)O MS-9649 COc1ccc(cc1OC)Nc2nc(cs2)C(=O)O MS-9650 Cc1c(sc(n1)Nc2ccc(c(c2)OC)OC)C(=O)O MS-9651 Cc1ccc2c(c1)CCN2C(=S)N MS-9653 c1ccc2c(c1)CCCN2C(=S)N MS-9654 Cc1ccc2c(c1)CCCN2C(=S)N MS-9655 Cc1cc(cc2c1[nH]c3c2nnc(n3)S)Cl MS-9656 Cc1cc(cc2c1N(C(=O)C2=O)C)Cl MS-9657 Cc1cc(cc\2c1NC(=O)/C2=N\NC(=S)NCC=C)Cl MS-9658 Cc1cc(cc\2c1N(C(=O)/C2=N\NC(=S)N)C)Cl MS-9659 COc1ccc(cc1OC)NC(=O)c2ccccc2N MS-9660 COc1cccc(c1)/C=C/C(=O)OC MS-9662 COc1ccccc1/C=C/C(=O)OC MS-9663 COc1ccc(cc1O)/C=C/C(=O)OC MS-9664 COc1cc(ccc1O)CCC(=O)OC MS-9665 COC(=O)c1ccc(c(c1F)O)F MS-9667 Cc1cc(cc(c1)/C=N/O)C MS-9668 c1cc(c(cc1Cl)Cl)S(=O)(=O)C/C(=N/O)/N MS-9669 c1c2c(cc3c1c(=O)[nH]c3=O)c(=O)[nH]c2=O MS-9670 CC(C(=O)NN)S(=O)(=O)c1ccc(cc1Cl)Cl MS-9671 COC(=O)c1cc(c(c(c1)F)O)F MS-9672 CC(C(=O)NN)S(=O)(=O)c1cc(ccc1Cl)Cl MS-9673 CC(C(=O)NN)S(=O)(=O)c1ccc2ccccc2c1 MS-9674 c1ccc2cc(ccc2c1)S(=O)(=O)C/C(=N/O)/N MS-9675 CC(=O)c1cccc(c1)NC(=O)c2cccc(c2)N MS-9676 c1ccc(cc1)Nc2ccc(cc2)NC(=O)c3cccc(c3)N MS-9677 c1ccc(cc1)Oc2ccc(cc2)NC(=O)c3cccc(c3)N MS-9678 COc1ccc(cc1OC)NC(=O)c2cccc(c2)N MS-9679 COc1ccc(c(c1)NC(=O)c2cccc(c2)N)OC MS-9680 c1cc(cc(c1)N)C(=O)Nc2ccc3c(c2)OCO3 MS-9681 c1ccc(c(c1)C(=O)Nc2ccccc2N3CCOCC3)N MS-9682 CCOC(=O)c1c(cccc1Cl)N MS-9683 c1ccc(cc1)Oc2ccccc2NC(=O)c3ccc(cc3)N MS-9684 c1ccc(c(c1)C(=O)Nc2ccc(cc2)OC(F)(F)F)N MS-9685 c1ccc(cc1)Nc2ccc(cc2)NC(=O)c3ccccc3N MS-9686 CCCCOc1ccc(cc1)CC(=O)OCCCC MS-9819 COc1cccc(c1OC)/C=C/[N+](=O)[O-] MS-9820 c1cc(cc(c1)[N+](=O)[O-])/C=C/C(=O)O MS-9821 CCOC(=O)c1cc(ccc1C)Br MS-9822 CCOC(=O)c1cc(cc(c1)O)O MS-9823 CCOC(=O)/C=C/c1ccc(cc1)[N+](=O)[O-] MS-9824 COC(=O)c1ccc(cc1F)C#N MS-9825 COc1ccc(cc1F)/C=C/C(=O)O MS-9826 c1cc(c(c(c1)F)Cl)CO MS-9827 COC(=O)c1cc(ccc1Br)O MS-9828 Cc1c(cc(cc1O)C(=O)OC)O MS-9829 c1cc(ccc1/C=C/C(=O)O)Cl MS-9830 COc1ccc(cc1OC)/C=C/C(=O)c2ccccc2 MS-9831 CC1(OC(=O)C(=CNc2nc(cs2)c3ccc(cc3)Br)C(=O)O1)C MS-9832 COc1ccc(cc1)NCC(=O)c2ccc(cc2)Br MS-9833 CC\1=NN(C(=O)/C1=C\c2ccc3c(c2)OCO3)c4ccccc4 MS-9834 CC(C)(C)C(=O)/C(=C\Nc1ccc(cc1)F)/C#N MS-9835 CC(C)(C)C(=O)/C(=C\c1cccnc1)/C#N MS-9836 c1ccc(cc1)N/N=C\2/c3ccccc3NC2=O MS-9837 c1ccc(cc1)N2CCN(CC2)C=C3C(=O)c4ccccc4C3=O MS-9838 CC(=O)Nc1ccccc1NC2=CC(=O)CC(C2)(C)C MS-9839 CC(C)C(=O)Nc1ccccc1NC2=CC(=O)CC(C2)(C)C MS-9840 c1ccc2c(c1)c(=O)c(=NNC(=O)COc3ccc(cc3)F)c2=O MS-9841 c1ccc2c(c1)c(=O)c(=NNC(=O)COc3ccc(cc3Cl)Cl)c2=O MS-9842 CC1CC(=CC(=O)C1)Nc2ccccc2N MS-9843 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3ccc(cc3)I MS-9844 CC1(CC(=CC(=O)C1)N2CCN(CC2)C)C MS-9845 CC(C)C(=O)Nc1ccccc1NC2=CC(=O)CC(C2)c3ccccc3 MS-9846 c1ccc-2c(c1)Cc3c2[nH]nc3c4cccs4 MS-9847 CC(C)C(=O)n1c-2c(c(n1)c3cccs3)Cc4c2cccc4 MS-9848 c1ccc-2c(c1)Cc3c2n(nc3c4cccs4)C(=O)c5cccs5 MS-9849 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3cc(cc(c3)Cl)Cl)C2=O MS-9850 CC(C)c1c2c(n[nH]1)-c3ccccc3C2 MS-9851 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)Cl)Cl)/C#N MS-9852 c1ccc(cc1)C2CC(=CC(=O)C2)Nc3cc(cc(c3)Cl)N MS-9853 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3ccc(c(c3)Cl)Cl)C2=O MS-9854 CCOC(=O)C(=CNc1nc[nH]n1)C#N MS-9855 CCOC(=O)C(=CNc1nc(cs1)c2ccc(cc2)Br)C(=O)OCC MS-9856 c1c(cc(cc1Cl)Cl)NC(=C(C#N)C#N)C#N MS-9857 Cc1cc(nc(n1)NC=C(C#N)C#N)C MS-9858 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccccc2F)/C(=O)C MS-9860 Cc1ccc(cc1)N/C=C(/C#N)\C(=O)C(C)(C)C MS-9861 CC(C)(C)C(=O)/C(=C\Nc1ccccc1)/C#N MS-9862 CC1(Cc2c(c(n[nH]2)Nc3ccccc3)C(=NN)C1)C MS-9863 CC(C)C(=O)Nc1ccc-2c(c1)C(=O)c3c2nn(c3C(C)(C)C)C MS-9864 CCOC(=O)/C(=C\Nc1[nH]c(nn1)SC)/C#N MS-9865 c1cc(ccc1N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2Cl)Cl)OC(F)(F)F MS-9866 Cc1cc(c2ccccc2n1)N/C=C(/C#N)\S(=O)(=O)c3ccc(cc3Cl)Cl MS-9867 COC(=O)c1c(ccs1)NC(=O)NC2CCCCC2 MS-9868 Cc1ccc(cc1)NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F MS-9869 c1cc(ccc1NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)Cl MS-9870 Cc1ccccc1NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F MS-9871 c1ccc(cc1)CNC(=S)Nc2cc(ccc2N3CCOCC3)C(F)(F)F MS-9872 c1cc(c(cc1C(F)(F)F)NC(=O)NC2CCCCC2)N3CCOCC3 MS-9873 COc1ccc(cc1)NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F MS-9874 c1cc(ccc1NC(=S)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)Cl MS-9875 COc1ccc(cc1)NC(=O)NNC(=O)c2ccncc2 MS-9876 c1ccc(c(c1)NC(=O)NNC(=O)COc2ccc(cc2)OC(F)(F)F)Cl MS-9878 c1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2)OC(F)(F)F MS-9879 Cc1ccc(cc1)NC(=O)NCc2cccc(c2)C(F)(F)F MS-9881 Cc1ccccc1NC(=O)NCc2cccc(c2)C(F)(F)F MS-9882 Cc1ccccc1NC(=S)NCc2cccc(c2)C(F)(F)F MS-9883 Cc1ccc(cc1)CNC(=O)NNC(=O)c2ccncc2 MS-9884 CCc1ccc(cc1)OCC(=O)NNC(=O)Nc2cccc(c2Cl)Cl MS-9886 CCc1ccc(cc1)OCC(=O)NNC(=O)Nc2cccc(c2)C(F)(F)F MS-9887 c1cc(c(c(c1)Cl)Cl)NC(=S)NNC(=O)COc2ccc(cc2)F MS-9888 c1cc(cc(c1)NC(=S)NNC(=O)COc2ccc(cc2)F)C(F)(F)F MS-9889 CC(C)c1cccc(c1NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)C(C)C MS-9890 c1cc(c(c(c1)Cl)Cl)NC(=S)Nc2cc(ccc2N3CCOCC3)C(F)(F)F MS-9891 c1cc(c(c(c1)Cl)Cl)NC(=S)NNC(=O)COc2ccc(cc2)OC(F)(F)F MS-9892 c1cc(cc(c1)NC(=S)NNC(=O)COc2ccc(cc2)OC(F)(F)F)C(F)(F)F MS-9893 Cc1cccc(c1NC(=S)NCc2ccccc2Cl)C MS-9894 Cc1cccc(c1NC(=S)NCc2cccc(c2)C(F)(F)F)C MS-9895 COc1ccccc1NC(=S)NCc2cccc(c2)C(F)(F)F MS-9896 Cc1ccccc1NC(=O)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-9897 CCOc1ccccc1NC(=O)NNC(=O)COc2ccc(cc2)F MS-9898 CCc1ccc(cc1)OCC(=O)NNC(=O)Nc2ccc(cc2)OCC MS-9900 CCc1ccc(cc1)OCC(=O)NNC(=O)Nc2ccccc2OCC MS-9901 CCCNC(=O)NNC(=O)COc1ccc(cc1)CC MS-9902 CCOc1ccccc1NC(=O)N2CCc3c2cccc3 MS-9903 CCCNC(=O)N1CCc2c1cccc2 MS-9904 CCOc1ccc(cc1)NC(=O)N2CCc3c2cccc3 MS-9905 c1ccc(cc1)NC(=S)N2CCc3c2cccc3 MS-9906 Cc1ccc(cc1)NC(=O)N2CCc3c2cccc3 MS-9907 c1ccc2c(c1)CCN2C(=S)Nc3cccc(c3)C(F)(F)F MS-9908 Cc1ccccc1NC(=O)N2CCc3c2cccc3 MS-9909 c1ccc2c(c1)CCN2C(=O)NC3CCCCC3 MS-9910 Cc1ccc(cc1)NC(=S)N2CCc3c2cccc3 MS-9911 COc1cc(ccc1NC(=O)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)[N+](=O)[O-] MS-9912 COc1cc(cc(c1)OC)NC(=O)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-9913 c1cc(c(cc1NC(=O)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)Cl)Cl MS-9914 c1cc(ccc1NC(=S)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)[N+](=O)[O-] MS-9915 COc1ccc(c(c1)[N+](=O)[O-])NC(=O)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl MS-9916 c1cc(c(c(c1)Cl)NC(=O)NNC(=O)c2ccncc2)C(F)(F)F MS-9917 c1cc(c(cc1C(F)(F)F)NC(=O)Nc2ccc(c(c2)Cl)Cl)N3CCOCC3 MS-9918 c1cc(c(cc1C(F)(F)F)NC(=S)Nc2ccc(cc2Cl)Cl)N3CCOCC3 MS-9919 c1cc(c(cc1C(F)(F)F)NC(=O)Nc2cc(ccc2Cl)Cl)N3CCOCC3 MS-9920 c1cc(ccc1NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)Br MS-9921 CCc1ccc(cc1)OCC(=O)NNC(=S)Nc2ccc(cc2Cl)Cl MS-9922 CCc1ccc(cc1)OCC(=O)NNC(=O)Nc2cc(ccc2OC)Cl MS-9923 c1cc(ccc1NC(=S)NNC(=O)COc2ccc(cc2)I)[N+](=O)[O-] MS-9924 c1ccc2c(c1)c(c[nH]2)CCNC(=S)Nc3cccc(c3)C(F)(F)F MS-9925 Cc1ccccc1NC(=S)NCCc2c[nH]c3c2cccc3 MS-9926 c1ccc(cc1)NC(=S)NCCc2c[nH]c3c2cccc3 MS-9927 CCc1cccc(c1NC(=O)NCCc2c[nH]c3c2cccc3)CC MS-9928 Cc1ccccc1NC(=O)NCCc2c[nH]c3c2cccc3 MS-9929 CCCCCCNC(=O)NCCc1c[nH]c2c1cccc2 MS-9930 Cc1cccc(c1NC(=S)NCCc2c[nH]c3c2cccc3)C MS-9931 c1ccc2c(c1)c(c[nH]2)CCNC(=S)Nc3ccc(cc3Cl)Cl MS-9932 CCc1ccc(cc1)OCC(=O)NNC(=O)NCC(=O)OCC MS-9933 CCCCOC(=O)CNC(=O)NNC(=O)c1ccncc1 MS-9934 CCOc1ccc(cc1)/C=C/2\C(=O)NC(=O)N2 MS-9935 Cc1ccccc1NC(=O)N2CCN(CC2)C(=O)Nc3ccccc3C MS-9936 Cc1ccc(cc1)NC(=O)N2CCN(CC2)C(=O)Nc3ccc(cc3)C MS-9937 Cc1ccccc1NC(=O)N2CCN(CC2)c3cc(ccc3C)Cl MS-9938 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccn3 MS-9939 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3cc(ccc3C)Cl MS-9940 CCOC(=O)N1CCN(CC1)C(=O)Nc2ccc(cc2)C MS-9941 Cc1ccc(cc1)NC(=O)NCCN2CCN(CC2)C(=O)Nc3ccc(cc3)C MS-9942 Cc1ccccc1NC(=O)N2CCN(CC2)C/C=C/c3ccccc3 MS-9943 Cc1ccccc1NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 MS-9944 Cc1ccccc1NC(=O)N2CCN(CC2)c3ccccc3 MS-9945 Cc1ccccc1NC(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl MS-9946 Cc1ccccc1NC(=O)N2CCN(CC2)c3ccc(cc3)F MS-9947 Cc1ccc(cc1)NC(=O)N2CCN(CC2)C/C=C/c3ccccc3 MS-9948 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3cc(ccc3C)C MS-9949 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(c(c3)Cl)Cl MS-9950 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cc3)F MS-9951 c1ccnc(c1)N2CCN(CC2)C(=S)NC3CCCCC3 MS-9952 c1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccn3 MS-9953 c1ccnc(c1)N2CCN(CC2)C(=S)Nc3ccc(cc3)Cl MS-9954 CCOC(=O)CNC(=O)N1CCN(CC1)c2ccccn2 MS-9955 CNC(=S)N1CCN(CC1)C=O MS-9956 c1cc2c(cc1CN3CCN(CC3)C(=O)NC4CCCCC4)OCO2 MS-9957 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=O)Nc3ccc4c(c3)OCO4 MS-9958 c1ccc(cc1)/C=C/CN2CCN(CC2)C(=S)Nc3ccc(cc3)Cl MS-9959 c1cc(sc1)CC(=O)NN MS-9960 COc1ccc(cc1)Nc2nnc(o2)c3ccccc3NC(=S)Nc4cccc(c4)C(F)(F)F MS-9961 CC1(CC(=CC(=O)C1)Nc2cccc(c2)N)C MS-9962 CC(C)(C)c1c2c(nn1C(=O)c3ccccc3)-c4ccccc4C2=O MS-9963 CC(=O)c1ccc(cc1)NC2=CC(=O)CC(C2)(C)C MS-9964 c1cc(cc(c1)[N+](=O)[O-])NC2=C(C(=O)CCC2)[N+](=O)[O-] MS-9965 CC1(CC(=C(C(=O)C1)C(=S)Nc2ccccc2)NCc3ccccc3)C MS-9966 Cc1c(sc(n1)Nc2ccccc2)/C(=N\O)/C MS-9967 CC(C)(C)c1c2c(nn1S(=O)(=O)c3ccccc3)-c4ccccc4C2=O MS-9968 CCCCCC(=O)n1c(c2c(n1)-c3ccccc3C2=O)C(C)(C)C MS-9969 c1ccc2c(c1)NC3(N2)CCCCC3 MS-9970 CC(=NO)c1ccc(cc1)NC=C2C(=O)CC(CC2=O)(C)C MS-9971 CC1(CC(=C(C(=O)C1)C(=O)Nc2ccccc2)Nc3ccc(cc3)Cl)C MS-9972 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)Cl)C MS-9973 c1ccc(cc1)c2c3c(nn2C(=O)c4ccccc4)-c5ccccc5C3=O MS-9974 c1ccc2c(c1)/C(=N/c3ccc(cc3)Cl)/C(=O)N2CN4CCOCC4 MS-9975 CC1(CC(=O)C(=CNc2ccc(cc2)Br)C(=O)C1)C MS-9976 c1ccc(c(c1)C(=O)O)NC2=C(C(=O)CCC2)Br MS-9977 CC1(CC(=C(C(=O)C1)Br)Nc2ccccc2[N+](=O)[O-])C MS-9978 c1cc(cc(c1)N/C(=C/C(=O)C(F)(F)F)/c2cccs2)C(F)(F)F MS-9979 c1cc(ccc1NC2=C(C(=O)CCC2)Cl)Cl MS-9980 c1ccc(cc1)NC2=CC(=[NH+]c3ccccc3)c4c2cccc4.[Cl-] MS-9981 c1ccc(cc1)NC2=CC(=O)c3c2cccc3 MS-9982 c1cc(ccc1N)NC2=CC(=O)CCC2 MS-9983 CC(=O)Nc1ccc(cc1)NC2=C(C(=O)CCC2)Cl MS-9984 c1cc(ccc1NC2=CC(=O)CCC2)Cl MS-9985 COc1cc(ccc1NC2=CC(=O)CCC2)[N+](=O)[O-] MS-9986 c1cc(ccc1NC2=C(C(=O)CCC2)Br)Cl MS-9987 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)N(c4ccccc4)C(C)C MS-9988 c1cc(cnc1)/C=N/c2ccc3c(c2)OCO3 MS-9989 CC(C)c1ccc(cc1)CNc2ccc3c(c2)OCO3 MS-9990 COc1ccc(cc1)Nc2nnc(o2)c3ccccc3N MS-9991 c1ccc(c(c1)C(=O)NNC(=S)Nc2ccc(cc2)Cl)N MS-9992 c1ccc(c(c1)c2nnc(o2)Nc3ccc(cc3)Cl)N MS-9993 c1ccc(cc1)NC(=O)NC(=S)NC(=O)c2ccc(cc2)Cl MS-9994 COc1ccc(cc1)NC(=S)NNC(=O)Cc2c[nH]c3c2cccc3 MS-9995 Cc1ccccc1NC(=S)NNC(=O)Cc2c[nH]c3c2cccc3 MS-9996 Cc1ccccc1NC(=S)NNC(=O)c2cccs2 MS-9997 CC(=O)Nc1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccccc2 MS-9998 Cc1ccccc1n2c(nnc2S)c3cccs3 MS-9999 c1cc2cccnc2c(c1)S(=O)(=O)Oc3c(cc(cc3Cl)Cl)Cl NA-0201 c1cc(ccc1S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl)Br NA-0202 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0209 c1cc(cc(c1)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl)C(F)(F)F NA-0211 c1cc(ccc1OC(F)(F)F)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0216 c1ccc(c(c1)C#N)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0219 c1cc(sc1S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl)Br NA-0226 c1ccc(cc1)CS(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0229 CCS(=O)(=O)Oc1c(cc(cc1Cl)Cl)Cl NA-0230 c1ccc(c(c1)F)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0233 c1cc(ccc1F)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0238 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0239 c1ccc2cc(ccc2c1)S(=O)(=O)Oc3c(cc(cc3Cl)Cl)Cl NA-0241 Cc1nc(cn1C)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0243 COc1ccc(cc1S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl)Br NA-0248 CCCCS(=O)(=O)Oc1c(cc(cc1Cl)Cl)Cl NA-0250 CCCS(=O)(=O)Oc1c(cc(cc1Cl)Cl)Cl NA-0251 c1ccc(cc1)/C=C/S(=O)(=O)Oc2c(cc(cc2Cl)Cl)Cl NA-0252 CC(C)(C)OC(=O)NCC(C(=O)OC)O NA-0260 c1cncc(c1C(=O)O)Br NA-0700 c1ccc2c(c1)CNC3(N2)c4ccccc4NC3=O NA-0701 c1cc(ccc1SC2CCNCC2)Br.Cl NA-0702 c1ccc2c(c1)c3c([nH]2)c4ccccc4[nH]c3=O NA-0704 c1cc(ccc1C(C=O)C=O)Cl NA-0705 c1cc(cc(c1)S)C(=O)O NA-0707 c1cc(c(cc1N2CCCC2)Cl)C(=O)NN NA-0708 CCOC(=O)c1c(con1)C(=O)c2ccc(cc2)Cl NA-0710 CCOC(=O)c1c(con1)C(=O)c2ccc3ccccc3c2 NA-0711 COC(=O)c1ccc(cc1Cl)N2CCCCC2 NA-0712 c1ccn(c1)c2ccc3c(c2)cn[nH]3 NA-0800 CC1CCCN(C1)C/C(=N/O)/N NA-0801 c1cc(c(cc1F)Br)NC(=O)CCl NA-0802 c1ccc(c(c1)C=O)n2cccn2 NA-0803 CCOC(=O)c1c(ccs1)Oc2ncc(cn2)Br NA-0804 c1cnc(nc1)Oc2ccc(cc2)C#N NA-0805 CCC(C)C(C(=O)O)N1Cc2ccccc2C1=O NA-0808 c1cc(cc(c1)n2cccn2)C=O NA-0809 CC(=O)c1ccc(c(c1)OC)Oc2ncccn2 NA-0810 CC(=O)N1CCCN(CC1)Cc2cnc(s2)Cl NA-0811 c1cc(c(nc1)C(=O)O)C(F)(F)F NA-0812 COC(=O)[C@@H]1C[C@@H](CCN1)O NA-0814 c1ccc2c(c1)nc(s2)C(=O)NN NA-0815 C/C(=C\C(=O)c1ccc(cc1)Oc2ncccn2)/N(C)C NA-0817 c1ccc(cc1)CN2CC3CCCC(C3C2)N NB-0206 CC(=O)c1ccc(nc1)N2CCOCC2 NB-0600 COc1cc(ccc1[N+](=O)[O-])N2CCNCC2 NB-0700 c1cc(ncc1[N+](=O)[O-])N2CCN(CC2)CCO NB-0701 c1cc(ncc1C#N)N2CCN(CC2)CCO NB-0702 c1cc(ccc1c2csc(n2)N3CCC(CC3)C(=O)O)Cl NB-0704 CNc1ccc(c(c1)OC)[N+](=O)[O-] NB-0705 CN(C)c1ccc(c(c1)OC)[N+](=O)[O-] NB-0707 COc1cc(ccc1[N+](=O)[O-])N2CCOCC2 NB-0708 c1ccc(cc1)c2c(sc(n2)N)Br.Br NB-0710 COC(=O)c1cc(cnc1N2CCOCC2)Br NB-0711 COC(=O)c1cc(cnc1N2CCCCC2)Br NB-0712 c1c(cnc(c1C(=O)O)N2CCOCC2)Br NB-0713 c1c(cnc(c1C(=O)O)N2CCCCC2)Br NB-0717 Cc1nc(cc(n1)Cl)N(C)C NB-0718 Cc1nc(cc(n1)Cl)NCCO NB-0720 Cc1nc(cc(n1)Cl)NCc2ccccc2 NB-0721 c1cc(ccc1CCl)n2cncn2 NB-0800 COC(=O)c1ccc(cc1)C2NCCS2 NB-0802 c1cc(c(cc1[N+](=O)[O-])CO)N2CCOCC2 NB-0803 c1cc(c(cc1Br)CO)N NB-0807 c1cc2c(cc1Br)COC(=O)N2 NB-0808 CSc1ccccc1OCC(=O)O NB-0810 c1ccnc(c1)CCCl NB-0813 c1c(cn[nH]1)[N+](=O)[O-] NB-0818 c1(c([nH]nc1Br)Br)[N+](=O)[O-] NB-0819 c1ccc(cc1)Cn2c(c(c(n2)Br)[N+](=O)[O-])Br NB-0821 c1cc(c(cc1[N+](=O)[O-])CO)N2CCCCC2 NB-0824 CNc1c(c(nn1Cc2ccccc2)Br)[N+](=O)[O-] NB-0828 c1cnc(cc1Cl)C=O NB-5000 CC(C)c1nc(no1)c2ccnc(n2)N3CCNCC3.Cl.Cl NC-0048 Cc1nc(no1)c2ccnc(n2)N3CCNCC3.Cl.Cl NC-0087 CCOC(=O)c1ccc(cc1)OC(F)F NC-0225 CCOC(=O)N/N=C/CCl NC-0700 CCc1ccc(cc1)c2cc([nH]n2)N NC-0703 COC(=O)c1ccc(nc1Cl)Cl NC-0704 c1ccc(cc1)c2c(cc(nn2)Cl)Br NC-0705 CCc1ccc(cc1)c2cc(on2)N NC-0706 COc1ccc(c(n1)Cl)C(=O)O NC-0707 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2cccc(c2)[N+](=O)[O-] NC-0709 c1cc(c(nc1)N2CCNCC2)C#N NC-0712 CC(C)(C)OC(=O)Nc1cnccc1C(=O)O NC-0713 CC(C)(C)OC(=O)N1CCN(CC1)CCOc2cccc(c2)N NC-0714 c1cncc(c1CO)N NC-0715 CCOC(=O)c1c(n2cc(ccc2n1)[N+](=O)[O-])Br NC-0716 CNc1ccc(c(c1)C(=O)OC)[N+](=O)[O-] NC-0717 COc1cnc(nc1Cl)c2ccccc2 NC-0718 c1cc(nc2c1c(n[nH]2)N)C3CC3 NC-0719 Cn1c2c(ccc(n2)C3CC3)c(n1)N NC-0720 c1cc2c(cc1F)cc(s2)CO NC-0721 c1cc2cc(sc2c(c1)F)CO NC-0722 CN(C)c1ccc(c(c1)C(=O)OC)[N+](=O)[O-] NC-0723 c1cc(cc2c1cc(s2)CO)Cl NC-0727 c1cc(c(cc1C(F)(F)F)O)[N+](=O)[O-] NC-0728 COC(=O)c1cc(ccc1[N+](=O)[O-])N2CCOCC2 NC-0729 COc1cc(ccn1)CO NC-0735 COC(=O)c1c(c2ccc(nc2s1)C3CC3)N NC-0737 Cc1cc(cc(c1)COc2ccc(cc2Br)C=O)C NC-0738 Cc1cc(c(cc1OC)N)Br NC-0740 c1cc2c(cc1C(F)(F)F)cc(s2)C=O NC-0741 c1cc(c(cc1N2CCOCC2)C(=O)O)[N+](=O)[O-] NC-0742 CC(C)(C)OC(=O)N1CCN(CC1)c2c(ccc(n2)C3CC3)C#N NC-0743 COC(=O)c1cc(ccc1OCC#C)Br NC-0744 c1ccc2c(c1)NCC(O2)C(=O)O NC-0746 c1cc(c(cc1N2CCOCC2)C(=O)NN)[N+](=O)[O-] NC-0749 CSc1nccc(n1)NN NC-0750 CCOC(=O)c1cc(c(nc1Cl)Cl)F NC-0751 CCOC(=O)N/N=C/CBr NC-0752 COC(=O)c1cc(ccc1O)C#N NC-0753 c1cc2c(cc(s2)CO)c(c1)Cl NC-0754 c1cc2nccn2cc1F NC-0755 CCOC(=O)c1cn2cc(ccc2n1)F NC-0761 CCOC(=O)CC(C(C)[N+](=O)[O-])C(=O)OCC NC-0762 Cc1cc(cc(c1)COc2ccc(cc2Br)CO)C NC-0763 COc1cc(cc(c1Cc2ccc(cc2)Br)OC)N NC-7058 Cc1cc(c(c(c1)[N+](=O)[O-])O)C(=O)OC ND-0003 CC(C)NC(=O)NCc1c(cc(cn1)Cl)C(F)(F)F ND-0004 CC(C)(C)[Si](C)(C)Oc1c(cc(c(c1Cl)O)Cl)Cl ND-0012 c1c(c(cc(c1O)Br)Cl)C(F)(F)F ND-0013 c1cc(c(cc1N2CCNCC2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-].Cl.Cl ND-0018 c1c(cc(c(c1C(F)(F)F)N)I)[N+](=O)[O-] ND-0021 CN(C)c1c(c2ccc(cc2[nH]1)Br)C=O ND-0025 Cc1cc(c(c(c1)N)O)C(=O)OC ND-0035 Cc1cc(c(c(c1)[N+](=O)[O-])OC)C(=O)OC ND-0036 CC(=O)N1CCN(CC1)c2ccc(c(c2)C(=O)NCc3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] ND-0038 COC(=O)c1cc(cc2c1OCC(=O)N2)Br ND-0042 c1c(cc(c(c1C(F)(F)F)N)Br)[N+](=O)[O-] ND-0047 Cc1cc(c(c(c1)N)OC)C(=O)OC.Cl ND-0048 Cc1cc(c(c(c1)N)OCc2ccccc2)C(=O)OC.Cl ND-0049 Cc1cc(c2c(c1)NC(=O)CO2)C(=O)OC ND-0052 c1cc2c(cc1Br)NC(=O)C23CCCCC3 ND-0055 COc1c(cc(cc1N)Br)C(=O)OC.Cl ND-0059 c1c(c(cc2c1nc(s2)CC#N)Cl)C(F)(F)F ND-0062 c1cc2c(cc1Br)[nH]c(c2C=O)Cl ND-0065 COc1cc(cc(c1O)[N+](=O)[O-])C(=O)OC ND-0066 Cc1cc(c2c(c1)[nH]c(=O)o2)C(=O)OC ND-0070 CN(CC(=O)NCc1c(cc(cn1)C(F)(F)F)Cl)c2ccc(cc2)Cl ND-0073 COC(=O)C1CC2(c3ccccc3NC2=O)NC1 ND-0200 c1cc(c(nc1)Cl)/C(=N/O)/N ND-0202 CNC(=O)c1cc(ccn1)Oc2ccc(cc2)N ND-0205 c1cc(c(nc1)Cl)c2nc(on2)C(F)(F)F ND-0206 c1c(c(cnc1Cl)C(F)(F)F)Cl ND-0209 CC(C)c1ccc(c(n1)N2CCN(CC2)C(=O)OC(C)(C)C)C#N ND-0229 c1cc2c(c(c1)[N+](=O)[O-])CCC2=O ND-0700 c1cc2c(c(c1)N)CCC2=O ND-0704 CNc1nc2ccc(cc2o1)[N+](=O)[O-] ND-0706 CC(C)c1c(cc(c(=O)[nH]1)C#N)I ND-0707 c1ccc(c(c1)NCc2ccc(cc2)N)[N+](=O)[O-] ND-0708 CC(C)(C)OC(=O)N1CCC2(CC1)NC(=O)CS2 ND-0710 COC(=O)c1cccc(c1)OCCN2CCN(CC2)Cc3ccccc3 ND-0711 CC(C)c1c(cc(c(=O)[nH]1)C#N)Cl ND-0713 c1ccc(c(c1)CNc2ccccc2[N+](=O)[O-])N ND-0714 CNc1cccc(c1C#N)F ND-0716 CC(C)c1c(cc(c(n1)Cl)C#N)I ND-0717 C1CNCCC12NC(=O)CS2.Cl ND-0718 CCNc1cccc(c1C#N)F ND-0719 c1ccc(cc1)C(CNc2ccc(cc2)Br)O ND-0720 CNc1cccc2c1c(nn2C)N ND-0721 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2ncnc3Cl NE-0001 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCN(CC2)Cc3ccc(cc3)OC.Cl NE-0010 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCN(CC2)Cc3cccc(c3)C(F)(F)F.Cl NE-0011 CN(C)c1c(c2c([nH]1)cccc2Br)C=O NE-0014 CC(=O)Nc1ccccc1C(=O)NCCc2c(cc(cn2)C(F)(F)F)Cl NE-0016 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC NE-0019 Cc1cccc(c1)S(=O)(=O)N2CCN(CC2)c3cc(c(cc3[N+](=O)[O-])F)C NE-0021 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCN(CC2)C(=O)c3ccc(cc3)C(F)(F)F NE-0022 CC(C)(C)OC(=O)N1CCC(CC1)COc2ccc(cc2OC)C(=O)OC NE-0025 COc1cc(ccc1OCC2CCNCC2)C(=O)OC.Cl NE-0026 CN1CCC(CC1)COc2ccc(cc2OC)C(=O)OC NE-0027 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCN(CC2)C(=O)Nc3ccc(cc3)OC NE-0029 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl NE-0030 Cc1cc(c(cc1F)[N+](=O)[O-])N2CCN(CC2)C(=O)OC(C)(C)C NE-0037 c1cc2c(c(c1)Br)CC(=O)N2 NE-0050 C[C@H]1CCN(C[C@H]1NC(=O)OC)Cc2ccccc2.Cl NE-0052 c1cc2c(c(c1)Br)c(c([nH]2)Cl)C=O NE-0053 CC(=O)c1ccc(c(c1)OC)OCCCCl NE-0054 c1ccc(cc1)C(c2ccccc2)SC(=N)N.Br NE-0059 CC(C)(C#N)NC(=O)OCc1ccccc1 NE-0200 CC(C)(c1[nH]nnn1)NC(=O)OCc2ccccc2 NE-0207 CC(C)(/C(=N/O)/N)NC(=O)OCc1ccccc1 NE-0208 CC(C)(c1nc(c(c(n1)O)O)C(=O)OC)NC(=O)OCc2ccccc2 NE-0215 Cn1c2ccc(cc2[nH]c1=O)[N+](=O)[O-] NE-0700 Cc1ncc(cn1)C(=O)OC NE-0701 c1cnc(nc1)C(=N)N.Cl NE-0702 COC(=O)c1cnc(nc1)SC NE-0705 c1cc(ccc1C2CN=C(O2)N)Br NE-0706 CNc1ccc(cc1[N+](=O)[O-])CO NE-0707 CN1C(c2cc(ccc2C1=O)Br)C#N NE-0709 COC(=O)c1cnc(nc1)S(=O)(=O)C NE-0711 c1cc(c(nc1)CCl)Br NE-0712 CNc1ccc(cc1[N+](=O)[O-])CCl NE-0713 COc1ccc(c(n1)Cl)C(=O)N NE-0714 CCOC(=O)c1cnc(nc1O)c2ccncc2 NE-0719 COC(=O)c1cc(nc(n1)Cl)N NE-0720 c1cc(c(nc1)Cl)c2ccnc(n2)N NE-0721 COc1ccc(c(n1)Cl)C#N NE-0722 c1cc(c(nc1)n2c(c(cn2)C#N)N)C(F)(F)F NE-0723 Cn1c2ccc(cc2nc1CCl)[N+](=O)[O-] NE-0724 CC(c1nc2cc(ccc2n1C)[N+](=O)[O-])O NE-0727 CNc1nc2cc(ccc2n1C)[N+](=O)[O-] NE-0728 c1c2cc([nH]c2ncc1C(F)(F)F)C(=O)NCC3CC3 NF-0003 COC(=O)N1CCN(CC1)C(=O)c2cc3cc(cnc3[nH]2)C(F)(F)F NF-0005 c1(nnc(s1)Br)Br NF-0010 Cc1cc2c(c(c1O)Br)C(=O)NC2 NF-0011 c1nnc(s1)N NF-0014 c1cc(c(cc1C(=O)O)S(=O)(=O)NC(=N)c2c(cc(cn2)C(F)(F)F)Cl)F NF-0015 CCc1cn(nn1)c2ccc(cc2)[N+](=O)[O-] NF-0019 Cc1ccc(cc1OC)C(=O)OC NF-0026 Cc1c(cccc1OC)C(=O)NC2CC2 NF-0027 Cc1c(cccc1OC)C(=O)OC NF-0031 C1CCN(CC1)c2nnc(s2)Br NF-0036 CCc1cn(nn1)c2ccc(cc2)N NF-0046 Cc1c(cccc1OC)C(=O)NC2CCCC2 NF-0049 Cc1ccc(cc1OC)C(=O)NC2CC2 NF-0052 COc1cc(ccc1F)C(=O)NC2CC2 NF-0053 C[C@@H]1CN(C[C@@H](O1)C)c2nnc(s2)Br NF-0054 CCN(CC)c1nnc(s1)Br NF-0055 c1ccc(cc1)COC(=O)N2CCC(=CC#N)CC2 NF-0215 c1c(n[nH]c1N)C#N NF-0227 c1ccc2c(c1)C(CS2(=O)=O)O NF-0702 c1c(cnc(c1Br)N2CCOCC2)Br NF-0705 c1cc(c(cc1C2OCCCO2)C#N)F NF-0707 c1cnc(c2c1[nH]nc2)Cl NF-0710 CS(=O)(=O)C1(CC1)C(=O)O NF-0711 CCOC(=O)c1cc(cc(n1)C)Cl NF-0713 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cc(cn2)Br)Br NF-0714 c1cc2c(cc1C3OCCCO3)c(n[nH]2)N NF-0716 c1ccc(cc1)c2nc(cc(n2)Cl)C(=O)O NF-0717 COc1cc(ccc1[N+](=O)[O-])C(=O)N NF-0718 CCOC(=O)c1cn(c(=O)c(c1Cl)Br)C NF-0720 Cc1cc(cc(n1)C(=O)O)Cl NF-0723 c1c([nH]nc1C(F)(F)F)C2CC2 NF-0724 c1cc(c(cc1C=O)C#N)N NF-0725 c1c(cnc2c1[nH]nc2N)C(F)(F)F NF-0730 c1cnc(c(c1I)C=O)F NF-0731 CNc1ncc(c(n1)C(=O)O)Br NF-0732 c1c(cc(nc1C(F)(F)F)C(F)(F)F)CO NF-0733 CCOC(=O)c1cnc(c(c1Cl)[N+](=O)[O-])OC NF-0734 c1c(c(cnc1Cl)Cl)C(F)(F)F NF-0737 c1ccc(cc1)c2ccc(cn2)CO NF-0738 CCOC(=O)c1c(nc2ccccc2n1)C NF-0739 c1cc2cn[nH]c2nc1 NF-0740 CC(C)/C=C\CCCCC(=O)NCc1ccc(c(c1)OC)O NG-0020 c1ccc(c(c1)C(F)(F)F)OCc2nnc3n2cc(cc3Cl)C(F)(F)F NG-0049 Cc1cc(nc(n1)NC(=O)NS(=O)(=O)c2ccccc2C(=O)OCC3COC(O3)C)C NG-0209 Cc1cc(no1)N NG-0401 Cc1cc(no1)C(=O)OC NG-0403 Cc1cc(on1)c2ccccc2 NG-0404 Cc1c(noc1N)C NG-0406 CC(C)(C)c1cc(no1)N NG-0408 Cc1cc(no1)CO NG-0409 c1cc2c(cc1Br)CCC(=O)N2 NG-0703 Cc1c(ccc(c1C#N)Br)OC NG-0704 COC(=O)c1cc2ccc(cc2s1)[N+](=O)[O-] NG-0706 CNc1c(c(nc(n1)Cl)C(=O)OC)Cl NG-0707 CCOC(=O)c1c(cccn1)C2OCCO2 NG-0708 c1(c(c(nc(c1Cl)Cl)C(F)(F)F)Cl)C(F)(F)F NG-0709 CNc1c(cc(cn1)Br)C(=O)NC NG-0710 c1c2c(cc(c1Br)C(F)(F)F)[nH]cc2I NG-0712 COC(=O)c1cc(ccc1F)CCl NG-0713 Cc1c(ccc(c1C(=O)NN)Br)OC NG-0714 CCOC(=O)c1c([nH]cn1)C(C)(C)C NG-0715 c1c2c(cc(c1I)O)NC(=O)CC2 NG-0716 c1c(c(cnc1N2CCNCC2)Cl)C(F)F NH-0224 C=Cc1ccc(nc1)Cl NK-0020 Cn1cc(c2c1cccc2)C=O NS-00004 COc1ccc(cc1)/C=N/c2ccc(cc2)OC NS-00005 COc1cccc(c1O)C=O NS-00006 CCOC(=O)c1c([nH]c2c1cc(cc2)O)C NS-00007 CCOC(=O)c1cc2cc(ccc2[nH]1)C NS-00008 c1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)C=O NS-00010 CCOC(=O)c1c([nH]c2c1cc(cc2)OS(=O)(=O)C(F)(F)F)C NS-00011 CC(C)[C@@H](C(=O)N)NC(=O)OCc1ccccc1 NS-00012 COc1ccc2c(c1O)cc3n2CCC3 NS-00013 Cc1cc2c(s1)ccc(c2C=O)OC NS-00014 COc1ccc(cc1OCc2ccccc2)[N+](=O)[O-] NS-00015 Cc1c2c(ccc(c2[N+](=O)[O-])OC)on1 NS-00016 CCSC(=N)Nc1ccc(cc1)O.I NS-00017 CC(=O)OC[C@@H](C(=O)OCc1ccc(cc1)[N+](=O)[O-])N.Cl NS-00018 Cc1cc(n(c1/C=C\2/c3ccccc3NC2=O)Cc4ccccc4)C NS-00019 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)S(=O)(=O)C NS-00020 CC(C)(C)OC(=O)N[C@H]1CC=C(C1)C(=O)O PS-1000 CC(C)(C)OC(=O)N[C@@H]1CC=C(C1)C(=O)O PS-1001 CC(C)(C)OC(=O)N[C@H]1CC[C@H](C1)CO PS-1002 CC(C)(C)OC(=O)N[C@@H]1CC[C@@H](C1)CO PS-1003 CC(C)(C)OC(=O)N[C@H]1CC[C@@H](C1)CO PS-1004 CC(C)(C)OC(=O)N[C@@H]1CC[C@H](C1)CO PS-1005 CC(C)(C)OC(=O)N[C@H]1CC=C(C1)CO PS-1006 CC(C)(C)OC(=O)N[C@@H]1CC=C(C1)CO PS-1007 CC(C)(C)OC(=O)N[C@@H]1CCC[C@@H]1CO PS-1008 CC(C)(C)OC(=O)N[C@@H]1CCC[C@H]1CO PS-1009 CC(C)(C)OC(=O)N[C@H]1CC[C@H](C1)C(=O)OC PS-1010 CC(C)(C)OC(=O)N[C@@H]1CC[C@@H](C1)C(=O)OC PS-1011 CC(C)(C)OC(=O)N[C@H]1CC[C@@H](C1)C(=O)OC PS-1012 CC(C)(C)OC(=O)N[C@@H]1CC[C@H](C1)C(=O)OC PS-1013 CC(C)(C)OC(=O)N[C@H]1CC=C(C1)C(=O)OC PS-1014 CC(C)(C)OC(=O)N[C@@H]1CC=C(C1)C(=O)OC PS-1015 CC(C)(C)OC(=O)N[C@@H]1C[C@@H](C=C1)C(=O)OC PS-1016 CC(C)(C)OC(=O)N[C@H]1C[C@H](C=C1)C(=O)OC PS-1017 CC(C)(C)OC(=O)N[C@H]1CCC[C@@H]1C(=O)OC PS-1018 Cc1ccc(cc1O)N PS-3000 c1cc(ccc1CCO)N PS-3001 C1C2CC3CC1CC(C2)C3=O PS-3002 c1cc(c(cc1Cl)C(=O)N)[N+](=O)[O-] PS-3004 CSc1ccccc1Cl PS-3005 c1cc(c(cc1Br)N)Br PS-3006 c1cc(c(c(c1)Cl)N)Cl PS-3007 CC(=O)c1ccccc1[N+](=O)[O-] PS-3008 COc1cc(ccc1N)[N+](=O)[O-] PS-3009 Cc1cc(cc(c1)S)C PS-3010 Cc1cc(cc(c1)N)C PS-3011 COc1ccc(c(c1)OC)CC(=O)O PS-3012 c1cc(c(c(c1)O)O)C(=O)O PS-3013 c1cc(c(cc1O)Cl)Cl PS-3014 c1c(cc(cc1Cl)Cl)O PS-3015 CC(=O)c1cccc(c1)C(=O)O PS-3016 Cc1cc(ccc1C#N)NC(=O)C PS-3017 Cc1cc(ccc1C(=O)C)NC(=O)C PS-3018 CN(C)c1ccc(c(n1)Cl)C(=O)O PS-3019 c1ccnc(c1)CCN2CCNCC2 PS-3020 Cc1c[n+](ccc1[N+](=O)[O-])[O-] PS-3021 c1cc(nnc1NN)Cl PS-3022 CCOC(CN1CCNCC1)OCC PS-3023 C1CCC(CC1)CCCN2CCNCC2 PS-3024 C1CN(CCN1)CCCC#N PS-3025 CC(=O)c1cc2c3ccccc3ccc2oc1=O PS-3026 CCOC(=O)c1c(c(sc1N)C)c2ccccc2 PS-3027 c1c(cnc(n1)N)[N+](=O)[O-] PS-3028 c1c(cncn1)Br PS-3029 Cc1cc(ccc1Br)N PS-3030 Cc1ccc(cc1O)[N+](=O)[O-] PS-3031 c1cc(cc(c1)Br)S(=O)(=O)N PS-3032 COc1cccc(c1)S PS-3033 c1cc(nc(c1N)Cl)Cl PS-3034 Cc1cc(c(cc1OC)Br)OC PS-3035 Cn1c(nnc1S)Cc2ccsc2 PS-3036 CC(C)(C)C(=CC#N)Cl PS-3037 C1C2CC3CC1CC(C2)(C3)CCC(=O)O PS-3038 c1c(nc(c(n1)N)Br)Br PS-3039 c1cc(c(nc1)NCCN)C(=O)O PS-3040 c1ccc(cc1)c2cc(n[nH]2)C(=O)O PS-3041 c1ccc(cc1)C(C(=O)O)Nc2ccccc2 PS-3042 c1ccc(cc1)CN2CCN(CC2)CCN PS-3043 c1ccnc(c1)C(CCCN)N PS-3044 c1cc(c(nc1)C=O)O PS-3045 C#Cc1ccccc1C=O PS-3046 C#Cc1cccc(c1)C=O PS-3047 C#Cc1ccc(cc1)C=O PS-3048 c1ccc(cc1)C2CCNc3ccccc3N2 PS-3049 c1ccc2c(c1)NCCC(=N2)c3ccco3 PS-3050 CC(C)[C@@H](C(=O)O)NC(=O)OCc1ccccc1 PS-3051 c1ccn2c(c1)ncc2[N+](=O)[O-] PS-3052 Cc1c2ccccn2cn1 PS-3053 c1cc(c(cc1C#N)[N+](=O)[O-])N PS-3054 CC(c1cccnc1)N PS-3055 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)C PS-3056 c1c(c(n[nH]1)C=O)Cl PS-3057 c1ccc(cc1)NC(C#N)c2ccncc2 PS-3058 Cc1csc(c1C#N)N PS-3059 CC(c1ccccn1)O PS-3060 c1cc(ccc1C(=O)N)C(=O)O PS-3061 c1cncc2c1ncc(c2)C(=O)O PS-3062 CC(C)(C)OC(=O)N(CCN)Cc1ccccc1 PS-3063 CC(C)(C)OC(=O)Cc1ccc(cc1)N PS-3064 COc1ccc(cc1)OCC(CN)O PS-3065 CC(c1ccco1)N PS-3066 c1ccc(cc1)CN2CCC(CC2)Nc3ccccc3N PS-3067 C1CCN2CCCC(C2C1)CO PS-3068 CC(=O)c1ccc(cc1)Br PS-3069 c1cc(ccc1NN)Br PS-3070 c1cc(cc(c1)S(=O)(=O)N)N PS-3071 c1cc(ncc1C(=O)O)NCCN PS-3072 COC(=O)Cc1ccc(cc1)N PS-3073 c1ccc2c(c1)NCCN2 PS-3074 Cc1cc(n(n1)C)C#N PS-3075 c1cc(c(cc1Cl)Cl)C2=NN=C(C2)C(=O)O PS-3076 CN1C2CCC1CC(C2)N PS-3077 c1ccc(cc1)C2CN(CCN2)c3ccc(cn3)C(=O)O PS-3078 Cc1[nH]c2cc(ccc2n1)C(=O)O PS-3079 c1ccc(cc1)N2CCNC2=O PS-3080 c1ccc(c(c1)N2CCNC2=O)[N+](=O)[O-] PS-3081 c1cc(ccc1CC#N)Br PS-3082 c1ccc(cc1)NC(C#N)c2cccc(c2)O PS-3083 c1c(cnc(c1Cl)N2CCNCC2)C(=O)O PS-3084 Cc1cc(n(n1)c2ccccc2C(=O)O)C PS-3085 c1ccc(cc1)c2[nH]c3cc(ccc3n2)C(=O)O PS-3086 c1c(nc(c(n1)N)N)Br PS-3087 COC(=O)c1cc([nH]n1)c2ccccc2 PS-3088 c1ccc(cc1)Nc2ccc(cn2)C(=O)O PS-3089 Cn1cc(c(n1)C=O)Br PS-3090 Cc1cc(cc(c1N)Cl)C(=O)O PS-3091 c1cc2nccn2nc1 PS-3092 c1cc(ncc1C(=O)O)Br PS-3093 c1cc2c(cc1Cl)sc(n2)N3CCNCC3 PS-3094 CC(C)(C)OCC(=O)O PS-3095 CN(C)C(=O)C(=O)O PS-3096 c1cc(ccc1C2SCCS2)OC/C(=N/O)/N PS-3097 c1cnccc1CN2CCC(CC2)C(=O)O PS-3098 c1cc(c(c(c1N)C#N)Cl)Cl PS-3099 COC(c1ccc(cc1)C(=O)OC)OC PS-3101 Cc1c(oc(c1C#N)N)C PS-3102 Cn1c2c(cn1)c(ncn2)Cl PS-3103 COC(=O)c1cccc(c1O)N PS-3104 c1cc2nc(cn2c(c1)Cl)C(=O)O PS-3105 c1ccn2c(c1)nc(c2Cl)C(=O)O.O.Cl PS-3106 c1c(c(cc(c1Cl)Cl)O)[N+](=O)[O-] PS-3107 c1cc(cc(c1)Cl)c2c(cc(=O)[nH]n2)Cl PS-3108 CCOC(=O)c1csc(n1)NC PS-3109 COc1ccc(c(c1)N)O PS-3110 CCOC(=O)c1cn2c(cccc2n1)N PS-3111 c1cc(c(cc1C#N)N)O PS-3112 CCCCc1[nH]cc(n1)CO PS-3113 CCOC(=O)c1c(n2ccccc2n1)Br PS-3114 Cn1c2ccc(cc2c(n1)N)Br PS-3115 Cn1cc(c(n1)/C(=N/O)/N)Br PS-3116 Cc1c2cc(c(nc2n(n1)C)Cl)C=O PS-3117 Cc1c(cn[nH]1)CCCN PS-3118 CC(C)(C)OC(=O)N1CCc2c(sc(n2)N)C1 PS-3119 CCNc1ccc(cc1N)Cl PS-3120 c1ccc(c(c1)CN2CCNCC2)C#N PS-3121 CCOC(=O)c1cnn(c1N)c2nc3ccccc3s2 PS-3122 c1ccc(cc1)S(=O)(=O)CC#N PS-3123 CN(C)C(=O)CN1CCNCC1 PS-3124 C1CCN(CC1)C(=O)CN2CCNCC2 PS-3125 Cc1cc(ccc1NC(=O)C)Cl PS-3126 Cc1ccc(cc1Cl)CN PS-3127 CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)O PS-3128 c1ccc2c(c1)cc(o2)C(=O)NN PS-3129 c1cc(ccc1OCCC#N)Br PS-3130 c1cc(ccc1CCCO)Cl PS-3131 CCCc1cnc(nc1)Cl PS-3132 c1cc(nc(c1)Cl)C(=O)O PS-3133 CCOC(=O)c1ccc(cc1)Br PS-3134 c1cscc1Cl PS-3135 c1ccc(cc1)/C=C/C=N/O PS-3136 c1ccc2c(c1)C(c3ccccc3S2)N4CCNCC4 PS-3137 CC(=O)Nc1ccc(cc1NC(=O)C)C(=O)O PS-3139 CC(=O)c1ccc-2c(c1)Cc3c2ccc(c3)C(=O)C PS-3140 c1cc(c(cc1C#N)N)N PS-3141 C1CCC2(CC1)C(=O)NC(=O)N2 PS-3142 c1c(cc(cc1Cl)Cl)C(=O)N PS-3143 c1c(cc(cc1Cl)Cl)S(=O)(=O)N PS-3144 c1c(cc(cc1Cl)Cl)C(=O)NN PS-3145 c1c(cc(c(c1C=O)O)Cl)Cl PS-3146 c1cc(nc(c1[N+](=O)[O-])Cl)Cl PS-3147 c1cc(c(cc1Cl)Cl)OC/C(=N/O)/N PS-3148 c1c(cc(nc1Cl)Cl)C(=O)O PS-3149 c1cc2c(cc1/C(=N/O)/N)CCO2 PS-3150 CC1(COC(=N1)c2cccnc2)C PS-3151 c1cc2c(cc[nH]2)cc1[N+](=O)[O-] PS-3152 Cc1cc(cc(n1)O)O PS-3153 COc1ccc(c(c1)S(=O)(=O)N)OC PS-3154 Cc1cc(n(n1)C)C(=O)N PS-3155 CCOC(=O)c1cc(nc(n1)Cl)C PS-3156 CCOC(=O)c1cc(c(c(c1)Cl)O)Cl PS-3157 c1cc(sc1)c2ccc(cc2)CO PS-3158 CCOC(=O)C(C)c1ccccc1 PS-3159 Cc1ccc2nc(c(n2c1)C(=O)O)C PS-3160 c1cc(c(nc1)N)O PS-3161 c1c2c(cc(c1Cl)S(=O)(=O)N)S(=O)(=O)NCN2 PS-3162 C1C2CC3(CC1CC(C2)(C3)O)C(=O)O PS-3163 Cc1ccc(c(n1)O)C(=O)O PS-3164 CCCCCn1c(nnc1S)O PS-3165 c1cc(cc(c1)O)CC(=O)O PS-3166 c1[nH]c2c(n1)[nH]cnc2=O PS-3167 Cc1cc(ccc1N)I PS-3168 CC(C)Oc1cc(ccc1OC)C(=O)O PS-3169 CC(C)c1cccc(c1)N PS-3170 CS(=O)(=O)c1ccc(cc1)O PS-3171 CC(C)n1c2ccc(cc2nn1)C(=O)O PS-3172 CC(C)c1ccc(c(c1)[N+](=O)[O-])N PS-3173 CCCOc1cc(ccc1OC)C(=O)O PS-3174 Cc1cccc(c1)/C(=N/O)/N PS-3175 COC(=O)c1ccc2c(c1)nns2 PS-3176 C[C@@]12[C@@](CC(=O)C1)(CC(=O)C2)C PS-3177 CC1(CCCCC1)C(=O)O PS-3178 CC1C(=O)CCC1=O PS-3179 COC(=O)Cc1ccc(c(c1)Cl)Cl PS-3180 Cc1ccc(cc1S(=O)(=O)N)[N+](=O)[O-] PS-3181 Cc1ccc(cc1)C#C PS-3182 CN1CCC(=O)CC1 PS-3183 CSc1ccccc1CN PS-3184 c1cc2c(cc1[N+](=O)[O-])c(c[nH]2)C=O PS-3186 CS(=O)(=O)c1ccc(cc1)Cl PS-3187 c1ccc(cc1)C#Cc2ccc(o2)C(=O)O PS-3191 c1ccc(cc1)c2nc(sn2)N3CCCNCC3 PS-3192 c1ccc(c(c1)C(=O)O)n2ccnc2 PS-3193 c1cc(cc(c1)N2CCCCC2)C(=O)O PS-3194 c1cc(ccc1N)S PS-3195 CSc1ccc(cc1)N PS-3196 CSc1ccc(cc1)C=O PS-3197 c1cc(cc(c1)S)O PS-3198 c1cc(ccc1[N+](=O)[O-])S PS-3199 CSc1ccc(cc1)[N+](=O)[O-] PS-3200 CC(=O)Nc1ccc(cc1)S PS-3201 c1cc(c(cc1Cl)N)S PS-3202 CC(C)(C)OC(=O)N1CCC(CC1)CC(=O)O PS-3203 C1CCN(C1)CCC2CCNCC2 PS-3204 C1CN(CCC1C(=O)O)C(=O)N PS-3205 COc1cccc(c1)C=O PS-3206 Cc1cc(nc(n1)C#N)C PS-3207 c1cc2ccnc(c2nc1)N PS-3208 CC(C)(C)OC(=O)NCc1ccc(cc1)C=O PS-3209 c1ccc(cc1)N(c2ccccc2)C(=O)N3CCNCC3 PS-3210 c1ncnc(n1)N2CCNCC2 PS-3211 CCCCCC(=O)N1CCNCC1 PS-3212 CS(=O)(=O)N1CCNCC1 PS-3213 CN(C)c1ccc(cc1)CO PS-3214 c1cc(c(cc1Br)Cl)N PS-3215 CC(C)(C)C(=O)N1CCNCC1 PS-3216 CCC(=O)N1CCNCC1 PS-3217 C1CCC(C1)CCCN2CCNCC2 PS-3218 C1CC(=O)N(C1=O)Cl PS-3219 COc1cc(ccc1C=O)O PS-3220 c1cc(c(cc1Br)N)Cl PS-3221 c1ccc(cc1)c2cccc(c2)N3CCNCC3 PS-3222 CC(C)(C)OC(=O)N1CCCC(C1)O PS-3223 c1cc(c(cc1[N+](=O)[O-])Cl)N2CCNCC2 PS-3224 CCN(CC)C1CCNCC1 PS-3225 CCOC(=O)c1c[nH]c(nc1=O)SC PS-3226 CN(C)C1CCNCC1 PS-3227 CCCN(CCC)C1CCNCC1 PS-3228 CN1CCN(CC1)CCO PS-3229 CN1CCN(CC1)CCCO PS-3230 CC1CCN(CC1)C2CCNCC2 PS-3231 Cc1ccnc(c1)N2CCNCC2 PS-3232 c1ccc(cc1)OCCCN2CCNCC2 PS-3233 CN(C)C(=O)N1CCNCC1 PS-3234 Cc1cc(nn1C)C(=O)O PS-3235 c1cc(c(cc1Cl)C(=O)O)[N+](=O)[O-] PS-3236 COc1ccc(c(c1)O)C=O PS-3237 COc1cc(c(cc1Br)OC)C=O PS-3238 Cc1cccnc1C(=O)O PS-3239 COc1ccc(cc1[N+](=O)[O-])N PS-3240 c1c(cc(cc1Cl)Cl)C(=O)O PS-3241 Cc1cc(ncc1[N+](=O)[O-])N PS-3242 CCOC(=O)c1ccc(cc1)N2CCNCC2 PS-3243 C1CN(CCN1)CCC(=O)O PS-3244 C1CCN(C1)C(=O)N2CCNCC2 PS-3245 CCOC(=O)CC1CCCNC1 PS-3246 C1CCN(CC1)S(=O)(=O)N2CCNCC2 PS-3247 CCCOCCN1CCNCC1 PS-3248 COc1ccc(c(c1)N)OC PS-3249 Cc1ccc(cc1)CN PS-3250 Cc1c(c(nnc1N)Cl)C PS-3251 COc1ccccc1O PS-3252 c1cc(nnc1)C(=O)O PS-3253 c1ccc2c(c1)c(cs2)CC(=O)O PS-3254 c1cc2ccc(nc2nc1)C(=O)O PS-3255 c1cc(cc(c1)S)N PS-3256 CN1CCN(C1=O)C PS-3257 c1cc2c(ccs2)cc1C=O PS-3258 c1cc(c(cc1O)C(=O)O)N PS-3259 c1c(cc(c(c1Cl)S(=O)(=O)N)Cl)Cl PS-3260 CC(=O)c1cccs1 PS-3261 c1cscc1CO PS-3262 Cc1ccc(s1)C PS-3263 c1cc(sc1)CCN PS-3264 c1cc(sc1)CC#N PS-3265 c1cc(sc1C(=O)O)C(=O)O PS-3266 c1cc(sc1[N+](=O)[O-])Br PS-3267 Cc1ccsc1Cl PS-3268 Cc1ccsc1C=O PS-3269 Cc1ccsc1C(=O)O PS-3270 Cc1cc(c(s1)N)C#N PS-3271 c1cc(c(cc1Cl)Cl)S(=O)(=O)N PS-3272 Cc1c(c2ccccc2[nH]1)C=O PS-3273 CC1Cc2ccccc2N1 PS-3274 c1ccc2c(c1)c(c[nH]2)CC#N PS-3276 c1cc2c(cc[nH]2)cc1O PS-3277 c1cc(cc2c1cc[nH]2)[N+](=O)[O-] PS-3278 Cc1cc(n(n1)C)CN PS-3279 c1cc2c(cc[nH]2)c(c1)O PS-3280 c1cc2cc[nH]c2c(c1)O PS-3281 CSc1nc2c(cc[nH]2)c(n1)O PS-3282 c1cc(ccc1NC(=O)C2CCCCC2C(=O)O)Cl PS-3283 CNC1CCOCC1 PS-3284 c1cc2c(ccc(n2)C(=O)O)nc1 PS-3285 c1cnc(cn1)c2c[nH]nc2 PS-3286 c1cnccc1c2c[nH]nc2 PS-3287 COc1cc2c(cc1OC)nc(nc2N)Cl PS-3289 c1cnc(cc1N)Cl PS-3290 c1c(sc(n1)N)C=O PS-3291 c1c(sc(n1)N)[N+](=O)[O-] PS-3292 c1ccc(cc1)n2c(c(cn2)C(=O)O)N PS-3293 C1COCCC1CCN PS-3294 C1COCCC1CN PS-3295 Cc1csc2c1ncnc2N3CCNCC3 PS-3296 c1cc2c(cc1N)CC(=O)N2 PS-3297 COc1ccsc1C=O PS-3298 c1ccc(cc1)C(=O)c2cc[nH]c2 PS-3299 c1c(csc1C(=O)O)C#N PS-3300 Cc1c(sc(c1C(=O)O)N)C PS-3301 c1cc(ccc1c2ccnc(n2)N)C(=O)O PS-3302 c1c(sc(n1)Br)C=O PS-3303 c1cnn2c1ncc(c2N)C(=O)O PS-3304 c1ccc2c(c1)nc(s2)CC(=O)O PS-3305 c1ccc2c(c1)nc(o2)CC(=O)O PS-3306 Cc1cc(nn1C)CN PS-3307 C1COC(CN1)CN PS-3308 c1cnc([nH]1)Br PS-3309 Cn1ccnc1Br PS-3310 c1csc2c1c(ncn2)N3CCNCC3 PS-3311 Cn1cncc1Br PS-3312 c1cc(ccc1S(=O)(=O)c2cscc2N)Cl PS-3313 Cc1[nH]cc(n1)Br PS-3314 c1c(nc[nH]1)Br PS-3315 c1c(c[nH]c1C=O)Br PS-3316 CSc1ccc(cc1)Br PS-3317 C1CCS(=O)(=O)NC1 PS-3318 c1cc2c(cc1C(=O)O)CC(=O)N2 PS-3319 CCOCn1ccnc1Cl PS-3320 Cn1ccnc1Cl PS-3321 c1cc2c(cc1C#N)CC(=O)N2 PS-3322 c1[nH]c(c(n1)C#N)C#N PS-3323 CN(C)S(=O)(=O)n1ccnc1 PS-3324 CCOCn1ccnc1I PS-3325 c1c(cnc(c1Br)Cl)N PS-3326 c1cc2c(cc[nH]2)cc1C=O PS-3327 c1cc(cc2c1cc[nH]2)C=O PS-3328 c1cc2c(ccc(c2nc1)O)Cl PS-3329 c1cc2cc[nH]c2c(c1)C=O PS-3330 COc1cc(cc(c1C=O)OC)O PS-3331 c1cc2c(cc[nH]2)cc1CO PS-3333 c1cc2cc[nH]c2c(c1)CO PS-3334 Cn1ccnc1I PS-3335 Cn1cc(nc1)I PS-3336 Cn1cncc1I PS-3337 c1cnc([nH]1)I PS-3338 c1c(nc[nH]1)I PS-3339 Cn1cncc1C=O PS-3340 Cn1ccnc1C(=O)O PS-3341 Cn1cc(nc1)C(=O)OC PS-3342 COC(=O)c1ccc2c(c1)CC(=O)N2 PS-3343 COC(=O)C1CCOCC1 PS-3344 CS(=O)(=O)c1ccc2c(c1)NC(=O)C2 PS-3345 c1cc2c(cc1[N+](=O)[O-])CC(=O)N2 PS-3346 c1cncc(c1N)C(=O)O PS-3347 C1COCCC1CO PS-3348 C1COCCC1CC(=O)O PS-3349 C1COCCC1C(=O)O PS-3350 c1c(scn1)C=O PS-3351 c1cc(ccc1N)Br PS-3352 c1cc(ccc1O)Br PS-3353 CC(C)c1cc(nc(n1)N)Cl PS-3354 CC(C)(C)Oc1ccc(cc1)O PS-3355 c1c(c(cc(c1Cl)Cl)C#N)C#N PS-3356 Cc1ccc(c(c1)Br)N PS-3357 c1cc(c(cc1Cl)N)Br PS-3358 Cc1cc(ccc1O)Cl PS-3359 CC(C)(C)OC(=O)NCC1CCNCC1 PS-3360 c1c(csc1Br)Br PS-3361 CN(C)C(=O)Cc1ccc(cc1)O PS-3362 CC1(N([C@@H](CO1)C=O)C(=O)OC(C)(C)C)C PS-3363 CN(C)C(=O)Nc1cccc(c1)C(=O)O PS-3364 CCOC(=O)Cc1ccc(cc1)N PS-3366 c1cc2c(cco2)cc1C=O PS-3367 CS(=O)(=O)Nc1cccc(c1)CC(=O)O PS-3368 c1cc(c(c(c1)Cl)Cl)C=O PS-3369 c1cc(c(cc1Cl)C=O)Cl PS-3370 c1cc(ccc1C#N)O PS-3371 c1cc(c(cc1Cl)C=O)[N+](=O)[O-] PS-3372 c1cc(c(cc1C#N)Cl)Cl PS-3373 c1cc(cc(c1)Cl)C(=O)O PS-3374 COc1ccc(cc1)O PS-3375 CCOC(=O)C1CCCN(C1)C(=O)OCc2ccccc2 PS-3376 c1ccc(c(c1)CO)N PS-3377 c1cc2c(cc1Cl)[nH]c(=O)s2 PS-3378 c1ccc(cc1)C(=O)c2ccccn2 PS-3379 c1cc(oc1)C(=O)O PS-3380 COc1ccc(cc1)CC(=O)O PS-3381 COc1ccc(cc1)C(=O)O PS-3382 COc1cc(nc(n1)N)Cl PS-3383 COc1cc(nc(n1)N)OC PS-3384 C[C@H]1[C@H](OC(=O)N1)c2ccccc2 PS-3385 c1ccc(cc1)N2C(=O)CSC2=S PS-3386 c1cc(cc(c1)[N+](=O)[O-])C=O PS-3388 c1cnc(cn1)C(=O)O PS-3389 c1c(cc(c(c1O)Br)O)C(=O)O PS-3390 c1cc2c(cc1O)CCC2=O PS-3391 CC(=O)c1ccc(cc1Cl)Cl PS-3392 CC(=O)c1cc(ccc1Cl)Cl PS-3393 c1cc(nc(c1)Cl)[N+](=O)[O-] PS-3394 CC(=O)c1ccc(cc1)OC PS-3395 CC(=O)c1ccccc1O PS-3396 CC(=O)c1ccc(c(c1)Cl)Cl PS-3397 c1ccc(c(c1)OCC(=O)NN)Cl PS-3398 CCOC(=O)c1cc(ccc1N)I PS-3399 COc1cc(ccc1Cl)[N+](=O)[O-] PS-3400 COc1cc(ccc1Cl)N PS-3401 c1cc(cc(c1)Br)C#N PS-3402 c1cc(c(c(c1)Cl)NC(=S)N)Cl PS-3403 c1cc(cc(c1)N)C#N PS-3404 Cc1ccc(cc1N)Br PS-3405 Cc1c(cccc1Br)N PS-3406 CC(=O)c1cc(cc(c1O)Br)Cl PS-3407 Cc1cccc2c1cc[nH]2 PS-3408 Cn1ccc(c1CC(=O)O)C(=O)O PS-3409 c1cc2c(cc1Cl)nccn2 PS-3410 c1cc2c(cc1Cl)nc(c(n2)O)O PS-3411 COc1cc2c(cc1OC)nc[nH]2 PS-3412 COc1ccc(c2c1CCC2)O PS-3413 CC(=O)c1cc(ccc1OC)OC PS-3414 c1c(c(=O)c(cn1CC(=O)O)Cl)Cl PS-3415 Cc1[nH]c2ccc(cc2n1)Cl PS-3416 Cc1[nH]c2ccc(cc2n1)OC PS-3417 Cc1cccc(c1N)[N+](=O)[O-] PS-3418 Cc1cccc(c1[N+](=O)[O-])OC PS-3419 Cc1ccc(cc1[N+](=O)[O-])OC PS-3420 c1cc2c(cc1[N+](=O)[O-])CCC2 PS-3421 CCC(=O)c1cccc(c1)[N+](=O)[O-] PS-3422 Cc1cc(nc(n1)Cl)C PS-3423 c1[nH]c2c(n1)c(ncn2)Cl PS-3424 c1ccc(cc1)CNc2c3c([nH]cn3)ncn2 PS-3425 c1ccc(cc1)C(=O)Nc2c3c([nH]cn3)ncn2 PS-3427 Cc1cccc(c1N)C PS-3428 Cn1c(c(cn1)C(=O)O)c2ccccc2 PS-3429 Cc1cc(sc1Br)C(=O)OC PS-3430 CC(=O)c1cccc(c1)O PS-3431 c1c(nc(nc1Cl)N)Cl PS-3432 c1c(ncnc1O)O PS-3433 c1ccc(c(c1)CC(=O)O)Br PS-3434 COc1cc(ccc1O)/C=C/C(=O)O PS-3435 CCCc1cc(nc(n1)S)O PS-3436 CCSc1[nH]nnn1 PS-3437 c1[nH]nc(n1)C(=O)N PS-3438 COc1cc(cc(c1)OC)CCC(=O)O PS-3439 Cc1ccc(cc1OC)C=O PS-3440 Cc1ccc(cc1OC)C#N PS-3441 COc1ccccc1Oc2ccc(cc2)N PS-3442 COc1ccc(cc1)Oc2ccc(cc2)N PS-3443 COc1ccnc(c1)C(=O)OC PS-3444 Cc1ccc(cc1C)S PS-3445 c1cc(ncc1Cl)C#N PS-3446 c1c(cnc(c1Cl)C#N)Cl PS-3447 c1cc(c(cc1[N+](=O)[O-])C#N)Br PS-3448 c1cc2c(cc1O)c(=O)[nH]cn2 PS-3449 c1c(ncnc1Cl)N2CCCC2 PS-3450 c1cc2c(cc1Br)c(=O)[nH]cn2 PS-3451 CCOC(=O)c1cc2cccc(c2[nH]1)[N+](=O)[O-] PS-3452 Cc1nccn1c2cc(ncn2)Cl PS-3453 Cc1cn(cn1)c2cc(ncn2)Cl PS-3454 c1cnn(c1)c2cc(ncn2)Cl PS-3455 c1cc(c(cc1[N+](=O)[O-])Br)C(=O)O PS-3456 CCOc1ccc2ccc(=O)oc2c1 PS-3457 COc1cc(ccc1N)Cl PS-3458 COc1c(cc(cn1)Br)C#N PS-3459 CC(C)(C)OC(=O)c1ccc(nc1)Br PS-3460 COc1cc(ccc1[N+](=O)[O-])Cl PS-3461 c1cc(c(cc1N)C#N)Br PS-3462 CNc1ccc(cc1OC)Cl PS-3463 Cc1c(ccc(n1)NC(=O)C)Br PS-3464 c1cc(nc(c1)Br)C(=O)N PS-3465 CCCNc1cc(ncn1)Cl PS-3466 c1cnc(nc1N2CCCC2)Cl PS-3467 CNC(=O)c1ccc(cc1)Br PS-3468 COc1cc(ccc1Br)C(=O)N PS-3469 Cc1ccc(c(c1)OC)[N+](=O)[O-] PS-3470 CNC(=O)c1cccc(c1)Br PS-3471 CS(=O)(=O)c1cc(cnc1)Br PS-3472 CCCc1c(cncn1)Br PS-3473 CCc1c(cncn1)Br PS-3474 CNC(=O)c1ccc(cn1)Br PS-3475 CCNC(=O)c1ccc(cn1)Br PS-3476 COc1cc(ccn1)Br PS-3477 c1c(nc(cn1)Cl)N PS-3478 c1c(ncnc1Cl)NC2CCCCC2 PS-3479 c1cnc(cc1C#N)Br PS-3480 COc1cc(cc(c1O)Br)C=O PS-3481 c1cc(ncc1[N+](=O)[O-])N PS-3482 CNc1ccc(nn1)Cl PS-3483 CCOC(=O)c1coc(n1)Br PS-3484 c1cc(c(cc1Cl)C=O)O PS-3485 c1cc(c(c(c1)Cl)Cl)c2c(nco2)C(=O)O PS-3486 c1cc(c(cc1Cl)Cl)c2c(nco2)C(=O)O PS-3487 CC(C)(C)N1CCC(=O)CC1 PS-3488 c1cc(ncc1Br)C(=O)N2CCCC2 PS-3489 CC(C)(C)OC(=O)n1cccn1 PS-3490 c1c(cc(cc1Br)Br)N PS-3491 c1cc(sc1)C2CCCN2 PS-3492 c1cc(oc1)C2CCCN2 PS-3493 c1cc(ccc1CO)O PS-3494 c1cc(c(c(c1)Br)N)[N+](=O)[O-] PS-3495 c1cc(c(c(c1)Br)N)N PS-3496 C1C(CO1)(CN)CO PS-3497 CC1CCN(C1=O)C PS-3498 c1cc(c(cc1C=O)Br)O PS-3499 COc1cc(c(cc1C(=O)OC)Br)Cl PS-3500 CCCNC(=O)c1ccc(cn1)Br PS-3501 c1cc(ncc1Br)C(=O)NC2CC2 PS-3502 CCN(CC)C(=O)c1ccc(cc1)Br PS-3503 CC(C)NC(=O)c1ccc(cn1)Br PS-3504 Cc1cnc(o1)c2ccccc2[N+](=O)[O-] PS-3505 Cc1ccc(c(c1Cl)N)Cl PS-3506 C#CCNC(=O)c1ccc(cc1)Br PS-3507 c1cc(c(cc1N)O)Cl PS-3508 c1cnn(c1)CCO PS-3509 COc1c(cnc(c1C#N)N)Br PS-3510 c1cc(cc(c1)Br)CC(=O)N2CCCC2 PS-3511 COc1ccn2ccnc2c1C#N PS-3512 c1c(cnc(c1[N+](=O)[O-])NN)Br PS-3513 c1c(nc(cn1)Cl)N2CCOCC2 PS-3514 c1c(ncnc1Cl)N2CCOCC2 PS-3515 CC(C)(C)Nc1cc(ncn1)Cl PS-3516 CCC[C@H]1CC[C@@H](CC1)C(=O)O PS-3517 CC(C)n1cc(cn1)Br PS-3518 c1cc(cc(c1)Br)C(=O)N PS-3519 c1cc(ccc1CN)N PS-3520 C1C=CCC1C(=O)O PS-3521 Cc1cc(cc(c1)C(=O)O)C(=O)O PS-3522 Cc1c[nH]c(n1)Br PS-3523 c1c(cc(cc1N)N)C(=O)O PS-3524 COc1ccc(cn1)Br PS-3525 c1c(c(nc(n1)Br)N)C#N PS-3526 Cc1ncc(n1C)Br PS-3527 Cn1cc(nc1)Br PS-3528 Cn1ccc(n1)CN PS-3529 c1cc(ccc1CN)OC2CCOCC2 PS-3530 CNCc1ccnc(c1)Cl PS-3531 CN(C)C1(CCOCC1)CN PS-3532 c1ccc2cnc(cc2c1)O PS-3533 Cn1ccc(n1)c2cccc(c2)C=O PS-3534 Cc1c(nc[nH]1)Br PS-3535 CNCc1ccc(cc1)OC2CCOCC2 PS-3536 Cc1cnc(c(n1)C)Cl PS-3537 Cn1cc(nc1Br)Br PS-3538 Cc1c(cco1)CNC PS-3539 c1cc2ccsc2c(c1)C(=O)O PS-3540 c1c(nc(s1)N2CCOCC2)C(=O)O PS-3541 Cn1ccc(n1)c2ccc(cc2)C=O PS-3542 c1cc2ccsc2c(c1)C=O PS-3543 c1cc2c(cco2)cc1CN PS-3544 c1cc2c(ccs2)cc1CN PS-3545 c1ccc(c(c1)CN)O PS-3546 CC1CCN(CC1)Cc2cccc(c2)CN PS-3547 C1CCN(CC1)C(=O)C2CCNCC2 PS-3548 C1CCCN(CC1)C(=O)C2CCNCC2 PS-3549 c1cc(ccc1CN2CCCNCC2)Br PS-3550 CC(C)(C)OC(=O)N1c2ccccc2CC1C(=O)O PS-3551 CC(C)(C)OC(=O)N1C2CCC1CC(=O)C2 PS-3552 c1cnc(cn1)CO PS-3553 c1ccc2c(c1)NCC(O2)C#N PS-3554 c1ccc2c(c1)c3cc(ccc3o2)C=O PS-3555 c1cc2c(cc1Br)[nH]cc2C=O PS-3556 Cc1nc(on1)c2ccccc2C=O PS-3557 Cc1cc(nc(n1)Cl)C(=O)OC PS-3558 CCOC(=O)c1cc(n[nH]1)c2cccs2 PS-3559 c1cc2c(cc1Cl)N(C(=O)CO2)CC(=O)O PS-3560 Cn1c(ccn1)c2cccc(c2)N PS-3561 Cc1cncc(n1)Oc2cccc(c2)N PS-3562 Cc1cncc(n1)Oc2cccc(c2)C=O PS-3563 c1coc(c1C=O)Br PS-3564 c1cc(nc(c1)N2CCCC2)CO PS-3565 Cn1c(ccn1)CO PS-3566 COC(=O)c1cc(cc(c1)O)N PS-3567 CNCC1CCN(CC1)c2c3c(ccs3)ncn2 PS-3568 CN1CCOc2c1ncc(c2)C=O PS-3570 c1csc2c1ncnc2N3CCC(CC3)C=O PS-3571 c1cc(c(cc1Br)[N+](=O)[O-])C(=O)O PS-3572 Cc1cc(ccc1N)OC PS-3574 c1c(ncc(n1)Br)Br PS-3575 c1cc(sc1C=O)Cl PS-3576 c1ccc(cc1)C2CCCN2 PS-3577 COc1ccc(cc1)C2CCCN2 PS-3578 c1ccc(cc1)CCC2CCCN2 PS-3579 c1ccnc(c1)C2CCCN2 PS-3580 c1cnccc1C2CCCN2 PS-3581 C1CCC(CC1)C2CCCN2 PS-3582 Cc1ccc(cc1)C2CNCC2NC(=O)OC(C)(C)C PS-3583 COC(=O)[C@@H]1CNC[C@H]1c2ccccc2 PS-3584 c1ccc(cc1)CCC2CCNC2 PS-3585 CNCCCc1ccccc1 PS-3586 CC(C)(C)OC(=O)N1CCCNCC1 PS-3588 c1ccnc(c1)c2cccc(c2)C=O PS-3589 c1cc(cc(c1)c2cccnc2)C=O PS-3590 Cc1cc(sc1)C=O PS-3591 Cc1cc(sc1)CO PS-3592 Cn1cc(cn1)C=O PS-3593 Cn1c(cc(n1)C(=O)O)O PS-3594 c1cc(ccc1C=O)c2cncnc2 PS-3595 c1ccnc(c1)c2ccc(cc2)C=O PS-3596 c1cc(cnc1)c2ccc(cc2)C=O PS-3597 c1cc(ccc1C=O)c2ccncc2 PS-3598 COc1ccc2c(n1)[nH]c(n2)S PS-3599 CS(=O)(=O)C1CCNC1 PS-3600 CN(C)C(CN)c1ccccc1 PS-3601 c1cc(cnc1)C(CN)N2CCOCC2 PS-3602 c1ccc(c(c1)C(CN)N2CCOCC2)Cl PS-3603 CN(C)CC(c1ccccc1)N PS-3604 c1ccc(cc1)C(CN2CCOCC2)N PS-3605 CNC(CN1CCOCC1)c2ccccc2 PS-3606 CC(CN)Oc1ccc(cc1)OC PS-3607 Cc1ccc(cc1)OC(C)CN PS-3608 COC(=O)c1cc(ccc1Br)C#N PS-3609 c1cc(c(c(c1)Br)C(=O)O)N PS-3610 CC(=O)CC(=O)c1ccccc1 PS-3611 Cc1cncc(c1N)C PS-3612 c1cc(cnc1)c2ncc(c(n2)N)C#N PS-3613 c1ccnc(c1)Oc2cccc(c2)C=O PS-3614 c1cc(cnc1)Oc2ccc(cc2)C=O PS-3615 c1ccc(c(c1)C=O)Oc2cnccn2 PS-3616 c1cc(cc(c1)Oc2cnccn2)C=O PS-3617 COc1ccccc1Oc2cccc(c2)C(=O)O PS-3619 COc1ccccc1Oc2ccc(cc2)C(=O)O PS-3620 Cc1ccc(cc1)c2ccn(n2)CC(=O)O PS-3621 c1ccc(cc1)C(CN2CCCCC2)N PS-3622 c1cc(cnc1)C2(CCNCC2)O PS-3623 Cc1ccc(cc1I)N PS-3624 COc1cc(ccc1O)CC(=O)O PS-3625 Cc1c(cccn1)Br PS-3626 c1c(c(ncn1)N)C(=O)O PS-3627 c1c(cc(c2c1c(cc(=O)o2)O)Cl)Cl PS-3628 c1cnc(cc1N)Br PS-3629 C#Cc1cc(cc(c1)C#C)C#C PS-3630 c1cc(ncc1C(=O)O)C#N PS-3631 c1cnccc1NC(=S)N PS-3632 c1c(ncs1)C=O PS-3633 Cc1cc(n(n1)c2ccc(cc2)C(=O)O)C PS-3634 c1cc(ccc1C=O)O PS-3635 COC(=O)c1ccncc1 PS-3636 C1COCCN1CCN PS-3637 CCOC(=O)c1c[nH]nc1 PS-3638 Cc1ccc(cc1Cl)C=O PS-3639 c1cc(ncc1Cl)N PS-3640 c1ccc(c(c1)C=O)C#N PS-3641 c1cc(ccc1C(C(=O)O)O)Cl PS-3642 CN(C)c1ccccc1C=O PS-3643 c1ccc2c(c1)[nH]nn2 PS-3644 c1cc2cc(cc(c2nc1)O)[N+](=O)[O-] PS-3645 c1c(cnc(c1Br)O)[N+](=O)[O-] PS-3646 CC(C)(C)NC(=O)c1ccccc1N PS-3647 Cn1c2ccccc2c(cc1=O)C=O PS-3648 CCOC(=O)c1c(c(ns1)C(=O)N)N PS-3649 c1ccc(cc1)n2nc(c(n2)N)C(=O)O PS-3650 c1cc2cc(cc(c2nc1)N)Br PS-3652 CCOC(=O)c1coc(n1)N PS-3653 Cc1cnc(n1C)Br PS-3654 c1cc(c(=O)[nH]c1)N PS-3655 Cc1nc2cccc(c2o1)C(=O)O PS-3656 c1cc(c(c2c1cn[nH]2)C(=O)O)N PS-3657 Cc1cc(n2c(n1)cc(n2)C(=O)O)C PS-3658 c1cc(cc2c1cc[nH]2)C#N PS-3659 c1cc(ncc1N)Cl PS-3660 CCOC(=O)c1cc(c(nc1)N)Br PS-3661 c1cnc(cc1Cl)C(=O)O PS-3662 c1ccc2c(c1)ccc(n2)C#N PS-3663 c1cc2c(nc1)nc([nH]2)S PS-3664 c1c(c(n[nH]1)[N+](=O)[O-])C#N PS-3665 Cc1cc(c(c(c1)C)S(=O)(=O)N)C PS-3666 c1cc(ccc1S(=O)(=O)NC(=O)N)Cl PS-3667 CC1CCCC(N1)C PS-3668 c1cnc(cc1[N+](=O)[O-])N PS-3669 Cc1ccnc(c1)Cl PS-3670 COCc1ccccn1 PS-3671 c1cc(c(nc1)O)Cl PS-3672 CCCc1ccncc1 PS-3673 CN1CCN(CC1)c2ccccc2CN PS-3674 CC(C)(C)OC(=O)N1CCC(CC1)C=O PS-3675 c1cc(c(cc1Cl)Cl)C(Cn2ccnc2)O PS-3676 C=C(c1ccccc1)C(=O)O PS-3677 c1cc2c(cc1O)cn[nH]2 PS-3678 CCOc1cc(c(nc1Br)Br)N PS-3679 c1ccc2c(c1)nco2 PS-3680 Cc1ccc(cn1)C(=O)O PS-3681 CC(C)c1cccc(c1)C(=O)O PS-3682 Cc1c(cc(s1)Br)Br PS-3683 Cc1c(ccs1)Br PS-3684 c1cc2c(cc1Cl)[nH]cc2C=O PS-3685 c1cc(c(cc1Br)N)C(=O)O PS-3686 CC(C)(C)OC(=O)N1CCC[C@@H]1CN PS-3687 c1cc(c2c(c1)NC(=O)CO2)N PS-3688 CC(C)(C)OC(=O)N1CCN(CC1)Cc2cccc(c2)N PS-3689 c1cc(cc(c1)N2CCCCC2)N PS-3690 COc1ccnc(c1)N PS-3691 c1cc(nc(c1)Br)NN PS-3692 c1cc(ccc1C=O)N2CCCC2 PS-3693 Cc1c(c(n(n1)C(=O)OC(C)(C)C)C)C=O PS-3694 CCOC(=O)C(c1ccc(cc1)O)O PS-3695 c1ccc(cc1)OCCC(=O)O PS-3696 c1ccc(c(c1)C=O)c2cccs2 PS-3697 C1CS(=O)(=O)CCN1 PS-3698 C1CC(CNC1)C(=O)N PS-3699 c1cc(cc(c1)C(=O)O)c2cc[nH]n2 PS-3700 c1cc(ncc1I)N2CCOCC2 PS-3701 c1cc(ncc1CO)N2CCCC2 PS-3702 CN1CCN(CC1)c2ccccc2C(=O)O PS-3703 CC(C)(C)OC(=O)N1CCSCC1C(=O)O PS-3704 CC(=O)c1cccc(c1)NC(=S)N PS-3705 c1cc(cc(c1)S(=O)(=O)N2CCCCC2)N PS-3707 CN(C)c1c(cc2ccccc2n1)C=O PS-3708 CS(=O)(=O)Nc1cccc(c1)C=O PS-3709 Cc1nc(cs1)c2cccc(c2)CO PS-3710 CC(C)N1CCc2c(sc(c2C#N)N)C1 PS-3711 Cc1c(cno1)C(=O)O PS-3713 c1cc(c(c(c1)Br)N)C(=O)O PS-3714 Cn1cncc1CN PS-3715 c1csc(n1)CO PS-3716 CN(C)c1cccc(c1)O PS-3717 c1cc(c(nc1)C(=O)O)O PS-3718 c1cc2cc(ccc2nc1)O PS-3719 COc1ccc(c(c1)O)C(=O)O PS-3720 COc1cccc(c1C(=O)O)O PS-3721 c1csc(n1)C=O PS-3722 Cc1c(cno1)I PS-3723 Cc1c(nc(o1)C)C(=O)O PS-3724 COC(=O)c1cccc(c1N)C(=O)O PS-3725 CC(C)(C)OC(=O)NCc1ccc(cc1)CO PS-3726 CCOC(=O)c1cnn2c1cccc2 PS-3727 CCOC(=O)c1c(c2cccnc2s1)N PS-3728 COC(=O)c1cccc(c1)c2cnco2 PS-3731 CCOc1ccc(cc1)c2c(c(=O)c3ccccc3o2)O PS-3732 COc1cccc2c1[nH]cc2 PS-3733 c1cc(c(c(c1)O)N)[N+](=O)[O-] PS-3734 c1cn(cn1)CCC(=O)O PS-3735 c1cnc(c2c1occ2)N3CCCNCC3 PS-3736 c1ccc2c(c1)CCC(O2)CO PS-3737 c1cc(ncc1CO)N PS-3738 c1ccnc(c1)/C(=N/O)/N PS-3739 CCOC(=O)c1cc([nH]n1)c2ccco2 PS-3740 CC(C)(C)OC(=O)N1CCC[C@H]1CO PS-3741 Cc1ccc(cc1)C[C@H](C(=O)O)NC(=O)OC(C)(C)C PS-3742 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@@H]1C(=O)O PS-3743 CC(C)(C)OC(=O)N[C@@H](Cc1cccs1)C(=O)O PS-3745 CC(C)(C)OC(=O)N1CCCCC1C(=O)O PS-3746 c1ccc2c(c1)cccc2C[C@H](C(=O)O)N PS-3747 c1cc(c(cc1Cl)Cl)C[C@H](C(=O)O)N PS-3748 c1cc(c(cc1C[C@H](C(=O)O)N)Cl)Cl PS-3749 c1ccnc(c1)C[C@H](C(=O)O)N PS-3750 c1cc(cnc1)C[C@@H](C(=O)O)N PS-3751 c1cc(cnc1)C[C@H](C(=O)O)N PS-3752 c1cnccc1C[C@@H](C(=O)O)N PS-3753 c1cnccc1C[C@H](C(=O)O)N PS-3754 c1ccc2c(c1)c(cs2)C[C@@H](C(=O)O)N PS-3755 c1cc(cc(c1)O)CN PS-3756 c1cc2c(c(c1)Br)CCCC2=O PS-3757 Cc1c(c(nc(n1)Cl)Cl)N PS-3758 COc1ccc(c(c1)C=O)[N+](=O)[O-] PS-3759 Cn1c(ccn1)CN PS-3760 CNCc1ccc2c(c1)CCN2C PS-3761 CN1CCc2c1ccc(c2)C(=O)O PS-3762 CN1CCc2c1ccc(c2)Br PS-3763 Cc1nc(on1)c2cccc(c2)C=O PS-3764 c1cc(ncc1C=O)OC2CCOCC2 PS-3765 Cc1c(sc(n1)c2ccncc2)C=O PS-3766 CN1CCc2c1ccc(c2)C=O PS-3767 Cc1cncc(n1)Oc2ccc(cc2)C=O PS-3768 c1cc(sc1)c2ncc(cn2)CO PS-3770 Cc1ccnc2c1cccc2 PS-3771 c1c(cncc1Br)CN PS-3772 Cc1cc(n(n1)c2ccc(cc2)CNC)C PS-3773 Cn1ccc2c1c(ccc2)Br PS-3774 c1cc(c(cc1[N+](=O)[O-])N)C#N PS-3775 CC(=O)c1ccc(nc1)Br PS-3776 c1ccc(cc1)c2ncc(cn2)C=O PS-3777 c1cc(sc1)c2ncc(cn2)C=O PS-3778 c1cc(sc1)CN2CCC(CC2)C=O PS-3779 c1c(cnc(n1)N2CCCC2)C=O PS-3780 C1COCCC1CCO PS-3781 c1c(cnc(n1)N2CCCC2)CO PS-3782 COC(=O)CC(=O)c1ccccc1Cl PS-3783 COc1ccc(nn1)N PS-3784 c1ccc(cc1)c2ccc(nn2)N PS-3785 COc1ccc(cc1)c2ccc(nn2)N PS-3786 Cc1ccc(cc1)c2nc(nc(n2)N)N PS-3787 c1cc(c(cc1[N+](=O)[O-])N)CO PS-3788 c1c[nH]nc1C(=O)O PS-3789 C[C@H](Cc1ccccc1)O PS-3790 COc1cc(ccc1Br)N PS-3791 c1cc(c(cc1Br)O)C(=O)O PS-3792 Cc1ccc(cc1OC)Cl PS-3793 COc1cc(ccc1Cl)Cl PS-3794 Cc1ccc(c(c1)Cl)N PS-3795 COc1ccc(cn1)C(=O)OC PS-3796 c1csc(c1Br)Cl PS-3797 c1cc(c(cc1Cl)Br)N PS-3798 c1cc(c(cc1Cl)[N+](=O)[O-])C#N PS-3799 c1cc(c(cc1Cl)N)C#N PS-3800 c1cc(c(cc1Cl)N)c2[nH]nnn2 PS-3801 Cc1cc(cc(c1)NC(=S)N)C PS-3802 c1cc(ccc1C#N)NC(=S)N PS-3803 COc1cc(ccc1OCc2ccccc2)C=O PS-3806 CCCc1ccc(cc1)C(=O)C PS-3807 CC(=O)c1ccc(cc1OC)OC PS-3811 CCCCc1[nH]c(c(n1)C=O)Cl PS-3814 CNCc1ccnn1C PS-3816 Cc1ccoc1C=O PS-3817 c1ccc(cc1)c2cc(on2)C=O PS-3818 c1c(c(nc(n1)Cl)N)Br PS-3821 CCOc1ncc(cn1)Br PS-3822 CC(C)Nc1ncc(cn1)Br PS-3823 CS(=O)(=O)c1ncc(cn1)Br PS-3824 COc1cc(ncn1)Cl PS-3825 CSc1ccnc(n1)Cl PS-3826 COc1cc(ncn1)I PS-3827 CSc1nccc(n1)I PS-3828 CSc1ncccn1 PS-3829 CCOC(=O)c1csc(n1)C(C)C PS-3830 Cc1nc(c(s1)Br)C(=O)OC PS-3831 CC(=O)Nc1ncc(s1)Br PS-3832 Cc1c(sc(n1)N)Cl PS-3833 CCOc1nc(cs1)Br PS-3834 CC(C)c1c(nc(s1)Cl)C(=O)OC PS-3835 CC(C)c1c(nc(s1)Br)C(=O)OC PS-3836 COc1nc(cs1)Br PS-3837 COc1ncc(s1)Br PS-3838 c1c(scn1)Br PS-3839 CC(C)(c1nc(cs1)Br)O PS-3840 CSc1nc(cs1)Br PS-3841 Cc1c(cccc1Cl)O PS-3842 COC(=O)c1cnc(o1)N PS-3843 CC(C)(C)OC(=O)NCc1cc(no1)Br PS-3844 CS(=O)(=O)c1ccc(cn1)Br PS-3845 CSc1ccc(cn1)Br PS-3846 CC1CN(CCN1)C(=O)OC(C)(C)C PS-3847 C[C@@H]1CN(CCN1)C(=O)OC(C)(C)C PS-3848 C[C@H]1CN(CCN1)C(=O)OC(C)(C)C PS-3849 CC(C)C[C@H]1CNCCN1C(=O)OC(C)(C)C PS-3850 CC(C)[C@H]1CNCCN1C(=O)OC(C)(C)C PS-3851 CC[C@H]1CNCCN1C(=O)OC(C)(C)C PS-3852 C1C[C@H]2CNCCN2C1 PS-3853 C1C[C@@H]2CNCCN2C1 PS-3854 C1CCN2CCNCC2C1 PS-3855 C1CC1N2CCNCC2 PS-3856 c1ccc(cc1)CN2CCCC(C2)N PS-3857 c1ccc(cc1)CN2CCC[C@@H](C2)N PS-3858 CC(C)(C)OC(=O)N[C@H]1CCCNC1 PS-3859 CC(C)(C)OC(=O)N1CCCC(C1)CN PS-3860 CC(C)(C)OC(=O)N1CCC[C@@H](C1)CN PS-3861 CC(C)(C)OC(=O)N1CCC[C@H](C1)CN PS-3862 CC(C)(C)OC(=O)N1CCC[C@H](C1)CO PS-3863 CC(C)(C)OC(=O)N1CCC[C@@H](C1)CO PS-3864 CC(C)(C)OC(=O)N1CCCC(C1)NC PS-3865 CC(C)(C)OC(=O)N1CCC(CC1)NC PS-3866 CC(C)(C)OC(=O)N1CCCC(C1)C=O PS-3867 CC(C)(C)OC(=O)NC1CCNC1 PS-3868 CC(C)(C)OC(=O)N1CC[C@H](C1)O PS-3869 CC(C)(C)OC(=O)N1CC[C@@H](C1)O PS-3870 CC(C)(C)OC(=O)N1CCC[C@H]1CN PS-3871 c1ccc(cc1)COC(=O)NC2CNC2 PS-3872 CC(C)(C)OC(=O)N1CC=CC(C1)O PS-3873 CSc1ccc(c(c1)C(=O)O)Cl PS-3874 Cc1cc(cc(n1)C)N PS-3875 c1c[nH]c2c1cc(c(c2)Cl)Cl PS-3876 c1cc2ccoc2c(c1)Br PS-3877 COC(=O)C1(CCC1)c2ccccc2 PS-3878 c1ccc(c(c1)S)Cl PS-3879 c1c(ncs1)C(=S)N PS-3880 c1csc(n1)C(=O)O PS-3881 Cc1ncc(s1)C=O PS-3882 c1ccc(cc1)[C@H]([C@@H](c2ccccc2)N)N PS-3883 c1nc(c(c(n1)Cl)Cl)Cl PS-3884 COc1c(ncnc1Cl)Cl PS-3885 CC(C)(C)OC(=O)N1CC=CC1 PS-3886 c1cnc(c(c1N)[N+](=O)[O-])Cl PS-3887 c1c(c(cnc1Cl)[N+](=O)[O-])Cl PS-3888 c1cnc(nc1)C(=O)O PS-3889 Cc1ccoc1CN PS-3890 c1cc(ncc1N2CCCC2)C(=O)O PS-3891 Cc1cncc(n1)N2CCCC(C2)C=O PS-3892 c1cc(cnc1)c2ccc(s2)Br PS-3893 CC1CNCCN1C(=O)OC(C)(C)C PS-3894 CS(=O)(=O)N1CCC(=O)CC1 PS-3895 CC(=O)c1ncccn1 PS-3897 c1cc(cc(c1)I)CO PS-3898 CCc1ccccc1C(=O)O PS-3899 c1cc2c(cc1N)[nH]nc2Br PS-3900 COc1cc(cnc1)C(=O)O PS-3901 CNCc1ccc(cc1)Cl PS-3902 c1ccc(c(c1)C=O)N2CCNCC2 PS-3903 COc1cccnc1C(=O)O PS-3904 c1cc(ccc1C=O)N2CCNCC2 PS-3905 Cc1c(ccs1)C(=O)O PS-3906 C1COCC1C(=O)O PS-3907 c1ccc2c(c1)c(c[nH]2)/C=C/C(=O)O PS-3908 Cc1ccc(cc1)CNC PS-3909 COc1ccc(c(c1)C#N)Br PS-3910 CS(=O)(=O)c1ccccc1N PS-3911 Cn1c2ccc3c(c2nc1N)cccn3 PS-3912 c1c(nc(s1)N2CCOCC2)Br PS-3914 CC(C)(CN)c1ccccc1 PS-3915 c1c(cnc(c1Br)C(=O)O)Cl PS-3916 c1cc(cc(c1)N2CCOCC2)CO PS-3917 c1ccc2c(c1)NC(=O)C(CS2)CC(=O)O PS-3918 c1cc2c(c(c1)Br)c(c[nH]2)C=O PS-3919 COc1nccc(n1)N PS-3920 Cc1ccc2c(c1)c(c[nH]2)C=O PS-3921 Cc1ccc2c(c1)[nH]cc2C=O PS-3922 c1cc2c(c[nH]c2c(c1)[N+](=O)[O-])C=O PS-3923 c1cn2cc(nc(c2n1)Br)Br PS-3924 c1c(c(cc(c1Cl)Cl)O)N PS-3925 Cc1cccc(c1[N+](=O)[O-])N PS-3927 c1cc(ccc1CC#N)C(=O)O PS-3928 c1c(cnc(c1Cl)C(=O)O)Br PS-3930 c1c(ncc(n1)Cl)Cl PS-3931 c1cc(cc(c1)Cl)c2cc[nH]n2 PS-3932 Cc1ccnc(c1C#N)N PS-3933 c1cc2c(c(c1)O)c(c[nH]2)C=O PS-3934 CCOC(=O)c1cnc(s1)C PS-3935 Cc1c(c2ccccc2n1C(=O)OC(C)(C)C)CO PS-3936 c1c(c2c([nH]1)nc[nH]c2=O)I PS-3937 c1c[nH]c2c1c(=O)[nH]cn2 PS-3938 CSc1[nH]c(=O)c2cc[nH]c2n1 PS-3939 c1c[nH]c2c1c(=O)[nH]c(n2)S PS-3940 c1c[nH]c2c1c(=O)[nH]c(n2)N PS-3941 c1c[nH]c2c1c(nc(n2)N)Cl PS-3942 CCOC(=O)c1ccc([nH]1)[N+](=O)[O-] PS-3943 c1cc(c2c(c1)[nH]cn2)C=O PS-3944 c1cc(c2c(c1)[nH]cn2)CO PS-3945 c1cnc(cc1Br)C#N PS-3946 Cc1cc(cc(n1)Br)N PS-3947 c1cc(cc2c1ccnc2)N PS-3948 c1cc(c2c(c1)nccn2)N PS-3949 c1cc2c(c(c1)Br)nccn2 PS-3950 CC(C)(C)OC(=O)N1CCNCC1 PS-3951 CS(=O)(=O)c1cccc(c1)N PS-3952 COc1cc(c(cc1Cl)N)Cl PS-3953 COc1ccc(c(c1)N)C(=O)O PS-3954 c1cc(c(c(c1)Br)N)C#N PS-3955 c1cc(c(c(c1)Br)C(=O)O)O PS-3956 c1cc(c(c(c1)Br)C#N)N PS-3957 CN(C)C1CCc2c(c3cc(ccc3[nH]2)Br)C1 PS-3958 c1c(cnc(n1)Cl)Cl PS-3959 c1cc(c(cc1O)C=O)[N+](=O)[O-] PS-3960 c1cc2c(nc1)CCCC2=O PS-3961 c1cc2c(cc1Cl)c(nc(=O)[nH]2)C3CC3 PS-3962 Cc1nc(co1)C(=O)NN PS-3963 CC(=O)SCC(Cc1ccccc1)C(=O)O PS-3964 Cc1cc(cnc1Br)Cl PS-3965 Cn1c(c(cn1)Br)CCN PS-3966 c1ccc2c(c1)c(cnc2O)Br PS-3968 Cc1c(sc(n1)Br)Br PS-3969 c1c2c(sc1Br)C(=O)NCC2 PS-3970 Cc1cc(nc(n1)Cl)N PS-3971 c1cc(ncc1[N+](=O)[O-])N2CCNCC2 PS-3972 COc1c(cccc1Br)N PS-3973 c1cc2c(ccnc2N)c(c1)Br PS-3974 c1c(c(nc(n1)Cl)N)N PS-3975 c1cc2c(cc1CC(=O)O)nccn2 PS-3976 c1cc2c(cc1C=O)nccn2 PS-3977 Cc1cc(nc(n1)N(C)c2ccc(cc2)N)C PS-3978 CCC(=O)c1ccccc1C PS-3979 c1ccc2c(c1)Nc3ccccc3S2 PS-3980 Cc1ccc(c(c1)C(=O)OC)[N+](=O)[O-] PS-3981 Cc1cc(cc(n1)C)Cl PS-3982 Cc1cc(cc(n1)C)Br PS-3983 Cc1cnc(nc1Cl)Cl PS-3984 Cn1cc(cn1)C(=O)O PS-3985 C#Cc1ccccc1C#N PS-3986 C#Cc1cccc(c1)C#N PS-3987 c1c(cnc(c1Cl)C#N)Br PS-3988 c1c(cnc(c1Br)C#N)Cl PS-3989 c1c(cncn1)CO PS-3990 CN(C)c1ccc(cc1)Cl PS-3991 c1cc2c(cc1Br)c(n[nH]2)Cl PS-3992 c1cc2c(cc1I)CCC2=O PS-3993 COC(=O)c1cc(no1)Br PS-3994 CC(C)n1ccnc1Cl PS-3995 c1cc2c(cco2)nc1 PS-3996 c1cc2c(c(c1)I)nc(s2)N PS-3997 c1cc2c(cc1O)nc(s2)N PS-3998 c1ccc2c(c1)c(ccn2)N PS-3999 CC(C)(C)OC(=O)NCCOc1ccc(cc1)N PS-4000 c1c(ncc(n1)N)C#N PS-4001 Cc1ccnc2c1cccc2N PS-4002 c1cc2c(c(c1)C#N)C(=O)CC2 PS-4003 Cc1ccc(cc1[N+](=O)[O-])CC(=O)O PS-4004 Cc1cccc(c1[N+](=O)[O-])CC(=O)O PS-4005 c12c([nH]nc1Br)nc(nc2Cl)N PS-4006 C=C(Cc1ccccc1)C(=O)O PS-4007 c1c2c(cc(s2)Br)sc1Br PS-4008 Cc1c(cnc(n1)Cl)C(=O)O PS-4009 COc1c(ccc(n1)Br)N PS-4010 Cn1ccc(n1)C(=O)O PS-4011 Cc1cn2c(n1)cccc2Br PS-4012 Cc1c(scn1)Br PS-4013 c1c(cnc(n1)N2CCOCC2)N PS-4014 CCCn1c(c(cn1)C=O)C PS-4015 COc1nc(cc(n1)Cl)Cl PS-4016 CN1CC(=O)NC1=O PS-4018 CCCCNc1ccccc1 PS-4019 c1ccc2c(c1)ccc(n2)O PS-4021 CCOC(=O)Cc1ccc(cc1)Br PS-4022 c1cnccc1SCC(=O)O PS-4023 c1cc2c(cc1[N+](=O)[O-])OCO2 PS-4024 CCN1CCC(=O)CC1 PS-4025 CC(=O)Oc1ccc(cc1)OC(=O)C PS-4026 c1ccc(c(c1)C#N)Cl PS-4027 CC1(C(=O)NC(=O)N1CO)C PS-4028 Cc1csc(n1)S PS-4029 CCOc1cc(ccc1O)C=O PS-4030 c1c(c(=O)[nH]c(=O)[nH]1)I PS-4031 CC(C)Sc1ccccc1 PS-4032 c1cc2cccc(c2c(c1)N)N PS-4034 CC(=O)c1cccc(c1)Cl PS-4035 CC(C)(c1ccccc1)O PS-4036 COc1ccc(cc1)CO PS-4037 c1cc(ccc1C#N)C(=O)O PS-4038 CCOc1ccc(cc1)OCC PS-4039 c1cc(cc(c1)Br)O PS-4040 COc1ccc(cc1OC)CCC(=O)O PS-4041 c1cc(sc1C=O)Br PS-4042 Cc1ccc(cc1)/C=C/C(=O)O PS-4043 c1cc2c(c(c1)O)CCC2=O PS-4044 c1ccc(cc1)Oc2cccc(c2)CO PS-4045 c1(nnc(s1)S)S PS-4046 C1CCC(C1)C(=O)O PS-4047 c1cc(ccc1CCO)[N+](=O)[O-] PS-4048 c1cc(c(cc1Cl)Cl)C(=O)O PS-4049 c1ccc2c(c1)[nH]c(n2)Cl PS-4050 c1c(cc(cc1O)O)C(=O)O PS-4051 c1cc(c(nc1)N)C(=O)O PS-4052 CCOC(=O)c1ccc(c(c1)O)O PS-4053 CC(=O)c1cccc(c1)C#N PS-4054 Cc1cc(nc(n1)C)O PS-4055 CCN(CC)c1ccc(cc1)C(=O)O PS-4056 c1cc(oc1)/C=N/O PS-4057 c1ccc(cc1)c2cc(c(s2)C(=O)N)N PS-4058 CNC(=O)c1ccccc1N PS-4059 CS(=O)(=O)c1ccccc1[N+](=O)[O-] PS-4060 c1ccc(cc1)SC2CC2 PS-4061 CCn1cc(cn1)C=O PS-4062 COc1cccc(c1OC)CN PS-4063 c1ccc(c(c1)N)I PS-4064 CCOC(=O)c1cnc(nc1C)Cl PS-4065 c1cc(ncc1N)[N+](=O)[O-] PS-4066 c1cc(nc2c1cc([nH]2)C(=O)O)Cl PS-4067 c1c[nH]c2c1c(c(cn2)C(=O)O)Cl PS-4068 CC1(CCC(=O)CC1)C PS-4069 CC(C)(C)c1cc(on1)N PS-4070 c1c(nc(s1)Br)C=O PS-4071 c1ccc2c(c1)c3ccccc3[nH]2 PS-4072 c1cc(c(cc1O)C=O)O PS-4073 c1cc(ccc1C(=O)O)Cl PS-4074 CCOC(=O)c1nc(cs1)C PS-4075 CCCC1CCNCC1 PS-4076 c1cc(c(c(c1)Cl)Cl)N PS-4077 c1nc(c(c(n1)Cl)Br)Cl PS-4078 c1cc2c(c(c1)O)nn[nH]2 PS-4079 COc1ccc(cc1O)[N+](=O)[O-] PS-4080 c1cnc(cc1C(=O)O)Br PS-4081 c1cc(nc(c1)Br)C(=O)O PS-4082 c1cc(nc(c1C(=O)O)Cl)Cl PS-4083 c1c(cnc(c1Cl)C(=O)O)Cl PS-4084 c1c[nH]c(=O)cc1C(=O)O PS-4085 COc1cc(ccn1)C(=O)O PS-4086 COc1ccc(cn1)C(=O)O PS-4087 c1c(cncc1N)C(=O)O PS-4088 c1cnc(cc1C(=O)O)N PS-4089 c1cc(nc(c1)N)C(=O)O PS-4090 c1ccc2c(c1)cc(cn2)Br PS-4091 c1c(cncc1Br)Br PS-4092 COCc1ccc(cc1)CC(=O)O PS-4093 COCc1ccc(cc1)CC(=O)OC PS-4094 Cc1ccc(cc1C)N PS-4095 CC(C)(C)OC(=O)N(C)C1CCNCC1 PS-4096 c1cnccc1N2CCCC2 PS-4097 C1CCC2=NCCCN2CC1 PS-4098 Cc1ccc(cc1)Nc2c(cccc2N)C(=O)O PS-4099 c1ccc(cc1)Nc2c(cccc2N)C(=O)O PS-4100 COC(=O)C(=O)CCc1ccccc1 PS-4101 c1ccc(c(c1)C=O)c2nccs2 PS-4102 COc1cccc(c1N)CCN2CCCC2 PS-4103 CCOC(=O)c1ccc(c(c1)N)N PS-4104 Cc1c(cccc1[N+](=O)[O-])CC(=O)O PS-4105 CCc1c(ccc(n1)C)O PS-4106 CCCc1ccc(cc1)CC(=O)O PS-4107 CC(=O)C1CCCCC1 PS-4108 c1cc(c(cc1Br)S(=O)(=O)N)N PS-4109 c1cc(c(cc1Cl)S(=O)(=O)N)N PS-4110 c1cc(cnc1)c2ccc(cc2)N PS-4111 c1cnccc1CCN PS-4112 c1cc(c(nc1)[N+](=O)[O-])Br PS-4113 c1cc(ncc1Cl)[N+](=O)[O-] PS-4114 COC(=O)c1ccc(c(c1)N)Cl PS-4115 c1ccc(cc1)COC(=O)CC#N PS-4116 c1cc2c(cc1CO)nc[nH]2 PS-4117 Cn1ccc(n1)CO PS-4118 c1cc2c(cc1C=O)nns2 PS-4119 c1cc2c(cc1C=O)nc[nH]2 PS-4120 c1ccc(cc1)c2ccc(cn2)C(=O)O PS-4121 Cn1ccc2c1cc(cc2)C(=O)O PS-4122 c1cnc(cc1C(=O)O)N2CCCCC2 PS-4123 c1c(cnc(c1[N+](=O)[O-])Cl)Cl PS-4124 c1ccc(cc1)c2ccc(cn2)C#N PS-4125 c1ccc(c(c1)CN2CCCNCC2)Cl PS-4126 c1ccc(c(c1)CO)Br PS-4127 COc1cccc(c1)Br PS-4128 c1cnccc1C(=O)NN PS-4129 Cc1ccc(cc1NC(=O)C)N PS-4130 c1cc(ccc1CC#N)N PS-4131 Cc1c([nH]c2c1cccc2[N+](=O)[O-])C PS-4132 Cc1ccc(c(c1)C(=O)NN)N PS-4133 c1ccc(c(c1)N)N2CCCCC2 PS-4134 c1cc(c(cc1[N+](=O)[O-])Br)N PS-4135 c1cc(cc(c1)Br)N PS-4136 COc1ccc(c(c1)C(=O)O)C#N PS-4137 Cc1cccc(c1O)OC PS-4138 Cc1cc(cc(c1O)C)C=O PS-4139 CCOC(=O)c1cc(c(c(c1)Cl)N)Cl PS-4140 C1CCC(C(C1)N)O PS-4141 c1c(cc(c(c1N)O)Cl)Cl PS-4142 c1cc(c(c(c1)Cl)C(=O)O)N PS-4143 c1cc(c(cc1Cl)N)C(=O)O PS-4144 Cc1cc(ccc1N)Br PS-4145 COC(=O)c1c(c2ccccc2s1)O PS-4146 c1cc(c(cc1Br)C=O)O PS-4147 c1cc(nnc1Cl)Cl PS-4148 c1cc(ccc1N)N2CCCCC2 PS-4149 c1cc2c(cc1O)[nH]cn2 PS-4150 c1cncc(c1C(=O)N)N PS-4151 CC1=NNC(=O)CC1 PS-4152 Cc1cc(no1)N/C=N/O PS-4153 CC(=O)Nc1cc(cc2c1cccc2)N PS-4154 C1CNC(=S)NC1 PS-4155 c1cc(c(=O)[nH]c1)C#N PS-4156 c1cncc2c1ccs2 PS-4157 c1cncc2c1c(cs2)N PS-4158 Cc1cc(ccc1NC(=O)C)N PS-4159 Cc1ccc(c(c1)C(=O)O)N PS-4160 Cc1c(c(c(cc1Br)[N+](=O)[O-])N)C PS-4161 Cc1c(c(c(cc1Br)N)N)C PS-4162 c1cc(cnc1)c2ccc(s2)N PS-4163 CC1=C(C(=O)OC1=O)C PS-4164 Cc1ccc(nn1)Cl PS-4165 Cc1c(c(nnc1O)O)C PS-4166 CC1=CC2C3CC(C2C1)C=C3C PS-4167 C1CC(=O)NN=C1C(=O)O PS-4168 Cn1c2cccc(c2cn1)N PS-4169 Cn1cc2c(cccc2n1)N PS-4170 c1cc(c(cc1Cl)CC(=O)O)Br PS-4171 Cc1cnc(c(n1)C)N PS-4172 c1cc(ccc1NN)[N+](=O)[O-] PS-4173 COc1ccc(cc1N)Cl PS-4174 CCOC(=O)Cc1cccc(c1)OC PS-4175 COc1cccc(c1)CC#N PS-4176 CCc1c(c([nH]c1C)C(=O)OCC)C PS-4177 Cc1c(c(c([nH]1)Cl)CC(=O)OC)C(=O)OC PS-4178 COC(=O)c1cc2ccccc2cn1 PS-4179 Cc1cc(cnc1Cl)[N+](=O)[O-] PS-4180 Cc1cc(cnc1)C(=O)O PS-4181 c1cc(c(nc1)[N+](=O)[O-])N PS-4182 c1c(cc(c(c1C(=O)O)O)Cl)Cl PS-4183 Cc1[nH]c(c(n1)[N+](=O)[O-])Br PS-4184 CCCOc1ccc(cc1)C#N PS-4185 CCc1ccc(cc1)C(=O)O PS-4186 COc1ccc(cc1)C#C PS-4187 C=CCc1c(cccc1O)C=O PS-4188 COc1ccc(cc1Br)C#N PS-4189 c1ccc2cnc(cc2c1)N PS-4190 CC(=O)c1ccc(cc1O)N PS-4191 CC(=O)c1c(cccc1OCC=C)O PS-4192 CC(=O)c1c(ccc(c1O)OC)OC PS-4193 COCC(=O)c1ccc(cc1O)O PS-4194 CCOc1ccc(cc1)C(=O)CCC(=O)O PS-4195 CCOc1cc(cc(c1O)Br)C=O PS-4196 CC(C)Cc1ccc(cc1)C(=O)C PS-4197 c1c(nc(nc1Cl)N)N PS-4198 c1ccc(cc1)c2c(c2=O)c3ccccc3 PS-4199 CCNc1ccc(cc1)C(=O)O PS-4200 CCCC(=O)c1ccc(cc1)O PS-4201 Cc1cc(nc(n1)C)NN PS-4202 COC(=O)c1ccc2c(c1)[nH]cc2C=O PS-4203 c1cc(c(cc1C=O)O)I PS-4204 Cc1cc(c(c(c1)CO)O)CO PS-4205 c1cc(c(c(c1)Br)[N+](=O)[O-])N PS-4206 c1ccc2c(c1)ccc(n2)N PS-4207 c1ccc(cc1)C=CC(=O)c2cccs2 PS-4208 c1cc(nnc1C=O)O PS-4209 c1ccc(c(c1)C(=O)NC2CCCCC2)N PS-4210 CN(C)S(=O)(=O)c1ccc(c(c1)N)O PS-4211 c1c(nc(nc1O)N)N PS-4212 C1[C@@H]2C=CC(=O)[C@H](O1)O2 PS-4213 CCOC(=O)c1cc2cc(ccc2[nH]1)[N+](=O)[O-] PS-4214 CCc1cccc(n1)N PS-4215 c1ccc(c(c1)S)Br PS-4216 CNCCc1ccccn1 PS-4217 CC(C)(C)OC(=O)NCC(Cc1ccccc1)C(=O)O PS-4218 CC(=O)/C=C/c1cn(c2c1cccc2)C PS-4219 c1c(c(sc1C(=O)O)Br)Br PS-4220 C1CC2CC1CC2C(=O)O PS-4221 Cn1c2ccccc2c(c(c1=O)[N+](=O)[O-])Cl PS-4222 CC(C)(C)OC(=O)N1CC(C1)CN PS-4223 CC(C)(C)OC(=O)N1CC(C1)I PS-4224 c1cc2c(cc1CCCC(=O)O)OCCO2 PS-4225 Cc1ccc2cc[nH]c2c1 PS-4226 CC(C)(C)OC(=O)NCCC1CCNCC1 PS-4227 CCOc1ccc(cc1)NC(=O)N PS-4228 c1c(cc(nc1Br)Br)C(=O)O PS-4229 c1cc(c(nc1)Br)N PS-4230 COc1cc(cc(c1OC)OCc2ccccc2)C=O PS-4231 CC(C)Cn1cnc2c1cccc2 PS-4232 c1ccc(cc1)C2(CCC2)C(=O)O PS-4233 CN1[C@@H]2CC[C@H]1C[C@H](C2)O PS-4234 c1ccnc(c1)c2ccc(s2)C(=S)N PS-4235 CC(C)(C)OC(=O)Nc1ccco1 PS-4236 Cc1c(c(on1)C)N PS-4237 Cc1c(c(on1)C)C#N PS-4238 c1cc(c(cc1Br)N)N PS-4239 Cc1c(c(no1)c2ccccc2)C=O PS-4240 Cc1c(c(no1)c2ccccc2)CO PS-4241 Cc1c(c(no1)c2ccccc2)CN PS-4242 Cc1c(c(on1)C)C=O PS-4243 Cc1cc(c(o1)C)CN PS-4244 c1cc2c(cc1C(=O)O)OCCO2 PS-4245 c1cc(c2c(c1)OCCO2)C(=O)O PS-4246 c1cocc1C(=O)O PS-4247 c1cc2c(cc1N)CCO2 PS-4248 c1cocc1Br PS-4249 c1ccnc(c1)c2ccc(s2)C=O PS-4250 c1ccnc(c1)c2ccc(s2)CO PS-4251 Cn1cccc1CN PS-4252 c1ccnc(c1)C(=O)O PS-4253 c1ccnc(c1)Br PS-4254 c1cc(cnc1)C(=O)O PS-4255 c1cncc(c1Cl)Br PS-4256 c1cc(cnc1)Br PS-4257 c1cc2cccnc2c(c1)C=O PS-4258 c1cc2cc(ccc2nc1)Br PS-4259 Cc1c(sc(n1)C)Br PS-4260 c1ccc2c(c1)nc(s2)CO PS-4261 c1cnc(nc1)Br PS-4262 Cc1cc(c(n1C)C)C(=O)O PS-4264 c1c(nc[nH]1)C(=S)N PS-4265 c1cc(c2c(c1)nsn2)C=O PS-4266 c1cc2c(cc1C(=O)O)nsn2 PS-4267 c1cc2c(cc1N)nsn2 PS-4268 c1csc(n1)Br PS-4269 c1ccc(cc1)c2c(nco2)C(=O)O PS-4270 c1ccc2c(c1)C[C@@H]([C@@H]2N)O PS-4272 c1ccc2c(c1)c(cs2)C=O PS-4273 c1ccc(cc1)CN2CCOC(C2)CO PS-4274 Cc1cc(n(n1)C)CO PS-4275 Cc1cc(nn1C)CO PS-4276 c1ccc(cc1)c2ccno2 PS-4277 c1cscc1CN PS-4278 CN1CCOc2c1ccc(c2)Br PS-4279 c1cc(ccc1c2cnco2)C(=O)O PS-4281 Cc1c(cnn1c2ccccc2)CO PS-4282 Cc1ccnn1c2ccccc2 PS-4283 Cc1c(nn(n1)c2ccccc2)CN PS-4284 c1cc(ccc1c2csnn2)C(=O)O PS-4285 c1cc(ncc1C(=O)NN)N2CCOCC2 PS-4286 Cc1cc([nH]c1C(=O)O)C PS-4287 Cc1nc(cs1)c2ccc(s2)C=O PS-4288 c1ccc(cc1)c2nc(cs2)C=O PS-4289 c1cnn(c1)c2ccc(cc2)C(=O)O PS-4290 c1cnn(c1)c2ccc(cc2)N PS-4291 c1cc(ccc1C(=O)O)n2ccnc2 PS-4292 c1cc(ccc1C(=O)O)n2cncn2 PS-4293 CN1CCN(CC1)c2ccc(cc2)C(=O)O PS-4294 Cc1nc(cs1)c2cccc(c2)C(=O)O PS-4295 c1ccc(cc1)Oc2ccc(cn2)N PS-4296 Cc1ncc(c(n1)c2ccccc2)C(=O)O PS-4297 c1cnc(nc1)N2CCC(CC2)CO PS-4298 c1ccn(c1)c2cccc(c2)C(=O)O PS-4299 c1ccn(c1)c2cccc(c2)C=O PS-4300 Cc1c2cc(sc2n(n1)C)C(=O)O PS-4301 Cn1c2ccc(cc2nn1)C(=O)O PS-4302 Cn1c2ccc(cc2nn1)CO PS-4303 c1ccc(c(c1)C(=O)O)N2CCOCC2 PS-4304 c1ccc(cc1)n2c(ccn2)C(=O)O PS-4305 c1ccc(cc1)n2c(ccn2)C=O PS-4306 c1cc(c(nc1)N2CCOCC2)CO PS-4307 c1ccn(c1)c2ccc(cc2)CN PS-4308 COc1ccc(cc1)C#N PS-4309 COc1cc2c(cc1OC)COC(=O)C2 PS-4310 CS(=O)(=O)c1cc(c(c(c1)Cl)O)Cl PS-4311 COc1cccc(c1CO)OC PS-4312 C1CCN(CC1)CC#N PS-4313 CSc1cc(ccc1[N+](=O)[O-])Cl PS-4314 Cc1c(snn1)C(=O)N PS-4315 CN(c1c(cccn1)[N+](=O)[O-])N PS-4316 c1cc(c(c(c1)Cl)Cl)C#N PS-4317 c1csc(c1Br)Br PS-4318 Cc1[nH]c2cc(c(cc2n1)Cl)Cl PS-4319 c1cc(c(cc1O)Cl)C(=O)O.O PS-4320 c1cc(ccc1N)n2ccnc2 PS-4321 c1ccc(cc1)CCCC(=O)O PS-4322 Cc1c(cco1)CO PS-4323 Cc1c(sc(n1)NC(=N)N)Br PS-4324 CC(=O)c1ccc(cc1)Oc2ccc(cc2)OC PS-4325 c1c(csc1[N+](=O)[O-])C=O PS-4326 c1c(csc1[N+](=O)[O-])C#N PS-4327 C#CCN1CCS(=O)(=O)CC1 PS-4328 c1cc(c(cc1Cl)C#N)Cl PS-4330 C1C(CC(=O)CC1=O)C(=O)O PS-4331 c1cc(ccc1CC(=S)N)[N+](=O)[O-] PS-4332 c1cc(cnc1)CNCCC#N PS-4333 c1cc(c(cc1S(=O)(=O)N)[N+](=O)[O-])Cl PS-4334 CC(C)(C)OC(=O)c1cccc(c1)N PS-4335 c1cc(c(cc1Cl)Cl)NN PS-4337 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NN PS-4338 c1cn[nH]c1[N+](=O)[O-] PS-4339 c1cc(nn2c1nnc2)Cl PS-4340 CCOC(=O)c1cnn(c1n2cccc2)C PS-4341 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)N PS-4342 c1ccc2c(c1)c(c(c(=O)[nH]2)C#N)Cl PS-4343 CCCc1c(cn[nH]1)C(=O)OCC PS-4344 c1cc2c(cc1Br)OCCO2 PS-4345 c1csc2c1[nH]c(=O)oc2=O PS-4346 Cc1csc(c1Cl)C(=O)NN PS-4347 c1csc2c1n3c(c(cn3)C(=O)O)nc2Cl PS-4348 CN(C)c1ccc(c(c1)Cl)C=O PS-4349 COC(=O)c1cscc1N PS-4350 COC(=O)c1c(csc1C(=O)OC)N PS-4351 c1csc2c1ncn(c2=O)N PS-4352 c1ccc2c(c1)ccc(c2O)[N+](=O)[O-] PS-4354 c1cc(cc(c1)Br)S PS-4355 CCC1CCCCC(=O)N1C PS-4356 c1c(csc1CC(=O)O)Br PS-4357 Cc1c(c(n(n1)Cc2ccc(o2)C(=O)O)C)Br PS-4358 c1ccc2c(c1)C(=O)CO2 PS-4359 CC1(C(N(C(S1)(C)C)C=O)C(=O)O)C PS-4360 c1cc(c(nc1)I)O PS-4361 c1cc2c(cc1CN)CCO2 PS-4362 CC(C)(C)c1c(=O)n(c(nn1)S)N PS-4363 Cc1nc(c(c(n1)Cl)N)Cl PS-4364 CCOC(=O)/C=C/c1ccc(c(c1)OC)O PS-4365 COc1cc(ccc1O)/C=C/CO PS-4366 Cn1c2c(cn1)c(=O)[nH]cn2 PS-4367 CCCCOc1ccc(cc1)S(=O)(=O)N PS-4368 CCCCc1[nH]cc(n1)C=O PS-4369 c1c(c(n[nH]1)C#N)Br PS-4370 COC(=O)c1cc(cc(c1)O)O PS-4371 c1ccc2c(c1)c(ccc2[N+](=O)[O-])N PS-4372 Cc1csc(n1)C=O PS-4373 c1cc(ccc1CCO)Cl PS-4374 CN(C)C(=N)NC(=O)c1cc(nc(c1)Cl)Cl PS-4375 CC(=O)c1ccc(c(c1)N)Cl PS-4376 COC(=O)C1CSCC1=O PS-4377 CCO/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl PS-4378 Cc1cc2c([nH]1)cccc2[N+](=O)[O-] PS-4379 COC(=O)c1c(c(cs1)C#N)N PS-4380 CCOC(=O)Cn1cnc(c1Cl)Cl PS-4381 c1nc(c(n1CC(=S)N)Cl)Cl PS-4382 c1c(nc[nH]1)[N+](=O)[O-] PS-4383 COC(=O)c1c(c(cs1)S(=O)(=O)C)N PS-4384 CCOC(=O)c1c[nH]c2cc(nn2c1=O)C PS-4385 Cc1ccc(cc1)S(=O)C PS-4386 c1nc(c(n1Cc2n[nH]nn2)Cl)Cl PS-4387 CCOC(=O)c1c2c(c(s1)SC)C(=O)CCC2 PS-4388 CC1(CCc2cc(ccc2O1)C=O)C PS-4389 c1cc(sc1)C2CC(=O)CS2 PS-4390 CC1(COC(=S)N1)C PS-4391 c1ccc(cc1)Oc2ccsc2C=O PS-4392 CSc1ccsc1 PS-4393 c1cc2c(cc1C(=S)N)non2 PS-4394 Cc1c(ccc(n1)N)[N+](=O)[O-] PS-4395 CC(C)(c1ccccn1)O PS-4396 Cc1ccc(c(n1)Br)N PS-4397 COC(=O)c1cc(nc(n1)Cl)Cl PS-4398 CN1CCN(C(C1)CO)C PS-4399 COc1cc2c(cc1OC)[nH]cnc2=O PS-4400 CCOC(=O)c1c(nc(s1)N)c2ccccc2 PS-4401 COc1ccc(cc1OC2CCCC2)C#N PS-4402 c1cc2c(c(c1)C(=O)O)NC(=O)C2=O PS-4403 c1cc(c(nc1)Cl)C(=O)NCCSCc2ccco2 PS-4404 CN(C)c1ccccc1[N+](=O)[O-] PS-4405 COc1ccc2c(c1)occ2CC(=O)O PS-4406 Cc1ccc(cc1N)I PS-4407 c1c(nc([nH]1)Cl)[N+](=O)[O-] PS-4408 c1ccc2c(c1)c(cc(n2)O)O PS-4409 COc1ccc(cc1)C(=S)N PS-4410 c1cnccc1I PS-4411 CS(=O)(=O)c1ccc(cc1)C(=O)O PS-4412 Cc1cc(cc(n1)O)C(=O)O PS-4413 CC(C)(C)C(=O)Nc1ccncc1C=O PS-4414 c1ccc(cc1)c2cc(ccn2)C(=O)O PS-4415 c1cscc1C(=S)N PS-4416 c1ccc(c(c1)N)n2cccn2 PS-4417 c1csc(c1O)C(=O)O PS-4418 c1c[nH]c(=O)c2c1occ2 PS-4419 CNc1ccc(cc1N)C#N PS-4420 c1cnc(c2c1occ2)Cl PS-4421 c1ccc2c(c1)c(no2)N PS-4422 COc1cccc2c1c(no2)N PS-4423 Cc1csc(n1)C(=O)O PS-4424 CC(=O)c1ccc(c(c1)N)NC PS-4425 Cc1cnc(s1)C(=O)O PS-4426 Cc1ccc(n1CCN2CCNCC2)C PS-4427 c1c2nc(cn2cc(n1)Br)C(=O)O PS-4428 Cc1c(c(n(n1)C)C(=O)O)Br PS-4430 c1cc(c2c(c1)OCCO2)C(=O)N PS-4431 c1cc2c(cc1[N+](=O)[O-])S(=O)(=O)C=C2 PS-4432 Cc1ccc2c(c1)ccs2 PS-4433 Cc1c2cc(ccc2sc1CC(=O)O)Cl PS-4434 C1C(=O)N=C(S1)CC#N PS-4435 Cc1cnc(s1)CO PS-4436 Cc1csc(n1)CO PS-4437 c1cc2c(cc1Cl)c(c(s2)Br)C=O PS-4438 c1ccc2c(c1)CC(C2O)N PS-4439 CC1=NN(C(=O)C1)C PS-4440 c1cc2cccc3c2c(c1)C(=O)N3 PS-4441 c1ccc(c(c1)CC(=O)O)I PS-4442 CC(=O)Nc1ccc2c(c1)CCCC2=O PS-4443 c1cc2c(cc1N)CCCC2=O PS-4444 c1cc2c(cc1N)CCC2=O PS-4445 COc1ccc2ccccc2c1[N+](=O)[O-] PS-4446 Cc1c(nns1)c2ccccc2 PS-4447 Cc1c(ccs1)C=O PS-4448 CC(=O)Nc1ccc(cc1)S(=O)(=O)N PS-4449 COc1ccccc1CO PS-4450 Cc1ccc(c(c1)N)Cl PS-4451 COc1cc(c(cc1N)Cl)[N+](=O)[O-] PS-4452 COc1ccc(cc1[N+](=O)[O-])C=O PS-4453 COc1ccc(cc1Cl)N PS-4454 c1ccc2c(c1)c(ns2)Cl PS-4455 COc1cccc(c1)S(=O)(=O)N PS-4457 c1c(nc([nH]c1=O)N)N PS-4458 c1cc(c(c(c1)Cl)N)[N+](=O)[O-] PS-4459 COc1ccc(c(c1)N)[N+](=O)[O-] PS-4460 CC(=O)N1CCc2c1c(ccc2)N PS-4461 c1ccc(cc1)c2[nH]nnn2 PS-4462 CC(=O)N1CCc2c1cc(cc2)N PS-4463 CC(=O)c1ccc(c(c1)[N+](=O)[O-])OC PS-4464 c1cc2c3c(ccc(c3c1)N)CC2 PS-4465 Cc1c(scn1)CCO PS-4466 COC(=O)c1ccc2c(c1)nn[nH]2 PS-4467 Cc1cccc2c1nsn2 PS-4468 c1cc(c(cc1Cl)C(=O)O)N PS-4469 CCOc1c(=O)c(=O)c1OCC PS-4470 COc1c(=O)c(=O)c1OC PS-4471 Cc1cc(cc(c1C#N)C)O PS-4472 Cc1cc(cc(c1O)C)C#N PS-4473 COc1cc(ccc1O)/C=C/[N+](=O)[O-] PS-4474 c1cc(ccc1c2ccc(o2)C=O)S(=O)(=O)N PS-4475 Cc1cc(nc(c1)O)C PS-4476 c1cc(c(cc1Cl)N)N PS-4477 c1ccc(cc1)C(=O)/C=N/O PS-4479 Cc1cc(nc(c1C(=O)N)Cl)Cl PS-4480 C1COCCN1CC(=O)N PS-4481 CCOC(=O)c1cc(nc(c1C#N)Cl)C PS-4482 c1c(cc(nc1Cl)Cl)C(=O)N PS-4483 Cc1ccc(c(c1)C(=O)OC)O PS-4484 COC(=O)c1cc(ccc1O)Cl PS-4485 c1ccc2c(c1)c(no2)O PS-4486 c1c(cc(nc1Cl)Cl)C#N PS-4487 c1cc(ccc1NN)I PS-4488 CC(C)(C)c1ccc(c(c1)N)N PS-4489 CC(C)(C)c1ccc(c(c1)N)NC(=O)CN2CCOCC2 PS-4490 c1ccc(cc1)S(=O)(=O)c2ccc(cc2)C=O PS-4491 CSc1nc(nc(n1)N)c2cccs2 PS-4492 c1cc(nc(c1NC(=O)CSCC(=O)O)Cl)Cl PS-4493 Cc1cccc2c1onc2O PS-4494 COC(c1cc[nH]n1)OC PS-4495 C1CSCCC1=O PS-4496 Cn1cc(c(n1)C=O)Cl PS-4497 c1c(c([nH]n1)C=O)Br PS-4498 c1c(cc(nc1Cl)Cl)N PS-4499 c1cncc(c1O)C(=O)O PS-4500 c1ccc2c(c1)C(c3ccccc3O2)C(=O)O PS-4501 c1cc(nnc1Br)Br PS-4502 Cn1ccc(=O)n(c1=O)C PS-4503 CCOC(=O)c1ccc2c(c1)nccn2 PS-4504 c1cc2c(nc1)sc(n2)S PS-4505 c1cc2c(cc[nH]2)cc1N PS-4506 c1ccc(c(c1)N)S(=O)(=O)N PS-4507 CCOc1cccc(c1)/C=C/C(=O)O PS-4508 c1cc2c(cc1N)[nH]cn2 PS-4509 Cc1cc(=O)[nH]c(=S)[nH]1 PS-4510 Cc1cc(c(cc1C)N)C PS-4511 Cc1ccc(cc1Cl)N2CCNC2=O PS-4512 Cc1ccc(c(n1)C)O PS-4514 c1cc(cc(c1)O)C(=O)c2cc(ccc2N)Cl PS-4515 c1cc(c(c(c1[N+](=O)[O-])Cl)C=O)Cl PS-4516 c1cc(c(c(c1[N+](=O)[O-])Cl)CO)Cl PS-4517 CN1C2CCC1CC(=O)C2 PS-4518 Cc1c(cccc1O)[N+](=O)[O-] PS-4519 CC(=O)Nc1cccc(c1)O PS-4520 CN1CCN(C1c2ccncc2)C PS-4521 C1CCC(CC1)C(=O)N PS-4522 Cc1cc(c2ccccc2n1)N3CCNCC3 PS-4523 COc1ncc(cn1)C=O PS-4524 c1cc(c(nc1)C(=O)O)N PS-4525 CCOC(=O)C1CCCC(=O)C1 PS-4526 c1c([nH]c(=O)[nH]c1=O)N PS-4527 COC(=O)c1ccc(cc1)C(=O)O PS-4528 c1cc2cc(ccc2nc1)N PS-4529 c1ccc2c(c1)N(C(=O)CS2)CC(=O)O PS-4530 c1cc2c(cc1N)scn2 PS-4531 COc1ccc(c(n1)Cl)[N+](=O)[O-] PS-4532 c1cc2cc[nH]c2nc1 PS-4533 CCOC(=O)c1cc2ccccc2cc1O PS-4534 C1C(=O)N=C(S1)N PS-4535 c1cncc(c1C#N)Cl PS-4536 Cc1ccc2c(c1)C(=O)CC2 PS-4537 c1cnc(nc1N)Cl PS-4538 CCOC(=O)c1c(sc(n1)N)Br PS-4539 CNC(=O)c1ccc(cc1)N PS-4540 Cc1ccc2c(c1)ocn2 PS-4542 c1cc(ccc1C(=O)O)S PS-4543 COC(=O)c1c(ccc(n1)Cl)Cl PS-4544 c1ccc2c(c1)cncc2N PS-4545 c1cc(c2c(c1)OCCO2)N PS-4546 c1cc(cnc1)C2CCCCN2 PS-4547 C=CCNC(=O)OCc1ccccc1 PS-4548 CCOC(=O)c1c(nco1)C PS-4549 COc1ccc(c(c1)OC)CO PS-4550 COCc1cc(=O)oc2c1ccc(c2)N PS-4551 c1cc(ccc1S(=O)(=O)N)I PS-4552 c1cc2cccnc2c(c1)O PS-4553 Cc1ccc2c(c1)nc([nH]2)C PS-4554 c1ccc(c(c1)NC(=S)N)Cl PS-4555 c1cc2c(cc1Cl)c(c[nH]2)C=O PS-4556 C1CC(=O)N(C1=O)O PS-4557 CSc1nnc(s1)N PS-4558 c1ccc(c(c1)N2CCOCC2)O PS-4559 Cc1cc(ccn1)Cl PS-4560 c1cc(c2c(c1Cl)C(=O)C(=O)N2)Cl PS-4561 c1cc(c(cc1C(=O)O)O)N PS-4562 c1cc(c(c(c1)Cl)C(=O)N)Cl PS-4563 c1cc2c(cc1N)OCO2 PS-4564 CC(C)c1ccccc1N PS-4565 c1cc2cccc3c2c(c1)C(=O)OC3=O PS-4566 c1cc(c(cc1Cl)[N+](=O)[O-])C(=O)O PS-4567 c1c(cc(cc1Cl)Cl)N PS-4568 CCOC(=O)Cc1ccc(c(c1)OC)OC PS-4569 c1cc(c(nc1)Cl)[N+](=O)[O-] PS-4570 Cc1cccc(c1C(=O)O)N PS-4571 c1cc(ccc1CC#N)O PS-4572 COc1ccccc1Br PS-4573 c1cc(ccc1C(=S)N)Cl PS-4574 CC(C)c1ccc(cc1)C(=O)C PS-4575 c1cc(cc(c1)[N+](=O)[O-])C#N PS-4576 c1cc(c(nc1)Cl)O PS-4577 Cc1c(c(=O)cco1)O PS-4578 CC(=O)c1ccccc1N PS-4579 Cc1ccccc1C=O PS-4581 c1cc(c(cc1Cl)N)[N+](=O)[O-] PS-4582 COC(=O)c1ccc(c(c1)N)C(=O)OC PS-4583 Cc1cnc(cn1)C(=O)O PS-4584 CCOC(=O)c1coc(n1)Cl PS-4585 CC(=O)c1ccco1 PS-4586 CC(=O)c1ccc(cc1)N PS-4587 c1ccc2c(c1)CCOC2 PS-4588 COc1ccc(cc1O)C=O PS-4589 COc1cccc(c1)N PS-4590 COc1ccc(c(c1OC)Cl)C=O PS-4591 Cc1ccc(c(c1)C(=O)O)O PS-4592 c1ccc(cc1)n2c(nnn2)S PS-4593 Cc1[nH]cc(n1)C=O PS-4594 CCc1[nH]c(c(n1)C)C=O PS-4595 Cc1c([nH]cn1)C=O PS-4596 Cc1nnc(s1)N PS-4597 Cc1ccc(c(c1)[N+](=O)[O-])O PS-4598 c1ccc2c(c1)CCO2 PS-4599 CN(C)c1ccncc1 PS-4600 C[C@@H](c1ccccc1)N PS-4601 c1cc(cc2c1cc[nH]2)N PS-4602 c1cc(c(cc1[N+](=O)[O-])N)O PS-4603 C1C2CC3CC1CC(C2)(C3)O PS-4604 Cn1c(nnn1)S PS-4606 COc1cccc(c1C(=O)O)N PS-4607 c1cc(ccc1c2cc[nH]n2)N PS-4608 c1cc(ccc1CC(=O)N)O PS-4609 CN(C)CCc1ccccn1 PS-4610 c1cc(c(cc1CC#N)Cl)Cl PS-4611 CC(=O)CCc1ccc(cc1)O PS-4612 c1ccc2c(c1)CC(C2)N PS-4613 CC(=O)c1ccc(cc1)[N+](=O)[O-] PS-4614 CCOC(=O)c1cccnc1Cl PS-4615 c1cc(ccc1c2cc[nH]n2)C(=O)O PS-4616 Cc1cccc(c1C=O)Cl PS-4617 c1cc(ccc1c2csnn2)N PS-4618 c1cnccc1c2cnco2 PS-4619 c1ccnc(c1)c2cnco2 PS-4620 c1cc(c(cc1C#N)Cl)NN PS-4621 Cc1c(oc(n1)C)C(=O)C PS-4622 c1cc(ccc1OCCC#N)Cl PS-4624 CCc1cnc(nc1)Cl PS-4625 Cc1cn(c2c1cccc2)CCC(=O)O PS-4626 CC(=O)Nc1cccc(c1)C#N PS-4627 Cc1ccnc(c1[N+](=O)[O-])Cl PS-4628 c1cc(cc(c1)C#N)C=O PS-4629 CN(c1cnc2ccccc2n1)N PS-4630 CC1(COC(=N1)c2ccc(cc2)OC)C PS-4631 c1cc2c(cc1O)c(co2)[N+](=O)[O-] PS-4632 CS(=O)(=O)c1ccc(s1)C(=O)O PS-4633 c1ccn(c1)c2ccc(cc2)N PS-4635 Cc1cc(c(c(c1)C(=O)O)N)C PS-4636 CCOC(=O)C1CCN(CC1)c2ccccc2C=O PS-4638 C1COCCN1CCCC#N PS-4639 c1ccc(c(c1)CSCCN)Cl PS-4640 c1cncc2c1C(=O)NC2=O PS-4641 Cc1cc(c(o1)C)C(=O)CC#N PS-4642 CCOC(=O)c1cc(oc1C)c2ccc(cc2)N PS-4643 Cc1nc(cs1)CC(=O)OC(C)C PS-4644 Cc1ccsc1CN PS-4645 c1cc2c(cc1Cl)c(cs2)C=O PS-4646 CC(C)n1c(nnc1S)O PS-4647 CC(C)(C)c1cc([nH]n1)C(=O)NN PS-4648 c1cc(sc1)C(=S)N PS-4649 COc1ccc2c(c1)nc(s2)N PS-4650 c1cc(ccc1C2=NCCS2)OCC#N PS-4651 c1cc(cc(c1)Cl)C(=S)N PS-4652 Cc1nc(cs1)C(=O)N PS-4653 Cc1nc(cs1)C#N PS-4654 c1ccc2c(c1)n(c(=O)o2)CCC(=O)O PS-4655 COc1ccc(c(c1)[N+](=O)[O-])C=O PS-4656 CCn1c(c(c(n1)C)Br)C(=O)OC PS-4657 COC(=O)c1ccc(cc1Cl)Cl PS-4659 Cc1cc(no1)/C(=N\O)/N PS-4660 COC(c1ccc(c(n1)S)C#N)OC PS-4661 CCOC(=O)c1ccc(nc1)Cl PS-4662 CC(c1ccccc1)C(=O)O PS-4663 COC(=O)c1ccc(nn1)Cl PS-4664 CCOC(=O)c1cnc(nc1Cl)c2cccs2 PS-4665 Cc1ccc(cn1)C(=S)N PS-4666 c1cncc(c1I)Cl PS-4667 COc1cc(ccn1)C(=O)N PS-4669 c1cc(cc(c1)Cl)C(=O)NN PS-4670 c1c(c(c(cn1)Cl)N2CCNCC2)Cl PS-4671 Cc1cc(nnc1)Cl PS-4672 c1c(cnc(c1N)Cl)Cl PS-4673 c1cnc(cc1C(=O)N)Cl PS-4674 Cc1c(ccnc1CO)[N+](=O)[O-] PS-4675 c1cnc(cc1C(=O)NN)Cl PS-4676 c1cc(ncc1C(=O)NN)Cl PS-4677 Cc1ccc(c(n1)Cl)[N+](=O)[O-] PS-4678 CSc1nc(cc(n1)Cl)Cl PS-4679 c1cnccc1C(=O)CC#N PS-4680 c1cc(c(cc1N)Cl)Br PS-4681 c1c(cnc(c1N)Cl)Br PS-4682 c1cnc(cc1O)O PS-4683 CCOC(=O)c1[nH]ccn1 PS-4684 c1cc(oc1)CNC(=O)c2ccnc(c2)Cl PS-4686 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)O PS-4687 CC(C)(C)OC(=O)N1CCC(CC1)CCCO PS-4688 c1cc(ccc1CCO)Br PS-4689 Cc1cccc(c1C)CN PS-4690 c1c(cc(cc1Cl)Cl)CN PS-4691 Cc1cccc(c1)C(=O)OC PS-4692 Cc1ccc(cc1C)C=O PS-4693 c1cc(cc(c1)O)N2CCOCC2 PS-4694 c1ccc(cc1)[C@@H](CN)O PS-4695 CNCc1cccnc1 PS-4696 c1c2c(cc(c1[N+](=O)[O-])Cl)C(=O)NC2=O PS-4697 c1cc(ccc1CC(=O)O)Br PS-4698 Cc1ccc(cc1)CS PS-4699 Cc1cccc(c1)CS PS-4700 c1cc(oc1)c2cc([nH]n2)N PS-4701 c1ccc(c(c1)S(=O)(=O)N)Br PS-4702 Cc1ccc(c(c1)N)C#N PS-4703 CC(=O)c1cccc(c1)Br PS-4704 Cc1ccc(c(c1)N)C(=O)O PS-4705 Cn1c(cc(n1)C2CC2)N PS-4706 c1cc2c(cc1C#N)OCCO2 PS-4707 c1ccc(cc1)c2c(c([nH]n2)N)Br PS-4708 Cc1cc(c(cc1Cl)N)N PS-4709 Cc1cc(c(cc1C)N)N PS-4710 CCc1ccc(cc1)C(=O)NN PS-4711 c1cc(c(cc1[N+](=O)[O-])Cl)C(=O)N PS-4712 COc1ccc(cc1OCc2ccccc2)C=O PS-4713 Cc1c(nc(s1)C)CC(=O)O PS-4714 Cc1c(c(no1)c2ccccc2)N PS-4715 C1C(=O)NCC(=O)N1 PS-4716 c1cc(sc1)S PS-4717 c1cc(cnc1)/C=C/C(=O)O PS-4718 CC1(CCCC(N1)(C)C)C PS-4719 CC(=O)c1cccc(c1)N(C)C(=O)C PS-4720 C=Cc1ccc(cc1)N PS-4721 c1cc(c(cc1C(=O)O)N)C(=O)O PS-4722 c1cc(ccc1S(=O)(=O)N)Br PS-4723 CSc1ccccc1Br PS-4724 c1c(cnc(n1)Cl)[N+](=O)[O-] PS-4725 c1cc(cc2c1ccnc2)O PS-4726 c1ccc2c(c1)CC(C2)O PS-4727 Cc1cc(ccc1[N+](=O)[O-])C=O PS-4728 CCOC(=O)Cc1ccccc1[N+](=O)[O-] PS-4729 c1c(cnc(n1)Cl)N PS-4730 c1cnc(nc1C(=O)N)Cl PS-4731 COc1nccc(n1)Cl PS-4732 COc1cc(ccn1)N PS-4733 c1cc2cnccc2c(c1)C=O PS-4734 c1cc2cnccc2cc1C=O PS-4735 c1cc2ccncc2c(c1)C=O PS-4736 c1cc2cnccc2cc1CO PS-4737 c1cc2ccncc2c(c1)CO PS-4738 c1cncc2c1scc2 PS-4739 c1cncc2c1c(cs2)Br PS-4740 c1cc2nccn2c(c1)Br PS-4741 c1cnc([nH]1)C(=O)O PS-4742 Cc1cc(c(cc1N)Br)C PS-4743 Cn1c2c(cn1)c(nc(n2)Cl)Cl PS-4744 Cc1c2c(nc(nc2Cl)Cl)n(n1)C PS-4745 COc1ccc(cc1[N+](=O)[O-])Br PS-4746 c1ccn2c(c1)nc(c2Cl)Br PS-4747 c1cncc2c1[nH]cc2Br PS-4748 c1ccc2c(c1)c(n[nH]2)C=O PS-4749 c1ccc2c(c1)cn[nH]2 PS-4750 c1cc2c(cn[nH]2)nc1 PS-4751 c1cncc2c1[nH]nc2 PS-4752 COC(=O)c1c[nH]cn1 PS-4754 CC(=O)c1cncnc1 PS-4755 COc1cccc(c1[N+](=O)[O-])Br PS-4756 Cn1c2cccc(c2cn1)C=O PS-4757 Cn1c2cc(ccc2cn1)C=O PS-4758 COC(=O)c1cccc2c1cn[nH]2 PS-4759 Cn1c2ccc(cc2cn1)C(=O)OC PS-4761 Cn1c2cc(ccc2cn1)C(=O)OC PS-4762 Cn1c2c(cccc2C(=O)OC)cn1 PS-4763 Cn1cc2c(cccc2n1)C(=O)OC PS-4764 Cn1cc2cccc(c2n1)C(=O)OC PS-4765 c1cc(c2cnn(c2c1)C3CCCCO3)C(=O)O PS-4766 c1cc2c(cc1C(=O)O)cnn2C3CCCCO3 PS-4767 c1cc2cnn(c2cc1C(=O)O)C3CCCCO3 PS-4768 c1cc2c(cc1CO)cn[nH]2 PS-4769 CC(C)(C)OC(=O)n1c2ccc(cc2cn1)N PS-4770 c1cc2c(cc1C#N)cn[nH]2 PS-4771 c1cc(cc(c1)Br)CC(=O)O PS-4772 Cc1cc2cn[nH]c2cc1Br PS-4773 c1cncc2c1c(n[nH]2)Br PS-4774 c1cc2c([nH]nc2Br)nc1 PS-4775 c1c[nH]c2c1c(ncc2)Cl PS-4776 c1cc(cc(c1)Br)CC#N PS-4777 CN1Cc2c(cccc2Br)C1=O PS-4778 CN1c2cccc(c2CC1=O)Br PS-4779 c1c(cc(nc1C(=O)O)Cl)Cl PS-4780 c1c(cc(nc1Br)Br)N PS-4781 Cc1cc(cc(n1)O)C(=O)OC PS-4782 CC1(CCCCC1)C=O PS-4783 CNCC1CCOCC1 PS-4784 c1cc2c(cc1N)oc(=O)[nH]2 PS-4785 Cc1c(oc(n1)c2ccccc2)CN PS-4786 c1c(cn[nH]1)C(=O)O PS-4787 c1cc2c(cc1CN)cn[nH]2 PS-4788 c1cc2cn[nH]c2cc1CN PS-4790 Cn1c2cccc(c2cn1)O PS-4791 Cn1c2cc(ccc2cn1)O PS-4792 Cn1c2ccc(cc2cn1)C#N PS-4793 Cn1c2cc(ccc2cn1)C#N PS-4794 c1cc(c2cn[nH]c2c1)CO PS-4795 c1cc2cn[nH]c2cc1CO PS-4796 c1cc(c2cn[nH]c2c1)CN PS-4797 c1cc2cn[nH]c2c(c1)CN PS-4798 Cn1c2ccc(cc2cn1)CN PS-4799 CN(C)c1ccc(cc1)N=O PS-4800 CC(=O)c1cccc2c1cn[nH]2 PS-4801 CC(=O)c1ccc2c(c1)cn[nH]2 PS-4802 CC(=O)c1ccc2cn[nH]c2c1 PS-4803 CC(=O)c1cccc2c1[nH]nc2 PS-4804 CC(=O)c1cccc2c1cnn2C PS-4805 CC(=O)c1ccc2c(c1)cnn2C PS-4806 CC(=O)c1ccc2cnn(c2c1)C PS-4807 CC(=O)c1cccc2c1n(nc2)C PS-4808 CC(=O)c1cccc2c1cn(n2)C PS-4809 CC(=O)c1ccc2cn(nc2c1)C PS-4810 CC(=O)c1cccc2c1nn(c2)C PS-4811 c1cc(c(cc1Br)C#N)[N+](=O)[O-] PS-4812 c1cc(c(cc1Br)O)[N+](=O)[O-] PS-4813 c1cc(c(cc1Br)O)N PS-4814 COc1cc(ccc1[N+](=O)[O-])Br PS-4815 COc1cc(ccc1N)Br PS-4816 c1cnc(nc1N)N PS-4817 Cc1cc(nc(c1)Cl)C PS-4818 Cc1ccnc(c1N)Br PS-4820 c1cnc(cc1N2CCCC2)N PS-4821 c1cncc(c1C#N)N PS-4822 COC(=O)c1ccnc(c1N)Cl PS-4823 Cc1cc(nc(c1N)Cl)Cl PS-4824 COc1ncc(cn1)N PS-4825 CCc1cc(nc(n1)N)O PS-4826 c1cc(c(cc1Cl)O)C=O PS-4828 Cn1ccc(n1)C=O PS-4829 Cc1ccc2cc(sc2c1)C(=O)O PS-4830 CC(C)(C)OC(=O)N1CCNCC1c2ccccc2 PS-4831 C[C@@H]1CNCCN1C(=O)OC(C)(C)C PS-4832 COc1c2c(cc[nH]2)ccn1 PS-4833 c1ccc(cc1)COc2cccnc2N PS-4834 COc1ccnc(c1[N+](=O)[O-])N PS-4835 COc1cccc(n1)Cl PS-4836 Cc1ccncc1C#N PS-4837 Cc1cc(ncc1[N+](=O)[O-])Cl PS-4838 c1ccc(cc1)S(=O)(=O)N(C2CC2)C3CCNCC3 PS-4839 c1cc(c(cc1C(=O)O)C(=O)O)Br PS-4840 c1cc(c(cc1Br)N)O PS-4841 CC(=O)c1cc(ccc1Cl)Br PS-4842 c1nc([nH]n1)C(=O)O PS-4843 CC(=O)c1cnn(c1)c2ccccc2 PS-4844 c1cc(sc1c2cc[nH]n2)Br PS-4845 Cc1cc(cnc1)Br PS-4846 c1cc(c(cc1Cl)[N+](=O)[O-])N2CCNCC2 PS-4847 c1c(cc(c(c1C#N)N)Cl)Cl PS-4848 COc1ccc(c(n1)OC)C=O PS-4849 CCCCc1ccco1 PS-4850 COC(=O)Cc1ccccc1Br PS-4851 c1c(sc(n1)N)C#N PS-4852 CC(C)(C)OC(=O)c1ccc(cc1)N PS-4853 COc1c(cc(cn1)Cl)Br PS-4854 Cc1cc(cnc1Br)[N+](=O)[O-] PS-4855 CO/C=N/C(=O)c1ccccc1O PS-4856 c1coc(c1Br)C=O PS-4857 c1c(coc1C=O)Br PS-4858 c1cc(c(cc1O)C=O)Br PS-4859 c1cc(ncc1C=O)Br PS-4860 c1cc2c(ccc(c2nc1)C=O)Br PS-4861 c1c(nc(s1)C=O)Br PS-4862 CC(C)c1[nH]c2ccccc2n1 PS-4863 c1cc(c(c(c1)O)Br)C=O PS-4864 c1nc(nc(n1)Cl)Cl PS-4865 c1ccc(cc1)C(=O)Nc2ccncc2 PS-4866 COc1ccc(cc1)c2ccn(n2)CC(=O)O PS-4867 CC(OC(=O)N[C@H]1CC[C@@H](CC1)O)(C)C PS-4868 COc1cccc(c1)c2cc[nH]n2 PS-4869 CS(=O)(=O)c1ccc(cc1)CCC(=O)O PS-4870 CS(=O)c1ccc(cc1)Br PS-4871 Cc1ccc(c(n1)N)[N+](=O)[O-] PS-4872 CC(=O)Oc1cc(c(cc1OC)C=O)Br PS-4873 c1cc(ncc1C#N)O PS-4874 COC(=O)c1cccnc1Cl PS-4875 c1cc(c(c(c1)Cl)C(=O)O)[N+](=O)[O-] PS-4876 c1cc(c(nc1)I)C#N PS-4877 c1cc(ncc1C(=O)N)Br PS-4878 COc1cccc(c1N)Br PS-4880 CN(C)Cc1ccc(cc1)Br PS-4881 c1cc(c(cc1Br)[N+](=O)[O-])O PS-4882 c1cc(c(cc1Br)C(=O)O)NN PS-4883 c1cc(cc(c1)NN)C#N PS-4884 COc1ccccc1c2cc[nH]n2 PS-4885 c1cnc(c(n1)C#N)Cl PS-4886 c1ccn(c1)c2ccc(cc2)C(=O)O PS-4888 CSc1ccc(cc1)Cl PS-4889 C1CCN(C1)CCCN2CCCNCC2 PS-4890 COc1ccc(cn1)C=O PS-4891 Cc1cccc(c1)C#C PS-4892 COc1ccnc(c1)C(=O)O PS-4893 c1cc(nc(c1Br)C(=O)O)Cl PS-4894 c1cc2cc[nH]c2c(c1)N PS-4895 COC(=O)c1cccc(n1)Br PS-4896 COC(=O)Cc1cccc(c1)Br PS-4897 COC(=O)c1cccnc1I PS-4898 c1cc2ccncc2c(c1)N PS-4899 CCOC(=O)c1cnco1 PS-4900 Cc1c(nco1)C(=O)OC PS-4901 CN(C)S(=O)(=O)c1ccc2c(c1)CCN2 PS-4902 c1c(cnc(n1)Cl)Br PS-4903 COc1ccc(c(c1)OC)[N+](=O)[O-] PS-4904 c1cc2c(c[nH]c2nc1)CC(C(=O)O)N PS-4905 C1CCN(C1)C(=O)C2CCNCC2 PS-4906 COc1ccc(nc1)Br PS-4907 CS(=O)(=O)c1ccc(nc1)Br PS-4908 Cc1c(ccc(n1)Cl)[N+](=O)[O-] PS-4909 c1c(cnc(c1[N+](=O)[O-])Cl)Br PS-4910 c1c(ocn1)C(=O)O PS-4911 Cc1ccccc1c2cc[nH]n2 PS-4912 CSc1cc(cnc1)Br PS-4913 c1cnc(cc1I)C(=O)O PS-4914 c1ccc(cc1)n2cc(cn2)C=O PS-4915 c1cc2c(cc1Br)cc(c(=N)o2)C#N PS-4917 c1cc(c(cc1Br)C(=O)O)N PS-4918 c1cc2c(cc1Br)c(ccn2)O PS-4919 COc1ccc2c(c1)c(ccn2)Cl PS-4920 Cc1cc(nc2c1cc(cc2)O)O PS-4921 Cc1cc(c2cc(ccc2n1)OC)O PS-4922 COc1ccc2c(c1)c(ccn2)N PS-4923 CC(C)(C)OC(=O)N1CCC(C1)C(=O)O PS-4924 c1cc2c(cc[nH]2)nc1 PS-4925 c1c[nH]c2c1ccnc2 PS-4926 CSc1c(cnc(n1)Cl)Br PS-4927 COc1c(cnc(n1)Cl)Br PS-4928 CN(C)c1c(cnc(n1)Cl)Br PS-4929 c1ccc(cc1)c2c(cccn2)N PS-4930 c1cncc(c1O)N PS-4931 c1cnc(nc1Cl)N PS-4932 c1[nH]c2c(nc(nc2n1)Cl)N PS-4933 c1[nH]c2c(n1)nc(nc2I)N PS-4934 c1ccc(cc1)CN2CCC(C2)CN PS-4935 c1cc(ncc1N)C(=O)O PS-4936 c1ccc(cc1)c2c(cccn2)C(=O)O PS-4937 c1cc(sc1C(=O)O)[N+](=O)[O-] PS-4938 c1cc2cnccc2c(c1)N PS-4940 CN(C)Cc1ccccc1Br PS-4941 CN(C)C(=O)c1ccccc1Br PS-4942 CCOC(=O)c1cc(cc(c1)Br)[N+](=O)[O-] PS-4943 C1CC1N2CCC(CC2)N PS-4944 c1ccc(c(c1)CN2CCOCC2)Br PS-4945 c1cc(cc(c1)Br)CN2CCOCC2 PS-4946 c1cc(ccc1CN2CCOCC2)Br PS-4947 CCOC(=O)c1cocn1 PS-4948 c1cc(ncc1Br)NN PS-4949 Cc1cc(c(cc1Br)C)N PS-4950 CNc1ccc(cc1)[N+](=O)[O-] PS-4951 Cn1c2ccccc2c(n1)C=O PS-4952 Cc1c(nc(o1)C)C=O PS-4953 c1cc(cc(c1)C=O)CN2CCOCC2 PS-4954 c1cc(cc(c1)OCCN2CCOCC2)C=O PS-4955 COc1ccc(cn1)O PS-4956 CSc1ncc(c(n1)C(=O)O)Cl PS-4957 c1cc(oc1)c2ccc(cc2)CO PS-4958 c1ccc(c(c1)C#N)Br PS-4959 COC(=O)c1ccc2c(c1)cccn2 PS-4960 c1cc(cc(c1)N)Cn2cncn2 PS-4961 c1cnc(cc1C(=O)O)N2CCOCC2 PS-4962 c1cc(oc1)CCC(=O)O PS-4963 c1c(c(nc(n1)Cl)Cl)[N+](=O)[O-] PS-4964 c1cc2c(cccn2)c(c1)[N+](=O)[O-] PS-4966 c1ccc(c(c1)CC(=O)O)[N+](=O)[O-] PS-4967 COc1ccc(cc1OC)c2cc[nH]n2 PS-4968 CCOc1ccc(cc1)C(=O)/C=C/C(=O)O PS-4969 COc1cc(cc(c1OC)OC)CC=C PS-4970 c1cc(c(c(c1)Cl)Cc2[nH]nnn2)Cl PS-4971 CS(=O)(=O)c1cccc(c1)Br PS-4973 CS(=O)(=O)c1cccc(c1)C=O PS-4974 c1c(cc(c(c1N)N)Cl)Br PS-4975 COc1ccnc(n1)N PS-4976 c1c(csc1C(=O)O)Cl PS-4978 Cc1cnc(cn1)Cl PS-4979 c1cn2cc(ncc2n1)Cl PS-4980 CCOc1cnc(cn1)N PS-4981 c1c(nc(c(n1)C(=O)O)Cl)Cl PS-4982 COc1cncc(n1)Br PS-4983 c1c(nc(c(n1)C#N)N)Cl PS-4984 Cc1cnc(cn1)C=O PS-4985 CC(=O)c1ccc(s1)C=O PS-4986 c1cc2c(c(c1)Br)nco2 PS-4987 CCCc1c(nc(s1)Br)C(=O)OC PS-4988 c1cc2c(cc1Br)[nH]nc2C(=O)O PS-4989 CCOc1ccc(cc1OCC)C#C PS-4990 CCOc1cc(ccc1OC)C#C PS-4991 COc1ccc(cc1OC)C#C PS-4992 c1cc(c2cccnc2c1)N PS-4993 COC(=O)C1(CC1)C(=O)OC PS-4994 Cc1ccc(c(c1)[N+](=O)[O-])OC PS-4995 c1cc2c(cc1Br)nc([nH]2)C(=O)O PS-4996 COc1ccc(c2c1nccc2)C(=O)O PS-4997 Cc1ccc2c(c1Br)cn[nH]2 PS-4998 Cc1cc2c(cn[nH]2)c(c1)Br PS-4999 Cc1ccc(c2c1[nH]nc2)Br PS-5000 Cc1ccc2c(c1Br)cnn2C PS-5001 Cc1ccc(c2c1n(nc2)C)Br PS-5002 Cc1c(ccc2c1cnn2C)Br PS-5003 Cc1cc2c(cc1Br)cnn2C PS-5004 CC(=O)c1ccc(s1)C(=O)O PS-5005 Cc1cc2cnn(c2cc1Br)C PS-5006 c1[nH]c2c(n1)c(nc(n2)N)S PS-5007 COc1ccc(cc1OC)C(=O)c2ccccc2 PS-5008 Cc1c(ccc(n1)Br)N PS-5009 c1cc(nc(c1N)Br)Br PS-5010 Cc1ccc(nc1C)N PS-5011 Cc1c(ncs1)C(=O)O PS-5012 c1ccc2cnc(cc2c1)Br PS-5013 c1cc2cn[nH]c2c(c1)C=O PS-5014 c1c(cnc(n1)Cl)C(=O)O PS-5015 Cc1c[nH]c2c1cc(cc2)Cl PS-5016 c1c(cc(nc1Cl)Cl)O PS-5017 c1ccc2cnc(cc2c1)C=O PS-5018 c1cn2c(n1)CNCC2 PS-5019 COC(=O)c1c(sc(n1)Br)Cl PS-5020 CCc1c(nc(s1)Br)C(=O)OC PS-5021 CCOc1ccc(cc1)C(=O)O PS-5022 CC(C)COc1ccc(cc1N)C(=O)O PS-5023 CCCCOc1ccc(cc1N)C(=O)O PS-5024 CC(C)CCOc1ccc(cc1N)C(=O)O PS-5025 c1cc(nc(c1Cl)CO)Cl PS-5026 c1cc(nc(c1Cl)C(=O)N)Cl PS-5027 c1cc(nc(c1Cl)C=O)Cl PS-5028 COc1ccc(c(n1)CO)Cl PS-5029 COc1ccc(c(n1)C=O)Cl PS-5030 COc1ccc(c(n1)C(=O)N)Cl PS-5031 CNC(=O)c1c(ccc(n1)OC)Cl PS-5032 COc1ccc(c(n1)C(=O)NN)Cl PS-5033 CCOC(=O)c1c(ccc(n1)Cl)Cl PS-5034 Cc1c(c(no1)c2ccccc2)C(C)O PS-5035 COc1cc(cc(c1)Br)C=O PS-5037 COc1cc(cc(c1)Br)N PS-5038 c1cc(c(cc1Cl)CO)[N+](=O)[O-] PS-5039 c1ccc(c(c1)C(=O)N)N PS-5040 c1cnc(cc1CO)N PS-5041 C1C(CC1=O)C(=O)O PS-5042 c1cncc(c1N)C=O PS-5044 COc1ccc(nc1)N PS-5045 CC(=O)Nc1ccc(c(c1)[N+](=O)[O-])N PS-5046 CC(=O)c1cccc(c1)C(=O)OC PS-5047 c1cc(c(c(c1)[N+](=O)[O-])C#N)C#N PS-5048 COC(=O)c1ccccc1Cl PS-5049 CC[C@@H]1CN(CCN1)C(=O)OC(C)(C)C PS-5050 c1csnc1Br PS-5051 c1csnc1C#N PS-5052 c1(c(nc([nH]1)Br)Cl)Cl PS-5053 CSc1cccs1 PS-5054 Cn1cc(c(n1)c2cccc(c2)N)Br PS-5055 c1ccc2c(c1)N(C(=O)CO2)CC#N PS-5056 CC(=C)C(=O)OC12CC3CC(C1)CC(C3)C2 PS-5057 CCCN1CCC(CC1)NC2CC2 PS-5058 COC(=O)CC(=O)c1cccnc1 PS-5059 c1ccc(c(c1)C#N)N2CCOCC2 PS-5060 CCS(=O)(=O)N1CCNCC1 PS-5061 c1c([nH]c(=O)[nH]c1=O)C=O.O PS-5062 CCCCCCN1CCNCC1 PS-5063 c1c([nH]c(=S)[nH]c1=O)CO PS-5064 CC(C)(C)OC(=O)CC(=O)OCc1ccccc1 PS-5065 COCCCCN1CCNCC1 PS-5066 COCCCN1CCNCC1 PS-5067 CN1CCCC(C1)CN2CCNCC2 PS-5068 CN1CCC(CC1)CN2CCNCC2 PS-5069 CN1CCC(CC1)N2CCNCC2 PS-5070 CCCCCN1CCNCC1 PS-5071 CCCC(C)N1CCNCC1 PS-5072 CCC(CC)N1CCNCC1 PS-5073 c1ccc(cc1)CCCCN2CCNCC2 PS-5074 CCOC(=O)CN1CCNCC1 PS-5075 CCOC(=O)C(C)N1CCNCC1 PS-5076 CCOC(=O)C1CCCNC1 PS-5077 CCOC(=O)c1cccnc1C PS-5078 Cc1ccc2nnc(n2n1)Cl PS-5079 Cc1ccc2nncn2n1 PS-5080 c1cc2c(cc1O)CCO2 PS-5081 c1cc2c(cco2)cc1O PS-5082 CC(C)(C)OC(=O)N1CC(C1)C(=O)OC PS-5083 c1ccc2c(c1)CCC[C@@H]2C(=O)O PS-5084 c1cc2cc(ccc2nc1)Cl PS-5085 c1cc(c(c(c1)Cl)C=O)O PS-5086 COC(=O)c1cc2ccsc2[nH]1 PS-5087 CS(=O)(=O)c1cc(ccc1C#N)Br PS-5088 c1cc2cc(ncc2c(c1)Br)O PS-5089 c1cc(cc2c1cc(nc2)O)Br PS-5090 Cc1ccc2cn[nH]c2c1Br PS-5091 CN(C)S(=O)(=O)c1ccc(cc1)c2csc(n2)N PS-5092 c1ccc2c(c1)nc(o2)N PS-5093 Cc1cc(cnc1Cl)N PS-5094 c1c(c(c(nc1Cl)Cl)[N+](=O)[O-])N PS-5095 CC(=O)N1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] PS-5096 COc1ccncc1N PS-5097 c1cc(ncc1O)C#N PS-5098 COc1cc(c(cn1)[N+](=O)[O-])N PS-5099 COC(=O)C1CCC(=O)C1 PS-5100 Cc1cc(cc(c1)Br)N PS-5101 COc1ccc(cc1OC)CCO PS-5102 c1cc(ccc1C=O)c2nnco2 PS-5103 CCc1nnc(o1)c2ccc(cc2)C=O PS-5104 CCCc1nnc(o1)c2ccc(cc2)C=O PS-5105 COC(=O)c1ccc(cc1N)Br PS-5106 Cc1ccc(cc1)SCC(=O)O PS-5107 c1cc2c(cc1Cl)oc(n2)Cl PS-5108 c1cc(c(cc1N)Cl)Cl PS-5109 CC(=O)Oc1cccc(c1)C=O PS-5110 c1cncc(c1N)I PS-5111 c1c(cnc(c1Cl)N)Cl PS-5112 c1cc(nc(c1)O)N PS-5113 Cc1cccnc1Br PS-5114 c1cc(oc1)/C=C/[N+](=O)[O-] PS-5115 c1cc(ncc1Cl)Cl PS-5116 c1ccc(c(c1)C(=O)NCC(=O)O)O PS-5117 c1cc(cc(c1)Br)[N+](=O)[O-] PS-5118 COc1ccc(cc1)Br PS-5119 c1ccc(cc1)/C=N/O PS-5120 c1cc(oc1)c2cc[nH]n2 PS-5121 c1cc(c(cc1N)C(=O)O)Br PS-5122 c1c(nc[nH]1)CCC(=O)O PS-5123 c1c(cc(c(c1Cl)N)Cl)N PS-5124 CC(=O)Nc1ccc(cc1)Cl PS-5125 Cc1ccc(c2c1cn[nH]2)Br PS-5126 Cc1cc2cn[nH]c2c(c1)Br PS-5127 c1c(ncc(n1)Cl)C#N PS-5128 CCOC(=O)c1cnc(nc1)SC PS-5129 Cc1cc(c(s1)Br)C(=O)OC PS-5130 Cc1cc(c(s1)C(=O)OC)Br PS-5131 Cc1ccc(cc1)S PS-5132 c1cc2cnn(c2cc1N)C3CCCCO3 PS-5133 c1cc2c(cc1Br)[nH]nc2Cl PS-5134 Cc1cc(cc2c1n(nc2)C)Br PS-5135 Cn1c2ccc(cc2cn1)Br PS-5136 c1cc2c(cn[nH]2)c(c1)O PS-5137 c1cc2cn[nH]c2cc1O PS-5138 c1ccc(c(c1)CN)n2ccnc2 PS-5139 CC(C)(c1cccc(c1)OC)C(=O)O PS-5140 CNCc1ccc(cc1)N2CCOCC2 PS-5141 Cc1cccc(c1)CC(=O)O PS-5142 c1cc(cc(c1)[N+](=O)[O-])C(=O)O PS-5143 CNCc1cccc(c1)c2cccnc2 PS-5144 CNCc1ccc(cc1)OCCN2CCOCC2 PS-5145 c1cc(cc(c1)N)c2ccncc2 PS-5146 CN1CCN(CC1)c2ccccc2N PS-5147 c1cc(cc(c1)N)c2cccnc2 PS-5148 c1cc(ccc1N)OCCN2CCOCC2 PS-5149 Cc1nc(cs1)c2ccc(cc2)N PS-5150 Cn1c(c2ccccc2n1)C(=O)O PS-5151 Cn1cncc1C(=O)OC PS-5152 CC(C)(C)OC(=O)N1CCCC(=O)CC1 PS-5153 Cc1ccc(c(c1O)Cl)N PS-5155 Cc1nc(no1)c2cccc(c2)C=O PS-5156 c1cc(ccc1C=O)OCCN2CCOCC2 PS-5157 Cn1ccc2c1ccc(c2)Br PS-5158 c1cc2nccn2cc1CO PS-5159 Cc1nc(no1)c2ccc(cc2)CO PS-5160 c1cc(oc1)c2cc(n[nH]2)CO PS-5161 c1cc(sc1)c2cc(n[nH]2)CO PS-5162 CC(C)(C)OC(=O)NCC1CCCCN1 PS-5163 c1cc(c(cc1C#N)N)Cl PS-5164 c1cc2c(ccc(c2N)N)nc1 PS-5165 c1cc(ncc1Br)[N+](=O)[O-] PS-5166 c1cc(c(nc1)Br)C(=O)O PS-5168 CC(=O)N1C=Cc2ccccc2C1CC(=O)O PS-5169 COc1cc(ccc1O)Cl PS-5170 COC(=O)c1ccnc(n1)Cl PS-5171 CCOC(=O)[C@H]1CCCN(C1)C(=O)OC(C)(C)C PS-5172 COc1c(cc(cc1Cl)[N+](=O)[O-])Cl PS-5173 COc1ccc(c(c1)Br)OC PS-5174 COc1cc(c(cc1OC)Br)C(=O)O PS-5175 c1ccc2c(c1)cc(nc2Br)N PS-5177 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccccc2 PS-5178 COc1cccc2c1cc[nH]2 PS-5179 c1ccc(cc1)C2(CCNCC2)O PS-5180 c1ccc(cc1)COC(=O)N2CCC(=O)CC2 PS-5181 CC(=O)n1cc(c2c1ccc(c2)Br)O PS-5183 c1cc(ccc1O)S PS-5184 Cc1cccc(n1)C(=O)CS(=O)(=O)C PS-5185 CC(C)(C)OC(=O)N1CCNC(=O)C1 PS-5186 CC(C)(C)OC(=O)N1CCC[C@@H](C1)O PS-5187 CC(C)(C)OC(=O)N1CCC[C@@H](C1)N PS-5188 CC(C)(C)OC(=O)N1CCC[C@H](C1)N PS-5189 c1ccc2c(c1)N(C(=O)CO2)CC(=O)O PS-5190 c1cnc(nc1C(=O)O)N PS-5191 CC(=O)Oc1ccc2c(c1)cc(cn2)Br PS-5192 c1cc(c(c(c1)Br)C#N)O PS-5193 Cc1ccc(c(n1)C)C=O PS-5194 Cc1ccc(cn1)C=O PS-5195 COc1cc(ccn1)C=O PS-5196 COc1cc(cnc1)O PS-5197 CCOc1ccc(cc1)CO PS-5198 COc1ccc(c(c1)OC)OC PS-5199 c1ccc(cc1)CN2CC[C@H](C2)N PS-5200 CSc1ncc(c(n1)N)C(=O)N PS-5201 CC(C)(C)OC(=O)N1CC[C@@H](C1)N PS-5202 CC(C)(C)OC(=O)N1CC[C@H](C1)N PS-5203 CC(C)(C)OC(=O)N[C@H]1CCNC1 PS-5204 CC(C)(C)OC(=O)N[C@@H]1CCNC1 PS-5205 CCOc1ccc(c(c1)S)OCC PS-5206 c1conc1Br PS-5207 CSc1cccc(c1)Br PS-5208 Cc1cc(cc(n1)C)C(=O)OC PS-5209 COC(=O)c1cc(ncc1N)Cl PS-5210 COc1ccc(cn1)N PS-5211 c1c(cc(c(c1[N+](=O)[O-])N)Br)C#N PS-5212 COc1ccc(c(c1)S)OC PS-5213 CC(C)C(=O)c1ccc(cc1)SC PS-5214 c1ccc(c(c1)N)Sc2ccccc2N PS-5215 CC(=O)c1ccc(cc1)NC(=O)C PS-5216 COC(=O)c1ccc(c(c1)Cl)N PS-5217 COc1cccc(c1N)OC PS-5218 CC(=O)c1ccccc1I PS-5219 COC(=O)c1cc(ccc1N)Br PS-5220 COC(=O)c1cc(ccc1N)I PS-5221 Cc1ccccc1NC(=O)C PS-5222 COC(=O)c1ccc(cc1O)I PS-5223 COc1cc(ccc1C(=O)OC)I PS-5224 c1c(cncc1Br)C=O PS-5225 c1cc(ncc1O)Br PS-5226 Cc1cc(c(c(c1)Br)N)C PS-5227 c1ccc(cc1)C(=O)c2ccccc2N PS-5228 c1(c(nc(nc1Cl)N)Cl)N PS-5229 c1c(cc(nc1C(=O)N)C(=O)N)Br PS-5230 c1cc(nc(c1N)Cl)Br PS-5231 C1CCN(CC1)C/C(=N/O)/N PS-5232 c1cc(nc(c1Br)N)N PS-5233 c1cnc(cc1[N+](=O)[O-])Cl PS-5234 c1cnc(cc1O)C(=O)O PS-5235 c1cc(nnc1N)Cl PS-5236 c1ccn(c1)c2cc(cnc2)C(=O)O PS-5238 CC(C)(C)c1cc(ncn1)N PS-5239 COC(c1ccc2cnccc2n1)OC PS-5240 c1cnc(cc1Br)N PS-5241 c1cc(oc1C(=O)NN)Br PS-5242 Cc1cc(ncc1C(=O)O)C PS-5243 c1ccc2c(c1)c(c(s2)C(=O)O)N PS-5244 COc1cc(cc(c1)Cl)Cl PS-5245 c1cc2c(ccs2)cc1N PS-5246 CCOc1cc(ncc1C(=O)OCC)Cl PS-5247 CCOC(=O)c1c(cc(cn1)Br)N PS-5248 COC(=O)c1cc(cc(n1)Cl)Cl PS-5249 COC(=O)c1cc(c(nc1)Br)Cl PS-5250 COC(=O)c1c(cc(cn1)Cl)Br PS-5251 Cc1cc(nc(c1)C)C PS-5252 c1cc2cn[nH]c2cc1C#N PS-5253 c1cc2cn[nH]c2c(c1)C#N PS-5254 c1cc2ccncc2c(c1)C#N PS-5255 c1ccc2c(c1)cncc2O PS-5256 c1cc2ccncc2c(c1)C(=O)O PS-5257 c1cc2cnccc2cc1C(=O)O PS-5258 c1cc(cc2c1ccnc2)C(=O)O PS-5259 COC(=O)c1c(nccn1)N PS-5260 c1cc(cc(c1)N)CC(=O)O PS-5261 CC(=O)c1cc2c(cc1Br)OCCO2 PS-5262 Cc1ccc(cc1N)C#N PS-5263 c1cc2c(cc1[N+](=O)[O-])cc([nH]2)C(=O)O PS-5264 c1ccc(c(c1)CC#N)C#N PS-5265 COc1cccc(c1)C#N PS-5266 c1ccc(c(c1)c2cnco2)Cl PS-5267 Cc1ccc(cc1[N+](=O)[O-])C#N PS-5268 c1csc(c1N)C(=O)N PS-5269 CC(=O)c1c(cc(cc1O)O)O PS-5270 c1cc(sc1)C(=O)NN PS-5271 COc1ccccc1S PS-5272 CCOc1ccc2c(cc(=O)oc2c1)C PS-5273 c1ccc(c(c1)C(=O)c2ccc(cc2)O)C(=O)O PS-5274 c1ccc(cc1)C(=O)NC(=S)N PS-5275 c1[nH]nc(n1)[N+](=O)[O-] PS-5276 Cc1c(n2cc(ccc2n1)Cl)C(=O)O PS-5277 c1ccc(cc1)c2c(n3cc(ccc3n2)Cl)C(=O)O PS-5278 c1c[nH]c(=O)[nH]c1=O PS-5279 c1cc(cc(c1)Cl)N PS-5280 COc1cc(c(cc1O)Br)CC(=O)O PS-5281 c1cc(ccc1N)Oc2ccc(cc2)N PS-5282 c1cc(ccc1c2ccnc(n2)N)Cl PS-5284 c1cc(cc(c1)I)N PS-5285 c1ccc(cc1)C(CO)C(=O)O PS-5286 CC(=O)c1cccc(c1)OC PS-5287 CC(=O)c1nccs1 PS-5288 CC(C)c1ccc(cc1)N PS-5289 CC(C)(C)c1ccc(cc1)N PS-5290 COc1ccc(cc1OC)N PS-5291 c1cc(ccc1C=O)C#N PS-5292 c1ccc(c(c1)CC#N)Cl PS-5293 c1ccc(c(c1)C=O)[N+](=O)[O-] PS-5294 c1cc(c(cc1C=O)[N+](=O)[O-])Cl PS-5295 CC(C)(C)c1ccc(c(c1)[N+](=O)[O-])N PS-5296 COc1ccc(c(c1OC)OC)C=O PS-5297 c1cc(ccc1C=O)C(=O)O PS-5298 c1ccc(c(c1)C(=O)O)Br PS-5299 CC(=O)N1CCC(CC1)NC2CC2 PS-5300 c1cc(ccc1C(=O)O)Br PS-5301 CC(=O)N/C(=C/c1ccccc1)/C(=O)O PS-5302 c1ccc(c(c1)C#N)[N+](=O)[O-] PS-5303 Cc1c(cc2cccnc2n1)C(=O)O PS-5304 c1cc(c(c(c1)Cl)C(=O)O)Cl PS-5305 c1cc(c(c(c1)Cl)C#N)Cl PS-5306 COc1ccc(cc1)C(=O)c2ccc(cc2)OC PS-5307 c1ccc(c(c1)CO)[N+](=O)[O-] PS-5308 c1cc(ccc1CO)[N+](=O)[O-] PS-5309 c1cc(cc(c1)[N+](=O)[O-])CO PS-5310 c1cc(cc(c1)Cl)CO PS-5311 c1cc(cc(c1)Br)CO PS-5312 c1cc(ccc1CO)Br PS-5313 c1cc(ccc1CO)Cl PS-5314 c1cc(c(cc1Cl)Cl)CO PS-5315 c1ccc(c(c1)CN)Cl PS-5316 c1cc(cc(c1)Cl)CN PS-5317 COc1ccccc1CN PS-5318 CCCC1CCC(=O)CC1 PS-5320 C1CC(=O)CCC1=O PS-5321 CC(=O)c1cccnc1 PS-5322 c1ccc2c(c1)c(c[nH]2)C=O PS-5323 c1cscc1C=O PS-5324 c1cscc1C(=O)O PS-5325 c1cc(sc1)CC(=O)O PS-5326 c1cscc1CC(=O)O PS-5327 c1c(nc(nc1Cl)Cl)Cl PS-5328 Cc1ccc(c(n1)Cl)C(=O)O PS-5329 c1cc(ncc1C(=O)O)Cl PS-5330 c1cc(ncc1C(=O)O)N PS-5331 c1cc(c(nc1)O)C(=O)O PS-5332 c1cc(c(nc1)Cl)C(=O)O PS-5333 CC(CCc1ccccc1)N PS-5334 c1ccc(cc1)CCCN PS-5335 CNc1ccccc1O PS-5336 c1ccc2cnccc2c1 PS-5337 c1cc(ccc1CC(=O)O)CO PS-5338 c1cnc(cc1Cl)N PS-5339 Cc1cccc(c1[N+](=O)[O-])O PS-5340 CC(=O)N1CCN(CC1)c2ccc(cc2)N PS-5341 COc1cc(cc(c1O)Br)CC(=O)O PS-5342 CC(C)(C)N1CCNCC1 PS-5343 C[C@@H]1CNC[C@@H](N1)C PS-5344 c1ccc(cc1)C(c2ccccc2N)O PS-5345 c1cncc(c1O)Cl PS-5346 CCOC(=O)c1ccncc1O PS-5348 c1ccc(c(c1)C(=O)O)Cl PS-5349 CCOC(=O)c1cc(cnc1)O PS-5350 c1c(c(cnc1Br)Cl)O PS-5351 c1c(c(cnc1Cl)O)Cl PS-5352 Cc1ccc(c(n1)Br)O PS-5353 c1cnc(c(c1O)Cl)Cl PS-5354 COc1c(cc(cn1)Br)O PS-5355 CNC(=O)c1ccc(cn1)O PS-5356 c1cc(c(nc1)Cl)Br PS-5357 c1cnoc1C(=O)O PS-5358 COc1cnc(nc1Cl)Cl PS-5359 Cc1nc(cs1)C=O PS-5360 c1ccc(c(c1)C=O)OC2CCOCC2 PS-5361 c1cc(c(cc1Br)N)C#N PS-5362 c1cc(ccc1C=O)OC2CCOCC2 PS-5363 Cc1ccc(cc1)C(=O)OC PS-5364 c1cc(c(c(c1)Br)O)C#N PS-5365 CC(C)(C)OC(=O)NC1CC1C(=O)OC PS-5366 c1cc(nc(c1)N2CCCC2)CN PS-5367 c1cc(cc(c1)C(=O)O)c2nccs2 PS-5368 Cn1c(ccn1)C(=O)O PS-5369 COC(=O)c1ccc(cn1)C#C PS-5370 COC(=O)c1c(cc(cn1)N)Cl PS-5371 COC(=O)c1c(cc(cn1)O)Cl PS-5372 Cc1c(cc2cnccc2n1)C(=O)O PS-5373 c1cc(cc(c1)N)c2cc[nH]n2 PS-5374 c1cc(c(cc1N)Br)[N+](=O)[O-] PS-5375 c1cc(cc(c1)Cl)S PS-5376 c1cc(c(cc1Cl)N)Cl PS-5377 c1ccc2c(c1)c3ccccc3o2 PS-5378 Cc1ccc(c(n1)O)[N+](=O)[O-] PS-5379 Cc1ccc(c(c1C)N)C(=O)O PS-5380 c1ccc(cc1)c2c(n3ccccc3n2)C(=O)O PS-5381 COC(=O)c1cc(cc(c1)Br)[N+](=O)[O-] PS-5382 c1cc2cccnc2c(c1)N PS-5383 C#Cc1ccc(cn1)Cl PS-5384 Cc1cc(cnc1)C#C PS-5385 Cc1cccnc1C#C PS-5386 C#Cc1ccc(nc1)C#N PS-5387 Cc1cc(ccn1)C#C PS-5388 Cc1ccc(nc1)C#C PS-5389 C#Cc1cccc(n1)Cl PS-5390 C#Cc1ccncc1Cl PS-5391 C#Cc1cn2ccnc2cn1 PS-5392 C#Cc1c(nccn1)Cl PS-5393 COc1c(nccn1)C#C PS-5394 COc1cnc(cn1)C#C PS-5395 Cc1cnc(cn1)C#C PS-5396 Cc1c(nccn1)C#C PS-5397 COC(=O)c1cccc(c1)O PS-5398 C#Cc1cccc2n1ccn2 PS-5399 CC(=O)Oc1ccccc1 PS-5400 CC(C)(C)c1cc(c(s1)C(=O)N)N PS-5401 c1cc(cc(c1)Br)C(=O)O PS-5402 Cc1ccc2c(c1)cc([nH]2)C PS-5403 c1c(cncn1)C(=O)O PS-5404 COc1ccccc1C(=O)O PS-5405 c1cc(cc(c1)O)C(=O)O PS-5406 COc1cc(ncn1)N PS-5407 c1cc(ccc1CC#N)Cl PS-5408 COc1cc2cc[nH]c2cc1OC PS-5409 c1ccc(c(c1)O)Br PS-5410 CC(C)(C)OC(=O)N1CCC(CC1)O PS-5411 COc1ccc(c(c1)[N+](=O)[O-])Cl PS-5413 COc1ccc(cc1I)N PS-5414 c1cc(oc1C#N)[N+](=O)[O-] PS-5415 c1cc(ccc1S)Cl PS-5416 Cc1cc(cc(n1)C)C(=O)O PS-5417 c1c(c(cnc1Cl)Cl)O PS-5418 CC(=O)c1c(cccc1Cl)Cl PS-5419 c1cc(cc(c1)[N+](=O)[O-])N2CCOCC2 PS-5420 c1ccc(cc1)COC2CCNC2 PS-5421 Cc1cc(ccc1CO)Br PS-5422 c1ccc2c(c1)c(no2)N3CCNCC3 PS-5423 C1CNCC1N2CCOCC2 PS-5424 Cc1ccccc1C(=O)OC PS-5425 c1ccc(cc1)[C@@H]([C@H](c2ccccc2)N)N PS-5426 c1cc(cc(c1)CO)CO PS-5427 Cc1cc(nc(n1)Sc2ccc(cc2)N)C PS-5428 COc1ccc(c(c1)C=O)Br PS-5429 c1ccc2c(c1)nc3cc(c(cc3n2)N)N PS-5430 c1cc(ccc1N)I PS-5431 c1cnc(nc1Cl)Cl PS-5432 c1cc(ncc1N)Br PS-5433 CS(=O)(=O)c1cccc(c1)C(=O)O PS-5434 COc1cc(nc(n1)c2cccc(c2)N)OC PS-5435 CC(=O)Nc1ccc(cc1Br)C#N PS-5436 c1c[nH]c2c1cncc2 PS-5437 COc1ccc(cc1Br)[N+](=O)[O-] PS-5438 c1cn2ccnc2cc1N PS-5439 CC(C)(C)OC(=O)NC1CCC(=O)CC1 PS-5440 CC1=CC(=O)OC1=O PS-5441 c1cc(c(c(c1O)Cl)[N+](=O)[O-])Cl PS-5442 COc1cc(ccn1)C#N PS-5443 c1cc(ncc1O)C(=O)O PS-5444 Cc1cccc(c1)S PS-5445 c1c(cncc1O)C(=O)O PS-5446 c1cc(c(nc1)[N+](=O)[O-])O PS-5447 c1cnc(cc1Br)C(=O)O PS-5448 Cc1ccnc(c1)NC(=O)C PS-5449 Cc1cc(c(nc1)O)[N+](=O)[O-] PS-5450 c1c(cnc(c1Br)N)[N+](=O)[O-] PS-5451 c1c(cnc(c1Br)Cl)[N+](=O)[O-] PS-5452 c1ccc(c(c1)O)S PS-5453 CC(=O)Nc1cc(ccn1)C(=O)O PS-5454 CC(=O)Nc1ccc(cn1)C(=O)O PS-5455 c1c([nH]cn1)C(=O)O PS-5456 c1c(scn1)C(=O)O PS-5457 CC(=O)c1cnccn1 PS-5458 c1c(ncs1)CO PS-5459 COC(=O)c1cscn1 PS-5460 CCOC(=O)c1c[nH]cn1 PS-5461 CCOC(=O)c1cnc(o1)N PS-5462 COC(=O)c1c(sc(n1)N)Br PS-5463 COc1ccnc(c1)Cl PS-5464 COC(=O)c1ccc2c(c1)NC(=O)C2 PS-5465 C1[C@@H](CC[C@H](C1)O)N PS-5466 COc1ccccc1NC(=S)N PS-5467 Cc1c([nH]c2c1cc(cc2)[N+](=O)[O-])C PS-5468 c1ccnc(c1)CNCc2cccnc2 PS-5469 Cc1ccc(cc1[N+](=O)[O-])C=O PS-5470 c1cc(cc(c1)n2cccn2)CN PS-5471 c1cc(cc(c1)n2cccn2)N PS-5472 c1ccc(cc1)CN2CCC(CC2)C(=O)O PS-5473 CNS(=O)(=O)c1ccc(cc1)Br PS-5474 CN(C)S(=O)(=O)c1ccc(cc1)Br PS-5475 c1cc(ccc1S(=O)(=O)NCCO)Br PS-5476 CCc1cccc(c1)C(=O)C PS-5477 c1cc(ccc1S(=O)(=O)N2CCCC2)Br PS-5478 c1cc(ncc1C#N)Br PS-5479 CC(=O)c1ccccc1Cl PS-5480 c1cnc(cc1Cl)C(=O)N PS-5481 CC(=O)Nc1ccccc1S(=O)(=O)C PS-5482 CC(C)(C)OC(=O)Nc1ccc(nc1)Br PS-5483 c1c(cc(cc1[N+](=O)[O-])Br)C(=O)O PS-5484 c1ccc(c(c1)CO)Cl PS-5485 CN1CCC(CC1)C(=O)O PS-5486 CC(=O)c1ccsc1 PS-5487 CN1CCCC(C1)C(=O)O PS-5488 c1cc(c(cc1Br)[N+](=O)[O-])NN PS-5489 C1CCN(CC1)C(=O)C2CCCNC2 PS-5490 c1cc(nc(c1)Br)Cl PS-5491 c1cc(nc(c1)Cl)N PS-5492 c1ccc(c(c1)C(=O)c2cc(ccc2N)[N+](=O)[O-])Cl PS-5493 COc1c(cccn1)C#N PS-5495 CN(C)C(=O)c1cccnc1S(=O)(=O)N PS-5496 c1cc(c(cc1Cl)Cl)CC(=O)O PS-5497 Cc1c(cccc1N)C(=O)OC PS-5498 c1ccc2c(c1)ccnc2C#N PS-5499 CC(=O)Nc1ccc(nc1)Br PS-5500 c1nnc(s1)Br PS-5501 c1cc(nc(c1[N+](=O)[O-])N)Cl PS-5502 c1cc(c(c(c1)[N+](=O)[O-])N)C(=O)O PS-5503 COc1ccc(c(n1)N)[N+](=O)[O-] PS-5504 Cc1cccc(c1N)N PS-5505 COc1c(cccn1)N PS-5506 CCN(CC)c1ccc(cc1)C PS-5507 COc1cc(cnc1)Br PS-5508 CC(=O)c1cc2cc(ccc2oc1=O)Br PS-5509 Cc1c(c(ncn1)C)C(=O)O PS-5510 CCOC(=O)C1CCC(=O)CC1 PS-5511 C[C@H](c1ccccc1)N PS-5512 CS(=O)(=O)c1ccc(cc1)/C=C/C(=O)O PS-5513 c1cc2cc(c(=O)n3c2c(c1)CC3)C=O PS-5514 c1cc(cnc1)c2cc(=O)oc3c2ccc(c3)O PS-5515 CN1CCC(CC1)CN PS-5516 CCOC(=O)CC(=O)c1ccncc1 PS-5517 CN(C)C1CCCNC1 PS-5518 c1cc(cc(c1)Cl)OCCN PS-5519 c1cc(cc(c1)Cl)OCCCN PS-5520 c1ccc(c(c1)C(=O)N2CCOCC2)N PS-5521 c1ccc(c(c1)CN2CCOCC2)N PS-5522 c1c(cc(c(c1C=O)O)Br)Cl PS-5523 Cc1cc2cc(ccc2[nH]1)N PS-5524 Cc1nnc(o1)c2cccc(c2)Br PS-5525 CNc1cncc(n1)Cl PS-5526 c1cc(ncc1Br)C(=O)N2CCOCC2 PS-5527 Cc1cc(c2ncnn2c1)Br PS-5528 c1cc(cc(c1)Cl)c2c(nco2)C(=O)O PS-5529 CC(=O)n1c2cccc(c2cn1)Cl PS-5530 CC(=O)n1c2cc(ccc2cn1)Cl PS-5531 CCOc1cccc(n1)Br PS-5532 c1cc(c(cc1C=O)O)O PS-5533 COc1ccncc1C(=O)OC PS-5534 c1cc(c(cc1[N+](=O)[O-])N)Br PS-5535 C[C@H]1CNCCN1C(=O)OC(C)(C)C PS-5536 COc1cccc(c1N)C(=O)O PS-5537 Cc1ncc(cn1)Br PS-5538 Cc1cc(ccc1C(=O)O)[N+](=O)[O-] PS-5539 c1ccc2c(c1)ccnc2Br PS-5540 c1c(ncc(n1)Cl)C(=O)O PS-5541 COC(=O)c1cnc(cn1)Cl PS-5542 CC1CCC(=O)CC1 PS-5543 c1c(c(=O)[nH]c(=O)[nH]1)C#N PS-5544 COC1CCNCC1 PS-5545 c1cc2c(ccc(c2nc1)O)[N+](=O)[O-] PS-5547 Cc1ccc(c(c1)N)O PS-5548 Cc1c(non1)CO PS-5549 Cc1cc(cs1)C(=O)O PS-5550 Cc1cc(no1)NC(=S)NC(=O)c2ccccc2 PS-5551 COc1cccc(c1)C#C PS-5552 c1cnc(c(n1)C#N)n2ccnc2 PS-5553 c1cncc(c1C(=O)O)I PS-5554 CSc1nccc(n1)N PS-5555 c1cc(c(c(c1)Cl)CN)Cl PS-5556 c1cc(c2cc[nH]c2c1)C#N PS-5557 c1c(c(cnc1N)Cl)Cl PS-5558 Cc1c(cccn1)C(=O)O PS-5559 Cc1c(nccn1)C(=O)O PS-5560 c1cc(cc(c1)Cl)C#N PS-5561 c1cc(ccc1C(=O)c2ccncc2)Cl PS-5562 CS(=O)(=O)c1ncccn1 PS-5563 COc1cccc(n1)N PS-5564 Cc1nc(co1)CO PS-5565 c1cnc(c2c1sc(c2)Br)Cl PS-5566 c1cc(nc(c1)C=O)CO PS-5567 c1cc(ccc1CC(=O)O)O PS-5568 Cc1ncc(s1)C(=O)O PS-5569 c1cc(sc1)CO PS-5570 CNCc1ccc(cn1)c2ccco2 PS-5571 c1cc(cc(c1)Cl)CC(=O)O PS-5572 COc1ccc(c(c1)N)Br PS-5573 COC(=O)c1ncccn1 PS-5574 c1cc(ncc1Cl)I PS-5575 c1ccc(cc1)c2ccc(nc2)C(=O)O PS-5576 c1cc(oc1)c2ccc(nc2)C(=O)O PS-5577 Cn1c2c(cccc2N)cn1 PS-5578 COc1cc(cc(c1OC)O)C=O PS-5579 Cc1nnc(o1)c2ccc(cc2)C=O PS-5580 CC(C)c1ccc(cc1)CC(=O)O PS-5581 c1cc(nc2c1cncc2)C(=O)O PS-5582 CC(C)(C)OC(=O)N1CCCC(C1)C(=S)N PS-5583 Cc1cccc(c1Cl)[N+](=O)[O-] PS-5584 Cc1cc(c(c(c1)N)O)C PS-5585 Cn1c2ccccc2[nH]c1=O PS-5586 c1c(cc(nc1N)Cl)Cl PS-5587 Cn1c2cccc(c2cn1)Br PS-5589 Cn1cc2c(n1)cccc2Br PS-5590 c1cnc(nc1C(=O)O)Cl PS-5591 c1cc(ccc1CO)I PS-5592 c1cc(nc(c1C#N)Cl)Cl PS-5593 CCOC(=O)c1c(sc(n1)Br)Cl PS-5594 c1cc2cn[nH]c2cc1C(=O)O PS-5595 c1cnc(cc1O)Cl PS-5596 c1cc(ncc1N)O PS-5597 c1cc2cnccc2cc1N PS-5598 c1cc2c(cccc2N)c(c1)N PS-5599 Cc1cc(ncn1)Cl PS-5600 Cc1cccnc1C=O PS-5601 c1cc(c(cc1N)Cl)O PS-5602 C1Cc2nnc(n2C1)CN PS-5603 CSc1ncc(n1Cc2ccccc2)C(=O)O PS-5604 Cc1cc(nc(c1)Cl)Cl PS-5605 Cc1cc(ccc1C=O)Br PS-5606 c1c(c(cnc1Cl)N)N PS-5607 c1c(c(cnc1O)[N+](=O)[O-])Cl PS-5608 COc1cc(ncc1[N+](=O)[O-])Cl PS-5609 c1c(ncc(n1)Br)Cl PS-5610 c1c2c(cnc1Cl)[nH]cn2 PS-5611 c1cnc2cnc(cc2n1)Cl PS-5612 Cc1cc(ncc1C#N)N PS-5613 CNCc1ccc(cc1)CN2CCCC2 PS-5614 CCCC(=O)c1ccccc1 PS-5615 COc1ccc(cc1O)Cl PS-5616 Cc1cncc(c1C#N)C PS-5617 COc1c(cc(cn1)Cl)C#N PS-5618 COc1cc(cnc1Cl)Br PS-5619 Cc1ccc(nc1C(=O)OC)Cl PS-5620 c1c2cn[nH]c2cnc1Br PS-5621 c1ccc2c(c1)cncc2C=O PS-5622 Cc1cc(c(nc1)C#N)N PS-5623 CC(C)(C)OC(=O)N1CC(C1)CNC PS-5624 c1cc2c(cc1N)c(ccn2)Br PS-5625 c1cc2c(ccnc2c(c1)O)Br PS-5626 c1cc(cc(c1)N2C(=O)C=CC2=O)N3C(=O)C=CC3=O PS-5627 c1c(cc(c(c1[N+](=O)[O-])N)Cl)Br PS-5628 Cc1c(nccn1)NN PS-5629 COc1c(nc(cn1)Br)NN PS-5630 c1c(nc(c(n1)NN)Cl)Br PS-5631 Cc1cc(c(nc1)NN)Br PS-5632 Cc1ccnc(c1)NN PS-5633 c1c(ncc(n1)Cl)NN PS-5634 Cc1cc(ncc1Br)NN PS-5635 c1cnc(cc1NN)Cl PS-5636 c1c(nc(cn1)Cl)NN PS-5637 c1cc(ccc1OCC#N)Cl PS-5638 c1cc2c(ccnc2Cl)c(c1)N PS-5639 c1cc2cnccc2cc1O PS-5640 COc1cccc2c1c(=O)oc(=O)[nH]2 PS-5641 CS(=O)(=O)c1ccc(c(c1)N)O PS-5643 Cc1cc(ncc1C#N)Cl PS-5644 c1cc(c2nnnn2c1)Cl PS-5645 CS(=O)(=O)c1ccc(c(c1)N)N PS-5647 c1c[nH]c2c1c(nc(n2)Cl)Cl PS-5648 c1c(cncc1Cl)C=O PS-5649 C1CCC(CC1)(CO)N PS-5650 CCOC1CCC(=O)CC1 PS-5651 c1ccc(cc1)NC(=O)N2CCNCC2 PS-5652 COc1c(nccn1)Cl PS-5653 c1c(ncc(n1)Cl)N PS-5654 c1c(nc(c(n1)O)Br)Br PS-5655 c1cnc(c(n1)NN)Cl PS-5656 c1cnc(cn1)Br PS-5657 COC(=O)c1cc(cc(c1)Cl)[N+](=O)[O-] PS-5658 c1cc(c(c(c1)Br)C=O)O PS-5659 CC(C)(c1ccc(cc1)Cl)N PS-5660 c1cc2c(c(c1)Br)sc(n2)N PS-5661 Cc1cc(nc(c1)N)C PS-5662 Cc1ccc(cc1)C=O PS-5663 c1cnc(c(n1)N)Cl PS-5664 c1cc(c(cc1Br)N)[N+](=O)[O-] PS-5665 c1c(nc(nc1Cl)Cl)N PS-5666 c1cc(c(c(c1)Cl)N)N PS-5667 Cc1ccc(c(c1)N)Br PS-5668 Cn1c(cc(n1)c2ccc(cc2)Cl)N PS-5669 c1ccc(cc1)C(c2ccccc2)N3CC(C3)N PS-5670 COc1ccc(c(c1)Br)N PS-5671 CC(C)(C)OC(=O)N1CC(C1)N PS-5672 Cc1[nH]c2c(n1)cc(cn2)Br PS-5673 CC(C)(C)OC(=O)NC1CNC1 PS-5674 Cc1c(cnc2c1nc([nH]2)C)Br PS-5675 CNc1cccc(c1[N+](=O)[O-])Br PS-5676 c1cc(c(c(c1)Br)[N+](=O)[O-])NC2CC2 PS-5677 CNc1cccc(c1N)Br PS-5678 c1cnc(nc1)c2ccc(cc2)C=O PS-5679 CNc1ccnc(c1[N+](=O)[O-])Br PS-5680 CNc1ccnc(c1N)Br PS-5681 c1cc(cc(c1)c2ncccn2)C=O PS-5682 c1cc(c(c(c1C=O)Cl)Cl)O PS-5683 c1ccc(c(c1)C(=O)CSC#N)O PS-5684 c1cc(c(nc1)Br)C=O PS-5685 Cc1ccnc(c1)C=O PS-5686 CC(C)(C)OC(=O)Nc1cnccc1C=O PS-5688 c1cc(ncc1Br)C=O PS-5689 c1cncc(c1C=O)Br PS-5690 c1ccc(cc1)COC(=O)N2CCCC2C=O PS-5692 Cc1c(c[nH]n1)C=O PS-5693 c1cc2cc(ccc2nc1)C=O PS-5694 c1c(n2c(n1)CCC2)C=O PS-5695 c1cc(ccc1CN)CO PS-5696 c1ccc(c(c1)CN)Br PS-5697 c1cc(ccc1CN)I PS-5698 Cc1ccnc(c1)CN PS-5699 COC(=O)c1c2cc(ccc2[nH]n1)Br PS-5700 COC(=O)c1c2ccc(cc2[nH]n1)Br PS-5701 COc1cc(cnc1Cl)C(=O)O PS-5702 Cc1nc(cs1)CN PS-5703 c1cc2cc[nH]c2c(c1)[N+](=O)[O-] PS-5704 COc1cccc(c1Br)[N+](=O)[O-] PS-5705 c1cnc(nc1)c2ccc(cc2)C(=O)O PS-5706 c1ccc(c(c1)c2ccncc2)C(=O)O PS-5707 c1cc(c(c(c1)[N+](=O)[O-])Br)C(=O)O PS-5708 c1cc(ccc1c2c[nH]cn2)C(=O)O PS-5709 c1ccc(c(c1)CC#N)C(=O)O PS-5710 CN1CCN(CC1)c2ccnc(c2)C(=O)O PS-5711 c1cnc(cc1n2ccnc2)C(=O)O PS-5712 c1cnc(cc1N)C(=O)O PS-5713 Cc1cnoc1C(=O)O PS-5715 c1c(nco1)C(=O)O PS-5716 c1cc(ccc1c2c(nco2)C(=O)O)Cl PS-5717 Cc1c(nco1)C(=O)O PS-5718 CCOC(=O)/C(=C/c1ccc(cc1)N(C)C)/C#N PS-5719 Cc1c(cnc(n1)N)C(=O)O PS-5720 Cc1ncc(cn1)C(=O)O PS-5721 c1c(cnc(n1)N)C(=O)O PS-5722 c1cc(nnc1C(=O)O)N2CCCCC2 PS-5724 Cc1cc(c(=O)[nH]n1)C(=O)O PS-5725 Cc1cc(c(nn1)Cl)C(=O)O PS-5726 c1cc(c(c(c1)Cl)[N+](=O)[O-])N PS-5727 C1CSCC(N1)C(=O)O PS-5728 c1cnccc1N2CC(CC2=O)C(=O)O PS-5729 C1CC(=O)CCC1C(=O)O PS-5730 C1CC1(C(=O)O)C(=O)O PS-5731 c1cc2nc(cn2nc1)C(=O)O PS-5734 c1cc(ccc1C#N)Br PS-5735 CCOC(=O)c1c(nsc1N)C PS-5736 COC(=O)c1cc(cnc1O)Br PS-5737 COC(=O)c1ccc(=O)oc1 PS-5739 Cn1cc(cn1)Br PS-5740 c1cncc(c1N)Cl PS-5741 CSc1nccc(n1)Cl PS-5742 c1c(n2c(n1)CCC2)Br PS-5743 c1cc(nnc1)CO PS-5744 C1CC(=O)CCC1CO PS-5745 Cc1cc(nc(n1)Nc2ccc(cc2)N)C PS-5746 Cc1cccc(n1)Br PS-5747 Cc1ccc(c(n1)C)Br PS-5748 CC(C)c1ccc(cc1)OC PS-5749 Cc1ccncc1Br PS-5750 c1cc(nc(c1)CO)CO PS-5751 c1c(nc(s1)Br)Br PS-5752 c1ccc(c(c1)NN)Cl PS-5753 C1CN2CCC1C(C2)O PS-5754 c1ccc2c(c1)CCN2 PS-5755 CCOC(=O)c1cc2ccccc2oc1=O PS-5756 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)O PS-5757 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)O PS-5758 C1CCCC(CC1)C(=O)O PS-5759 c1cc(ccc1CCC(=O)O)O PS-5760 c1c(c(cc(c1Cl)Cl)[N+](=O)[O-])N PS-5761 c1cc(c(nc1)Cl)N PS-5762 C1CCN(C1)CC#N PS-5763 c1ccc2c(c1)cco2 PS-5764 c1ccc2c(c1)[nH]cn2 PS-5765 c1ccc2c(c1)[nH]c(n2)O PS-5766 Cc1cc(nc(n1)Nc2ccccc2C(=O)O)C PS-5767 Cc1cc(nc(n1)Nc2cccc(c2)C(=O)O)C PS-5768 c1ccc2c(c1)-c3ccccc3C2=O PS-5769 c1ccc2c(c1)CCC2=O PS-5770 COc1ccc2c(c1)CCCC2=O PS-5771 c1cc(sc1)Br PS-5772 c1cscc1Br PS-5773 c1cc(sc1)CCO PS-5774 c1ccc2c(c1)ccs2 PS-5775 COc1cccc(c1)/C=C/C(=O)O PS-5776 COc1ccc(cc1)/C=C/C(=O)O PS-5777 c1cc(ccc1/C=C/C(=O)O)Br PS-5778 c1ccnc(c1)C=CC(=O)O PS-5779 C#Cc1cccc(c1)Cl PS-5780 COc1ccc(cc1)[N+](=O)[O-] PS-5781 CC(=O)c1cccc(c1)NC(=O)C PS-5782 COc1ccc(cc1C#N)Br PS-5783 COc1cc(ccc1Br)[N+](=O)[O-] PS-5784 c1cnc(cc1C#N)N PS-5786 Cc1ccc(c(n1)N)Br PS-5787 COc1cc(ccc1N)C(=O)O PS-5788 c1cc(c(nc1)C#N)Cl PS-5789 C1CCC(C1)CC(=O)O PS-5790 Cc1ccc(cc1[N+](=O)[O-])NC(=O)C PS-5791 Cc1ccc(c(c1)[N+](=O)[O-])N PS-5792 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])Cl PS-5793 c1ccc(cc1)COc2ccccc2N PS-5794 Cc1ccc(c(c1)S)C PS-5796 c1ccc(cc1)CNc2ccccc2N PS-5797 c1ccc(c(c1)C=O)I PS-5798 c1ccc(cc1)COc2ccc(cc2)N PS-5799 Cn1cc(cn1)I PS-5800 COc1c(cnc(n1)OC)Br PS-5801 c1cc(oc1)c2cc(on2)N PS-5802 Cc1cccc(c1C)C=O PS-5803 c1cc(cc(c1)O)C#N PS-5804 Cc1nc(no1)c2ccc(cc2)CNC PS-5805 c1ccc(c(c1)CN)n2cccn2 PS-5806 C1[C@H](CN[C@@H]1C(=O)O)O PS-5807 CC(CN)c1ccccc1 PS-5808 Cc1c(n2ccccc2n1)C=O PS-5809 CCOC(=O)C(=O)c1ccc(s1)Br PS-5810 Cc1nc(cs1)c2ccc(cc2)C(=O)O PS-5811 Cc1c(nc(o1)C)CO PS-5812 c1cc(ccc1CN2CCCCC2)CO PS-5813 c1cc(c(c(c1)Br)O)C=O PS-5814 c1cc(c(c(c1)[N+](=O)[O-])N)N PS-5815 COc1cc(cc(c1OC)OC)Br PS-5816 Cn1ccc2c1ccc(c2)N PS-5817 c1cc(cc(c1)N2CCCC2)N PS-5818 c1cc(sc1)CN PS-5819 COc1cccc(c1)CC(=O)O PS-5820 c1cc2c(cc1CC(=O)O)OCO2 PS-5821 c1cc(c(cc1CC(=O)O)Cl)O PS-5822 c1cnc(cc1Cl)Cl PS-5824 CC(=O)n1cc(c2c1cccc2)C=O PS-5825 CN(C)c1ccccc1C#N PS-5826 C1CC(OC1)C(=O)N2CCNCC2 PS-5827 c1ccc(c(c1)N2CCNCC2)[N+](=O)[O-] PS-5828 c1cc(ccc1N2CCNCC2)[N+](=O)[O-] PS-5829 CCOC(=O)N1CCN(CC1)CCO PS-5830 C1CN(CCN1)CC(=O)N2CCOCC2 PS-5831 C1CCN(C1)C(=O)CN2CCNCC2 PS-5832 C1CCN(C1)CCCN2CCNCC2 PS-5833 C1CCN(CC1)CCCN2CCNCC2 PS-5834 CCCCN1CCNCC1 PS-5835 CCCCCCCN1CCNCC1 PS-5836 COCCN1CCNCC1 PS-5837 CCOCCN1CCNCC1 PS-5838 C=CCN1CCNCC1 PS-5839 CC(C)N1CCNCC1 PS-5840 C1CCCC(CCC1)N2CCNCC2 PS-5841 C1CCC(CC1)CN2CCNCC2 PS-5842 C1CCCC(CC1)N2CCNCC2 PS-5843 CN(C)CCN1CCNCC1 PS-5844 C=CCN(CCN1CCNCC1)CC=C PS-5845 C1CN(CCN1)CCN2CCOCC2 PS-5846 Cc1cc(cc(c1N)[N+](=O)[O-])Cl PS-5847 CCN(CC)CCCN1CCNCC1 PS-5848 CCCN(CCC)CCCN1CCNCC1 PS-5849 C1CNCCC1C(=O)O PS-5850 C1CCNC(C1)C(=O)O PS-5851 CCOC(=O)C1CCN(CC1)Cc2ccccc2 PS-5852 CCOC(=O)C1CCCN(C1)C PS-5853 CCOC(=O)C1CCCN(C1)Cc2ccccc2 PS-5854 CC1(CC(CC(N1)(C)C)N)C PS-5855 CC1(CC(CC(N1)(C)C)O)C PS-5856 COC(=O)c1cccc2c1c(ccc2)O PS-5857 C1CNCCC12OCCO2 PS-5858 C1COC2(CCNCC2)OC1 PS-5859 Cc1ccc(cn1)Br PS-5860 CS(=O)(=O)c1ccccc1Cl PS-5861 CS(=O)(=O)c1ccccc1Br PS-5862 Cc1cc(c(cc1N)[N+](=O)[O-])C PS-5863 COC(=O)c1ccc(c(c1)C=O)O PS-5864 c1cc(c(c(c1)Cl)O)C=O PS-5865 CCc1cc(ccc1NC(=O)C)C#N PS-5866 c1ccc(c(c1)c2ccc(cc2)C(=O)O)S(=O)(=O)N PS-5867 c1c(csc1Br)C=O PS-5868 c1cc(ccc1C2CC2)O PS-5869 CS(=O)(=O)c1cc(ccc1N)Br PS-5870 COc1ccc(cc1/C=C/C(=O)O)Br PS-5871 c1cc(ccc1C(=O)CC#N)O PS-5872 c1c(cc(c(c1[N+](=O)[O-])N)Br)Cl PS-5873 CCN(CC)C(=O)c1ccc(c(c1)OC)Br PS-5874 Cc1cc(nc(c1N)Br)C PS-5875 Cc1ccnc(c1N)C PS-5876 Cc1cc(ncc1N)C PS-5877 C1CCC2C(C1)C2C(=O)O PS-5878 Cc1ccc2c(c1Br)C(=O)C(=O)N2 PS-5879 C1CCC(C1)N2CCC2C(=O)O PS-5880 c1cc(sc1C=O)C(=O)O PS-5881 Cc1c(con1)C(=O)O PS-5882 c1ccc(cc1)C2CC(=O)C2 PS-5883 c1ncn(n1)CC(=O)O PS-5884 c1ncn(n1)CCC(=O)O PS-5885 Cc1ccc(cc1Br)N PS-5886 CC(OC(=O)N[C@H]1CC[C@@H](CC1)N)(C)C PS-5887 COc1cc(cc(c1OC)OC)N PS-5888 c1c(cc(c(c1Br)N)Br)C#N PS-5889 Cc1ccsc1C PS-5890 CC(C)CC1CC(=O)CC(=O)C1 PS-5891 CCCC(=O)c1cc(c(cc1O)O)O PS-5892 c1ccc2c(c1)cccc2N3C(=O)C=CC3=O PS-5893 CC(=O)c1ccc(cc1)c2ccc(cc2)C(=O)O PS-5894 C=Cc1ccc(cc1)C(=O)O PS-5895 c1cc(cc(c1)Cl)c2ccc(o2)C(=O)O PS-5896 c1ccc(c(c1)C#CCO)Cl PS-5897 c1cc(cc(c1)Cl)C#CCO PS-5898 c1ccc(c(c1)C=O)c2ccco2 PS-5899 c1cc(cc(c1)c2ccco2)C=O PS-5900 c1ccc(c(c1)c2ccco2)C(=O)O PS-5901 c1cc(cc(c1)C(=O)O)c2ccco2 PS-5902 Cn1cnc2c1cc(cc2)Br PS-5903 c1ccc(c(c1)C#CCO)C#N PS-5904 CS(=O)(=O)c1ccc(cc1)C#N PS-5905 CC(=O)N1CCc2c1ccc(c2)N PS-5906 CC(=O)c1ccccc1c2ccc(cc2)OC PS-5907 CC(=O)c1ccc(cc1)c2cccc(c2)OC PS-5908 COc1cccc(c1)c2ccc(o2)C(=O)O PS-5909 c1cc2c(cc1C(=O)O)nns2 PS-5910 C=CCc1cccc(c1O)C=O PS-5911 Cc1ccc(o1)c2ccc(cc2)C=O PS-5912 c1c(c(=O)c(c[nH]1)Cl)Cl PS-5913 C#Cc1ccccc1Cl PS-5914 c1cc(c(nc1)C#N)O PS-5915 Cc1ccc(o1)c2ccc(cc2)C(=O)O PS-5916 c1cc(cc2c1cc(cc2)C(=O)O)C(=O)O PS-5917 COC(=O)c1cccc(c1)C#CCO PS-5918 COC(=O)c1ccc(cc1)C#CCO PS-5919 CC(C)(C)c1cc([nH]n1)N PS-5920 c1cc(cc(c1)C(=O)O)c2ccsc2 PS-5921 c1ccc2c(c1)c(cc(=O)[nH]2)CC(C(=O)O)N PS-5922 c1c(cnc(n1)N2CCN(CC2)CCO)Br PS-5923 c1cc(ccc1CN)O PS-5924 c1cc(cc2c1cc[nH]2)O PS-5925 CC(C)(C)c1c(c2ccccc2[nH]1)C=O PS-5926 c1cc(c(cc1C#N)Br)N PS-5927 Cc1c(c2ccccc2n1C)C=O PS-5928 C#Cc1ccc(cc1)Cl PS-5929 CC(=O)Nc1ccccc1Cl PS-5930 c1cc(cc(c1)Cl)c2cnco2 PS-5931 CNCc1ccc(cc1)N PS-5932 CNc1cccc(c1)CN PS-5933 CS(=O)(=O)c1ccc(c(c1)N)C(=O)O PS-5934 CN(C)CCCc1ccc(cc1)N PS-5935 Cn1cc(c(n1)N)Br PS-5936 CN1CCC(CC1)NC2CCN(CC2)C PS-5937 CS(=O)(=O)c1cc(cc(c1)S(=O)(=O)C)N PS-5938 CN1CCCC(C1)CO PS-5939 c1c(cnc(n1)N2CCCNCC2)Br PS-5940 CCc1ccc(cc1)C(=O)OC PS-5941 CC(C)(C)OC(=O)N1CCC(CC1)NC2CC2 PS-5942 CC(C)(C)OC(=O)Nc1cccc(c1)CN PS-5943 CC(C)(C)c1cc2cc(ccc2[nH]1)N PS-5944 CC(C)(C)c1cc2cc(ccc2[nH]1)NC3CCNCC3 PS-5945 Cc1cc(c(cc1S(=O)(=O)C)N2CCNCC2)Cl PS-5946 CN(C)Cc1cc(ccc1Br)O PS-5947 c1cc(c2c(c1)non2)N PS-5948 Cc1cc(c(cc1N)S(=O)(=O)C)C PS-5949 Cc1ccc(c(c1N)C)S(=O)(=O)C PS-5950 CN(C)c1ccc(cn1)Br PS-5951 Cc1ccc(cc1N)O PS-5952 Cc1csc(n1)N PS-5953 Cc1ccc(cc1C(=O)O)[N+](=O)[O-] PS-5954 Cc1ccc(cc1C#N)[N+](=O)[O-] PS-5955 c1cc(c(c(c1)N)O)C(=O)O PS-5956 Cc1ccc(cc1[N+](=O)[O-])N PS-5957 CC(=O)c1ccc(cc1)I PS-5958 c1cc(ccc1C(=O)O)NN PS-5959 c1cc(nc(c1)Br)N PS-5960 CN(C)S(=O)(=O)c1ccccc1Br PS-5961 c1cc(ccc1S(=O)(=O)CC#N)Br PS-5962 CC(=O)C(=O)c1ccc(cc1)Cl PS-5963 CC(C)Oc1ccccc1CN PS-5964 CC(c1ccc(cc1)S(=O)(=O)C)NCCOC PS-5965 CS(=O)(=O)c1ccc(c(c1)[N+](=O)[O-])N PS-5967 c1c(con1)Br PS-5968 COc1ncc(c(n1)SC)Br PS-5969 c1ccc(cc1)c2nnc(o2)C3CCNCC3 PS-5970 c1cc(sc1)c2nc(on2)C3CCNCC3 PS-5971 CS(=O)(=O)c1cc(ccc1C(=O)O)Br PS-5972 c1cc(nc2c1cncc2Br)C(=O)O PS-5973 c1c(cnc(n1)N2CCCC(C2)C(=O)O)Br PS-5974 CC(C)(C)OC(=O)Nc1cccc(c1)CCC(=O)O PS-5975 CC(C)(C)OC(=O)c1cccc(c1)C(=O)O PS-5976 CC(C)(C)OC(=O)c1ccc(cc1)C(=O)O PS-5977 CS(=O)(=O)c1cc(ccc1C(=O)O)Cl PS-5978 CN1CCN(CC1)c2ccc(cn2)Br PS-5979 c1ccc(cc1)COC(=O)NN PS-5980 Cc1cc(nc(n1)N2CCC(CC2)C(=O)O)C PS-5981 c1cc2c(cc[nH]2)c(c1)[N+](=O)[O-] PS-5982 CS(=O)(=O)c1cccc(c1)CC(=O)O PS-5983 c1cc2cc(c(=O)n3c2c(c1)CCC3)C(=O)O PS-5984 C1CN(CCNC1=O)C(=O)CCC(=O)O PS-5985 COc1cc(nc(n1)c2ccc(cc2)N)OC PS-5986 c1cnncc1C(=O)O PS-5987 c1c(ncs1)C(=O)O PS-5988 c1ccc(c(c1)N)Br PS-5989 c1c(cnc(n1)NN)Br PS-5990 COc1ccc(cc1)c2cnc(nc2)Cl PS-5991 COC(=O)C1=CCc2c1cccc2 PS-5992 CS(=O)(=O)c1ccc(c(c1)Br)NN PS-5993 c1cc(cc2c1cc[nH]2)C(=O)N3CCNCC3 PS-5994 CS(=O)(=O)c1ccc(cc1)C=O PS-5995 c1cc(nn2c1nc(c2)C(=O)O)Cl PS-5996 c1cc(c(nc1)N2CCC(CC2)C#N)[N+](=O)[O-] PS-5997 COc1cccc(c1CN2CCC(=O)CC2)OC PS-5998 C1CCC(=O)C(C1)C#N PS-5999 Cc1ccc(c(c1)C)S PS-6000 c1ccc(cc1)C(=O)Cc2cnccn2 PS-6001 CS(=O)(=O)c1cc(ccc1C=O)Br PS-6002 Cc1cc(ccc1N)[N+](=O)[O-] PS-6003 c1cc(c(cc1Cl)Cl)C=O PS-6004 Cc1c(cccc1[N+](=O)[O-])C(=O)O PS-6005 c1cc(c(c(c1)Cl)C=O)Cl PS-6006 Cc1cc(c(cc1S(=O)(=O)C)Cl)Cl PS-6007 CC(=O)Oc1ccc(cc1)C(=O)O PS-6008 Cc1c(cc(c(c1[N+](=O)[O-])Cl)Cl)S(=O)(=O)C PS-6009 CNc1ccc(cc1[N+](=O)[O-])S(=O)(=O)C PS-6010 CS(=O)(=O)c1cccc(c1)C#N PS-6011 Cc1ccc(n1C)CN PS-6012 Cc1csc(c1c2nc3ccccc3s2)N PS-6013 c1ccc2c(c1)ncn2Cc3ccc(cc3)C(=O)O PS-6014 c1ccc2c(c1)c(on2)C(=O)O PS-6015 c1ccc2c(c1)cc(s2)C=O PS-6016 CC(C)(C)OC(=O)NC1(CC1)C(=O)O PS-6017 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)O PS-6018 CC(C)(C)OC(=O)[N@]1CSC[C@H]1C(=O)O PS-6019 Cc1ccsc1Br PS-6020 CC(C)(C)OC(=O)N1CCC(CC1)CN PS-6021 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)N PS-6022 c1cc(ccc1c2cncnc2N)Cl PS-6023 c1cc2c(ccnc2cc1Cl)SCC(=O)NN PS-6024 CCOc1cc(c(cc1N2CCOCC2)OCC)N PS-6025 CCOC(=O)C1CCN(CC1)Cc2cccc(c2)N PS-6026 CCOC(=O)CCc1ccc(cc1)O PS-6027 Cc1c(c(n(n1)C)C)N PS-6028 c1ccc2c(c1)C[C@H](NC2)CO PS-6029 c1cc(oc1C=O)I PS-6030 c1cc(nc(c1Cl)C(=O)O)Cl PS-6031 Cc1ccc(o1)c2cccc(c2)N PS-6032 c1cc(cnc1)NC(=O)CCC(=O)O PS-6033 c1c(nns1)C=O PS-6034 COC(=O)c1cccc(c1N)[N+](=O)[O-] PS-6035 c1cc(c(cc1C(=O)O)[N+](=O)[O-])Br PS-6036 COC(=O)c1ccc(c(c1)[N+](=O)[O-])Br PS-6037 c1ccnc(c1)c2c3ccccn3nn2 PS-6038 Cc1cn(nn1)Cc2ccccc2 PS-6039 c1cc(cc(c1)I)C=O PS-6040 COc1ccc(c(c1)OC)I PS-6041 c1cc(cc(c1)Cl)O PS-6042 c1cc(c(cc1[N+](=O)[O-])C#N)C#N PS-6043 COc1ccc(c(c1)C(=O)O)N PS-6044 CC(=O)c1cccc(c1Cl)Cl PS-6045 Cc1c(ncnc1Cl)Cl PS-6046 c1c(ncnc1Cl)N PS-6047 c1ccc(cc1)COc2cccc(c2)N PS-6048 COc1ccc2c(ccnc2c1)O PS-6049 Cc1cccc2c1nc[nH]c2=O PS-6050 c1cc2c(cc1Cl)sc(=S)[nH]2 PS-6051 c1cc2c(cc1[N+](=O)[O-])CCN2 PS-6052 CCCOC(=O)c1ccc(cc1)N PS-6053 CCC(C)N1CCNCC1 PS-6054 c1c(nc(s1)Cl)C=O PS-6055 c1c(nc(s1)Cl)CO PS-6056 c1c[nH]c2c1cnc(n2)Cl PS-6057 c1c(sc(n1)Br)Br PS-6058 C1CSCCC1N PS-6059 c1ccc(cc1)c2ncccn2 PS-6060 c1cncc(c1Cl)N PS-6061 COc1c(cc(cn1)[N+](=O)[O-])Br PS-6062 Cc1c(ccc(n1)Br)[N+](=O)[O-] PS-6063 c1c(cc(cc1Cl)Cl)C=O PS-6064 C1CC[C@H]([C@@H](C1)O)O PS-6065 Cc1c(nc(nc1O)c2ccccn2)C PS-6066 C1CCc2c(c(nc(n2)N)O)C1 PS-6067 CN1CCN(CC1)c2ncc(cn2)Br PS-6068 Cc1nc(cs1)Br PS-6069 CSc1ncc(cn1)Br PS-6070 c1cc(cc(c1)Br)N2CCOCC2 PS-6071 c1c(cnc(n1)N2CCOCC2)Br PS-6072 CCOC(=O)COc1ccc(cc1)Br PS-6073 COc1c(cnc(n1)N2CCNCC2)Br PS-6074 c1cc(ncc1Br)N2CCNCC2 PS-6075 Cn1ccc2c1cccc2OC PS-6076 c1c(ncs1)Br PS-6077 c1c(csc1C2OCCO2)Br PS-6078 c1cc2ccncc2c(c1)Cl PS-6079 c1c(cc(cc1N)Cl)C#N PS-6080 COc1c(cccn1)Cl PS-6081 c1cc2ccncc2c(c1)O PS-6082 COc1ccc2ccncc2c1 PS-6083 COc1cccc2c1cncc2 PS-6084 Cc1ccc2cnccc2c1 PS-6085 Cc1cc(c(nc1)OC)[N+](=O)[O-] PS-6086 c1c[nH]c(=O)c(c1O)C#N PS-6087 C1CC(CNC1)C(=O)O PS-6088 c1cc(ccc1CCC(=O)O)[N+](=O)[O-] PS-6089 c1cc(ncc1Br)N2CCOCC2 PS-6090 c1c(cnc(=O)[nH]1)Br PS-6091 c1c(cnc(n1)N2CCCC2)Br PS-6092 c1cc(ncc1Br)N2CCCC2 PS-6093 c1cc2c(cccn2)c(c1)Br PS-6094 c1cc(c(nc1)N)C#N PS-6095 c1c(cnc(c1[N+](=O)[O-])N)Cl PS-6096 Cc1cc(cc(n1)Cl)C(=O)OC PS-6097 c1c(cncc1Br)O PS-6098 CC(=O)CSc1ccccc1 PS-6099 COc1cccc(c1)CN PS-6100 COc1ccc(c(c1)O)C(=O)OC PS-6101 Cc1nc(c(s1)C=O)c2ccccc2 PS-6102 c1cnc(cc1C=O)N2CCCC2 PS-6103 c1cc(cc(c1)C=O)CN2CCCC2 PS-6104 CN1CCCN(CC1)c2ccc(cc2)C=O PS-6105 Cn1ccc2c1cccc2CN PS-6106 c1ccc(cc1)OCc2ccccc2CN PS-6107 COC(=O)CC(=O)c1cc(cnc1)Br PS-6108 COc1cc(c(cc1OC)OC)C=O PS-6109 Cc1cccc(c1C=O)C PS-6110 CC(C)[C@H]1COC(=O)N1 PS-6111 c1ccc(cc1)[C@H](CO)N PS-6112 c1ccc(cc1)C[C@H]2COC(=O)N2 PS-6113 Cc1cc(c(c(n1)C)[N+](=O)[O-])Cl PS-6114 c1c(c(nc(n1)Cl)Cl)Cl PS-6115 CCC(=O)c1cccc(c1)Cl PS-6116 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)N PS-6117 CCOC(=O)N1CCC(CC1)O PS-6118 CCN(CC)c1ccc(cc1)C=O PS-6119 CC(=O)c1ccc(c(c1O)OC)OC PS-6120 c1ccc(cc1)c2cccc(c2)CN PS-6121 Cc1cccc(n1)Cl PS-6122 c1cncc(c1Cl)Cl PS-6123 COc1ccc(nc1)C#N PS-6124 c1cc(c(nc1)Br)Cl PS-6125 CCC(=O)c1ccc(cc1)OC PS-6126 c1cc2c(ccc(=O)o2)cc1C=O PS-6127 c1cc(c(cc1[N+](=O)[O-])N)C(=O)O PS-6128 COc1cccnc1N PS-6129 c1cnc(cc1C=O)Br PS-6130 CCCN1CCC(=O)CC1 PS-6131 COc1ccc(cc1CO)Br PS-6132 COc1cc(ccc1O)O PS-6133 c1cc(ccc1CN)C#N PS-6134 c1cc(c(cc1N)[N+](=O)[O-])[N+](=O)[O-] PS-6135 CC(=O)c1cccc(c1)Oc2ccccc2 PS-6136 C1[C@H](CN[C@H]1C(=O)O)O PS-6137 C1CC(=O)N[C@@H]1C(=O)O PS-6138 C1C[C@H](CNC1)C(=O)O PS-6139 c1cc(cc(c1)N)CCC(=O)O PS-6140 CCN(CC)c1ccccc1 PS-6141 c1cc(ncc1O)Cl PS-6142 c1c(cnc(c1C(=O)O)C#N)Br PS-6143 c1c(cnc(c1[N+](=O)[O-])O)Cl PS-6144 c1cc(ccc1CO)N PS-6145 Cc1ccnc(c1)C#N PS-6146 Cc1ccnc(c1O)C PS-6147 Cc1cc(ncc1[N+](=O)[O-])C PS-6148 c1c(c(c(cn1)Br)N)Br PS-6149 COc1cccnc1[N+](=O)[O-] PS-6150 COc1c(cccn1)C(=O)O PS-6151 Cc1cncc(n1)N2CCNCC2 PS-6152 CC1CC(=O)CCN1C(=O)OC(C)(C)C PS-6153 c1ccc(cc1)COC(=O)N2CCC(CC2)O PS-6154 CC(C)C1CC(=O)CCN1C(=O)OC(C)(C)C PS-6155 CC(C)(C)OC(=O)N1CCC(=C)CC1 PS-6156 C1COCCN1c2c(nsn2)O PS-6157 CC1CC(=O)CC(O1)C PS-6158 CC(C)(C)OC(=O)N1CC(C1)O PS-6159 CC(C)(C)OC(=O)N1CC(=O)C1 PS-6160 c1cc(ccc1C#N)N PS-6161 Cc1ccn2c(c1)nc(c2C(=O)O)c3ccccc3 PS-6162 c1cc(cc(c1)[N+](=O)[O-])c2cc[nH]n2 PS-6163 C1CNCCNC1=O PS-6164 Cc1c(nc(o1)C)CN PS-6165 CNCc1cc(nn1C)c2ccccc2 PS-6166 c1cc(cc(c1)C=O)Cn2ccnc2 PS-6167 c1cc(ccc1Cn2ccnc2)C=O PS-6168 Cn1ccc2c1ccc(c2)C=O PS-6169 Cn1c(cc(n1)c2ccccc2)C=O PS-6170 c1cc(cc(c1)CO)Cn2cncn2 PS-6171 Cn1c(cc(n1)c2ccccc2)CO PS-6172 c1c(cc(nc1Cl)Cl)CN PS-6173 Cc1cc(ccn1)Br PS-6174 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)C=O PS-6175 C#Cc1ccc2c(c1)nccn2 PS-6176 C#Cc1ccc(cc1)c2cnco2 PS-6177 Cn1c(cc(n1)c2ccccc2)CN PS-6178 CNCC1CCN(CC1)C(=O)OCc2ccccc2 PS-6179 c1cnc2c(n1)c(cs2)N PS-6180 c1cc(nc(c1)N2CCOCC2)C=O PS-6181 c1cc(cc(c1)n2cncn2)C=O PS-6182 c1cc(cc(c1)C=O)Cn2cncn2 PS-6183 Cn1c(cc(n1)C=O)c2ccco2 PS-6184 Cn1c(cc(n1)CO)c2ccco2 PS-6185 CSc1cccc(c1)C(=O)O PS-6186 c1cc(c(cc1C=O)[N+](=O)[O-])O PS-6187 c1cc(cc(c1)c2ccco2)CN PS-6188 Cn1c(cc(n1)c2cccs2)C=O PS-6189 c1cc(nc(c1)N2CCOCC2)C(=O)O PS-6190 Cc1ccc(c(c1)C)OCC(=O)NN PS-6191 COC(=O)c1ccc(c(c1)[N+](=O)[O-])Cl PS-6192 c1csc(n1)Cl PS-6193 c1ccc(c(c1)CO)c2ccco2 PS-6194 c1cc(c(cc1C(=O)O)Br)C(=O)O PS-6195 C1COCCN1c2n[nH]nn2 PS-6196 COc1cc(c(cc1OC)N)C#N PS-6197 c1ccc2c(c1)CCN2CCC(=O)O PS-6198 COc1c(cccc1Cl)N PS-6199 C1COCCC1C=O PS-6200 C1COCCC1C(=O)N PS-6201 Cc1cc(cc(c1N)C)Br PS-6202 c1c(sc(n1)N)C(=O)O PS-6203 COc1ccc(cc1S(=O)(=O)N)Br PS-6204 Cc1cc(=O)oc2c1ccc(c2)N PS-6205 C1CCN(CC1)c2[nH]nnn2 PS-6206 Cc1ccccc1OC PS-6207 c1ccc(cc1)c2ccn(n2)CC(=O)O PS-6208 c1ccnc(c1)Cl PS-6209 c1ccnc(c1)S PS-6210 CCS(=O)(=O)c1ccc2c(c1)NC(=O)CO2 PS-6211 COc1c(cc(cn1)Br)C(=O)O PS-6212 CC(=O)Nc1cc(cnc1)C(=O)O PS-6213 Cc1ccc(c(n1)C)[N+](=O)[O-] PS-6214 C1C2CC3(CC1CC(C2)(C3)O)N PS-6215 CS(=O)(=O)c1cccc(c1)S(=O)(=O)C PS-6216 Cn1c(nnc1S)c2ccncc2 PS-6217 Cc1ccc(c(n1)C)N PS-6218 c1cc(ccc1C[C@@H](C(=O)O)N)I PS-6219 CC(=O)NNc1ccncc1[N+](=O)[O-] PS-6221 Cc1c(n2ccccc2n1)C(=O)NN PS-6222 CCOc1cc(ccc1NC(=O)C)[N+](=O)[O-] PS-6223 c1(nc(sn1)Cl)Br PS-6224 COC(=O)c1ccc(nc1)O PS-6225 COC(=O)c1ccnc(c1)Br PS-6226 COC(=O)c1ccc(nc1)Br PS-6227 COC(=O)c1cc(ccn1)I PS-6228 COC(=O)c1cc(ccn1)Br PS-6229 c1c(cncc1Br)Cl PS-6230 COc1ccc2c(c1)nc([nH]2)S PS-6231 c1cc(c(cc1O)C(=O)O)O PS-6232 c1cnccc1c2[nH]nnn2 PS-6233 c1ccc2c(c1)c(c[nH]2)CC(=O)NN PS-6234 CCOc1ccccc1Br PS-6235 CC(=O)c1cc(ccc1Br)OC PS-6236 Cc1cc(cc(c1)OC)C PS-6237 CC(C)Oc1ccc(cc1)C(=O)O PS-6238 Cc1ccc2nc(c(n2c1)C(=O)O)c3ccccc3 PS-6239 c1ccc2c(c1)c(nc(n2)c3ccncc3)O PS-6240 Cn1ccc2c1cc(cc2)Br PS-6241 CN(C)CCOc1ccccc1C=O PS-6242 Cn1c2ccccc2nc(c1=O)CCC(=O)O PS-6243 c1ccc(c(c1)C=O)N2CCCC2 PS-6244 CN1CCN(CC1)c2cccc(c2)N PS-6245 Cc1nc(no1)c2ccc(cc2)N PS-6246 Cc1nnc(s1)S PS-6247 Cc1cc(no1)C=O PS-6248 c1cc(c(cc1Cl)Cl)N PS-6249 Cc1cc(sc1)CN PS-6250 CSc1cccc(c1)Cl PS-6251 COc1ccccc1SC PS-6252 CCS(=O)(=O)c1ccccc1 PS-6253 c1cc(c(cc1[N+](=O)[O-])C=O)O PS-6254 c1cc(cc(c1)n2ccnc2)C(=O)O PS-6255 CC(C)(C)OC(=O)NCc1cccc(c1)C=O PS-6256 c1cc(c(c(c1)Br)[N+](=O)[O-])O PS-6257 c1cc(c(c(c1)Br)O)[N+](=O)[O-] PS-6258 c1cc(c(c(c1)Br)N)O PS-6259 c1cc(c(c(c1)Br)O)N PS-6260 c1cnc(cc1Br)Cl PS-6261 c1cc(c(cc1C#N)Cl)N PS-6262 COC(=O)c1ccc(c(c1)Br)N PS-6263 c1cc(c(cc1C(=O)O)I)O PS-6264 Cc1ccnc(c1N)Cl PS-6265 c1ccnc(c1)C(C=O)C=O PS-6266 CC(=O)C(=O)c1ccc(cc1)[N+](=O)[O-] PS-6267 Cc1cncc(n1)Cl PS-6268 Cc1ccc2cc(ccc2n1)C=O PS-6269 c1cnc(cc1C=O)N2CCOCC2 PS-6270 Cc1ccc(s1)C(=O)C PS-6271 c1cc(ccc1N)Cl PS-6272 CC(C)(C)OC(=O)N1CCC(CC1)N PS-6274 c1cc(c(cc1C#N)O)O PS-6276 c1cc(cc(c1)NN)C(=O)O PS-6277 Cc1nc(cc(n1)O)c2ccccc2 PS-6278 c1ccc(cc1)S(=O)(=O)c2ccccc2N PS-6279 c1cc(c(cc1Cl)O)N PS-6280 c1ccc(c(c1)[N+](=O)[O-])Br PS-6281 CCOC(=O)c1c(c([nH]c1C)C=O)C PS-6285 CCOC(=O)c1c(c(c([nH]1)C)C(=O)OC(C)(C)C)C PS-6287 COc1ccc(c(c1)C=O)OC PS-6288 Cc1cccc(n1)OC PS-6289 Cc1cccc(c1N)C(=O)O PS-6290 COc1ccnc(c1OC)CO PS-6291 c1cc2c(cc1[N+](=O)[O-])C(=O)CCO2 PS-6292 Cc1c(cccc1[N+](=O)[O-])N PS-6293 c1cc(c(cc1[N+](=O)[O-])O)Cl PS-6294 c1c(cc(c(c1Cl)N)Cl)Cl PS-6295 c1c(c(nc(n1)Cl)Cl)Br PS-6296 Cc1cc(nc(n1)SC)I PS-6297 Cc1ccc(c(c1)C(=O)O)[N+](=O)[O-] PS-6298 COc1cc2c(cc1OC)ncnc2Cl PS-6299 Cc1ccccc1S PS-6300 c1ccc(cc1)c2cnco2 PS-6301 COC(=O)CN1c2ccccc2SCC1=O PS-6302 c1cc(c(cc1/C=C/C(=O)O)Cl)F PS-6304 c1cc(c(cc1C(C(=O)O)N)Cl)F PS-6305 c1cc2c(cc1C(F)(F)F)nc([nH]2)C(=O)O PS-6306 c1cc(c(cc1C(F)(F)F)CC(=O)O)Cl PS-6307 c1cc(ccc1c2nnc(o2)C3CCNCC3)F PS-6308 c1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)O PS-6309 COc1ccnn2c1nnc2c3ccc(cc3)C(F)(F)F PS-6310 COc1ccc(cc1C(=O)O)F PS-6311 c1ccc(cc1)CN2CCC(C2)NC(=O)C(F)(F)F PS-6317 c1cc(c(cc1F)[N+](=O)[O-])N2CCCC2 PS-6318 COc1c(cc(cc1F)C(=O)O)F PS-6320 CCOC(=O)c1cnn(c1C(F)(F)F)C PS-6321 c1cc(ccc1/C=C/C(=O)N)C(F)(F)F PS-6322 Cc1cc(ccc1F)c2csc(n2)N PS-6323 C[C@H](c1cccc(c1)C(F)(F)F)O PS-6325 CC(=O)c1cc(ccc1O)OC(F)(F)F PS-6327 Cc1ccc2ccc(cc2n1)F PS-6328 CCOC(=O)C1CCC(CC1)(F)F PS-6331 C1COC(=O)C1C(F)(F)F PS-6333 COc1c(cccc1F)C(=O)O PS-6334 c1cc2c(cc1/C=C/C(=O)O)OC(O2)(F)F PS-6335 COc1cccc(c1CC#N)F PS-6336 c1c(cnc(c1Cl)N2CCCNCC2)C(F)(F)F PS-6338 CC(C)(C)C(=O)Nc1ccc(c(c1C(=O)O)F)F PS-6339 c1ccc(c(c1)C(=O)O)Nc2ccccc2F PS-6341 CS(=O)(=O)c1ccc(c(c1)F)N2CCCNCC2 PS-6342 c1cc(ncc1/C=C/C(=O)O)C(F)(F)F PS-6344 CCOC(=O)c1cc2cccnc2nc1C(F)(F)F PS-6349 c1cnc(cc1C(F)(F)F)S PS-6367 c1cc(sc1)C(=O)C(F)(F)F PS-6370 c1cc(c(nc1)Cl)C(F)(F)F PS-6371 CC(C)(C)OC(=O)c1c2ccc(nc2[nH]n1)F PS-6372 c1c(cnc(c1F)C(=O)O)F PS-6373 c1c(cnc(c1Br)C(=O)O)F PS-6376 c1c(cnc(c1F)Cl)C#N PS-6377 c1c(cnc(c1F)Cl)C(=O)O PS-6378 Cc1cc(ncc1C(=O)O)F PS-6379 Cc1ccc(c(n1)C(=O)O)F PS-6380 c1cc2c(cc1S(=O)(=O)C(F)(F)F)nc[nH]2 PS-6381 c1c(cnc(c1Cl)N)C(F)(F)F PS-6382 c1cc(c(nc1)Oc2ccc(cc2F)F)N PS-6384 c1cc(c(cc1c2csc(n2)N)F)F PS-6385 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCCN PS-6386 c1ccc(c(c1)Oc2c(cccn2)N)F PS-6387 c1c(cncc1Br)C(F)(F)F PS-6390 CNc1c(cc(cn1)C(F)(F)F)N PS-6391 c1cc2c(cc(=O)oc2cc1N)C(F)(F)F PS-6393 c1cc(c(cc1C(F)(F)F)N)N2CCCC2 PS-6394 c1ccc(c(c1)c2ccc(o2)C(=O)O)F PS-6398 c1cc(cc(c1)F)c2ccc(o2)C(=O)O PS-6399 c1cc(cc(c1)F)C#CCO PS-6400 COc1ccc(c(c1C(=O)O)F)F PS-6401 CS(=O)(=O)c1cc(cc2c1[nH]c(c2)C(=O)O)F PS-6402 CS(=O)(=O)c1cc(ccc1N2CCNCC2)F PS-6403 CS(=O)(=O)c1ccc(cc1C(=O)O)F PS-6404 c1cc(ccc1c2cc(c(s2)C(=O)N)N)F PS-6405 COc1ccc(c(c1F)C(=O)O)F PS-6406 c1cc(cc(c1)OC(F)(F)F)CN2CCNCC2 PS-6407 c1c(c(nc(n1)Cl)N)F PS-6408 C1Cn2c(nnc2C(F)(F)F)CN1 PS-6410 c1cc(nc(c1)F)C(F)(F)F PS-6412 c1ccc(c(c1)OCCC(=O)O)F PS-6413 c1[nH]c2c(n1)c(nc(n2)F)N PS-6414 Cc1cc(c(nc1)Cl)F PS-6415 c1ccc(c(c1)CN2CCNCC2)OC(F)(F)F PS-6416 c1cc(ccc1CN2CCNCC2)OC(F)(F)F PS-6417 c1cc(c(cc1Br)F)/C=C/C(=O)O PS-6418 COc1ccc(cc1C#N)F PS-6422 c1cc(ccc1Nc2ncnc(n2)N)F PS-6423 CC(=O)Nc1ccc(cc1Br)C(F)(F)F PS-6424 CC(=O)Nc1ccc(c(c1)C(F)(F)F)Br PS-6425 c1c(cc(c2c1[nH]cn2)Br)C(F)(F)F PS-6426 CC(=O)C(=O)c1cccc(c1)C(F)(F)F PS-6428 c1cc2c(cc1C(F)(F)F)CC(=O)N2 PS-6431 c1c2c(cc(c1Cl)F)nc[nH]2 PS-6434 c1cc(c(c(c1)Cl)CSCCN)F PS-6435 c1cc(c(cc1Cl)F)/C=C/C(=O)O PS-6436 c1cc(nc(c1C(=O)O)O)C(F)(F)F PS-6437 CC(=O)/C=C/c1ccc(cc1)C(F)(F)F PS-6438 c1c2c(cc(=O)oc2cc(c1Cl)O)C(F)(F)F PS-6439 COc1c(cc(cn1)C(F)(F)F)Cl PS-6441 c1c(cnc(c1F)N)Cl PS-6442 Cc1c(c(n(n1)C(=O)C)C(F)(F)F)[N+](=O)[O-] PS-6443 c1cc2c(cc1C(=O)CC(=O)C(F)(F)F)OCO2 PS-6444 c1cc(cc(c1)F)CCC(=O)O PS-6446 Cc1c(c(n[nH]1)C(F)(F)F)Cl PS-6447 c1c(cncc1Cl)C(F)(F)F PS-6449 c1ccc2c(c1)c(ccc2F)C#N PS-6453 c1cc(ccc1c2cc(nc(n2)N)N)F PS-6456 c1c2c(cc(c1OC(F)F)OC(F)F)sc(n2)N PS-6457 c1cc(nc(c1C(=O)O)Cl)C(F)(F)F PS-6458 c1cc(c(c2c1[nH]cn2)F)F PS-6459 c1ccc(cc1)c2nc(c(o2)C(F)(F)F)C(=O)O PS-6460 c1ccc(cc1)CN2CCC(CC2)(F)F PS-6461 COc1cc(c(c(c1)F)C(=O)O)F PS-6462 Cc1c(c(nn1C)C(F)(F)F)Br PS-6463 c1cnc(cc1C(F)(F)F)Cl PS-6464 c1cc(ccc1C(F)(F)F)SCC(=O)O PS-6465 CS(=O)(=O)c1cc(ccc1F)C#N PS-6468 CS(=O)(=O)c1cc(ccc1F)C(=O)O PS-6469 c1cc(c(c(c1)F)F)/C=C/C(=O)O PS-6471 c1cc(c(cc1F)F)/C=C/C(=O)O PS-6472 c1cc(c(cc1F)/C=C/C(=O)O)F PS-6473 c1cc(c(c(c1)F)/C=C/C(=O)O)F PS-6474 c1cc(c(cc1/C=C/C(=O)O)F)F PS-6475 c1c(cc(cc1F)F)/C=C/C(=O)O PS-6476 c1cc(c(cc1CO)F)C(=O)O PS-6478 CCC(=O)c1cc(c(c(c1)F)O)F PS-6479 c1cc(c(cc1F)F)C(C(=O)O)O PS-6481 c1c(cc(cc1F)F)C(C(=O)O)O PS-6482 c1cc2c(cccc2F)c(c1)C(=O)O PS-6483 c1cc(c(c(c1)F)F)CC(C(=O)O)N PS-6484 c1cc(c(cc1F)F)CC(C(=O)O)N PS-6485 c1cc(c(cc1CC(C(=O)O)N)F)F PS-6486 c1c(cc(cc1F)F)CC(C(=O)O)N PS-6487 c1cc(c2c(c1)[nH]cn2)C(F)(F)F PS-6488 c1c(cc2c(c1C(F)(F)F)nc[nH]2)Br PS-6489 c1cc2c(cc1C(F)(F)F)NC(=O)CS2 PS-6490 Cc1c(ccc(n1)C(F)(F)F)C(=O)N PS-6491 c1cc2c(cc1C(F)(F)F)NC(=O)CO2 PS-6493 CC1C(=O)Nc2cc(ccc2O1)C(F)(F)F PS-6494 c1cc2c(cc1C(F)(F)F)nco2 PS-6495 Cc1nc2cc(ccc2o1)C(F)(F)F PS-6496 Cc1c[nH]c2c1cc(cc2)F PS-6498 Cc1c(ccc(n1)C(F)(F)F)C(=O)OC PS-6500 c1cc(c(cc1Br)F)CN2CCCNCC2 PS-6501 Cc1cc(c(o1)C(F)(F)F)CN PS-6502 c1c(cc(c2c1COCO2)CO)F PS-6504 c1cc(ccc1C(Cc2cnccn2)O)C(F)(F)F PS-6505 CC(=O)Nc1ccc(cc1)OC(F)F PS-6506 CCOC(=O)c1cnc(=O)[nH]c1C(F)(F)F PS-6509 CCOC(=O)c1cnc(nc1C(F)(F)F)Cl PS-6510 c1cc2cccnc2c(c1)F PS-6513 c1cc(ncc1C(=O)O)OCC(F)(F)F PS-6514 CN(C)c1c(cc(cn1)N)C(F)(F)F PS-6515 CCOC(=O)c1cnn(c1C)c2ccc(cc2F)F PS-6516 c1cc2c(cc1C(F)(F)F)nsn2 PS-6517 C1(=O)C(SC(=N1)N)(C(F)(F)F)F PS-6518 c1cc(ccc1N)S(=O)(=O)Nc2ccc(cc2F)F PS-6519 c1cc(cc(c1)N2CC(CC2=O)C(=O)O)C(F)(F)F PS-6520 c1cc(ccc1c2n[nH]nn2)C(F)(F)F PS-6521 c1cnc(cc1C(F)(F)F)Br PS-6522 c1c(cn2cc(nc2c1Cl)C(=O)O)C(F)(F)F PS-6525 c1cc2c(cc1F)sc(n2)S PS-6527 CCOC(=O)Cc1c(cccc1F)F PS-6528 c1cc(c(cc1F)Cl)CC(=S)N PS-6529 c1ccc2c(c1)nc(o2)C(F)(F)Br PS-6530 c1ccn2c(c1)ncc2C(=O)C(F)(F)Cl PS-6531 CCOC(=O)C(c1ccccn1)(F)F PS-6533 COC(=O)/C=C/c1cccc(c1)F PS-6535 CC(=O)c1cc(c(c(c1)F)OC)F PS-6536 CCOC(=O)Cc1ccccc1C(F)(F)F PS-6537 COC(=O)c1cnccc1C(F)(F)F PS-6540 CC(=O)/C=C/c1cccc(c1)C(F)(F)F PS-6541 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)O PS-6543 c1cc2ccncc2c(c1)F PS-6546 c1cc(c(cc1F)[N+](=O)[O-])N2CCCCC2 PS-6547 c1cc(c(c2c1[nH]cc2)F)O PS-6549 c1cc(ccc1F)S(=O)(=O)CC#N PS-6550 c1cc(c(nc1)OCC(F)(F)F)C#N PS-6552 c1cc\2c(c(c1)F)NC(=O)/C2=N\O PS-6553 c1cc2c(cc1F)c(c(cn2)C(=O)O)O PS-6554 c1cc(c(c(c1C#N)F)F)O PS-6557 COc1cc(cc(c1)C(F)(F)F)C(=O)O PS-6558 c1c(c(n[nH]1)C(F)(F)F)Br PS-6559 CCOC(=O)C(=O)c1ccc(cc1)F PS-6560 c1cc(cc(c1)F)/C=C/C(=O)O PS-6565 c1cc(ccc1/C=C/C(=O)O)F PS-6566 c1cc(ccc1c2[nH]c3ccc(cc3n2)C(=O)O)F PS-6567 c1cc(c(cc1F)[N+](=O)[O-])N2CCOCC2 PS-6571 c1cc(cc(c1)F)c2[nH]nnn2 PS-6573 COc1ccc(cc1F)C#N PS-6574 COc1ccc(cc1F)CO PS-6575 c1c(cc2c(c1F)nc(s2)N)F PS-6577 c1cc(ccc1C(C(=O)O)O)F PS-6578 CSc1ccc(cc1F)C(=O)N PS-6580 c1ccc(c(c1)c2[nH]nnn2)F PS-6583 c1cc(cc(c1)S(=O)(=O)N)OC(F)(F)F PS-6586 C1CC1(C(=O)O)C(F)(F)F PS-6587 CN(C)c1ccncc1C(=O)C(F)(F)F PS-6588 c1cc(ccc1C(=O)N)SC(F)(F)F PS-6589 c1cc(ccc1OCC(=O)NN)F PS-6592 CCc1cc(c(cc1F)O)OC PS-6594 c1cc(ccc1OCCC(=O)O)F PS-6597 c1cc(c(cc1F)C(C(=O)O)O)F PS-6598 c1cc(c(c(c1)F)C(C(=O)O)O)F PS-6599 c1cc(cc(c1)F)CC(C(=O)O)N PS-6600 c1cc(sc1)C(=O)c2ccc(cc2)F PS-6602 c1cc(c(c(c1)F)C(=O)O)C(=O)O PS-6605 c1cc2c(cc1F)C(=O)OC2=O PS-6606 c1cc2c(cc1F)c(=O)c(co2)C(=O)O PS-6609 c1cc(c(cc1C(=O)C#N)Cl)F PS-6610 c1cc(cc(c1)NC(=O)N)C(F)(F)F PS-6612 c1cc2c(cc1C(=O)O)OC(O2)(F)F PS-6613 c1cc(ncc1C(F)(F)F)F PS-6614 c1cc2c(cc1F)c(c[nH]2)CC(C(=O)O)N PS-6615 c1cc(c(c(c1)F)CC(C(=O)O)N)F PS-6617 c1cc(ccc1c2[nH]nnn2)F PS-6618 CC(=O)c1cc(c(cc1F)O)OC PS-6620 c1cc2c(cc1F)c(ccn2)Cl PS-6622 CS(=O)(=O)CC(=O)c1cccc(c1)F PS-6623 c1ccc2c(c1)cc(c(=O)o2)C(=O)C(F)(F)F PS-6629 COc1cc(ccc1C#N)C(F)(F)F PS-6630 COc1cc(ccc1C(=O)O)C(F)(F)F PS-6631 C1CCNC(C1)CC(C(=O)O)C(F)(F)F PS-6635 c1cc2c(c(c1)F)NCCC2=O PS-6636 COc1ccc(cc1)c2cc(n[nH]2)C(F)(F)F PS-6637 c1c(c(cnc1Cl)F)N PS-6639 COc1ccc(c(c1)C(F)(F)F)C(=O)OC PS-6640 CCOC(=O)c1cc(cnc1Cl)F PS-6641 c1c(cc(cc1C(F)(F)F)O)C#N PS-6642 COC(=O)C(=O)c1ccc(c(c1)F)F PS-6643 COc1ccc(cc1)c2cc(n[nH]2)C(F)F PS-6644 c1c(cnc(c1[N+](=O)[O-])O)C(F)(F)F PS-6646 c1c(cnc(c1C(F)(F)F)O)[N+](=O)[O-] PS-6647 c1cc2c(cc1C(F)(F)F)c(c(cn2)C(=O)O)O PS-6651 c1c(cnc(c1Cl)C#N)F PS-6653 c1c(cnc(c1Cl)C(=O)O)F PS-6654 Cc1cn2cc(cc2c(=O)[nH]1)C(F)(F)F PS-6655 c1cc2cc(cc(c2nc1)F)Br PS-6656 COC(=O)c1c(cc(cn1)F)Cl PS-6657 c1cc2c(cccn2)c(c1)F PS-6658 C#Cc1ccc(nc1)C(F)(F)F PS-6660 C#Cc1ccc(cn1)C(F)(F)F PS-6661 c1c(cnc(c1Br)C#N)F PS-6662 c1c(cc(c2c1[nH]cn2)Br)F PS-6663 c1c(cnc(c1C(F)(F)F)NN)Br PS-6664 Cn1c(cc(n1)c2ccc(s2)C(=O)O)C(F)(F)F PS-6665 c1cc(sc1C(F)F)Br PS-6666 c1csc(c1Br)C(F)F PS-6667 c1cnc(cc1CN)C(F)(F)F PS-6668 c1cnc(cc1C#N)C(F)(F)F PS-6669 c1cnc(c(c1C(=O)O)F)F PS-6673 COC(=O)c1cc(ncc1C(F)(F)F)Cl PS-6674 COc1cccc(c1C#N)OCC(F)(F)F PS-6676 CO[C@@](c1ccccc1)(C(=O)O)C(F)(F)F PS-6677 COC(=O)c1c(cc(s1)c2ccc(cc2)F)N PS-6680 Cn1c2cc(c(cc2cn1)F)Br PS-6683 Cn1cc2cc(c(cc2n1)Br)F PS-6684 c1c2cnn(c2cc(c1F)Br)C3CCCCO3 PS-6685 c1cnc(c(c1CO)F)Cl PS-6686 c1cnc(c(c1O)F)Cl PS-6687 c1cc2c(cc1C(F)(F)F)NCCO2 PS-6688 COC(=O)CC(=O)c1cccc(c1)C(F)(F)F PS-6691 c1cc(c(cc1OC(F)(F)F)C(=O)O)O PS-6692 c1cc(c(cc1C(=O)CCC(=O)O)Cl)F PS-6693 CC(=O)Nc1ccc(cc1[N+](=O)[O-])OC(F)(F)F PS-6694 c1cncc2c1nc(c(c2)C(=O)O)C(F)(F)F PS-6695 Cc1nc(c(o1)C(F)(F)F)C(=O)O PS-6696 c1cc(c(cc1F)F)C(C(=O)O)N PS-6697 Cc1cc(c(o1)C(F)(F)F)C(=O)N PS-6698 c1cc(cc(c1)C(F)(F)F)CCC(=O)O PS-6700 c1cc(c(c(c1)Cl)/C=C/C(=O)O)F PS-6701 c1cc(nc(c1C#N)Cl)C(F)(F)F PS-6702 c1cc(cc(c1)C(F)(F)F)c2[nH]nnn2 PS-6703 c1c(cnc(c1F)N)C(F)(F)F PS-6704 c1c(cc(c2c1C(=O)CC2)F)F PS-6706 c1c(c(cnc1F)N)C(=O)O PS-6707 c1cc(c(cc1F)F)OCCC(=O)O PS-6709 c1cc2c(cc1F)c(n[nH]2)Br PS-6710 c1cc2c(cc1F)[nH]nc2Br PS-6711 Cc1cc(cc(n1)NN)C(F)(F)F PS-6713 c1cnc(nc1C(F)(F)F)N2CCC(CC2)C(=O)N PS-6714 c1cc(nc(c1N)Cl)C(F)(F)F PS-6715 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCNCC2 PS-6716 c1ccc(c(c1)c2csc(n2)N)F PS-6718 c1cc(c(cc1F)F)c2csc(n2)N PS-6720 c1cc(nnc1C(F)(F)F)Cl PS-6722 Cn1c2cccc(c2c(n1)N)F PS-6723 Cn1c2ccc(cc2c(n1)N)F PS-6724 c1cc2c(cc1OC(F)(F)F)cn[nH]2 PS-6725 COC(=O)c1cc(ncc1F)Cl PS-6726 COC(=O)c1cc(ncc1F)Br PS-6727 COC(=O)c1c(cc(cn1)F)F PS-6728 COC(=O)c1c(cc(cn1)F)Br PS-6729 COC(=O)c1c(cc(cn1)Br)F PS-6730 COC(=O)c1cc(c(nc1)Cl)F PS-6731 CS(=O)(=O)c1ccc(cc1C#N)C(F)(F)F PS-6732 c1cc(c(cc1F)/C=C/C(=O)O)Br PS-6734 c1cn(cn1)C(=O)C(C(F)(F)F)(F)F PS-6735 c1ccc(c(c1)CC(=O)C2CC2)F PS-6736 c1c(nc(s1)C(=O)O)C(F)(F)F PS-6737 c1cc(nc(c1C(=O)N)Cl)C(F)(F)F PS-6739 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCNCC3 PS-6740 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCCNCC3 PS-6741 c1cc(c(cc1C#N)C(=O)O)F PS-6742 c1cc(c(cc1C(=O)O)F)C#N PS-6743 C#Cc1cccc(c1)OC(F)F PS-6744 c1cc2cc(c(nc2nc1)C(F)(F)F)C(=O)O PS-6745 c1c(cnc(c1F)C#N)Cl PS-6748 c1c(cnc(c1F)C#N)Br PS-6749 CS(=O)(=O)c1ccc(cc1F)C#N PS-6750 c1c(cnc(c1F)C(=O)O)Cl PS-6751 c1c(cnc(c1F)C(=O)O)Br PS-6752 c1c(cnc(c1F)Br)Br PS-6753 c1cc(c(cc1C(=O)O)C#N)F PS-6754 CC(=O)Nc1ccc(cc1Cl)OC(F)(F)F PS-6758 CS(=O)(=O)c1ccc(cc1C(F)(F)F)C#N PS-6759 c1cc2c(cc1F)C(=O)CO2 PS-6761 c1cc2c(cc1F)OCC2=O PS-6762 c1cc2cc(ccc2cc1C#N)F PS-6764 COc1cc(ccc1F)/C=N/O PS-6769 c1cnc(nc1C(F)(F)F)NN PS-6771 c1cc(ncc1C(F)(F)F)c2[nH]nnn2 PS-6772 CCOC(=O)Cc1cccc(c1)C(F)(F)F PS-6773 c1cc(cc2c1cc(cc2)F)C(=O)O PS-6775 c1cc(cc(c1)C(F)(F)F)c2nc(nc(n2)N)N PS-6776 c1cc(ccc1c2nc(nc(n2)N)N)C(F)(F)F PS-6777 c1ccc2c(c1)OC(O2)(F)F PS-6778 c1cc(ncc1/C(=N\O)/N)C(F)(F)F PS-6779 CN(C(=O)c1ccc(cc1)F)N PS-6782 CC(C)(C)OC(=O)N1C[C@H](C[C@H]1C(=O)O)F PS-6783 c1cc(ccc1n2c(c(cn2)C(=O)O)N)F PS-6784 c1cc(ccc1c2nnc(n2N)S)F PS-6785 c1cc(c2cc[nH]c2c1F)Br PS-6787 c1cc(c(cc1F)[N+](=O)[O-])N2CCNCC2 PS-6788 c1cc(sc1)C(=O)CC(=O)C(F)(F)F PS-6790 c1cc2c(cc1OC(F)(F)F)CC(=O)N2 PS-6792 Cc1cc(c2cccc(c2n1)F)O PS-6793 Cc1cc(c2ccc(cc2n1)C(F)(F)F)N PS-6794 c1cc(ccc1C(=O)C(F)(F)F)C(=O)O PS-6795 CN(c1c(cccn1)C(F)(F)F)N PS-6796 c1cc(c(cc1F)C(C(=O)O)N)F PS-6797 c1c2c(cc(c1F)Cl)n(cc(c2=O)C(=O)O)C3CC3 PS-6798 c1c(cc(c2c1[nH]cn2)F)F PS-6799 c1cn(cn1)C(=O)C(F)(F)F PS-6800 C1COCCN1C(=O)C(F)(F)F PS-6801 c1cc2c(ccnc2c(c1)F)Cl PS-6802 c1cc(oc1)C(=O)CC(=O)C(F)(F)F PS-6803 CC(=O)Nc1ccc(cc1C(F)(F)F)Br PS-6804 c1cc(ccc1C(=O)N)OC(F)(F)F PS-6806 c1ccc(c(c1)C(=O)NN)OC(F)(F)F PS-6807 CS(=O)(=O)c1ccc(cc1C(=O)O)C(F)(F)F PS-6809 c1cc(ccc1/C(=N/O)/N)C(F)(F)F PS-6811 CS(=O)(=O)c1ccc(cc1F)C(=O)O PS-6814 Cc1cc2cc(ccc2[nH]1)F PS-6821 c1cc(c(cc1F)F)Nc2ncnc(n2)N PS-6823 c1cc(cc(c1)C(F)(F)F)/C=C/C(=O)O PS-6824 c1cc(ccc1C=CC(=O)O)C(F)(F)F PS-6825 C1CC(CCC1C(=O)O)C(F)(F)F PS-6826 C1CC(CC(=O)C1)C(F)(F)F PS-6827 C1CC(=O)CCC1C(F)(F)F PS-6828 C1=C(C(=O)OC1=O)C(F)(F)F PS-6829 c1cc(ccc1CC(=O)O)OC(F)F PS-6831 c1cncc(c1C(F)(F)F)Br PS-6833 COc1ccc(cc1CC(=O)O)F PS-6836 C1C(=NNC1=O)C(F)(F)F PS-6838 c1cncc(c1C(F)(F)F)C(=S)N PS-6839 c1cc(c2c(c1F)C(=O)OC2=O)F PS-6842 c1c[nH]c2c1cc(c(c2)F)F PS-6843 c1c[nH]c2c1c(cc(c2)F)F PS-6844 c1cnoc1c2cc(cc(c2)F)F PS-6845 c1cnc(nc1C(F)(F)F)S PS-6846 CN(C)Cc1cc(ccc1O)F PS-6848 c1cc(c(cc1F)C(=O)O)C(=O)O PS-6851 c1[nH]c2c(n1)c(nc(n2)F)Cl PS-6852 c1c(cnc(c1Br)O)C(F)(F)F PS-6854 COC(=O)Cc1ccc(cc1[N+](=O)[O-])C(F)(F)F PS-6855 COc1ccc(nc1)C(F)(F)F PS-6858 c1cc(c(cc1C=CC(=O)O)F)Cl PS-6862 c1cc(ccc1C(F)(F)F)OCC(=O)O PS-6863 c1csc2c1nc(c(c2)C(=O)O)C(F)(F)F PS-6865 COc1cc(c(c(c1)F)C#N)F PS-6866 c1c(cc(c(c1F)C(=O)O)F)O PS-6867 c1cc(ccc1CSCCN)F PS-6869 CC(C)n1c2ccc(cc2nc1C(F)(F)F)C(=O)O PS-6882 c1cc2c(c(c1)F)[nH]c(=O)oc2=O PS-6888 c1cc(c(cc1F)CO)C#N PS-6890 COc1ccc(cc1C(=O)O)OC(F)(F)F PS-6891 c1cc(c(c(c1)Cl)CN2CCCNCC2)F PS-6894 c1cc(c2ncc(n2c1)Br)F PS-6895 c1cc(ccc1C2CCCN2)F PS-6897 c1cc(ccc1C2CCCN2)C(F)(F)F PS-6898 c1cc2c(cc1F)c(cc(n2)C(F)(F)F)N3CCNCC3 PS-6900 COC(=O)c1ccnc(n1)C(F)(F)F PS-6901 c1cc(c(cc1F)F)C2CC2C(=O)O PS-6902 c1cc(nc(c1C(F)(F)F)C(=O)O)Cl PS-6906 c1c(c(cnc1Cl)C(F)(F)F)C(=O)O PS-6907 Cc1cc(nn1C(=O)C)C(F)(F)F PS-6910 c1c(cnc(c1C(=O)O)Cl)F PS-6915 c1c(cnc(c1C(=O)O)Cl)C(F)(F)F PS-6917 c1cc(c(nc1)C(F)(F)F)C#N PS-6919 c1cc(nc(c1C(=O)O)F)F PS-6921 c1cc(c(cc1Br)F)C2CC2C(=O)O PS-6922 c1cc(ccc1CN2CCN(CC2)CCO)F PS-6926 c1cc(c(cc1F)F)c2nc(cs2)C(=O)N PS-6933 c1cc2c(cc1F)[nH]cc2CC(C(=O)O)N PS-6938 COC(C#N)(c1ccccc1)C(F)(F)F PS-6941 COc1cc(cc(c1)C(F)(F)F)C#N PS-6942 c1c[nH]c2c1cc(c(c2)Cl)F PS-6948 c1(c(nc([nH]1)Br)Br)C(F)(F)F PS-6950 c1cc(ccc1N)Oc2ccc(cc2)F PS-6951 c1cnc(nc1C(F)(F)F)N2CCC(CC2)C(=O)O PS-6952 c1cc2c(cc1OC(F)F)nc([nH]2)S PS-6955 C1CC(C1)(C(=O)O)C(F)(F)F PS-6956 Cc1cc(ccc1NC(=O)C)OC(F)(F)F PS-6958 c1cc(c(nc1)F)C(F)(F)F PS-6960 CC(=O)c1ccc(c2c1cccc2)F PS-6961 c1cc2c(ccnc2c(c1)C(F)(F)F)S PS-6962 c1cc(c(cc1F)F)c2ccno2 PS-6963 c1cc(c(c(c1)F)c2ccno2)F PS-6965 CS(=O)(=O)CC(=O)c1ccc(nc1)C(F)(F)F PS-6966 c1ccc(c(c1)c2cc[nH]n2)F PS-6967 c1cc(ccc1F)SCCC(=O)O PS-6968 c1cc(c(cc1F)F)c2cc[nH]n2 PS-6969 c1cc(c(c(c1)F)c2cc[nH]n2)F PS-6970 c1ccc(c(c1)c2csc(n2)Nc3ccc(cc3C(F)(F)F)Br)O.Br PS-6971 CCCCCc1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl PS-6972 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)OCc3ccccc3)I PS-6973 c1c(cc(cc1C(F)(F)F)NC(=N)Nc2nc(cc(n2)O)C(F)(F)F)C(F)(F)F PS-6974 c1cc(ccc1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)I PS-6975 c1cnc(nc1)N2CCN(CC2)C(=O)C(=O)c3c[nH]c4c3cc(cc4)Br PS-6976 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2C(F)(F)F)Br PS-6977 CC(C)(C)OC(=O)n1cc(c2c1cccc2OCc3ccccc3)Br PS-6978 CCOc1cc(cc(c1OCC)OCC)c2c3cc(c(cc3ccn2)OC)OC PS-6979 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCCSCc3ccco3 PS-6980 c1ccc(c(c1)c2csc(n2)Nc3cc(ccc3F)F)O.Br PS-6981 c1ccc(c(c1)c2csc(n2)Nc3c(cccc3F)F)O.Br PS-6982 COc1ccc(cc1OC)C[C@H]2c3cc(c(cc3CCN2)OC)OC.Cl PS-6983 c1c(cc(c(c1I)O)I)C=O PS-6984 c1ccc(c(c1)c2csc(n2)Nc3ccccc3F)O.Br PS-6985 c1ccc(c(c1)c2csc(n2)Nc3cccc(c3)F)O.Br PS-6986 c1ccc(c(c1)c2csc(n2)Nc3ccc(cc3)F)O.Br PS-6987 c1cc(c(cc1Br)OC(F)(F)F)I PS-6988 c1cc(c(c(c1)Cl)Cl)NC(=N)Nc2nc(cc(n2)O)C(F)(F)F PS-6989 Cc1ccc2c(c1)c(cn2C(=O)OC(C)(C)C)I PS-6990 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccc(cc3)c4ccccc4 PS-6991 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)OCc3ccccc3)CO PS-6992 CC(C)(C)OC(=O)n1cc(c2c1c(ccc2)OCc3ccccc3)CO PS-6993 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)OCc3ccccc3)C=O PS-6994 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)Cl)Cl PS-6995 c1cc(c(cc1I)C(F)(F)F)Br PS-6996 c1c(cc(cc1C(F)(F)F)NC(=N)NC(=N)N)C(F)(F)F.Cl PS-6997 CC(=O)N1CCc2c1cc(cc2)NC3CCN(CC3)Cc4ccccc4 PS-6998 c1cc2c(cc1C(F)(F)F)c(cc(n2)C(F)(F)F)N3CCNCC3 PS-6999 c1cc(cc(c1)S(=O)(=O)N(C2CC2)C3CCNCC3)C(F)(F)F PS-7000 CCOC(=O)CSc1nnc(n1C)c2cc(nc(c2)Cl)Cl PS-7001 c1cc2c(cc1Br)cc(c(c2Br)O)C(=O)O PS-7002 c1c(c(c(cn1)I)N)I PS-7003 Cc1c(cc(n1CCNC(=O)OC(C)(C)C)c2ccccc2)C(=O)O PS-7004 CSc1c(c2nc(cc(n2n1)C(F)(F)F)C(F)(F)F)C(=O)N PS-7005 CCOC(=O)c1cc(=O)c2cc(ccc2o1)I PS-7006 CCOC(=O)c1cnc2c(c1Oc3ccc(cc3)OC)c(nn2C)C PS-7007 CC(C)(C)OC(=O)N1CCN(CC1)c2ccccc2Br PS-7008 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)Br PS-7009 COC(=O)c1cc(ccc1I)Br PS-7010 c1c2c(cc(c1F)Br)[nH]nc2I PS-7011 c1ccc(c(c1)N2CCNCC2)O.Br.Br PS-7012 Cc1c(cc(n1CCCNC(=O)OC(C)(C)C)C(C)(C)C)C(=O)O PS-7013 c1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)Br PS-7014 c1cc2c(c(c1)C(=O)O)-c3ccc(cc3C2)I PS-7015 c1c(cc(c(c1Br)N)Br)OC(F)(F)F PS-7016 COC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F PS-7017 COC(=O)C(=CNC1CC1)C(=O)c2cc(c(cc2Cl)Cl)F PS-7018 c1cc(c(cc1C(=O)O)OC(F)(F)F)I PS-7019 c1cc(ccc1Oc2ccc(cc2)I)Cl PS-7020 c1cc(cnc1)NC(=O)CN2CCNCC2.Cl.Cl.Cl PS-7021 CC(=O)Nc1ccc(cc1C(F)(F)F)I PS-7022 Cc1c(cc(n1CCCN2CCOCC2)c3ccccc3)C(=O)O PS-7023 c1cc(ccc1C(=O)C=Cc2cc(cs2)Br)Cl PS-7024 CC(C)(C)c1cc2nc(cc(n2n1)N3CCNCC3)C(F)(F)F PS-7025 c1c(cc(cc1Br)I)C(=O)O PS-7026 c1cc(c(cc1I)C(=O)O)Br PS-7027 CCOC(=O)c1c(csc1N)c2ccc(cc2)Br PS-7028 CC(C)(C)OC(=O)n1cc(c2c1cccc2Br)CO PS-7029 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)Br)CO PS-7030 Cc1ccc(cc1)S(=O)(=O)n2ccc(c2)C(=O)c3ccccc3 PS-7031 c1c(cc2c(c1C(F)(F)F)c(c(cn2)C(=O)O)O)C(F)(F)F PS-7032 c1cc2c3ccc(cc3[nH]c2cc1Br)Br PS-7033 CC(C)(C)OC(=O)n1cc(c2c1cccc2Br)C=O PS-7034 c1c(c(cc(c1Br)C(=O)O)Br)C(=O)O PS-7035 COc1cccc(c1CN2CCC(CC2)N)OC.Cl.Cl PS-7036 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)OC)C)Br PS-7037 c1cc(ccc1OC([C@@H](C(F)(F)F)F)(F)F)Br PS-7038 c1cc2c(cc1Br)c(n[nH]2)I PS-7039 c1cc(c(cc1OC(F)(F)F)Cl)I PS-7040 c1cc(ccc1C(c2ccc(cc2)Cl)N3CCNCC3)Cl PS-7041 c1cc(ccc1N)Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F PS-7042 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)C#N)Br PS-7043 COc1ccc(cc1)CNC(=O)c2ccc(cn2)Br PS-7044 COC(=O)c1ccc(c(c1)OCc2ccccc2)Br PS-7045 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cc2)C(=O)OC PS-7046 CC(C)(C)OC(=O)N1CCN(CC1)Cc2cccc(c2)C(=O)O PS-7047 c1cc(c(cc1c2ccc(c(c2)C(F)(F)F)N)C(F)(F)F)N PS-7048 c1c(cc(c(c1Br)O)Br)C(F)(F)F PS-7049 c1[nH]c(c(n1)I)I PS-7050 CC(C)(C)OC(=O)NCCNc1ccc(cc1N)C(F)(F)F PS-7051 c1cc(ccc1C[C@@H](C(=O)O)NC=O)I PS-7052 c1cc(ccc1Oc2nccc(n2)C(F)(F)F)Br PS-7053 c1c(cc(c(c1Br)N)Br)C(F)(F)F PS-7054 c1c(cc(c(c1C(F)(F)F)N)Br)Br PS-7055 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)Cl PS-7056 c1cc(cc(c1)C(F)(F)F)C(=O)c2ccc(cc2)C(F)(F)F PS-7057 c1cc(cc(c1)C(F)(F)F)C(=O)c2cccc(c2)C(F)(F)F PS-7058 CCOC(=O)c1c(nc(s1)c2ccc(cc2Cl)Cl)O PS-7059 c1cc(c(cc1OCC(F)(F)F)C(=O)O)OCC(F)(F)F PS-7060 c1cc(ccc1c2ccc(cc2)Br)OC(F)(F)F PS-7061 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)Cl PS-7062 c1cc(ccc1C(F)(F)F)NS(=O)(=O)c2ccc(cc2)N PS-7063 CCOC(=O)c1c(c2cc(ccc2nc1SC)Cl)Cl PS-7064 CC(C)(C)c1c(sc(n1)N)Br.Br PS-7065 c1cc(c(cc1C(=O)O)C(F)(F)F)I PS-7066 c1cc2c(cc1Cl)c(cc(n2)C(F)(F)F)N3CCNCC3 PS-7067 c1cc2c(cc(nc2c(c1)OC(F)(F)F)C(F)(F)F)Cl PS-7068 CCOC(=O)c1c(sc(n1)Br)Br PS-7069 c1cc(ccc1S(=O)(=O)N(C2CC2)C3CCNCC3)Cl PS-7070 c1cc(ccc1c2ccc(cc2)I)Cl PS-7071 COc1ccc(c(c1)O)C(=O)C=Cc2ccc(c(c2)OC)OC PS-7072 c1cc(ccc1Oc2ccc(cc2)I)F PS-7073 c1cc2c(cc1F)c(cc(n2)C(F)(F)F)N3CCCNCC3 PS-7074 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2[nH]c(=S)[nH]n2 PS-7075 c1cc(c(cc1C#N)OC(F)(F)F)I PS-7076 COc1cc(ccc1I)Br PS-7077 Cc1c(sc(n1)C2CCN(CC2)C(=O)OC(C)(C)C)CO PS-7078 c1ccc(cc1)COc2ccccc2c3ccccc3N.Cl PS-7079 c1ccc(cc1)c2ccccc2N3CCNCC3.Cl.Cl PS-7080 c1cc(ccc1OCCCN2CCNCC2)F.Cl.Cl PS-7081 Cc1ccc2c(c1Br)cnn2C(=O)OC(C)(C)C PS-7082 Cc1cc(cc(c1I)C)Br PS-7083 c1cc2c(cc(nc2c(c1)Br)C(F)(F)F)Cl PS-7084 c1cc2c(cc1Br)c(cc(n2)C(F)(F)F)Cl PS-7085 c1ccc(cc1)C(c2ccccc2)OCCN3CCCNCC3 PS-7086 Cc1c(c2ccccc2n1C(=O)OC(C)(C)C)Br PS-7087 Cc1cccc2c1n(cc2Br)C(=O)OC(C)(C)C PS-7088 Cc1ccc2c(c1)c(cn2C(=O)OC(C)(C)C)Br PS-7089 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)O)C)Br PS-7090 COC(=O)c1cc(c(c(c1)Br)N)Br PS-7091 c1cc(cc(c1)S(=O)(=O)C(F)(F)F)NC2CCNCC2 PS-7092 c1c(cc(c(c1C(F)(F)F)Br)N)C(F)(F)F PS-7093 c1c(c(cc(c1N)Br)C(F)(F)F)C(F)(F)F PS-7094 Cc1c(cc(cc1Br)C(=O)OC)Br PS-7095 c1c(c(cnc1Cl)C(F)(F)F)I PS-7096 CS(=O)(=O)c1ccc(cc1)c2nc(on2)C3CCNCC3 PS-7097 c1ccc2c(c1)nc(o2)C[C@@H](c3ccc(cc3)C(F)(F)F)O PS-7098 c1ccc2c(c1)nc(o2)C[C@@H](c3cccc(c3)C(F)(F)F)O PS-7099 c1cc2c(cc1C(F)(F)F)nnn2C3CCNCC3.Cl PS-7100 Cc1ccc(cc1Nc2nccc(n2)c3cccnc3)C(=O)O PS-7101 c1ccc(cc1)CNC(=O)CN2CCNCC2.Cl.Cl PS-7102 CCOC(=O)C1CCC(N1Cc2ccccc2)C(=O)OCC PS-7103 CC(C)(C)OC(=O)Nc1ccc(cc1C=O)OC(F)(F)F PS-7104 CN(C)[C@@H](CN)c1ccc(cc1)C(F)(F)F.Cl.Cl PS-7105 c1cc(sc1)CNC(=O)c2cc(c(nc2Cl)Cl)F PS-7106 CCOC(=O)C(c1ccc(cc1Cl)Cl)C(=O)OCC PS-7107 CCOC(=O)CNc1ccc(cc1)I PS-7108 c1ccc(cc1)COc2ccc(cc2)N3CCNCC3.Cl PS-7109 CCOC(=O)C(c1cccc(c1)C(F)(F)F)C(=O)OCC PS-7110 COc1cccc2c1nc(c(c2Cl)c3ccccc3)Cl PS-7111 c1cc(c(cc1Br)C(F)(F)F)S(=O)(=O)N PS-7112 c1cc(c(cc1C(F)(F)F)Br)S(=O)(=O)N PS-7113 c1cc(c(cc1C(F)(F)F)S(=O)(=O)N)Br PS-7114 c1cc(c(cc1S(=O)(=O)N)C(F)(F)F)Br PS-7115 c1c(cc(cc1Br)Br)C(F)(F)F PS-7116 c1cc(c(cc1Br)C(F)(F)F)Br PS-7117 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)Cl PS-7118 c1cc(ncc1C(F)(F)F)SCc2ccc(o2)C(=O)O PS-7119 c1cc(c(cc1OC(F)(F)F)I)N PS-7120 c1ccc(cc1)[C@H](CC(=O)c2ccccc2)c3ccccc3O PS-7121 CC(C)(C)OC(=O)n1c2ccc(cc2cn1)OC(F)(F)F PS-7122 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)F PS-7123 COC(=O)c1cccc2c1c(n[nH]2)I PS-7124 COC(=O)c1ccc2c(c1)[nH]nc2I PS-7125 Cc1cc(ccc1I)OC(F)(F)F PS-7126 c1cc(ccc1OCC(F)(F)F)I PS-7127 CCOC(=O)c1cnc2c(c1O)cccc2OC(F)(F)F PS-7128 CCOC(=O)c1cnc2ccc(cc2c1O)OC(F)(F)F PS-7129 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C[C@@H](C(=O)O)N PS-7130 Cc1c(c(n[nH]1)C)CCN.Br.Br PS-7131 C1COc2c(c(sc2Br)Br)O1 PS-7132 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1Cl)C(=O)O PS-7133 c1cc2c(cc(nc2c(c1)C(F)(F)F)C(F)(F)F)Cl PS-7134 c1cnc2cc(cc(c2c1Cl)C(F)(F)F)C(F)(F)F PS-7135 CCCc1c(cnn1c2cc(cc(c2)Cl)Cl)C(=O)O PS-7136 c1cc(c(cc1Br)C(F)(F)F)NC(=S)N PS-7137 c1cc(c(cc1OC(F)(F)F)CC(=O)O)Br PS-7138 c1cc(c(cc1Br)I)O PS-7139 c1cc(ccc1C(=S)N)Oc2ccc(cn2)C(F)(F)F PS-7140 CC(=O)Nc1ccc(c(c1)Br)OC(F)(F)F PS-7141 c1cc(c(cc1Br)I)N PS-7142 CCOC(=O)[C@@H]1CN(CCC1=O)Cc2ccccc2.Cl PS-7143 CCOC(=O)[C@@H]1CCN(CC1=O)Cc2ccccc2.Cl PS-7144 c1cc(ccc1NC(=N)NC(=N)N)OC(F)(F)F.Cl PS-7145 c1cc(cc(c1)C(F)(F)F)c2nc(on2)C3CCNCC3 PS-7146 CC(C)(C)OC(=O)n1c2cc(ccc2cn1)Br PS-7147 CC(C)(C)OC(=O)n1c2ccc(cc2cn1)Br PS-7148 CC(C)(C)OC(=O)n1c2cccc(c2cn1)Br PS-7149 c1ccc(cc1)Oc2ccc(cn2)I PS-7150 c1cc(c(cc1C#N)C(F)(F)F)I PS-7151 c1cc(c(cc1I)C(F)(F)F)C#N PS-7152 CC(C)(C)OC(=O)n1cc(c2c1cccc2)Br PS-7153 CC(C)(C)OC(=O)n1ccc2c1cccc2Br PS-7154 CC(C)(C)OC(=O)n1ccc2c1c(ccc2)Br PS-7155 COc1cc(c(cc1Br)OC)Br PS-7156 c1c(cc(c(c1C(=O)O)O)Br)Br PS-7157 CCO[C@H](C)Oc1ccc2cc(ccc2c1)Br PS-7158 c1c(nc(nc1N2CCOCC2)N3CCOCC3)C(=O)O PS-7159 c1ccc(c(c1)C(=O)c2cc(ccc2N)Br)F PS-7160 c1cc(c2c(c1Br)nsn2)Br PS-7161 COC(=O)c1cc(cc(c1)Br)Br PS-7162 Cc1c(cc(cc1Br)C(=O)O)Br PS-7163 c1c2c(cc(c1F)Br)[nH]nc2Br PS-7164 CC(C)(C)c1ccc(cc1)C(=O)Cc2nc3ccccc3o2 PS-7165 c1ccnc(c1)CN2CCC[C@@H](C2)C(=O)O.Cl.Cl PS-7166 c1ccc(cc1)C(=O)NC(=S)Nc2cc(ccc2F)F PS-7167 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2F)F PS-7168 c1ccc(cc1)C(=O)NC(=S)Nc2cccc(c2F)F PS-7169 c1ccc2c(c1)c(c(c(n2)C(F)(F)F)Br)O PS-7170 COc1ccc(cc1)C(=O)c2cccc(c2)Br PS-7171 c1cc(ccc1n2c(c(cn2)C(=O)O)C(F)(F)F)Cl PS-7172 c1ccc(cc1)c2ccc(cc2)c3nnc(o3)C(F)(F)F PS-7173 c1cc(ccc1c2c(c[nH]n2)c3ccncc3)C(F)(F)F PS-7174 CCOC(=O)C(c1ccc(cc1F)Cl)C(=O)OCC PS-7175 c1ccc2c(c1)c(=O)n(c(n2)C(=O)NC[C@H]3CCCO3)N PS-7176 c1cc(ccc1OC(F)(F)F)I PS-7177 c1ccc(c(c1)OC(F)(F)F)I PS-7178 c1cc(cc(c1)I)OC(F)(F)F PS-7179 c1c(cc(cc1Br)Br)N.Cl PS-7180 c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)Br PS-7181 c1cc(c(cc1C(F)(F)F)N)I PS-7182 c1cc(c(cc1I)C(F)(F)F)N PS-7183 c1cc(c2cnccc2c1Br)Br PS-7184 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccccc2 PS-7185 c1cc(cnc1)NC(=O)c2cc(c(nc2Cl)Cl)F PS-7186 CC(C)(C)CC(C)(C)c1ccc(c(c1)Br)O PS-7187 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)Br PS-7188 Cc1c(c(on1)c2ccc(cc2)C(F)(F)F)C(=O)OC PS-7189 c1ccc2c(c1)cccc2N3CCNCC3.Cl.Cl PS-7190 c1ccc(c(c1)Cn2cncn2)I PS-7191 Cc1c(c(no1)c2ccccc2)I PS-7192 c1c(cc(cc1OC(F)(F)F)Br)C(=O)O PS-7193 c1cc(c(cc1C(=O)O)OC(F)(F)F)Br PS-7194 c1cc(c(cc1C(=O)O)Br)OC(F)(F)F PS-7195 c1cc(c(cc1OC(F)(F)F)C(=O)O)Br PS-7196 c1c(cnc(n1)I)Br PS-7197 c1c(ncc(n1)I)Br PS-7198 Cc1cc(cc(c1)NC(=S)NC(=O)c2ccccc2)C PS-7200 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccccc2 PS-7201 c1cc(ccc1C(=O)O)Oc2nccc(n2)C(F)(F)F PS-7202 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=C/C(=O)O PS-7203 c1ccc(c(c1)S(=O)(=O)O)I PS-7204 c1cc(c(cc1C(=O)N)Br)OC(F)(F)F PS-7205 c1c(cnc(c1CO)N)Br.Br PS-7206 c1cc(nc(c1)I)Br PS-7207 CC(C)(C)OC(=O)N[C@@H](Cc1cccc(c1)F)C(=O)O PS-7208 COc1ccccc1Oc2ccc(cc2N)C(F)(F)F PS-7209 COc1ccc(cc1)Oc2ccc(cc2N)C(F)(F)F PS-7210 c1cnoc1c2nnc(o2)c3cc(nc(c3)Cl)Cl PS-7211 COC(=O)c1ccc(c(c1)C(F)(F)F)Br PS-7212 c1cc(c(cc1CC(=O)O)C(F)(F)F)Br PS-7213 c1cc(c(c(c1)Br)CC(=O)O)C(F)(F)F PS-7214 c1cc(c(cc1C(F)(F)F)Br)CC(=O)O PS-7215 c1cc(c(cc1Cl)Cl)NC(=N)NC(=N)N.Cl PS-7216 c1cc(c(cc1NC(=N)NC(=N)N)Cl)Cl.Cl PS-7217 c1cc(c(c(c1)Cl)NC(=N)NC(=N)N)Cl.Cl PS-7218 c1cc(c(c(c1)Cl)Cl)NC(=N)NC(=N)N.Cl PS-7219 c1c(cc(cc1Cl)Cl)NC(=N)NC(=N)N.Cl PS-7220 c1cc(c(cc1Cl)NC(=N)NC(=N)N)Cl.Cl PS-7221 c1c(cc(cc1Cl)I)C(=O)O PS-7222 c1cc(c(cc1I)C(=O)O)Cl PS-7223 c1ccc(c(c1)c2ccc(c(c2)C(=O)O)O)C(F)(F)F PS-7224 c1cc(ccc1C(F)(F)F)NC(=N)NC(=N)N.Cl PS-7225 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)C#N PS-7226 CC(C)(C)OC(=O)NCCNc1ccc(cn1)C(=O)O PS-7227 c1cc2c(cc(nc2c(c1)C(F)(F)F)C(F)(F)F)O PS-7228 c1cnc2cc(cc(c2c1O)C(F)(F)F)C(F)(F)F PS-7229 c1ccc(cc1)COc2ccc(c(c2)F)Br PS-7230 c1cc2c(cc1OC(F)(F)F)c(n[nH]2)Br PS-7231 CC(C)(C)OC(=O)N1C[C@@H](C[C@H]1C(=O)OC)N.Cl PS-7232 c1c(c(nc(n1)Cl)C(F)(F)F)C(=O)OCC2CC2 PS-7233 CC(C)(C)OC(=O)N1CCN(CC1)CC(=O)O.O.O PS-7234 c1ccc(cc1)c2cc(c(c(n2)S)C#N)C(F)(F)F PS-7235 c1ccc(cc1)n2c(cc(n2)C(F)(F)F)C(F)(F)F PS-7236 c1c(nc2c(cnn2c1C(F)(F)F)C#N)C(F)(F)F PS-7237 c1cc(c(cc1OC(F)(F)F)CC#N)Br PS-7238 c1c(cc(cc1Br)Br)C(=O)O PS-7239 CC(C)(C)OC(=O)n1cc(c2c1cccc2Cl)C=O PS-7240 c1c(c(nc(c1F)Cl)Cl)C(=O)N2CCOCC2 PS-7241 CC(=O)Nc1ccc(cc1F)I PS-7242 c1cc2c(ccc3c2c(c1)C(=O)OC3=O)Br PS-7243 COc1cc(nc(n1)Oc2cccc(c2)C(=O)O)OC PS-7244 CCOC(=O)c1ccc(cc1)I PS-7245 Cc1ccc(cc1I)C(=O)OC PS-7246 Cc1cc(ccc1I)C(=O)OC PS-7247 c1cc(ccc1CCC(=O)O)I PS-7248 c1ccc2c(c1)c(cc(n2)C(F)(F)F)Br PS-7249 Cn1c2cccc(c2c(n1)I)F PS-7250 c1cc2c(cc1Br)c(co2)Br PS-7251 c1ccc(cc1)C(c2ccccc2)N3CC(C3)O.Cl PS-7252 c1ccc(cc1)COc2ccc(cc2)c3ccccc3N PS-7253 CC(C)(C)OC(=O)n1ccc2c1c(ccc2)C(=O)OC PS-7254 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)O PS-7255 CCOC(=O)c1cc(c(nc1N2CCNCC2)C)C#N PS-7256 c1ccc(cc1)C(=O)NC(=S)Nc2cccc(c2)F PS-7257 c1ccc(cc1)c2c(n3c(n2)cccn3)Br PS-7258 c1ccc(cc1)C2(CCNCC2)c3ccccc3.Cl PS-7259 c1cc(ccc1c2ccc(cc2)N)C(F)(F)F.Cl PS-7260 c1cc(cc(c1)N)c2ccc(cc2)C(F)(F)F.Cl PS-7261 c1ccc(c(c1)c2cccc(c2)C(F)(F)F)N.Cl PS-7262 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)C(=O)O PS-7263 CCS(=O)(=O)c1cc(c(cc1N)OC)C(=O)OC PS-7264 CC(C)(C)OC(=O)CN1CCNCC1.Cl.Cl PS-7265 c1cc(ccc1OC(C(F)F)(F)F)Br PS-7266 c1cc(cc(c1)Br)OC(C(F)F)(F)F PS-7267 c1cnc(cc1I)C(F)(F)F PS-7268 c1ccc2c(c1)c(ccn2)c3c[nH]nc3c4ccccn4 PS-7269 c1ccc(cc1)c2cc(=O)c3ccc4ccccc4c3o2 PS-7270 c1cc(ccc1c2nnn(n2)CC(=O)O)C(F)(F)F PS-7271 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C(=N/O)/N PS-7272 COC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F PS-7273 c1cc(c(cc1C(F)(F)F)C(F)(F)F)CC(=O)O PS-7274 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CC(=O)O PS-7275 CC(C)(C)OC(=O)Nc1ccc(cc1)Br PS-7276 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O PS-7277 Cc1ccc2c(c1)n(nc2I)C PS-7278 C[C@@H](c1cc(cc(c1)C(F)(F)F)C(F)(F)F)NC PS-7279 c1c(c(cc(c1OC(F)(F)F)Br)N)N PS-7280 c1c(cc(c(c1N)N)OC(F)(F)F)Br PS-7281 c1c(cc(c(c1N)N)Br)OC(F)(F)F PS-7282 c1cc(cc(c1)C(F)(F)F)c2ccn(n2)CC(=O)O PS-7283 c1cc(ccc1OC(F)F)I PS-7284 COc1c(cc(cc1F)I)F PS-7285 c1cc(ccc1CN)I.Cl PS-7286 c1cc(cc(c1)I)CN.Cl PS-7287 CN(C)c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)F PS-7288 c1cc(c(cc1C=O)Br)OC(F)(F)F PS-7290 c1cc(c(cc1C=O)OC(F)(F)F)Br PS-7291 c1c(cc(cc1OC(F)(F)F)Br)C=O PS-7292 c1c(cc(c(c1C=O)O)C(F)(F)F)Br PS-7293 c1cc(c(cc1C(=O)O)C(F)(F)F)Br PS-7294 c1cc(c(c(c1)C(F)(F)F)Br)C(=O)O PS-7295 c1cc(c(c(c1)Br)C(=O)O)C(F)(F)F PS-7296 c1c(cc(cc1C(F)(F)F)Br)C(=O)O PS-7297 c1cc(c(cc1Br)C(F)(F)F)C(=O)O PS-7298 Cc1cc(cc(c1O)I)Cl PS-7299 c1ccc(c(c1)c2ccc3cnccc3n2)C(=O)O.O PS-7300 c1ccc(cc1)C(=O)c2cc(ccc2F)C(F)(F)F PS-7301 c1ccc(cc1)C(=O)c2cccc(c2F)C(F)(F)F PS-7302 c1ccc(cc1)C(=O)c2ccc(cc2F)C(F)(F)F PS-7303 c1cc(ccc1C=O)Oc2nccc(n2)C(F)(F)F PS-7304 c1ccc(c(c1)N)SCc2c(cccc2Cl)F PS-7305 c1cnc(c(c1I)C=O)Cl PS-7307 CN(C)c1ccc(cc1)/C=C/C(=O)c2ccccc2O PS-7308 c1cc(cc(c1)Oc2cc(cc(c2)Cl)Cl)C=O PS-7309 COc1cc(nc(n1)C2CCCCC2C(=O)O)OC PS-7310 Cc1c2ccc(cc2oc(=O)c1Cc3ccccc3)O PS-7311 CCOC(=O)C(c1ccc(cc1)OC)C(=O)OCC PS-7312 Cc1ccc(cc1)S(=O)(=O)n2cc(nc2)C(=O)O PS-7313 c1ccc(c(c1)c2ccc(cc2)C(F)(F)F)C(=O)O PS-7314 c1cc(cc(c1)C(F)(F)F)c2ccc(cc2)C(=O)O PS-7315 c1cc(oc1)C(=O)/C=C/c2ccc(cc2)C(F)(F)F PS-7316 c1ccc2cc(ccc2c1)C(=O)CC(=O)C(F)(F)F PS-7317 c1ccc(c(c1)C(=O)c2cc(ccc2N)Cl)Cl PS-7318 c1cc(c(c(c1)Cl)F)NC(=N)NC(=N)N.Cl PS-7319 c1cc2c(cc1Cl)c(cc(n2)C(F)(F)F)Cl PS-7320 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)Cl PS-7321 c1cc(c(cc1Br)OC(F)(F)F)C#N PS-7322 c1cc(c(cc1Br)C#N)OC(F)(F)F PS-7323 c1cc(c(c(c1)I)C(=O)O)F PS-7324 c1cc(c(cc1I)F)C(=O)O PS-7325 c1cc(c(cc1I)C(=O)O)F PS-7326 c1cc(c(cc1F)I)C(=O)O PS-7327 c1cc(c(cc1F)C(=O)O)I PS-7328 c1c(cc(cc1F)I)C(=O)O PS-7329 c1cc(c(cc1C(=O)O)I)F PS-7330 Cc1c(cnc(c1Br)N)Br PS-7331 c1cc(c(cc1Br)Br)CO PS-7332 c1cc2c(c(c1)Br)nc([nH]2)C(F)(F)F PS-7333 C#Cc1ccc(cc1Br)OC(F)(F)F PS-7334 Cc1cc(c(c(c1)Br)N)Br PS-7335 c1cc(ccc1c2cc3c(s2)c(ncn3)Cl)F PS-7336 c1cc(ccc1c2csc3c2c(ncn3)Cl)F PS-7337 COC(=O)C=Cc1ccc(cc1Cl)C(F)(F)F PS-7338 CS(=O)(=O)c1cc(cc(c1)S(=O)(=O)C)CO PS-7339 CC(=O)c1cccc(c1)c2ccc(cc2)C(F)(F)F PS-7340 c1cc(c(cc1CC#N)C(F)(F)F)Br PS-7341 c1cc(c(cc1C(F)(F)F)Br)CC#N PS-7342 CC(=O)c1cc(ccc1F)I PS-7343 c1c(cc(cc1Br)Br)C=O PS-7344 c1cc(c(cc1C=O)Br)Br PS-7345 CCOC(=O)c1cc(ccc1Cl)Br PS-7346 Cn1c2cc(c(cc2c(n1)Cl)F)Br PS-7347 c1c(cc(cc1Cl)I)C#N PS-7348 c1cc(c(cc1I)C#N)Cl PS-7349 c1ccc(cc1)COc2ccc(cc2)Br PS-7350 c1ccc(cc1)COc2cccc(c2)Br PS-7351 c1ccc(cc1)OCc2ccccc2Br PS-7352 c1ccc(cc1)[C@@H](c2ccc(cc2)Br)O PS-7353 c1cc(ccc1C(=O)c2ccc(cc2C(=O)O)F)F PS-7354 Cc1ccc(cc1I)C(=O)O PS-7355 Cc1c(cccc1I)C(=O)O PS-7356 Cc1ccc(c(c1)C(=O)O)I PS-7357 c1cc2c(cc1F)[nH]nc2I PS-7358 CSc1c(c(nc(n1)c2ccccc2)Cl)C#N PS-7359 c1cc(c(c(c1)F)C#N)OCc2ccc(cc2)Cl PS-7360 Cc1c2cc(ccc2sc1Br)Cl PS-7361 c1c(c(nc(=O)n1[C@H]2[C@@H]([C@@H]([C@H](O2)CO)O)O)N)F PS-7362 c1c(cc(cc1Br)Br)C#N PS-7363 Cc1c2c(ncnc2Cl)sc1c3ccccc3 PS-7364 c1cc(nc(c1Br)Cl)C(F)(F)F PS-7365 c1c(cnc(c1Br)Cl)C(F)(F)F PS-7366 COCCCCC(=O)c1ccc(cc1)C(F)(F)F PS-7367 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)C=O PS-7368 CCOC(=O)CC(=O)c1ccc(cc1)C(F)(F)F PS-7369 CC(C)(C)c1ccc(cc1)I PS-7370 c1c(sc(n1)N)Br.Br PS-7371 CSc1ccc(cc1)Oc2cccc(c2C#N)F PS-7372 CC1(N([C@H](CO1)C(=O)OC)C(=O)OC(C)(C)C)C PS-7373 CC(C)(C)OC(=O)NC1(CCOCC1)CC(=O)O PS-7374 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)O PS-7375 c1cc(c(cc1Br)OC(F)(F)F)F PS-7376 c1cc(c(cc1OC(F)(F)F)Br)F PS-7377 c1cc(c(cc1Br)F)OC(F)(F)F PS-7378 c1ccc(cc1)COc2ccc(cc2)NC(=S)N PS-7379 c1ccc(cc1)c2ccc(cc2)C(=O)c3ccccc3 PS-7380 CC(C)(C)OC(=O)N1CCN(CC1)CCC(=O)O PS-7382 CCS(=O)(=O)c1ccc(c(c1)C(=O)OC)OC PS-7383 C1CCc2c(c(c(c(n2)S)C#N)C(F)(F)F)C1 PS-7384 C[C@@H](c1cc(cc(c1)C(F)(F)F)C(F)(F)F)O PS-7385 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)O PS-7386 c1cc(c(cc1C(F)(F)F)C(=O)O)C(F)(F)F PS-7387 Cc1c(c(no1)c2c(cccc2Cl)Cl)CO PS-7388 c1c(cc(c(c1C(F)(F)F)N)F)Br PS-7389 Cc1cc(nc(n1)N(C)c2ccc(cc2)C(=O)O)C PS-7391 CCNc1cc(cc(c1)C(F)(F)F)C(F)(F)F PS-7392 C[C@H](c1cc(cc(c1)C(F)(F)F)C(F)(F)F)N PS-7393 c1cc2c(c(c1)C(F)(F)F)ncc(c2O)C(=O)O PS-7394 c1cc(ccc1c2nnc(o2)S)Br PS-7395 c1cc(ccc1SC(F)(F)F)Br PS-7396 c1cc(c(cc1O)Br)OC(F)(F)F PS-7397 c1cc2c(cc1F)c(no2)C3CCNCC3.Cl PS-7398 Cc1cc(c2cc(ccc2n1)Br)Cl PS-7399 Cc1cc(cc(c1)Nc2c(cccc2N)C(=O)O)C PS-7400 c1cc(ccc1C(=O)O)n2ccc(n2)C(F)(F)F PS-7401 CC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F PS-7402 c1cc(c(cc1Br)OC(F)(F)F)N PS-7403 c1cc(c(cc1OC(F)(F)F)N)Br PS-7404 c1cc(c(cc1N)OC(F)(F)F)Br PS-7405 c1cc(c(cc1N)Br)OC(F)(F)F PS-7406 c1c(cc(cc1OC(F)(F)F)Br)N PS-7407 c1cc(c(cc1OC(F)(F)F)Br)N PS-7408 c1cc(c(cc1Br)N)OC(F)(F)F PS-7409 c1cc2cc(ccc2nc1)I PS-7410 c1c(cc(c(c1N)N)Br)C(F)(F)F PS-7411 c1c(cc(c(c1C(F)(F)F)N)N)Br PS-7412 Cc1cc(ccc1Br)OC(F)(F)F PS-7413 Cc1cc(cc(c1)Br)OC(F)(F)F PS-7414 Cc1cc(ccc1OC(F)(F)F)Br PS-7415 c1cc(cc(c1)Br)OCC(F)(F)F PS-7416 COc1ccc(cc1C(F)(F)F)Br PS-7417 c1cc(c(cc1CO)C(F)(F)F)Br PS-7418 c1cc(c(cc1C(F)(F)F)CO)Br PS-7419 c1cc(c(cc1C(F)(F)F)Br)CO PS-7420 c1c(cnc(c1Br)F)Br PS-7421 c1c(cnc(c1Br)Br)F PS-7422 c1cc(c(cc1Cl)I)O PS-7424 c1cc(c(cc1O)I)Cl PS-7425 c1cc(c(cc1I)O)Cl PS-7426 c1cc(ccc1F)S(=O)(=O)c2ccc(cc2)F PS-7428 c1cc2c(cc1F)sc3n2cc(n3)C(=O)O.O PS-7429 c1cc(ccc1CN2CCCCC2)Br PS-7430 Cc1c(sc(n1)c2ccccc2)Br PS-7431 Cc1nc(c(s1)Br)c2ccccc2 PS-7432 c1cc(ccc1N)Oc2ccc(c(c2)Cl)Cl PS-7433 c1cc(c(cc1F)Br)S(=O)(=O)N PS-7434 c1cc(c(cc1CN)C(F)(F)F)Br PS-7435 c1cc(c(cc1Cl)I)N PS-7436 c1cc(c(cc1N)I)Cl PS-7437 c1cc(c(cc1N)Cl)I PS-7438 c1c(c(cc(c1F)Br)Cl)C(=O)O PS-7439 COc1cc(ccc1OCc2ccccc2)CC#N PS-7440 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CC#N PS-7441 c1cc(c(cc1C(F)(F)F)CC#N)C(F)(F)F PS-7442 c1cc(c(cc1C(F)(F)F)C(F)(F)F)CC#N PS-7443 CS(=O)(=O)c1ccc(cc1F)Br PS-7444 CS(=O)(=O)c1cc(ccc1F)Br PS-7445 c1c(cnc(c1Br)N)S(=O)(=O)O PS-7446 c1cc(c(cc1C=O)C(F)(F)F)Br PS-7447 c1c(cc(cc1C(F)(F)F)Br)C=O PS-7448 c1cc(c(cc1C(F)(F)F)C=O)Br PS-7449 c1cc(cc(c1)Br)C(=O)C(F)(F)F PS-7450 c1ccc(cc1)CN2CCC(CC2)(C#N)O.Cl PS-7451 CCOc1cc(ccc1Br)N.Cl PS-7452 Cc1c(cccc1I)Cl PS-7453 c1ccc(cc1)C=CC=CC(=O)c2ccc(cc2)F PS-7454 CCOc1cc(ccc1C(=O)OCC)CC(=O)O PS-7455 c1ccc(cc1)COc2cccc(c2)C(F)(F)F PS-7456 c1ccc(cc1)COc2ccc(cc2)C(F)(F)F PS-7457 CS(=O)(=O)c1ccc(c(c1)C(F)(F)F)C=O PS-7458 COc1cccc(c1I)F PS-7459 c1cc(c(cc1Br)Br)O PS-7460 c1cc(c(cc1Br)O)Br PS-7461 CN(C)c1ccc(cc1)C=CC(=O)c2ccccc2 PS-7462 c1ccc(cc1)COc2ccc3c(c2)c(c[nH]3)C=O PS-7463 c1ccc(cc1)COc2ccc3c(c2)[nH]cc3C=O PS-7464 Cc1cc(n(n1)c2ccc(cc2)Br)C PS-7465 c1ccc(cc1)C(=O)c2cc(ccc2Cl)Cl PS-7466 c1cc(ccc1c2ccc(cc2)Br)F PS-7467 c1ccc(cc1)c2ccc(cc2F)Br PS-7468 Cc1c(ccc(n1)Br)Br PS-7469 Cc1cc(ncc1Br)Br PS-7470 Cc1cc(cnc1Br)Br PS-7471 Cc1cc(c(nc1)Br)Br PS-7472 c1cc(c(cc1C=CC(=O)O)C(F)(F)F)Cl PS-7473 CCOC(=O)[C@H](Cc1c[nH]c2c1cc(cc2)F)N PS-7474 c1cc2c(cc1SC(F)(F)F)sc(n2)N PS-7475 c1cc(cc(c1)c2ccc(cc2)C(F)(F)F)C=O PS-7476 c1ccc(cc1)C(=O)c2ccc(cc2)C(F)(F)F PS-7477 c1ccc(cc1)C(=O)c2ccccc2C(F)(F)F PS-7478 c1ccc(cc1)C(=O)c2cccc(c2)C(F)(F)F PS-7479 c1cnccc1N2CCCNCC2.Cl.Cl PS-7480 c1cc(c(cc1Br)C(F)(F)F)C#N PS-7481 c1cc(c(cc1C#N)C(F)(F)F)Br PS-7482 c1cc(c(c(c1)C(F)(F)F)Br)C#N PS-7483 c1cc(c(cc1C(F)(F)F)C#N)Br PS-7484 c1cc(c(c(c1)I)C=O)F PS-7485 c1cc(c(cc1I)F)C=O PS-7486 c1cc(c(cc1I)C=O)F PS-7487 Cc1cc(cc(c1)Br)Br PS-7488 c1ccc(c(c1)c2cccc(c2)C(=O)O)N.Cl PS-7489 c1ccc(c(c1)c2ccc(cc2)C(=O)O)N.Cl PS-7490 c1cc(cc(c1)C(=O)O)c2cccc(c2)N.Cl PS-7491 c1cc(ccc1c2ccc(cc2)N)C(=O)O.Cl PS-7492 c1cc(c(cc1F)NC(=N)NC(=N)N)F.Cl PS-7493 c1cc(c(cc1NC(=N)NC(=N)N)F)F.Cl PS-7494 c1c(cc(cc1F)F)NC(=N)NC(=N)N.Cl PS-7495 CN1CCN(CC1)CCCCl.Cl.Cl PS-7496 c1cc2c(cc1F)c(cc(n2)C(F)(F)F)Cl PS-7497 COC(=O)c1cc(ccc1Br)Cl PS-7498 c1c2c(cc(c1F)Br)[nH]nc2Cl PS-7499 c1ccc(cc1)Oc2cccc(c2)Br PS-7500 c1ccc(cc1)Oc2ccc(cc2)Br PS-7501 c1c(onc1C(=O)O)CN2CCOCC2.Cl PS-7502 c1cc2nc(cn2cc1Br)N.Cl PS-7503 CC(=O)c1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C PS-7504 c1cc(ccc1OC2CCNCC2)Cl.Cl PS-7505 c1cc(ccc1NC(=N)NC(=N)N)Cl.Cl PS-7506 c1cc(cc(c1)Cl)NC(=N)NC(=N)N.Cl PS-7507 c1ccc(c(c1)NC(=N)NC(=N)N)Cl.Cl PS-7508 c1cc(cc(c1)I)C(=O)O PS-7510 Cc1cc(c2nccn2c1)Br.Cl PS-7511 COC(=O)CC(=O)c1ccc(nc1)C(F)(F)F PS-7512 c1cc(c(c(c1)I)C#N)F PS-7513 c1cc(c(cc1C#N)I)F PS-7514 c1cc(c(cc1I)F)C#N PS-7515 c1cc(c(cc1C#N)F)I PS-7516 c1cc(c(cc1I)C#N)F PS-7517 c1cc(c(cc1F)I)C#N PS-7518 c1ccc(cc1)COc2ccc(cc2Cl)C=O PS-7519 c1c(c(=O)[nH]c(=O)n1[C@H]2C[C@@H]([C@H](O2)CO)O)F PS-7520 COC(=O)CC(=O)c1ccc(cc1)C(F)(F)F PS-7521 CCOC(=O)CC(=O)c1cc(c(cc1F)F)F PS-7522 c1c(cc(cc1C(F)(F)F)S)C(F)(F)F PS-7523 CC(=O)n1c(cc(n1)C(F)(F)F)C(F)(F)F PS-7524 c1ccc2c(c1)c3ccc(cc3[nH]2)Br PS-7525 CC(C)c1ccc(cc1)I PS-7526 CN(C)C(=O)c1cc(ccc1Br)F PS-7527 c1c(cc(c(c1Cl)N)Cl)OC(F)(F)F PS-7528 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)Cl PS-7529 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CC#N PS-7530 COc1ccc(cc1C(=O)OC)S(=O)(=O)N PS-7531 c1cc2c(cc1I)NCC2 PS-7532 CC(=O)c1cc(cc2c1CCC2(C)C)C(C)(C)C PS-7533 CC(C)(C)OC(=O)Nc1nc(cs1)C(=O)O PS-7534 COc1ccc(cc1C(=O)OC)S(=O)(=O)C PS-7535 c1cc(cc(c1)C(F)(F)F)c2csc(n2)N PS-7536 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)F)F PS-7537 c1cc(c(cc1C(F)(F)F)C(F)(F)F)CO PS-7538 c1c(c(c(nc1Cl)Cl)C=O)C(F)(F)F PS-7539 COc1ccc2c(c1)c(c3ccccc3n2)Cl PS-7540 c1ccc2cc(ccc2c1)c3cc4ccccc4[nH]3 PS-7541 Cc1ccc(cc1)Sc2cccc(c2C#N)F PS-7542 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CN PS-7543 C[C@@H](Cc1ccc(cc1)Br)C(=O)O PS-7544 c1cc2c(cc[nH]2)cc1I PS-7545 c1cc(c(cc1C(F)(F)F)F)Br PS-7546 c1cc(c(cc1F)C(F)(F)F)Br PS-7547 c1cc(c(cc1Br)C(F)(F)F)F PS-7548 c1cc2cccc(c2c(c1)S(=O)(=O)O)Cl PS-7549 CNCc1cscc1Br.Cl PS-7550 c1c(cc(c(c1C(=O)O)F)Cl)C(F)(F)F PS-7551 c1cc(cc2c1ccc(n2)Cl)Br PS-7552 c1cc2cnc(cc2c(c1)Br)Cl PS-7553 c1cc2cc(ncc2c(c1)Br)Cl PS-7554 c1cc(cc2c1cc(nc2)Cl)Br PS-7555 c1cc(c2ccncc2c1Cl)Br PS-7556 c1ccc(cc1)C(c2ccccc2)NC(=S)N PS-7557 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)N PS-7558 c1ccc(cc1)COc2ccc(cc2)CC(=O)O PS-7559 c1ccc(c(c1)C=CC(=O)c2ccc(cc2)F)O PS-7560 c1cc(ccc1c2ccc(cc2)C(=O)O)C(=O)O PS-7561 c1cnc(cn1)c2nc(cc(n2)O)C(F)(F)F PS-7562 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C=O PS-7563 c1cc(c(cc1C(F)(F)F)C=O)C(F)(F)F PS-7564 c1cc(c(cc1C(F)(F)F)C(F)(F)F)C=O PS-7565 c1ccc(cc1)Oc2nc(nc(n2)Cl)Cl PS-7566 c1cc(sc1Br)Br PS-7567 c1c(c(cs1)Br)Br PS-7568 COc1ccc(cc1)CC2CCNCC2.Cl PS-7569 c1c(cc(c(c1C(=O)N)F)Cl)C(F)(F)F PS-7570 c1c(cnc(c1F)CN)Br.Cl PS-7571 c1c(cnc(c1Br)CN)F.Cl PS-7572 c1ccc(c(c1)OC(F)(F)F)S(=O)(=O)N PS-7573 c1c(c(cc2c1OC(C(O2)(F)F)(F)F)F)N PS-7574 c1cc(ccc1n2cc(cn2)Br)F PS-7575 c1ccc(c(c1)OC(F)(F)F)Br PS-7576 c1cc(ccc1OC(F)(F)F)Br PS-7577 c1cc(c(cc1C(F)(F)F)Br)O PS-7578 c1cc(c(cc1O)C(F)(F)F)Br PS-7579 c1cc(nc(c1I)F)F PS-7580 c1cc(c(cc1C(=O)O)Cl)OC(F)(F)F PS-7581 c1cc(c(cc1CN)Br)F.Cl PS-7582 c1cc(c(cc1Br)F)CN.Cl PS-7583 c1cc(c(cc1F)Br)CN.Cl PS-7584 c1cc(c(cc1F)CN)Br.Cl PS-7585 c1ccc(cc1)c2nc(cc(n2)O)C(F)(F)F PS-7586 c1cc(ccc1N2CCCCC2)Br PS-7587 c1cc(c(cc1N)C(F)(F)F)Br PS-7588 c1cc(c(cc1C(F)(F)F)Br)N PS-7589 c1cc(c(c(c1)N)Br)C(F)(F)F PS-7590 c1c(cc(cc1N)Br)C(F)(F)F PS-7591 c1cc(c(c(c1)Br)N)C(F)(F)F PS-7592 c1cc(c(cc1C(F)(F)F)N)Br PS-7593 c1cc(c(cc1Br)C(F)(F)F)N PS-7594 c1cc(c(c(c1)Cl)CC(=N)N)Cl.Cl PS-7595 c1cc(c(nc1)Cl)I PS-7596 c1cc(ncc1I)Cl PS-7597 c1cnc(cc1I)Cl PS-7598 Cc1ccc(n1c2ccc(cc2)C(F)(F)F)C PS-7599 CS(=O)(=O)c1ccc(cc1C(F)(F)F)N PS-7600 CS(=O)(=O)c1ccc(cc1N)C(F)(F)F PS-7601 c1ccc(cc1)c2cc(nc(n2)N)C(F)(F)F PS-7602 c1cc(n(c1)c2ccc(cc2)C(F)(F)F)C=O PS-7603 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C#N PS-7604 c1cc(c(c(c1)C(F)(F)F)C#N)C(F)(F)F PS-7605 c1cc(c(cc1C(F)(F)F)C#N)C(F)(F)F PS-7606 c1cc(c(cc1C(F)(F)F)C(F)(F)F)C#N PS-7607 Cc1c(cccc1Br)C(F)(F)F PS-7608 Cc1ccc(cc1Br)C(F)(F)F PS-7609 Cc1ccc(cc1C(F)(F)F)Br PS-7610 c1ccc2c(c1)nnn2C3CCNCC3.Cl PS-7611 c1c(ccc(c1)Cl)[C@H]2CC[C@@H](CC2)C(=O)O PS-7612 c1cc(ccc1OCCCN2CCNCC2)F PS-7613 COc1cc(nc(n1)CN2CCNCC2)OC PS-7614 COc1ccccc1C=CC(=O)c2ccccc2 PS-7615 c1cc(sc1)c2nc(on2)CCCC(=O)O PS-7616 c1ccc(cc1)C#Cc2ccc(c(c2)C(=O)O)O PS-7617 CC(=O)Oc1cc(cc(c1)OC(=O)C)C(=O)O PS-7618 c1cc(c(cc1OC(F)(F)F)CC(=O)O)F PS-7619 c1cc(c(c(c1)OC(F)(F)F)F)CC(=O)O PS-7620 c1cc(cc(c1)OC(C(F)F)(F)F)C(=O)O PS-7621 c1cc(ccc1C(=O)O)OC(C(F)F)(F)F PS-7622 C#Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F PS-7623 c1cc(ccc1c2cc(cc(c2)Cl)Cl)N PS-7624 COc1ccc2cc(ccc2n1)Br PS-7625 COc1cccc2c1nccc2Br PS-7626 c1ccc(cc1)C(c2ccccc2)N3CC(=O)C3 PS-7627 c1ccc(cc1)Cn2cc(cn2)Br PS-7628 COc1ccc2cc(ccc2c1)Br PS-7629 Cc1cc(c(nc1)F)I PS-7630 c1cc(c(cc1N)F)I PS-7631 c1cc(c(cc1I)F)N PS-7632 c1cc(c(cc1F)I)N PS-7633 c1cc(c(c(c1)I)N)F PS-7634 c1cc2c(c(c1)Br)OC(O2)(F)F PS-7635 c1cc2c(cc1Br)OC(O2)(F)F PS-7636 c1cc(c(c(c1C(=O)O)F)F)Br PS-7637 c1cc(c(nc1)Br)Br PS-7638 c1cnc(cc1Br)Br PS-7639 CC(C)(C)OC(=O)N(C)CC1CNC1.Cl PS-7640 CS(=O)(=O)Nc1ccc(cc1)CN.Cl PS-7641 Cn1c(cc(n1)C(=O)Nc2cccnc2)Cl PS-7642 c1ccc2c(c1)n3cc(nc3s2)C(=O)O.O PS-7643 COc1ccccc1C2C(CC(=O)O2)C(=O)O PS-7644 c1cc(ccc1NC(=S)N)OC(F)(F)F PS-7645 c1cc(ccc1OCC(=O)O)OC(F)(F)F PS-7646 CN1CCC=C(C1)C(=O)OC.Br PS-7647 Cc1cc(ccc1I)F PS-7648 CS(=O)(=O)c1ccc(cc1)CCN.Cl PS-7649 COc1ccc(cc1)c2ccc(cc2)N.Cl PS-7650 COc1cccc(c1)c2ccccc2N.Cl PS-7651 COc1ccc(cc1)c2cccc(c2)N.Cl PS-7652 COc1ccccc1c2cccc(c2)N.Cl PS-7653 COc1cccc(c1)c2ccc(cc2)N.Cl PS-7654 c1ccc(cc1)COc2ccc(cc2)N.Cl PS-7655 c1cc(c(cc1Br)C(=O)O)Cl PS-7656 c1cc(c(cc1Cl)C(=O)O)Br PS-7657 c1cc(c(cc1Br)Cl)C(=O)O PS-7658 c1c(cc(cc1Cl)Br)C(=O)O PS-7659 c1cc(c(cc1Cl)Br)C(=O)O PS-7660 c1ccc(cc1)Cn2cc(c3c2cccc3)C=O PS-7661 C1CNCCC1C(=O)N2CCOCC2.Cl PS-7662 CC(C)(C)c1cc(c(c(c1)C(C)(C)C)O)C=O PS-7663 CCOC(=O)[C@H](C)c1ccc(cc1)CC(C)C PS-7664 c1ccc(cc1)COc2ccc(cc2)C(F)F PS-7665 CCOC(=O)c1cc(=O)c2ccc(cc2o1)O PS-7666 CCOC(=O)c1cc(=O)oc2c1ccc(c2)O PS-7667 c1cc(ccc1c2ccc(cc2F)F)C(=O)O PS-7668 c1cc(ccc1CCC(=O)O)OC(F)(F)F PS-7669 c1cc(cc(c1)OC(F)(F)F)CCC(=O)O PS-7670 c1cc(c(cc1C(F)(F)F)/C=C/C(=O)O)F PS-7671 c1cc(c(cc1F)C(F)(F)F)/C=C/C(=O)O PS-7672 c1cc(c(cc1/C=C/C(=O)O)C(F)(F)F)F PS-7673 c1cc(c(c(c1)C(F)(F)F)F)C=CC(=O)O PS-7674 c1cc(c(cc1C=CC(=O)O)F)C(F)(F)F PS-7675 COC(=O)c1cc(c(nc1)Br)F PS-7676 c1c(c(cc(c1Br)F)N)C(=O)O PS-7677 c1c(cc(c(c1C(=O)O)N)Br)F PS-7678 CC(C)(C)OC(=O)n1c2cc(ccc2cn1)N PS-7679 Cc1c(cc(o1)S(=O)(=O)N(C)C)C(=O)O PS-7680 Cc1c(c(no1)c2ccc(cc2)OC)C(=O)O PS-7681 c1ccc(cc1)c2ccc(cc2)Br PS-7682 c1ccc(cc1)c2ccccc2Br PS-7683 CC(C)Oc1ccc(cc1Br)F PS-7684 COC(=O)c1ccc(c(c1)Br)F PS-7685 COC(=O)c1ccc(c(c1)F)Br PS-7686 COC(=O)c1cc(ccc1Br)F PS-7687 c1cc(c(c(c1)Br)F)CC(=O)O PS-7688 c1cc(c(cc1Br)F)CC(=O)O PS-7689 c1c(cc(cc1F)Br)CC(=O)O PS-7690 c1cc(c(cc1CC(=O)O)Br)F PS-7691 c1ccc(c(c1)c2ccccc2Cl)C(=O)O PS-7692 c1cc(ccc1F)S(=O)(=O)C/C(=N/O)/N PS-7693 c1ccc(c(c1)/C=C/C(=O)O)OC(F)(F)F PS-7694 c1cc(ccc1[C@@H]2CCCCN2)Cl.Cl PS-7696 CC(=O)Nc1ccc(c(c1)F)Br PS-7697 c1cc(cc(c1)F)OC2CCNCC2.Cl PS-7698 c1cc(ccc1NC(=N)NC(=N)N)F.Cl PS-7699 c1cc(cc(c1)F)NC(=N)NC(=N)N.Cl PS-7700 c1ccc(c(c1)NC(=N)NC(=N)N)F.Cl PS-7701 c1ccc2c(c1)c(cc(n2)C(F)(F)F)Cl PS-7702 c1cc2c(cc1C(F)(F)F)c(ccn2)Cl PS-7703 c1cnc(cn1)c2nc(on2)C3CCNCC3 PS-7704 COc1ccc(cc1C(=O)O)S(=O)(=O)N PS-7705 c1cc(c(c(c1)F)C#N)Oc2ccc(cc2)F PS-7706 c1cc2c(cc1F)c(cc(n2)C(F)(F)F)O PS-7707 CCCCC(=O)c1ccc(c(c1)Cl)Cl PS-7708 c1cc(c(c(c1)Cl)C2CC2C(=O)O)Cl PS-7709 CCC(=O)c1ccc(c(c1)Br)F PS-7710 c1c(c(c(nc1Cl)Cl)N)C(F)(F)F PS-7711 c1ccc2c(c1)c(cs2)C(=N)N.O.Cl PS-7712 CC(=O)c1ccc(cc1)c2ccc(cc2)Cl PS-7713 CC(=O)c1cccc(c1)c2ccccc2Cl PS-7714 CC(C)C(=O)c1ccc(cc1)C2CCCCC2 PS-7715 c1cc(cnc1)c2nc(on2)C3CCNCC3 PS-7716 CCCCc1nnc(o1)c2ccc(cc2)C=O PS-7717 CCCc1c(cnn1c2ccccc2)C(=O)O PS-7718 C[C@H](c1ccc2cc(ccc2c1)OC)C(=O)O PS-7719 COc1ccc(cc1C(=O)O)S(=O)(=O)C PS-7720 c1cc(ccc1COc2ccc(cc2)C=O)F PS-7721 CC(C)(C)c1ccc(cc1)C(=O)C(F)(F)F PS-7722 Cc1cncc(n1)Oc2cccc(c2)C(=O)O PS-7723 Cc1cncc(n1)Oc2ccc(cc2)C(=O)O PS-7724 c1c(cc(cc1C(F)(F)F)O)C(F)(F)F PS-7725 c1c(cc(c(c1C(F)(F)F)N)Cl)Cl PS-7726 COc1cc2c(cc1OC)CNCC2.Cl PS-7727 c1cc(c(cc1C(F)(F)F)N)S.Cl PS-7728 CC(C)(C)c1ccc(cc1)c2cc(n(n2)C)N PS-7729 CC(C)(C)c1cc(nc(n1)c2ccccn2)O PS-7730 CC(C)(C)OC(=O)N1CC(=O)C[C@H]1C(=O)O PS-7731 c1ccc2c(c1)cc([nH]2)c3ccc(c(c3)F)F PS-7732 c1cc2c(cc1OC(F)(F)F)c(ccn2)O PS-7733 c1cc(c(cc1C(F)(F)F)N)C(F)(F)F PS-7734 c1cc(c(cc1N)C(F)(F)F)C(F)(F)F PS-7735 c1c(cc(cc1C(F)(F)F)N)C(F)(F)F PS-7736 CCCCCc1c(cncn1)Br PS-7737 CCCCOc1ccc(cc1)Br PS-7738 CC(C)(C)c1ccc(c(c1)Br)O PS-7739 Cc1cc(ccc1Br)C(=O)OC PS-7740 c1cc(cc(c1)I)C#N PS-7741 c1cc(ccc1C#N)I PS-7742 c1ccc(c(c1)C#N)I PS-7743 c1c(nc2c(nc(nc2n1)N)N)CO.Cl PS-7744 CN(C)c1cc(nc(n1)N(C)C)C(=O)O.O PS-7745 COC(=O)c1cccc(c1)Oc2ccccc2 PS-7746 COc1ccc(cc1)c2ccccc2C(=O)O PS-7747 CCOC(=O)C(=O)c1ccc2ccccc2c1 PS-7748 CCOC(=O)C(=O)c1cccc2c1cccc2 PS-7749 c1cn(c(=O)[nH]c1=O)[C@H]2C[C@@H]([C@H](O2)CO)O PS-7750 c1cc(ccc1c2cc[nH]n2)OC(F)(F)F PS-7751 c1ccc(cc1)N2C(=O)CC(=N2)C(F)(F)F PS-7752 Cc1ccc2c(cc(c(c2n1)O)Cl)Cl PS-7753 COc1ccc2c(c1)cc(nc2Cl)Cl PS-7754 c1ccc2c(c1)cc([nH]2)c3ccc(cc3)Cl PS-7755 CCCOc1ccc(cc1N)c2ccccc2 PS-7756 c1ccc(c(c1)c2nc3ccccc3s2)O PS-7757 Cc1ccc(cc1)Oc2cccc(c2C#N)F PS-7758 CC1=C([C@@H](C(=O)N1)CC(=O)OC)C(=O)OC PS-7759 [Li+].c1ccc(c(c1)CN2CCOCC2)C(=O)[O-] PS-7760 c1c(cc(c(c1C=O)F)Cl)C(F)(F)F PS-7761 CC(C)Nc1ccc(cc1)Nc2ccccc2 PS-7762 CCOC(=O)c1cccc(c1)c2ccccc2 PS-7763 COC(c1ccccc1)C(=O)c2ccccc2 PS-7764 c1ccc(cc1)C(=O)C=Cc2ccc(cc2)F PS-7765 c1cc(cc(c1)c2cccc(c2)C(=O)O)C=O PS-7766 c1ccc(c(c1)C=O)c2cccc(c2)C(=O)O PS-7767 Cc1c(c(n[nH]1)C)CCNC.Cl.Cl PS-7768 c1cc(c(c(c1C(=O)O)F)F)C(F)(F)F PS-7769 c1cc(c(nc1)Br)C(F)(F)F PS-7770 c1cc(c(nc1)C(F)(F)F)Br PS-7771 c1cnc(cc1Br)C(F)(F)F PS-7772 Cc1ccc(cc1)CC2CCNCC2.Cl PS-7773 c1ccc(cc1)C(=O)C2CCNCC2.Cl PS-7774 c1cc(ncc1C(=N)N)C(F)(F)F.Cl PS-7775 c1cc(cc(c1)S(=O)(=O)C(F)(F)F)N PS-7776 c1cc(ccc1N)S(=O)(=O)C(F)(F)F PS-7777 c1cc(cc(c1)S(=O)(=O)N)C(F)(F)F PS-7778 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)N PS-7779 Cc1cc2cn(nc2cc1Br)C PS-7780 Cc1cc(cc2c1nn(c2)C)Br PS-7781 Cc1cc2c(cc1Br)cn(n2)C PS-7782 Cc1c(ccc2c1cn(n2)C)Br PS-7783 Cc1ccc2c(c1Br)cn(n2)C PS-7784 c1cc2c(cc1Br)CCC(=O)C2 PS-7785 c1ccc2c(c1)c(ccc2Br)F PS-7786 c1cc(c(cc1C=O)Cl)OC(F)(F)F PS-7787 c1cc(c(cc1C(=O)O)C(F)(F)F)Cl PS-7788 c1cc(c(c(c1)C(F)(F)F)Cl)C(=O)O PS-7789 c1c(cc(cc1C(F)(F)F)Cl)C(=O)O PS-7790 CC(=O)c1ccc(c(c1F)C(F)(F)F)F PS-7791 c1cc(c(cc1C(=O)O)OC(F)(F)F)F PS-7792 c1cc(c(c(c1)OC(F)(F)F)F)C(=O)O PS-7793 CC(C)(C#N)c1ccc(cc1)Br PS-7794 c1cc2c(ccnc2c(c1)Br)O PS-7795 c1cc(cc(c1)N)c2cccc(c2)F.Cl PS-7796 c1cc(c(cc1Cl)C(=O)N)C(F)(F)F PS-7797 c1ccc(cc1)COc2ccc3cc[nH]c3c2 PS-7798 c1ccc(cc1)COc2cccc3c2cc[nH]3 PS-7799 c1cc(ncc1C(=O)O)OC2CCOCC2 PS-7800 c1cc(cc(c1)Br)c2cc[nH]n2 PS-7801 c1cc(ccc1c2cc[nH]n2)Br PS-7802 c1cc(ccc1n2ccnc2)Br PS-7803 c1ccc(c(c1)n2cccn2)Br PS-7804 c1cc(ccc1OC(F)F)Br PS-7805 c1cc(cc(c1)Br)OC(F)F PS-7806 c1ccc(c(c1)OC(F)F)Br PS-7807 c1cnc(cc1I)F PS-7808 c1cc(ncc1I)F PS-7809 c1cc(c(nc1)F)I PS-7810 c1c(cncc1I)F PS-7811 c1cncc(c1I)F PS-7812 CC(=O)c1ccc(c(c1)C(F)(F)F)Cl PS-7813 CC(=O)c1cc(ccc1Cl)C(F)(F)F PS-7814 Cc1cncc(c1Br)C.Cl PS-7815 Cc1ccc(c(c1)Br)N.Cl PS-7816 Cc1cc(cc(c1)Br)N.Cl PS-7817 c1cc(cc(c1)Br)CN.Cl PS-7818 c1cc(ccc1CN)Br.Cl PS-7819 CC(C)(C)c1cc(c(c(c1)O)O)C(C)(C)C PS-7820 CC(C)(C)c1cc(c(cc1O)O)C(C)(C)C PS-7821 CC(C)(C)c1cc(c(cc1O)C(C)(C)C)O PS-7822 c1ccc(c(c1)c2ccc3cccnc3n2)O PS-7823 c1cc(cc(c1)SC(F)(F)F)C(=O)O PS-7824 c1ccc(c(c1)C(=O)O)SC(F)(F)F PS-7825 c1cc(ccc1C(=O)O)SC(F)(F)F PS-7826 c1cc(cc(c1)OC(C(F)F)(F)F)C=O PS-7827 c1cc(ccc1C=O)OC(C(F)F)(F)F PS-7828 c1cc(c(cc1CC(=O)O)C(F)(F)F)F PS-7829 c1cc(c(cc1F)C(F)(F)F)CC(=O)O PS-7830 c1cc(c(c(c1)F)CC(=O)O)C(F)(F)F PS-7831 c1cc(c(cc1CC(=O)O)F)C(F)(F)F PS-7832 c1cc(c(cc1C(F)(F)F)CC(=O)O)F PS-7833 c1cc(c(c(c1)C(F)(F)F)F)CC(=O)O PS-7834 c1cc(c(c2c1[nH]c(n2)C(F)(F)F)F)F PS-7835 Cc1ccc2cc(ccc2n1)Br PS-7836 Cc1c(ccc2c1nccc2)Br PS-7837 Cc1cncc2c1c(ccc2)Br PS-7838 c1cc2c(cccc2Br)c(c1)N PS-7839 c1cc(cc2c1cc(cc2)Br)N PS-7840 CS(=O)(=O)c1cccc(c1)CN.Cl PS-7841 CS(=O)(=O)c1ccc(cc1)CN.Cl PS-7842 c1cc(c(cc1C#N)Cl)OC(F)(F)F PS-7843 Cc1cc(cc(c1O)Cl)Br PS-7844 COc1cc(ccc1Cl)Br PS-7845 COc1ccc(c(c1)Br)Cl PS-7846 COc1ccc(c(c1)Cl)Br PS-7847 COc1cc(ccc1Br)Cl PS-7848 COc1ccc(cc1Br)Cl PS-7849 CSCc1cccc(c1N)C(F)(F)F PS-7850 c1cc(c(c(c1)OC(F)(F)F)N)C(=O)O PS-7851 c1cc(c(cc1C(=O)O)OC(F)(F)F)N PS-7852 c1cc(c(cc1OC(F)(F)F)C(=O)O)N PS-7853 Cc1c(ccc(c1Cl)Br)N PS-7854 Cc1cc(cc(c1N)Cl)Br PS-7855 C[C@H](c1ccc(cc1)CC(C)C)C(=O)OC PS-7856 c1ccc(cc1)c2cc3ccccc3nc2N PS-7857 c1ccc(c(c1)C(F)(F)F)NC(=S)N PS-7858 Cc1ccc(cc1)SC(=O)C(F)(F)F PS-7859 c1cnc(cn1)c2nc(on2)CCC(=O)O PS-7860 CCC(=O)c1cc(cc(c1)F)C(F)(F)F PS-7861 CCC(=O)c1cc(ccc1F)C(F)(F)F PS-7862 CCC(=O)c1ccc(cc1F)C(F)(F)F PS-7863 CCC(=O)c1cccc(c1F)C(F)(F)F PS-7864 CCC(=O)c1ccc(c(c1)C(F)(F)F)F PS-7865 CCC(=O)c1ccc(c(c1)F)C(F)(F)F PS-7866 COC(=O)c1ccc(cc1)OC(F)(F)F PS-7867 COC(=O)c1cccc(c1)OC(F)(F)F PS-7868 COC(=O)c1ccccc1OC(F)(F)F PS-7869 COc1ccc(cc1C=O)OC(F)(F)F PS-7870 COc1ccc(cc1OC(F)(F)F)C=O PS-7871 Cc1cc(ccc1C(=O)O)OC(F)(F)F PS-7872 c1cc(cc(c1)OC(F)(F)F)CC(=O)O PS-7873 c1ccc(c(c1)CC(=O)O)OC(F)(F)F PS-7874 c1cc(ccc1CC(=O)O)OC(F)(F)F PS-7875 c1ccc(c(c1)O)I PS-7876 c1cc(cc(c1)I)O PS-7877 Cc1ccccc1c2ccccc2N.Cl PS-7878 Cc1ccccc1c2ccc(cc2)N.Cl PS-7879 c1cc(ccc1N)Oc2ccc(cc2)Cl PS-7880 c1ccc(c(c1)Oc2ccc(cc2)N)Cl PS-7881 c1cc(c(cc1C(F)(F)F)CC#N)Cl PS-7882 c1cc(c(cc1Br)Cl)C=O PS-7883 c1cc(c(cc1Cl)C=O)Br PS-7884 c1cc(c(cc1Br)C=O)Cl PS-7885 CCOC(=O)C(=Cc1ccc(cc1)F)C#N PS-7886 CN(C)Cc1ccccc1OC(F)(F)F PS-7887 COC(=O)c1ccc(o1)Oc2cccnc2 PS-7888 COc1ccc(cc1)c2c(nco2)C(=O)O PS-7889 c1cc(c(c(c1)OC(F)(F)F)F)CC#N PS-7890 CCOC(=O)c1cc(cc(c1)Cl)Cl PS-7891 c1cc(c(c(c1)Br)F)C(=O)O PS-7892 c1cc(c(cc1C(=O)O)F)Br PS-7893 c1cc(c(c(c1)F)Br)C(=O)O PS-7894 c1cc(c(cc1F)Br)C(=O)O PS-7895 c1cc(c(cc1C(=O)O)Br)F PS-7896 c1cc(c(cc1Br)C(=O)O)F PS-7897 c1cc(c(cc1Br)F)C(=O)O PS-7898 c1c(cc(cc1F)Br)C(=O)O PS-7899 c1cc(c(c(c1)Br)C(=O)O)F PS-7900 CC(C)(C)c1cc(cc(c1)C(C)(C)C)C=O PS-7901 c1ccc(cc1)[C@@H](C2CCCCC2)C(=O)O PS-7902 C=CCn1c(n[nH]c1=S)c2ccccn2 PS-7903 CSc1nc(cc(n1)O)c2ccccc2 PS-7904 c1ccc(cc1)C(=O)c2cc(cc(c2)F)F PS-7905 c1ccc(cc1)C(=O)c2cc(ccc2F)F PS-7906 c1ccc(c(c1)C(=O)c2ccc(cc2)F)F PS-7907 CC(=O)Nc1ccc(cc1C(F)(F)F)N PS-7908 CC(=O)Nc1ccc(cc1N)C(F)(F)F PS-7909 c1cc(c(cc1/C=N/O)Br)F PS-7910 c1cc(c(c(c1)Br)C(=O)N)F PS-7911 c1cc(c(cc1Br)F)C(=O)N PS-7912 c1cc(c(cc1C(=O)N)Br)F PS-7913 c1cc(c(cc1Br)C(=O)N)F PS-7914 c1cc(c(cc1F)C(=O)N)Br PS-7915 c1cncc(c1Cl)C(F)(F)F.Cl PS-7916 c1cc(c(c(c1C#N)F)F)Br PS-7917 c1ccc(c(c1)CC#N)SC(F)(F)F PS-7919 Cc1cc(ccc1Br)SC PS-7920 c1cc(c(cc1C=CC(=O)O)Cl)Cl PS-7921 CC(=O)c1ccc(cc1F)Br PS-7922 CC(=O)c1cccc(c1F)Br PS-7923 c1c(c(nc(n1)Cl)Cl)C(F)(F)F PS-7924 c1ccc(cc1)C(=O)c2ccc(cc2)Cl PS-7925 c1cc(c(cc1Br)C#N)Cl PS-7926 c1c(cc(cc1Cl)Br)C#N PS-7927 c1cc(c(cc1Cl)C#N)Br PS-7928 Cc1c(c(=O)n(n1C)c2ccccc2)C=O PS-7929 c1ccc(cc1)Oc2cc(ccc2F)C=O PS-7930 c1cc(cc(c1)C(=O)O)c2cccc(c2)F PS-7931 c1ccc(c(c1)c2cccc(c2)F)C(=O)O PS-7932 c1c(cc(nc1Cl)Cl)C(F)(F)F PS-7933 C[C@@H](C12CC3CC(C1)CC(C3)C2)N.Cl PS-7934 CCOC(=O)[C@@H](c1ccccc1)N.Cl PS-7935 c1ccc(cc1)[C@@H](CC(=O)O)CN.Cl PS-7936 c1cc(ncc1Cl)CN.Cl.Cl PS-7937 c1ccc(cc1)Oc2ccc(cn2)C(=O)O PS-7938 CC(C)(C)N1CCNCC1.Cl.Cl PS-7939 c1cc(nc(c1)C(F)(F)F)C(F)(F)F PS-7940 c1cc(c(nc1)C(F)(F)F)C(F)(F)F PS-7941 c1c(cncc1C(F)(F)F)C(F)(F)F PS-7942 CC(C)Oc1ccccc1Br PS-7943 Cc1cc(cc(c1OC)C)Br PS-7944 Cc1cccc(c1Br)C(=O)O PS-7945 Cc1cc(ccc1Br)C(=O)O PS-7946 Cc1cccc(c1C(=O)O)Br PS-7947 Cc1cc(ccc1C(=O)O)Br PS-7948 Cc1c(cccc1Br)C(=O)O PS-7949 Cc1ccc(cc1C(=O)O)Br PS-7950 Cc1ccc(c(c1)C(=O)O)Br PS-7951 c1c(c(cc(c1Br)F)N)C#N PS-7952 c1cc(c(c(c1)Cl)C(F)(F)F)Cl PS-7953 C1C2CC3CC1CC(C2)(C3)C(=N)N.Cl PS-7954 CC(=O)N(C)c1cccc(c1)CN.Cl PS-7955 c1cc2c(cc1F)c(c[nH]2)CCN.Cl PS-7956 c1c(cc(c(c1O)F)Cl)C(F)(F)F PS-7957 Cc1cccc(c1C)Oc2c(cccn2)N PS-7958 c1ccc(cc1)CC(=O)c2ccc(cc2)F PS-7959 c1ccc(cc1)OC(=O)c2ccccc2O PS-7960 c1ccc(cc1)Oc2ccc(cc2)C(=O)O PS-7961 CCOC(=O)C(=O)c1ccc(c(c1)F)F PS-7962 c1cc(c(cc1c2ccno2)Cl)Cl PS-7963 Cc1cc(c(cc1F)Br)C#N PS-7964 c1cc(c(cc1F)CC#N)Br PS-7965 c1cc(c(c(c1)Br)F)CC#N PS-7966 c1cc(c(cc1Br)F)CC#N PS-7967 c1c(cc(cc1F)Br)CC#N PS-7968 c1ccc(cc1)OC2CCNCC2.Cl PS-7969 c1cc(ccc1N)OC(F)(F)F.Cl PS-7970 c1ccc(cc1)Oc2cccc(c2C#N)F PS-7971 c1ccc2c(c1)c(cc(n2)C(F)(F)F)O PS-7972 c1ccc(cc1)[C@@H](C#N)C(=O)C(F)(F)F PS-7973 CN1C2CCC1CC(C2)N.Cl.Cl PS-7974 CC(C)Cc1ccc(cc1)Br PS-7975 c1cc2c(ccs2)cc1Br PS-7976 c1cc2c(ccs2)c(c1)Br PS-7977 c1cc(c(cc1Cl)Cl)c2cc[nH]n2 PS-7978 COC(=O)c1ccc2nccn2c1.Cl PS-7980 c1cc(ncc1C(F)(F)F)CN.Cl PS-7981 c1cc(c(nc1)CN)C(F)(F)F.Cl PS-7982 Cc1ccccc1NCCc2ccccn2 PS-7983 COc1cccc(c1)c2cccc(c2)C=O PS-7984 Cc1ccc(cc1)C=CC(=O)c2ccco2 PS-7985 COc1ccccc1C(=O)c2ccccc2 PS-7986 COc1ccc(cc1)C(=O)c2ccccc2 PS-7987 CCOC(=O)c1nc(cc(n1)OC)OC PS-7988 COc1cc(cc(c1OC)OC)C(=O)O PS-7989 COC(=O)c1ccc(c(c1)F)C(=O)OC PS-7990 c1ccc(c(c1)c2cc[nH]n2)C(F)(F)F PS-7991 c1ccc(c(c1)C(F)(F)F)n2ccnc2 PS-7992 c1cc(cc(c1)n2ccnc2)C(F)(F)F PS-7993 c1cc(ccc1OC(C(F)F)(F)F)F PS-7994 Cc1ccc(cc1C)CNC2CC2.Cl PS-7995 Cc1ccc(c(c1)C)CNC2CC2.Cl PS-7996 Cc1cccc(c1C)CNC2CC2.Cl PS-7997 c1cc(sc1)c2ccc(cc2)N.Cl PS-7998 c1ccc2c(c1)ncn2CCCN.Cl PS-7999 c1cc2c(cc1N)c(c[nH]2)C(=O)N.Cl PS-8000 c1cc(c(cc1N)Cl)OC(F)(F)F PS-8001 c1cc(c(cc1OC(F)(F)F)Cl)N PS-8002 c1c(cc(c(c1N)O)Cl)C(F)(F)F PS-8003 c1ccc2c(c1)cc([nH]2)c3ccc(cc3)F PS-8004 CC(C)(C)OC(=O)Nc1cccc(c1)F PS-8005 CC(C)(C)OC(=O)Nc1ccc(cc1)F PS-8006 COc1ccc(cc1)C(C(C(=O)O)N)O PS-8007 Cc1ccc2c(c1)c(c[nH]2)CCN.Cl PS-8008 c1cc(c(cc1Cl)C2CCCCC2)O PS-8009 c1cc(c(cc1C(F)(F)F)CO)Cl PS-8010 c1cc(c(cc1CO)Cl)C(F)(F)F PS-8011 c1cc(c(cc1Cl)CO)C(F)(F)F PS-8012 c1cc(c(cc1CO)C(F)(F)F)Cl PS-8013 COc1ccc(cc1)/C=C/c2ccccc2 PS-8014 CC(=O)c1ccc(cc1)Cc2ccccc2 PS-8015 c1cc(ccc1C(=O)CCCC(=O)O)F PS-8016 c1cc(c(c(c1)OC(F)(F)F)F)CO PS-8017 c1cc(cc(c1)OC(C(F)F)(F)F)O PS-8018 Cc1c[nH]c2c1cc(cc2)Br PS-8019 Cc1ccc(o1)c2ccccc2N.Cl PS-8020 Cc1ccc(o1)c2ccc(cc2)N.Cl PS-8021 c1cc(c(cc1Cl)S(=O)(=O)N)F PS-8022 c1cc(c(c(c1)Cl)F)S(=O)(=O)N PS-8023 c1cc(c(cc1C(F)(F)F)CN)Cl PS-8024 CC1=Nc2ccc3ccccc3c2C1(C)C PS-8025 c1cc(nnc1C(=O)O)N2CCOCC2 PS-8026 c1cc(cc(c1)OC(C(F)F)(F)F)N PS-8027 c1ccc(c(c1)N)OC(C(F)F)(F)F PS-8028 c1cc(ccc1N)OC(C(F)F)(F)F PS-8029 c1c(c(cc(c1Cl)Cl)F)C(=O)O PS-8030 c1cc(c(cc1Cl)C(F)(F)F)C=O PS-8031 c1cc(c(cc1C=O)C(F)(F)F)Cl PS-8032 c1cc(c(c(c1)Cl)C=O)C(F)(F)F PS-8033 c1cc(c(cc1C(F)(F)F)C=O)Cl PS-8034 c1cc(c(c(c1)C(F)(F)F)Cl)C=O PS-8035 Cc1cnccc1Br.Cl PS-8036 CC(C)(C)c1ccc(cc1OC)C(=O)O PS-8037 c1cc(ccc1CO)SC(F)(F)F PS-8038 Cc1cc(no1)c2c(c(no2)C)C(=O)O PS-8039 c1c(cc(cc1F)F)c2c(c[nH]n2)C=O PS-8040 c1cc(c(cc1OC(F)(F)F)C=O)F PS-8041 c1cc(c(cc1C=O)OC(F)(F)F)F PS-8042 c1cc(c(c(c1)OC(F)(F)F)F)C=O PS-8043 c1cc(c(cc1C(=O)O)F)C(F)(F)F PS-8044 c1cc(c(cc1C(=O)O)C(F)(F)F)F PS-8045 c1c(cc(cc1C(F)(F)F)F)C(=O)O PS-8046 c1cc(c(cc1C(F)(F)F)F)C(=O)O PS-8047 c1cc(c(c(c1)F)C(=O)O)C(F)(F)F PS-8048 c1cc(c(cc1F)C(F)(F)F)C(=O)O PS-8049 c1cc(c(c(c1)C(F)(F)F)F)C(=O)O PS-8050 c1cc(c(cc1C(F)(F)F)C(=O)O)F PS-8051 c1ccc2c(c1)ccc(n2)Br PS-8052 c1cc2ccc(cc2nc1)Br PS-8053 CS(=O)(=O)c1ccccc1N.Cl PS-8054 CS(=O)(=O)c1cccc(c1)N.Cl PS-8055 CS(=O)(=O)c1ccc(cc1)N.Cl PS-8056 c1cc(c(cc1Cl)S(=O)(=O)O)N PS-8057 c1cc(c(cc1C(=O)CN)F)F.Cl PS-8058 c1cc(c(cc1F)F)C(=O)CN.Cl PS-8059 c1cc(c(cc1O)Cl)Br PS-8060 c1cc(c(cc1Br)O)Cl PS-8061 c1cc(c(cc1Br)Cl)O PS-8062 c1cc(c(cc1O)Br)Cl PS-8063 c1cc(ccc1CN)SC(F)(F)F PS-8064 c1c(cc(cc1C(F)(F)F)F)C(=O)N PS-8065 c1cc(c(cc1C(F)(F)F)F)C(=O)N PS-8066 c1ccc2cc(ccc2c1)Br PS-8067 C=Cc1cc(ccc1Cl)C(F)(F)F PS-8068 c1cc(c(cc1Cl)C=O)OC(F)F PS-8069 Cc1c(ccc(n1)Cl)Br PS-8070 Cc1cc(ncc1Br)Cl PS-8071 Cc1cc(cnc1Cl)Br PS-8072 c1ccc(cc1)c2[nH]cc(n2)C(=O)O.O PS-8073 Cc1cc(ccc1CO)OC(F)(F)F PS-8074 CC(=O)c1ccc(cc1C(F)(F)F)F PS-8075 CC(=O)c1cc(ccc1F)C(F)(F)F PS-8076 CC(=O)c1ccc(cc1F)C(F)(F)F PS-8077 CC(=O)c1cccc(c1F)C(F)(F)F PS-8078 CC(=O)c1ccc(c(c1)C(F)(F)F)F PS-8079 CC(=O)c1c(cccc1F)C(F)(F)F PS-8080 c1cc(c(c(c1)OC(F)(F)F)O)C=O PS-8081 c1cc(c(cc1OC(F)(F)F)C=O)O PS-8082 c1ccc(c(c1)C(=O)O)OC(F)(F)F PS-8083 c1cc(c(cc1O)C(F)(F)F)C(=O)O PS-8086 c1cc2c(c[nH]c2nc1)N.Cl.Cl PS-8087 c1cncc2c1[nH]cc2N.Cl.Cl PS-8088 c1c(cc(c(c1N)O)F)Br PS-8089 c1cc(c(c(c1N)O)Br)F PS-8090 c1cnc(cn1)I PS-8091 c1csc2c1sc(c2)CN.Cl PS-8092 Cc1ccc2cc(c(nc2c1)Cl)C=O PS-8093 c1cc(c(cc1C#N)C(F)(F)F)Cl PS-8094 c1cc(c(cc1C(F)(F)F)C#N)Cl PS-8095 c1cc(c(cc1C(F)(F)F)Cl)C#N PS-8096 c1c(cc(cc1C(F)(F)F)Cl)C#N PS-8097 c1cc(c(cc1Cl)C(F)(F)F)C#N PS-8098 Cc1ccc(cc1Cl)Br PS-8099 Cc1cc(ccc1Cl)Br PS-8100 c1ccc(cc1)c2c(=O)nc([nH]n2)S PS-8101 CCNc1ccc(cc1)OC(F)(F)F PS-8102 CCNc1ccccc1OC(F)(F)F PS-8103 C[C@@H](c1ccc(cc1)OC(F)(F)F)N PS-8104 c1cc(ccc1/C=N/O)OC(F)(F)F PS-8105 c1cc(c(cc1N)C(F)(F)F)C(=O)O PS-8106 c1cc(c(c(c1)C(F)(F)F)N)C(=O)O PS-8107 c1cc(c(cc1C(F)(F)F)C(=O)O)N PS-8108 c1cc(c(c(c1)N)C(=O)O)C(F)(F)F PS-8109 c1cc(c(cc1C(F)(F)F)N)C(=O)O PS-8110 c1c(cc(cc1C(F)(F)F)N)C(=O)O PS-8111 c1cc(c(cc1C#N)OC(F)(F)F)F PS-8112 c1cc(c(cc1C#N)F)OC(F)(F)F PS-8113 c1c(c(cc(c1F)Br)N)N PS-8114 c1cc(c(c(c1N)N)F)Br PS-8115 c1c(cc(c(c1N)N)F)Br PS-8116 c1cc(c(c(c1N)N)Br)F PS-8117 c1c(cc(c(c1N)N)Br)F PS-8118 COc1ccc(c(c1)F)Br PS-8119 COc1cc(ccc1F)Br PS-8120 COc1cc(cc(c1)Br)F PS-8121 COc1ccc(cc1Br)F PS-8122 COc1ccc(c(c1)Br)F PS-8123 COc1ccc(cc1F)Br PS-8124 c1cc(c(cc1F)Br)CO PS-8125 c1cc(c(cc1Br)CO)F PS-8126 c1cc(c(cc1Br)F)CO PS-8127 c1cc(c(cc1CO)Br)F PS-8128 c1c(cc(cc1F)Br)CO PS-8129 c1cc(c(cc1F)CO)Br PS-8130 c1ccc(cc1)Oc2ccc(cc2)Cl PS-8132 c1cc(ccc1Cc2ccc(cc2)F)F PS-8133 CC[C@@H](c1ccc(cc1)C(F)(F)F)O PS-8134 CC[C@@H](c1ccccc1C(F)(F)F)O PS-8135 Cc1nc(on1)c2ccccc2C(=O)O PS-8136 Cc1nc(no1)c2ccc(cc2)C(=O)O PS-8137 Cc1nc(on1)c2cccc(c2)C(=O)O PS-8138 Cc1cc(cc(c1)OC(F)(F)F)C=O PS-8139 Cc1cc(ccc1C=O)OC(F)(F)F PS-8140 CC(=O)c1cccc(c1)OC(F)(F)F PS-8141 CC(=O)c1ccccc1OC(F)(F)F PS-8142 COC(=O)c1cccc(c1)C(F)(F)F PS-8143 COC(=O)c1ccc(cc1)C(F)(F)F PS-8144 COC(=O)c1ccccc1C(F)(F)F PS-8145 COc1ccc(c(c1)C(F)(F)F)C=O PS-8146 COc1ccc(cc1C(F)(F)F)C=O PS-8147 COc1cc(ccc1C=O)C(F)(F)F PS-8148 Cc1c(cccc1C(F)(F)F)C(=O)O PS-8149 Cc1ccc(cc1C(F)(F)F)C(=O)O PS-8150 Cc1cc(cc(c1)C(F)(F)F)C(=O)O PS-8151 Cc1ccc(cc1C(=O)O)C(F)(F)F PS-8152 c1ccc(c(c1)CC(=O)O)C(F)(F)F PS-8153 c1cc(cc(c1)C(F)(F)F)CC(=O)O PS-8154 C#Cc1ccc(c(c1)F)OC(F)(F)F PS-8155 c1c([nH]nc1C(F)(F)F)C(F)(F)F PS-8156 Cc1cc(c(cc1N)Br)F PS-8157 Cc1cc(c(cc1F)N)Br PS-8158 Cc1cc(cc(c1N)Br)F PS-8159 c1c(cnc(c1C=O)F)Br PS-8160 c1cc(nc(c1F)C=O)Br PS-8161 CNCCc1ccc(c(c1)O)O.Cl PS-8162 Cc1ccc(cc1C(F)(F)F)C(=O)N PS-8163 c1cc(c(c(c1)C(F)(F)F)F)CC#N PS-8164 c1cc(c(cc1CC#N)F)C(F)(F)F PS-8165 c1cc(c(cc1CC#N)C(F)(F)F)F PS-8166 c1c(cc(cc1C(F)(F)F)F)CC#N PS-8167 CCC(=O)c1ccc(c(c1)Cl)Cl PS-8168 c1cc(c(c(c1)F)Br)C=O PS-8170 c1cc(c(cc1Br)C=O)F PS-8171 c1cc(c(cc1F)C=O)Br PS-8172 c1cc(c(cc1F)Br)C=O PS-8173 c1cc(c(cc1C=O)Br)F PS-8174 c1cc(c(cc1Br)F)C=O PS-8175 c1c(cc(cc1F)Br)C=O PS-8176 c1cc(c(cc1C=O)F)Br PS-8177 c1ccc(cc1)SCC(=N)N.Cl PS-8178 CCOC(=O)c1ccc(c(c1)Cl)F PS-8179 CCOC(=O)c1ccc(cc1F)Cl PS-8180 CCOC(=O)c1ccc(cc1Cl)F PS-8181 Cc1ccc(c(c1Cl)CC(=O)O)F PS-8182 Cc1ccc2c(c1)C(CCC2(C)C)(C)C PS-8183 c1ccc(cc1)COc2ccc(cc2)F PS-8184 c1ccc(c(c1)C(=O)O)S(=O)(=O)O PS-8185 CCC(=O)c1cccc(c1)C(F)(F)F PS-8186 CCC(=O)c1ccccc1C(F)(F)F PS-8187 c1cc(ccc1CCC=O)C(F)(F)F PS-8188 c1cc(cc(c1)OC(F)F)CC(=O)O PS-8189 c1cc(c(cc1C#N)OC(F)(F)F)N PS-8190 c1c(c(cc(c1F)F)F)C=CC(=O)O PS-8191 CCOc1ccc(nc1)Br PS-8192 COC(=O)Cc1cccc(c1)N.Cl PS-8193 COC(=O)c1ccc(cc1)CN.Cl PS-8194 COC(=O)c1ccccc1CN.Cl PS-8195 COC(=O)c1cccc(c1)CN.Cl PS-8196 COc1cc(cnc1Cl)C(=O)OC PS-8197 c1ccc(cc1)COc2ccnc(c2)O PS-8198 c1cnccc1c2ncc(cn2)C(=O)O PS-8199 Cc1cc(ccc1C#N)OC(F)(F)F PS-8200 c1cc(ccc1CC#N)OC(F)(F)F PS-8201 c1cc(cc(c1)OC(F)(F)F)CC#N PS-8202 c1ccc(c(c1)CC#N)OC(F)(F)F PS-8203 Cc1cc(cc(c1O)C)Br PS-8204 Cc1cc(cc(c1Br)C)O PS-8205 Cc1cc(ccc1Br)OC PS-8206 Cc1ccc(c(c1)Br)OC PS-8207 C=Cc1ccc(cc1Br)F PS-8208 C=Cc1cccc(c1F)Br PS-8209 C=Cc1ccc(cc1F)Br PS-8210 CC(=O)Nc1cccc(c1)CN.Cl PS-8211 c1ccc2c(c1)cccc2CCC(=O)O PS-8212 c1ccc(cc1)COc2ccc(cc2)O PS-8213 c1cc(c(cc1Br)C#N)F PS-8214 c1c(cc(cc1F)Br)C#N PS-8215 c1cc(c(cc1F)Br)C#N PS-8216 c1cc(c(c(c1)Br)F)C#N PS-8217 c1cc(c(cc1C#N)F)Br PS-8218 c1cc(c(cc1F)C#N)Br PS-8219 c1cc(c(c(c1)Br)C#N)F PS-8220 c1cc(c(cc1Br)F)C#N PS-8221 c1cc(c(cc1C#N)Br)F PS-8222 c1cc(c(c(c1)F)Br)C#N PS-8223 c1ccc2c(c1)c(cs2)CN.Cl PS-8224 c1ccc(cc1)[C@@H]2CNCCO2.Cl PS-8225 c1cnc2c(c1Cl)cc(cc2F)F PS-8226 c1cnc(c(c1C(F)(F)F)F)Cl PS-8227 Cc1ccccc1Oc2ccc(cc2)N PS-8228 Cc1ccc(cc1)Oc2ccc(cc2)N PS-8229 c1cc(cc(c1)C(F)(F)F)CCC#N PS-8230 C1CC1N2CCNCC2.Cl.Cl PS-8231 CC(=O)c1ccccc1Br PS-8232 C#Cc1ccc(cc1F)Br PS-8233 C#Cc1ccc(c(c1)F)Br PS-8234 C#Cc1ccc(cc1Br)F PS-8235 C#Cc1cc(ccc1F)Br PS-8236 c1cc(c(cc1Cl)F)C(F)(F)F PS-8237 c1cc(c(cc1F)Cl)C(F)(F)F PS-8238 CCCCC[C@H]1CC[C@@H](CC1)C(=O)O PS-8239 c1ccc(cc1)Oc2ccc(cc2)C=O PS-8240 c1ccc(cc1)c2cccc(c2)C(=O)O PS-8241 c1ccc(cc1)C(=O)c2ccc(cc2)O PS-8242 COc1c(cnc(n1)OC)C(=O)OC PS-8243 COc1cc(cc(c1O)OC)C(=O)O PS-8244 c1c(c(c(nc1F)N)F)C(F)(F)F PS-8245 c1ccc2c(c1)c(cc(n2)Cl)Cl PS-8246 c1cc2c(ccnc2cc1Cl)Cl PS-8247 c1cc2c(cc1Cl)c(ccn2)Cl PS-8248 c1cc(c(c2c1ccnc2)Cl)Cl PS-8249 c1c(cnc(c1C(F)F)Cl)Cl PS-8250 c1ccc2c(c1)ncn2CCN.Cl PS-8251 C[C@@H](c1ccc(cc1)c2ccccc2)N PS-8252 C1CCN(C1)c2nnn(n2)CC(=O)O PS-8253 CCOC(=O)c1c(cc(nc1O)C)O PS-8254 c1c(cc(c(c1N)C(F)(F)F)F)F PS-8255 c1c(c(cc(c1F)N)F)C(F)(F)F PS-8256 c1cc(cc(c1)Br)C2CC2 PS-8257 C=CCc1cccc(c1)Br PS-8258 c1c(cnc(c1F)CN)Cl.Cl PS-8259 CCCCC(=O)c1ccc(cc1)Cl PS-8260 C1C(=O)N(C(=O)S1)CCN.Cl PS-8261 c1ccc(c(c1)OC(F)(F)F)Cl PS-8262 c1cc(cc(c1)Cl)OC(F)(F)F PS-8263 c1cc(c(cc1O)C(F)(F)F)Cl PS-8264 c1cc(c(cc1C(F)(F)F)Cl)O PS-8265 c1cc(c(cc1C(F)(F)F)O)Cl PS-8266 Cc1ccc(cc1)C(=O)c2ccccc2 PS-8267 Cc1ccccc1C(=O)c2ccccc2 PS-8268 CC(C)(C)OC(=O)c1ccc(cc1)F PS-8269 c1cc(ccc1CCCCC(=O)O)F PS-8270 COC(=O)c1cc(ccc1O)C(=O)O PS-8271 c1cc(c(cc1Cl)F)CN.Cl PS-8272 Cc1ccc(c(c1)C#N)Br PS-8273 Cc1cc(ccc1C#N)Br PS-8274 Cc1ccc(cc1Br)C#N PS-8275 Cc1cc(ccc1Br)C#N PS-8276 c1ccc(c(c1)c2ccco2)N.Cl PS-8277 c1cc(cc(c1)N)c2ccco2.Cl PS-8278 c1cc(c(cc1N)C(F)(F)F)Cl PS-8279 c1cc(c(cc1C(F)(F)F)Cl)N PS-8280 c1cc(c(cc1N)Cl)C(F)(F)F PS-8281 c1cc(c(cc1C(F)(F)F)N)Cl PS-8282 c1cc(c(cc1Cl)C(F)(F)F)N PS-8283 c1cc(ccc1C#N)c2ccc(cc2)O PS-8284 c1cc(c(c(c1)OC(F)(F)F)F)N PS-8285 c1cc(c(cc1OC(F)(F)F)N)F PS-8286 CNc1ccccc1N.Cl.Cl PS-8287 Cc1ccc(c(c1)Cl)C(F)(F)F PS-8288 c1cnccc1Br.Cl PS-8289 c1ccc2cc(ccc2c1)c3cc[nH]n3 PS-8290 c1ccc2c(c1)cccc2c3cc[nH]n3 PS-8291 C[C@@H](C(=O)O)N1CCNCC1.O.O PS-8292 c1cc(ccc1O)SC(F)(F)F PS-8293 c1cc(cc(c1)S)OC(F)(F)F PS-8294 c1cc(ccc1OC(F)(F)F)S PS-8295 c1ccc(c(c1)OC(F)(F)F)S PS-8296 c1c(c(cc(c1N)N)F)C(F)(F)F PS-8297 Cc1cc(ccc1F)OC(F)(F)F PS-8298 COc1ccc(c(c1)C(F)(F)F)F PS-8299 c1cc(c(cc1F)CO)C(F)(F)F PS-8300 c1cc(c(cc1CO)C(F)(F)F)F PS-8301 c1c(cc(cc1C(F)(F)F)F)CO PS-8302 c1cc(c(cc1F)C(F)(F)F)CO PS-8303 c1cc(c(c(c1)F)C(F)(F)F)CO PS-8304 c1cc(c(c(c1)F)CO)C(F)(F)F PS-8305 c1cc(c(cc1C(F)(F)F)CO)F PS-8306 c1cc(c(c(c1)C(F)(F)F)F)CO PS-8307 c1cc(c(cc1CO)F)C(F)(F)F PS-8308 COc1ccc(c(c1)N)Cl.Cl PS-8309 CC1=Nc2ccc(cc2C1(C)C)Cl PS-8310 COC(=O)CC1CCNCC1.Cl PS-8311 COC(=O)c1cscc1N.Cl PS-8312 c1ccc(c(c1)N)SC(F)(F)F PS-8313 c1cc(ccc1N)SC(F)(F)F PS-8314 c1c(cc(cc1F)S(=O)(=O)N)F PS-8315 c1cc(c(cc1S(=O)(=O)N)F)F PS-8316 c1cc(c(cc1F)S(=O)(=O)N)F PS-8317 c1cc(c(cc1F)F)S(=O)(=O)N PS-8318 c1cc(c(c(c1)C(F)(F)F)F)CN PS-8319 c1c(cc(cc1C(F)(F)F)F)CN PS-8320 c1cc(c(c(c1)F)CN)C(F)(F)F PS-8321 c1cc(c(cc1F)C(F)(F)F)CN PS-8322 c1cc(c(cc1CN)F)C(F)(F)F PS-8323 c1cc(c(cc1C(F)(F)F)F)CN PS-8324 c1cc(c(cc1OC(F)(F)F)N)O PS-8325 Cc1csc(n1)NC(=N)N.Cl PS-8326 CCCCCc1ccc(cc1)C(=O)O PS-8327 CC(C)(C)c1ccc(cc1)CC(=O)O PS-8328 c1cc(cc(c1)C(F)(F)F)CS PS-8329 CN(C)c1ccc(c(c1C#N)F)C=O PS-8330 CS(=O)(=O)c1ccc(c(c1)F)F PS-8331 CS(=O)(=O)c1cc(ccc1F)F PS-8332 c1cc(c(cc1OC(F)(F)F)N)N PS-8333 COc1ccccc1OC(F)(F)F PS-8334 c1cc(cc(c1)OC(F)(F)F)CO PS-8335 c1ccc(c(c1)CO)OC(F)(F)F PS-8336 c1cc(ccc1CO)OC(F)(F)F PS-8337 c1cc(c(c(c1)F)C=O)C(F)(F)F PS-8338 c1cc(c(cc1F)C(F)(F)F)C=O PS-8339 c1c(cc(cc1C(F)(F)F)F)C=O PS-8340 c1cc(c(cc1C(F)(F)F)F)C=O PS-8341 c1cc(c(cc1C=O)F)C(F)(F)F PS-8342 c1cc(c(cc1C=O)C(F)(F)F)F PS-8343 c1cc(c(c(c1)C(F)(F)F)F)C=O PS-8344 c1cc(ccc1C(=O)C(F)(F)F)F PS-8345 c1cc(cc(c1)F)C(=O)C(F)(F)F PS-8346 c1(c([nH]c(=O)[nH]c1=O)C(=O)O)F.O PS-8347 c1cnc(c(c1O)F)Br PS-8348 c1c(c(cnc1Br)F)O PS-8349 c1c(c(c(cn1)Br)O)F PS-8350 Cc1ccc2c(c1)c(cc(n2)C)Cl PS-8351 C1CC2(CCNCC2)OC1=O.Cl PS-8352 Cc1cc(ccc1N)OC(F)(F)F PS-8353 c1cc(ccc1N)OCC(F)(F)F PS-8354 c1ccc(c(c1)N)OCC(F)(F)F PS-8355 c1cc(cc(c1)OC(F)(F)F)CN PS-8356 c1ccc(c(c1)CN)OC(F)(F)F PS-8357 COc1ccc(cc1N)C(F)(F)F PS-8358 COc1cc(cc(c1)N)C(F)(F)F PS-8359 COc1ccc(c(c1)C(F)(F)F)N PS-8360 c1c(cnc(c1Br)N)F PS-8361 c1c(cnc(c1N)F)Br PS-8362 c1c(cc(cc1F)Br)O PS-8363 c1cc(c(cc1O)F)Br PS-8364 c1cc(c(c(c1)Br)F)O PS-8365 c1cc(c(cc1F)Br)O PS-8366 c1cc(c(cc1Br)O)F PS-8367 c1cc(c(c(c1)Br)O)F PS-8368 c1cc(c(cc1F)O)Br PS-8369 c1cc(c(cc1O)Br)F PS-8370 c1cc(c(cc1Br)F)O PS-8371 c1ccc(cc1)c2ccnc(n2)Cl PS-8372 CCOC(=O)c1c(cc[nH]1)N.Cl PS-8373 c1cc(c(cc1F)S(=O)(=O)N)N PS-8376 c1cc(ccc1c2ccc(cc2)F)F PS-8377 Cc1ccc(cc1C(F)(F)F)CO PS-8378 Cc1ccc(cc1CO)C(F)(F)F PS-8379 C[C@@H](c1ccccc1C(F)(F)F)O PS-8380 C=Cc1cc(ccc1F)C(F)(F)F PS-8381 C=Cc1cccc(c1F)C(F)(F)F PS-8382 c1cc(ccc1C=O)OC(F)(F)F PS-8383 c1cc(cc(c1)OC(F)(F)F)C=O PS-8384 c1ccc(c(c1)C=O)OC(F)(F)F PS-8385 c1cc(c(cc1C=O)C(F)(F)F)O PS-8386 c1cc(cc(c1)C(F)(F)F)C(=O)O PS-8388 Cc1c(ccc(n1)F)Br PS-8390 Cc1cc(cnc1F)Br PS-8391 Cc1cc(ncc1Br)F PS-8392 Cc1ccc(c(n1)Br)F PS-8393 Cc1cc(cnc1Br)F PS-8394 c1cc(c(cc1Br)F)N PS-8395 c1cc(c(c(c1)F)Br)N PS-8396 c1cc(c(cc1N)Br)F PS-8397 c1cc(c(cc1N)F)Br PS-8398 c1cc(c(cc1Br)N)F PS-8399 c1cc(c(cc1F)N)Br PS-8400 c1cc(c(c(c1)Br)N)F PS-8401 c1cc(c(cc1F)Br)N PS-8402 c1cc(c(c(c1)Br)F)N PS-8403 COc1cc(ccc1O)CN.Cl PS-8404 c1cc(cc(c1)F)C(=O)CN.Cl PS-8405 c1ccc(c(c1)C(=O)CN)F.Cl PS-8406 Cc1cc(ccc1S(=O)(=O)N)F PS-8407 CS(=O)(=O)c1ccc(cc1F)N PS-8408 CS(=O)(=O)c1cc(ccc1F)N PS-8409 CS(=O)(=O)c1ccc(c(c1)N)F PS-8410 C[C@@H](c1ccc(cc1)C(F)(F)F)N PS-8411 C[C@@H](c1cccc(c1)C(F)(F)F)N PS-8412 c1ccnc(c1)c2cc(n[nH]2)C(=O)O PS-8413 c1cc(ccc1C(=O)N)C(F)(F)F PS-8414 c1ccc(c(c1)C(=O)N)C(F)(F)F PS-8415 c1cc(c(cc1C#N)C(F)(F)F)F PS-8416 c1cc(c(c(c1)F)C#N)C(F)(F)F PS-8417 c1cc(c(cc1C#N)F)C(F)(F)F PS-8418 c1cc(c(cc1F)C(F)(F)F)C#N PS-8419 c1c(cc(cc1C(F)(F)F)F)C#N PS-8420 c1cc(c(cc1C(F)(F)F)C#N)F PS-8421 c1cc(c(cc1C(F)(F)F)F)C#N PS-8422 c1cc(c(cc1F)C#N)C(F)(F)F PS-8423 c1cc(c(c(c1)C(F)(F)F)F)C#N PS-8424 c1cc(c(c(c1)F)C(F)(F)F)C#N PS-8425 c1c[nH]c2c1c(c(c(c2F)F)F)F PS-8426 c1cc2nccn2cc1Cl.Cl PS-8427 Cc1ccc(c(c1)F)Br PS-8428 Cc1c(cccc1Br)F PS-8429 c1ccc(cc1)c2ccccc2Cl PS-8430 c1ccc(cc1)c2ccc(cc2)Cl PS-8431 COC(=O)c1ccc(c(c1)F)Cl PS-8432 COC(=O)c1ccc(cc1F)Cl PS-8433 Cc1ccc(c(c1Cl)C(=O)O)F PS-8434 c1cc(c(cc1CC(=O)O)Cl)F PS-8435 c1cc(c(cc1CC(=O)O)F)Cl PS-8436 c1c(cc(cc1F)Cl)CC(=O)O PS-8437 c1cc(c(c(c1)F)NC(=S)N)F PS-8438 c1cc(c(cc1F)NC(=S)N)F PS-8439 c1cc(c(cc1F)F)NC(=S)N PS-8440 c1c(cc(cc1F)F)NC(=S)N PS-8441 c1ccc(cc1)Oc2ccc(cc2)F PS-8442 CC(=O)c1cccc(c1)C(F)(F)F PS-8443 CC(=O)c1ccccc1C(F)(F)F PS-8444 c1ccc(c(c1)C(=O)O)OC(F)F PS-8445 COc1c(ccc(c1C(=O)O)F)F PS-8446 COc1c(ccc(c1F)F)C(=O)O PS-8447 COc1ccnc(c1)Br PS-8448 C1C2CC3CC1CC(C2)C3N.Cl PS-8449 c1ccc(cc1)COCCN.Cl PS-8450 c1cc(cc(c1)C(=O)O)CN.Cl PS-8451 CC(=O)Nc1ccc(cc1F)Cl PS-8452 CC(=O)Nc1ccc(cc1Cl)F PS-8453 c1cc(c(cc1F)Cl)CC(=O)N PS-8454 CCc1cccc2c1nc(cc2O)C PS-8455 Cc1cc(ccc1N)S(=O)(=O)O PS-8456 c1ccc(cc1)Nc2ccc(cc2)F PS-8457 c1ccc(cc1)Nc2cccc(c2)F PS-8458 COC(=O)c1c(ccc(c1F)N)F PS-8459 c1cc(ccc1C#N)OC(F)(F)F PS-8460 c1ccc(c(c1)C#N)OC(F)(F)F PS-8461 c1cc(cc(c1)OC(F)(F)F)C#N PS-8462 CN1CCCC(C1)N.Cl.Cl PS-8463 Cc1ccc(cc1O)Br PS-8464 Cc1cc(ccc1O)Br PS-8465 Cc1ccc(c(c1)Br)O PS-8466 Cc1ccc(c(c1Cl)C(=O)C)F PS-8468 CC(=O)Cc1ccc(cc1Cl)F PS-8469 c1ccc(cc1)Cc2ccc(cc2)F PS-8470 c1ccc(cc1)Oc2ccc(cc2)O PS-8471 c1ccc(cc1)C2(CC2)C(F)(F)F PS-8472 CCOC(=O)c1ccc(c(c1)F)F PS-8473 CCOC(=O)c1ccc(cc1F)F PS-8474 CCOc1ccc(c(c1F)F)C=O PS-8475 Cc1ccc(c(c1F)F)CC(=O)O PS-8476 Cc1ccc(c(c1F)CC(=O)O)F PS-8477 c1cc(c(cc1C#N)C(F)(F)F)N PS-8478 c1cc(c(cc1N)C(F)(F)F)C#N PS-8479 c1cc(c(c(c1)N)C#N)C(F)(F)F PS-8480 c1cc(c(cc1C(F)(F)F)C#N)N PS-8481 c1cc(c(c(c1)C(F)(F)F)N)C#N PS-8482 C#Cc1cccc(c1)OC(F)(F)F PS-8483 C#Cc1ccc(cc1)OC(F)(F)F PS-8484 c1cc(c2c(c1)OC(O2)(F)F)C=O PS-8485 CC(C)(C)c1cccc(c1)N.Cl PS-8486 c1cc2c(cc1CN)CCO2.Cl PS-8487 CCSc1ncc(c(n1)N)CO PS-8489 Cc1c(nc(s1)C)CC(=O)OC PS-8490 CCc1ccc(cc1)S(=O)(=O)N PS-8491 Cc1ccc(cc1)c2ccnc(n2)N PS-8492 Cc1nccc(n1)c2cccc(c2)N PS-8493 c1cncc2c1nc3c(c2)CNCC3 PS-8494 c1ccc(cc1)c2ccc(c(c2)N)O PS-8495 CC(C)(C#C)Oc1ccc(cc1)C#N PS-8496 c1cc(cc(c1)c2cccnc2)CO PS-8497 c1cc(cnc1)c2ccc(cc2)CO PS-8498 CC(C)(C)OC(=O)N1CCC(=O)C1 PS-8499 CC(C)(C)OC(=O)N1CC(C1)C=O PS-8500 Cc1c(cccc1C(F)(F)F)C#N PS-8501 Cc1ccc(c(c1)C(F)(F)F)C#N PS-8502 Cc1ccc(cc1C(F)(F)F)C#N PS-8503 Cc1cc(cc(c1)C(F)(F)F)C#N PS-8504 Cc1ccc(cc1C#N)C(F)(F)F PS-8505 c1ccc(c(c1)CC#N)C(F)(F)F PS-8506 c1cc(cc(c1)C(F)(F)F)CC#N PS-8507 c1ccc(c(c1)C=O)Br PS-8508 c1cc(cc(c1)Br)C=O PS-8509 c1cc(ccc1C=O)Br PS-8510 c1cc2c(cc1Cl)sc(n2)N PS-8511 c1cc(sc1c2cc[nH]n2)Cl PS-8512 Cc1cc(c(c(c1Cl)C)C=O)O PS-8513 COc1cc(c(cc1OC)F)C=O PS-8514 COc1cc(nc(n1)OC)C(=O)O PS-8515 COc1cc(c(nn1)OC)C(=O)O PS-8516 c1cn(cn1)CCN.Cl.Cl PS-8517 CC(C)(C)c1ccc(c(c1)Cl)N PS-8518 c1ccc(cc1)Cc2cccc(c2)N PS-8519 c1cnc(c(c1C(F)(F)F)F)F PS-8520 C=Cc1ccc(cc1)Br PS-8521 c1cnc(nc1C(F)(F)F)Cl PS-8522 c1c(cnc(n1)Cl)C(F)(F)F PS-8523 c1ccc(cc1)c2ccccc2C=O PS-8524 c1ccc(cc1)c2cccc(c2)C=O PS-8525 CCOC(=O)Cc1ccccc1F PS-8526 c1c(cc(c2c1COCO2)C=O)F PS-8527 c1cc(c(cc1C(=O)O)O)C(=O)O PS-8528 COC(=O)[C@@H]1C[C@H](CN1)O.Cl PS-8529 C1COCCN1CC(=O)O.Cl PS-8530 c1cnc(c(c1C(F)F)F)Cl PS-8531 COc1cc(c(cc1OC)F)C#N PS-8532 c1cc(c(c(c1)C(=O)O)N)C(=O)O PS-8533 c1cc(c(cc1F)F)C(=O)CC#N PS-8534 c1c(cc(cc1F)F)C(=O)CC#N PS-8535 c1ccc(c(c1)OC(F)(F)F)F PS-8538 c1cc(c(cc1F)C(F)(F)F)O PS-8539 c1cc(c(cc1O)C(F)(F)F)F PS-8540 c1cc(c(cc1C(F)(F)F)O)F PS-8541 c1cc(c(cc1F)O)C(F)(F)F PS-8542 C1CCN(CC1)CC(=O)O.Cl PS-8543 CN1CCCC[C@H]1C(=O)O.Cl PS-8544 CN1CCC(CC1)C(=O)O.Cl PS-8545 c1cc(c(cc1N)F)C(F)(F)F PS-8546 c1cc(c(c(c1)F)N)C(F)(F)F PS-8547 c1cc(c(cc1C(F)(F)F)F)N PS-8548 c1cc(c(cc1N)C(F)(F)F)F PS-8549 c1cc(c(cc1C(F)(F)F)N)F PS-8550 c1c(cc(cc1N)F)C(F)(F)F PS-8551 c1cc(c(cc1F)C(F)(F)F)N PS-8552 c1cc(c(cc1Cl)S)Cl PS-8553 c1cc(c(cc1S)Cl)Cl PS-8554 Cc1cc(c(c(c1)C(C)(C)C)O)C PS-8555 CC(C)(C)c1ccc(c(c1)O)C=O PS-8556 c1cc(cc(c1)S)C(F)(F)F PS-8557 c1ccc(c(c1)C(F)(F)F)S PS-8558 c1cc(ccc1C(F)(F)F)S PS-8559 Cn1c2cc(c(cc2cn1)F)C=O PS-8560 Cc1c(cccc1F)C(F)(F)F PS-8561 c1cc(cc(c1)OC(F)(F)F)O PS-8562 c1cc(ccc1O)OC(F)(F)F PS-8563 c1ccc(c(c1)O)OC(F)(F)F PS-8564 Cc1ccc2ccc(cc2n1)Cl PS-8565 Cc1cccc2c1nccc2Cl PS-8566 COc1cc(ccc1N)F.Cl PS-8567 Cc1cccc(c1N(C)C)C(C)C PS-8568 c1cc(cc(c1)OC(F)(F)F)N PS-8569 c1cc(ccc1N)OC(F)(F)F PS-8570 c1ccc(c(c1)N)OC(F)(F)F PS-8571 c1cc(c(c(c1)N)O)C(F)(F)F PS-8572 c1cc(c(cc1C(F)(F)F)N)O PS-8573 Cc1cc(cc(c1O)Cl)Cl PS-8574 Cc1cc(c(c(c1)Cl)O)Cl PS-8575 c1c(cnc(n1)F)Br PS-8576 c1c(cnc(n1)Br)F PS-8577 Cc1ccc(c(n1)CN)F.Cl PS-8578 c1cc(ccc1C2CCCCC2)O PS-8579 CCCCc1ccc(cc1)C(=O)C PS-8580 COc1ccc2c(c1)CCC(=O)C2 PS-8581 c1cc(c(cc1C(F)(F)F)N)N PS-8582 c1c(cc(cc1N)N)C(F)(F)F PS-8583 c1cc(c(c(c1)N)N)C(F)(F)F PS-8584 c1cc(c(cc1N)C(F)(F)F)N PS-8585 COc1cccc(c1)C(F)(F)F PS-8586 COc1ccc(cc1)C(F)(F)F PS-8587 COc1ccccc1C(F)(F)F PS-8588 c1cc(cc(c1)C(F)(F)F)CO PS-8589 c1ccc(c(c1)CO)C(F)(F)F PS-8590 c1cc(nc(c1)Br)F PS-8591 c1cc(ncc1Br)F PS-8592 c1cnc(cc1Br)F PS-8593 c1cc(c(nc1)Br)F PS-8594 c1cnc(cc1F)Br PS-8595 c1c(cncc1Br)F PS-8596 c1cncc(c1F)Br PS-8597 c1cncc(c1Br)F PS-8598 c1cc(ccc1C2CCCCC2)N PS-8599 c1ccc(cc1)NC2CCCCC2 PS-8600 c1cc(ccc1N)SC(F)F PS-8601 c1cc(ccc1F)S(=O)(=O)N PS-8602 c1cc(cc(c1)S(=O)(=O)N)F PS-8603 c1ccc(c(c1)F)S(=O)(=O)N PS-8604 Cc1cc(ccc1N)C(F)(F)F PS-8605 Cc1ccc(cc1N)C(F)(F)F PS-8606 Cc1c(cccc1N)C(F)(F)F PS-8607 Cc1cc(cc(c1)N)C(F)(F)F PS-8608 c1cc(cc(c1)C(F)(F)F)CN PS-8609 c1ccc(cc1)C(=N)N.O.Cl PS-8610 CCOc1cc(ccc1F)Cl PS-8611 Cc1ccc(c(c1Cl)OC)F PS-8612 Cc1ccc(c(c1F)CO)Cl PS-8613 Cc1ccc(c(c1Cl)CO)F PS-8614 c1c(cc(c(c1F)O)Cl)C=O PS-8615 c1c(cc(c(c1C=O)O)Cl)F PS-8616 c1c(cc(cc1F)Cl)C(=O)O PS-8617 c1cc(c(cc1C(=O)O)F)Cl PS-8619 c1cc(c(c(c1)Cl)F)C(=O)O PS-8620 c1cc(c(cc1Cl)F)C(=O)O PS-8621 c1cc(c(c(c1)F)Cl)C(=O)O PS-8624 CS(=O)(=O)c1ccc(cc1)F PS-8627 CS(=O)(=O)c1ccccc1F PS-8628 c1cc(c2cccc(c2c1)F)C=O PS-8629 Cc1ccc(cc1C)C(F)(F)F PS-8630 c1cc(ccc1C=O)C(F)(F)F PS-8631 c1cc(cc(c1)C(F)(F)F)C=O PS-8632 c1ccc(c(c1)C=O)C(F)(F)F PS-8633 c1c([nH]c(=O)[nH]c1=O)C(=O)O.O PS-8634 c1c(cc(c(c1C(=O)O)O)F)F PS-8635 c1cc(c(c(c1O)C(=O)O)F)F PS-8636 c1cc(c(c(c1C(=O)O)F)F)O PS-8637 c1cc(c(c(c1F)C(=O)O)O)F PS-8638 c1cc(c(c(c1O)F)C(=O)O)F PS-8639 Cc1ccc(c(c1F)CN)Cl PS-8640 c1cnn(c1)C(=O)NCCCl PS-8641 c1cc(cnc1)CC(=O)O.Cl PS-8642 c1cc(c(cc1C(=O)N)Cl)F PS-8643 c1cc(c(cc1Cl)C(=O)N)F PS-8644 c1cc(c(cc1F)Cl)C(=O)N PS-8645 c1cc(c(c(c1)Cl)F)C(=O)N PS-8646 c1cc(c(cc1F)F)C(=S)N PS-8647 c1cc2ccc(cc2nc1)C(=O)O PS-8648 c1cc2c(cc1N)OC(O2)(F)F PS-8649 C1C[C@H](CNC1)N.Cl.Cl PS-8651 Cc1cncc(n1)Br PS-8652 c1cc(ccc1C(=N)N)O.Cl PS-8653 CC(=O)c1ccc(c(c1)Cl)F PS-8654 CC(=O)c1cc(ccc1F)Cl PS-8655 CC(=O)c1cc(ccc1Cl)F PS-8656 CC(=O)c1ccc(cc1Cl)F PS-8657 CC(=O)c1c(cccc1Cl)F PS-8658 CC(=O)c1ccc(cc1F)Cl PS-8659 CC(C)C1CC(=O)CC(=O)C1.O PS-8660 C=Cc1ccc(cc1)C(F)(F)F PS-8661 C=Cc1cccc(c1)C(F)(F)F PS-8662 C=Cc1ccccc1C(F)(F)F PS-8663 c1cc(cc(c1)C(=O)O)C(F)F PS-8664 COC(=O)c1c(cccc1F)F PS-8665 COC(=O)c1cc(ccc1F)F PS-8666 COC(=O)c1cc(cc(c1)F)F PS-8667 COC(=O)c1ccc(cc1F)F PS-8668 c1cc(cc(c1)OC(F)F)C=O PS-8669 COc1ccc(c(c1F)C=O)F PS-8670 COc1cc(c(c(c1)F)C=O)F PS-8671 COc1ccc(c(c1C=O)F)F PS-8672 COc1cc(c(cc1C=O)F)F PS-8673 CC(=O)c1cc(cc(c1O)F)F PS-8674 c1c(cc(cc1F)F)CC(=O)O PS-8675 c1cc(c(c(c1)F)CC(=O)O)F PS-8676 c1cc(c(cc1F)CC(=O)O)F PS-8677 c1cc(c(cc1CC(=O)O)F)F PS-8678 c1cc(c(cc1F)F)CC(=O)O PS-8679 c1cc(c(c(c1)F)F)CC(=O)O PS-8680 c1ccc(cc1)C(C(=O)O)(F)F PS-8681 C1CS(=O)(=O)C[C@H]1N.Cl PS-8682 c1ccc(cc1)C(=O)CN.Cl PS-8683 C1CC(CCC1N)(F)F.Cl PS-8684 Cc1cc(ncc1C(=O)O)Cl PS-8685 c1cc(ncc1CC(=O)O)Cl PS-8686 CC(=C)CCc1ccccc1C#N PS-8687 COc1cc(c(cc1N)F)OC PS-8688 CC(=O)Nc1ccc(c(c1)F)F PS-8689 CC(=O)Nc1cc(cc(c1)F)F PS-8690 c1cc(ccc1C#N)C(F)(F)F PS-8691 c1cc(cc(c1)C(F)(F)F)C#N PS-8692 c1ccc(c(c1)C#N)C(F)(F)F PS-8693 Cc1ccc(cc1)C(=N)N.Cl PS-8694 c1ccc2c(c1)CCN2N.Cl PS-8695 c1cc(cc(c1)F)NC(=S)N PS-8696 c1ccc(c(c1)NC(=S)N)F PS-8697 c1ccc(cc1)c2ccccc2O PS-8698 CCC(=O)c1cc(cc(c1)F)F PS-8699 CCC(=O)c1ccc(cc1F)F PS-8700 CCC(=O)c1cccc(c1F)F PS-8701 Cc1ccc(c(c1F)F)C(=O)C PS-8702 COC(=O)c1ccc(c(c1)O)F PS-8703 COC(=O)c1cc(ccc1O)F PS-8704 COc1cc(cc(c1O)F)C=O PS-8705 COc1ccc(c(c1)C(=O)O)F PS-8706 C#Cc1ccc(cc1)C(F)(F)F PS-8707 C#Cc1ccccc1C(F)(F)F PS-8708 C#Cc1cccc(c1)C(F)(F)F PS-8709 c1c(cc(c(c1O)O)O)C(=O)O PS-8710 c1ccc2c(c1)CC(C2)N.Cl PS-8712 c1cc(c(cc1Cl)F)CC#N PS-8713 c1c(cc(cc1F)Cl)CC#N PS-8714 c1cc(c(cc1CC#N)Cl)F PS-8715 c1cc(c(c(c1)Cl)F)CC#N PS-8716 COC(=O)c1cc(ccc1N)F PS-8717 c1cc(c(cc1N)CC(=O)O)F PS-8718 Cc1cc(c(c(n1)O)C(=O)O)O PS-8719 c1cc(cc(c1)OC(F)F)C#N PS-8720 COc1cc(c(cc1F)C#N)F PS-8721 COc1c(cc(cc1F)F)C#N PS-8722 CC(C)(Cc1ccc(cc1)F)O PS-8723 CC(=O)Nc1ccc(c(c1)N)F PS-8724 CCOC(=O)c1ccc(cc1)F PS-8725 CCOC(=O)c1cccc(c1)F PS-8726 CCOC(=O)c1ccccc1F PS-8727 Cc1ccc(c(c1)F)CC(=O)O PS-8728 Cc1[nH]c2ccc(c(c2n1)F)F PS-8729 c1cc(c(cc1C=O)F)C(=O)O PS-8730 c1c(c(cnn1)C(=O)O)C(=O)O PS-8731 c1cnc(c(n1)C(=O)O)C(=O)O PS-8732 CC(C)(Cc1ccc(cc1)F)N PS-8733 Cc1ccc(c(c1F)CC#N)F PS-8734 Cc1ccc(c(c1F)F)CC#N PS-8735 c1cc(nc(c1)C(=O)O)C(=O)O PS-8736 CC(C)(C)c1ccc(cc1)S PS-8737 c1cc2c(c(c1)F)C(=O)OC2=O PS-8738 C1CCN(C1)CC(=O)O.Cl PS-8740 COc1cc(nc(n1)C#N)OC PS-8741 CCCN1CCNCC1.Cl PS-8742 c1cc(c(c(c1F)O)F)Cl PS-8743 CC(C)C[C@H]1CCCN1.Cl PS-8744 Cc1ccc(s1)CN.Cl PS-8745 c1cscc1CCN.Cl PS-8746 c1cc2c(cc1F)[nH]cc2C=O PS-8748 c1cc(ccc1C(=O)CC#N)F PS-8749 c1cc(c(cc1F)Cl)S PS-8750 c1[nH]c(c(n1)C(=O)N)N.Cl PS-8751 Cc1ccc2c(c1)c(cs2)C PS-8752 CC(C)(C)c1ccc(cc1)C=O PS-8753 C1CN(CCN1)CC(=O)O.O PS-8754 C1CCC(=CC1)C(=C(F)F)F PS-8755 c1ccc(c(c1)C(F)(F)F)O PS-8756 c1cc(cc(c1)O)C(F)(F)F PS-8757 CCn1c(c(cn1)N)C.Cl PS-8758 CCn1cc(c(n1)C)N.Cl PS-8759 c1c(cc(cc1O)O)N.Cl PS-8760 c1cc(c(nc1)CO)O.Cl PS-8761 c1c([nH]c(=S)[nH]c1=O)N.O PS-8762 c1cc(cc(c1)N)C(F)(F)F PS-8763 c1ccc(c(c1)C(F)(F)F)N PS-8764 c1cc(ccc1C(F)(F)F)N PS-8765 c1cc(ncc1O)CN.Cl PS-8766 c1c(c(cc(c1F)Cl)N)N PS-8767 Cc1ccc(c(c1Cl)O)F PS-8768 COc1c(cccc1Cl)F PS-8769 COc1cccc(c1F)Cl PS-8770 COc1ccc(c(c1)F)Cl PS-8771 c1cc(c(cc1CO)F)Cl PS-8772 c1cc(c(cc1CO)Cl)F PS-8773 c1c(cc(cc1F)Cl)CO PS-8774 c1cc(c(cc1Cl)CO)F PS-8775 c1cc(c(c(c1)Cl)F)CO PS-8776 c1ccc2cc(ccc2c1)S PS-8777 COc1cc(c(c(c1)F)O)F PS-8778 Cc1cc(c(cc1F)Cl)N PS-8779 c1cc(c(cc1F)Cl)CN PS-8780 c1cc(c(cc1Cl)CN)F PS-8781 c1cc(c(cc1CN)Cl)F PS-8782 c1cc(c(c(c1)Cl)CN)F PS-8783 c1cc(c(c(c1)Cl)F)CN PS-8784 c1cnc(c(c1C=O)F)Cl PS-8785 CC(C)[C@H](C#N)c1ccccc1 PS-8786 c1ccc2c(c1)ccc(n2)CO PS-8787 c1cnccc1S(=O)(=O)O PS-8788 c1cc(cc(c1)OC(F)F)N PS-8789 c1ccc(c(c1)N)OC(F)F PS-8790 c1cc(ccc1N)OC(F)F PS-8791 COc1cc(c(c(c1)F)N)F PS-8792 COc1c(cc(cc1F)N)F PS-8793 COc1c(ccc(c1F)F)N PS-8794 Cc1ccnc(c1)CN.Cl PS-8795 c1cnc(cn1)C(=N)N.Cl PS-8796 c1cc(c(cc1Cl)F)C=O PS-8797 c1cc(c(cc1F)Cl)C=O PS-8798 c1cc(c(cc1C=O)Cl)F PS-8799 c1cc(c(c(c1)Cl)F)C=O PS-8800 c1cc(c(cc1C=O)F)Cl PS-8801 c1cc(c(cc1F)C=O)Cl PS-8802 c1c(cc(cc1F)Cl)C=O PS-8803 c1cc(c(cc1Cl)C=O)F PS-8804 c1cc(c(c(c1)Cl)C=O)F PS-8805 CC(C)(C)c1ccc(cc1)C#C PS-8806 CCOc1cccc(c1F)F PS-8807 c1cc(cc(c1)C(F)F)CO PS-8808 c1cc(=O)[nH]nc1C(=O)O.O PS-8809 c1cc(c(c(c1O)F)C=O)F PS-8810 c1c(cc(c(c1F)C=O)F)O PS-8811 c1c(cc(c(c1F)O)F)C=O PS-8812 c1cc(c(c(c1F)C=O)O)F PS-8813 c1c(c(cc(c1F)F)O)C=O PS-8814 c1c(cc(c(c1C=O)O)F)F PS-8815 c1cc(c(c(c1)F)F)C(=O)O PS-8817 c1c(cc(cc1F)F)C(=O)O PS-8818 c1cc(c(cc1F)F)C(=O)O PS-8819 c1ccnc(c1)C(=N)N.Cl PS-8822 c1cnccc1C(=N)N.Cl PS-8823 C1CNCCC1(F)F.Cl PS-8824 CSc1ccc(c(c1)F)N PS-8825 c1ccc2c(c1)c(ccn2)C=O PS-8826 Cc1ccc(c(c1F)F)CN PS-8827 C[C@@H](c1cc(cc(c1)F)F)N PS-8828 c1cc(c(c(c1)F)F)C(=O)N PS-8829 c1cc(c(c(c1)F)C(=O)N)F PS-8830 c1c(cc(cc1F)F)C(=O)N PS-8831 c1cc(c(cc1F)C(=O)N)F PS-8832 c1cc(c(cc1C(=O)N)F)F PS-8833 C1CC2(CCC1=O)OCCO2 PS-8834 COc1ccc(cc1OC)F PS-8835 COc1cccc(c1F)CO PS-8836 COc1cc(cc(c1)F)CO PS-8837 COc1cccc(c1CO)F PS-8838 COc1ccc(cc1CO)F PS-8839 c1cc(cc(c1)C(F)F)C=O PS-8840 Cc1ccc(c(c1F)F)C=O PS-8841 Cc1ccc(c(c1F)C=O)F PS-8842 CC(=O)c1ccc(c(c1)F)F PS-8843 CC(=O)c1cc(cc(c1)F)F PS-8844 CC(=O)c1c(cccc1F)F PS-8845 CC(=O)c1cc(ccc1F)F PS-8846 CC(=O)c1ccc(cc1F)F PS-8847 CC(=O)c1cccc(c1F)F PS-8848 c1cc(c(c(c1)O)F)C(=O)O PS-8849 c1cc(c(cc1F)C(=O)O)O PS-8850 C#Cc1cc(c(c(c1)F)F)F PS-8851 c1cc(oc1C(=O)O)C(=O)O PS-8853 c1cc(c(cc1C#N)F)Cl PS-8854 c1cc(c(cc1C#N)Cl)F PS-8855 c1cc(c(cc1Cl)C#N)F PS-8856 c1cc(c(c(c1)Cl)C#N)F PS-8857 c1cc(c(c(c1)Cl)F)C#N PS-8858 c1cc(c(cc1F)Cl)C#N PS-8859 c1cc(c(cc1Cl)F)C#N PS-8860 c1c(cc(cc1F)Cl)C#N PS-8861 c1cc(c(c(c1)F)Cl)C#N PS-8862 c1cc(c(cc1F)C#N)Cl PS-8863 c1cc(c(cc1C(=O)O)N)F PS-8864 c1cc(c(cc1N)C(=O)O)F PS-8865 c1cc(c(cc1F)C(=O)O)N PS-8866 c1cc(c(cc1F)N)C(=O)O PS-8867 CC(=O)c1cc(no1)C(=O)O PS-8870 c1c(cc(c(c1C#N)O)F)F PS-8871 CC(C)(c1ccc(cc1)F)O PS-8873 c1cc(cc(c1)F)NC(=O)N PS-8874 c1cc(c(cc1F)C(=O)N)N PS-8875 c1cc(c(c(c1)F)C(=O)N)N PS-8876 CC(=O)Oc1ccccc1F PS-8877 Cc1cc(cc(c1O)C=O)F PS-8878 COC(=O)c1cccc(c1)F PS-8879 COC(=O)c1ccc(cc1)F PS-8880 COC(=O)c1ccccc1F PS-8881 COc1ccc(cc1C=O)F PS-8882 COc1cc(cc(c1)F)C=O PS-8883 COc1cc(ccc1C=O)F PS-8884 COc1ccc(cc1F)C=O PS-8885 COc1cc(ccc1F)C=O PS-8886 COc1ccc(c(c1)F)C=O PS-8887 COc1cccc(c1C=O)F PS-8888 COc1cccc(c1F)C=O PS-8889 COC(=O)c1cncnc1O PS-8892 COc1ccc(nn1)C(=O)O PS-8893 COc1cnc(cn1)C(=O)O PS-8894 c1cc(c(c(c1C#N)F)F)N PS-8895 c1cc(c(c(c1C#N)N)F)F PS-8896 c1c(c(cc(c1F)N)F)C#N PS-8897 C1CNCCC1=O.O.Cl PS-8898 CC(C)(c1ccc(cc1)F)N PS-8899 C[C@@H](c1cccc(c1)F)NC PS-8900 CC(=O)Nc1cccc(c1)F PS-8901 CC(=O)c1cc(ccc1F)N PS-8902 c1cc(cc(c1)C(F)F)C#N PS-8903 Cc1c(ccc(c1F)C#N)F PS-8904 c1c(cc(cc1F)F)CC#N PS-8905 c1cc(c(cc1F)CC#N)F PS-8906 c1cc(c(cc1CC#N)F)F PS-8907 c1cc(c(c(c1)F)CC#N)F PS-8908 c1cc(c(cc1F)F)CC#N PS-8909 c1cc(c(c(c1)F)F)CC#N PS-8910 c1ccc(cc1)C(C#N)(F)F PS-8911 C1C(=O)N=C(S1)N.Cl PS-8912 CC(C)c1ccc(cc1)S PS-8913 C#Cc1ccc2ccccc2c1 PS-8914 CCC(=O)c1cccc(c1)F PS-8915 CCC(=O)c1ccc(cc1)F PS-8916 CCC(=O)c1ccccc1F PS-8917 Cc1ccc(c(c1)F)C(=O)C PS-8918 Cc1ccc(c(c1)C(=O)C)F PS-8919 CC(=O)Cc1ccc(cc1)F PS-8920 CC(=O)Cc1ccccc1F PS-8921 C1[C@@H](CC[C@H](C1)O)N.Cl PS-8922 COc1cc(cc(c1)F)C#N PS-8923 C1CNCCNC1=O.Cl PS-8924 Cc1cc(c(c(c1)C)OC)C PS-8925 CC(C)[C@@H]1CCCN1.Cl PS-8926 C1CC(=O)CCNC1.Cl PS-8927 c1cc(c(cc1C=O)C#N)F PS-8928 c1cc(c(cc1C#N)F)C=O PS-8929 c1cc(c(cc1F)C#N)C=O PS-8930 c1cnc(c(n1)Cl)Cl PS-8931 Cc1c([nH]cn1)CO.Cl PS-8932 Cc1c(cn(n1)C)N.Cl PS-8933 c1cnccc1C(F)(F)F PS-8934 c1cc(cnc1)C(F)(F)F PS-8935 Cc1ccnc(n1)O.Cl PS-8936 c1cc(ncc1O)N.Cl PS-8937 c1cncc(c1N)O.Cl PS-8938 CC(=O)c1ccn[nH]1.Cl PS-8939 c1cc(c(c(c1)Cl)O)F PS-8940 c1cc(c(cc1O)Cl)F PS-8941 c1cc(c(cc1F)Cl)O PS-8942 c1cc(c(c(c1)Cl)F)O PS-8943 c1cc(c(cc1O)F)Cl PS-8944 c1cc(c(cc1F)O)Cl PS-8945 c1c(cc(cc1F)Cl)O PS-8946 c1cc(c(cc1Cl)F)O PS-8947 c1cc(c(cc1S)F)F PS-8948 C1CCC(CC1)(C(=O)O)F PS-8949 c1cc(c(cc1C#N)C#N)F PS-8950 Cc1cc(cnc1Cl)F PS-8951 c1cc(c(c(c1)F)Cl)N PS-8952 c1cc(c(c(c1)Cl)N)F PS-8953 c1cc(c(cc1N)F)Cl PS-8954 c1cc(c(cc1N)Cl)F PS-8955 c1cc(c(c(c1)Cl)F)N PS-8956 c1cc(c(cc1Cl)F)N PS-8957 c1cc(c(cc1F)Cl)N PS-8958 c1cc(c(cc1Cl)N)F PS-8959 c1c(cc(cc1F)Cl)N PS-8960 Cc1cc(c(c(c1)C)C#N)C PS-8961 CC(C)(C#N)c1ccccc1 PS-8962 c1c(cc(c(c1O)N)F)F PS-8963 c1c(c(cc(c1F)F)O)N PS-8964 c1c(cc(c(c1N)O)F)F PS-8965 c1c(cc(c(c1F)O)F)N PS-8966 c1c(c(cc(c1F)O)F)N PS-8967 c1cc(c(c(c1N)O)F)F PS-8968 Cc1cc(cnc1)N.Cl PS-8969 C#CCCCc1ccccc1 PS-8970 C1CC[C@@H]([C@H](C1)CO)CO PS-8971 C#Cc1ccc(c(c1)F)C#C PS-8972 c1cc(c(c(c1N)N)F)F PS-8973 c1c(cc(c(c1N)N)F)F PS-8974 Cc1ccc(c(c1F)O)F PS-8975 Cc1ccc(c(c1F)F)O PS-8976 COc1cc(cc(c1)F)F PS-8977 COc1cccc(c1F)F PS-8978 COc1ccc(c(c1)F)F PS-8979 COc1ccc(cc1F)F PS-8980 COc1cc(ccc1F)F PS-8981 c1cc(c(c(c1)F)F)CO PS-8982 c1cc(c(cc1F)CO)F PS-8983 c1c(cc(cc1F)F)CO PS-8984 c1cc(c(cc1CO)F)F PS-8985 c1cc(c(c(c1)F)CO)F PS-8986 c1cc(c(cc1F)F)CO PS-8987 COc1ncc(c(n1)O)F PS-8988 C1CNCC1(F)F.Cl PS-8989 c1cc(c(c(c1)F)F)CN PS-8990 c1c(cc(cc1F)F)CN PS-8991 c1cc(c(c(c1)F)CN)F PS-8992 c1cc(c(cc1F)CN)F PS-8993 c1cc(c(cc1CN)F)F PS-8994 c1cc(c(cc1F)F)CN PS-8995 COc1cc(c(cn1)F)O PS-8996 c1cc(nc(c1C=O)F)F PS-8997 c1c(c(c(cn1)F)C=O)F PS-8998 CSc1cccc(c1)F PS-8999 CSc1ccc(cc1)F PS-9000 c1cc(ccc1CS)F PS-9001 CCc1c(c(ncn1)O)F PS-9002 COc1ccc(cc1F)O PS-9003 COc1ccc(cc1O)F PS-9004 COc1ccc(c(c1)F)O PS-9005 COc1cc(ccc1O)F PS-9006 COc1cccc(c1O)F PS-9007 CCOC(=O)c1ncon1 PS-9008 c1cc(c(c(c1)F)F)C=O PS-9009 c1c(cc(cc1F)F)C=O PS-9010 c1cc(c(c(c1)F)C=O)F PS-9011 c1cc(c(cc1F)C=O)F PS-9012 c1cc(c(cc1F)F)C=O PS-9013 c1cc(c(cc1C=O)F)F PS-9014 Cc1cc(c(nc1)Cl)C PS-9015 COc1ccc(cc1F)N PS-9016 COc1cc(ccc1F)N PS-9017 COc1cccc(c1N)F PS-9018 COc1ccc(cc1N)F PS-9019 COc1c(cccc1F)N PS-9020 COc1cc(cc(c1)F)N PS-9021 c1cc(nc(c1)F)C(=O)O PS-9022 c1cnc(cc1C(=O)O)F PS-9023 c1cc(c(nc1)F)C(=O)O PS-9024 c1cc(ncc1C(=O)O)F PS-9025 c1cc(ncc1F)C(=O)O PS-9026 c1c(cncc1F)C(=O)O PS-9027 c1cncc(c1C(=O)O)F PS-9028 c1cc(ccc1C=O)Cl PS-9029 c1cc(c(c(c1)F)CN)N PS-9030 CCOc1ccc(cc1)F PS-9031 Cc1cc(ccc1F)OC PS-9032 Cc1ccc(cc1F)OC PS-9033 Cc1ccc(cc1OC)F PS-9034 Cc1ccc(c(c1)OC)F PS-9035 c1cc(ccc1CCO)F PS-9036 Cc1ccc(cc1CO)F PS-9037 Cc1ccc(c(c1)F)CO PS-9038 Cc1cccc(c1CO)F PS-9039 Cc1cc(cc(c1)F)CO PS-9040 Cc1c(cccc1F)CO PS-9041 C[C@@H](c1ccc(cc1)F)O PS-9042 C[C@H](c1cccc(c1)F)O PS-9043 C=Cc1ccc(cc1F)F PS-9044 C=Cc1cc(cc(c1)F)F PS-9045 C=Cc1ccc(c(c1)F)F PS-9046 C=Cc1cc(ccc1F)F PS-9047 C=Cc1c(cccc1F)F PS-9048 c1cc(nc(c1)F)C(=O)N PS-9049 c1cc(c(c(c1)F)O)C=O PS-9050 c1cc(c(cc1O)F)C=O PS-9051 c1cc(c(cc1F)O)C=O PS-9052 c1cc(c(cc1F)C=O)O PS-9053 c1cc(c(c(c1)F)C=O)O PS-9054 c1cc(c(cc1C=O)F)O PS-9055 c1cc(ccc1C(=O)O)F PS-9056 c1c(ncnc1O)C(=O)O PS-9059 C1C[C@@H](CNC1)F.Cl PS-9060 C1CNCCC1F.Cl PS-9061 CCNc1ccccc1F PS-9062 Cc1cc(ccc1F)CN PS-9063 Cc1ccc(cc1CN)F PS-9064 C[C@H](c1ccc(cc1)F)N PS-9065 C[C@H](c1cccc(c1)F)N PS-9066 CC(c1ccccc1F)N PS-9067 CC(=O)c1cccnc1F PS-9068 c1cc(cc(c1)F)C(=O)N PS-9069 c1ccc(c(c1)C(=O)N)F PS-9070 c1cc(ccc1C(=O)N)F PS-9071 C1C[C@H](NC1)C(F)(F)F PS-9072 c1c(cc(cc1F)F)C#N PS-9073 c1cc(c(c(c1)F)C#N)F PS-9074 c1cc(c(cc1C#N)F)F PS-9075 c1cc(c(cc1F)F)C#N PS-9076 c1cc(c(cc1F)C#N)F PS-9077 C=Cc1ccccc1Cl PS-9078 Cc1cccc(c1C=O)F PS-9079 Cc1cc(cc(c1)F)C=O PS-9080 Cc1ccc(cc1C=O)F PS-9081 Cc1cc(ccc1F)C=O PS-9082 Cc1cccc(c1F)C=O PS-9083 Cc1ccc(c(c1)F)C=O PS-9084 Cc1ccc(c(c1)C=O)F PS-9085 Cc1cc(ccc1C=O)F PS-9086 Cc1ccc(cc1F)C=O PS-9087 Cc1c(cccc1F)C=O PS-9088 c1cc2c(cc1F)CCO2 PS-9089 CC(=O)c1ccccc1F PS-9090 CC(=O)c1ccc(cc1)F PS-9091 CC(=O)c1cccc(c1)F PS-9092 C#Cc1ccc(c(c1)F)F PS-9093 c1cc2c(cc1F)CCN2 PS-9095 Cc1ccnc(c1)C(=O)O PS-9096 c1c(cnc(c1N)C#N)F PS-9097 c1c(cnc(c1F)C#N)N PS-9098 c1cc2c(cc1F)nco2 PS-9099 c1cc(c(cc1C#N)F)O PS-9100 CCc1cccc(c1O)C PS-9101 c1cc2c(c(c1)F)nc[nH]2 PS-9104 Cc1c(ccc(n1)F)C#N PS-9105 Cc1ccc(c(n1)C#N)F PS-9106 c1cc2c(cc1F)cn[nH]2 PS-9107 c1cc(c(cc1C#N)F)N PS-9108 c1c(cc(cc1N)F)C#N PS-9109 c1cc(c(cc1F)C#N)N PS-9110 c1cc(c(cc1N)C#N)F PS-9111 c1cc(c(c(c1)F)N)C#N PS-9112 c1cc(c(cc1F)N)C#N PS-9113 c1cc(c(cc1C#N)N)F PS-9114 c1cc(c(cc1N)F)C#N PS-9115 c1c(nc[nH]1)C(F)(F)F PS-9116 c1c[nH]nc1C(F)(F)F PS-9117 C1CC(=O)CNC1.Cl PS-9118 Cc1ccc(cc1F)C#N PS-9119 Cc1cccc(c1C#N)F PS-9120 Cc1cc(cc(c1)F)C#N PS-9121 Cc1ccc(c(c1)F)C#N PS-9122 Cc1ccc(cc1C#N)F PS-9123 Cc1c(cccc1F)C#N PS-9124 Cc1cc(ccc1C#N)F PS-9125 Cc1ccc(c(c1)C#N)F PS-9126 c1cc2c(cc[nH]2)c(c1)F PS-9127 c1cc2cc[nH]c2c(c1)F PS-9128 c1cc(cc(c1)F)CC#N PS-9129 c1ccc(c(c1)CC#N)F PS-9130 c1cc(ccc1CC#N)F PS-9131 c1c(nc[nH]1)CO.Cl PS-9132 c1cocc1CN.Cl PS-9133 c1cnc(nc1)O.Cl PS-9134 c1c(c(ncn1)Cl)F PS-9135 c1cncnc1N.Cl PS-9136 c1cc(nc(c1)Cl)F PS-9137 c1cc(ncc1Cl)F PS-9138 c1cc(c(nc1)F)Cl PS-9139 c1cc(c(nc1)Cl)F PS-9140 c1cc(ncc1F)Cl PS-9141 c1cncc(c1Cl)F PS-9142 c1cc(nc(c1O)F)F PS-9143 C1CC1CNC(=S)N PS-9144 c1c(cnc(c1F)N)F PS-9145 c1c(cc(cc1F)F)O PS-9146 c1cc(c(c(c1)F)O)F PS-9147 c1cc(c(c(c1)F)F)O PS-9148 c1cc(c(cc1O)F)F PS-9149 c1cc(c(cc1F)O)F PS-9150 c1cc(c(cc1F)F)O PS-9151 C1CN(C(=O)N1)CCN PS-9152 c1c(cc(cc1F)F)N PS-9153 c1cc(c(c(c1)F)F)N PS-9154 c1cc(c(cc1F)F)N PS-9155 c1cc(c(cc1N)F)F PS-9156 c1cc(c(c(c1)F)N)F PS-9157 c1cc(c(cc1F)N)F PS-9158 c1cc(cc(c1)S)F PS-9159 c1ccc(c(c1)F)S PS-9160 c1cc(c(c(c1)F)O)O PS-9161 c1cc(c(cc1F)O)O PS-9162 Cc1cc(cnc1F)O PS-9164 COc1ccc(cn1)F PS-9165 c1cc(c(cc1F)O)N PS-9166 c1cc(c(cc1N)F)O PS-9167 c1cc(c(cc1F)N)O PS-9168 c1cc(c(c(c1)F)O)N PS-9169 c1cc(c(c(c1)F)N)O PS-9170 c1cc(c(cc1O)N)F PS-9171 c1cc(c(cc1O)F)N PS-9172 Cc1ccc(c(n1)F)N PS-9173 Cc1cc(ncc1N)F PS-9174 c1cc(c(c(c1)F)N)N PS-9175 Cc1cc(ccc1O)F PS-9176 Cc1c(cccc1F)O PS-9177 Cc1cc(ccc1F)O PS-9178 Cc1ccc(c(c1)F)O PS-9179 Cc1ccc(c(c1)O)F PS-9180 Cc1ccc(cc1O)F PS-9181 Cc1cc(cc(c1)F)O PS-9182 Cc1cccc(c1F)O PS-9183 Cc1ccc(cc1F)O PS-9184 COc1cccc(c1)F PS-9185 COc1ccc(cc1)F PS-9186 COc1ccccc1F PS-9187 c1cc(ccc1CO)F PS-9188 c1ccc(c(c1)CO)F PS-9189 C1CNC[C@H]1F.Cl PS-9190 Cc1cc(ccc1F)N PS-9191 Cc1ccc(cc1N)F PS-9192 Cc1cccc(c1N)F PS-9193 Cc1ccc(cc1F)N PS-9194 Cc1cc(cc(c1)F)N PS-9195 Cc1ccc(c(c1)N)F PS-9196 Cc1c(cccc1F)N PS-9197 Cc1ccc(c(c1)F)N PS-9198 Cc1cccc(c1F)N PS-9199 Cc1cc(ccc1N)F PS-9200 CNc1ccccc1F PS-9201 c1cc(cc(c1)F)CN PS-9202 c1cc(ccc1CN)F PS-9203 c1cc(nc(c1)F)C=O PS-9204 c1cc(ncc1C=O)F PS-9205 c1cc(c(nc1)F)C=O PS-9206 c1cc(ncc1F)C=O PS-9207 c1c(cncc1F)C=O PS-9208 c1cncc(c1C=O)F PS-9209 c1cc(ccc1C=O)F PS-9210 c1cc(cc(c1)F)C=O PS-9211 c1ccc(c(c1)C=O)F PS-9212 C1CNC[C@H]1O.Cl PS-9213 C[C@@H](c1ccccn1)N PS-9214 C=Cc1ccccc1F PS-9215 C=Cc1ccc(cc1)F PS-9216 C=Cc1cccc(c1)F PS-9217 c1cc(nc(c1)F)C#N PS-9218 c1cc(c(nc1)F)C#N PS-9219 c1cnc(cc1C#N)F PS-9220 c1c(cncc1F)C#N PS-9221 C1CC1S(=O)(=O)N PS-9222 c1cc(ccc1C#N)F PS-9223 c1cc(cc(c1)F)C#N PS-9224 c1ccc(c(c1)C#N)F PS-9225 C1CC1C(=N)N.Cl PS-9226 C#Cc1ccc(cc1)F PS-9227 C#Cc1ccccc1F PS-9228 C#Cc1cccc(c1)F PS-9229 c1cnc(cc1C#N)O PS-9230 c1cc(sc1)Cl PS-9231 c1cc(ncc1F)F PS-9232 c1cc(c(nc1)F)F PS-9233 c1c(cncc1F)F PS-9234 c1cnc(cn1)Cl PS-9235 c1c(c(ncn1)O)F PS-9237 c1c(non1)C(=O)O PS-9238 c1cc(cnc1)Cl PS-9239 C1CNCCC1C=O PS-9240 c1cc(c(nc1)F)O PS-9241 c1cc(c(nc1)O)F PS-9242 c1cc(ncc1F)O PS-9243 c1cc(ncc1O)F PS-9244 c1cc(sc1)C=O PS-9245 c1cc(nc(c1)F)N PS-9246 c1cc(c(nc1)F)N PS-9247 c1cc(ncc1N)F PS-9248 c1cc(c(nc1)N)F PS-9249 c1cc(ncc1F)N PS-9250 c1cncc(c1N)F PS-9251 c1c(cncc1F)N PS-9252 c1cc(ccc1O)F PS-9253 c1ccc(c(c1)O)F PS-9254 c1cc(cc(c1)F)O PS-9255 Cc1cccc(n1)F PS-9256 Cc1ccnc(c1)F PS-9257 Cc1cccnc1F PS-9258 Cc1ccc(nc1)F PS-9259 Cc1ccc(cn1)F PS-9260 Cc1ccncc1F PS-9261 c1cc(cc(c1)F)N PS-9262 c1cc(ccc1N)F PS-9263 c1cc(ncc1O)N PS-9264 C1C(CN1)O.Cl PS-9265 c1cc(sc1)C#N PS-9266 c1cscc1C#N PS-9267 c1cc(nc(c1)N)N PS-9269 Cc1ccc(nn1)N PS-9270 Cc1cnc(cn1)N PS-9271 Cc1cncc(n1)N PS-9272 c1cncc(c1N)N PS-9273 c1cnc(cn1)CN PS-9274 COc1ccccn1 PS-9275 Cc1c(cccn1)O PS-9276 Cc1cc(cnc1)O PS-9277 Cc1ccncc1O PS-9278 c1cc(cc(c1)O)N PS-9279 COc1ccncc1 PS-9280 COc1cccnc1 PS-9281 C1C[C@@H](C(=O)C1)C#N PS-9282 C#Cc1cccs1 PS-9283 Cc1ccc(nc1)N PS-9284 Cc1ccnc(c1)N PS-9285 Cc1c(cccn1)N PS-9286 Cc1ccc(cn1)N PS-9287 Cc1cc(ccn1)N PS-9288 Cc1ccncc1N PS-9289 Cc1cc(cnc1)N PS-9290 Cc1cnccc1N PS-9291 c1ccnc(c1)CN PS-9292 Cc1c(ocn1)C#N PS-9293 c1cncnc1C=O PS-9294 c1c(cncn1)C=O PS-9295 c1cnc(nc1)C=O PS-9296 c1cnncc1C=O PS-9297 c1cnc(cn1)C=O PS-9298 Cc1cccc(c1)N PS-9299 Cn1ccc(n1)C#N PS-9300 c1ccnc(c1)C=O PS-9301 c1c(cncn1)C#N PS-9302 c1cnc(nc1)C#N PS-9303 c1cc(nnc1)C#N PS-9304 c1cnc(cn1)C#N PS-9305 C#Cc1ccccn1 PS-9306 c1([nH]nnn1)N.O PS-9307 C1CSCC1=O PS-9308 C1COCCN1N PS-9309 C1CC1(C(=O)O)O PS-9310 C1CN(CCN1)N PS-9311 C1C[C@@H](NC1)CO PS-9312 C1COCCC1N PS-9313 C1COC[C@H]1CN PS-9314 c1[nH]nc(n1)S PS-9315 c1cs[nH]c1=O PS-9316 C1CNC(=O)[C@H]1O PS-9317 C1[C@@H](CNC1=O)O PS-9318 C1CC1(C(=O)O)N PS-9319 C[C@@H]1CNCCN1 PS-9320 CN1CCNCC1 PS-9321 C1CCC(C1)CO PS-9322 c1csc(n1)N PS-9323 c1cnc([nH]1)S PS-9324 c1c(scn1)N PS-9325 C1CNC(=O)CN1 PS-9326 C1CC1CC(=O)O PS-9327 CC1(CC1)C(=O)O PS-9328 C1COCCC1=O PS-9329 C[C@H]1C(=O)CCO1 PS-9330 CC1CCNCC1 PS-9331 c1c(ocn1)CO PS-9332 c1c(nco1)CO PS-9333 Cc1cc(=O)[nH]o1 PS-9334 c1coc(n1)CO PS-9335 Cc1ccsc1 PS-9336 c1cnc(cn1)F PS-9337 Cc1cc(n[nH]1)N PS-9338 Cn1ccc(n1)N PS-9339 c1cc(oc1)CN PS-9340 c1c(nco1)C=O PS-9341 C1=CC(=O)NC1=O PS-9342 Cc1c[nH]c(n1)C PS-9343 C1CCN(C1)C#N PS-9344 CCn1ccnc1 PS-9345 Cc1ccnn1C PS-9346 Cc1ccc(o1)C PS-9347 c1c(nc[nH]1)C=O PS-9348 c1cc(=O)[nH]nc1 PS-9349 c1cnc([nH]1)C=O PS-9350 c1cc(nnc1)N PS-9352 c1cnc(cn1)N PS-9353 c1cnncc1N PS-9354 c1cc([nH]c1)C=O PS-9355 c1c[nH]cc1C=O PS-9356 Cc1cncnc1 PS-9357 c1cc(cnc1)N PS-9358 c1[nH]nc(n1)C#N PS-9359 c1c(nco1)C#N PS-9360 c1cn(cn1)C#N PS-9361 C1COC[C@H]1O PS-9362 C1CNC[C@H]1O PS-9363 C1COCC1=O PS-9364 C[C@@H]1CCCN1 PS-9365 c1nncn1N PS-9366 c1[nH]nc(n1)N PS-9367 c1conc1N PS-9368 c1c[nH]nc1N PS-9369 c1cn[nH]c1N PS-9370 c1c(cn[nH]1)N PS-9371 Cn1ccnc1 PS-9372 C1CC(=O)C=C1 PS-9373 C1CC(C1)N PS-9374 C1CNC1=O PS-9375 C1CC(=O)C1 PS-9376 c1[nH]ncn1 PS-9377 c1cnn[nH]1 PS-9378 C1CN[C@H](CN1)C(=O)O.Cl.Cl PS-9379 CC(C)(C)OC(=O)N[C@@H]1CCCNC1 PS-9380 CC(c1cccc(c1)F)N PS-9382 C[C@@H](c1ccc(cc1)F)N PS-9383 C[C@@H](c1cccc(c1)F)N PS-9384 C[C@@H](c1ccccc1F)N PS-9385 C1CNC[C@@H]1F.Cl PS-9387 C1C[C@H](NC1)CO PS-9388 C[C@H]1CNCCN1 PS-9389 C1COC[C@@H]1O PS-9390 C1CN[C@@H](CC12OCCO2)C(=O)O PS-9393 C1CNC12COC2.C(=O)(C(=O)O)O PS-9397 CN(C)c1c(c(ncn1)Cl)N RS-0002 CC1(CC2=C(C(=O)C1)Sc3c(c(=O)[nH]cn3)N2)C RS-0003 CC1(CC(=C2C(=Nc3c(ncnc3S2)OC)C1)NCc4ccccc4)C RS-0004 Cc1c(c(nc(n1)N)SCc2ccc(cc2)[N+](=O)[O-])N RS-0005 c1nc(c(c(n1)Cl)N)N2CCCCC2 RS-0007 c1ccc(cc1)CNC(=O)c2csc3c2C4CCN3CC4 RS-0009 c1ccc(cc1)C(c2ccccc2)C(=O)Cc3csc4c3C5CCN4CC5.Cl RS-0010 Cc1[nH]c2c(n1)cnc3c2c(=O)n(c(=O)n3C)C RS-0012 COc1c2c(ncn1)SCC(=N2)N.Cl RS-0014 COc1c2c(ncn1)SCC(=O)N2 RS-0019 c1ccc2c(c1)c3c(n2CN4CCCCC4)nc5ccccc5n3 RS-0020 c1ccc2c(c1)c3c(n2CC(=O)NN)nc4ccccc4n3 RS-0021 Cn1c2c(c(=O)n(c1=O)C)nc3c4ccccc4[nH]c3n2 RS-0023 CCOC(=O)/C(=C/1\C=CN(C=N1)C)/C#N RS-0025 CCN(CC)C(=O)N1CCN(CC1)CC(=O)c2c(n(c(=O)n(c2=O)C)C)N RS-0026 Cn1c(c(c(=O)n(c1=O)C)C(=O)CN2CCOCC2)N RS-0027 CC(=O)Nc1cc(=O)c2c([nH]1)n(c(=O)n(c2=O)C)C RS-0028 Cn1c2c(c(c(c(n2)NNC(=O)c3ccccc3)N)O)c(=O)n(c1=O)C RS-0029 Cn1c2c(c(c(cn2)[N+](=O)[O-])Nc3ccccc3C(=O)OC)c(=O)n(c1=O)C RS-0031 Cn1cnc2c1c3c(nc2)n(c(=O)n(c3=O)C)C RS-0032 COc1ccc2c(c1)[nH]cc2CCN RS-0033 CN(C)c1nc(nc(n1)Oc2ccc(cc2)OCC#C)OC RS-0035 CC(=O)Nc1ccc(cc1)Nc2c(cc(cc2[N+](=O)[O-])C(=O)N3CC(=O)Nc4c3cccc4)[N+](=O)[O-] RS-0037 CC1(CC(=C2C(=Nc3c(ncnc3S2)OC)C1)NCCCCCC(=O)O)C RS-0040 CC1(CC(=C(C(=O)C1)Br)Nc2ccc(cc2)CCCC(=O)OC)C RS-0041 c1cc(ccc1NC(=O)/C=N/O)S(=O)(=O)N RS-0042 c1cc(ccc1C2C3COCN3CO2)[N+](=O)[O-] RS-0045 CC(=O)N1C2CC(NC1=O)N(C(=O)N2)C(=O)C RS-0046 c1ccc(cc1)C2=NOC(C2(Cl)Cl)(c3ccccc3)O RS-0048 C1C2(COCN2CO1)CO RS-0049 CC(C1CC1)N(c2ccccc2)C(=O)CN3CCOCC3.Cl RS-0050 c1cc(ccc1C(=O)/C(=C/c2ccc(cc2Cl)Cl)/n3cncn3)Cl RS-0051 Cc1c(c(nc(n1)N)C(F)(F)F)Br RS-0053 Cc1cc(nc(n1)N)C(F)(F)F RS-0054 Cc1ccc(cc1)NC(=O)O/N=C(/C(C)C)\Cl RS-0055 CC(C)CCOc1ccc2c(c1)nc([nH]2)NC(=O)OC RS-0056 c1ccc(cc1)Cn2cnc3c2c(=O)[nH]c(n3)NCCCCCC(=O)O.O RS-0057 CN(C)c1ccnc2c1c3c(s2)c(=O)[nH]cn3 RS-0058 Cn1c(c(c(=O)n(c1=O)C)C(=O)CN2CCC(C2)c3ccccc3)N RS-0062 CC(C)(C)N(C=C(Cl)Cl)C(=O)n1ccnc1 RS-0065 CC1(C(N1N2C(=O)c3ccccc3C2=O)C#Cc4ccccc4)C RS-0066 c1ccc2c(c1)c3cc(ccc3[nH]2)N RS-0067 c1cc(ccc1/C=C(/C=N/N2C(=O)CSC2=S)\Cl)[N+](=O)[O-] RS-0068 Cc1c(c(n(n1)C)C)/C=C(/C(=O)C(C)C)\n2cncn2 RS-0069 c1ccc(cc1)C(=O)NC2C(=C(C(=O)O2)Cl)N RS-0070 CC(=O)NC1=C(C(=O)OC1NC(=O)c2ccccc2)Cl RS-0071 Cc1ccccc1S(=O)(=O)NC2C(=C(C(=O)O2)Oc3ccccc3)Br RS-0072 c1cc(cc(c1)[N+](=O)[O-])/C=C(\C(=O)c2ccc(cc2Cl)Cl)/n3cncn3 RS-0073 CC(C)COC(=O)c1c(snn1)NC(=O)Nc2ccccc2 RS-0074 CCCCOC(=O)c1c(snn1)NC(=O)Nc2ccccc2 RS-0075 CSC\1CS(=O)(=O)C/C1=N/OC(=O)Nc2ccccc2 RS-0077 CSC\1CS(=O)(=O)C/C1=N\OC(=O)Nc2ccc(cc2)[N+](=O)[O-] RS-0078 Cc1ccc(cc1)NC(=O)O/N=C\2/CS(=O)(=O)CC2SC RS-0079 CSC\1CS(=O)(=O)C/C1=N/OC(=O)Nc2cccc(c2)[N+](=O)[O-] RS-0080 c1ccc(cc1)c2c(nc(s2)c3ccccc3)C(=O)N/N=C/4\N(C(=O)CS4)c5ccccc5 RS-0082 CC(C)(C)N(C=C(Cl)Cl)C(=O)n1cnc2c1cccc2 RS-0083 c1ccc(cc1)c2n[n-]nn2.c1cc(ccc1CC[NH3+])O.O RS-0084 CCCCCCCCOc1ccc(cc1)NS(=O)(=O)c2ccc3c(c2)nc([nH]3)NC(=O)OC RS-0085 CCCOc1c(c(c2n1c(cc(n2)C)C)C#N)C#N RS-0088 CC1OCC(CO1)(/[N+](=N/c2ccccc2[N+](=O)[O-])/[O-])[N+](=O)[O-] RS-0090 Cc1c(n(n[n+]1[O-])c2ccc(cc2)Br)N RS-0091 CCCCCCCCCCCC(=O)NC(CC)C(=O)O RS-0092 CCCCCCCCCCCC(=O)NC(CO)C(=O)O RS-0093 CCCCCCCCCCCCN(CCC(=O)O)C(=O)C RS-0094 Cc1ccccc1C(=N)Nc2[nH]nnn2.Cl RS-0099 CN(C)S(=O)(=O)c1ccccc1/C=N/O RS-0100 C(COc1c(non1)N)OCCOc2c(non2)N RS-0101 CC(C)(C)N(C=C(Cl)Cl)C(=O)OCc1cccc(c1)Oc2ccccc2 RS-0103 c1(c(non1)N)N RS-0105 c12c(c(n[nH]1)[N+](=O)[O-])[nH]nc2C(=O)N RS-0106 CCOCCN(C(C)C1CC1)C(=S)Nc2ccccc2 RS-0107 CC(C1CC1)N(Cc2ccccc2)C(=S)Nc3ccccc3 RS-0108 c1[nH]c(=S)[nH]n1 RS-0110 CCOC(=O)c1c(n(c2c1cc(cc2)O)C)C RS-0114 C(CCCN(CC(=O)O)CC(=O)O)CCN(CC(=O)O)CC(=O)O RS-0115 c1ccc(cc1)COC(=O)ON2C(=O)CCC2=O RS-0117 CC(C)/N=C\1/SCC(S1)(C)/C=N/O RS-0118 CCN(CC)C(=S)SCC(CN1C(=O)CCC1=O)S(=O)(=O)C RS-0122 CN(C)c1ccc(cc1)/C=C(/C(=O)c2ccc(cc2Cl)Cl)\n3ccnc3 RS-0124 CC(C)(C)OC(=O)N/C(=C\c1c[nH]c2c1cccc2)/C(=O)O RS-0125 c1cc(ccc1C23CC4CC(C2)CC(C4)(C3)C(=O)[O-])C56CC7CC(C5)CC(C7)(C6)C(=O)[O-].[Na+].[Na+] RS-0126 CC1(S(=O)(=O)CCS1(=O)=O)c2ccc(cc2Cl)Cl RS-0129 COc1cc(cc(c1)OC)/C=C/2\C=CC(=O)O2 RS-0130 COC(=O)c1c(sc(n1)n2c(=O)ccc(n2)O)c3ccccc3 RS-0131 COC(=O)c1c(sc(n1)NNC=O)c2ccccc2 RS-0132 COC(=O)Nc1[nH]c2ccc(cc2n1)S(=O)(=O)N3CCCCCC3 RS-0133 CCOC(=O)CC1=C(C(C(=C(O1)N)C#N)c2cccnc2)C(=O)OCC RS-0134 CC(OC(=O)N1CC2C(=CC1)C(=C([C@@]([C@@H]2c3ccc(cc3)C(F)(F)F)(C#N)C#N)N)C#N)(C)C RS-0137 COc1ccc(cc1Cn2cc(cn2)[N+](=O)[O-])C3C(=C(OC4=C3C(=O)CCC4)N)C#N RS-0139 CCCc1c2c(n[nH]1)OC(=C(C2c3ccoc3)C#N)N RS-0141 CC1CN(C(C(C1=O)/C=C(\C#N)/C(=S)N)C)C RS-0142 Cc1ccc(cc1)n2c3c(c(n2)C)C(C(=C(O3)N)C#N)c4ccccc4F RS-0145 Cc1ccc(cc1)n2c3c(c(n2)C)C(C(=C(O3)N)C#N)c4cccc(c4)Cl RS-0146 c1ccc(cc1)n2c3c(c(n2)C(F)(F)F)C(C(=C(O3)N)C#N)c4cccs4 RS-0147 Cc1ccc(cc1)n2c3c(c(n2)C)C(C(=C(O3)N)C#N)c4ccncc4 RS-0148 Cc1ccc(cc1)n2c3c(c(n2)C)C(C(=C(O3)N)C#N)c4ccco4 RS-0149 c1cc(cnc1)C2c3c([nH]nc3OC(=C2C#N)N)C(F)(F)F RS-0150 Cc1ccc(cc1)n2c3c(c(n2)C)C(C(=C(O3)N)C#N)c4c(cccc4Cl)F RS-0153 c1ccc(cc1)n2c3c(c(n2)C(F)(F)F)C(C(=C(O3)N)C#N)c4cccnc4 RS-0155 COc1ccccc1C2c3c([nH]nc3OC(=C2C#N)N)C(F)(F)F RS-0156 Cc1c(c(n(n1)Cc2cc(ccc2OC)C3c4c([nH]nc4OC(=C3C#N)N)c5ccccc5)C)[N+](=O)[O-] RS-0157 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(c(c3)Cn4cc(cn4)[N+](=O)[O-])OC)C(=O)C1)C RS-0158 CCO.Cc1c(c(n(n1)c2ccccc2)Cl)C3c4c([nH]nc4OC(=C3C#N)N)C(C)(C)C RS-0160 Cc1c(c(n(n1)c2ccccc2)Cl)C3c4c(c5ccccc5oc4=O)OC(=C3C#N)N RS-0161 CN1CCC2(CC1)c3c([nH]nc3OC(=C2C#N)N)c4ccccc4 RS-0162 CCOc1ccc(cc1)C2C3=C(CCCC3=O)OC(=C2[N+](=O)[O-])N RS-0163 CC(=O)n1c2ccccc2c3c1C(C(=C(O3)N)C#N)c4ccc(cc4)F RS-0164 COc1ccc2c(c1)oc3c2c(c(c(c3c4cccnc4)C#N)N)C#N RS-0165 C/C(=N/O)/C1C(OC(O1)(C)C)(C)C RS-0167 CC(C)(C)C(=O)CSc1[nH]cc([nH+]1)c2ccccc2.[Cl-] RS-0169 CCOC(=O)C1C2CC(C(C1Cl)Br)OC2=O RS-0170 CC1=C(C2(c3ccccc3NC2=O)C(=C(O1)N)C(=O)OC)C(=O)OC RS-0171 c1ccc(cc1)/[N+](=N/N2CCOC2=O)/[O-] RS-0172 c1ccc(cc1)CN2CCN(CC2)C(=O)C(C(F)(F)F)C(F)(F)F RS-0173 Cc1cc(n(n1)c2nc(c3c(n2)-c4ccccc4CC3)c5ccc(cc5)Br)C RS-0174 c1ccc(cc1)CNc2cc(nc(n2)c3ccc(cc3)[N+](=O)[O-])c4ccccc4 RS-0175 c1ccc(cc1)c2cc(nc(n2)c3ccc(cc3)[N+](=O)[O-])Nc4ccccc4 RS-0176 Cc1c(c(n[nH]1)C)CCCOc2ccc(cc2)OC.Cl RS-0178 CNC(=O)C1(CCON1OC)C(=O)NC RS-0179 Cc1ccc(cc1)S(=O)(=O)C(C#N)c2c(nc3ccccc3n2)Cl RS-0180 CN(CN1CC(CC1=O)c2ccccc2)S(=O)(=O)C RS-0181 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)Nc3ccc-4c(c3)C(=O)c5c4cccc5 RS-0182 CCOC(=O)CN1C(=O)N(C(C1(C)C)N(C(=O)Nc2ccc(cc2)Cl)O)c3ccc(cc3)Cl RS-0187 CC(C)(/C=N/O)NCC(=O)OC RS-0189 CC[N+](CC)(CCS(=O)(=O)CC)Cc1ccccc1.[I-] RS-0192 c1cc2c(cc(c(c2nc1)NNC(=O)c3ccco3)[N+](=O)[O-])[N+](=O)[O-] RS-0194 Cc1ccc(cc1)S(=O)(=O)NNc2c(cc(c3c2nccc3)[N+](=O)[O-])[N+](=O)[O-] RS-0196 Cc1cc(nc(n1)NCc2ccccc2)Oc3ccccc3 RS-0198 Cc1cc(nc(n1)N2CCOCC2)N3CCOCC3 RS-0199 CCC(=O)C1=C(CC(CC1=O)c2ccccc2)Nc3ccc(cc3)OC RS-0202 CCC(=O)C1=C(CC(CC1=O)c2ccccc2)NC(C)C(=O)O RS-0203 c1ccc(cc1)c2cc(nc(n2)N3CCOCC3)c4ccc(cc4)[N+](=O)[O-] RS-0204 Cc1cc(n(n1)c2nc(c(c(n2)c3ccccc3)[N+](=O)[O-])c4ccccc4)C RS-0205 c1ccc(cc1)c2c(c(nc(n2)N3CCCCC3)c4ccccc4)Oc5ccccc5 RS-0206 CN(C)c1nc(c(c(n1)c2ccccc2)NC(=O)c3ccc(cc3)Cl)c4ccccc4 RS-0207 CCOC(=O)c1ccccc1Nc2nc(c3c(n2)-c4ccccc4CC3)c5ccccc5 RS-0208 CCOC(=O)c1ccc(cc1)NC(=O)c2c(cn(n2)C)I RS-0211 Cc1cccc(c1n2c(nnn2)C3(CCCCC3)Nc4cc(on4)C)C RS-0212 CCCC1(N(N=C(S1)NC(=O)C)C(=O)C)C RS-0213 c1ccc(cc1)N2C(SCC2=O)c3ccccc3F RS-0214 COc1ccc(cc1)C2C3=C(CN(C3=O)Cc4ccccc4)NC(=O)N2 RS-0215 CCOC(=O)C1=C(NC(=O)NC1c2ccccc2)CBr RS-0216 c1ccc(cc1)CN2CC3=C(C2=O)C(NC(=O)N3)c4ccccc4 RS-0217 COc1ccc(cc1)OCCN2CCNCC2.Cl RS-0222 c1ccc(cc1)N2CN(CNC2=S)Cc3ccco3 RS-0223 COc1ccc(cc1)N2CNC(=S)N(C2)c3ccccc3 RS-0224 c1cc(cc(c1)Nc2nc(nc(n2)N)C(F)(F)F)C(F)(F)F RS-0225 CCn1cc(c(n1)C(=O)Nc2cccc(c2)SC)Br RS-0226 CC(C)CC1(N(N=C(S1)NC(=O)C)C(=O)C)c2ccccc2 RS-0227 CCCCSC(CO)CS(=O)CCCC RS-0228 CCCCS(=O)CC(CO)Sc1ccccc1 RS-0229 CCCCCCCCS(=O)CC(CS(=O)CCCCCCCC)O RS-0230 CCCCCCCCS(=O)CC(CO)S(=O)CCCCCCCC RS-0231 Cc1cccc(c1NC(=O)C2(CCCCC2)NC(=O)c3cccnc3)C RS-0232 Cc1cccc(c1NC(=O)C2(CCCCC2)N(C)C(=O)c3cccnc3)C RS-0233 Cc1ccccc1NC(=O)C2(CCCCC2)N(Cc3ccco3)C(=O)c4cccnc4 RS-0234 c1c(c(c2c(c1Cl)non2)[N+](=O)[O-])N3CCN(CC3)CCO RS-0236 CCCc1c2c([nH]n1)OC(=C(C2c3cc(c(c(c3)Br)O)OC)C#N)N RS-0237 c1ccc2c(c1)cccc2c3c4c([nH]n3)OC(=C(C4c5cc(ccc5O)Br)C#N)N RS-0238 CCN1CN(C(=S)SC1)CCOc2ccccc2 RS-0240 c1c2c(c3c(c1Br)non3)nno2 RS-0241 CC(c1ccc(cc1)C(C)(C)C)S(=O)CC(CO)O RS-0242 c1cc(ccc1CS(=O)CC(CO)O)Cl RS-0243 c1ccc(cc1)Oc2ccc(cc2)CS(=O)CC(CO)O RS-0244 COc1cc(c(cc1OC)Br)CC(=O)O RS-0245 COc1cc(c(cc1OC)[N+](=O)[O-])CC#N RS-0246 COc1ccc(cc1OC)/C(=C/c2ccccc2)/C(=O)O RS-0247 c1cc(c(c(c1)Cl)Cn2cc(cn2)N)F RS-0248 CCn1c(c(cn1)[N+](=O)[O-])C(=O)O RS-0249 CCn1cc(c(n1)C(=O)O)Cl RS-0250 Cc1c(cnn1CCC(=O)O)Cl RS-0251 CCOC(=O)Cn1c(c(c(n1)C(F)(F)F)Br)C RS-0252 c1cc(ccc1OCn2ccc(n2)C(=O)O)Br RS-0253 COc1ccc(cc1)OCCCl RS-0254 Cc1[nH]c(=S)[nH]n1 RS-0255 CCCCSc1[nH]ncn1 RS-0256 c1ccc2c(c1)nc(o2)SCC(=O)O RS-0257 c1nc(c(c(n1)Cl)N)NN RS-0258 Cc1c(c(n(n1)C(C)C(=O)Nc2cc(ccc2OC)Cl)C)[N+](=O)[O-] RS-0259 Cc1c(c(n(n1)C(C)C(=O)Nc2cc(ccc2Cl)Cl)C)[N+](=O)[O-] RS-0260 c1ccc(cc1)c2c(nc(nn2)c3ccccc3)NN RS-0264 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)O)C)[N+](=O)[O-] RS-0266 c1cc(c(c2c1non2)[N+](=O)[O-])SCC(=O)O RS-0268 COc1cc(c(cc1OC)I)CC(=O)O RS-0269 c1ccc(c(c1)C2N=C(Nc3n2c4ccccc4n3)N)O RS-0271 c1ccc2c(c1)cccc2C3N=C(Nc4n3c5ccccc5n4)N RS-0272 c1cc(oc1)/C=N/OCC(=O)O RS-0273 Cc1c(n(c2c1cccc2)C(=O)CCl)C RS-0274 Cc1c(cnn1CCC(=O)O)Br RS-0275 Cc1c(cn(n1)CCC(=O)O)Cl RS-0276 c1c(n(nc1C(F)(F)F)CCC(=O)O)C2CC2 RS-0277 Cc1nc([nH]n1)SCCO RS-0280 Cc1cc(=O)[nH]c(n1)SCC(=O)O RS-0282 CCn1cc(c(n1)C(=O)O)I RS-0284 C(C1C(=O)N=C(S1)N)C(=O)O RS-0285 CCOc1ccc(cc1)C2N=C(Nc3n2c4ccccc4n3)N RS-0286 COc1cc(cc(c1OC)OC)C2N=C(Nc3n2c4ccccc4n3)N RS-0287 Cc1cc(nn1Cc2ccc(cc2)Br)[N+](=O)[O-] RS-0288 c1c(c(n[nH]1)C(F)(F)F)Cl RS-0290 c1ccc(c(c1)OCn2ccc(n2)C(=O)O)Cl RS-0291 c1c(nc(s1)CCN)C(=O)O RS-0292 c1ccc(cc1)Cn2cc(c(n2)N)Cl RS-0294 Cc1cc(nn1Cc2ccccc2Cl)N RS-0295 Cc1ccc(cc1)Cn2c(c(c(n2)C)N)C RS-0296 CCc1c2ccccc2[nH]c1C(=O)OCC RS-0297 Cc1nc(cs1)CCN RS-0298 CCOC(=O)Cn1cc(c(n1)C)Br RS-0299 c1nc([nH]n1)SCCO RS-0301 CCn1c(c(cn1)I)C(=O)O RS-0302 c1cc(c(cc1Cl)Cl)OCn2ccc(n2)C(=O)NN RS-0303 Cc1c(cn(n1)CC(=O)NN)Br RS-0304 Cc1c(c(n(n1)C)C(=O)NN)Cl RS-0305 Cc1c(c(nn1CC(=O)NN)C(F)(F)F)Cl RS-0306 CCn1c(c(c(n1)C(=O)O)Cl)Br RS-0307 C1C(N=C2N1C=CC=C2)CBr.Br RS-0308 Cc1c(sc(c1C(=O)N)N)C RS-0309 Cn1c(c(cn1)I)C(=O)O RS-0310 Cn1cc(c(n1)C(=O)O)I RS-0311 C1CS(=O)(=O)CC1CC(=O)O RS-0314 CN(CC(=O)O)C1CCS(=O)(=O)C1 RS-0315 Cc1cc(nc(n1)CN)C.Cl RS-0317 Cc1cc(c2c(c1)cc(c(n2)Cl)C=O)C RS-0318 CCOc1ccc2c(c1)cc(c(n2)Cl)C=O RS-0319 Cc1csc2n1cc(n2)CCN.Cl RS-0320 COc1ccc(cc1)Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F RS-0321 COC(=O)c1cc2cc(ccc2[nH]1)Cl RS-0322 COC(=O)c1cc2cc(ccc2[nH]1)F RS-0323 COC(=O)c1cc2ccc(cc2[nH]1)Cl RS-0324 COC(=O)c1cc2ccc(cc2[nH]1)F RS-0325 Cn1c2ccc(cc2cc1C(=O)O)Cl RS-0326 Cn1c2ccc(cc2cc1C(=O)O)Br RS-0328 Cn1c2ccc(cc2cc1C(=O)O)F RS-0329 Cn1c2cc(ccc2cc1C(=O)O)Cl RS-0330 Cn1c2cc(ccc2cc1C(=O)O)Br RS-0331 COc1ccc2c(c1OC)cc([nH]2)C(=O)O RS-0332 Cn1c2ccc(c(c2cc1C(=O)O)OC)OC RS-0333 COc1cc2cc([nH]c2cc1OC)C(=O)O RS-0335 Cn1c(cc2c1c(c(c(c2)OC)OC)OC)C(=O)O RS-0336 Cc1ccc2c(c1)cc([nH]2)C(=O)NN RS-0337 COc1cc2cc([nH]c2cc1OC)C(=O)NN RS-0338 CCOc1ccc2c(c1)cc([nH]2)C(=O)NN RS-0339 c1cc2c(cc1Br)cc([nH]2)C(=O)NN RS-0340 CC1c2c(c3ccc(cc3[nH]2)OC)CCN1 RS-0341 c1ccn(c1)c2ccc(c(c2)C(=O)O)Cl RS-0342 c1cc(oc1)c2nnc(n2N)S RS-0344 Cc1c(c2ncc(c(n2n1)N)C#N)c3ccccc3 RS-0345 c1ccc(cc1)c2cnn3c2ncc(c3N)C#N RS-0346 c1c(nc(s1)CCN)C(F)(F)F.Cl RS-0347 Cc1c(sc(n1)CN)C RS-0348 CCc1nc(cs1)CN.Cl.Cl RS-0349 Cc1ccc(n1Cc2ccc(cc2)C(=O)O)C RS-0350 CN(Cc1ccc(o1)C=O)S(=O)(=O)C RS-0351 CCCn1cc(c(n1)C(=O)O)Br RS-0352 Cc1c(c(n(n1)C)Br)Br RS-0353 COC(=O)c1c(c[nH]n1)[N+](=O)[O-] RS-0354 Cc1c(c(n[nH]1)C(=O)O)Cl RS-0355 Cc1c(c(n[nH]1)C(=O)O)I RS-0357 c1(c([nH]nc1C(F)F)C(F)F)[N+](=O)[O-] RS-0358 C(C(=O)O)n1c(c(c(n1)C(F)F)[N+](=O)[O-])C(F)F RS-0359 Cc1c(cnn1C)C(=O)O RS-0360 CCn1cc(c(n1)C)C(=O)O RS-0361 CCn1c(c(cn1)Br)C(=O)O RS-0362 c1ccc(c(c1)Cn2cc(c(n2)C(=O)O)[N+](=O)[O-])Cl RS-0363 COC(=O)c1c(cn(n1)Cc2ccccc2Cl)[N+](=O)[O-] RS-0364 c1cc(cc(c1)Cl)Cn2cc(c(n2)C(=O)O)[N+](=O)[O-] RS-0365 c1ccc(c(c1)Cn2cc(c(n2)C(=O)O)Cl)Cl RS-0366 c1cc(cc(c1)Cl)Cn2c(cc(n2)[N+](=O)[O-])C(=O)O RS-0367 c1cc(c(cc1F)Cl)Cn2c(cc(n2)[N+](=O)[O-])C(=O)O RS-0368 Cc1ccc(o1)C(=O)O RS-0369 c1ccc(c(c1)c2nnc(o2)CCl)Br RS-0370 CC1CCCN(C1)c2ccc(cc2C#N)N RS-0371 c1cc(c(cc1N)C#N)N2CCOCC2 RS-0372 c1c[nH]nc1[N+](=O)[O-] RS-0374 Cc1c(cn(n1)CC(=O)O)Cl RS-0376 c1cnn(c1)Cc2ccc(o2)C(=O)O RS-0377 C1COCCC1N.Cl RS-0383 Cn1c2ccc(cc2nc1CN)C(F)(F)F.Cl RS-0384 Cc1c(c(n[nH]1)[N+](=O)[O-])I RS-0385 Cc1c(c(n(n1)c2ccc(cc2)C(=O)O)N)c3ccc(cc3)Cl RS-0386 CC(=O)N1CCOc2c1cc(cc2)S(=O)(=O)Cl RS-0387 c1ccc(c(c1)Cn2cc(c(n2)C(=O)O)Br)Cl RS-0388 c1cc(c(c(c1)Cl)Cn2cc(c(n2)C(=O)O)Br)F RS-0389 c1cc(ccc1Cn2cc(c(n2)C(=O)O)Cl)Cl RS-0390 Cc1c(c(n[nH]1)C(=O)OC)Cl RS-0391 Cc1c(c(n[nH]1)C(=O)OC)[N+](=O)[O-] RS-0393 c1c(cn(n1)CC(=O)O)Cl RS-0394 Cc1c(c(n(n1)CC(=O)O)C)Br RS-0395 c1c(cn(n1)CC(=O)O)Br RS-0396 Cc1ccc(c(c1N2CCCC2=O)C)S(=O)(=O)Cl RS-0397 Cc1ccc(cc1S(=O)(=O)Cl)N2CCCC2=O RS-0398 C1CC(COC1)C(=O)N RS-0399 Cc1cc(n(n1)CC(C)C(=O)O)C RS-0400 c1ccc(cc1)c2c(cn[nH]2)CN.Cl RS-0401 c1cn(cn1)CC(=O)O RS-0402 c1cc(cc(c1)N)c2nc3ccc(cc3o2)Cl RS-0404 Cc1nc(no1)CN.Cl RS-0406 CC(C(=O)[O-])N1CCOCC1.[Na+] RS-0407 c1cc(c(cc1F)Cl)Cn2cc(cn2)N.Cl RS-0409 c1ccc(cc1)C2=C[C@@H]3CC[C@H]2C=C3c4ccccc4 RS-1000 c1ccc2c(c1)c(c3ccccc3n2)N.O RS-1001 C(CCN)CC(=O)O RS-1002 c1cc(ccc1C#N)c2ccc(cc2)C#N RS-1004 c1c(sc(n1)Br)[N+](=O)[O-] RS-1007 C=Cc1ccccc1Br RS-1008 CCCCc1cc2cc(ccc2o1)C(=O)O RS-1009 COc1cc(nc(n1)OC)Cl RS-1011 c1cc(c(cc1C=O)Cl)[N+](=O)[O-] RS-1013 c1cc(ccc1C2(CC2)CO)Cl RS-1014 c1cc(ccc1C#N)C(=O)N RS-1015 c1ccc(cc1)C(=O)c2ccc(cc2)C#N RS-1016 c1ccc(cc1)COc2ccc(cc2OCc3ccccc3)C=O RS-1017 c1cc(c(cc1CC(=O)O)O)O RS-1018 Cc1c(sc(n1)C)C=O RS-1020 CCOC(=O)CC1CCCCC1=O RS-1022 CC(=O)CC(=O)c1ccco1 RS-1024 COC(=O)CC(=O)c1ccc(cc1)F RS-1029 c1ccc(cc1)C(=O)c2ccc3ccccc3c2 RS-1030 c1cc(ccc1/C=C/CO)[N+](=O)[O-] RS-1031 CCCCCOC(=O)c1cc(c(c(c1)OC)O)OC RS-1032 c1ccc(cc1)CC(=O)NN RS-1033 CC(C)(CCCC(C)(C)C(=O)O)C(=O)O RS-1035 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3cc(ccc3Cl)Cl)CO)N SS-0001 COC(=O)C1=C(Oc2c(=O)cc(oc2C1c3cc(ccc3Cl)Cl)CO)N SS-0002 CCOc1ccc(cc1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0003 COc1ccc(c(c1)OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0004 COc1cc(cc(c1)OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0005 COc1ccc(c(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)OC SS-0006 COc1cc(ccc1OCc2ccccc2)C3c4c(c(=O)cc(o4)CO)OC(=C3C#N)N SS-0007 c1cc(ccc1C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)OCC(=O)N SS-0008 Cc1cccc(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0009 c1cc(ccc1C(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)F SS-0010 c1cc(ccc1C(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)Cl SS-0011 c1cc(ccc1C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)O SS-0012 c1cc2c(cc1CNC(=O)c3c(c4cc5c(nc4s3)C6CCN5CC6)N)OCO2 SS-0013 CC(C)NC(=O)c1c(c2cc3c(nc2s1)C4CCN3CC4)N SS-0014 CC(=O)c1ccc(cc1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0016 c1cc(ccc1NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)F SS-0018 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)F)N)C(F)(F)F)C1 SS-0019 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)NCCc4ccc(cc4)F)N)C(F)(F)F)C1 SS-0020 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccccc4OC)N)C(F)(F)F)C1 SS-0021 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)OC)N)C(F)(F)F)C1 SS-0022 c1c2c(nc3c1c(c(s3)C(=O)N)N)CCCCCC2 SS-0023 CC(C)N1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccc5c(c4)OCO5)N)C1 SS-0024 c1c2c(nc3c1c(c(s3)C#N)N)CCCCCC2 SS-0026 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)N)N)C(F)(F)F)C1 SS-0027 c1c(c2c3c(c(cc(=O)[nH]3)O)sc2nc1C4CC4)C(F)(F)F SS-0028 CC(C)Oc1ccccc1C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0029 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)c4ccc(cc4)Cl)N)C(F)(F)F)C1 SS-0030 CC(=O)N1c2ccccc2C3(C1=O)c4c(c(=O)cc(o4)CO)OC(=C3C#N)N SS-0031 c1ccc2c(c1)C3(c4c(c(=O)cc(o4)CO)OC(=C3C#N)N)C(=O)N2Cc5cccc(c5)Br SS-0032 c1ccc(cc1)CNC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0034 c1cc(c(cc1NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)Cl)F SS-0035 c1csc(n1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0036 c1c(c(nc2c1N3CCC2CC3)SCC(=O)NC4CCCC4)C#N SS-0037 c1cc(c(cc1NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)C(F)(F)F)Cl SS-0038 c1cc(cc(c1)NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)C#N SS-0039 c1cc(c(cc1NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)Cl)F SS-0040 c1cc(ccc1NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)OC(F)(F)F SS-0041 c1cc(ccc1CNC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)F SS-0042 c1cc(cc(c1)F)NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N SS-0043 c1cc(cc(c1)Br)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0044 CC(C)N1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)OC)N)C1 SS-0045 CCc1c(c(c(c(n1)SCc2[nH]c3ccccc3n2)C#N)C(F)(F)F)C SS-0047 CC(C)N1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)OC(F)(F)F)N)C1 SS-0048 c1cc(cnc1)c2cc(c3c4c(c(cc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0050 c1cc2c(cc1C(=O)CSc3c(cc4c(n3)C5CCN4CC5)C#N)OCO2 SS-0051 c1ccc2c(c1)CCN(C2)C(=O)c3c(c4cc5c(nc4s3)C6CCN5CC6)N SS-0052 c1cc(oc1)c2cc(c3c4c(c(cc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0053 COc1ccc(cc1OC)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0054 COc1ccc(cc1NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)Cl SS-0055 CCOc1cccc(c1)NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N SS-0056 c1c(cc(cc1Cl)Cl)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0057 c1cc(ccc1CNC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)F SS-0058 c1c2c(nc3c1c4c(s3)c(ncn4)N)CCCCCC2 SS-0060 c1ccc2c(c1)[nH]c(n2)CSc3c(c(cc(n3)c4ccncc4)C(F)(F)F)C#N SS-0061 c1ccc2c(c1)[nH]c(n2)CSc3c(c(cc(n3)C4CC4)C(F)(F)F)C#N SS-0062 COc1ccccc1NC(=O)c2c(c3c(cc(nc3s2)Cc4ccccc4)C(F)(F)F)N SS-0063 COc1ccc(c(c1)c2cc(c(c(n2)SCc3[nH]c4ccccc4n3)C#N)C(F)(F)F)OC SS-0064 c1ccc(cc1)Cc2cc(c3c(c(sc3n2)C(=O)N)N)C(F)(F)F SS-0065 COc1ccc(c(c1)NC(=O)c2c(c3c(cc(nc3s2)Cc4ccccc4)C(F)(F)F)N)OC SS-0066 c1ccc(cc1)Cc2cc(c3c(c(sc3n2)C(=O)Nc4ccccc4F)N)C(F)(F)F SS-0067 c1ccc(cc1)Cc2cc(c(c(n2)SCC(=O)NCC(=O)O)C#N)C(F)(F)F SS-0068 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(cc3)Cl)CO)N SS-0069 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(cc3)OCC(=O)N SS-0070 Cc1ccc2c(c1)nc([nH]2)CSc3c(ccc(n3)c4ccncc4)C#N SS-0071 CN(C)c1nc(nc(n1)N)CSc2c(cc3c(n2)CCCCCC3)C#N SS-0072 c1cc(ccc1NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)OC(F)(F)F SS-0073 c1cc(ccc1CCNC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)Cl SS-0074 Cc1cc(no1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0075 COc1ccc(cc1OC)CCNC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N SS-0076 c1cc(c(cc1NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)F)F SS-0077 c1c2c(c(sc2nc3c1N4CCC3CC4)C(=O)N)N SS-0078 c1c2c(c(sc2nc3c1N4CCC3CC4)C(=O)Nc5nncs5)N SS-0079 CCOC(=O)c1ccc(cc1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0080 c1cc(ncc1CSc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N)Cl SS-0082 c1ccc(cc1)Cc2cc(c(c(n2)SCC(=O)N)C#N)C(F)(F)F SS-0083 CC(C)NC(=O)CSc1c(c(cc(n1)Cc2ccccc2)C(F)(F)F)C#N SS-0084 c1ccc(cc1)Cc2cc(c(c(n2)SCC(=O)NC3CC3)C#N)C(F)(F)F SS-0085 c1cc(ccc1NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)Cl SS-0086 COc1ccc(cc1OC)NC(=O)c2c(c3c(cc(nc3s2)Cc4ccccc4)C(F)(F)F)N SS-0087 c1c2c(nc3c1c(ns3)Br)CCCCC2 SS-0088 Cc1ccc2c(c1)nc([nH]2)CSc3c(c(cc(n3)c4ccco4)C(F)(F)F)C#N SS-0089 CCN(CC)C(=O)CSc1c(c(cc(n1)Cc2ccccc2)C(F)(F)F)C#N SS-0091 CCN(CC)C(=O)c1c(c2c(cc(nc2s1)Cc3ccccc3)C(F)(F)F)N SS-0092 c1c(cc(cc1Cl)Cl)NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N SS-0093 c1cc(cc(c1)F)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0095 c1cc(ccc1C(F)(F)F)NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N SS-0097 c1cc(ccc1NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)Cl SS-0098 c1cc(c(cc1Cl)NC(=O)CSc2c(cc3c(n2)C4CCN3CC4)C#N)Cl SS-0099 c1cc(cnc1)c2cc(c3c(c(sc3n2)C(=O)NCC(=O)O)N)C(F)(F)F SS-0100 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3c(c4ccc(nc4s3)c5cccnc5)N SS-0101 Cc1cc2c(c(=O)o1)C3(c4ccccc4N(C3=O)Cc5ccccc5Cl)C(=C(O2)N)C#N SS-0102 CCC1CCc2c(cc(c(n2)SCC(=O)N3CCCC3C(=O)O)C#N)C1 SS-0103 Cc1ccc(c(c1)F)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0106 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3c(c4cc5c(nc4s3)C6CCN5CC6)N SS-0107 COCCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(cc3)C(=O)OC)CO)N SS-0108 COCCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3cccc(c3Cl)Cl)CO)N SS-0109 CN1CCc2c(cc3c(c(sc3n2)C(=O)NCCc4c[nH]c5c4cccc5)N)C1 SS-0110 COCCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(c(c3)Cl)Cl)CO)N SS-0111 CCOc1ccccc1NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0112 c1ccc(c(c1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N)Cl SS-0113 c1ccc(cc1)COC(=O)C2=C(Oc3c(=O)cc(oc3C2c4ccc(cc4)F)CO)N SS-0114 c1ccc(cc1)COC(=O)C2=C(Oc3c(=O)cc(oc3C2c4cccnc4)CO)N SS-0115 CCOc1cccc(c1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0116 CN(C)c1ccc(cc1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0117 c1cnccc1c2cc(c3c4c(c(cc(n4)O)O)sc3n2)C(F)(F)F SS-0118 c1cc(ccc1CSc2c(cc3c(n2)C4CCN3CC4)C#N)Cl SS-0119 CC(C)OC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(c(c3)F)F)CO)N SS-0121 c1cc(cc(c1)F)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0122 c1ccc(cc1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0123 Cc1ccccc1C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0124 c1ccc(cc1)Oc2ccc(cc2F)C3c4c(c(=O)cc(o4)CO)OC(=C3C#N)N SS-0125 COc1cc(c(cc1OC)OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0126 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)OC(F)(F)F)N)C(F)(F)F)C1 SS-0127 c1cc(sc1)c2cc(c3c4c(c(cc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0128 c1ccc(cc1)Nc2nc3c(s2)c(cc(=O)[nH]3)O SS-0129 CCNc1nc2c(s1)c3c(c(=O)[nH]2)C(C(=C(O3)N)C#N)c4ccc(cc4)C SS-0130 Cc1c(c2c3c(c(cc(=O)[nH]3)O)sc2nc1C)C SS-0131 c1ccc(cc1)Nc2nc3c(s2)c4c(c(=O)[nH]3)C(C(=C(O4)N)C#N)c5ccc(cc5)Br SS-0132 Cc1cc(c(c(n1)SCC(=O)Nc2cc(c(cc2C(=O)OC)OC)OC)C#N)C(F)(F)F SS-0133 COC(=O)c1ccc(cc1NC(=O)CSc2c(cc3c(n2)CCCCC3)C#N)Cl SS-0134 CN(C)CCSc1c(c(cc(n1)c2ccc(cc2)Br)C(F)(F)F)C#N SS-0135 COC(=O)CC(=O)CSc1c(cc2c(n1)CCCCC2)C#N SS-0136 COc1cccc(c1)c2ccc3c4c(c(nc(=O)[nH]4)O)sc3n2 SS-0137 Cc1c(c2c3c(c(nc(=O)[nH]3)O)sc2nc1C)C SS-0138 COc1ccc(cc1)c2cc(nc3c2c4c(s3)c(nc(=O)[nH]4)O)c5cccs5 SS-0139 c1cc(sc1)c2cc(c3c4c(c(nc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0140 CN1CCc2c(cc3c4c(c(nc(=O)[nH]4)O)sc3n2)C1 SS-0141 COc1ccc(cc1OC)c2cc(c3c4c(c(nc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0142 COc1ccc(cc1)c2cc(c(c(n2)SCc3ccc(nc3)Cl)C#N)C(F)(F)F SS-0143 c1cc(ccc1c2cc(c(c(n2)SCc3ccc(nc3)Cl)C#N)C(F)(F)F)Cl SS-0144 Cc1cc(c(c(n1)SCc2ccc(nc2)Cl)C#N)C(F)(F)F SS-0145 c1cc(ncc1CSc2c(cc3c(n2)CCCCC3)C#N)Cl SS-0146 CC(C)(C)C1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4nccs4)N)C(F)(F)F)C1 SS-0147 CCOC(=O)C(C)Sc1c(c(cc(n1)Cc2ccccc2)C(F)(F)F)C#N SS-0148 Cc1ccc(c(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)C SS-0149 c1ccc(c(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)OCc4ccc(cc4)Cl SS-0150 c1ccc(c(c1)COc2ccccc2C3c4c(c(=O)cc(o4)CO)OC(=C3C#N)N)Cl SS-0151 CC(C)Oc1ccc(cc1OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0152 COc1ccc(c(c1OC)OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0153 COc1cccc(c1OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0154 COc1ccc(cc1)CNC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N SS-0155 C1Cc2c(nc3c(c2C(F)(F)F)c(c(s3)C(=O)NC45CC6CC(C4)CC(C6)C5)N)C1 SS-0156 Cc1cccc2c1nc(s2)NC(=O)c3c(c4c(c5c(nc4s3)CCC5)C(F)(F)F)N SS-0157 CSc1ccc(cc1)NC(=O)c2c(c3cc4c(nc3s2)CCCCC4)N SS-0158 CCN(CC)C(=O)CSc1c(c(cc(n1)C2CC2)C(F)(F)F)C#N SS-0159 CN1CCC2(CC1)c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0160 CCc1c(c(c2c(c(sc2n1)C(=O)NCc3ccc(cc3)F)N)C(F)(F)F)C SS-0161 CCc1c(c(c(c(n1)SCC(=O)Nc2ccc(cc2C)Br)C#N)C(F)(F)F)C SS-0162 CCc1c(c(c(c(n1)SCC(=O)NCc2ccc(cc2)OC)C#N)C(F)(F)F)C SS-0163 CC1CCc2c(c(c3c(c(sc3n2)C(=O)NCc4ccc(cc4)OC)N)C(F)(F)F)C1 SS-0164 COC(=O)c1ccc(cc1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0165 CC(=O)N1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4cccc(c4)C#N)N)C(F)(F)F)C1 SS-0166 Cc1ccc(cc1)CNC(=O)CSc2c(c(c3c(n2)CCC(C3)C(C)(C)C)C(F)(F)F)C#N SS-0167 CC(=O)N1CCc2c(c(c(c(n2)SCC(=O)Nc3ccccc3C(=O)OC)C#N)C(F)(F)F)C1 SS-0168 CC(=O)N1CCc2c(c(c(c(n2)SCC(=O)Nc3cccc(c3)C#N)C#N)C(F)(F)F)C1 SS-0169 COc1ccc(cc1OC)c2ccc3c4c(c(nc(=O)[nH]4)O)sc3n2 SS-0170 COc1ccc(cc1OC)CNC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N SS-0171 c1c2c(nc3c1c4c(s3)c(nc(=O)[nH]4)O)CCCC2 SS-0172 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3cc(ccc3Cl)[N+](=O)[O-])CO)N SS-0173 c1cc(oc1)c2cc(c3c(c(sc3n2)C(=O)c4ccc5c(c4)OCO5)N)C(F)(F)F SS-0174 c1cc2c(cc1c3cc(c4c(c(sc4n3)C(=O)c5ccc6c(c5)OCCO6)N)C(F)(F)F)OCO2 SS-0175 COC(=O)c1ccccc1NC(=O)CSc2c(cc3c(n2)CCCCC3)C#N SS-0176 Cc1ccc(cc1)CNC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N SS-0177 CC1CCc2c(c(c3c(c(sc3n2)C(=O)NCc4ccc(c(c4)OC)OC)N)C(F)(F)F)C1 SS-0178 CC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccccc4F)N)C(F)(F)F)C1 SS-0179 c1ccc(cc1)c2cc(c3c4c(c(c(c(=O)[nH]4)Br)O)sc3n2)c5ccc(cc5)Cl SS-0180 CC(C)(C)C1CCc2c(c(c(c(n2)SCC(=O)NCc3ccc(cc3)F)C#N)C(F)(F)F)C1 SS-0181 Cc1cc(c(c(n1)SCC(=O)Nc2ccc(cc2)SC)C#N)C(F)(F)F SS-0182 c1ccc(cc1)C2CCc3c(c(c(c(n3)SCC(=O)Nc4ccc(cc4)F)C#N)C(F)(F)F)C2 SS-0183 c1ccc(cc1)C2CCc3c(c(c(c(n3)SCCN4CCCC4)C#N)C(F)(F)F)C2 SS-0184 Cc1coc(n1)NC(=O)CSc2c(c(c3c(n2)CCC(C3)c4ccccc4)C(F)(F)F)C#N SS-0185 CC(=O)N1CCc2c(c(c(c(n2)SCC(=O)NCc3ccc(cc3)Cl)C#N)C(F)(F)F)C1 SS-0186 CC(C)(C)C1CCc2c(c(c(c(n2)SCC(=O)Nc3nccs3)C#N)C(F)(F)F)C1 SS-0187 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3c(cccc3Cl)F)CO)N SS-0188 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(c(c3)Cl)Cl)CO)N SS-0189 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(c(c3)F)F)CO)N SS-0190 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(cc3)F)CO)N SS-0191 COc1cccc(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0192 c1cc(c(cc1F)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)F SS-0193 c1cc(c(c(c1)Cl)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)Cl SS-0194 Cc1ccc(o1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0195 CCCOc1ccc(cc1OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0196 c1ccc(c(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)Cl SS-0197 c1ccc(c(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)F SS-0198 CNc1nc2c(s1)c3c(c(=O)[nH]2)C(C(=C(O3)N)C#N)c4cccc(c4)F SS-0199 CCC1CCc2c(c(c(c(n2)SCC(=O)Nc3nccs3)C#N)C(F)(F)F)C1 SS-0200 CCC1CCc2c(c(c(c(n2)SCC(=O)Nc3cccc(c3)OC)C#N)C(F)(F)F)C1 SS-0201 CCC1CCc2c(c(c(c(n2)SCC(=O)NCc3ccc(cc3)C)C#N)C(F)(F)F)C1 SS-0202 CCc1c(c(c(c(n1)SCC(=O)Nc2c(cccc2Cl)Cl)C#N)C(F)(F)F)C SS-0203 CCC1CCc2c(c(c(c(n2)SCc3ccc(cc3)C(=O)O)C#N)C(F)(F)F)C1 SS-0204 CCc1c(c(c2c(c(sc2n1)C(=O)NCCc3ccc(c(c3)OC)OC)N)C(F)(F)F)C SS-0205 CCc1c(c(c2c(c(sc2n1)C(=O)NCc3ccc(cc3)C)N)C(F)(F)F)C SS-0206 CCc1c(c(c2c(c(sc2n1)C(=O)Nc3ccccc3Cl)N)C(F)(F)F)C SS-0207 CCc1c(c(c(c(n1)SCC(=O)Nc2nc(cs2)C)C#N)C(F)(F)F)C SS-0208 CCc1c(c(c(c(n1)SCC(=O)NCc2ccc(cc2)F)C#N)C(F)(F)F)C SS-0209 CCc1c(c(c(c(n1)SCC(=O)Nc2ccc(c(c2)Cl)F)C#N)C(F)(F)F)C SS-0210 CCc1c(c(c(c(n1)SCC(=O)NC(C)c2ccccc2)C#N)C(F)(F)F)C SS-0211 CCc1c(c(c(c(n1)SCc2cccc(c2)F)C#N)C(F)(F)F)C SS-0212 CCc1c(c(c(c(n1)SCc2ccccc2Cl)C#N)C(F)(F)F)C SS-0213 CCc1c(c(c(c(n1)SCC(=O)Nc2c(c3c(s2)CCC3)C#N)C#N)C(F)(F)F)C SS-0214 Cc1cccc2c1nc(s2)NC(=O)c3c(c4c(c5c(nc4s3)CCCC5)C(F)(F)F)N SS-0215 Cc1cc(c2c3c(c(nc(=O)[nH]3)O)sc2n1)C(F)(F)F SS-0216 c1cc(ccc1Nc2nc3c(s2)c(cc(=O)[nH]3)O)F SS-0217 c1cc(ccc1Nc2c(c3c(s2)c(cc(=O)[nH]3)O)C#N)F SS-0218 c1cc(c(nc1)Cl)NC(=O)CSc2c(c(cc(n2)c3ccc4c(c3)OCO4)C(F)(F)F)C#N SS-0219 Cc1ccc(cc1)CNC(=O)CSc2c(c(c3c(n2)CCCCCC3)C(F)(F)F)C#N SS-0221 CC(C(=O)O)Sc1c(ccc(n1)c2cccnc2)C#N SS-0222 Cc1csc(n1)NC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N SS-0223 Cc1cc(ccc1NC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N)Br SS-0224 Cc1csc(n1)NC(=O)c2c(c3c(c4c(nc3s2)CCCC4)C(F)(F)F)N SS-0225 c1cc(cc(c1)NC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N)C#N SS-0226 Cc1ccccc1NC(=O)c2c(c3c(c4c(nc3s2)CCCCCC4)C(F)(F)F)N SS-0227 c1cc(cc(c1)NC(=O)c2c(c3c(c4c(nc3s2)CCCCC4)C(F)(F)F)N)C#N SS-0228 CCOC(=O)N1CCC(CC1)NC(=O)c2c(c3c(c4c(nc3s2)CCC(C4)C)C(F)(F)F)N SS-0229 c1cc(cc(c1)NC(=O)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N)C#N SS-0230 C1Cc2c(nc(c(c2C(F)(F)F)C#N)SCC(=O)NC34CC5CC(C3)CC(C5)C4)C1 SS-0231 COc1ccccc1NC(=O)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N SS-0232 c1cc(cc(c1)NC(=O)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N)C#N SS-0233 c1cc(c(cc1NC(=O)CSc2c(c(c3c(n2)CCCCCC3)C(F)(F)F)C#N)F)F SS-0234 CC1CCc2c(c(c(c(n2)SCC(=O)NCc3ccccc3)C#N)C(F)(F)F)C1 SS-0235 CC1CCc2c(c(c(c(n2)SCC(=O)NCc3ccccc3Cl)C#N)C(F)(F)F)C1 SS-0236 c1cc(ccc1NC(=O)CSc2c(c(c3c(n2)CCCCCC3)C(F)(F)F)C#N)F SS-0237 CN(C)c1ccc(cc1)NC(=O)CSc2c(c(c3c(n2)CCCCCC3)C(F)(F)F)C#N SS-0238 CC1CCc2c(c(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)C#N)C(F)(F)F)C1 SS-0239 CC1CCc2c(c(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)C#N)C(F)(F)F)C1 SS-0240 CCCCSc1c(c(c2c(n1)CCC(C2)C)C(F)(F)F)C#N SS-0241 CCCSc1c(c(c2c(n1)CCCCCC2)C(F)(F)F)C#N SS-0242 c1cc(cc(c1)F)CSc2c(c(c3c(n2)CCCCCC3)C(F)(F)F)C#N SS-0243 c1cc(ccc1CSc2c(c(c3c(n2)CCCCCC3)C(F)(F)F)C#N)C(=O)O SS-0244 COc1cc2c(cc1OC)CN(CC2)C(=O)c3c(c4c(c5c(nc4s3)CCC5)C(F)(F)F)N SS-0245 CCOC(=O)CCCSc1c(c(c2c(n1)CCC(C2)C)C(F)(F)F)C#N SS-0246 CC1CCc2c(c(c(c(n2)SCc3ccccc3F)C#N)C(F)(F)F)C1 SS-0247 CC(C(=O)C)Sc1c(c(c2c(n1)CCCCCC2)C(F)(F)F)C#N SS-0248 CC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4c(c5c(s4)CCCC5)C#N)N)C(F)(F)F)C1 SS-0249 CCOc1ccc(cc1)c2cc(c(c(n2)SCC(=O)Nc3nccs3)C#N)C(F)(F)F SS-0250 COc1cccc(c1)c2cc(c(c(n2)SCC(=O)Nc3nncs3)C#N)C(F)(F)F SS-0251 c1cc2c(cc1NC(=O)CSc3c(c(cc(n3)c4ccncc4)C(F)(F)F)C#N)OCCO2 SS-0252 CCOC(=O)c1ccc(cc1)NC(=O)CSc2c(c(cc(n2)c3ccncc3)C(F)(F)F)C#N SS-0253 Cc1coc(n1)NC(=O)CSc2c(c(cc(n2)c3ccncc3)C(F)(F)F)C#N SS-0254 COc1ccc(cc1OC)c2cc(c(c(n2)SCC(=O)Nc3nncs3)C#N)C(F)(F)F SS-0255 Cc1cccc2c1nc(s2)NC(=O)CSc3c(c(cc(n3)c4ccc(cc4)OC)C(F)(F)F)C#N SS-0256 CCOC(=O)N1CCC(CC1)NC(=O)CSc2c(c(cc(n2)c3ccc(cc3)Br)C(F)(F)F)C#N SS-0257 Cc1ccc(o1)c2cc(c3c(c(sc3n2)C(=O)c4ccc5c(c4)OCO5)N)C(F)(F)F SS-0258 c1cc(c(cc1c2cc(c3c(c(sc3n2)C(=O)N)N)C(F)(F)F)Cl)Cl SS-0260 c1ccc(cc1)c2cc(c(c(n2)SCC(=O)N3CCc4ccccc4C3)C#N)C(F)(F)F SS-0261 CC(=O)CSc1c(c(cc(n1)c2ccc3c(c2)OCO3)C(F)(F)F)C#N SS-0262 CC(c1ccccc1)Sc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0263 CC1CCc2c(c(c3c(c(sc3n2)C(=O)NCCc4ccccc4)N)C(F)(F)F)C1 SS-0265 c1cc(ccc1NC(=O)c2c(c3c(c4c(nc3s2)CCCCCC4)C(F)(F)F)N)F SS-0266 c1ccc(c(c1)NC(=O)c2c(c3c(c4c(nc3s2)CCCCCC4)C(F)(F)F)N)Cl SS-0267 c1cc2c(cc1C(=O)c3c(c4c(cc(nc4s3)c5ccncc5)C(F)(F)F)N)OCCO2 SS-0268 COc1ccc(c(c1)c2cc(c3c4c(c(cc(=O)[nH]4)O)sc3n2)C(F)(F)F)OC SS-0269 c1c(c2c(c3c(c4c(nc3s2)CCCCC4)C(F)(F)F)[nH]c1=O)O SS-0270 COc1ccc(c(c1)c2cc(c3c(c(sc3n2)C(=O)Nc4c(c5c(s4)CCCC5)C#N)N)C(F)(F)F)OC SS-0271 COc1ccc(c(c1)c2cc(c3c(c(sc3n2)C(=O)N4CCc5ccccc5C4)N)C(F)(F)F)OC SS-0272 c1ccc2c(c1)CCN(C2)C(=O)c3c(c4c(cc(nc4s3)c5ccc6c(c5)OCO6)C(F)(F)F)N SS-0273 COc1ccc(c(c1)c2cc(c(c(n2)SCC(=O)N3CCc4cc(c(cc4C3)OC)OC)C#N)C(F)(F)F)OC SS-0274 Cc1ccc(cc1)NC(=O)c2c(c3c(c4c(nc3s2)CCCC4)C(F)(F)F)N SS-0275 c1ccc2c(c1)CCN(C2)C(=O)c3c(c4c(c5c(nc4s3)CCCCC5)C(F)(F)F)N SS-0276 Cc1cc(ccc1NC(=O)CSc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N)Br SS-0277 Cc1ccccc1NC(=O)CSc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N SS-0278 Cc1ccc(cc1NC(=O)CSc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N)Cl SS-0279 c1ccc2c(c1)CCN(C2)C(=O)CSc3c(c(cc(n3)c4cccnc4)C(F)(F)F)C#N SS-0280 Cc1ccc(cc1NC(=O)c2c(c3c(c4c(nc3s2)CCCC4)C(F)(F)F)N)Cl SS-0281 COc1ccc(c(c1)OC)NC(=O)c2c(c3c(c4c(nc3s2)CCCC4)C(F)(F)F)N SS-0282 c1cc(c(cc1F)F)NC(=O)c2c(c3c(c4c(nc3s2)CCCC4)C(F)(F)F)N SS-0283 Cc1ccc(cc1)CSc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N SS-0284 c1cc(c(cc1CNC(=O)CSc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N)Cl)Cl SS-0285 COc1ccc(cc1)NC(=O)c2c(c3c(cc(nc3s2)c4ccc5c(c4)OCO5)C(F)(F)F)N SS-0286 Cc1ccc(o1)c2cc(c3c(c(sc3n2)C(=O)N)N)C(F)(F)F SS-0287 Cc1ccc(o1)c2cc(c3c(c(sc3n2)C(=O)OC)N)C(F)(F)F SS-0288 CCOC(=O)CCCSc1c(c(cc(n1)c2ccc(o2)C)C(F)(F)F)C#N SS-0289 Cc1ccc(o1)c2cc(c(c(n2)SCCC#N)C#N)C(F)(F)F SS-0290 Cc1csc(n1)NC(=O)c2c(c3c(c4c(nc3s2)CCCCC4)C(F)(F)F)N SS-0291 c1cc(c(cc1NC(=O)c2c(c3c(c4c(nc3s2)CCCCC4)C(F)(F)F)N)Cl)F SS-0292 CCOC(=O)CCSc1c(c(c2c(n1)CCCCC2)C(F)(F)F)C#N SS-0293 C1CCc2c(nc(c(c2C(F)(F)F)C#N)SCCN3CCCC3)CC1 SS-0294 c1ccc(c(c1)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N)Cl SS-0295 COc1ccc(cc1)CNC(=O)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N SS-0296 c1ccc(cc1)CNC(=O)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N SS-0297 c1cc(c(cc1Cl)Cl)CNC(=O)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N SS-0298 c1cc(c(cc1F)Cl)NC(=O)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N SS-0299 c1cc(c(cc1F)F)NC(=O)c2c(c3c(c4c(nc3s2)CCCCC4)C(F)(F)F)N SS-0300 CCN(CC)C(=O)CSc1c(c(c2c(n1)CCCCC2)C(F)(F)F)C#N SS-0301 Cc1cccc(c1)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N SS-0302 Cc1cc(ccc1NC(=O)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N)Br SS-0303 c1cc(ccc1CNC(=O)CSc2c(c(c3c(n2)CCCCC3)C(F)(F)F)C#N)Cl SS-0304 CC(C)(C)c1cc(c(c(n1)SCC(=O)N2CCc3ccccc3C2)C#N)C(F)(F)F SS-0305 c1cc(ccc1CNC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N)Cl SS-0307 c1cc(c(c(c1)Cl)NC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N)Cl SS-0308 COc1ccc(c(c1)OC)NC(=O)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N SS-0309 c1cc(c(c(c1)Cl)NC(=O)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N)Cl SS-0310 c1cc(ccc1CNC(=O)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N)Cl SS-0311 c1cc(c(cc1NC(=O)c2c(c3c(c4c(nc3s2)CCC4)C(F)(F)F)N)Cl)F SS-0312 c1cc(cc(c1)NC(=O)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N)C(F)(F)F SS-0313 CCN(CC)C(=O)CSc1c(c(c2c(n1)CCC2)C(F)(F)F)C#N SS-0314 c1cc(c(cc1NC(=O)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N)Cl)F SS-0316 c1cc(cc(c1)F)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N SS-0317 Cc1cccc(c1)CSc2c(c(c3c(n2)CCC3)C(F)(F)F)C#N SS-0318 CCOC(=O)CCSc1c(c(c2c(n1)CCC2)C(F)(F)F)C#N SS-0319 CCOC(=O)C(C)Sc1c(c(cc(n1)C2CC2)C(F)(F)F)C#N SS-0320 CCOC(=O)CCSc1c(c(cc(n1)C(C)(C)C)C(F)(F)F)C#N SS-0321 CCOC(=O)CCSc1c(c(cc(n1)C)C(F)(F)F)C#N SS-0322 CCOC(=O)CCCSc1c(c(cc(n1)c2ccc3c(c2)OCO3)C(F)(F)F)C#N SS-0323 CCOC(=O)CCSc1c(c(cc(n1)c2ccc3c(c2)OCO3)C(F)(F)F)C#N SS-0324 COc1ccc(cc1OC)c2cc(c(c(n2)SC(c3ccccc3)C(=O)O)C#N)C(F)(F)F SS-0326 CCOC(=O)NC(=O)CSc1c(c(cc(n1)c2ccc(c(c2)OC)OC)C(F)(F)F)C#N SS-0327 COc1ccc(cc1OC)c2cc(c3c4c(c(cc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0328 c1ccc(c(c1)CNC(=O)CSc2c(c(cc(n2)c3ccc(cc3)Cl)C(F)(F)F)C#N)Cl SS-0329 c1cc(cnc1)c2cc(c3c(c(sc3n2)C(=O)c4ccc(cc4)F)N)C(F)(F)F SS-0331 CNc1c(c2c(s1)c(cc(=O)[nH]2)O)C#N SS-0332 CCOC(=O)c1c2c(sc1NC(=O)c3c(c4c(cc(nc4s3)C5CC5)C(F)(F)F)N)CCCC2 SS-0333 Cc1ccc(cc1Br)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0334 CC(=O)c1c(c2c(cc(nc2s1)c3ccc4c(c3)OCO4)C(F)(F)F)N SS-0335 c1cc2c(cc1C(=O)CSc3c(c(cc(n3)c4ccncc4)C(F)(F)F)C#N)OCO2 SS-0336 c1cnccc1c2cc(c(c(n2)SCCN3CCCCCC3)C#N)C(F)(F)F SS-0337 Cc1coc(n1)NC(=O)c2c(c3c(cc(nc3s2)c4ccncc4)C(F)(F)F)N SS-0338 c1cnccc1c2cc(c3c4c(c(nc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0340 c1cc2c(cc1C(=O)c3c(c4c(cc(nc4s3)c5ccncc5)C(F)(F)F)N)OCO2 SS-0341 c1ccnc(c1)CSc2c(c(cc(n2)c3ccc4c(c3)OCCO4)C(F)(F)F)C#N SS-0342 c1ccc(cc1)CCSc2c(c(cc(n2)c3ccc4c(c3)OCCO4)C(F)(F)F)C#N SS-0343 c1c(c(c(nc1C23CC4CC(C2)CC(C4)C3)SCCC(=O)O)C#N)C(F)(F)F SS-0344 CC(C(=O)C)Sc1c(c(cc(n1)C23CC4CC(C2)CC(C4)C3)C(F)(F)F)C#N SS-0345 CCOC(=O)NC(=O)CSc1c(c(cc(n1)C23CC4CC(C2)CC(C4)C3)C(F)(F)F)C#N SS-0346 c1cc2c(cc1c3cc(c4c5c(c(nc(=O)[nH]5)O)sc4n3)C(F)(F)F)OCCO2 SS-0347 CCOC(=O)c1c(c(c(s1)NC(=O)c2c(c3c(cc(nc3s2)c4ccc5c(c4)OCCO5)C(F)(F)F)N)C#N)C SS-0348 c1cc2c(cc1c3cc(c4c(c(sc4n3)C(=O)N)N)C(F)(F)F)OCCO2 SS-0349 CC(=O)c1c(c2c(cc(nc2s1)c3ccc4c(c3)OCCO4)C(F)(F)F)N SS-0350 c1cc2c(cc1c3cc(c(c(n3)SCC#N)C#N)C(F)(F)F)OCCO2 SS-0351 CC(C(=O)C)Sc1c(c(cc(n1)c2ccc3c(c2)OCCO3)C(F)(F)F)C#N SS-0352 CC(c1ccccc1)Sc2c(c(cc(n2)c3ccc4c(c3)OCCO4)C(F)(F)F)C#N SS-0353 c1cc2c(cc1c3cc(c4c5c(c(cc(=O)[nH]5)O)sc4n3)C(F)(F)F)OCCO2 SS-0354 CCc1nnc(s1)NC(=O)CSc2c(c(cc(n2)c3cccnc3)C(F)(F)F)C#N SS-0355 CCc1nnc(s1)NC(=O)CSc2c(c(cc(n2)c3cccc(c3)OC)C(F)(F)F)C#N SS-0356 CC(C)(C)C(=O)c1c(c2c(cc(nc2s1)c3cccnc3)C(F)(F)F)N SS-0357 c1cc(cnc1)c2cc(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)C#N)C(F)(F)F SS-0358 c1cc2c(cc1C(=O)c3c(c4c(cc(nc4s3)C5CC5)C(F)(F)F)N)OCO2 SS-0360 c1c(c(c(nc1C2CC2)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)C#N)C(F)(F)F SS-0361 CCOC(=O)c1c2c(sc1NC(=O)CSc3c(c(cc(n3)C4CC4)C(F)(F)F)C#N)CCCC2 SS-0362 COc1cccc(c1)C(=O)CSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0363 COc1ccc(cc1)C(=O)CSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0364 c1cc(ccc1C(=O)CSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N)Cl SS-0365 COC(=O)CSc1c(c(cc(n1)C2CC2)C(F)(F)F)C#N SS-0366 CC(=O)CSc1c(c(cc(n1)C2CC2)C(F)(F)F)C#N SS-0367 CCSc1c(c(cc(n1)C2CC2)C(F)(F)F)C#N SS-0368 c1c(c(c(nc1C2CC2)SCCN3CCCCC3)C#N)C(F)(F)F SS-0369 c1ccc(cc1)CSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0370 c1cc(cc(c1)F)CSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0371 CC(C)(C)c1cc(c(c(n1)SCC(=O)c2ccc3c(c2)OCO3)C#N)C(F)(F)F SS-0372 COc1ccc(c(c1)OC)c2cc(c3c(c(sc3n2)C(=O)c4ccccc4)N)C(F)(F)F SS-0373 Cc1cc(c(c(n1)SCC(=O)C(C)(C)C)C#N)C(F)(F)F SS-0374 CCN(CC)C(=O)CSc1c(c(cc(n1)c2ccc(cc2)Br)C(F)(F)F)C#N SS-0375 Cc1ccc(cc1)S(=O)(=O)CCSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0376 COc1cccc(c1)c2cc(c3c(c(sc3n2)C(=O)N)N)C(F)(F)F SS-0377 COc1cccc(c1)c2cc(c3c(c(sc3n2)C(=O)OC)N)C(F)(F)F SS-0378 COc1cccc(c1)c2cc(c3c(c(sc3n2)C#N)N)C(F)(F)F SS-0379 CC(=O)c1c(c2c(cc(nc2s1)c3cccc(c3)OC)C(F)(F)F)N SS-0380 COC(=O)c1c(c2c(cc(nc2s1)c3ccc4c(c3)OCO4)C(F)(F)F)N SS-0381 c1cc2c(cc1c3cc(c(c(n3)SCC(=O)Nc4c(c5c(s4)CCCC5)C#N)C#N)C(F)(F)F)OCO2 SS-0382 CCOC(=O)c1c(c(c(s1)NC(=O)CSc2c(c(cc(n2)C(C)(C)C)C(F)(F)F)C#N)C#N)C SS-0383 CC(C)(C)c1cc(c(c(n1)SCC(=O)Nc2c(c3c(s2)CCCC3)C#N)C#N)C(F)(F)F SS-0384 COc1cccc(c1)c2cc(c(c(n2)SCC(=O)N)C#N)C(F)(F)F SS-0385 COc1cccc(c1)c2cc(c(c(n2)SCCN3CCOCC3)C#N)C(F)(F)F SS-0386 c1cnccc1c2cc(c(c(n2)SCC(=O)Nc3nccs3)C#N)C(F)(F)F SS-0387 COc1ccc(cc1)c2cc(c(c(n2)SCC(=O)Nc3cc(c(c(c3)OC)OC)OC)C#N)C(F)(F)F SS-0388 c1cnccc1c2cc(c3c(c(sc3n2)C(=O)C45CC6CC(C4)CC(C6)C5)N)C(F)(F)F SS-0389 COC(=O)c1c(c2c(cc(nc2s1)c3ccncc3)C(F)(F)F)N SS-0390 c1cnccc1c2cc(c3c(c(sc3n2)C#N)N)C(F)(F)F SS-0391 COc1ccc(cc1OC)C(=O)c2c(c3c(cc(nc3s2)c4ccco4)C(F)(F)F)N SS-0392 c1cc(ccc1c2cc(c3c(c(sc3n2)C#N)N)C(F)(F)F)Br SS-0393 c1cc(ccc1c2cc(c(c(n2)SCCC(=O)O)C#N)C(F)(F)F)Br SS-0394 COc1ccc(cc1)c2cc(c(c(n2)SCCCn3c4ccccc4[nH]c3=O)C#N)C(F)(F)F SS-0395 Cc1ccc(cc1)S(=O)(=O)CCSc2c(c(cc(n2)c3ccc(cc3)OC)C(F)(F)F)C#N SS-0396 COc1ccc(cc1OC)CCNC(=O)CSc2c(c(cc(n2)c3cccs3)C(F)(F)F)C#N SS-0397 COc1ccc(cc1OC)CCNC(=O)CSc2c(c(cc(n2)c3ccc4c(c3)OCO4)C(F)(F)F)C#N SS-0398 COC(=O)CSc1c(c(cc(n1)c2ccco2)C(F)(F)F)C#N SS-0399 CCOC(=O)CC(=O)CSc1c(c(cc(n1)c2ccc3c(c2)OCO3)C(F)(F)F)C#N SS-0401 c1cc2c(cc1c3cc(c(c(n3)SCCN4CCCCC4)C#N)C(F)(F)F)OCO2 SS-0402 C=CCSc1c(c(cc(n1)c2ccc3c(c2)OCO3)C(F)(F)F)C#N SS-0403 c1cc2c(cc1c3cc(c(c(n3)SCC(=O)Nc4ccc(c(c4)F)F)C#N)C(F)(F)F)OCO2 SS-0404 Cc1coc(n1)NC(=O)CSc2c(c(cc(n2)c3ccc4c(c3)OCO4)C(F)(F)F)C#N SS-0405 c1ccc(c(c1)NC(=O)CSc2c(c(cc(n2)c3ccc4c(c3)OCO4)C(F)(F)F)C#N)F SS-0406 CC(c1ccccc1)NC(=O)CSc2c(c(cc(n2)c3ccc4c(c3)OCO4)C(F)(F)F)C#N SS-0407 CC(C(=O)C)Sc1c(c(cc(n1)c2ccco2)C(F)(F)F)C#N SS-0408 CCOC(=O)C(C)Sc1c(c(cc(n1)c2ccco2)C(F)(F)F)C#N SS-0409 CSc1c(c(cc(n1)c2ccco2)C(F)(F)F)C#N SS-0410 CC(C(=O)C)Sc1c(c(cc(n1)c2ccc(c(c2)OC)OC)C(F)(F)F)C#N SS-0411 COc1ccc(cc1OC)c2cc(c(c(n2)SCC(=O)c3ccc(c(c3)O)O)C#N)C(F)(F)F SS-0412 CNc1nc2c(s1)c3c(c(=O)[nH]2)C(C(=C(O3)N)C#N)c4ccccc4 SS-0413 CCOC(=O)NC(=O)CSc1c(c(cc(n1)C)C(F)(F)F)C#N SS-0415 c1cc(c(c(c1)Cl)NC(=O)c2c(c3ccc(nc3s2)c4cccnc4)N)Cl SS-0416 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4nnc(s4)SCC(C)C)N)C1 SS-0417 CCC1CCc2c(cc3c(c(sc3n2)C(=O)c4ccc5c(c4)OCO5)N)C1 SS-0418 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cc(ccc4C)F)N)C1 SS-0419 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCCc4ccc(c(c4)OC)OC)N)C1 SS-0420 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4Cl)Cl)N)C1 SS-0421 COc1ccc(cc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)C(F)(F)F SS-0422 c1cc(c(cc1Br)F)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0423 COc1ccc(c(c1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)Cl SS-0424 Cc1ccc(cc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)Cl SS-0425 Cc1ccc(cc1Cl)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0426 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cc(cc(c4)Cl)Cl)N)C1 SS-0427 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCCc4ccc(cc4)Cl)N)C1 SS-0428 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)Cl)N)C1 SS-0429 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NC4CCCC4)N)C1 SS-0430 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4Cl)F)N)C1 SS-0431 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4F)Cl)N)C1 SS-0432 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4F)Br)N)C1 SS-0433 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(c(c4)F)C)N)C1 SS-0434 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cccc(c4)OCC)N)C1 SS-0435 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCCc4ccc(cc4)OC)N)C1 SS-0436 CCc1cccc(c1)NC(=O)c2c(c3cc4c(nc3s2)CCC(C4)CC)N SS-0437 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(c(c4)C)Br)N)C1 SS-0438 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(c(c4)C)C)N)C1 SS-0439 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4Br)C)N)C1 SS-0440 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(c(c4)Cl)C)N)C1 SS-0441 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cccc(c4C)Cl)N)C1 SS-0442 c1ccc(cc1)Oc2cc(ccc2F)C3C(=C(OC4=C3C(=O)CCC4)N)C#N SS-0443 c1ccc(cc1)COC(=O)CSc2c(c(cc(n2)c3ccco3)C(F)(F)F)C#N SS-0444 c1cc(oc1)c2cc(c(c(n2)SCc3ccncc3)C#N)C(F)(F)F SS-0445 c1ccnc(c1)CSc2c(c(cc(n2)c3ccco3)C(F)(F)F)C#N SS-0446 CCN(CC)C(=O)CSc1c(c(cc(n1)c2ccco2)C(F)(F)F)C#N SS-0447 c1ccc(cc1)C(C(=O)O)Sc2c(c(cc(n2)c3ccc(cc3)Br)C(F)(F)F)C#N SS-0448 c1cc2c(cc1[N+](=O)[O-])C3(c4c(c(=O)cc(o4)CO)OC(=C3C#N)N)C(=O)N2 SS-0449 COc1cc(c(cc1OC)[N+](=O)[O-])C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0450 c1ccc(c(c1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)[N+](=O)[O-] SS-0451 c1cc(cnc1)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0452 COc1cc(cc(c1OC)OC)C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N SS-0453 c1ccc2c(c1)C3(c4c(c(=O)cc(o4)CO)OC(=C3C#N)N)C(=O)N2 SS-0454 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)CC(C)C SS-0455 CCCCOc1ccc(cc1OC)C2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0456 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)C3CCC=CC3 SS-0457 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)Cc3ccccc3 SS-0458 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2cccc(c2)OCC(=O)N)C(=O)OC SS-0459 COc1ccc(cc1OC)c2cc(c3c(c(sc3n2)C(=O)NC4CC4)N)C(F)(F)F SS-0460 COc1ccc(cc1OC)c2cc(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)F)N)C(F)(F)F SS-0461 COc1ccc(cc1OC)c2cc(c3c(c(sc3n2)C(=O)c4ccc(c(c4)OC)OC)N)C(F)(F)F SS-0462 COc1ccc(cc1OC)c2cc(c(c(n2)SCC(=O)N)C#N)C(F)(F)F SS-0463 COc1ccc(cc1OC)NC(=O)c2c(c3c(cc(nc3s2)C45CC6CC(C4)CC(C6)C5)C(F)(F)F)N SS-0464 COc1ccc(cc1)NC(=O)c2c(c3c(cc(nc3s2)C45CC6CC(C4)CC(C6)C5)C(F)(F)F)N SS-0465 CCN(CC)C(=O)c1c(c2c(cc(nc2s1)C34CC5CC(C3)CC(C5)C4)C(F)(F)F)N SS-0466 c1cc2c(cc1C(=O)c3c(c4c(cc(nc4s3)C56CC7CC(C5)CC(C7)C6)C(F)(F)F)N)OCO2 SS-0467 c1c(c2c(c(sc2nc1C34CC5CC(C3)CC(C5)C4)C(=O)N)N)C(F)(F)F SS-0468 c1c(c2c(c(sc2nc1C34CC5CC(C3)CC(C5)C4)C(=O)O)N)C(F)(F)F SS-0469 c1ccc(cc1)C(C(=O)O)Sc2c(c(cc(n2)C34CC5CC(C3)CC(C5)C4)C(F)(F)F)C#N SS-0470 c1c(c2c3c(c(cc(=O)[nH]3)O)sc2nc1C45CC6CC(C4)CC(C6)C5)C(F)(F)F SS-0471 CCOC(=O)CSc1c(c(cc(n1)C23CC4CC(C2)CC(C4)C3)C(F)(F)F)C#N SS-0472 CCOC(=O)c1c(c2c(cc(nc2s1)C34CC5CC(C3)CC(C5)C4)C(F)(F)F)N SS-0473 c1c(c2c(c(sc2nc1C34CC5CC(C3)CC(C5)C4)C#N)N)C(F)(F)F SS-0474 c1c(c(c(nc1C23CC4CC(C2)CC(C4)C3)SCC(=O)NC5CC5)C#N)C(F)(F)F SS-0475 c1c(c2c(c(sc2nc1C34CC5CC(C3)CC(C5)C4)C(=O)NC6CC6)N)C(F)(F)F SS-0476 c1cc(ccc1C2c3c(c(=O)cc(o3)CO)OC(=C2C#N)N)Cl SS-0477 c1cc(ccc1c2cc(c3c(c(sc3n2)C(=O)NC4CC4)N)C(F)(F)F)Br SS-0478 Cc1cc(c(c(n1)SCC(=O)Nc2c(c3c(s2)CCC3)C#N)C#N)C(F)(F)F SS-0479 Cc1cc(no1)NC(=O)CSc2c(ccc(n2)c3cccnc3)C#N SS-0480 Cc1ccc(cc1)c2cc(c3c(c(sc3n2)C(=O)NC4CC4)N)C(F)(F)F SS-0481 Cc1ccc(cc1)c2cc(c3c(c(sc3n2)C(=O)c4ccc5c(c4)OCO5)N)C(F)(F)F SS-0482 Cc1ccc(cc1)c2cc(c(c(n2)SCC(=O)NC3CC3)C#N)C(F)(F)F SS-0483 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3ccccc3OC(F)(F)F)C#N)c4ccsc4)C1 SS-0484 c1c(c(c(nc1C23CC4CC(C2)CC(C4)C3)SCCC#N)C#N)C(F)(F)F SS-0485 COc1ccc(cc1OC)c2cc(c3c(c(sc3n2)C(=O)NC45CC6CC(C4)CC(C6)C5)N)C(F)(F)F SS-0486 COc1ccc(cc1)NC(=O)c2c(c3c(cc(nc3s2)c4ccc(c(c4)OC)OC)C(F)(F)F)N SS-0487 COc1ccc(cc1OC)c2cc(c3c(c(sc3n2)C(=O)c4ccc5c(c4)OCO5)N)C(F)(F)F SS-0488 COc1ccc(cc1)C(=O)c2c(c3c(cc(nc3s2)c4ccc(c(c4)OC)OC)C(F)(F)F)N SS-0489 c1cc(cnc1)c2ccc(c(n2)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)C#N SS-0490 c1cc(ccc1c2cc(c3c(c(sc3n2)C(=O)NC4CC4)N)C(F)(F)F)F SS-0491 c1cc(ccc1c2cc(c3c(c(sc3n2)C(=O)c4ccc5c(c4)OCO5)N)C(F)(F)F)F SS-0492 CCOC(=O)c1c(c(c(s1)NC(=O)CSc2c(c(cc(n2)c3ccc(cc3)F)C(F)(F)F)C#N)C#N)C SS-0493 c1cc(ccc1c2cc(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)C#N)C(F)(F)F)F SS-0494 COc1ccc(cc1)c2cc(c3c4c(c(cc(=O)[nH]4)O)sc3n2)C(F)(F)F SS-0495 COc1ccc(cc1)c2cc(c3c(c(sc3n2)C(=O)NC45CC6CC(C4)CC(C6)C5)N)C(F)(F)F SS-0496 COc1ccc(cc1)c2cc(c3c(c(sc3n2)C(=O)Nc4ccc(c(c4)OC)OC)N)C(F)(F)F SS-0497 CC(c1ccccc1)NC(=O)c2c(c3c(cc(nc3s2)c4ccc(cc4)OC)C(F)(F)F)N SS-0498 COc1ccc(cc1OC)c2cc(c(c(n2)SCC(=O)NC34CC5CC(C3)CC(C5)C4)C#N)C(F)(F)F SS-0499 CCOC(=O)C(C)Sc1c(c(cc(n1)c2ccc(c(c2)OC)OC)C(F)(F)F)C#N SS-0500 CCOC(=O)c1c(c(c(s1)NC(=O)CSc2c(c(cc(n2)c3ccc(c(c3)OC)OC)C(F)(F)F)C#N)C#N)C SS-0501 COc1ccc(cc1OC)c2cc(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)C#N)C(F)(F)F SS-0502 COc1ccc(cc1OC)c2cc(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)C#N)C(F)(F)F SS-0503 COc1ccc(cc1)c2cc(c(c(n2)SCC(=O)NC34CC5CC(C3)CC(C5)C4)C#N)C(F)(F)F SS-0504 CCOC(=O)c1c(c(c(s1)NC(=O)CSc2c(c(cc(n2)c3ccc(cc3)OC)C(F)(F)F)C#N)C#N)C SS-0505 COc1ccc(cc1)c2cc(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)C#N)C(F)(F)F SS-0506 COc1ccc(cc1)NC(=O)CSc2c(cc3c(n2)CCCCCC3)C#N SS-0507 c1c(c(c(nc1C23CC4CC(C2)CC(C4)C3)SCC#N)C#N)C(F)(F)F SS-0508 COC(=O)CSc1c(c(cc(n1)C23CC4CC(C2)CC(C4)C3)C(F)(F)F)C#N SS-0509 CCN(CC)C(=O)CSc1c(c(cc(n1)C23CC4CC(C2)CC(C4)C3)C(F)(F)F)C#N SS-0510 c1c(c(c(nc1C23CC4CC(C2)CC(C4)C3)SCC(=O)N)C#N)C(F)(F)F SS-0511 CCOC(=O)c1c(c(c(s1)NC(=O)CSc2c(cc3c(n2)CCN(C3)C)C#N)C#N)C SS-0512 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)C(C)C SS-0513 CCOC(=O)c1c(c(c(s1)NC(=O)CSc2c(cc3c(n2)CCCCCC3)C#N)C#N)C SS-0514 c1cc(ccc1CSc2c(cc3c(n2)CCCCCC3)C#N)C(=O)O SS-0515 CC(C)OC(=O)CC(=O)CSc1c(cc2c(n1)CCCCCC2)C#N SS-0516 c1c2c(nc(c1C#N)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)CCCCCC2 SS-0517 c1c2c(nc(c1C#N)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)CCCCCC2 SS-0518 CCOC(=O)c1c2c(sc1NC(=O)c3c(c4cc5c(nc4s3)CCCCCC5)N)CCCC2 SS-0519 c1cc2c(cc1C(=O)c3c(c4cc5c(nc4s3)CCCCC5)N)OCCO2 SS-0520 CN1CCc2c(cc(c(n2)SCC(=O)Nc3ccc(cc3)OC(F)(F)F)C#N)C1 SS-0521 CCOC(=O)c1c(c(c(s1)NC(=O)CSc2c(c(c3c(n2)CCN(C3)C)c4cccs4)C#N)C#N)C SS-0522 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCC4)C#N)C#N)c5cccs5)C1 SS-0523 CN1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)OC(F)(F)F)N)c5cccs5)C1 SS-0524 c1cc(ccc1NC(=O)c2c(c3cc4c(nc3s2)CCCCC4)N)OC(F)(F)F SS-0525 COc1ccccc1CSc2c(cc3c(n2)CCCCC3)C#N SS-0526 c1cc(cc(c1)Cl)CSc2c(cc3c(n2)CCCCC3)C#N SS-0527 c1ccc(c(c1)CSc2nnc(s2)NC(=O)c3c(c4ccc(nc4s3)c5ccncc5)N)Cl SS-0528 c1cc(ccc1CSc2nnc(s2)NC(=O)c3c(c4ccc(nc4s3)c5ccncc5)N)Cl SS-0529 CC(C)CSc1ccccc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0530 CCCSc1nnc(s1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0531 CCSc1ccccc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0532 CCCSc1nc2ccc(cc2s1)NC(=O)c3c(c4ccc(nc4s3)c5ccncc5)N SS-0533 CCSc1nc2ccc(cc2s1)NC(=O)c3c(c4ccc(nc4s3)c5ccncc5)N SS-0534 CCCCSc1nc2ccc(cc2s1)NC(=O)c3c(c4ccc(nc4s3)c5ccncc5)N SS-0535 C=CCSc1nc2ccc(cc2s1)NC(=O)c3c(c4ccc(nc4s3)c5ccncc5)N SS-0536 CN1CCc2c(c(c(c(n2)SCc3ccccc3OC)C#N)c4cccs4)C1 SS-0537 COc1ccc(cc1)C(=O)c2c(c3cc4c(nc3s2)CCCCC4)N SS-0538 CN1CCc2c(c(c(c(n2)SCC(=O)c3ccc(cc3)c4ccccc4)C#N)c5cccs5)C1 SS-0539 CC(C)OC(=O)CSc1c(c(c2c(n1)CCN(C2)C)c3cccs3)C#N SS-0540 CC(C)OC(=O)CSc1c(cc2c(n1)CCCCC2)C#N SS-0541 c1ccc(cc1)OCCSc2c(cc3c(n2)CCCCC3)C#N SS-0542 COc1ccc(c(c1)C2C(=C(OC(=C2C(=O)OC)CSc3c(cc4c(n3)CCCCC4)C#N)N)C#N)F SS-0543 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)C(C)(C)C)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0544 CC(C)OC(=O)C1=C(OC(=C(C1c2cc(cc(c2)OC)OC)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0545 CCOC(=O)C1=C(OC(=C(C1c2c(cccc2Cl)F)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0546 CCOC(=O)C1=C(OC(=C(C1c2ccsc2)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0547 Cc1ccc(c(n1)SCC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)OC)C(=O)OC)C#N SS-0548 CCOC(=O)C1=C(OC(=C(C1c2cccs2)C#N)N)CSc3c(c(c4c(n3)CCC(C4)C(C)(C)C)c5ccc(cc5)OC)C#N SS-0549 CC(C)OC(=O)C1=C(OC(=C(C1c2ccncc2)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0550 COc1cccc(c1)C2C(=C(OC(=C2C(=O)OC)CSc3c(cc4c(n3)CCCCC4)C#N)N)C#N SS-0551 CCOC(=O)C1=C(OC(=C(C1c2ccc(c(c2)Cl)Cl)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0552 CC(C)OC(=O)C1=C(OC(=C(C1c2ccccc2Cl)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0553 COc1cc2c(cc1OC)CN(CC2)C(=O)CSc3c(cc4c(n3)CCCCC4)C#N SS-0554 CN1CCc2c(cc(c(n2)SCc3cccc(c3)Br)C#N)C1 SS-0555 COc1ccc(cc1OC)NC(=O)CSc2c(cc3c(n2)CCCCC3)C#N SS-0556 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)C#N)c5ccsc5)C1 SS-0557 CCOC(=O)c1c2c(sc1NC(=O)CSc3c(c(c4c(n3)CCN(C4)C)c5cccs5)C#N)CCCC2 SS-0558 CCOC(=O)c1c2c(sc1NC(=O)CSc3c(c(cc(n3)C)C(F)(F)F)C#N)CCC2 SS-0559 c1c2c(nc(c1C#N)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)CCCCC2 SS-0560 CCOC(=O)c1c2c(sc1NC(=O)CSc3c(cc4c(n3)CCCCC4)C#N)CCC2 SS-0561 c1cc(ccc1NC(=O)c2c(c3cc4c(nc3s2)CCCCC4)N)F SS-0562 c1ccc(c(c1)NC(=O)c2c(c3cc4c(nc3s2)CCCCC4)N)OC(F)(F)F SS-0563 CN1CCc2c(cc(c(n2)SCc3ccccc3C(F)(F)F)C#N)C1 SS-0564 COc1cccc(c1)CSc2c(cc3c(n2)CCCCC3)C#N SS-0565 c1cc(cc(c1)F)NC(=O)CSc2c(cc3c(n2)CCCCC3)C#N SS-0566 c1cc(ccc1NC(=O)CSc2c(cc3c(n2)CCCCC3)C#N)F SS-0567 CC(C)Oc1ccc(cc1)C2c3c(c4c(c5cc6c(nc5s4)CCCCC6)[nH]c3=O)OC(=C2C#N)N SS-0568 CCCSc1ccccc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0569 CCN1CCc2c(cc(c(n2)SCC(=O)Nc3ccc(cc3)OC)C#N)C1 SS-0570 Cc1cc2c(c(=O)o1)C3(c4ccccc4NC3=O)C(=C(O2)N)C(=O)OC SS-0571 Cc1cc(nc2c1c3c(s2)c(cc(=O)[nH]3)O)C SS-0573 CC(c1ccccc1)NC(=O)CSc2c(c(c3c(n2)CCN(C3)C)c4cccs4)C#N SS-0574 Cc1cc(c(c(n1)SCC(=O)Nc2ccc(cc2)F)C#N)C(F)(F)F SS-0575 Cc1cc(c(c(n1)SCC(=O)Nc2nccs2)C#N)C(F)(F)F SS-0576 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(c(c4)F)F)N)C1 SS-0577 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4C)C)N)C1 SS-0578 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)C)N)C1 SS-0579 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(c(c4)Cl)F)N)C1 SS-0580 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cc(ccc4OC)Cl)N)C1 SS-0581 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cc(c(c(c4)OC)OC)OC)N)C1 SS-0582 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccc(cc4)C)N)C1 SS-0583 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NC(C)c4ccccc4)N)C1 SS-0584 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4C)OC)N)C1 SS-0585 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccc(cc4)OC)N)C1 SS-0586 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4OC)OC)N)C1 SS-0587 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccc(cc4)Cl)N)C1 SS-0588 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccccc4Cl)N)C1 SS-0589 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)C(F)(F)F)N)C1 SS-0590 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cc(ccc4F)F)N)C1 SS-0591 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccccc4C)N)C1 SS-0592 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccccc4OC)N)C1 SS-0593 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccc(cc4)F)N)C1 SS-0594 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4cccc(c4)Cl)N)C1 SS-0596 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccccc4OCC)N)C1 SS-0597 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cc(ccc4Cl)Cl)N)C1 SS-0598 COc1ccc(cc1)CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0599 c1cc(c(cc1Cl)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)Cl SS-0600 COCCOC(=O)C1=C(OC2=C(C1c3ccc(cc3)C(=O)OC)C(=O)CCC2)N SS-0601 c1ccc(c(c1)C(F)(F)F)NC(=O)c2c(c3cc4c(nc3s2)CCCCCC4)N SS-0603 COc1ccc(cc1)NC(=O)CS/C(=N\C#N)/Nc2ccccc2F SS-0604 c1cc(c(c(c1)F)NC(=O)CSc2c(c(cc(n2)c3cccs3)C(F)(F)F)C#N)F SS-0606 COC(=O)C1=C(OC(=C(C1c2ccc(cc2)F)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0607 COC(=O)C1=C(OC(=C(C1c2cccc(c2)F)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0608 COC(=O)C1=C(OC(=C(C1c2ccccc2F)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0609 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NC(C)C45CC6CC(C4)CC(C6)C5)N)C1 SS-0610 CCC1CCc2c(cc3c(c(sc3n2)C(=O)c4ccc(cc4)Br)N)C1 SS-0611 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NC4CC4)N)C1 SS-0612 CCC1CCc2c(cc3c(c(sc3n2)C(=O)c4ccc(cc4)F)N)C1 SS-0613 CCC1CCc2c(cc3c(c(sc3n2)C(=O)c4ccc(c(c4)OC)OC)N)C1 SS-0614 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4nc(cs4)C)N)C1 SS-0615 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cccc(c4)C(F)(F)F)N)C1 SS-0616 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cccc(c4)F)N)C1 SS-0617 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(c(c4)OC)OC)N)C1 SS-0618 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4F)F)N)C1 SS-0619 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCc4ccccc4)N)C1 SS-0620 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCCc4ccc(cc4)F)N)C1 SS-0621 COc1cc(cc(c1OC)OC)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0622 c1cc(cc(c1)F)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0623 Cc1ccc(cc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)F SS-0624 c1cc(c(cc1CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)Cl)Cl SS-0625 c1cc(nc2c1c(c(s2)C(=O)Nc3cc(cc(c3)Cl)Cl)N)c4ccncc4 SS-0626 c1cc(ccc1CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)Cl SS-0627 COc1ccc(cc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)Cl SS-0629 Cc1ccc(cc1F)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0630 Cc1cc(ccc1Br)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0631 c1ccc(cc1)C(=O)c2c(c3cc4c(nc3s2)CCCCC4)N SS-0632 c1cc(cc(c1)Cl)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0633 COc1cccc(c1OC)CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0634 CC(c1ccccc1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0635 Cc1cccc(c1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0636 c1cc(ccc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)F SS-0637 c1ccc(c(c1)CCNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)Cl SS-0639 CC(=O)c1ccc(cc1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0641 Cc1ccc(cc1)CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0642 Cc1cc(ccc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)OC SS-0643 c1cc(oc1)CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0644 COc1ccc(cc1OC)CCNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0646 c1cc(c(cc1F)F)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0647 COc1cccc(c1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0648 COc1ccccc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0649 COc1ccc(cc1OC)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0650 c1cc(c(cc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)C(F)(F)F)Cl SS-0651 c1ccc(c(c1)C(F)(F)F)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0652 c1cc(cc(c1)Cl)CCNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0653 COc1cc(cc(c1)OC)CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0654 c1cc(ccc1CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)C(F)(F)F SS-0655 Cc1ccc(c(c1)C)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0656 Cc1ccc(cc1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0657 c1ccc(cc1)CNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0658 c1cc(ccc1CCNC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)F SS-0659 c1cc(cc(c1)Br)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0660 COc1ccc(c(c1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)OC SS-0661 CCOc1ccccc1NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N SS-0662 Cc1ccc(c(c1)NC(=O)c2c(c3ccc(nc3s2)c4ccncc4)N)C SS-0663 CN1CCc2c(cc3c(c(sc3n2)C(=O)Nc4c(cccc4Cl)Cl)N)C1 SS-0664 c1cc(cnc1)c2ccc(c(n2)SCC#N)C#N SS-0665 Cc1cc(c(c(n1)S(=O)(=O)C)C#N)C(F)(F)F SS-0666 CN1CCc2c(c(c3c(c(sc3n2)C(=O)c4ccc(cc4)c5ccccc5)N)c6cccs6)C1 SS-0667 c1ccc(cc1)C(=O)CCCSc2c(cc3c(n2)CCCCC3)C#N SS-0668 CN1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)Cl)N)C1 SS-0669 CN1CCc2c(cc(c(n2)SCc3ccccc3F)C#N)C1 SS-0670 CC(C)(C)C(=O)c1c(c2cc3c(nc2s1)CCN(C3)C)N SS-0671 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3ccc(c(c3)OC)OC)C#N)c4cccs4)C1 SS-0672 CN1CCc2c(cc(c(n2)SCc3ccccc3Br)C#N)C1 SS-0673 c1cc(cnc1)CSc2c(cc3c(n2)CCCCCC3)C#N SS-0674 CCc1ccc(cc1)C2C(=C(OC(=C2C(=O)OC)CSc3c(ccc(n3)C)C#N)N)C#N SS-0675 CCOC(=O)c1c2c(sc1NC(=O)CSc3c(c(c4c(n3)CCN(C4)C)c5ccsc5)C#N)CCCC2 SS-0676 Cc1ccc(c(n1)SCC2=C(C(C(=C(O2)N)C#N)c3ccccc3Cl)C(=O)OC)C#N SS-0678 CCOC(=O)C1=C(OC(=C(C1c2cccc(c2)F)C#N)N)CSc3c(cc4c(n3)CCCCCC4)C#N SS-0679 c1cc(cc(c1)F)NC(=O)CSc2c(cc3c(n2)CCCCCC3)C#N SS-0680 CCOC(=O)c1c2c(sc1NC(=O)CSc3c(c(cc(n3)C)C(F)(F)F)C#N)CCCC2 SS-0681 COc1cc2c(cc1OC)CN(CC2)C(=O)CSc3c(ccc(n3)c4cccnc4)C#N SS-0682 c1ccc(c(c1)C(F)(F)F)NC(=O)c2c(c3cc4c(nc3s2)CCCCC4)N SS-0683 CN1CCc2c(c(c(c(n2)SCc3cccnc3)C#N)c4cccs4)C1 SS-0684 c1cc(cnc1)c2ccc(c(n2)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)C#N SS-0685 CN1CCc2c(cc(c(n2)SCC(=O)Nc3c(c4c(s3)CCCC4)C#N)C#N)C1 SS-0686 Cc1cc(c(c(n1)SCC(=O)Nc2c(c3c(s2)CCCC3)C#N)C#N)C(F)(F)F SS-0687 CN1CCc2c(c(c3c(c(sc3n2)C(=O)c4cccc(c4)OC)N)c5cccs5)C1 SS-0688 CN1CCc2c(c(c(c(n2)SCc3ccc(cc3)Cl)C#N)c4cccs4)C1 SS-0689 Cc1ccccc1CSc2c(c(c3c(n2)CCN(C3)C)c4cccs4)C#N SS-0690 CC(=O)CSc1c(c(c2c(n1)CCC(C2)C(C)(C)C)c3cccs3)C#N SS-0691 CN1CCc2c(c(c(c(n2)SC/C=C/c3ccccc3)C#N)c4cccs4)C1 SS-0692 CN1CCc2c(c(c3c(c(sc3n2)C(=O)c4ccc5c(c4)OCO5)N)c6cccs6)C1 SS-0693 CCc1c2c(n[nH]1)OC(=C(C2c3ccc(c(c3)OCC)OCCN4CCOCC4)C#N)N SS-0694 CCOC(=O)C1=C(OC(=C(C1c2cccc(c2)F)C#N)N)CSc3c(c(cc(n3)C)C)C#N SS-0695 c1cc(ccc1NC(=O)c2c(c3cc4c(nc3s2)CCCCCC4)N)F SS-0696 c1cc(ccc1NC(=O)c2c(c3cc4c(nc3s2)CCCCCC4)N)Cl SS-0697 c1cc(ccc1NC(=O)CSc2c(cc3c(n2)CCCCCC3)C#N)Cl SS-0698 Cc1ccc2c(c(sc2n1)C(=O)Nc3c(cccc3Cl)Cl)N SS-0699 c1cc(c(c(c1)Cl)NC(=O)c2c(c3cc4c(nc3s2)CCCCCC4)N)Cl SS-0700 c1cc(c(c(c1)Cl)NC(=O)c2c(c3cc4c(nc3s2)CCCCC4)N)Cl SS-0701 CC(C)(C)OC(=O)CSc1c(cc2c(n1)CCCCCC2)C#N SS-0702 Cc1ccccc1CSc2c(cc3c(n2)CCN(C3)C)C#N SS-0703 CN1CCc2c(cc(c(n2)SCCOc3ccccc3)C#N)C1 SS-0704 CN1CCc2c(c(c3c(c(sc3n2)C(=O)c4ccc(cc4)OC)N)c5cccs5)C1 SS-0705 CC1(CC2=C(C(=O)C1)C3(c4ccccc4N(C3=O)Cc5ccccc5)C(=C(O2)N)C#N)C SS-0706 Cc1c2c(n[nH]1)OC(=C(C23c4ccccc4N(C3=O)Cc5ccccc5)C#N)N SS-0707 Cc1c2c(n(n1)c3ccccc3)OC(=C(C24c5ccccc5N(C4=O)Cc6ccccc6)C#N)N SS-0708 CN1CCc2c(cc(c(n2)SCc3c(cccc3Cl)Cl)C#N)C1 SS-0709 CC(C)OC(=O)c1c(c2c(c3c(nc2s1)CCN(C3)C)c4cccs4)N SS-0710 Cc1cccc(c1NC(=O)CSc2c(c(c3c(n2)CCN(C3)C)c4cccs4)C#N)C SS-0711 CN1CCc2c(cc(c(n2)SCC(=O)Nc3ccc(cc3)F)C#N)C1 SS-0712 CCOC(=O)c1c2c(sc1NC(=O)CSc3c(c(c4c(n3)CCC4)c5cccs5)C#N)CCCC2 SS-0714 CN1CCc2c(cc(c(n2)SCC3=C(C(C(=C(O3)N)C#N)c4cccc(c4)OC)C(=O)OC)C#N)C1 SS-0715 CCOC(=O)C1=C(OC(=C(C1c2cccnc2)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0716 COC(=O)C1=C(OC(=C(C1c2cccc(c2)Br)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0717 COC(=O)C1=C(OC(=C(C1c2ccccc2)C#N)N)CSc3c(cc4c(n3)CCCCCC4)C#N SS-0718 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)F)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0719 CCc1c(cc(c(n1)SCc2cccnc2)C#N)C SS-0721 CCc1c(cc(c(n1)SCC(=O)O)C#N)C SS-0722 c1ccc(c(c1)/C=C/2\COCC3=C2OC(=C(C3c4ccccc4C(F)(F)F)C#N)N)C(F)(F)F SS-0723 CCCCOc1ccccc1C2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0724 CCOC1CC(=CC=C1OC(C)C)C2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0725 CC(C)c1c2c(n[nH]1)OC(=C(C2c3cc(c(c(c3)OC)OC)OC)C#N)N SS-0726 CCCc1c2c(n[nH]1)OC(=C(C2c3ccnc4c3cccc4)C#N)N SS-0727 CC(C)(C)c1c2c(n[nH]1)OC(=C(C2c3c(cccc3F)F)C#N)N SS-0728 CC(C)(C)c1c2c(n[nH]1)OC(=C(C2c3ccc(cc3)OC(F)(F)F)C#N)N SS-0729 c1cc(cc(c1)NC(=O)CSc2c(c(cc(n2)c3ccco3)C(F)(F)F)C#N)C(F)(F)F SS-0731 Cc1ccc(cc1)SCc2c3c(n[nH]2)OC(=C(C3c4ccc(c(c4)OC)OC(C)C)C#N)N SS-0732 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cc(ccc3F)OC)C(=O)C1)C SS-0733 CCCc1c2c(n[nH]1)OC(=C(C2c3cc(ccc3OC)OC)C#N)N SS-0734 CCCc1c2c(n[nH]1)OC(=C(C23CCN(CC3)C(=O)OCc4ccccc4)C#N)N SS-0735 Cc1c2c(n[nH]1)OC(=C(C23CCN(CC3)C(=O)OCc4ccccc4)C#N)N SS-0736 CC(C)Oc1ccc(cc1)[C@@H]2[C@H]3CN(CC=C3C(=C(C2(C#N)C#N)N)C#N)C SS-0737 CCOC(=O)N1CC=C2[C@H](C1)[C@H](C(C(=C2C#N)N)(C#N)C#N)c3cc(cc(c3)OC)OC SS-0738 CCOc1cc(ccc1OC(C)C)C2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0739 COc1ccc(cc1OC)NC(=O)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0740 COC(=O)C1=C(OC(=C(C1c2cccc(c2)Br)C#N)N)CSc3c(cc4c(n3)CCCCCC4)C#N SS-0742 COC(=O)C1=C(OC(=C(C1c2ccc(cc2)F)C#N)N)CSc3c(cc4c(n3)CCCCCC4)C#N SS-0743 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)COc4cccc(c4)OC)OC SS-0744 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C(=O)OC(C)C)c3ccc(cc3)C(F)(F)F SS-0745 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)c4ccc(c(c4)F)F SS-0746 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)F)F SS-0747 COCCOC(=O)C1=C(OC2=C(C1c3ccc(c(c3)F)F)C(=O)CCC2)N SS-0748 CC(C)(C)C1CCc2c(c(c3c(c(sc3n2)C(=O)c4ccc(cc4)OC)N)c5ccc(cc5)OC)C1 SS-0749 CC(C)(C)C1CCc2c(c(c(c(n2)SCc3ccccn3)C#N)c4cccs4)C1 SS-0750 CN1CCc2c(c(c(c(n2)SCc3c(cccc3Cl)Cl)C#N)c4cccs4)C1 SS-0751 Cc1cc(c2c(c(sc2n1)C(=O)c3ccc(cc3)F)N)C(F)(F)F SS-0752 CC(C)(C)C1CCc2c(c(c(c(n2)SCc3ccncc3)C#N)c4cccs4)C1 SS-0753 Cc1cc(c2c(c(sc2n1)C(=O)Nc3cc(no3)C)N)C(F)(F)F SS-0754 CC(C)(C)C1CCc2c(c(c(c(n2)SCC(=O)c3cccc(c3)OC)C#N)c4cccs4)C1 SS-0756 CC(C)(C)C1CCc2c(c(c(c(n2)SCCCC(=O)c3ccc(cc3)F)C#N)c4cccs4)C1 SS-0757 CN1CCc2c(c(c(c(n2)SCCS(=O)(=O)c3ccc(cc3)Cl)C#N)c4ccsc4)C1 SS-0758 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3ccc(c(c3)OC)OC)C#N)c4ccccc4)C1 SS-0759 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)OC)OCc4ccccc4 SS-0760 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)OC)OC(C)C SS-0761 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)Br)F SS-0762 CN1CCc2c(c(c(c(n2)N)C#N)c3ccccc3)C1 SS-0764 CCOC(=O)C1=C(OC2=C(C1c3cc(ccc3F)OC)C(=O)CC(C2)(C)C)N SS-0765 COc1cc2c(cc1OC)CN(CC2)C(=O)CSc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N SS-0766 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(cc3)F SS-0767 CC1(CC2=C(C(C(=C(O2)N)C(=O)OCCOC)c3ccc(cc3)C(=O)OC)C(=O)C1)C SS-0768 CC1(CC2=C(C(C(=C(O2)N)C(=O)OC)c3ccc(cc3)C(=O)OC)C(=O)C1)C SS-0769 CO/N=C(\c1csc(n1)NC(=O)CSc2c(c(cc(n2)c3ccccc3)C(F)(F)F)C#N)/C(=O)O SS-0771 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C(=O)OCCOC)c3ccc(cc3)C(F)(F)F SS-0772 CCCCOc1ccccc1C2C3=C(CCCC3=O)OC(=C2C(=O)OCC)N SS-0773 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C(=O)OC(C)C)c3cccc(c3)C(F)(F)F SS-0774 CN1CCc2c(c(c(c(n2)SCC(=O)CC(=O)OC)C#N)c3cccs3)C1 SS-0775 CC(C)(C)C1CCc2c(c(c(c(n2)SCC(=O)Nc3cccc(c3)F)C#N)c4cccs4)C1 SS-0776 CC(C)(C)C1CCc2c(c(c(c(n2)SCc3cccc(c3)OC)C#N)c4ccc(cc4)OC)C1 SS-0777 CC1(CC2=C(C(C(=C(O2)N)C(=O)OCCOC)c3ccc(c(c3)F)F)C(=O)C1)C SS-0778 COc1ccc(cc1OC)c2ccc3c4c(c(cc(=O)[nH]4)O)sc3n2 SS-0779 CC(C)(C)C1CCc2c(c(c(c(n2)SCC(=O)Nc3ccc(cc3)F)C#N)c4cccs4)C1 SS-0780 Cc1cc(nc(c1C#N)SCC2=C(C(C(=C(O2)N)C#N)c3ccccc3F)C(=O)OC)C SS-0781 Cc1cc(nc(c1C#N)SCC2=C(C(C(=C(O2)N)C#N)c3cccnc3)C(=O)OC)C SS-0782 CC(C)OC(=O)C1=C(OC2=C(C1c3ccc(c(c3)F)F)C(=O)CC(C2)(C)C)N SS-0783 CC(C)OC(=O)C1=C(OC2=C(C1c3ccc(c(c3)F)F)C(=O)CCC2)N SS-0784 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3c(cccc3Cl)F SS-0785 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3cccc(c3)OC SS-0786 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccccc3C(F)(F)F SS-0787 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccncc3 SS-0788 CC(C)(C)C1CCc2c(c(c3c(c(sc3n2)C(=O)c4ccc(cc4)F)N)c5cccs5)C1 SS-0789 CC(C)(C)C(=O)c1c(c2c(c3c(nc2s1)CCN(C3)C)c4cccs4)N SS-0790 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(cc3)Br SS-0791 CCOc1ccc(cc1OCC)C2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0792 CCOc1cc(ccc1O)C2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0795 CC(C)(C)C1CCc2c(c(c(c(n2)SCc3ccccc3Cl)C#N)c4ccccc4)C1 SS-0796 CCOC(=O)CC1=C(C(C(=C(O1)N)C#N)c2ccsc2)C(=O)OCC SS-0797 Cc1cc(c(c(n1)SCCN2CCCCC2)C#N)C(F)(F)F SS-0798 CCOC(=O)C1=C(Oc2cc(oc(=O)c2C1c3c(cccc3Cl)Cl)C)N SS-0799 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(cc3)OCc4ccccc4 SS-0800 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3cc(c(c(c3)OC)O)[N+](=O)[O-] SS-0801 Cc1ccc(o1)[C@@H]2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0802 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)OCc4ccccc4)OC SS-0803 CC(C)(C)C1CCc2c(c(c(c(n2)SCC(=O)OC)C#N)c3cccs3)C1 SS-0804 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3cccc(c3)[N+](=O)[O-] SS-0805 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3cccc(c3)Cl SS-0806 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3c(cccc3Cl)Cl SS-0807 Cc1cc2c(c(=O)o1)[C@H](C(=C(O2)N)C#N)c3ccccc3[N+](=O)[O-] SS-0808 CCOc1ccc(cc1)C2c3c(cc(oc3=O)C)OC(=C2C#N)N SS-0809 CCOC(=O)CC1=C([C@H](C(=C(O1)N)C#N)c2ccccc2[N+](=O)[O-])C(=O)OCC SS-0810 COCC1=C(C(C(=C(O1)N)C#N)c2cccc(c2)Br)C(=O)OC SS-0811 COCC1=C(C(C(=C(O1)N)C#N)c2ccccc2F)C(=O)OC SS-0812 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)COc4ccc(cc4F)F)OC SS-0813 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3cc(ccc3F)Br SS-0814 COc1cc(cc(c1OC)OC)C2c3c(c4ccccc4oc3=O)OC(=C2C#N)N SS-0816 CC(C)(C)c1c2c(n[nH]1)OC(=C(C2c3ccc(cc3)SC)C#N)N SS-0817 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)Cl)Cl SS-0818 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(cc3)c4ccccc4 SS-0819 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3ccc(c(c3)[N+](=O)[O-])Cl SS-0820 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3cccc(c3)F SS-0821 Cc1cc2c(c(=O)o1)C(C(=C(O2)N)C#N)c3cccc(c3Cl)Cl SS-0822 CCOC(=O)C1=C(OC(=C(C1c2ccc(s2)[N+](=O)[O-])C#N)N)CSc3c(cc4c(n3)CCC4)C#N SS-0823 CC(C)OC(=O)CC(=O)CSc1c(ccc(n1)c2cccnc2)C#N SS-0824 CC(C)(C)OC(=O)CSc1c(cc2c(n1)CCCCC2)C#N SS-0825 CC(C)OC(=O)CC(=O)CSc1c(cc2c(n1)CCCCC2)C#N SS-0826 c1ccc(cc1)COC(=O)c2c(c3cc4c(nc3s2)CCCCC4)N SS-0827 CC(C)OC(=O)c1c(c2cc3c(nc2s1)CCCCC3)N SS-0828 c1ccc(c(c1)CSc2c(cc3c(n2)CCCCC3)C#N)C(F)(F)F SS-0829 c1cc(cnc1)c2ccc(c(n2)SCCC3OCCO3)C#N SS-0830 CC(C)(C)C1CCc2c(c(c(c(n2)SCCOC3CCCCO3)C#N)c4cccs4)C1 SS-0831 CC(C)(C)C1CCc2c(c(c(c(n2)SCc3ccc(cc3)[N+](=O)[O-])C#N)c4cccs4)C1 SS-0832 c1cc(ccc1CSc2c(cc3c(n2)CCCCC3)C#N)[N+](=O)[O-] SS-0833 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)Br)N)C1 SS-0835 CCC1CCc2c(cc3c(c(sc3n2)C(=O)c4ccc(cc4)C)N)C1 SS-0836 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4ccc(cc4)OC)N)C1 SS-0837 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cccc(c4)C)N)C1 SS-0838 CCC1CCc2c(cc3c(c(sc3n2)C(=O)NCCc4ccccc4)N)C1 SS-0839 CCC1CCc2c(cc3c(c(sc3n2)C#N)N)C1 SS-0840 CCC1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cccc(c4)Br)N)C1 SS-0841 Cc1cc(c2c3c(c(cc(=O)[nH]3)O)sc2n1)c4ccccc4 SS-0842 CN1CCc2c(cc3c(c(sc3n2)C(=O)Nc4cccc(c4)F)N)C1 SS-0843 CC(C)OC(=O)CC(=O)c1c(c2cc3c(nc2s1)CCN(C3)C)N SS-0844 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)C#N)N)CSc3c(ccc(n3)c4ccncc4)C#N SS-0845 COc1cccc(c1)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0846 c1c2c(nc(c1C#N)SCC(=O)O)CCCCC2 SS-0848 Cc1cc(c(c(n1)SCC(=O)CC(=O)OC)C#N)C(F)(F)F SS-0849 Cc1cc(c(c(n1)SCC(=O)CC(=O)OC(C)C)C#N)C(F)(F)F SS-0850 CC(C)(C)c1ccc(cc1)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0851 CC(C)NC(=O)c1c(c2c(cc(nc2s1)c3cccs3)C(F)(F)F)N SS-0852 c1ccc(cc1)C(=O)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0853 Cc1cc(c(c(n1)SCC(=O)NCc2ccccc2)C#N)C(F)(F)F SS-0854 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3ccc(cc3)F)C#N)c4ccccc4)C1 SS-0855 CCOC(=O)C1=C(OC(=C(C1c2cccnc2)C#N)N)CSc3c(ccc(n3)c4ccccc4)C#N SS-0856 c1cc(cnc1)c2c3c(nc4c2c(c(s4)C(=O)c5ccc(cc5)F)N)CCCC3 SS-0857 CCCCOc1ccc(cc1OC)c2c(c(nc(c2C#N)SCC(=O)C34CC5CC(C3)CC(C5)C4)N)C#N SS-0858 CCOC(=O)C1=C(NC(=S)[C@]([C@@H]1c2cccs2)(CC=C)C#N)C SS-0859 c1cc(cnc1)c2c3c(nc4c2c(c(s4)C(=O)C56CC7CC(C5)CC(C7)C6)N)CCCC3 SS-0860 CN1CCc2c(cc3c(c(sc3n2)C(=O)N)N)C1 SS-0861 c1cc2c(cc1[N+](=O)[O-])sc(n2)NC(=O)CSc3c(ccc(n3)C45CC6CC(C4)CC(C6)C5)C#N SS-0862 Cc1cc(c2c3c(c(cc(=O)[nH]3)O)sc2n1)c4cccs4 SS-0863 c1cc(cc(c1)F)NC(=O)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0864 Cc1cc(nc2c1c(c(s2)C(=O)NC(C)c3ccccc3)N)C SS-0865 Cc1cc(nc2c1c(c(s2)C(=O)Nc3ccc(cc3)F)N)C SS-0866 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)SC)C#N)N)CSc3c(ccc(n3)c4ccccc4)C#N SS-0867 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)OC)C#N)N)CSc3c(ccc(n3)c4ccncc4)C#N SS-0868 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)F)C#N)N)CSc3c(cc4c(n3)CCN(C4)C)C#N SS-0869 CCOC(=O)C1=C(OC(=C(C1c2cccnc2)C#N)N)CSc3c(ccc(n3)c4ccncc4)C#N SS-0870 CCOC(=O)C1=C(OC(=C(C1c2ccccc2C(F)(F)F)C#N)N)CSc3c(cc4c(n3)CCN(C4)C)C#N SS-0871 CCOC(=O)C1=C(OC(=C(C1c2ccccc2)C#N)N)CSc3c(cc4c(n3)CCN(C4)C)C#N SS-0872 c1c2c(nc3c1c4c(s3)c(cc(=O)[nH]4)O)CCCCCC2 SS-0874 Cc1cc(c2c3c(c(cc(=O)[nH]3)O)sc2n1)C(F)(F)F SS-0875 CCOC(=O)CC(=O)CSc1c(c(c2c(n1)CCC(C2)C(C)(C)C)c3cccs3)C#N SS-0876 CCN1CCc2c(c(c3c(c(sc3n2)C(=O)c4ccccc4)N)C(=O)OCC)C1 SS-0877 CN1CCc2c(cc3c(c(sc3n2)C(=O)c4ccc(cc4)OC)N)C1 SS-0878 CN1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccccc4)N)c5cccs5)C1 SS-0880 Cc1cccc(c1)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0882 c1cc(cnc1)c2ccc3c(c(sc3n2)C(=O)c4ccc(cc4)F)N SS-0883 Cc1cc(c2c(c(sc2n1)C(=O)Nc3ccc(cc3)F)N)C(F)(F)F SS-0884 Cc1cc(nc(c1C#N)SCc2c3c([nH]n2)OC(=C(C3c4ccccc4[N+](=O)[O-])C#N)N)C SS-0885 CN1CCN(CC1)C(=O)CSc2c(ccc(n2)c3cccs3)C#N SS-0886 CN1CCN(CC1)C(=O)CSc2c(c(cc(n2)c3cccs3)c4ccc(cc4)Cl)C#N SS-0887 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2F)Br)C#N)N)CSc3c(c(cc(n3)C)C)C#N SS-0888 c1cc(sc1)c2cc(c3c4c(c(cc(=O)[nH]4)O)sc3n2)c5ccc(cc5)F SS-0890 c1cc(sc1)c2cc(c(c(n2)SCc3ccncc3)C#N)c4ccc(cc4)F SS-0894 Cc1cc(n(n1)C(=O)CSc2c(c(cc(n2)c3ccccc3)C(F)(F)F)C#N)C SS-0895 Cc1cc(n(n1)C(=O)CSc2c(c(cc(n2)c3cccs3)c4cccs4)C#N)C SS-0896 Cc1cc(n(n1)C(=O)CSc2c(c(cc(n2)c3cccs3)c4ccc(cc4)OC)C#N)C SS-0897 COc1ccccc1c2cc(nc3c2c4c(s3)c(cc(n4)O)O)c5cccs5 SS-0898 CCOC(=O)C1=C(OC(=C(C1c2cccnc2)C#N)N)CSc3c(c(cc(n3)c4cccs4)c5ccc(cc5)Cl)C#N SS-0899 CN1CCc2c(cc3c4c(c(cc(=O)[nH]4)O)sc3n2)C1 SS-0900 c1cc(nc2c1c3c(s2)c(cc(n3)O)O)C45CC6CC(C4)CC(C6)C5 SS-0901 c1cc(nc(c1C#N)SCCN2CCCCC2)C34CC5CC(C3)CC(C5)C4 SS-0903 c1cc(cnc1)c2ccc(c(n2)SCC(=O)c3ccc(cc3)Cl)C#N SS-0904 c1ccc(cc1)C(=O)CSc2c(ccc(n2)c3cccnc3)C#N SS-0905 CCOC(=O)CSc1c(ccc(n1)c2cccnc2)C#N SS-0906 Cc1cc(nc2c1c(c(s2)C(=O)Nc3ccc(cc3)OC)N)C SS-0907 CCOC(=O)c1c(c2ccc(nc2s1)c3cccnc3)N SS-0910 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3nc4ccccc4s3)C#N)c5ccsc5)C1 SS-0911 CN1CCc2c(c(c(c(n2)SCC(=O)Nc3ccccc3)C#N)c4ccsc4)C1 SS-0912 c1ccc2c(c1)nc(s2)NC(=O)CSc3c(ccc(n3)C45CC6CC(C4)CC(C6)C5)C#N SS-0913 Cc1csc(n1)NC(=O)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0914 CCc1nnc(s1)NC(=O)CSc2c(ccc(n2)C34CC5CC(C3)CC(C5)C4)C#N SS-0915 CCOC(=O)CC(=O)CSc1c(c(cc(n1)C)C(F)(F)F)C#N SS-0917 COc1ccc(cc1)c2cc(nc(c2C#N)SCCN3CCCCC3)c4ccccc4 SS-0918 CCOC(=O)C1=C(OC(=C(C1c2ccccc2I)C#N)N)CSc3c(c(c(c(n3)C)C)C)C#N SS-0920 C=CCOc1ccc(cc1)C2c3c(c4ccccc4oc3=O)OC(=C2C#N)N SS-0922 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)OCc4ccccc4)C(=O)C1)C SS-0923 c1cc(cc(c1)NC(=O)CSc2c(cc3c(n2)CCCCCC3)C#N)C(F)(F)F SS-0924 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0925 CCc1c(cc(c(n1)SCC2=C(C(C(=C(O2)N)C#N)c3ccccc3)C(=O)OCC)C#N)C SS-0926 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)C#N)N)CSc3c(cc4c(n3)CCCCCC4)C#N SS-0927 CCOC(=O)C1=C(OC(=C(C1c2ccccc2F)C#N)N)CSc3c(cc4c(n3)CCCCCC4)C#N SS-0928 CCOC(=O)C1=C(OC(=C(C1c2ccccc2Cl)C#N)N)CSc3c(cc4c(n3)CCCCCC4)C#N SS-0929 CCOC(=O)C1=C(OC(=C(C1c2ccccc2)C#N)N)CSc3c(cc4c(n3)CCCCC4)C#N SS-0931 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)C#N)N)CSc3c(c(cc(n3)C)C)C#N SS-0932 c1cc(nc(c1C#N)SCC(=O)NC23CC4CC(C2)CC(C4)C3)C56CC7CC(C5)CC(C7)C6 SS-0934 c1ccc(cc1)NC(=O)c2c(c3cc4c(nc3s2)C5CCN4CC5)N SS-0935 CC(C)c1ccc(cc1)C2C(=C(OC3=C2C(=O)CC(C3)(C)C)N)C#N SS-0936 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cccc(c3)OC)C(=O)C1)C SS-0937 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccccc3OC)C(=O)C1)C SS-0938 Cc1cc(c2c(c(sc2n1)C(=O)OC)N)C(F)(F)F SS-0939 c1cc(cnc1)c2ccc(c(n2)SCC(=O)O)C#N SS-0940 c1ccc(cc1)C(=O)CSc2c(cc3c(n2)CCCCCC3)C#N SS-0941 CC1=C(C(C(=C(N1)SCc2ccc(cc2)[N+](=O)[O-])C#N)c3ccccc3[N+](=O)[O-])C(=O)C SS-0942 c1cc(cnc1)c2ccc3c(c(sc3n2)C#N)N SS-0943 CCCN1c2ccccc2C3(C1=O)c4c([nH]nc4OC(=C3C#N)N)CC SS-0944 CCCCc1c2c(n[nH]1)OC(=C(C23c4ccccc4N(C3=O)CCC)C#N)N SS-0945 CCCN1c2ccccc2C3(C1=O)C(=C(OC(=C3C(=O)OC)C)N)C#N SS-0946 CCCN1c2ccccc2C3(C1=O)C(=C(OC(=C3C(=O)OCCOC(=O)C(=C)C)C)N)C#N SS-0947 c1ccnc(c1)CSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0948 c1cc(cnc1)CSc2c(c(cc(n2)C3CC3)C(F)(F)F)C#N SS-0949 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)NC(C)C)N)C(F)(F)F)C1 SS-0950 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)NC4CC4)N)C(F)(F)F)C1 SS-0951 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)NCC(=O)O)N)C(F)(F)F)C1 SS-0952 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccccc4F)N)C(F)(F)F)C1 SS-0953 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)F)N)C(F)(F)F)C1 SS-0954 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(c(c4)F)F)N)C(F)(F)F)C1 SS-0955 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)C(=O)OCC)N)C(F)(F)F)C1 SS-0956 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4cc(ccc4OC)Cl)N)C(F)(F)F)C1 SS-0957 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(cc4OC)OC)N)C(F)(F)F)C1 SS-0958 CCC1CCc2c(c(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)C(=O)C)N)C(F)(F)F)C1 SS-0959 Cc1ccc(o1)c2cc(c(c(n2)SCC(=O)NCC(=O)O)C#N)C(F)(F)F SS-0960 CC1=C(C(C(=C(O1)N)C#N)c2ccccc2)C(=O)OCCOC(=O)C(=C)C SS-0961 CC1=C(C(C(=C(O1)N)C#N)c2c(cccc2Cl)F)C(=O)OCCOC(=O)C(=C)C SS-0962 CC1=C(C(C(=C(O1)N)C#N)c2c(cccc2Cl)Cl)C(=O)OCCOC(=O)C(=C)C SS-0963 CC1=C(C(C(=C(O1)N)C#N)c2ccc(c(c2)Cl)Cl)C(=O)OCCOC(=O)C(=C)C SS-0964 CC1=C(C(C(=C(O1)N)C#N)c2ccc(cc2Cl)Cl)C(=O)OCCOC(=O)C(=C)C SS-0965 CC1=C(C(C(=C(O1)N)C#N)c2cccc(c2Cl)Cl)C(=O)OCCOC(=O)C(=C)C SS-0966 CC1=C(C(C(=C(O1)N)C#N)c2ccc(c(c2)Cl)[N+](=O)[O-])C(=O)OCCOC(=O)C(=C)C SS-0967 CC1=C(C(C(=C(O1)N)C#N)c2ccccc2[N+](=O)[O-])C(=O)OCCOC(=O)C(=C)C SS-0968 CC1=C(C(C(=C(O1)N)C#N)c2ccc3c(c2)OCO3)C(=O)OCCOC(=O)C(=C)C SS-0969 CC1=C(C(C(=C(O1)N)C#N)c2ccc(cc2)Br)C(=O)OCCOC(=O)C(=C)C SS-0970 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2ccccc2Cl)C(=O)OC SS-0971 COC(=O)CC1=C(C(C(=C(O1)N)C#N)c2ccncc2)C(=O)OC SS-0972 Cc1cccc2c1NC(=O)C23C(=C(OC(=C3C(=O)OCCOC(=O)C(=C)C)C)N)C#N SS-0973 CC1=C(C2(c3ccccc3NC2=O)C(=C(O1)N)C#N)C(=O)OCCOC(=O)C(=C)C SS-0974 CC1=C(C2(c3cc(ccc3NC2=O)[N+](=O)[O-])C(=C(O1)N)C#N)C(=O)OCCOC(=O)C(=C)C SS-0975 Cc1c2c(n[nH]1)OC(=C(C2c3ccc(c(c3)OC)OC4CCCC4)C#N)N SS-0976 CC(C)c1c2c(n[nH]1)OC(=C(C2c3ccc(c(c3)OC)OC4CCCC4)C#N)N SS-0977 COc1cc(ccc1OC2CCCC2)C3c4c([nH]nc4OC(=C3C#N)N)c5ccc(cc5)Cl SS-0978 Cc1ccc(c(c1)C)c2c3c(n[nH]2)OC(=C(C3c4ccc(c(c4)OC)OC5CCCC5)C#N)N SS-0979 CCCc1c2c(n[nH]1)OC(=C(C2c3c[nH]nc3c4ccc(cc4)F)C#N)N SS-0980 COC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccccc3[N+](=O)[O-])CO)N SS-0981 COC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(c(c3)Cl)[N+](=O)[O-])CO)N SS-0982 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccccc3[N+](=O)[O-])CO)N SS-0983 CCOC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(c(c3)Cl)[N+](=O)[O-])CO)N SS-0984 CC(C)OC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccccc3[N+](=O)[O-])CO)N SS-0985 CC(C)OC(=O)C1=C(Oc2c(=O)cc(oc2C1c3ccc(c(c3)Cl)[N+](=O)[O-])CO)N SS-0986 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccccc4Cl)N SS-0987 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(cc4)Cl)N SS-0988 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(cc4Cl)Cl)N SS-0989 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4c(cccc4Cl)Cl)N SS-0990 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4c(cccc4Cl)F)N SS-0991 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(cc4)F)N SS-0992 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4cccc(c4)[N+](=O)[O-])N SS-0993 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(cc4)[N+](=O)[O-])N SS-0994 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(c(c4)Cl)[N+](=O)[O-])N SS-0995 CCOC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4cccnc4)N SS-0996 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccccc4Cl)N SS-0998 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(cc4Cl)Cl)N SS-0999 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4c(cccc4Cl)Cl)N SS-1000 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4c(cccc4Cl)F)N SS-1001 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4cccnc4)N SS-1002 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4cccc(c4)[N+](=O)[O-])N SS-1003 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(cc4)[N+](=O)[O-])N SS-1004 COC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(c(c4)Cl)[N+](=O)[O-])N SS-1005 CC(C)OC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4cccc(c4)[N+](=O)[O-])N SS-1006 CC(C)OC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccccc4Cl)N SS-1008 CC(C)OC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4ccc(cc4Cl)Cl)N SS-1009 CC(C)OC(=O)C1=C(Oc2c3ccccc3sc(=O)c2C1c4c(cccc4Cl)F)N SS-1011 CCc1c(c(c2c(c(sc2n1)C(=O)NCC(=O)O)N)C(F)(F)F)C SS-1012 c1c(c2c(c(sc2nc1C3CC3)C(=O)N)N)C(F)(F)F SS-1013 COc1ccc(cc1OC)Cc2cc(c3c(c(sc3n2)C(=O)N)N)C(F)(F)F SS-1014 COc1ccc(cc1OC)Cc2cc(c3c(c(sc3n2)C(=O)NC4CC4)N)C(F)(F)F SS-1015 COc1ccc(cc1OC)Cc2cc(c3c(c(sc3n2)C(=O)NCc4ccccc4Cl)N)C(F)(F)F SS-1016 COc1ccc(cc1OC)Cc2cc(c3c(c(sc3n2)C(=O)NCc4ccc(cc4)F)N)C(F)(F)F SS-1017 COc1ccc(cc1OC)Cc2cc(c3c(c(sc3n2)C(=O)NCc4ccc5c(c4)OCO5)N)C(F)(F)F SS-1018 COc1ccc(cc1)CNC(=O)c2c(c3c(cc(nc3s2)Cc4ccc(c(c4)OC)OC)C(F)(F)F)N SS-1019 COc1ccc(cc1OC)Cc2cc(c3c(c(sc3n2)C(=O)Nc4ccc(cc4)F)N)C(F)(F)F SS-1020 CCc1c(cc2c3c(sc2n1)C(=O)NCC(=O)N3)C SS-1021 CCc1c(c(c2c3c(sc2n1)C(=O)NCC(=O)N3)C(F)(F)F)C SS-1022 Cc1cc(nc2c1c3c(s2)C(=O)N4CCC[C@H]4C(=O)N3)C SS-1023 CCc1c(cc2c3c(sc2n1)C(=O)N4CCC[C@H]4C(=O)N3)C SS-1024 c1c2c(nc3c1c4c(s3)C(=O)N5CCC[C@H]5C(=O)N4)CCCC2 SS-1025 Cc1ccc(cc1)C(C(=O)O)O SS-2000 CC(C)(C)OC(=O)N1CCC2(CC1)C(=O)NC(=O)N2 SS-2050 CCC(c1ccc(cc1)Br)C(=O)O SS-2067 CCOc1cccnc1N SS-2093 CCC(C)(c1cccs1)C(=O)O SS-2109 COc1ccc(cc1)OCCO SS-2122 CC(CSC(=O)C)C(=O)N SS-2160 Cc1ccc(cn1)CO SS-2181 Cc1cccc[n+]1C.[I-] SS-2183 c1cc(ccc1SCCO)Cl SS-2220 c1cc([nH]c1)C2=NCCC2 SS-2224 CC(C)(CO)C(c1ccco1)O SS-2262 c1cc(c(cc1Cl)Cl)C2(CC2)C(=O)O SS-2283 Cc1nc2cc3c(cc2s1)nc(s3)C SS-2286 COC(=O)C1C(O1)c2ccc(cc2)[N+](=O)[O-] SS-2293 COC(=O)C1C(O1)c2ccc(cc2)C#N SS-2332 COc1cc(cc(c1OC)Br)/C=C/C(=O)O SS-2341 CC(C)(c1ccc(cc1)Cl)C(=O)OC SS-2349 CC(C)(CS(=O)c1ccc(cc1)O)C(=O)O SS-2360 CCCCCCCCN1CNC(=S)NC1 SS-2382 c1ccc(cc1)Sc2ccc(cc2)N SS-2399 COc1ccc(cc1)/C=C/C(=O)C(=O)OC SS-2403 c1ccc(cc1)C(C2CCC2)(C(=O)O)O SS-2407 CC(=O)N/C(=C/c1ccc(cc1)OC)/C(=O)O SS-2408 CCC(c1ccc(c(c1)OC)OC)C(=O)O SS-2423 CC1CN(CCN1)c2ccccc2OC SS-2433 c1ccc(cc1)S(=O)(=O)n2ccc(c2)C(=O)CCCl SS-2455 CC(C)NCC(c1cc(cc(c1)OC)OC)O SS-2483 CCCCn1c2ccc(cc2c3c1ccc(c3)Br)Br SS-2581 CCC(c1ccc(cc1)C2CCCCC2)C(=O)O SS-2597 C=CCC(c1ccccc1)(c2ccccc2)C(=O)O SS-2630 CC(C)C(=O)C(C)(C)C(c1ccccc1)NC(=O)OC SS-2640 c1ccc(cc1)C(=O)N(c2ccccc2)c3ccc(cc3)N SS-2690 COc1ccc(cc1)/C=C(\C#N)/C(=O)OC SS-2939 CC(CSC(=O)c1ccccc1)C(=O)O SS-2940 COc1cccc(c1)C(CC(=O)O)CC(=O)O SS-2946 CSC(=S)N1CCOCC1 SS-2948 CCCC1(c2cc(ccc2-c3c1cc(cc3)Br)Br)CCC SS-2954 Cc1cccc(c1I)[N+](=O)[O-] SS-2957 c1cc2c(c(c1)C(=O)O)[nH]c(=O)oc2=O SS-2958 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)c3ccccc3N SS-2959 COC(=O)CN1C(=O)c2ccccc2C1=O SS-2960 c1ccc(c(c1)C(=O)O)NCc2ccc(cc2)Cl SS-2961 C#CC[C@@H](c1ccccc1)N.Cl SS-2962 COCC(C(=O)O)N SS-2963 CC1=C(c2cc(ccc2C1)F)CC(=O)O SS-2964 COc1c(cc2ccccc2c1Br)C#N SS-2965 Cc1cc(n[nH]1)[N+](=O)[O-] SS-2966 c1ccc(cc1)NC(=O)C(=O)O SS-2967 C1COC(O1)CCCC=O SS-2968 COc1cnc(nc1O)O SS-2971 CC(C)(C)OC(=O)N1CCC(CC1)c2nc(cs2)C(=O)O SS-2972 C1CC2C=CC1C(C2C(=O)O)C(=O)O SS-2973 COc1cc2cc(sc2cc1OC)/C(=N\O)/N.Cl SS-2975 COc1cc2cc(sc2cc1OC)C(=O)O SS-2976 CC(CCSCc1ccccc1)(C(=O)O)N SS-2978 Cc1cc(cc(c1C#N)C)Br SS-2979 c1c(nc2n1CCS2)C=O SS-2982 COc1cccc(c1OC)C(c2ccncc2)O SS-2983 Cc1ccc(c2c1sc(n2)N)OC SS-2985 C=C(CC(=O)OCc1ccccc1)C(=O)O SS-2986 c1ccc2c(c1)/C(=C\N)/C(=O)OC2=O SS-2987 c1ccc2c(c1)c(cnc2N)Br SS-2988 CC1(COP(=O)(O[C@H]1c2ccccc2OC)O)C SS-2992 CC1(COP(=O)(O[C@@H]1c2ccccc2OC)O)C SS-2993 CC1(COP(=O)(O[C@@H]1c2ccccc2)O)C.O SS-2994 CC1(COP(=O)(O[C@H]1c2ccccc2Cl)O)C SS-2995 CC1(COP(=O)(O[C@H]1c2ccccc2)O)C.O SS-2996 CC1(COP(=O)(O[C@@H]1c2ccccc2Cl)O)C SS-2997 c1ccc(cc1)c2ccc(cc2)CCO SS-2998 c1cc(ccc1N)SCC#N SS-2999 c1cc(c(cc1S(=O)(=O)O)N)F SS-3000 c1ccc2c(c1)CC(C2)(CC(=O)O)O SS-3001 c1cc2c(cc1Cl)c3ccncc3[nH]2 SS-3002 C[C@@H]1C[C@@H](c2ccccc2N1)C(=O)OC SS-3003 CCC(C(=O)O)NC(=O)OC(C)(C)C SS-3006 c1ccc(cc1)C[C@@H]([C@@H](C(=O)O)O)N SS-3011 COC(=O)c1c(cccn1)Br SS-3013 Cc1nc(cc(n1)O)c2ccc(cc2Cl)Cl SS-3014 CC(C)(c1ccc(cc1)[N+](=O)[O-])C(=O)O SS-3015 CC(C)(c1ccc(c(c1)I)N)C(=O)OC SS-3016 c1ccc2c(c1)CNC(=S)N2 SS-3017 CSC1=NCc2ccccc2N1.Cl SS-3018 CCOC(=O)c1ccc(cc1Cl)N SS-3019 c1cc2c(ccc(c2Cl)CO)nc1 SS-3020 c1cc2cc(c(cc2nc1)Cl)C=O SS-3021 Cc1c(cncc1OC)N.Cl SS-3022 c1cc(c(cc1O)CCCC(=O)O)O SS-3024 c1ccc(cc1)C(=O)CC(=O)CCC(=O)O SS-3025 c1cc(c(cc1S(=O)(=O)N)N)C(=O)O SS-3028 Cn1cnc2c1c(ncn2)Cl SS-3029 c1cc(nc(c1)Br)CBr SS-3030 Cc1nc(cc(n1)Cl)N SS-3031 CC1CCN(CC1)c2cc(ccc2N)N3CCN(CC3)C SS-3034 c1c[nH]c2c1ncnc2Cl SS-3037 c1c(cc(c(c1[N+](=O)[O-])O)O)/C=C(\C#N)/C(=O)O SS-3041 c1c(c(c(c(c1F)C(=O)O)Cl)F)O SS-3042 c1c(c(cc(c1[N+](=O)[O-])Cl)Cl)N SS-3043 c1cc(c(cc1Br)CBr)I SS-3044 CC(=O)c1ccnc(n1)SC SS-3045 COc1ccc(cc1)C(=O)CCCC(=O)OC SS-3047 Cc1ccc(cc1OC(F)F)[N+](=O)[O-] SS-3048 Cc1cc(=O)c2cc(ccc2[nH]1)C#N SS-3049 Cc1cc(c2cc(ccc2n1)C#N)Cl SS-3050 CNC1(CCN(CC1)Cc2ccccc2)C#N SS-3051 c1cc(c(cc1S(=O)(=O)O)O)N SS-3052 CN(C)C(=O)C1(CCNCC1)N2CCCCC2.Cl SS-3053 CS(=O)(=O)Nc1ccccc1I SS-3055 CC(C(=O)O)OC1CCN(CC1)C(=O)OC(C)(C)C SS-3056 C[C@H](C(=O)O)OC1CCN(CC1)C(=O)OC(C)(C)C SS-3057 c1c(cc(c2c1C(=O)CCO2)Br)Cl SS-3058 COC(=O)/C(=C/C(=O)O)/Br SS-3060 c1cncc2c1sc(n2)N SS-3062 c1cc(ccc1COCC(=O)O)Br SS-3063 Cc1c(nc[nH]1)CC#N SS-3067 CCOC(=O)c1ccc(cc1)c2ccc(cc2)O SS-3068 c1cc(c(c(c1)F)F)[N+](=O)[O-] SS-3069 CCOC(=O)CC1C(=O)NCCN1Cc2ccccc2 SS-3070 c1ccc2c(c1)C(CC2=O)C(=O)O SS-3073 Cn1cnc2c1ncnc2Cl SS-3075 CC(C)(C)OC(=O)NC(CO)(CO)CO SS-3076 CSc1nccc(n1)CC(=O)c2ccc(cc2)F SS-3077 CC(C)(C)[C@@H](C(=O)O)NC(=O)OCc1ccccc1 SS-3079 COC(=O)C1CC1c2ccc(cc2)F SS-3080 COc1cc(c(cc1OC)Br)CCN SS-3082 C[C@H]1CN[C@@H](CN1Cc2ccc(cc2)F)C SS-3083 COCOc1c(ccc(c1[Si](C)(C)C)F)F SS-3085 CCCCc1nc(c(n1Cc2ccc(cc2)Br)CO)Cl SS-3086 CC(=O)Nc1ccccc1Br SS-3087 c1cc(nc(c1)Br)CN2CCCCC2 SS-3088 C[C@]12CC[C@@H]3c4ccc(cc4CC[C@H]3[C@@H]1C=C[C@@H]2O)OCc5ccccc5 SS-3089 Cc1cc(c2cc(ccc2n1)C(=O)NCc3ccccc3)O SS-3090 CC(C)(C)OC(=O)N1CCN(CC1)C2(CCOCC2)C#N SS-3093 CC(C)(C)OC(=O)N1CCC1C(=O)N(C)OC SS-3095 Cc1ccc2c(c1)c3c([nH]2)CCN(C3)C SS-3096 CN(C)CCO/N=C(/C=C/c1ccc(cc1)O)\c2ccccc2F SS-3097 c1c[nH]c2c1c(ncn2)N.OS(=O)(=O)O SS-3099 c1ccc2c(c1)CN(C(=O)N2)C3CCNCC3 SS-3104 CC(C)(C)OC(=O)N(CCO)Cc1ccccc1 SS-3110 c1[nH]c2c(n1)CC(CC2)C(=O)O SS-3113 c1cc(c(c(c1)Br)C=O)Br SS-3114 c1ccc(c(c1)C(=O)O)n2cncn2.Cl SS-3116 c1cc(ccc1c2cc3c(o2)CCNC3)Br.Cl SS-3118 c1cc(c(cc1Cl)O)[N+](=O)[O-] SS-3119 CC(=O)c1cc(ccc1F)Br SS-3120 C1C[C@@H]2C[C@@H](N[C@@H]2C1)C(=O)O SS-3122 c1ccc(c(c1)C(=O)O)NC(=O)CCl SS-3146 c1cc(ccc1CC(CO)(CO)[N+](=O)[O-])F SS-3152 COc1ccccc1CC(C(=O)O)N SS-3154 c1ccc2c(c1)C(c3ccccc3NC2=O)Cl SS-3167 COC(=O)c1cc(c2cccc(c2c1)OCc3ccccc3)CCO SS-3176 COC(=O)C[C@H]1CCc2c1n(c3c2cc(cc3S(=O)(=O)C)F)Cc4ccc(cc4)Cl SS-3179 CC(C)(C)OC(=O)N1CC2CC1C2C(=O)O SS-3182 c1ccc(cc1)CN2CC3(CC(=O)NC3)CC2=O SS-3183 CCOC(=O)c1cc(n(n1)C)C SS-3184 c1cc(cc(c1)N)C(=O)Nc2cccnc2 SS-3186 c1ccc(cc1)[C@@H]2COC(=O)N2 SS-3215 c1cc(ccc1N2CCC(CC2)Oc3ccc(cc3)OC(F)(F)F)O SS-3227 C1=CSC2C1C2C(=O)O SS-3231 CSc1nccc(n1)c2c[nH]nc2 SS-3250 c1csc(c1Br)c2c(ccs2)Br SS-3253 c1cc(sc1)CC(=O)N SS-3258 c1cc(sc1)C(=O)N SS-3260 COc1ccc2c(c1)cccc2OC SS-3261 c1ccc(c(c1)C(=O)c2cc(ccc2NC(=O)CCl)Cl)Cl SS-3265 COC(=O)c1ccc2c(c1)C(CC(=O)O2)c3ccccc3 SS-3270 COC(=O)c1ccc2c(c1)[C@H](CC(=O)O2)c3ccccc3 SS-3272 CCOP(=O)(Cc1ccc(cc1)C(=O)Nc2ccc(cc2C#N)Br)OCC SS-3273 c1ccc(cc1)CN2CCCC(=O)CC2 SS-3274 CCOc1ccnc2c1cc[nH]2 SS-3279 COc1ccnc2c1cc[nH]2 SS-3281 CC(C)(C)OC(=O)N1CCCC1 SS-3295 CC(C)CC(=O)N1C(COC1=O)Cc2ccccc2 SS-3300 CCSC1C(C(C2C(O1)COC(O2)c3ccccc3)O)NC(=O)C SS-3302 CC(C)CC(=O)N(C)C(C)C(c1ccccc1)O SS-3305 CC(C)C1CC(OC1=O)CO SS-3308 CC1C(OC2(N1C)C(CC(O2)CBr)C(C)C)c3ccccc3 SS-3309 COC1C[C@@H]([C@@H](CO1)O)O SS-3337 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCCCBr SS-3339 c1ccc(c(c1)c2c3cc(ccc3[nH]c(=O)n2)Cl)Cl SS-3341 CC(C)(C)[Si](C)(C)OCC(C(=O)OC)OC1CCCCO1 SS-3348 CC(C)(C)OC(=O)NCC#C SS-3353 c1ccc(cc1)C(C(C(=O)O)N)O SS-3359 Cn1c(=O)c(c([nH]c1=O)N)N SS-3364 CSc1[nH]c(=O)ccn1 SS-3370 c1ccc(cc1)COc2ccc3c(c2)c(cc(=O)o3)O SS-3371 C[C@]12CC[C@@H]3c4ccc(cc4CC[C@H]3[C@@H]1C=CC2=O)OCc5ccccc5 SS-3378 CC1(C=Cc2cc(ccc2O1)CC(=O)O)C SS-3383 CC(C)(C)OC(=O)NCC1CC1 SS-3387 c1cc(ccc1/C=N/c2ccc(cc2)F)O SS-3393 C[C@@H](CO)CO[Si](c1ccccc1)(c2ccccc2)C(C)(C)C SS-3394 c1ccc(cc1)COC(=O)N2CCCC(C2)CO SS-3395 C1CC1C(=O)C(=O)[O-].[K+] SS-3396 CC(=O)O.c1cc2c([nH]cn2)[n+](c1)[O-] SS-3397 CN(Cc1cnc2c(n1)c(nc(n2)N)N)c3ccc(cc3)C(=O)O SS-3399 C[C@@H](C(=O)O)NC(=O)Cc1cc(cc(c1)F)F SS-3400 CC(C)(C)OC(=O)N1CCCC1=O SS-3403 COc1ccc(cc1)C(CN)C2(CCCCC2)O SS-3413 C[C@@H]1CC2C3C[C@@H](C4=CC(=O)C=C[C@@]4([C@]3([C@H](C[C@@]2([C@]1(C(=O)S)O)C)O)F)C)F SS-3414 CN1CC[C@@]23CCCC[C@@H]2[C@@H]1C(=O)c4c3cc(cc4)OC SS-3417 COC(=O)Cc1cc(=O)n2c(c1C(=O)OC)CCC2 SS-3424 Cc1ccc(cc1)S(=O)(=O)OC2CCN(CC2)C(=O)OCc3ccccc3 SS-3431 c1ccc2c(c1)c(cc(n2)N3CCNCC3)c4cccc(c4)F.C(=C/C(=O)O)\C(=O)O SS-3433 c1ccc2c(c1)c(cc(n2)Cl)c3ccc(cc3)F SS-3434 c1ccc2c(c1)ccn2C(=O)O SS-3438 COc1cccc2c1nc(s2)NC(=O)c3ccccc3 SS-3439 c1cc(c2c(c1)sc(n2)N)O SS-3440 c1ccc(cc1)CNc2ccccc2Br SS-3448 CC(C)(C)OC(=O)N1CCCC(C1)C(=O)O SS-3449 COc1c(cccc1Br)[N+](=O)[O-] SS-3458 CC(c1nc2ccccc2c(=O)n1c3ccc(cc3)C#N)Br SS-3463 COc1c(cccc1)C(=O)NC[C@]2(CC[C@@H](CC2)O)c3ccccc3 SS-3468 COC(=O)c1ccccc1SSc2ccccc2C(=O)OC SS-3470 CNC(=O)C(c1ccccc1)N SS-3472 CNCC(c1ccccc1)N.Cl.Cl SS-3473 Cc1c(n(c2c1cccc2)S(=O)(=O)c3ccccc3)C SS-3474 CN1CCc2c(c3cc(ccc3[nH]2)Cl)C1 SS-3475 CC(C)(C)OC(=O)N1Cc2ccc(cc2C1)CO SS-3479 c1cc(ccc1c2cc3c(o2)CCNC3)[N+](=O)[O-] SS-3482 CNCc1ccccc1.Cl SS-3494 C[C@@H](c1ccccc1)N2CCNCC2 SS-3510 c1ccc(c(c1)C(=O)CCCl)F SS-3519 COc1cccc2c1CC[C@@H](C2)NCc3ccccc3 SS-3530 CCCN[C@H]1CCc2c(cccc2O)C1.Br SS-3533 CCOC(c1ccc(cc1Br)F)OCC SS-3534 Cc1c2cc(ccc2[nH]c1c3ccc(cc3)OCc4ccccc4)OCc5ccccc5 SS-3549 CCn1c2ccccc2c3c1ccc(c3)C#N SS-3554 c1cc(cc2c1cc(c(c2)C(=O)O)O)Br SS-3555 C(C(CCl)(CCl)C(=O)O)Cl SS-3556 CCOC(=O)Cc1[nH]c(nn1)C SS-3566 CCCCc1ncc(n1Cc2ccc(cc2)C(=O)O)C=O SS-3568 CN1CCN(CC1)c2ccc(cc2Cl)N SS-3590 c1cc(ccc1C2(CCC(=O)CC2)C#N)F SS-3591 c1ccc(cc1)C2(CCC(=O)CC2)CO SS-3592 COC(=O)C1(CCC(=O)CC1)c2ccc(cc2)F SS-3593 c1cc2c(cc1Br)cn[nH]2 SS-3596 Cc1c(c(=O)n(n1C)c2ccccc2)C(=O)O SS-3597 c1ccc(c(c1)C2(CCC(=O)CC2)C#N)F SS-3605 c1ccc(cc1)COc2cc(ncc2OCc3ccccc3)C(=O)OCc4ccccc4 SS-3617 CCc1ccc(cc1F)Br SS-3619 CC1(C=Cc2cc(ccc2O1)C(=O)O)C SS-3624 CCOC(=O)C(Cc1ccccc1C(=O)OC)C#N SS-3625 Cc1ccc(cc1)C(c2ccc(cc2)C)N SS-3626 CCOC(=O)CCCc1nc2cc(ccc2n1C)N SS-3629 c1cc(ccc1CCCC(=O)O)Cl SS-3645 COc1ccc2c(c1)C(CC2=O)CC(=O)O SS-3646 COc1cc(ccc1OCCN2CCCC2)N SS-3647 c1ccc2c(c1)C(=O)N(C2=O)Cc3ccc(cc3)C(=O)O SS-3677 c1ccc(cc1)C(c2ccccc2)N3CC(C3)CN SS-3680 CC(C)(C)OC(=O)NC1CCc2ccccc2NC1=O SS-3682 CC(C)(C)OC(=O)N[C@@H](c1ccc(cc1)OS(=O)(=O)C(F)(F)F)C(=O)OC SS-3695 c1cc2c(c(c1)C=O)OCC2 SS-3697 CCOC(=O)c1cnn(c1C(F)(F)F)c2cccc(c2)Cl SS-3704 c1cc(cc(c1)Cl)n2c(c(cn2)CC(=O)O)C(F)(F)F SS-3705 c1cc(cc(c1)Cl)n2c(c(cn2)CC#N)C(F)(F)F SS-3706 c1cc(c(cc1Cl)Cl)NN.Cl SS-3729 c1ccc(cc1)Cn2ccc3c2ccc(c3)Br SS-3732 c1ccc(c(c1)CN)F SS-3747 c1ccc(cc1)N2CCN(CC2)C(=S)N SS-3792 CNC1(CCN(CC1)Cc2ccccc2)c3ccccc3 SS-3795 CC(C)Sc1c(cccn1)CO SS-3811 COC(c1ccc2cccnc2n1)OC SS-3813 CCNCc1nnc(o1)C SS-3821 c1ccc(cc1)S(=O)(=O)CCCN.Cl SS-3822 CC(C)(C)OC(=O)Nc1ccccc1CC(=O)O SS-3824 Cn1ccc(n1)CCN.Cl.Cl SS-3827 c1c(scn1)CN.Cl.Cl SS-3828 CN1CCCN=C1CN.Cl.Cl SS-3831 CCOC(=O)N1CCCC1C(=O)O SS-3834 C(c1[nH]nc(n1)N)C(=O)O SS-3835 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC4CCC(c5c4cccc5)C(=O)O SS-3840 c1cc(c(cc1C(=N)N)F)F.Cl SS-3844 COc1cc(ccc1O)C(=N)N.Cl SS-3845 c1cc(ccc1CCC(=N)N)O.Cl SS-3846 c1cc(cc(c1)O)C(=N)N.Cl SS-3847 c1ccc2c(c1)-c3ccccc3C2COC(=O)Nc4ccc(cc4)SCC(=O)O SS-3849 COc1cc(c(cc1OC)NC(=O)OCC2c3ccccc3-c4c2cccc4)C(=O)O SS-3850 CC(C)(C)OC(=O)Nc1nc(cs1)CC(=O)O SS-3851 c1ccc2c(c1)ccn2C3CCNCC3.Cl SS-3855 c1ccc2c(c1)cccc2C3CCNCC3.Cl SS-3856 c1ccc2c(c1)C=CC23CCNCC3.Cl SS-3857 c1ccc2cc(ccc2c1)C3CCNCC3.Cl SS-3858 c1ccc2c(c1)COC23CCNCC3.Cl SS-3860 c1ccc2c(c1)C(=O)OC23CCNCC3.Cl SS-3861 c1ccc2c(c1)CSC23CCNCC3.Cl SS-3862 CN(C)C(=O)Oc1ccc(cc1)CC(=O)O SS-3863 CCS(=O)(=O)Nc1ccccc1C(=O)O SS-3864 CC(=O)O.CN(C)c1ccc(cc1)C2CCCN2 SS-3871 c1ccc2c(c1)ccc(=O)n2C3CCNCC3.Cl SS-3872 c1ccc2c(c1)CCC23CCNCC3.Cl SS-3873 c1ccc2c(c1)COC(=O)N2C3CCNCC3.Cl SS-3874 c1ccc2c(c1)CCC(=O)N2C3CCNCC3.Cl SS-3875 CC(=O)Nc1ccc(cc1)OCCCC(=O)O SS-3876 CCNC(=O)Nc1cccc(c1)C(=O)O SS-3880 CCOC(=O)Nc1ccc(cc1)CC(=O)O SS-3881 CS(=O)(=O)N1CCCC(C1)O SS-3883 CCOC(=O)Nc1cccc(c1)CC(=O)O SS-3885 CN(C)C(=O)Nc1ccc(cc1)CC(=O)O SS-3888 c1cc(ccc1CC(=O)O)NC(=O)CCl SS-3889 CCNC(=O)Nc1cccc(c1)CCC(=O)O SS-3890 CS(=O)(=O)N1CC2(CCNCC2)c3c1cccc3.Cl SS-3893 CN(C)C(=O)COc1ccccc1C(=O)O SS-3894 CS(=O)(=O)NC(Cc1ccccc1)C(=O)O SS-3895 CC(=O)Nc1ccc(cc1)OCC(=O)O SS-3896 c1cc(ccc1n2c(nc(n2)C(=O)O)CCl)F SS-3899 c1ccc(cc1)n2c(nc(n2)C(=O)O)CCl SS-3900 Cc1ccn2c(c1)ncc2CCN SS-3901 CN(C)C(=O)Oc1ccc(cc1)C(=O)O SS-3903 CN(C)C(=O)Oc1cccc(c1)C(=O)O SS-3904 CCOC(=O)N1CCN(CC1)c2ccccc2O SS-3906 CS(=O)(=O)N1CCN(CC1)c2ccccc2O SS-3907 CCNC(=O)N1CCN(CC1)c2ccc(cc2)O SS-3908 CCOC(=O)N1CCN(CC1)c2cccc(c2)O SS-3909 CCNC(=O)N1CCN(CC1)c2ccccc2O SS-3910 CCNC(=O)N1CCN(CC1)c2cccc(c2)O SS-3911 CS(=O)(=O)N1CCN(CC1)c2ccc(cc2)O SS-3912 CS(=O)(=O)N1CCN(CC1)c2cccc(c2)O SS-3913 CC(=O)Nc1ccc(cc1)S(=O)(=O)CC#N SS-3915 CC(C)(C)c1ccc(cc1)CC(C(=O)O)NC(=O)OC(C)(C)C SS-3916 CC(C)(C)OC(=O)NC(Cc1ccco1)C(=O)O.C1CCC(CC1)NC2CCCCC2 SS-3919 CC(C)(C)OC(=O)NC(C(c1ccccc1)c2ccccc2)C(=O)O SS-3920 c1ccc2c(c1)c3c([nH]2)CN(C(C3)C(=O)O)C(=O)OCC4c5ccccc5-c6c4cccc6 SS-3921 c1ccc(cc1)/C=C/CC(C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SS-3922 c1ccc(cc1)C(c2ccccc2)C(C(=O)O)NC(=O)OCC3c4ccccc4-c5c3cccc5 SS-3923 C=CCC(C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 SS-3924 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(Cc4ccncc4)C(=O)O SS-3925 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(Cc4ccsc4)C(=O)O SS-3926 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(Cc4ccccn4)C(=O)O SS-3927 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(Cc4ccco4)C(=O)O SS-3928 CC(C)(C)c1ccc(cc1)CC(C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SS-3929 c1ccc2c(c1)c(cs2)CC(C(=O)O)NC(=O)OCC3c4ccccc4-c5c3cccc5 SS-3931 c1ccc2c(c1)C(CCC2=O)C(=O)O SS-3938 CC(C)(CNS(=O)(=O)C)CO SS-3940 CN(C)C(=O)CCCC(=O)O SS-3941 CS(=O)(=O)CCCN.Cl SS-3945 c1cc(cc(c1)NC(=O)CCl)CC(=O)O SS-3946 c1cc(cc(c1)NC(=O)CCl)CCC(=O)O SS-3947 c1cc(ccc1CCC(=O)O)NC(=O)CCl SS-3948 CS(=O)(=O)N1CCCCC1C(=O)O SS-3952 CCS(=O)(=O)NCCCC(=O)O SS-3953 CS(=O)(=O)N1CCCC(C1)C(=O)O SS-3954 CCOC(=O)NC(C)C(=O)O SS-3955 CCOC(=O)NCCCC(=O)O SS-3956 CCOC(=O)N1CCCCC1C(=O)O SS-3957 CCOC(=O)N1CCCC(C1)C(=O)O SS-3958 CCS(=O)(=O)NCCC(=O)O SS-3961 CCS(=O)(=O)N1CCCC1C(=O)O SS-3962 CCN(CC)C(=O)OCC(=O)O SS-3963 CS(=O)(=O)Oc1cccc(c1)CC(=O)O SS-3964 CC(=O)Nc1ccc(cc1)OCCO SS-3965 c1ccc2c(c1)ncn2CCO SS-3966 c1ccc2c(c1)ncn2CCCN SS-3967 c1cn(nn1)CC(=O)O.Cl SS-3969 CC(=O)Nc1ccccc1OCCCC(=O)O SS-3970 CC(=O)NCCc1ccc(cc1)OCC(=O)O SS-3971 CC(=O)Nc1cccc(c1)OCC(=O)O SS-3972 CN(C)CCNC(=O)c1ccc(cc1)N SS-3976 c1ccc(cc1)CN2CCN(CC2)C(=O)C3CCNCC3 SS-3977 C1CNCCC1C(=O)NCCCN2CCOCC2 SS-3979 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)CCl SS-3980 CCN(CC)C(=O)Oc1cc(nc2c1cccc2)C(=O)O SS-3986 CN(C)C(=O)CCc1cccc(c1)C(=O)O SS-3990 Cn1ccnc1SCC(=O)O SS-3993 CN(C)S(=O)(=O)CCCN.Cl SS-3996 CN(C)C(=O)CCCCN.C(=O)(C(=O)O)O SS-3997 CCNC(=O)N1CCCCC1CO SS-3999 CCNC(=O)N1CCCC(C1)CO SS-4001 CCNC(=O)N1CCC(CC1)O SS-4002 CCNC(=O)N[C@H]1CC[C@@H](CC1)O SS-4003 c1cc(ccc1CCC(=O)N)C(=O)O SS-4006 c1cnccc1COCC(=O)O.O.Cl SS-4007 CN(C)C(=O)CCc1ccc(cc1)C(=O)O SS-4009 CCOC(=O)N[C@H]1CC[C@@H](CC1)O SS-4014 CCOC(=O)NCCCCCO SS-4015 CCNC(=O)N1CCCCC1CCO SS-4016 CCNC(=O)NCCCCCO SS-4017 COc1cccc(c1)OCCN SS-4020 CCOC(=O)Cn1cnc(c1C#N)C#N SS-4021 c1ccc(cc1)c2ccn(n2)CCN SS-4022 CC(C)(C)OC(=O)N1CCc2c(cccc2N)C1 SS-4025 c1c([nH]nc1C(=O)O)C2CC2 SS-4027 C(=C/C(C(F)(F)F)(OC(F)(F)F)F)\C(=O)O SS-4028 c1cc(c2c(c1)nccn2)C(=O)O SS-4030 c1cc-2c(cc1)C(c3c2cccc3)COC(=O)N[C@H]4CC[C@H](CC4)CC(=O)O SS-4035 CCOC(=O)N1CCCC(C1)O SS-4036 CS(=O)(=O)Nc1ccc(cc1)CC(=O)O SS-4037 CCOC(=O)NCCc1ccc(cc1)O SS-4038 CC(C)(C)OC(=O)NC(Cc1ccncc1)C(=O)O SS-4040 CN(C)C(=O)Nc1ccc(cc1)C(=O)O SS-4041 CS(=O)(=O)N1CCN(CC1)CCO SS-4042 CCNC(=O)NCCc1ccc(cc1)O SS-4043 CS(=O)(=O)Oc1ccc(cc1)CC(=O)O SS-4044 c1ccc2c(c1)nnn2CCC(=O)O SS-4045 c1ccc2c(c1)ncn2CC(=O)O SS-4046 CS(=O)(=O)NCCc1ccc(cc1)O SS-4048 CN(C)C(=O)c1ccc(cc1)N SS-4049 CC(CC(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 SS-4050 CC(C)(C)OC(=O)Nc1cc(c(cc1C(=O)O)OC)OC SS-4051 CS(=O)(=O)Oc1cccc(c1)CCC(=O)O SS-4053 c1ccc(cc1)C(CC(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SS-4057 c1ccc2c(c1)-c3ccccc3C2COC(=O)N[C@@H]4CCC[C@H](C4)C(=O)O SS-4059 c1cc(cc(c1)C(F)(F)F)C(=N)N.Cl SS-4066 c1c(cc(cc1F)F)C(=N)N.Cl SS-4067 CN(C)CCNC(=O)C1CCNCC1 SS-4068 CCNC(=O)N1CCN(CC1)CCO SS-4069 CC(C)(C)OC(=O)C1CCNCC1.Cl SS-4070 CC(C)(C)OC(=O)C1CCCNC1.Cl SS-4071 CSc1ccccc1N2CCNCC2 SS-4074 c1cc-2c(cc1)C(c3c2cccc3)COC(=O)N[C@H]4CC[C@@H](CC4)C(=O)O SS-4077 Cc1ccc(n1C)C(=N)N.Cl SS-4078 c1cc(ccc1C(=O)C=O)N2CCOCC2.O SS-4080 c1cnccc1CCCN SS-4081 COc1ccc(cc1)S(=O)(=O)N2CCNCC2 SS-4090 Cn1ccnc1SCCN SS-4092 CS(=O)(=O)N1CCc2c1ccc(c2)N SS-4093 CC(C)(C)OC(=O)NCCc1ccc(cc1)C(=O)O SS-4094 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCC(CC4)CN.Cl SS-4097 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCC(CC4)N.Cl SS-4098 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCCC(C4)CN.Cl SS-4099 c1ccc2c(c1)ncn2C3CCNCC3.Cl SS-4101 CC(c1cccc(c1)NC(=O)OC(C)(C)C)N SS-4102 C(C(=O)O)n1c(nnn1)N SS-4104 COc1ccc(cc1OC)CCNC(=O)C/C(=N/O)/N SS-4106 CC(C)(C)OC(=O)[C@H](CCC(=O)ON1C(=O)CCC1=O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SS-4109 c1ccc2c(c1)-c3ccccc3C2COC(=O)N[C@@H](Cc4cn(cn4)c5ccc(cc5[N+](=O)[O-])[N+](=O)[O-])C(=O)O SS-4110 CCSSC[C@@H](C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 SS-4112 CC(C)(C)OC(=O)N[C@@H](CC(=O)OCC1c2ccccc2-c3c1cccc3)C(=O)O SS-4125 c1ccc(cc1)C(=O)c2ccc(cc2)C[C@@H](C(=O)O)NC(=O)OCC3c4ccccc4-c5c3cccc5 SS-4126 CC(C)(C)OC(=O)NC(Cc1ccccn1)C(=O)O SS-4128 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC4(CC4)C(=O)O SS-4133 CC(C)(C)Oc1ccc(cc1)C(=O)O SS-4137 CC(C)(C)OC(=O)N[C@@H]1CCC[C@H](C1)CC(=O)O SS-4157 Cn1nc(nn1)S SS-4159 CCOc1ccc(cc1)CC[C@@H](C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SS-4165 c1c(cc(c(c1O)O)Br)C=O SS-4168 CC(C)[C@@H](CO)N.Cl SS-4171 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCC(=O)NCC(=O)NCC(=O)O SS-4172 CC(C)(C)OC(=O)N1CCC(CC1NC(=O)OCC2c3ccccc3-c4c2cccc4)C(=O)O SS-4180 CC(C)(C)OC(=O)NC1CC(CCN1C(=O)OC(C)(C)C)C(=O)O SS-4182 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCOC(C4)C(=O)O SS-4189 CC(C)(C)OC(=O)NCc1ccc(cc1)C[C@@H](C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SS-4190 c1cc(ccc1C(CC(=O)O)C(=O)O)N SS-4202 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(Cc4ccc(cc4)F)C(=O)O SS-4208 CC(C)(C)OC(=O)NCc1ccc(cc1)C[C@H](C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SS-4209 CC(OC(=O)N[C@H]1CC[C@H](CC1)CC(=O)O)(C)C SS-4217 c1ncn(n1)CCO SS-4218 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC4(CCS(=O)(=O)CC4)C(=O)O SS-4228 CC(C)(C)OC(=O)NC1(CCC(CC1)O)C(=O)O SS-4229 CS(=O)(=O)Nc1ccc(cc1)C(=O)O SS-4236 C(CNC(=O)CCl)C(=O)O SS-4240 CNCCCCCCO SS-4245 CC(OC(=O)N[C@H]1CC[C@@H](CC1)C(=O)O)(C)C SS-4248 CNC(=O)CCC(=O)O SS-4259 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCC4CCCNC4 SS-4275 CC(c1cccc(c1)N)NC(=O)OC(C)(C)C SS-4308 COc1ccc(cc1)C2CNCCN2 SS-4311 CN(C)C(=O)COc1cccc(c1)C(=O)O SS-4316 CCNC(=O)N1CCC(CC1)C(=O)O SS-4318 c1cc2c(cc1Cl)CCCN2 SS-4320 CC(C)(C)OC(=O)N1CCC(CC1)CNC.CC(C)(C)OC(=O)N1CCC(CC1)CNC.C(=C/C(=O)O)\C(=O)O SS-4321 COCC1CCNCC1.Cl SS-4322 c1cc(c2c(c1O)CCC2)F SS-4323 CC(C)(C)OC(=O)N1CCC(=O)C(C1)F SS-4324 Cc1c(c(n(n1)C)C)CN.Cl SS-4325 COc1ccc2cc[nH]c2n1 SS-4327 CN(C)C/C=C/C(=O)O.Cl SS-4328 CC(C)(C)OC(=O)NC(C/C=C/c1ccccc1)C(=O)O.C1CCC(CC1)NC2CCCCC2 SS-4329 CC1(OCC(O1)C2C(OC(O2)(C)C)C3COC(O3)(C)C)C SS-4330 c1cn2ccnc(c2n1)Cl SS-4331 CCc1cnn2c1nc(cc2Cl)Cl SS-4332 CN(C(=O)c1cncc(n1)Cl)OC SS-4333 CC(C)(C)OC(=O)Nc1nccs1 SS-4334 CNC(=O)c1cccc(c1)CN.Cl SS-4335 CC(C)(C)OC(=O)N1CCC(CC1)(C(=O)N)N SS-4336 c1c(nc(cn1)Cl)C(=O)O SS-4337 CC(C)(C)C(=O)Nc1cccc(n1)Br SS-4338 CC(C)(C)OC(=O)N1CCC(=CC(=O)O)CC1 SS-4339 CC(C)(C)OC(=O)N1CCO[C@@H](C1)CO SS-4340 c1c[nH]c(=O)cc1I SS-4341 Cc1c(nc[nH]1)C2CCNCC2.Cl.Cl SS-4342 c1csc2c1nc(nc2Cl)Cl SS-4343 CCOC(=O)Cc1c(ncnc1O)O SS-4344 CC(C)(C)OC(=O)C1CCCC(C1)C(=O)N(C)OC SS-4345 CC(C)(C)OC(=O)N1C[C@@H](C[C@H]1C(=O)N(C)C)O SS-4346 CC(C)(CC1Cc2ccccc2C1)N.Cl SS-4347 CC(C)(C)[Si](C)(C)Oc1ccc2cc[nH]c2c1 SS-4348 C[C@@H](c1c(ccc(c1Cl)F)Cl)O SS-4349 C[C@H](c1c(ccc(c1Cl)F)Cl)O SS-4350 CC(C)(C)OC(=O)N[C@H]1CCCC[C@H]1N SS-4351 CC(C)(C)OC(=O)N[C@@H]1CCCC[C@@H]1N SS-4352 C1[C@@H]2[C@H]1[C@@H](NC2)C(=O)O SS-4354 C1[C@H]2[C@H]1[C@H](NC2)C(=O)O SS-4355 c1ccc2c(c1)c3ccccc3n2CN4CCCC4 SS-4356 C=CCOC(=O)N1CCN([C@@H](C1)C(=O)O)C(=O)OCC2c3ccccc3-c4c2cccc4 SS-4357 c1cc(ccc1CNc2ccc(cc2)F)F SS-4358 CCOC(=O)C(=CNc1ccc(nc1)OC)C(=O)OCC SS-4359 CNC(=O)Cc1ccc(cc1Br)Cl SS-4360 CCOP(=O)(Cc1ccc(cn1)Br)OCC.Cl SS-4361 CNC(=O)Cc1cc(ccc1Br)OC SS-4362 CCC[C@H]1C(=O)N2CCC[C@H]2C(=O)N1 SS-4363 c1ccc(cc1)c2cccc(c2)CCO SS-4364 Cc1cc2c(cc1C(=O)C)C(C(C2(C)C)C)(C)C SS-4365 CCCCCCC(C)(C)c1cc(cc(c1)O)O SS-4366 C[C@@H]1C[C@H](N(C1)C(=O)OC(C)(C)C)C(=O)O SS-4367 CN1C(=O)COC1=O SS-4369 CC(C)(C)OC(=O)N1CCC2(CC1)CC(=O)c3ccccc3O2 SS-4370 c1ccc(cc1)[C@H]2CCN[C@@H]2C(=O)O.Cl SS-4371 c1c[nH]c2c1ccnc2Cl SS-4372 C1CC2CCC1[C@H]3[C@@H]2C(=O)NC3=O SS-4373 c1ccc(cc1)SCC(CSc2ccccc2)O SS-4374 CCOC(=O)/C=C/c1cc(ccc1F)[N+](=O)[O-] SS-4375 CC(C)(C)O[C@H]1CCN([C@@H]1C(=O)O)C(=O)OCC2c3ccccc3-c4c2cccc4 SS-4376 Cc1ccc(cc1)/C=C/C(=O)N2[C@H](COC2=O)c3ccccc3 SS-4377 CC(C)(C)OC(=O)N1CCC2(CC1)CC(CO2)O SS-4378 Cc1ccc(cc1F)c2ncon2 SS-4379 c1ccc(cc1)COC(=O)N[C@@H]2CC[C@@H](C2)CO SS-4380 c1ccc(cc1)COC(=O)N[C@@H]2CC[C@@H](C2)C(=O)O SS-4381 c1ccc(cc1)COC(=O)N[C@@H]2CC[C@@H](C2)N.C(=O)(C(=O)O)O SS-4382 CC(C)(C)OC(=O)N[C@@H]1CC[C@@H](C1)C(=O)O SS-4383 COC(=O)[C@H]1CC[C@H](C1)NC(=O)OCc2ccccc2 SS-4384 C[C@@H]1C[C@H](NC1)C(=O)O.Cl SS-4385 c1(c(non1)N)C(=N)NO SS-4387 CC1(Cc2c(cc(cc2O1)C(=O)OC)O)C SS-4388 CC(C)(C)OC(=O)N1CCO[C@@H](C1)C(=O)O SS-4389 CC(C)/C(=C\c1ccc(c(c1)OCCCOC)OC)/C(=O)O SS-4390 CS(=N)(=O)C SS-4392 c1ccc(cc1)COCON SS-4393 C[C@@H](CN)CO SS-4394 CN(C)C(=O)CC1CCCC1=O SS-4395 CC1(CN1)C SS-4396 c1ccc(cc1)[C@H]2COCC(=O)N2 SS-4399 c1cc(ccc1S(=O)(=O)Nc2nccs2)Br SS-4400 COc1ccc2c(c1)cc(cn2)F SS-4402 COc1ccc2c(n1)c(ccn2)Br SS-4403 CC1C(=O)Nc2ccc(cc2C(=N1)c3ccccc3)Cl SS-4406 COC(=O)C(=O)/C=C/c1ccccc1Br SS-4407 COC(=O)/C=C(\C(=O)OC)/Nc1c[nH]c(=O)[nH]c1=O SS-4408 CCC(=O)c1ccc(cc1)OC(=O)C(C)(C)C SS-4410 c1cc(c(c(c1)F)SCC(=O)O)[N+](=O)[O-] SS-4412 COc1cc(c(cc1Cl)OCC=C)[N+](=O)[O-] SS-4413 COC(=O)C(=O)/C=C/c1cccc(c1)Cl SS-4414 CCOC(=O)c1ccc(c(c1)Br)C(=O)OCC SS-4415 CN(C(=O)C1CCN(CC1)C(=O)OCc2ccccc2)OC SS-4416 COc1cc(c(cc1OC)Br)CCC#N SS-4417 c1ccc(c(c1)C(=N)N)Cl SS-4420 CC(C)(C)OC(=O)Nc1ccccc1OC SS-4421 COC(=O)c1cc(cc(c1)F)C#N SS-4423 CC(=O)c1cc2cc(ccc2[nH]1)F SS-4424 CC[C@@H](c1ccc(c(c1)F)F)N.Cl SS-4425 c1ccc2c(c1)c(nn2Cc3ccc(cc3)F)C(=O)O SS-4426 c1cc(ccc1C(=O)c2cc(cs2)Cl)F SS-4427 c1cc(ccc1CC2CCNCC2)F SS-4428 c1cc(ccc1C(c2ccncc2)O)F SS-4429 CC(=O)Oc1ccc2c(c1)CC[C@@H]3[C@@H]2CC[C@]4([C@H]3CCC4=O)C SS-4431 c1c[nH]c2c1cc(cn2)F SS-4432 CC(C)(C)OC(=O)N(c1ncc(cn1)Br)C(=O)OC(C)(C)C SS-4436 CC(C)(C)OC(=O)n1c2ccccc2c(n1)I SS-4437 CC(=O)/C(=C\c1ccccc1[N+](=O)[O-])/C(=O)OC SS-4438 c1cc(ccc1S(=O)(=O)Nc2nncs2)Br SS-4440 c1cc2ccc(nc2c(c1)Br)Cl SS-4441 c1cc2ccc(=O)[nH]c2c(c1)Br SS-4442 COC(=O)c1ccc(cc1)c2n[nH]nn2 SS-4444 CCN(CC)C(=O)CS(=O)(=O)c1ccccc1 SS-4446 CCOC(=O)c1cccn2c1nnc2CC3CCN(CC3)C(=O)OC(C)(C)C SS-4447 CC[C@H](c1ccc(c(c1)Cl)Cl)N.Cl SS-4449 CN(CCC(=O)O)Cc1ccccc1 SS-4451 c1cc(ccc1C#N)c2ccc(c(c2)I)O SS-4452 CC(=O)c1cnn(c1N)C SS-4454 CC(C)(C)OC(=O)N1C2C=CC1c3c2cccc3 SS-4455 Cc1c(ncnn1)O SS-4457 c1cc(nc2c1nc(s2)N)Br SS-4460 CCOC(=O)c1c2ccc(cc2sn1)Br SS-4462 c1ccc2cc(ccc2c1)CCCC(=O)O SS-4463 COc1cc(ccc1CC(=O)OC)O SS-4464 CC(C)(C)OC(=O)N1CCC(CC1)COC SS-4465 CC(C)(C)OC(=O)N1CC2C(C1)O2 SS-4524 Cc1cc(ccc1OCc2ccccc2)C=O SS-4525 CC(C)(C)OC(=O)N1CCC(CC1)Nc2cc(ncn2)Cl SS-4526 CN(C)CC[C@H](c1ccccc1)O.C(=O)(C(=O)O)O SS-4527 C1C(CN1)F.Cl SS-4528 CC(C)(C#N)c1cc(ccn1)I SS-4529 CC(C)(C)O[C@@H]1CCN([C@@H]1C(=O)O)C(=O)OCC2c3ccccc3-c4c2cccc4 SS-4530 COc1ccc2c(c1)c(cs2)C(=O)O SS-4531 CC(C)(C)OC(=O)N1CC2CC1C(C2)O SS-4532 CC(C)(C)OC(=O)NCC(=O)NN SS-4533 Cc1c(c(n(n1)c2ccccc2)N)C#N SS-4534 c1c(sc(n1)Br)C(=O)N2CCCC2 SS-4535 Cc1ccc(cc1)C(=O)c2ncccn2 SS-4536 COC(=O)C(=O)/C=C/c1ccc(cc1)Br SS-4537 COC(=O)C(=O)/C=C/c1cccc(c1)Br SS-4538 C[Sn](C)(C)c1cc(ncc1Cl)Cl SS-4539 COC(=O)CCC1=C(NC(=O)C1)c2ccc(cc2)Cl SS-4540 c1c(cc(c2c1[nH]c(=O)o2)[N+](=O)[O-])Cl SS-4541 c1ccc2c(c1)CCC(C(=O)N2)N3C(=O)c4ccccc4C3=O SS-4542 c1cc(cc(c1)[N+](=O)[O-])C(=O)C(F)(F)F SS-4545 CC1(Cc2c(ccc(c2O1)OC)Br)C SS-4546 Cc1cc(c(nc1)Br)C SS-4547 COc1ccc2cc(cnc2c1)Cl SS-4548 Cc1c2ccccc2nc(n1)NC(=N)N SS-4549 c1ccc2c(c1)c3cc(ccc3[nH]2)c4[nH]nnn4 SS-4550 CC(C)(C)OC(=O)Nc1c(cccc1OC(F)(F)F)C(=O)O SS-4551 COc1c2cc(c(cc2ccn1)F)Cl SS-4552 c1cc(c(cc1[N+](=O)[O-])F)Oc2ccnc(c2)NC(=O)N3CCOCC3 SS-4553 CCOC(=O)CC1(Cc2ccccc2C1)N.Cl SS-4554 C1CC2(CC(=C1)/C=C/C(=O)O)OCCO2 SS-4555 c1cc2c(cc1O)c3c(c(=O)o2)CCC3 SS-4556 CSc1c(cnc(n1)Cl)F SS-4557 CC1(C(=O)Nc2c(ccc(n2)[N+](=O)[O-])O1)C SS-4558 COP(=O)(N1CCOCC1)OC SS-4559 CC1(OCCO1)CN SS-4560 CC(C)(C)OC(=O)N1CCC(CC1)CS(=O)(=O)c2cc(cc(c2)F)C(F)(F)F SS-4561 CC(C)(C)OC(=O)CC(C=C)O SS-4562 B1(OC(C(O1)(C)C)(C)C)c2ccnc(c2)C(C)(C)C#N SS-4563 Cc1ccccc1NC(=O)OC(C)(C)C SS-4564 c1ccc(cc1)[C@@H]2COCC(=O)N2 SS-4565 CC(C)(C)OC(=O)N1CC2CC1CC2O SS-4566 C[Si](C)(C)Oc1cc(cc(c1)Br)Br SS-4567 c1cc(ccc1NCC(=O)O)[N+](=O)[O-] SS-4568 CCCc1c(c([nH]n1)C(=O)N)[N+](=O)[O-] SS-4569 C=CCNC(=O)OCC1c2ccccc2-c3c1cccc3 SS-4570 c1cnn2c1ncc(c2)Br SS-4574 COc1ccc(cc1)N2CCN(CC2)c3ccc(cc3)N SS-4575 CN(C)CC[C@@H](c1ccccc1)O.C(=O)(C(=O)O)O SS-4576 CCOC(=O)c1ccc(nc1)NC(=O)OC(C)(C)C SS-4577 Cc1c(sc(n1)C)CC(=O)O SS-4578 c1ccc2c(c1)c(n[nH]c2=O)Cc3ccc(c(c3)C(=O)O)F SS-4579 CCOC(=O)C(c1c(cc(c(n1)Cl)[N+](=O)[O-])Cl)C(=O)OCC SS-4580 c1ccc(cc1)COC(=O)CCCCCCCCCCCCCCCCC(=O)O SS-4581 CC(C)(C)OC(=O)CCCCCCCCCCCCCCC(=O)O SS-4582 CC(C)(C)OC(=O)CCCCCCCCCCCCC(=O)O SS-4583 CCOC(=O)CCCc1nc2cc(ccc2n1C)[N+](=O)[O-] SS-4584 c1c(c[nH]c1C(=O)O)C#N SS-4585 c1ccc2c(c1)CCCC23CCNCC3.Cl SS-4586 CC(C)(C)OC(=O)CCCCCCCCCCCCCCCCCCC(=O)O SS-4587 CC(C)(Cc1c[nH]c2c1cccc2)N SS-4588 c1cc(c(c(c1)Br)Cl)C(=O)O SS-4589 COC(=O)[C@H]1C[C@H](CCN1)O.Cl SS-4590 c1cc(cnc1)C(=O)N2CCCCC2C(=O)O SS-4591 COC(=O)c1ccc(s1)Br SS-4592 c1c(c(nc(n1)Cl)NCC(F)(F)F)C#N SS-4593 C=CCc1cccc(c1O)C(=O)O SS-4594 CC(C)(C)OC(=O)CCCCCCCCCCCCCCCCC(=O)O SS-4595 C[C@@H](CO)C(C)C SS-4597 CC(C)(C)OC(=O)Nc1ccc2c(c1)NC(=O)C2 SS-4598 c1cc(nc2c1ncc(=O)[nH]2)N SS-4599 c1ccc(cc1)c2nc(on2)c3cccs3 SS-4600 c1(c([nH]c(=O)[nH]c1=O)N)Br SS-4601 CN(C(=O)c1c(ncnc1Cl)Cl)OC SS-4602 Cc1c(c(nc(n1)N)O)[N+](=O)[O-] SS-4603 Cc1cccc(c1NC)C SS-4604 Cc1c(c(sn1)N)C(=O)O SS-4605 c1cnccc1c2cc(c(=O)[nH]c2)C(=O)O SS-4606 c1ccc(cc1)c2nc(on2)c3ccco3 SS-4607 Cc1nc(c(s1)c2ccccc2F)C(=O)O SS-4608 CN(C)C(=S)Oc1cc(ccc1C(=O)OC)OC SS-4609 CC(C)(C(=O)N1CCCC1)Br SS-4610 CC(C)COc1cc(cc(c1)OC(C)C)C(=O)O SS-4612 c1ccc(cc1)COC2CC(=O)C2 SS-4613 Cc1nnc(o1)CCl SS-4614 C[C@@H]1C[C@@H](c2ccccc2N1)C(=O)OC SS-4615 B1(OCC(CO1)(C)C)c2ccccc2C#N SS-4616 C[C@@H](c1ccccc1)NO.C(=O)(C(=O)O)O SS-4617 C=C[C@@H](c1ccc(cc1)C(F)(F)F)N.Cl SS-4618 CN(C)c1ccc(cc1)C(C(=O)c2ccccc2)O SS-4619 c1ccc(c(c1)NC(=O)[C@H]([C@@H](C(=O)O)O)O)Cl SS-4621 CC(C)(C)OC(=O)CCCCNC(=O)OCc1ccccc1 SS-4622 CC(c1ccc(cc1)F)C(=O)O SS-4623 Cc1cc(c(nc1)[N+](=O)[O-])O SS-4625 CC(C)(C)c1ccc2c(c1)CC[C@H]2N SS-4626 C[C@@H]1C[C@H]1C(=O)O SS-4627 Cc1cccc(c1)/C=C/C(=O)c2ccccc2 SS-4629 C1CC(=COC1)C(=O)O SS-4630 COc1ccc(cc1OCCCCl)C=O SS-4631 COc1ccc2c(c1I)CCCC2=O SS-4632 CC(C)(CO)C(c1ccccc1)N SS-4634 CC(C)(CO)C(c1ccccc1)N SS-4635 COc1c2c(ncn1)CCNC2 SS-4636 CC(C)(CO)[C@H](c1ccccc1)N SS-4638 COC(=O)c1c2ccccc2[nH]n1 SS-4639 Cn1c(c(cn1)C(=O)O)Br SS-4640 c1c2cn[nH]c2ncc1Cl SS-4641 CCOC(=O)c1cnn(c1)c2ccc(cn2)C=O SS-4642 CC(C)(C)OC(=O)Nc1ncc(s1)Br SS-4643 COc1ccc(cc1)C(=O)ON.CS(=O)(=O)O SS-4644 CCCCCCCCOc1ccc(cc1)c2cccs2 SS-4645 c1cc(c2c(c1)OCCO2)N.Cl SS-4646 CN1C2CCC1CNC(=O)C2 SS-4647 Cc1c(c(cc2c1OCO2)[N+](=O)[O-])C(=O)O SS-4648 COc1ccc(c(c1)OC)CNc2ncns2 SS-4649 C/C(=N\c1ccccc1C#N)/N(C)C SS-4650 c1cc2nc(cn2cc1Br)C(=O)O SS-4651 C[C@@H](CO)C(C)(C)O SS-4652 COc1ccc(c(c1)OC)CNCC#N.Cl SS-4653 C[n+]1ccc(cc1)N.[I-] SS-4654 c1c(c(n(n1)C2CCOCC2)N)C(=O)N SS-4655 Cc1cc(c(cc1C(=O)O)F)F SS-4656 COc1ccccc1c2c[nH]c3c2cc(cn3)Br SS-4657 CC(C)(C)OC(=O)N[C@H](c1ccc(cc1)OS(=O)(=O)C(F)(F)F)C(=O)OC SS-4658 Cc1c(n(cn1)C(c2ccccc2)(c3ccccc3)c4ccccc4)C SS-4659 c1cc(ccc1[C@@H](C(=O)O)O)Br SS-4660 CC(C)(CCC(C)(C)Cl)Cl SS-4661 c1cc(ccc1[C@H](C(=O)O)O)Br SS-4662 CN1CCN(CC1)C(=O)c2ccc(cc2)[N+](=O)[O-] SS-4663 CC(C)(C)NCC(=O)COc1ccccc1.Cl SS-4664 CN1C(=O)C(=C(C1=O)Br)Br SS-4665 c1cncc2c1cc(c(c2)Cl)F SS-4666 c1ccc(cc1)C2(CCC3(CC2)OCCO3)C=O SS-4667 C[C@@H]1CN(C[C@H]1C(=O)OC)Cc2ccccc2 SS-4668 Cc1cn(cn1)c2ccc(nc2OC)Br SS-4669 C1CNC[C@@H]1C(=O)O SS-4670 CC(C)(C)[Si](c1ccccc1)(c2ccccc2)OCCC=C SS-4671 Cc1ccc(cc1)S(=O)(=O)n2cc(c3c2ncnc3Cl)Br SS-4672 C1CC2=C(CC(=O)N2)C(=O)C1 SS-4673 c1c(c(nc(c1F)Cl)Cl)C(=O)N SS-4674 CCOC(=O)C1Cc2cccc(c2O1)[N+](=O)[O-] SS-4675 Cc1cc(c2cc(ccc2n1)NC(=O)C)OC SS-4676 COc1cc(cc(c1OC)OC)C(=O)C(=O)O SS-4677 c1ccc(cc1)COC(=O)NCCc2ccc(cc2)O SS-4678 C1CC/C=C\C(CC1)N SS-4679 CCCCCCc1ccc(c(c1)C(=O)C)O SS-4680 CC(C)(C)OC(=O)N1CC2CC(=O)CC2C1 SS-4681 c1cc(c2c(c1)[nH]c(=O)o2)CCO SS-4682 c1ccc(c(c1)Oc2c(cccn2)Br)Cl SS-4683 c1ccc(c(c1)Oc2c(cccn2)Br)F SS-4684 CC(C(=O)c1ccc(cc1)OC(=O)C(C)(C)C)Br SS-4685 Cc1cn(cn1)c2ccc(nc2OC)C(=O)OC SS-4686 C[C@@H](C(=O)NN)NC(=O)OC(C)(C)C SS-4687 CCOC(=O)C(=C1SCS1)C(=O)C SS-4688 COc1cc(ccc1c2ccnc(c2)Cl)F SS-4689 c1cc(cc(c1)Nc2cc(ncn2)Cl)C(F)(F)F SS-4690 C=CCCCCC[C@@H](C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 SS-4691 COC(=O)c1cc(c(c(c1Nc2ccccc2)F)N)[N+](=O)[O-] SS-4692 C[C@H](C(=O)NN)NC(=O)OCc1ccccc1 SS-4693 CCc1c(ncnc1O)O SS-4694 Cn1cnc2c1cc(c(c2F)N)C(=O)OC SS-4695 COc1cccc(c1O)[N+](=O)[O-] SS-4696 C1CNCCC1NN.Cl.Cl SS-4697 Cc1cc(c(cc1C(=O)O)[N+](=O)[O-])Cl SS-4698 COC(=O)[C@@H]1[C@H]2[C@@H]1CC/C=C\CC2 SS-4699 c1csc2c1scc2Br SS-4700 c1ccc(c(c1)C(=O)O)Nc2ccnc3c2cccc3C(F)(F)F SS-4701 CCOC(=O)c1cc2n(n1)CCN(C2)C(=O)OCc3ccc(cc3)[N+](=O)[O-] SS-4702 COC(=O)[C@H]1[C@H]2[C@@H]1CC/C=C\CC2 SS-4703 c1ccc(cc1)Nc2ccnc3c2cccc3 SS-4706 Cc1c(cccc1I)CO SS-4707 c1c(c(cc(c1F)[N+](=O)[O-])Br)N SS-4708 c1ccc2c(c1)CCC(=O)CC2 SS-4709 CC(C)OC(=O)c1ccc(s1)Br SS-4710 CCOC(=O)Cn1c(cc2c1CCCC2=O)C SS-4711 C1C(=O)N=C2N1C=CC=C2.Br SS-4713 CCOC(=O)C1Cc2c(nc(n2C)C)C(=O)C1 SS-4714 CCOC(=O)c1ccc(cc1)N2C[C@H](N[C@H](C2)C)C SS-4715 CCCc1ccc(s1)C(=O)NC(C)(C)C SS-4717 COc1ccc(cc1)C(=O)C2CCNCC2.Cl SS-4719 COC(=O)c1cc(cc(c1)OCc2ccccc2)O SS-4720 Cc1cc(cc(c1C(=O)c2ccc(cc2)C(=O)c3c(cc(cc3C)C(C)(C)C)C)C)C(C)(C)C SS-4721 c1c(cc(cc1F)F)NC(=O)C(F)(F)F SS-4722 CC1(O[C@@H]2[C@@H]3[C@@H]([C@H](C(=O)O3)O)O[C@@H]2O1)C SS-4723 c1cc(ccc1N2C(=O)C=CC2=O)[N+](=O)[O-] SS-4724 Cc1ccc(cc1)S(=O)(=O)N2CCC3(CC2)OCCO3 SS-4725 CC(=O)Cc1cc(c(cc1[N+](=O)[O-])OC)OC SS-4726 CCC(c1ccccc1)C(=O)c2ccc(cc2)OCCCl SS-4727 CN1C=Cc2ccc(cc2CC1=O)OC SS-4729 Cc1ccc(cc1)S(=O)(=O)n2cc(c3c2ncc(c3)Cl)Br SS-4731 C1C2CC1(C2)C(=O)O SS-4732 CC(C)(C)OC(=O)N1Cc2ccc(cc2C1)CCO SS-4733 CC1(COC2(CC3CC(=C(C3C2)C(=O)OC)O)OC1)C SS-4737 CC1=CCC(CC1)C(=O)O SS-4738 Cc1cc(ccc1Cl)c2cc(n[nH]2)C(=O)OC SS-4739 CC(C)n1c2cc(cc(c2cn1)C(=O)OC)Br SS-4740 CCOC(=O)c1cc(n(n1)C)c2ccc(cc2)Cl SS-4741 CC1(COC2(CC3CC=CC3C2)OC1)C SS-4742 CCOC(=O)c1cc(n(n1)C)c2ccc(c(c2)F)F SS-4743 CC(C)(CO)[C@H](c1ccccc1)O SS-4745 CCOC(=O)c1cnn(c1N)Cc2ccccc2 SS-4747 CCOC(=O)c1cc(n(n1)C)c2cc(cc(c2)Cl)Cl SS-4748 c1ccc(cc1)C2C[C@@H]2N.Cl SS-4749 c1ccc(c(c1)NC(=O)[C@@H]([C@H](C(=O)O)O)O)Cl SS-4750 c1ccc(cc1)c2ccccc2C(=O)Nc3ccc(c(c3)Cl)C(=O)O SS-4751 CC(OC(=O)N[C@H]1CC[C@H](CC1)N)(C)C SS-4753 C[C@@H](CO)COCc1ccc(cc1)OC SS-4755 CC1=CCC(CC1)C(=O)OC SS-4756 c1cc(cc(c1)[N+](=O)[O-])c2ncccn2 SS-4757 c1ccc(c(c1)C(=O)c2cnc(s2)N)Cl SS-4758 CCn1c2c(cncc2Br)nc1c3c(non3)N SS-4759 c1cc(ccc1Cn2cc(cn2)CO)F SS-4760 c1ccc2c(c1)c(cc(c2N)Br)Br SS-4764 CCCC[C@@H](C(=O)OCc1ccccc1)N.Cc1ccc(cc1)S(=O)(=O)O SS-4765 CC1(COC2(CC3CC(=O)CC3C2)OC1)C SS-4766 C=C[C@H](c1ccc(cc1)C(F)(F)F)N.Cl SS-4767 C1C[C@@H]2C[C@H]1C[C@H]2N.Cl SS-4768 c1ccc(cc1)c2ccc3ccccc3c2 SS-4770 Cc1c(c2ccccc2n1C(=O)OC(C)(C)C)I SS-4771 CCCC(CC1(CCCC1)C(=O)O)C(=O)OCc2ccccc2 SS-4772 C[C@]12CCC(=O)C=C1CCCC2=O SS-4773 CCOC(=O)c1c(c2c(o1)CCCC2=O)C SS-4774 Cc1cc(cc(c1O)C)C(=O)OCc2ccccc2 SS-4775 C[C@H](CO)C1CCC2[C@@]1(CCCC2O)C SS-4776 C1C[C@H]2C[C@@H]1C[C@@H]2N.Cl SS-4778 c1cc(cc(c1)Cl)c2ccnc(n2)N SS-4779 CCOC(=O)c1c2c([nH]n1)CCN(C2)C(=O)OC(C)(C)C SS-4780 c1ccc2c(c1)CC(C2)(CC(=O)O)N SS-4781 c1ccc(cc1)COc2ccccc2C3CCC3=O SS-4782 Cc1cn(cn1)c2ccc(cc2OC)C#N SS-4784 c1ccc(cc1)COC(=O)Nc2ccc(c(c2)F)N3CCSCC3 SS-4785 CCCSc1nc(c2c(n1)n(cn2)[C@H]3[C@@H]([C@@H]([C@H](O3)CO)O)O)N SS-4786 CCCSc1nc(cc(n1)N)N SS-4789 Cc1ccc(cc1)S(=O)(=O)O[C@@H]2CO[C@H]3[C@@H]2OC[C@@H]3OS(=O)(=O)c4ccc(cc4)C SS-4790 c1c(cc(c2c1C(=O)CCO2)Br)Br SS-4791 c1ccc(c(c1)CN2CCC(=O)CC2)C(F)(F)F SS-4792 c1ccc(cc1)COC(=O)N2CCC3(CCC(=O)CC3)CC2 SS-4793 c1ccc2c(c1)[nH]c(n2)CN(Cc3[nH]c4ccccc4n3)Cc5[nH]c6ccccc6n5 SS-4794 CNCCCc1[nH]c2ccccc2n1 SS-4795 CCOC(=O)c1c2c(sc1NC(=O)C)C(=O)CCC2 SS-4796 c1ccc2c(c1)c(=O)nc(o2)c3ccccc3O SS-4797 Cc1ccc(cc1)S(=O)(=O)NCCNS(=O)(=O)c2ccc(cc2)C SS-4798 Cc1cc(cc(c1NN)C)Br.Cl SS-4799 c1ccc2c(c1)c(=O)cc(o2)c3ccncc3 SS-4800 c1ccc(cc1)COC2CCC(=O)CC2 SS-4801 CC(C)(C)OC(=O)N1CC[C@@H]([C@@H](C1)F)O SS-4802 CC(C)(C)OC(=O)N1CC[C@H]([C@H](C1)F)O SS-4803 c1cc2c3c(c1)[nH]c(=O)n3CCC2=O SS-4804 c1cc2c(cc1O)c(cs2)C(=O)O SS-4805 CC(C)(C1CCNCC1)S(=O)(=O)c2cc(cc(c2)F)C(F)(F)F.Cl SS-4806 CC(C)(C)OC(=O)NCC(=O)OCc1ccccc1 SS-4808 c1ccc(c(c1)C(C(=O)N)N)Cl.Cl SS-4809 CCOC(=O)c1cnc2n(c1=O)ccs2 SS-4810 c1c(c(c(nc1Br)Cl)O)Br SS-4811 COc1cc(c(nc1)CO)F SS-4812 CCCCCNS(=O)(=O)c1ccc(cc1)CC SS-4813 CC(C)(C)C(=O)OCc1cc(ccc1OC)c2ccc3c(n2)nc(nc3Cl)Cl SS-4815 COC(=O)C(c1ccccc1Cl)N.Cl SS-4816 c1cnc2c(c1Cl)cc(cc2C(F)(F)F)I SS-4817 COC(=O)c1c(noc1C2CC2)c3c(cccc3Cl)Cl SS-4818 CC(C)(CO)[C@@H](c1ccccc1)O SS-4819 COc1cc(cnc1CO)F SS-4820 CC(C)(CO)C(c1ccccc1)O SS-4823 C(c1nc([nH]n1)N)C(=O)O SS-4824 COc1ccc(cc1)Cn2c3ccccc3c(n2)C(=O)OC SS-4825 COc1ccc(cc1)Cn2c3ccccc3c(n2)C(=O)O SS-4828 C[C@@]12CC[C@@H]3c4ccc(cc4CC[C@H]3[C@@H]1C=C[C@@H]2O)OC SS-4829 CCOC(=O)c1cnn2c1CN(CC2)C(=O)OC(C)(C)C SS-4830 c1c(c(cc(c1F)Br)F)C=O SS-4831 c1ccc(cc1)Cc2ccc(cc2)CO SS-4832 c1ccc(c(c1)C2=NCCN2)N SS-4833 c1ccc(cc1)[C@@H]2COC(=O)N2C(=O)CBr SS-4834 CC(C)(C#N)c1c(cccc1Cl)Cl SS-4835 CCOC(=O)c1c(nc(nc1C)C)C SS-4836 c1ccc(cc1)CN2CCOC(C2)CN SS-4839 Cc1cc(c(c(c1)C)Nc2ccnc(n2)Cl)C SS-4840 CC(C)(C)[Si](c1ccccc1)(c2ccccc2)O[C@H]3CCC(=O)[C@@H](C3)F SS-4841 c1ccc(cc1)[C@@H](CC(=O)O)C(=O)O SS-4842 COc1cccc2c1CC[C@@H](C2)N.Cl SS-4843 c1ccc(cc1)[C@H](CC(=O)O)C(=O)O SS-4844 C[S@@](=N)(=O)c1ccccc1 SS-4845 C[S@](=N)(=O)c1ccccc1 SS-4846 Cc1cc(cc(c1)NC(C)C)C SS-4847 c1ccc(cc1)CN2CC3(CCCNCC3)OC2=O.Cl SS-4848 Cc1cn(cn1)c2ccc(cc2OC)C(=O)O SS-4849 Cc1cc(c(=O)n(c1)C)C SS-4850 CC(C)(C)OC(=O)N1CCC2(CC1)CN(C(=O)CC2=O)Cc3ccc(cc3)OC SS-4852 CN1CCCN=C(C1=O)c2ccccc2 SS-4853 C[C@@H](c1ccccc1)NC(=O)c2ccccc2C(=O)O SS-4856 C[C@H](c1ccccc1)NC(=O)c2ccccc2C(=O)O SS-4857 COc1cc2cc[nH]c2cc1F SS-4859 Cc1c(c2c(c(c1O)C)CC[C@](O2)(C)C(=O)O)C SS-4860 CC(C)(C)c1ccc2c(c1)CC[C@@H]2N SS-4863 Cc1c(c2c(c(c1O)C)CC[C@@](O2)(C)C(=O)O)C SS-4864 C1C[C@@H](C[C@H](C1)O)N.Cl SS-4867 C1C2CC(=O)NCC2CC1=O SS-4868 C1C[C@H](C[C@@H](C1)O)N.Cl SS-4869 c1ccc(cc1)CO[C@H]2CCC(=O)[C@H](C2)F SS-4870 c1ccc(cc1)CO[C@H]2CCC(=O)[C@@H](C2)F SS-4871 C[C@H]1C[C@@H]1C(=O)O SS-4872 c1cc(ccc1C#N)C2CCNCC2.Cl SS-4873 CCOC(=O)/C=C/c1ccc(cc1Br)F SS-4874 CC(=O)CCCO[Si](C)(C)C(C)(C)C SS-4875 C[C@H](c1ccccc1)N2CCCC2=O SS-4876 CC(=O)Nc1ccc(nn1)Cl SS-4877 c1cc(ccc1c2nc(on2)c3ccc(o3)Br)F SS-4878 C[C@@H](c1cccc(c1)N)N SS-4879 C/C(=C\c1ccc(c(c1)F)Cl)/C(=O)O SS-4880 c1cc(ccc1C=O)Oc2ccc(cc2)Oc3ccc(cc3)C=O SS-4881 Cc1ccc(cc1)S(=O)(=O)O[C@H](CNC(=O)OCc2ccccc2)[C@@H]3C=CCO3 SS-4882 Cc1ccc(cc1)S(=O)(=O)ON=C2CCOCC2 SS-4883 c1c(c(nc(c1[N+](=O)[O-])Cl)C(F)(F)F)[N+](=O)[O-] SS-4884 c1ccc(cc1)CN2CCO[C@H](C2)CN SS-4885 CC(C)(C)C(=O)N1CCN(CC1)Cc2ccccc2 SS-4886 c1ccc(cc1)CN2CCO[C@@H](C2)CN SS-4887 CC(C)(C)OC(=O)N1CC(=C)C1 SS-4888 CC(C)(C)OC(=O)N1CCC2(CC1)CC(=O)C2 SS-4889 COc1ccccc1NC(=O)[C@@H]([C@H](C(=O)O)O)O SS-4890 c1ccc(cc1)NC(=O)[C@H]([C@@H](C(=O)O)O)O SS-4891 c1ccc(cc1)NC(=O)[C@@H]([C@H](C(=O)O)O)O SS-4892 COc1ccccc1NC(=O)[C@H]([C@@H](C(=O)O)O)O SS-4893 Cc1ccccc1NC(=O)[C@H]([C@@H](C(=O)O)O)O SS-4894 C1CCN(CC1)CCCS(=O)(=O)O SS-4895 CC(=O)Oc1ccc2c(c1)CC=C3[C@@H]2CC[C@]4([C@H]3CCC4=O)C SS-4896 CC(C)(C)OC(=O)N1CC2(C1)CC(=O)C2 SS-4897 COc1cncc(n1)C(=O)OC SS-4898 C1C2CC3CC1CC(C2)(C3)C(=O)NN SS-4899 c1ccc(cc1)COc2ccc(cc2OCc3ccccc3)C[C@@H](C(=O)O)NC(=O)OCc4ccccc4 SS-4900 Cn1c(cc(n1)O)C(=O)OC SS-4901 c1ccc(cc1)COC(=O)N[C@H]2CCCC[C@H]2N.C(=O)(C(=O)O)O SS-4902 c1cc2c(cc1I)c(ncn2)O SS-4903 c1ccc(cc1)COc2ccc3c(cc(=O)oc3c2)O SS-4904 CC(C)(C)OC(=O)N1CCC2(C1)CC(=O)C2 SS-4905 Cc1c(c2c(c(c1O)C)CCC(O2)(C)C(=O)N3CCNCC3)C.Cl SS-4906 c1ccc(cc1)C[C@H](c2ccccc2)N SS-4907 c1ccc(cc1)C[C@@H](c2ccccc2)N SS-4908 CC(C)(C)OC(=O)N1CCC2(CC1)CC(=O)N2 SS-4909 CC(C)(C)OC(=O)N1CCC2(CC1)Cc3cc(ccc3O2)C(=O)O SS-4910 c1ccc2c(c1)CC3(O2)CCNCC3 SS-4912 c1c(c(c(cn1)Br)Cl)F.Cl SS-4913 CC(C)(CN=[N+]=[N-])C(=O)O SS-4925 CS(=N)(=O)C1CC1 SS-4928 c1c(cnc(n1)C(F)(F)F)C=O SS-4929 c1c(cnc(n1)C2CC2)C=O SS-4930 C1CC1NC(=O)C(=O)O SS-4931 C1C2CC1(NC2)C(=O)O.Cl SS-4932 COC(=O)C12CC(C1)CN2.Cl SS-4933 c1cc(ccc1CCl)OCCN2CCCCCC2.Cl SS-4934 CCOC(=O)[C@H]([C@H](c1ccccc1)N)O SS-4935 Cc1c(n2c(n1)C(=O)CCC2)C SS-4936 CCOC(=O)[C@@H]([C@@H](c1ccccc1)N)O SS-4937 CC(C)(C)OC(=O)N1CCC(CC1)Oc2ccc(nc2)Br SS-4939 CC(C)(C)OC(=O)Nc1ccc(c(c1)C(F)(F)F)OC SS-4941 CC1CC(NC1)(C)C.Cl SS-4942 CC(C)(C(=O)OC)n1cc(nc1)[N+](=O)[O-] SS-4943 COC(=O)CCCCCCCCCCCBr SS-4946 CC(=C)CNC(=O)OC(C)(C)C SS-4947 COCCON SS-4948 CS(=NCC(=O)O)(=O)C SS-4951 CC1CC(NC1=O)(C)C SS-4953 c1cc(ncc1Br)OCC(F)(F)F SS-4954 c1c[nH]nc1O SS-4955 c1cc2nc(cn2nc1)CCl.Cl.Cl SS-4956 c1ccc2c(c1)c(nc(n2)C(F)F)O SS-4957 c1cc2c(nc1C#N)CCCC2=O SS-4958 c1ccc(cc1)c2cc(nc(n2)Cl)N3CCOCC3 SS-4959 C1C[C@H](C[C@H]1N)O SS-4960 CC1(CC(=C)C(=O)N1)C SS-4961 CC(C)(C)OC(=O)Nc1nc(ns1)Cl SS-4962 CCCCC(=O)c1ccccc1O SS-4963 c1ccc2c(c1)ccc3c2C(=O)CCC3 SS-4964 C[C@](CCCCCCC=C)(C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 SS-4965 CC(C)(CNC(=O)c1cccnc1)S SS-4967 c1ccc(cc1)S(=N)(=O)c2ccccc2 SS-4968 COC(=O)CCc1ccc(c(c1)[N+](=O)[O-])F SS-4969 CCCCCC[C@H](CC(=O)OC)O SS-4970 c1cc(sc1)C(=O)CCC(=O)c2cccs2 SS-4971 CC(C)(C)OC(=O)Nc1cccc(c1)N SS-6000 CCC(C(=O)c1ccc2c(c1)OCO2)NC.Cl SS-6001 c1ccc2c(c1)cc(o2)C(=O)O SS-6002 CC(Cc1ccc2c(c1)cco2)N.Cl SS-6003 Cc1cc2c(cc1C)nc([nH]2)C(=O)C SS-6004 CC(C)(C)OC(=O)n1c2cccc(c2cn1)[N+](=O)[O-] SS-6005 CC(C)(C)OC(=O)n1c2ccc(cc2c(n1)I)[N+](=O)[O-] SS-6006 c1cc2c(cc1N=[N+]=[N-])c(n[nH]2)I SS-6007 c1cc2c(cc1I)c(n[nH]2)I SS-6008 COC(=O)c1cccc2c1[nH]nc2 SS-6009 c1cc(c2c(c1)[nH]nc2C(=O)O)C=O SS-6010 Cc1c2c(cccc2OCc3ccccc3)[nH]n1 SS-6011 Cc1c2c(cccc2Cl)[nH]n1 SS-6012 COC(=O)c1cc(cc2c1cn[nH]2)Br SS-6013 c1c(cc(c2c1[nH]nc2N)Br)Br SS-6014 COC(=O)c1cc2c(cc1Br)cn[nH]2 SS-6015 COC(=O)c1cc(cc2c1[nH]nc2)Br SS-6016 COc1c(ccc2c1cn[nH]2)Br SS-6017 CCc1cc(cc2c1[nH]nc2)Br SS-6018 COc1ccc2c(c1)cn[nH]2 SS-6019 COc1cc(cc2c1cn[nH]2)Br SS-6020 CCOC(=O)/C=C/c1cnc2n1cccc2 SS-6021 CC(C)(C)OC(=O)n1cc(c2c1ccc(c2)Br)I SS-6022 CC(C)(C)OC(=O)N1CC(=O)c2c1cc(cc2)Br SS-6023 c1cc(c2cc[nH]c2c1)C(=O)NN SS-6024 COC(=O)c1cccc2c1cc[nH]2 SS-6025 c1cc(c2cc[nH]c2c1)CO SS-6026 COC(=O)c1ccc2c(c1)cc[nH]2 SS-6027 CC(C)(C)OC(=O)n1ccc2c1ccc(c2)C=O SS-6028 CC(C)(C)OC(=O)n1ccc2c1ccc(c2)C(=O)OC SS-6029 CC(C)(C)OC(=O)N1CCc2c1cc(cc2)C(=O)OC SS-6030 CC(C)(C)OC(=O)N1CCc2c1ccc(c2)CCCl SS-6031 c1cc2c(c(c1)Br)CNC2=O SS-6032 c1c(cc(c2c1C(=O)NC2)Br)O SS-6033 COC(=O)c1ccc2c(c1)CNC2=O SS-6035 c1cc2c(cc1[N+](=O)[O-])CNC2=O SS-6036 c1cc2c(cc1Br)CNC2=O SS-6037 c1cc2c(cc1C(=O)O)CNC2=O SS-6038 c1cc2c(cc1Br)C(=O)NC2 SS-6039 c1cc2c(cc1[N+](=O)[O-])C(=O)NC2 SS-6040 c1ccc2c(c1)CNC2=O SS-6041 c1cc2c(c(c1)I)C(=O)NC2 SS-6042 c1[nH]c2c(c(=O)n1)[nH]nc2I SS-6043 c1cc(ccc1CN2CCNCC2)C(F)(F)F SS-6044 COC(=O)c1cc2c(cn1)c(n[nH]2)Br SS-6045 c1c2c(cn[nH]2)c(nc1Cl)Cl SS-6046 COC(=O)c1cc2c(nc1)N(C(=O)C2)COCC[Si](C)(C)C SS-6047 c1c2c(c(cn1)Br)c(n[nH]2)N SS-6048 c1cncc2c1cn[nH]2 SS-6049 c1c(cncn1)N SS-6051 c1c(cncn1)O SS-6052 c1c(cncn1)I SS-6053 COC(=O)c1c(nc(c(n1)Cl)Cl)N SS-6054 c1c(cncc1I)Br SS-6056 C1CCNC1 STR00030 c1ccc(c(c1)N)Cl STR00033 CCOC(=O)CC#N STR00038 c1c[nH]nc1 STR00103 c1cc(cnc1)C=O STR00136 c1ccc(c(c1)C=O)Cl STR00143 c1cc(cc(c1)Cl)C=O STR00144 c1ccc(cc1)S STR00162 C=CCBr STR00178 C#CCBr STR00180 CC(=N)N.Cl STR00189 CC(C)(C)N STR00192 C1COCCN1 STR00194 c1ccc(cc1)CN STR00195 c1cc(ccc1CN)Cl STR00198 c1ccnc(c1)N STR00201 c1ccc(cc1)S(=O)(=O)NN STR00208 c1ccc(c(c1)C(=O)NN)O STR00212 c1ccc(cc1)N STR00216 COc1ccc(cc1)N STR00220 Cc1ccc[n+](c1)[O-] STR00249 CC(C)(C)C(=O)CC#N STR00250 CN(C)C(OC)OC STR00254 CC1(OC(=O)CC(=O)O1)C STR00259 c1cc[nH]c1 STR00296 C1C(=O)NC(=S)S1 STR00300 c1cc(c(cc1Cl)Cl)O STR00302 c1ccc(c(c1)NN)Cl.Cl STR00333 c1ccc(c(c1)N)O STR00335 COC(CN)OC STR00343 c1cc(oc1)C=O STR00358 c1ccc(cc1)/C=C/C(=O)O STR00363 c1cc(ccc1Cl)I STR00382 C1CSC(=N1)N STR00410 CC(=S)N STR00411 c1cc(ccc1NN)Cl.Cl STR00429 c1cc(c(cc1Cl)Cl)C(=O)Cl STR00436 C1CC1N STR00451 C1CCC(=O)C1 STR00465 c1ccc(c(c1)C(=O)O)S STR00467 COC(=O)c1ccc(cc1)Cl STR00479 c1cnc(nc1)S STR00484 c1ccc(c(c1)C(=O)N)Cl STR00491 c1cc(cc(c1)Cl)C(=O)N STR00492 Cc1cc(=O)[nH]c(=O)[nH]1 STR00504 c1cc(cnc1)CN STR00537 CCOC(=O)CC(=O)c1ccccc1 STR00545 c1cnccc1C(=O)N STR00561 CSc1ccccc1N STR00572 CSc1cccc(c1)N STR00573 c1ccc(cc1)c2ccccc2N STR00574 COc1ccc(c(c1)OC)N STR00575 C1CC(=O)CC(=O)C1 STR00599 C1CCN(CC1)N STR00611 C(C(=O)O)C(=O)O STR00614 COc1cccc(c1)OC STR00616 c1cc(ccc1CC(=O)O)[N+](=O)[O-] STR00634 CCOC(=O)C(=O)CBr STR00638 c1ccc(cc1)Br STR00651 c1cc(ccc1Cl)Br STR00662 c1cc(cc(c1)N)C(=O)O STR00672 c1cc(cc(c1)O)[N+](=O)[O-] STR00679 c1ccc2c(c1)Cc3ccccc3C2=O STR00681 CC(C)(C)C(=O)CC(=O)OC STR00744 COc1ccc(cc1)S STR00751 CC(C)(C)NN.Cl STR00762 C(#N)C(Cl)(Cl)Cl STR00776 c1cc(c(cc1C=O)Cl)Cl STR00782 CCOC(=O)C1CCCC1=O STR00828 c1c[n+](ccc1[N+](=O)[O-])[O-] STR00842 c1cc(ccc1S)Br STR00881 COc1ccc(cc1)NN.Cl STR00890 Cc1cc(c(c(c1)C)N)C STR00896 Cc1ccc(c(c1)C)N STR00897 c1cc(ccc1C=O)[N+](=O)[O-] STR00898 CC(=O)Nc1ccc(cc1)O STR00901 c1ccc(c(c1)[N+](=O)[O-])O STR00905 C(C(=O)O)O STR00936 COC(=O)CO STR00937 CC(=O)c1cccc(c1)[N+](=O)[O-] STR00971 COc1ccc(cc1)C(=O)CBr STR00973 c1cnc(nc1)Cl STR00974 c1cc(c(cc1Cl)Cl)CC#N STR00977 C1C2CC3CC1CC(C2)(C3)N.Cl STR01017 c1cc(oc1)CO STR01021 COC(=O)C=CCBr STR01036 c1ccc(c(c1)C=O)C=O STR01056 CC(=O)N STR01066 c1cc(ccc1C(=O)Cl)[N+](=O)[O-] STR01076 C1CCC(=CC1)N2CCCC2 STR01084 Cc1ccc(cc1)CBr STR01086 c1cc(ccc1N)N STR01091 c1ccc2c(c1)c(ncn2)O STR01100 c1c(c(n[nH]1)N)C#N STR01102 c1ccc(cc1)C=CC#N STR01107 c1ccc(cc1)C(=O)CBr STR01109 CC(=O)c1ccc(cc1)O STR01114 Cc1c(cccc1Cl)Cl STR01117 c1cc(ccc1C(=O)CBr)Cl STR01162 c1cc(ccc1C#N)Cl STR01164 COC(=O)CC#N STR01166 CS(=O)(=O)CC(=O)O STR01174 CCOC(=O)CN.Cl STR01178 C1CC=COC1 STR01188 C(CBr)O STR01207 C(C(CO)O)N STR01210 c1cc(ccc1CC#N)[N+](=O)[O-] STR01247 C1CC(=O)OC1=O STR01303 CN(C)c1ccc(cc1)C=CC=O STR01311 CCNC(=O)N STR01353 c1cc(ccc1C(=O)O)[N+](=O)[O-] STR01385 CC1(C(=O)N(C(=O)N1Br)Br)C STR01390 COC(=O)Cc1ccc(cc1)O STR01403 Cc1ccc(cc1)S(=O)[O-].[Na+] STR01406 Cc1ccccc1Br STR01411 Cc1cccc(c1)Br STR01412 Cc1ccc(cc1)Br STR01413 c1cc(cc(c1)O)C=O STR01419 C1CCCNCC1 STR01425 c1c[nH]c(=O)nc1N STR01426 CCCN STR01427 C1CC1CN STR01428 CC(C)(CN)N STR01438 c1ccc(cc1)C(=O)CC(=O)c2ccccc2 STR01439 CC1(CC(=O)NC(=O)C1)C STR01447 c1ccc(cc1)C(=O)CCl STR01480 CC(C)(C)c1ccc(cc1)CO STR01483 c1c(c(nc(n1)O)O)Br STR01501 c1cc(c(cc1O)O)C=O STR01512 Cc1ccc(cc1)S(=O)(=O)OC STR01542 c1ccc2c(c1)cccn2 STR01546 C=Cc1ccccn1 STR01590 c1cc(c(cc1[N+](=O)[O-])Cl)Cl STR01633 Cc1cccc(c1)C#N STR01636 Cc1cc(ccc1N)Cl STR01685 CC(C)(CO)N STR01693 c1ccc(cc1)C(=O)c2cc(ccc2N)Cl STR01705 c1cc(c(c(c1)Cl)O)Cl STR01713 c1c(cc(cc1[N+](=O)[O-])[N+](=O)[O-])C(=O)O STR01728 c1cc(c(cc1CN)Cl)Cl STR01748 c1ccc2c(c1)c(ccc2Cl)O STR01788 c1cc(c(c(c1)Br)N)Br STR01809 c1ccc(c(c1)C#N)O STR01814 C1C(=CC(=O)O1)O STR01860 c1ccc2c(c1)c(cc(=O)o2)O STR01861 c1c(c(cc(c1Cl)Cl)N)N STR01907 c1cc(cc(c1)[N+](=O)[O-])N STR01954 c1ccc2c(c1)c(=O)c(co2)C=O STR02001 c1cocc1CO STR02020 c1cc(ccc1CS)Cl STR02043 CCOC(=O)C(Cc1ccccc1)C(=O)C STR02085 Cc1cccc(c1)NN.Cl STR02094 COc1ccc(c(c1)[N+](=O)[O-])N STR02098 c1cc(sc1)I STR02125 c1c(cc(c(c1C(=O)O)N)Cl)Cl STR02151 Cc1cccc(c1C)O STR02184 c1ccc2c(c1)ccc(n2)C=O STR02188 Cc1[nH]ccn1 STR02220 C1CCC(=CC1)N2CCOCC2 STR02225 CCn1c2ccccc2c3c1ccc(c3)C=O STR02256 C1CC(OC1)CN STR02270 c1cc(ccc1NN)Br.Cl STR02278 CC(=O)CC(=O)c1ccc(cc1)Cl STR02310 CC1=CC(=O)CC1 STR02311 CC(C)(C)OC(=O)CBr STR02323 COc1cc(ccc1O)C(=O)O STR02334 Cc1ccccc1NN.Cl STR02353 CN1CCOCC1 STR02354 CN(C)c1cccc(c1)N.Cl.Cl STR02355 c1ccc(cc1)I STR02365 c1c(cc(cc1C(=O)O)O)C(=O)O STR02376 c1cc(ccc1C=O)C=O STR02396 C1CCC(=O)NCC1 STR02412 c1cc2c(cc1[N+](=O)[O-])scn2 STR02426 Cc1ccc(c(c1)N)N STR02446 c1cc(c(cc1Cl)[N+](=O)[O-])N STR02491 Cc1ccc2c(c1[N+](=O)[O-])cccn2 STR02499 COc1ccc(cc1)OC STR02500 CC(C)([C@H](C(=O)O)N)S STR02534 CNCc1ccccc1 STR02536 c1ccc2c(c1)C(=O)N(C2=O)CO STR02558 c1ccc(c(c1)c2[nH]c3ccccc3n2)N STR02578 C([C@@H](C(=O)O)N)S STR02584 Cc1ccc(o1)C=O STR02593 c1ccc2c(c1)C(=O)N(C2=O)CCCBr STR02619 COC(=O)c1ccc(cc1N)Cl STR02665 COc1ccc(c(c1)N)N STR02678 COc1ccc(cc1)C(=O)NN STR02684 c1(nnc(s1)S)N STR02713 CCC(c1ccccc1)O STR02714 c1ccc2c(c1)c(c[nH]2)C[C@@H](C(=O)O)N STR02722 CCCCc1ccc(cc1)Br STR02736 c1ccc(cc1)[C@H](CO)O STR02743 C(CO)CBr STR02760 c1ccc(cc1)C(c2ccccc2)C(=O)O STR02769 C1CCC(CC1)C(=O)O STR02844 c1ccc(cc1)c2ccc(cc2)C#N STR02867 CCCCc1ccc(cc1)c2ccccc2 STR02879 CN(C)C1CCCCC1 STR02891 c1cc(c(cc1O)[N+](=O)[O-])N STR02932 c1ccc(cc1)CN.Cl STR02952 C(C#N)C(=S)N STR02955 c1cc(c(cc1CC(=O)O)Cl)Cl STR02969 CC(=O)NC(=S)N STR02973 CC(=O)c1cccc(c1)N STR02986 C1C(=O)OC(=O)CS1 STR03033 C1CCCC(=O)CCC1 STR03048 CCc1ccc(cc1)C=O STR03104 CN(C)C(=O)N STR03134 c1cc(ccc1C(=O)N)Br STR03150 CN1CCCCC1 STR03153 c1ccc2c(c1)C(=O)CC2=O STR03163 CC(=O)c1ccc(cc1)C#N STR03197 COc1cc(cc(c1OC)OC)C=O STR03224 Cc1ccccc1C(=O)C STR03226 c1ccc(cc1)COC(=O)N STR03232 c1ccc2c(c1)CCCC2=O STR03237 c1cc(c(c(c1)[N+](=O)[O-])C(=O)O)C(=O)O STR03241 CC(=CC(=O)O)C STR03265 C1CCN(C1)CCN STR03276 CSc1ccccc1 STR03277 CCc1cccc(c1)Br STR03317 CC[C@@H](C(=O)O)N STR03331 CCC(=O)c1ccc(cc1)Cl STR03376 CCOC(=O)NN STR03390 c1ccc2c(c1)cccc2[N+](=O)[O-] STR03423 c1cc(ccc1[N+](=O)[O-])Br STR03424 CC(C)(C)CC(=O)O STR03445 Cc1cc(c(c(c1)Br)N)C(=O)O STR03467 c1cc(c(cc1[N+](=O)[O-])C(=O)O)N STR03468 c1ccc(c(c1)C=CC(=O)O)Cl STR03476 C(=C\C(=O)O)\C(=O)O STR03481 CNc1ccc(cc1)C(=O)O STR03499 c1ccc2c(c1)nccn2 STR03544 C1CCN(CC1)CCN STR03551 c1cc(c(c(c1)[N+](=O)[O-])N)[N+](=O)[O-] STR03602 c1c(c(cc(c1Cl)Cl)Cl)O STR03605 c1cc(c(cc1Cl)Br)O STR03609 c1cc(cc(c1)Br)Cl STR03612 c1c(ncnc1Cl)Cl STR03622 Cc1cccs1 STR03626 CCC(C)Br STR03634 CC(C)(C)C1CCC(CC1)O STR03673 c1cc(ccc1C#N)[N+](=O)[O-] STR03675 c1cc(c(c(c1)Cl)C#N)N STR03690 c1ccc(cc1)N2C(=O)C=CC2=O STR03760 c1ccc2c(c1)cccc2CN STR03771 c1cc2c(cc1N)C(=O)NC2=O STR03779 C1CC1C(=O)C2CC2 STR03807 COC(=O)c1ccccc1I STR03826 c1([nH]nc(n1)N)C(=O)O STR03830 Cc1cc(c(c(c1)C)Br)C STR03864 c1ccc(cc1)C(=O)c2ccc(c(c2)N)N STR03869 Cc1ccc(cn1)O STR03888 CCNC STR03903 CCOC(=O)Cc1cccs1 STR03971 COc1ccc2c(c1)c(ccn2)[C@H]([C@@H]3C[C@@H]4CCN3C[C@@H]4C=C)O STR03990 c1ccc2c(c1)c(cs2)CC#N STR04035 c1ccc(cc1)C2(c3ccccc3-c4c2cccc4)Br STR04110 C1COC(C(O1)O)O STR04115 CC(=O)c1ccc(cc1)C2CCCCC2 STR04122 c1c(c(=O)[nH]c(=O)[nH]1)[N+](=O)[O-] STR04133 CCOc1cc(ccc1OC)C=O STR04189 c1c(cc(c(c1Cl)N)Cl)Br STR04191 Cc1ccno1 STR04226 c1ccc2c(c1)C=Cc3ccccc3N2 STR04241 C1COC=C1 STR04249 c1ccc2c(c1)CCC2 STR04252 c1ccc2c(c1)c(ccc2Br)N STR04257 C1CCC(=O)C(=O)C1 STR04269 c1ccc(c(c1)CS)Br STR04271 c1cc(c(c(c1)Cl)N)C(=O)O STR04272 COc1cc(c(c(c1)OC)[N+](=O)[O-])OC STR04290 COC(=O)C1CCCC1=O STR04302 c1cnccn1 STR04325 Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C STR04334 c1nc2c(=O)[nH]c(nc2n1[C@H]3[C@@H]([C@@H]([C@H](O3)CO)O)O)N STR04471 Cc1cc(c(c(c1)O)C)C STR04504 CC1(C(=O)NC(=O)N1)C STR04524 c1ccc(cc1)OCCO STR04582 C(=S)(N)NC(=S)N STR04620 c1cc(ccc1O)Sc2ccc(cc2)O STR04624 C1CC(CC(C1)N)C(=O)O STR04646 c1cc(ccc1C(=N)N)Cl.Cl STR04649 c1cc(ccc1CCl)C(=O)O STR04662 C1C2CC3CC1CC(C2)(C3)N STR04703 C=C[C@H]1CN2CC[C@H]1C[C@H]2[C@@H](c3ccnc4c3cccc4)O STR04708 Cc1cccc(c1)CN STR04724 CC(=O)Nc1ccc(c(c1)C(=O)O)[N+](=O)[O-] STR04792 c1ccc(cc1)COC(=O)C(c2ccccc2)C(=O)O STR04796 CC1CCC(=O)C1=O STR04813 c1cc2c(c(c1)N)c(=O)[nH][nH]c2=O STR04818 c1cc(cc2c1ccc(=O)o2)O STR04824 c1cc(ccc1C=C(C#N)C#N)O STR04828 CC(=O)c1c(cccc1OC)O STR04840 COc1ccccc1C#N STR04854 c1ccc(cc1)C2=CCNCC2.Cl STR04870 C1C=CCN1 STR04876 c1c(c(cc2c1OCO2)[N+](=O)[O-])C=CC(=O)O STR04910 c1cc(c(cc1C(=O)O)O)[N+](=O)[O-] STR04954 c1ccc(cc1)COC(=O)CBr STR04959 Cc1cc(ccc1Cl)Cl STR04993 c1cc(c(cc1O)[N+](=O)[O-])Cl STR05013 COC1C=CC(O1)(CN)OC STR05014 c1ccc(cc1)C(c2ccccc2)O STR05017 c1cc(cc(c1)N)N.Cl.Cl STR05055 CNc1ccccc1C(=O)OC STR05066 c1ccc(cc1)c2c[nH]cn2 STR05069 COc1cccnc1Cl STR05101 COc1cc(c(cc1OC)[N+](=O)[O-])C=O STR05106 Cc1cc(=O)oc2c1cc(cc2)O STR05149 c1cc(c(nc1)C(=O)N)O STR05164 c1cnccc1C(=O)Cl.Cl STR05181 c1ccc(c(c1)CCO)[N+](=O)[O-] STR05203 c1cc(c(cc1C(=O)O)[N+](=O)[O-])[N+](=O)[O-] STR05213 CCC(C#N)c1ccccc1 STR05239 c1(c(c(=O)c1=O)O)O STR05257 Cc1ccc(cc1Br)C(=O)O STR05274 Cc1cc(ccc1[N+](=O)[O-])C(=O)O STR05311 Cn1c2ccccc2nc1N STR05341 COc1ccc(cc1)C(=O)CN.Cl STR05370 c1c(n[nH]c1O)N STR05383 COc1ccc(nn1)Cl STR05479 c1ccc2c(c1)c(=O)c3ccccc3o2 STR05546 Cc1c(c(=O)n(n1C)c2ccccc2)N STR05569 c1ccc2c(c1)nnn2CO STR05581 Cc1cc(cnc1)C#N STR05585 CCc1[nH]ccn1 STR05623 Cc1cn(c(=O)[nH]c1=O)[C@H]2C[C@@H]([C@H](O2)CO)O STR05630 c1ccc(cc1)c2[nH]ccn2 STR05632 COc1cc(cc(c1)OC)C=O STR05637 Cc1cccc(n1)C=O STR05660 c1ccc(cc1)CNC(=S)N STR05661 CC(=O)Nc1cccc(c1)N STR05687 CCOC(=O)CCCBr STR05803 COc1ccc(c(c1)C(=O)O)[N+](=O)[O-] STR05879 CNCc1cccc2c1cccc2.Cl STR05882 COCCBr STR05916 C#Cc1cccc(c1)N STR05978 c1c(cc(c(c1Br)N)Br)[N+](=O)[O-] STR06005 c1c(cc(cc1Cl)Cl)NN STR06028 CC(=O)Cc1ccccc1Cl STR06041 CC(=O)Cc1ccc(cc1)Cl STR06042 Cc1cc(n(n1)C)Cl STR06047 c1c(cnc(c1[N+](=O)[O-])N)Br STR06048 c1ccc(cc1)COc2ccccc2CC(=O)O STR06066 c1ccc(cc1)CON.Cl STR06086 CCc1ccccc1O STR06133 c1cc2c(cc1Cl)c(cs2)CC#N STR06146 c1ccc2c(c1)cn[nH]c2=O STR06150 c1c(csc1C=O)Br STR06172 CCOC(=O)N1[C@@H]2CC[C@H]1CC(=O)C2 STR06174 COc1cc(cc(c1)OC)O STR06179 CC(=O)c1ccc(cc1)c2ccc(cc2)Br STR06203 c1cc2cc(ccc2nc1)[N+](=O)[O-] STR06205 Cc1ccc(cc1C)O STR06236 c1cc(ccc1[N+](=O)[O-])I STR06257 c1c(cc(cc1C(=O)O)N)C(=O)O STR06298 Cc1c(cccc1Br)[N+](=O)[O-] STR06300 c1cc(c(c(c1)Cl)Cl)OCC(=O)O STR06337 COc1ccc(c(c1)OC)C=O STR06383 c1ccc(c(c1)CO)CO STR06426 c1ccc2c(c1)cccc2Br STR06472 C1CC(CCC1C(=O)O)N STR06482 C=CCSc1c(cccn1)C(=O)O STR06487 c1ccc(cc1)OCC#N STR06531 c1ccc(cc1)/C=C/C(=O)c2ccccc2 STR06550 c1ccc2c(c1)c(ccc2Br)Br STR06577 COC(=O)c1cscc1c2ccccc2 STR06588 C[C@H](c1cccc2c1cccc2)N STR06625 CC(=O)c1ccc(cc1)OCc2ccccc2 STR06633 c1cc(oc1C=O)Br STR06646 c1cc(c(nc1)Cl)C(=O)N STR06653 Cc1cc(ccc1Br)[N+](=O)[O-] STR06684 c1ccc(cc1)NCCO STR06691 CCC(=O)c1ccc(cc1)OCc2ccccc2 STR06699 COc1ccc(cc1C=O)Br STR06720 CC(C)(C)c1ccc(cc1)OC STR06745 c1ccc(cc1)C(=N)c2ccccc2 STR06747 c1ccc2c(c1)c(ccc2O)N.Cl STR06764 Cc1cccc2c1NC(=O)C2=O STR06774 CC1(CC(=O)CC(N1)(C)C)C STR06804 c1ccc(cc1)C(c2ccccc2)N3CC(C3)O STR06841 CC(C)(C)c1cc2c(s1)c(ncn2)Cl STR06850 Cc1csc2c1ncnc2Cl STR06851 Cc1ccc(c(c1)C)C(=O)C STR06914 Cc1cccc(c1Br)[N+](=O)[O-] STR06977 Cc1cc[nH]n1 STR06996 c1cc(ccc1NN)S(=O)(=O)O STR07041 B(c1ccc(c(c1)Cl)Cl)(O)O STR07093 CCOC(=O)c1cccc(c1)Br STR07102 COC(=O)c1ccccc1Br STR07133 Cc1cn(c(n1)Br)C STR07137 C1CN1 STR07159 c1ccc(c(c1)Cl)Br STR07176 CC(C)(C)c1ccc(cc1)Br STR07177 c1ccc2c(c1)nc(s2)CBr STR07213 c1ccc(cc1)c2c(nco2)CBr STR07214 c1ccc2c(c1)ccc(n2)Cl STR07222 Cc1nc(cs1)C(=S)N STR07268 CC(C)(C)C(=O)OCC(=S)N STR07269 c1cnn(c1)C(=N)N.Cl STR07295 COc1ccccc1I STR07301 c1ccc2c(c1)c(cs2)CO STR07371 COc1cc(cc(c1)OC)C(=O)OC STR07374 c1c(cnc2c1c(c[nH]2)I)Br STR07406 c1cc(oc1)C(=O)CC#N STR07414 C1CCC(C1)O STR07441 Cn1c(=O)c(c(cn1)Cl)Cl STR07454 CC1(Cc2c(sc(c2C(=O)C1)SC)C#N)C STR07502 CCCc1ccccc1N STR07512 COc1ccnc(n1)Cl STR07516 Cc1cc(no1)C(=S)N STR07527 c1ccc2c(c1)cc(o2)CO STR07538 Cc1ccnc(c1)C STR07571 c1ccc(cc1)c2nc(no2)CCl STR07631 c1ccc(cc1)c2nc(on2)CCl STR07632 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)CCl STR07663 C1CC(=O)CC1=O STR07692 Cc1cccc(c1)I STR07696 c1ccc(cc1)S(=O)(=O)O STR07703 CC(C)(C)[C@@H](C(=O)O)N STR07808 c1cc(c(c(c1)Cl)Cl)/C=C/C(=O)O STR07856 c1ccc(cc1)C(=O)c2cc(ccc2O)Br STR07864 C1CCC(CC1)C#N STR07874 COC(=O)C1=CCCC1 STR07915 c1ccc(cc1)Oc2cccc(c2)O STR07918 c1ccc2c(c1)CC[C@@H]2N STR07992 c1ccc(cc1)c2ccc(cc2)CN STR08023 c1ccc(cc1)CCCCCC(=O)O STR08043 C1C(CN1)O STR08059 c1ccc2c(c1)CCC[C@@H]2N STR08071 c1ccc(cc1)[C@H](C(=O)O)O STR08136 c1ccnc(c1)CCO STR08146 CC(C)C(=O)C1CCCCC1=O STR08161 CC(C)c1ccc(cc1)O STR08167 CC(C)(C)OC(=O)N1CC(=O)O[C@@H]([C@@H]1c2ccccc2)c3ccccc3 STR08272 COc1cc(ccc1I)[N+](=O)[O-] STR08281 CCOC(=O)CCN1CCNCC1 STR08341 c1ccc(cc1)CON STR08364 c1cc(c(cc1CBr)Cl)Cl STR08450 CNc1ccncc1 STR08498 c1ccc2c(c1)c(ccn2)Cl STR08502 CNc1ccccc1[N+](=O)[O-] STR08505 Cc1cc(c(cc1C)[N+](=O)[O-])N STR08532 C1CC(CCC1O)O STR08594 COc1ccc(cc1)I STR08687 c1cc(c(c(c1)O)O)O STR08708 CNC(=O)c1cc(cc(c1)Br)[N+](=O)[O-] STR08721 C1CCOC(=O)C1 STR08736 c1cc(c(cc1N)[N+](=O)[O-])N STR08741 CC1CCCO1 STR08776 c1cc(c(cc1O)[N+](=O)[O-])NCCO STR08779 c1[nH]c2c(n1)ncnc2Br STR08792 CCOC(=O)c1c(cccc1Cl)Cl STR08820 CCOC(=O)C(=S)N STR08851 c1cnoc1 STR08895 COc1cc(c(cc1OC)[N+](=O)[O-])[N+](=O)[O-] STR08903 CC(C)(C)OC(=O)NCC1CNC1 STR08904 c1ccc(c(c1)S(=O)(=O)N)Cl STR08928 C1C(=O)CO1 STR08949 Cc1ccc(c(c1)C)C#N STR08989 COc1ccc(c(c1)C(=O)OC)Br STR09008 Cc1cccc(c1O)O STR09012 COC(=O)c1ccccc1S(=O)(=O)N STR09073 c1nnc(s1)S STR09095 COc1cc(cc(c1O)OC)C=O STR09162 C1CCNCC1.Cl STR09186 Cc1ccc(cc1)C(=O)c2ccc(cc2)C STR09191 CC(C)(C)c1ccccc1 STR09192 c1ccc(c(c1)Br)I STR09197 B(c1ccc2cc[nH]c2c1)(O)O STR09340 Cc1cccc(c1)OC STR09347 c1c(c(c(cn1)Cl)N)Cl STR09436 C1COCC(=O)N1 STR09474 c1c(cc(cc1N)Br)C(=O)O STR09568 COc1cc(nc(n1)C(=O)O)OC STR09587 Cc1ccc(cc1C)NN.Cl STR09614 C1C[C@H](CNC1)O.Cl STR09634 C1C[C@@H](CNC1)O.Cl STR09635 C#Cc1ccc(cc1)C#C STR09668 CC1CCCCC1O STR09785 c1cncc(c1Cl)S(=O)(=O)N STR09801 Cc1cc(cc(c1)I)C STR09819 C#CCCO STR09821 COC(=O)[C@@H]1CCCC[C@H]1C(=O)O STR09867 B(/C=C/c1ccccc1)(O)O STR09885 B(c1cccc(c1)N(C)C)(O)O STR09904 B(c1ccnc(c1)C)(O)O STR09910 B(c1cccc(c1)C(=O)NC2CC2)(O)O STR09927 c1ccc2c(c1)nc(s2)C=O STR10004 CNCc1ccc(cc1)c2ccn(n2)C STR10013 c1[nH]nc(n1)C(=O)O TS-00001 c1nc(no1)C(=O)O TS-00002 c1cnnc(n1)C(=O)O TS-00003 c1cnc(c(c1O)N)O TS-00004 Cc1nc(nc(n1)O)N TS-00005 Cn1c(ncn1)C(=O)O TS-00008 c1nnnn1CC(=O)N TS-00009 Cc1c(nno1)C(=O)O TS-00010 C1C(=NNC1=O)C(=O)O TS-00011 c1c(nc(o1)N)C(=O)O TS-00012 Cc1nc(no1)C(=O)O TS-00013 c1nnnn1CC(=O)O TS-00014 c1csc(n1)C(=O)N TS-00015 c1c(ncs1)C(=O)N TS-00016 C1CN[C@@H](CN1)C(=O)N TS-00017 C1CN[C@@H](CN1)C(=O)O TS-00018 c1c(sc(n1)N)CO TS-00019 CSc1[nH]nc(n1)N TS-00020 COc1nc(sn1)N TS-00021 C(#N)c1c(nc([nH]1)N)C#N TS-00022 c1c2c(nc[nH]2)nc(n1)N TS-00023 c1c2c(ncnc2[nH]n1)N TS-00024 c1cc2nncn2nc1N TS-00025 c1cnc2c(n1)c(n[nH]2)N TS-00026 c1[nH]c(c(n1)C(=O)N)C#N TS-00027 c1c2c([nH]n1)nc[nH]c2=O TS-00028 c1c2c([nH]c(=O)[nH]2)ncn1 TS-00029 c1nc(c2c(n1)[nH]nn2)N TS-00030 c1c(c(nc(n1)O)O)C#N TS-00031 c1nc2c(c(n1)O)nn[nH]2 TS-00032 c1cc(ncc1C(=O)N)N TS-00033 c1cc(c(nc1)N)C(=O)N TS-00034 c1c(cncc1N)C(=O)N TS-00035 c1cnc(c(n1)C(=O)N)N TS-00036 c1cc(nnc1C(=O)O)N TS-00037 c1cnnc(c1C(=O)O)N TS-00038 c1cc(=O)[nH]nc1C(=O)N TS-00039 c1c(ncc(n1)O)C(=O)O TS-00040 c1cnc(c(n1)C(=O)O)O TS-00041 Cn1c(ncn1)C(=O)OC TS-00042 CN1C(=O)CC(=N1)C(=O)O TS-00043 COc1c(ncnc1O)O TS-00044 COC(=O)Cn1cnnn1 TS-00045 COC(=O)c1cc(no1)O TS-00046 C1(C(=O)NC(=O)NC1=O)N TS-00047 c1csc(c1C(=O)O)N TS-00048 c1c(nc(s1)N)C(=O)N TS-00050 c1c(nc(s1)N)C(=O)O TS-00051 C1CN[C@H](CN1)CC(=O)O TS-00052 COC(=O)[C@@H]1COC(=O)N1 TS-00053 COCc1nc(sn1)N TS-00054 c1ccnc(c1)c2[nH]nnn2 TS-00055 C(C#N)c1c(c(n[nH]1)N)C#N TS-00056 CSc1nc(ns1)N TS-00057 Cn1cnc2c1c(ncn2)N TS-00058 Cn1cnc2c1nc[nH]c2=O TS-00059 c1[nH]c2c(n1)c(nc(n2)N)N TS-00060 c1c[nH]c2c1c(nc(n2)O)O TS-00061 c1cc(oc1)c2nnc(o2)N TS-00062 c1c[nH]n2c1nc(c2)C(=O)O TS-00063 c1c[nH]c2c1[nH]c(=O)[nH]c2=O TS-00064 c1con2c1nc(c2)C(=O)O TS-00065 c1csc(n1)C(=O)CC#N TS-00066 Cc1ncc(c(n1)N)C(=O)O TS-00067 COC(=O)c1cncnc1N TS-00068 CCOC(=O)c1nccnn1 TS-00069 CNCc1cc(ccc1O)O TS-00070 COC(=O)c1ccc(=O)[nH]n1 TS-00071 Cc1nc(nc(n1)OC)NC TS-00072 CCCCc1[nH]c(cn1)CO TS-00073 COc1cc(nc(n1)OC)N TS-00075 COc1c(c(ncn1)OC)N TS-00076 CCOC(=O)c1c[nH]nc1N TS-00077 c1c([nH]c(=O)[nH]c1=O)C(=O)O TS-00078 c1[nH]c(c(n1)C(=O)O)C(=O)O TS-00079 CCOC(=O)c1c(onn1)C TS-00080 CCOC(=O)C1=NNC(=O)C1 TS-00081 COC(=O)C1=NNC(=O)CC1 TS-00082 CCOC(=O)c1cn[nH]c1O TS-00083 CCOC(=O)c1nnc(o1)C TS-00084 COCc1nc(cc(n1)O)O TS-00085 COc1nc(nc(n1)OC)N TS-00086 Cc1csc(c1C(=O)N)N TS-00087 Cc1cc(c(s1)N)C(=O)N TS-00088 Cc1csc(n1)CC(=O)N TS-00089 COC(=O)c1cc(on1)CO TS-00090 CC(=O)Oc1c(ccs1)N TS-00092 Cc1csc(c1C(=O)O)N TS-00093 Cc1cc(c(s1)N)C(=O)O TS-00094 COc1ccsc1C(=O)N TS-00095 C1CNC(=O)[C@@H](N1)CC(=O)O TS-00096 Cc1c(nc(s1)N)C(=O)O TS-00099 Cc1c(snn1)C(=O)OC TS-00100 c1cnn2c1ncc(c2N)C#N TS-00101 C1C(=O)N=C(S1)CC(=O)O TS-00102 c1cc(c2cc[nH]c2c1)C(=N)N TS-00103 CC(C)(C)c1cccc(c1)C#N TS-00104 C1CC(OC1C(=O)O)C(=O)O TS-00105 c1cc(cc(c1)N)c2[nH]nnn2 TS-00106 c1cnccc1CNCCC#N TS-00107 C1CSCCC1(C(=O)O)N TS-00108 c1cc2c(cc1C(=O)N)nn[nH]2 TS-00109 c1cnccc1c2nc(no2)N TS-00110 c1cc2c(cc1C(=O)O)nn[nH]2 TS-00111 c1cnc2c(cnn2c1)C(=O)O TS-00112 c1cn2cc(nc2cn1)C(=O)O TS-00113 c1cncn2c1nc(c2)C(=O)O TS-00114 c1cnn2c1nc(cc2)C(=O)O TS-00115 c1cnc2ncc(n2c1)C(=O)O TS-00116 c1cnc(cn1)c2nc(no2)N TS-00117 c1cnc2c(n1)c(nc(n2)N)O TS-00118 C1[C@H](NC(=S)S1)C(=O)O TS-00120 c1cc2c(cc1C(=O)O)non2 TS-00121 COCc1ncc(c(n1)N)C#N TS-00122 CN(CCCN)c1ccccc1 TS-00123 CC(=O)NC(=O)c1cnccn1 TS-00125 CC(=O)c1cnc(cn1)C(=O)N TS-00126 COc1c2c([nH]cn2)nc(n1)N TS-00127 c1ccc(cc1)CNCC(=O)O TS-00128 c1cc2c(cc1N)nc(s2)N TS-00129 c1cc(sc1)c2cc(n[nH]2)N TS-00130 CNCCc1ccc(cc1)OC TS-00131 CNCCc1ccccc1OC TS-00132 CNCCc1cccc(c1)OC TS-00133 CNCC[C@@H](c1ccccc1)O TS-00134 c1c(ncc(n1)C(=O)N)C(=O)N TS-00135 CC(=O)Nc1c(ccs1)C#N TS-00136 CCCOc1ccc(cc1)CO TS-00137 c1cnc(c(n1)C(=O)N)C(=O)O TS-00138 Cc1cc(c(cc1O)C(=O)O)N TS-00139 CCOC(=O)c1cnc(nc1)N TS-00140 CCOC(=O)c1cncnc1N TS-00141 c1csc2c1[nH]c(c2)C(=O)O TS-00142 C1[C@H](CN[C@@H]1C(=O)O)O.Cl TS-00143 c1c(nc(cn1)C(=O)O)C(=O)O TS-00144 c1c(ncc(n1)C(=O)O)C(=O)O TS-00145 CCOC(=O)c1ccc(=O)[nH]n1 TS-00146 COc1c(c(ccn1)C(=O)O)N TS-00147 c1csc2c1c(=O)[nH]c(=O)[nH]2 TS-00149 C1COCCN1c2nnc(o2)N TS-00150 c1(c(nc([nH]1)N)C(=O)O)C(=O)O TS-00151 C1CC(=O)N(C1)CCCC(=O)O TS-00152 CN(C)CCCN1CCNCC1 TS-00156 c1c(cnc(c1N)C(=O)N)Cl TS-00157 c1cnc(c(c1C(=O)N)N)Cl TS-00159 c1cc(nc(c1N)C(=O)N)Cl TS-00160 CCOC(=O)CC1CCOCC1 TS-00161 CCOC(=O)[C@@H](C)C1(CCC1)O TS-00162 Cc1ccc(n1c2ccccn2)C TS-00163 CC(=O)N1C[C@@H](C[C@H]1C(=O)O)O TS-00164 c1ccc(c(c1)N)S(=O)(=O)O TS-00165 COCc1nc(cs1)C(=O)O TS-00166 c1cc(ccc1O)S(=O)(=O)N TS-00167 c1cncc(c1N)S(=O)(=O)N TS-00168 c1c(cncc1S(=O)(=O)O)N TS-00169 CSc1ccc(s1)C(=O)O TS-00170 Cc1cc(sc1)c2ccccc2 TS-00171 c1cnc2c(n1)cc(cn2)C(=O)O TS-00172 c1cc2c(nc1)ncc(n2)C(=O)O TS-00173 c1cc(ccc1Cc2[nH]nnn2)N TS-00174 c1cc2c(cc1N)sc(n2)C#N TS-00175 Cc1c(n2cccnc2n1)C(=O)O TS-00176 Cc1cncc2n1cc(n2)C(=O)O TS-00177 c1cc(c2nc(cn2c1)C(=O)O)N TS-00178 Cc1cc(cc(c1N)C)C(C)(C)C TS-00179 CC(C)c1ccc(cc1)CCNC TS-00180 Cc1cc2ccccc2nc1Cl TS-00181 C1CCC(CC1)NC(=N)N.Cl TS-00182 c1cc2c(cc1C(=O)O)[nH]c(=O)[nH]2 TS-00183 Cc1cc(cc(c1)C(=O)N)C(=O)N TS-00184 c1cc(ccc1CCNCC#N)F TS-00185 CCCCc1ccc(cc1)C(=O)O TS-00187 C[C@@H](C(=O)C)OCc1ccccc1 TS-00189 c1cc(oc1)c2c(nco2)C(=O)O TS-00190 c1cc(oc1)c2cc(no2)C(=O)O TS-00191 COC(=O)CCNc1ccccc1 TS-00192 COC(=O)CNCc1ccccc1 TS-00193 CC(C)(C)c1ccc([nH]1)C(C)(C)C TS-00194 c1cocc1c2nc(no2)C(=O)O TS-00195 c1cc(c(cc1O)O)/C=C/C(=O)O TS-00196 c1cc(c(cc1O)/C=C/C(=O)O)O TS-00197 c1cc2c(nc1)NC[C@H](O2)C(=O)O TS-00198 c1cc(ccc1CCCC(=O)O)O TS-00199 CCOC(=O)Cc1cccc(n1)N TS-00200 COC(=O)c1cccc(n1)CCN TS-00201 COC(=O)c1c(cccn1)C(=O)O TS-00202 COC(=O)c1cccc(n1)C(=O)O TS-00203 c1cc(c(cc1CCC(=O)O)N)O TS-00204 CCOC(=O)c1cccc(n1)CO TS-00205 COc1ccccc1OCC(=O)N TS-00206 CCOC(=O)c1cnc(nc1C)N TS-00207 CCOC(=O)c1cnc(nc1N)C TS-00208 COc1ccc2c(n1)sc(n2)N TS-00209 CNCc1c(cccc1OC)OC TS-00210 c1conc1N2CC[C@@H](C2)C(=O)O TS-00211 c1cc(ccc1CCCC(=O)O)F TS-00212 c1ccc(c(c1)C#N)S(=O)(=O)N TS-00214 CCCc1c(c(n(n1)C)C(=O)N)N TS-00215 COc1cc(ccc1Cl)C2CC2 TS-00216 COc1ccc(c(n1)OC)C(=O)O TS-00217 COc1cc(cc(n1)OC)C(=O)O TS-00218 CCOC(=O)c1cnc(nc1O)N TS-00219 Cc1nn2cc(nc2s1)C(=O)O TS-00220 COC(=O)c1ccc(o1)C(=O)OC TS-00221 c1cc(sc1)C(=O)CCC(=O)O TS-00222 CCOC(=O)C[C@H]1CCCCC1=O TS-00223 Cc1ccc(cc1)c2ccc(cc2)O TS-00224 c1cc(nc(c1N)C#N)n2ccnc2 TS-00226 CCCCN1C[C@H](CC1=O)C(=O)O TS-00227 CCOC(=O)CC1CCN(CC1)C TS-00229 CCOC(=O)[C@@H](C)C1CCNCC1 TS-00230 Cc1cc(cc(c1C#N)Cl)Cl TS-00231 Cc1cc(ccc1N)S(=O)(=O)N TS-00232 c1cc2nc(cn2cc1C#N)C(=O)O TS-00233 Cc1c(sc(n1)COC)C(=O)O TS-00234 c1cc(ncc1C(=O)N)n2ccnc2 TS-00235 C1C[C@@H](C(=O)C1)SCCC(=O)O TS-00236 CCC[C@H]1CCc2ccccc2C1=O TS-00237 CCCCc1[nH]c(c(n1)CO)Cl TS-00238 c1cnccc1c2cc(n[nH]2)C(=O)O TS-00239 c1cc(nc(c1)n2ccnc2)C(=O)O TS-00240 c1cc(c(nc1)n2ccnc2)C(=O)O TS-00241 c1cnc(cc1C(=O)O)n2ccnc2 TS-00242 c1ccc2c(c1)nc(c(n2)O)C(=O)O TS-00243 c1cnccc1c2c(nco2)C(=O)O TS-00244 c1cc(cnc1)c2c(nco2)C(=O)O TS-00245 c1ccc(cc1)c2nnc(o2)C(=O)O TS-00246 c1cnc(c(n1)C(=O)O)n2ccnc2 TS-00247 c1cc(nnc1C(=O)O)n2ccnc2 TS-00248 c1cnc(c(n1)C#N)N2CCOCC2 TS-00249 c1cnc(cn1)c2c(nco2)C(=O)O TS-00250 c1cnccc1c2nc(no2)C(=O)O TS-00251 c1cc(cnc1)c2nc(no2)C(=O)O TS-00252 CCOC(=O)c1cnc2n1cccn2 TS-00253 Cc1cc(n2cc(nc2n1)C(=O)O)C TS-00254 Cc1cc2ncc(c(n2n1)C)C(=O)O TS-00255 Cc1c(nc2c(n1)c(nc(n2)N)O)C TS-00256 CC(=O)Nc1ccc(cc1)OCC=C TS-00257 Cc1cc2nnc(c(n2n1)C)C(=O)O TS-00258 c1csc(c1[S@](=O)O)C(=O)O TS-00259 CCCCc1ccc(cc1)C(=O)OC TS-00260 CCC(C)C(c1ccccc1)C(=O)O TS-00261 CC(C)(C)c1cccc(c1)C(=O)OC TS-00262 CCc1ccc(cc1)CCCC(=O)O TS-00263 CCOC(=O)C(C)(C)c1ccccc1 TS-00264 c1cc2c(cc1C(=O)O)NC(=O)CO2 TS-00265 COC(=O)c1c(c2c(o1)nccn2)N TS-00266 c1nc(c2c(n1)n(cn2)CC(=O)O)N.Cl.Cl TS-00267 CC(=O)Nc1[nH]c(=O)c2c(n1)[nH]cn2 TS-00268 c1cc(cc(c1)SC(F)(F)F)N TS-00269 c1cnc(cc1C(=O)O)OCC2CC2 TS-00270 c1cc(ncc1C(=O)O)OCC2CC2 TS-00271 c1cc(nc(c1)OCC2CC2)C(=O)O TS-00272 c1cc2c(cc1O)C[C@H](NC2)C(=O)O TS-00273 c1cc(cc(c1)O)C2CC2(C(=O)O)N TS-00274 c1cnc(c(n1)C(=O)O)N2CCCC2 TS-00275 C1CS(=O)(=O)C[C@H]1NCC(=O)O TS-00276 c1cscc1c2c[nH]cc2C(=O)O TS-00277 COC(=O)CCc1ccc(cc1)CN TS-00278 COC(=O)CCNCc1ccccc1 TS-00279 CC[C@H](C)NCc1ccccc1OC TS-00280 CC(=O)Nc1cc(ccn1)C(=O)OC TS-00281 CCOC(=O)/C=C/c1cccc(c1)F TS-00282 c1ccc2c(c1)c(c(s2)C(=O)O)O TS-00283 c1cc(sc1)c2cc(n[nH]2)C(=O)O TS-00284 c1cc(sc1c2c[nH]nc2)C(=O)O TS-00285 c1cc(sc1c2c[nH]cn2)C(=O)O TS-00286 COC(=O)c1ccc2c(c1)nsn2 TS-00287 c1cc(ccc1Nc2nnns2)O TS-00288 CCCCOc1ccc(cc1)C(=O)O TS-00289 COc1ccc(cc1)CCCC(=O)O TS-00290 COc1ccccc1CCNC(=O)N TS-00291 c1ccc(c(c1)C(=O)N)OCC(=O)O TS-00292 COC(=O)c1ccc(c(c1)N)C(=O)O TS-00293 c1ccc(cc1)C(=O)N[C@H](C(=O)O)O TS-00294 c1cc(sc1)c2c(nco2)C(=O)O TS-00295 c1cc(oc1)c2c(ncs2)C(=O)O TS-00296 c1cc(oc1)c2nc(cs2)C(=O)O TS-00297 COC(=O)C[C@@H](c1ccc(cc1)O)N TS-00298 COC(=O)C[C@@H](c1cccc(c1)O)N TS-00299 CCOC(=O)c1cn2c(n1)CNCC2 TS-00300 CCOc1cc(ccc1OC)CNC TS-00301 c1cn(cn1)c2c(c(ncn2)Cl)N TS-00302 COc1ccc(c(c1)C(=O)O)C(=O)O TS-00303 COC(=O)Oc1ccc(cc1)C(=O)O TS-00304 COC(=O)c1ccc(c(c1)O)C(=O)O TS-00305 Cc1cc(no1)NC(=O)/C=C/C(=O)O TS-00306 c1conc1N2C[C@H](CC2=O)C(=O)O TS-00307 COC(=O)c1cnc(cn1)C(=O)OC TS-00308 COc1cccc(c1OC)C(=O)OC TS-00309 COC(=O)C[C@@H](c1cccc(c1)O)O TS-00310 CC(C)(C)OC(=O)c1ccc(=O)[nH]n1 TS-00311 CCOc1cc(cc(c1)OCC)CO TS-00312 c1cc2c(cc1Br)CCC2 TS-00313 c1ccn2c(c1)ncc2S(=O)(=O)N TS-00314 CCOC(=O)CCNCc1ccco1 TS-00315 COc1ccc(c(c1)[C@H](CN)O)OC TS-00317 CCOC(=O)c1nc(cs1)C2CC2 TS-00318 CCCSc1c(cccn1)C(=O)O TS-00319 c1cc(nn2c1ncc2C(=O)O)Cl TS-00320 c1c(c(cc(c1O)C(=O)O)O)C(=O)O TS-00321 CCCc1[nH]c(c(n1)C(=O)O)C(=O)O TS-00322 Cc1c(c(no1)C(=O)OC)/C(=N/O)/C TS-00323 c1ccc2c(c1)[nH]c(n2)S(=O)(=O)O TS-00324 c1ccn2c(c1)ncc2S(=O)(=O)O TS-00325 CC(C)(C)OC(=O)C1=NNC(=O)CC1 TS-00326 c1ccc(cc1)CNCc2ccncc2 TS-00327 CS(=O)(=O)c1ccc(cc1)C(=O)N TS-00328 CCCCN1C[C@H](CC1=O)C(=O)OC TS-00329 CC(C)(C)c1ccccc1n2cccc2 TS-00330 c1ccc2c(c1)c3c([nH]2)CCCCCC3 TS-00331 CNCCC(=O)c1ccccc1.Cl TS-00332 CCOC(=O)Cc1cc(ccc1F)F TS-00333 CNS(=O)(=O)Cc1ccc(cc1)N TS-00334 CC(=O)N1CCC(CC1)NCCOC TS-00335 c1cc(ccc1OCCC(=O)O)Cl TS-00336 c1cc(cc(c1)C(=O)O)C(=N)N.Cl TS-00337 c1ccc(c(c1)C(=O)O)S(=O)(=O)N TS-00338 CC(COC)N1CC(CC1=O)C(=O)O TS-00339 CCOC(=O)c1csc(n1)COC TS-00340 Cc1[nH]cc(n1)CNCc2ccccc2 TS-00341 COC(=O)c1cc(c(nc1N)N)Cl TS-00342 COc1ccc(cc1)NC(=N)N.Cl TS-00343 COC(=O)c1ccccc1OC(F)F TS-00344 c1c(n2c(n1)CCCC2)S(=O)(=O)O TS-00345 Cc1cc(cc(c1F)C)Br TS-00346 C1CNC(CN1)C(=O)O.Cl.Cl TS-00347 c1cc(cc(c1)SC(F)(F)F)C#N TS-00348 Cc1c(nn(n1)c2ccccc2)C(=O)O TS-00349 c1ccc(cc1)c2c(nc(nc2O)N)O TS-00350 c1cc(ccc1Cn2cncn2)C(=O)O TS-00351 Cc1c(nnn1c2ccccc2)C(=O)O TS-00352 COC(=O)[C@@H]1CSCC(=N1)C(=O)O TS-00353 CCOC(=O)Cc1cc2ccccc2[nH]1 TS-00354 CN1CCN(CC1)c2c(nccn2)C#N TS-00355 Cc1c(c(n(n1)C)C)NS(=O)(=O)C TS-00356 COC(=O)CSc1c(ccs1)N TS-00357 c1ccc(cc1)Cc2nc(on2)C(=O)O TS-00358 c1cc(nc(c1N)C#N)N2CCOCC2 TS-00359 c1ccnc(c1)c2ccc(s2)C(=O)N TS-00360 c1ccc(cc1)CCCN2CCNCC2 TS-00361 c1ccnc(c1)c2nnn(n2)CC(=O)O TS-00362 CCOC(=O)c1cn2cccc(c2n1)N TS-00363 CCCCc1ccc(c(c1)C)NC(=O)C TS-00364 Cc1cc(nc(c1)C(C)(C)C)C(C)(C)C TS-00365 c1ccc2c(c1)c(c(o2)C(=O)O)C(=O)O TS-00366 c1cc(cnc1)N2C[C@H](CC2=O)C(=O)O TS-00368 CCOC(=O)c1c(c2cccnc2o1)N TS-00369 c1cc(sc1c2cncnc2)C(=O)O TS-00370 c1cnc(nc1)c2ccc(s2)C(=O)O TS-00371 c1cc(cnc1)c2csc(n2)C(=O)O TS-00373 c1ccnc(c1)c2nc(cs2)C(=O)O TS-00374 c1cc(cnc1)c2c(ncs2)C(=O)O TS-00375 CCc1ccc(cc1)C(=O)CCC(=O)O TS-00376 c1ccc(cc1)C(=O)CCCCC(=O)O TS-00377 CCOC(=O)[C@@H](C)C(=O)c1ccccc1 TS-00378 Cc1cc(cc(c1C(=O)O)C)C(C)(C)C TS-00379 CCCc1ccc(cc1)CCCC(=O)O TS-00380 CCOC(=O)c1cc(on1)c2ccco2 TS-00381 c1cnc(nc1)N2C[C@H](CC2=O)C(=O)O TS-00382 c1cnc(cn1)N2C[C@H](CC2=O)C(=O)O TS-00383 Cc1ccc(cc1N)SC(F)(F)F TS-00384 c1cc(cc(c1)SC(F)(F)F)CN TS-00385 CC(C)OC(=O)c1c(cccn1)C(=O)C TS-00386 c1cnc(cc1C(=O)O)OCC2CCC2 TS-00387 c1cc(ncc1C(=O)O)OCC2CCC2 TS-00388 c1cc(nc(c1)OCC2CCC2)C(=O)O TS-00389 c1cc(c(nc1)OCC2CCC2)C(=O)O TS-00390 CC(=O)N[C@@H](Cc1ccccc1)C(=O)O TS-00391 c1cc(c(nc1)N2CCNCC2)C(=O)O TS-00392 c1cnc(cc1C(=O)O)N2CCNCC2 TS-00393 c1c(nc(cn1)N2CCCCC2)C(=O)O TS-00394 COc1ccc(cc1)c2nnc(s2)N TS-00395 C1CNCCC1CCCC(=O)O.Cl TS-00396 CCOC(=O)c1nc(on1)c2ccoc2 TS-00398 c1ccc(cc1)COCC(=O)CC(=O)O TS-00399 Cc1cc(cc(c1)C(=O)OC)C(=O)OC TS-00400 CC(=O)c1c(cc(cc1O)OCC=C)O TS-00401 c1cnc(cc1N2CCOCC2)C(=O)O TS-00402 Cn1ccnc1c2ccc(s2)C(=O)O TS-00403 CC(=O)Nc1cccc(c1)OCCCN TS-00404 Cn1c2ccccc2nc1c3ccccc3 TS-00405 CCC(C)(C)c1ccc(cc1)OCCO TS-00406 CNCc1ccc(cc1)OCCN(C)C TS-00407 COC(=O)[C@@H]1CCn2c1c(cc2)C(=O)O TS-00408 C=CCOc1nc(nc(n1)OCC=C)O TS-00409 c1c(nc(cn1)N2CCOCC2)C(=O)O TS-00410 c1c(cnc(n1)N2CCOCC2)C(=O)O TS-00411 c1cnc(c(n1)C#N)SCCC(=O)O TS-00412 c1ccc(cc1)Oc2cccc(c2)CC#N TS-00413 c1cnc([nH]1)CN2CCC(CC2)C(=O)O TS-00414 c1c(nc[nH]1)CN2CCC(CC2)C(=O)O TS-00415 CN(C)CCCOc1ccc(cc1)CO TS-00416 c1ccc(c(c1)[C@@H](CC(=O)O)C(=O)O)O TS-00419 CCOC(=O)c1ccc(c(c1)O)C(=O)O TS-00420 COC(=O)CC(=O)Cc1ccccc1F TS-00421 c1cc(oc1)c2c(nc(s2)N)C(=O)O TS-00422 Cc1c(cc(cc1OC)C(=O)OC)OC TS-00423 CCOc1cccc(c1C(=O)O)OCC TS-00424 COc1ccc(cc1OC)CC(=O)OC TS-00425 Cc1ccc(c(c1)C)C(=O)c2ccccc2 TS-00426 Cc1c(c(n(n1)C)Cl)S(=O)(=O)O TS-00427 CNCc1cc(c(c(c1)OC)OC)OC TS-00428 c1cc(sc1c2nccs2)C(=O)O TS-00429 Cc1c(n2c(n1)ccc(n2)Cl)C(=O)O TS-00430 c1(c(sc(n1)N)C(F)(F)F)C(=O)O TS-00431 CCOC(=O)c1ccc(o1)C(=O)OCC TS-00432 CCOC(=O)c1ccc(o1)COC(=O)C TS-00433 CCCc1nc(c(n1C)C(=O)O)C(=O)O TS-00434 c1csc(n1)N2C[C@H](CC2=O)C(=O)O TS-00435 c1ccc(cc1)CCc2ccccc2CO TS-00436 c1ccc(cc1)COc2ccc(cc2)CN TS-00437 COC(=O)c1cc(c(s1)SC)C#N TS-00438 CC[C@H]1CCCCN1C(=O)OC(C)(C)C TS-00439 CC(C)N(CCN1CCNCC1)C(C)C TS-00440 CCOC(=O)[C@@H](c1ccccc1Cl)N TS-00441 c1cc(c(cc1F)C(=O)O)OCC(=O)O TS-00442 COC(=O)CC(=O)c1ccc(cc1F)F TS-00443 c1ccc(cc1)S(=O)(=O)CCC(=O)O TS-00444 COc1ccc(cc1)CNc2ccccn2 TS-00445 CC(C)(C)OC(=O)N1CC[C@@H](C1)CNC TS-00446 COC(=O)CCc1ccc(c(c1)Cl)O TS-00447 CCOC(=O)C(c1c(cccn1)C)(F)F TS-00448 CCOC(=O)C(c1ccc(cn1)C)(F)F TS-00449 CCOC(=O)C(c1cccc(n1)C)(F)F TS-00450 c1cc2cccc(c2c(c1)C(=O)N)C(=O)O TS-00452 c1cc(ccc1c2cnc(nc2)N)C(=O)O TS-00455 c1cc(cc(c1)C(=O)O)c2cnc(nc2)N TS-00456 c1cc(cc(c1)C(=O)O)c2ccnc(n2)N TS-00457 c1cc2c(cc1S(=O)(=O)N)OCCO2 TS-00459 COC(=O)c1ccc(cc1)S(=O)(=O)N TS-00460 CC(COC)N1CC(CC1=O)C(=O)OC TS-00461 CCOC(=O)c1c(nc(s1)COC)C TS-00463 c1c(c(c(cn1)Br)C(=O)N)N TS-00464 COC(=O)c1ccccc1Cn2ccnc2 TS-00465 COC(=O)c1cccc(c1)Cn2cccn2 TS-00466 C[C@@H](c1ccc(c(c1)F)c2ccccc2)O TS-00467 CC(C)(C)OC(=O)N1CCN[C@H](C1)CO TS-00468 Cc1c(cc(s1)c2ccccc2)C(=O)C TS-00469 c1ccc(cc1)c2cnc(o2)CCC(=O)O TS-00470 CCOC(=O)c1coc(n1)c2ccccc2 TS-00471 Cc1c(nnn1Cc2ccccc2)C(=O)O TS-00472 c1ccc2c(c1)nc(s2)c3cnoc3N TS-00473 CC(C)(C)OC(=O)N1CCO[C@H](C1)CO TS-00474 COC(=O)CCCc1c[nH]c2c1cccc2 TS-00475 CN1CCN(CC1)c2ccc(c(n2)C#N)N TS-00476 COC(=O)CCSc1c(ccs1)N TS-00477 c1ccc(cc1)c2nnc(o2)CCC(=O)O TS-00478 CCOC(=O)c1nnc(o1)c2ccccc2 TS-00479 CCOC(=O)C1(CC1)C(=O)c2ccccc2 TS-00481 c1ccc(cc1)CN2CCC(CC2)CCN TS-00483 CCOC(=O)c1cc2ccncc2c(=O)o1 TS-00484 CCOC(=O)c1nc(on1)c2ccncc2 TS-00485 CCOC(=O)c1nc(on1)c2cccnc2 TS-00486 CCOC(=O)c1cn2ccc(c(c2n1)N)C TS-00487 CC(C)(C)OC(=O)Nc1ccc(nc1)C#N TS-00488 CCOC(=O)CNc1ccc2c(c1)CCC2 TS-00489 c1ccc(cc1)CNC2CCCC2C(=O)O TS-00490 COC(=O)c1cccc(c1)CN2CCCC2 TS-00491 CN[C@@H](Cc1c[nH]cn1)C(=O)OC.Cl TS-00492 c1cc(c(nc1)NCC(=O)O)C(F)(F)F TS-00493 c1cc(ncc1C(F)(F)F)NCC(=O)O TS-00494 c1cc(nc(c1)NCC(=O)O)C(F)(F)F TS-00495 c1ccc(cc1)c2nn(c(=O)o2)CC(=O)O TS-00496 c1cc(cnc1)CN2C[C@H](CC2=O)C(=O)O TS-00497 CCOC(=O)c1cc(c(c(c1O)C)N)C#N TS-00498 c1ccc(cc1)c2c(nc(s2)N)C(=O)O TS-00499 CCCc1ccc(cc1)C(=O)CCC(=O)O TS-00500 c1cc(ncc1C(=O)O)CCN2CCCC2 TS-00501 c1ccc(cc1)c2c[nH]c(n2)c3ccccc3 TS-00502 c1ccc(cc1)COc2ccsc2CO TS-00503 CNCc1ccc(cc1)CN2CCOCC2 TS-00504 CSc1c(c(sn1)SC)C(=O)N TS-00505 CCOC(=O)c1nnc(o1)Br TS-00506 c1cc(ccc1N2C[C@H](CC2=O)C(=O)O)O TS-00507 CCOC(=O)Cn1cnc2c1ncnc2N TS-00508 Cc1ccnc(n1)N2CCC(CC2)C(=O)O TS-00510 CN1CCN(CC1)c2cc(ccn2)C(=O)O TS-00511 CN1CCN(CC1)c2ccc(cn2)C(=O)O TS-00512 CN1CCN(CC1)c2cccc(n2)C(=O)O TS-00513 CN1CCN(CC1)c2c(cccn2)C(=O)O TS-00514 Cc1cncc(n1)N2CCC(CC2)C(=O)O TS-00515 c1cc(ccc1c2nc(nc(n2)N)N)Cl TS-00516 c1cc(ccc1c2cc(ccc2N)F)Cl TS-00517 Cc1cc(no1)c2c(c(no2)C)C(=O)OC TS-00518 COC(=O)c1ccc(c(c1)[C@H](C2CC2)O)O TS-00519 COc1ccc(c(c1)/C=C/C(=O)OC)OC TS-00520 c1ccc(cc1)C#Cc2ccc(cc2)C(=O)O TS-00521 c1cnc(cc1C(=O)O)OC2CCNCC2 TS-00522 c1cc(ncc1C(=O)O)OC2CCNCC2 TS-00523 c1cc(nc(c1)OC2CCNCC2)C(=O)O TS-00524 c1cc(c(nc1)OC2CCNCC2)C(=O)O TS-00525 CC(C)(C)C(=O)Nc1ccncc1C(=O)O TS-00526 CCOC(=O)c1cc([nH]n1)c2cccs2 TS-00527 CC(C)CCOc1cccc(c1C(=O)C)O TS-00528 Cc1ccc(cc1)C(=O)/C=C/c2ccccc2 TS-00529 CCc1cccnc1NC(=O)OC(C)(C)C TS-00530 CC(C)(C)OC(=O)NCCc1ccccn1 TS-00531 c1ccc2c(c1)ccc(c2Br)O TS-00532 c1ccc2c(c1)ccc(c2O)Br TS-00533 c1cc2ccc(cc2c(c1)Br)O TS-00534 c1cc(cc2c1cc(cc2)Br)O TS-00535 c1cnc(cc1C(=O)O)OC2CCOCC2 TS-00538 c1cc(nc(c1)OC2CCOCC2)C(=O)O TS-00539 c1cc(c(nc1)OC2CCOCC2)C(=O)O TS-00540 CCOC(=O)c1cccc(n1)C(=O)OCC TS-00541 CCOC(=O)c1c(c2c(s1)nccn2)N TS-00542 COC(=O)CCSc1c(nccn1)C#N TS-00543 Cc1[nH]cc(n1)CN2CCC(CC2)C(=O)O TS-00544 CC(C)(C)c1ccc(cc1)CSCCN TS-00545 c1c(c(c(o1)C(F)(F)F)C(=O)O)C(=O)O TS-00546 CCOC(=O)c1cnc(cn1)C(=O)OCC TS-00547 COC(=O)c1c(sc(n1)N)c2ccco2 TS-00548 CC(C)(C)OC(=O)N1CCC(=O)[C@H](C1)C#N TS-00549 CC(C)(C)OC(=O)Nc1cc(cnc1)OC TS-00550 c1cc(sc1)[C@H](C(=O)c2cccs2)O TS-00551 c1cc(ccc1C2(CCCCC2)CO)Cl TS-00552 C1CNCCC1(C(=O)O)N.Br TS-00553 CCOC(=O)c1c(scn1)C(F)(F)F TS-00554 c1cnc(cc1C(=O)O)OC2COCOC2 TS-00555 c1cc(ncc1C(=O)O)OC2COCOC2 TS-00556 c1cc(nc(c1)OC2COCOC2)C(=O)O TS-00557 COC(=O)CC[C@@H](C(=O)OC)n1cccc1 TS-00558 CSc1ncc(c(n1)NC2CC2)C(=O)O TS-00560 c1ccc2c(c1)nc(s2)SCC(=O)O TS-00561 CCOC(=O)C1CCN(CC1)C2CCCC2 TS-00562 CCOC(=O)C1CCCC1NC2CCCC2 TS-00563 CCOC(=O)c1cn2c(n1)ccc(n2)Cl TS-00564 COC(=O)c1c(sc(n1)N)C(F)(F)F TS-00565 CCOC(=O)Cc1cnc(nc1O)COC TS-00566 CC(C)(C)OC(=O)NCc1c(cccn1)F TS-00567 COC(=O)C1CC(=O)N(C1)C2CCCNC2 TS-00568 COC(=O)[C@H]1CC(=O)N(C1)C2CCNCC2 TS-00569 c1csc(n1)CN2CCC(CC2)C(=O)O TS-00570 Cc1c2cc(ccc2sc1C(=O)O)Cl TS-00571 Cc1csc2c1cc(cc2)Br TS-00572 CC(C)(c1nc(c(c(n1)O)O)C(=O)OC)N TS-00573 CNCCc1ccc(cc1)Oc2ccccc2 TS-00574 CN1CCN(CC1)c2c(c(ncn2)Cl)N TS-00575 c1ccc(c(c1)C(=O)c2cnccn2)C(=O)O TS-00576 c1ccc(cc1)OCc2ccccc2C(=O)O TS-00577 c1ccc(cc1)Oc2ccc(cc2)CC(=O)O TS-00578 c1ccc(cc1)COc2ccccc2C(=O)O TS-00579 CCOC(=O)C[C@H]1C(=O)NCCN1C(=O)C TS-00580 CCOC(=O)c1ccc(cc1)S(=O)(=O)C TS-00581 COc1ccc(cc1OC)SCC(=O)O TS-00582 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)N TS-00583 COC(=O)c1c(c(c(s1)SC)C#N)N TS-00584 CC(C)(C)OC(=O)N1CCC(CC1)CNC TS-00585 CCNC1CCN(CC1)C(=O)OC(C)(C)C TS-00586 Cc1cc(ccc1OCCCC(=O)O)Cl TS-00587 c1cnc(nc1C(F)(F)F)n2cc(cn2)N TS-00588 c1ccc(cc1)COc2ccc(cn2)C(=O)O TS-00589 c1ccc(cc1)COc2cc(ccn2)C(=O)O TS-00590 c1ccc(cc1)COc2cccc(n2)C(=O)O TS-00591 COC(=O)c1ccnc(c1)Oc2ccccc2 TS-00592 COC(=O)c1ccc(cc1)c2ccnc(n2)N TS-00593 COC(=O)c1cccc(c1)c2ccnc(n2)N TS-00594 COC(=O)c1ccccc1CS(=O)(=O)N TS-00595 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)O TS-00596 COc1ccc(cc1)Nc2ccc(cc2)OC TS-00598 CC(C)(C)OC(=O)N1CCC(CC1)CCO TS-00599 c1cc(cc(c1)Cl)Oc2ccc(cc2)C#N TS-00600 c1ccc(cc1)c2c3cc(ccc3no2)Cl TS-00601 CCOC(=O)[C@H](Cc1ccccc1)N.Cl TS-00602 CCN[C@@H](C)Cc1ccc(cc1)OC.Cl TS-00603 COc1ccc(nn1)c2ccc(cc2)C(=O)O TS-00604 COc1ccc(nn1)c2cccc(c2)C(=O)O TS-00605 COc1ccc2cccc(c2c1)CC(=O)OC TS-00606 CC(C)(C)OC(=O)N1CCN[C@@H](C1)C(=O)O TS-00607 CC[C@@H](c1ccc(cc1)c2ccccc2F)O TS-00608 CSc1c(c(n(n1)c2ccccc2)N)C#N TS-00609 CC(=O)c1ccc2c(c1)C(CCC2(C)C)(C)C TS-00610 c1cc(oc1c2n[nH]c(=O)o2)Br TS-00611 CCOC(=O)C(c1cccc(n1)OC)(F)F TS-00612 COc1ccc2c(c1)cc([nH]2)c3n[nH]c(=O)o3 TS-00613 CC(C)(C)OC(=O)N1CCOC[C@H]1C(=O)O TS-00614 CC(C)(C)OC(=O)N1C[C@H](C[C@H]1C(=O)O)O TS-00616 CC(C)(C)OC(=O)N1CCO[C@@H](C1)C(=O)O TS-00617 CCOC(=O)c1c(n(nn1)c2ccccc2)C TS-00618 c1cc(ncc1C#N)OCCC2CCNCC2 TS-00619 c1cnc(cc1C#N)OCCC2CCNCC2 TS-00620 c1cc(nc(c1)OCCC2CCNCC2)C#N TS-00621 c1c(cc(c(c1C(=O)O)OCC(=O)O)F)F TS-00622 Cc1cc(n(n1)C)Oc2ccc(cc2)C(=O)O TS-00623 CCOC(=O)c1nc(on1)Cc2ccccc2 TS-00624 Cc1c(nnn1Cc2cccc(c2)N)C(=O)O TS-00625 c1cc(cc(c1)N)Cn2c(c(nn2)C(=O)N)N TS-00626 c1ccc(c(c1)C#N)OCCN2CCOCC2 TS-00627 CC(C)(C)OC(=O)Nc1ccc(cc1)CC#N TS-00628 CCCNCc1ccc(cc1)N2CCCCC2 TS-00629 c1cc(oc1)C(=O)/C=C/c2ccc(cc2)Cl TS-00630 Cc1c(nc(o1)c2ccc(cc2)OC)C(=O)O TS-00631 c1ccc(cc1)CCN2C[C@H](CC2=O)C(=O)O TS-00632 Cc1c(ccc(n1)NC(=O)OC(C)(C)C)C#N TS-00633 CC(C)(C)OC(=O)N1CSC[C@H]1C(=O)O TS-00634 c1ccc(cc1)Cc2nc(cs2)CC(=O)O TS-00636 CC(C)(C)OC(=O)Nc1ccc2c(c1)CCC2 TS-00637 COC(=O)c1cccc(c1)CN2CCCCC2 TS-00638 COC(=O)C[C@H]1CCN(C1)Cc2ccccc2 TS-00639 CCOC(=O)C1CCCC1Nc2ccccc2 TS-00640 CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)N TS-00641 COc1ccc(c(c1)[C@H](CN)O)OC.Cl TS-00642 c1ccc(cc1)c2cc(cnc2)Br TS-00644 c1ccc(cc1)c2cccc(n2)Br TS-00645 COc1cccc(c1)Cc2nc(on2)C(=O)O TS-00646 c1cnc(cc1C(=O)O)NCC2CCCCC2 TS-00647 c1cc(ncc1C(=O)O)NCC2CCCCC2 TS-00648 c1cc(nc(c1)NCC2CCCCC2)C(=O)O TS-00649 c1cc(c(nc1)NCC2CCCCC2)C(=O)O TS-00650 COc1cccc(c1)N2C[C@H](CC2=O)C(=O)O TS-00652 c1ccc(cc1)COC(=O)NC2(CC2)C(=O)O TS-00653 COC(=O)c1c(sc(n1)N)c2cccnc2 TS-00654 C=CCSc1c(cccn1)c2n[nH]c(=O)o2 TS-00655 c1ccc(cc1)CN2CCO[C@H](C2)CC(=O)O TS-00656 COc1ccc(cc1)CN2CC[C@@H](C2)C(=O)O TS-00657 COc1cccc(c1)CN2CC[C@@H](C2)C(=O)O TS-00658 COC(=O)c1cccc(c1)CN2CCOCC2 TS-00659 COC(=O)[C@@H]1CN(CCO1)Cc2ccccc2 TS-00660 c1ccc(cc1)COC(=O)N2CC[C@@H](C2)CO TS-00661 CN1CCN(CC1)c2ccc(cc2C(=O)O)N TS-00662 CCOC(=O)C1CCN(CC1)c2ncccn2 TS-00663 CCOC(=O)c1c(csc1n2cccc2)C TS-00664 c1cc(c(nc1)N(CCO)C2CCCCC2)N TS-00665 COc1ccc(cc1OC2CCCC2)C(=O)O TS-00666 c1cc(ccc1C(=O)O)OCC2CCOCC2 TS-00667 c1cc(cc(c1)OCC2CCOCC2)C(=O)O TS-00668 CCCOc1ccc(cc1)C(=O)CCC(=O)O TS-00669 c1cc(ncc1C(=O)O)OCC2CCNCC2 TS-00670 c1cnc(cc1C(=O)O)OCC2CCNCC2 TS-00671 c1cc(nc(c1)OCC2CCNCC2)C(=O)O TS-00672 c1cc(c(nc1)OCC2CCNCC2)C(=O)O TS-00673 c1ccc(cc1)c2c(noc2N)c3ccccc3 TS-00674 c1ccc2c(c1)c(nc(n2)CSCCO)O TS-00675 Cc1c(c2c(s1)CC(CC2=O)(C)C)C(=O)C TS-00676 CCOC(=O)c1nnc(s1)Br TS-00677 COc1c2ccccc2ccc1Br TS-00678 c1cnc(cc1C(=O)O)OC[C@H]2CCCCO2 TS-00680 c1cc(ncc1C(=O)O)OC[C@H]2CCCCO2 TS-00681 c1cc(nc(c1)OC[C@H]2CCCCO2)C(=O)O TS-00682 c1cc(ncc1C(=O)O)OCC2CCOCC2 TS-00683 c1cc(c(nc1)OCC2CCOCC2)C(=O)O TS-00684 c1cnc(cc1C(=O)O)OCC2CCOCC2 TS-00685 COC(=O)[C@H]1CC(=O)N(C1)CCn2ccnc2 TS-00686 c1cc(ccc1CNC2CCCC2C(=O)O)F TS-00687 CC(C)(C)OC(=O)NC[C@@H](c1ccccc1)O TS-00688 CN(C)CCCOc1ccc(cc1)C(=O)OC TS-00689 Cc1cc(ccc1NC(=O)OC(C)(C)C)OC TS-00690 Cc1c(ccc(n1)NC(=O)OC(C)(C)C)CN TS-00691 CCNS(=O)(=O)c1c(nn(c1Cl)C)C TS-00692 Cc1nc(c(o1)Br)c2ccccc2 TS-00693 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(=O)O TS-00694 CC(C)(C)OC(=O)Nc1cccnc1C(=O)O TS-00695 CC(C)(C)OC(=O)Nc1ccc(nc1)C(=O)O TS-00696 c1ccc(cc1)c2ccc(cc2F)c3cc[nH]n3 TS-00697 CC(=O)c1ccc(cc1)c2ccc(cc2)C(=O)C TS-00698 COc1ccc(cc1)C(=O)/C=C/c2ccccc2 TS-00699 CN(C)CCCCOc1ccc(cn1)C(=O)O TS-00700 CN(C)CCCCOc1cccc(n1)C(=O)O TS-00701 CN(C)CCCCOc1cc(ccn1)C(=O)O TS-00702 c1cc(ccc1c2ccc(s2)Cl)C(=O)O TS-00703 c1cc(cc(c1)C(=O)O)c2ccc(s2)Cl TS-00704 CC1(C=Cc2cc(ccc2O1)Br)C TS-00705 c1ccc(cc1)c2ccc(s2)Br TS-00706 CC(=O)N[C@@H](CSc1ccccc1)C(=O)O TS-00707 c1ccc2c(c1)nc(s2)SCCC(=O)O TS-00708 COC(=O)c1c(cc(s1)c2cccs2)N TS-00709 CCOC(=O)C1CCN(CC1)C2CCCCC2 TS-00710 CCOC(=O)C1CCCC1NC2CCCCC2 TS-00711 c1ccnc(c1)c2ccc(s2)Br TS-00712 CC(C)(C)OC(=O)Nc1cc(n(c1)C)C(=O)O TS-00713 c1cc(ccc1c2ccc(cc2)C(=O)N)C(=O)N TS-00714 CC(C)(C)OC(=O)N[C@H]1CCN(C1)C2CCC2 TS-00715 CCOC(=O)c1cc2c(s1)cccc2Cl TS-00716 c1cc(ccc1Oc2ccnc(n2)Cl)Cl TS-00717 Cc1cc(c(c2c1CCC2)OC)Br TS-00718 COc1cc(c(c(c1OC)OC)N)C(=O)OC TS-00719 CCOC(=O)Cn1nc(nn1)N2CCOCC2 TS-00720 c1cc(cc2c1cc(cc2)O)C(=O)N3CCCC3 TS-00721 c1ccc2c(c1)ccc(c2CN3CCCCC3)O TS-00724 Cc1c(cccc1Cl)NC(=O)OC(C)(C)C TS-00725 COC(=O)COc1ccc(cc1C(=O)OC)F TS-00726 Cc1c(cnn1c2ccccc2)c3n[nH]c(=O)o3 TS-00727 c1cc(ccc1Cn2c3c(c(ncn3)O)nn2)N TS-00728 CC(C)NC1CCN(CC1)C(=O)OC(C)(C)C TS-00729 CC(C)(C)c1ccc(cc1)OCC(=N)N.Cl TS-00730 Cc1c(nn(n1)c2ccccc2)c3n[nH]c(=O)o3 TS-00731 CCOC(=O)c1cccc(c1)NS(=O)(=O)C TS-00734 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)OC TS-00735 CC(C)(C)OC(=O)N(CCO)C1CCCCC1 TS-00736 c1ccc(cc1)/C=C/C(=O)c2cc(ccc2F)F TS-00737 COc1ccc(cc1)Nc2cc(ccn2)C(=O)O TS-00738 CC(C)(C)OC(=O)N1CCNC[C@H]1C(=O)OC TS-00739 CC(C)(C)OC(=O)N1CCN[C@@H](C1)C(=O)OC TS-00740 CC(C)(C)OC(=O)N[C@@H]1C[C@H](NC1)C(=O)OC TS-00741 c1ccc(cc1)Sc2ccccc2CC(=O)O TS-00742 CC(C)(C)OC(=O)N1CCO[C@H](C1)CC(=O)O TS-00744 COC(=O)c1ccc(nc1)Sc2ccccc2 TS-00745 c1ccc(cc1)CSc2c(cccn2)C(=O)O TS-00746 c1cc(cc(c1)Br)CSCCN TS-00747 CCOc1cccc2c1oc(c2)c3n[nH]c(=O)o3 TS-00748 C1C2CC3CC1CC(C2)(C3)c4nc(nc(n4)O)N TS-00749 c1ccc2c(c1)cc(nc2N3CCCCC3)Cl TS-00751 c1ccc(cc1)NCC[C@H](C(=O)O)C(F)(F)F TS-00753 CC(C)(C)OC(=O)N1CSCC[C@H]1C(=O)O TS-00755 CC(C)(C)OC(=O)N1CCS[C@@H](C1)C(=O)O TS-00756 CCOC(=O)c1cc(sc1N)c2ccccc2 TS-00757 CCOC(=O)C1CCCC1NCc2ccccc2 TS-00758 c1ccc(cc1)c2cc(cnc2C#N)C(F)(F)F TS-00759 CC(=O)N1CCN(CC1)c2ccc(cc2)C(=O)O TS-00760 CC(=O)N1CCN(CC1)c2cccc(c2)C(=O)O TS-00761 CCOC(=O)Cc1ccc(cc1)N2CCNCC2 TS-00762 CC(=O)c1cc(cc(c1O)C(C)(C)C)C(C)(C)C TS-00763 c1cc(cc(c1)Cl)Oc2ccc(cc2)C(=O)O TS-00764 Cn1c(c(nc1Br)C(=O)O)C(=O)O TS-00765 c1cc(ccc1N)S(=O)(=O)Nc2ccncc2 TS-00769 c1cc(cnc1)NS(=O)(=O)c2ccc(cc2)N TS-00770 COc1ccc(cc1)CN2CCC(CC2)C(=O)O TS-00771 CCOC(=O)c1cccnc1N2CCN(CC2)C TS-00772 c1ccc(c(c1)n2cc(c(=O)[nH]c2=O)C#N)Cl TS-00773 CCOC(=O)[C@H](CCC1CCCCC1)N.Cl TS-00774 c1cc(c(cc1C(=O)O)OC(F)(F)F)C(=O)O TS-00775 Cc1nc(cs1)c2cc(no2)c3n[nH]c(=O)o3 TS-00776 c1cc2c(cc1C(=O)CCC(=O)O)OCCCO2 TS-00777 CCCCOc1ccc(cc1)C(=O)CCC(=O)O TS-00778 c1cc(ncc1C(=O)O)OCCC2CCNCC2 TS-00779 c1cnc(cc1C(=O)O)OCCC2CCNCC2 TS-00780 c1cc(nc(c1)OCCC2CCNCC2)C(=O)O TS-00781 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(=O)O TS-00782 Cc1ccc(cc1)S(=O)(=O)NCCN.Cl TS-00783 c1cc2cccc(c2c(c1)C(=O)O)Br TS-00784 c1cc(c(nc1)SC/C(=N/O)/N)C(F)(F)F TS-00785 COC(=O)N1Cc2ccc(cc2C[C@H]1C(=O)O)O TS-00786 c1ccc(cc1)S(=O)(=O)n2ccc(c2)C(=O)O TS-00787 CCc1cc(c(nc1)C(=O)OCC)C(=O)OCC TS-00788 c1cc(ccc1C(=O)O)OCCN2CCOCC2 TS-00789 c1cc(cc(c1)OCCN2CCOCC2)C(=O)O TS-00790 c1ccc(c(c1)C(=O)O)OCCN2CCOCC2 TS-00791 CC(C)(C)OC(=O)Nc1ccc(cc1)CC(=O)O TS-00792 CCOC(=O)c1cccc(c1)CN(C)CC(=O)O TS-00793 CSc1ccc(cc1)N2C[C@H](CC2=O)C(=O)O TS-00794 c1ccc(c(c1)C#N)S(=O)(=O)N2CCNCC2 TS-00795 CC(C)(C)OC(=O)N1CCC(CC1)c2[nH]ccn2 TS-00796 COc1ccc(cc1)/C=C\2/C(=O)NC(=S)S2 TS-00797 c1cc(cc(c1)F)COc2ccc(cc2Cl)N TS-00798 COC(=O)c1c(csc1C(=O)OC)N.Cl TS-00799 c1cc(ccc1c2cc(cnc2)Br)F TS-00800 c1ccc(cc1)/C=C/C(=O)c2ccc(cc2)C(=O)O TS-00801 CC(C)(C)OC(=O)Nc1ccc(nc1)C(=O)OC TS-00802 c1ccc(c(c1)C#N)S(=O)(=O)N2CCOCC2 TS-00803 CC(C)Oc1cc(cc(c1)OC(C)C)C(=O)OC TS-00804 Cc1ccc(cc1)C(=O)/C=C/c2ccc(cc2)OC TS-00805 COC(=O)C1(CCCCC1)c2ccc(cc2)Cl TS-00806 COc1ccc(cc1)/C=C/C(=O)c2cccc(c2)N TS-00807 CCOC(=O)c1cnc(nc1NC2CC2)SC TS-00808 CC(C)(C)N[C@]1(CC(=O)C=C1)C(=O)OC(C)(C)C TS-00809 CC(C)(C)OC(=O)N1CCC(CC1)C2=NCCN2 TS-00810 CCOC(=O)c1c(csc1N)c2cccs2 TS-00811 c1cc(ccc1Oc2ccc(cc2N)Cl)Cl TS-00812 CC(C)(C)c1ccc(c(c1)C(=O)c2ccccc2)O TS-00813 COC(=O)[C@H](Cc1c[nH]c2c1cccc2)N.Cl TS-00814 COc1ccc(cc1Br)C(F)(F)F TS-00815 c1ccc(c(c1)C(=O)O)S(=O)(=O)N2CCCC2 TS-00816 c1cc(cc2c1cc(cc2)O)C(=O)N3CCCCC3 TS-00817 Cn1c(nnc1SCC(=O)O)c2cccs2 TS-00818 CS(=O)(=O)N1CCN(CC1)c2ccc(cc2)N TS-00819 Cc1ccc2c(ccnc2c1Br)Cl TS-00820 c1cc(ccc1C(=O)CCC(=O)O)Br TS-00821 CC(C)(c1ccc(cc1)Br)C(=O)OC TS-00822 CC(C)(C)OC(=O)c1cccc(c1)Br TS-00823 CNCc1ccc(cc1C(F)(F)F)C(F)(F)F TS-00824 CNCc1cc(ccc1C(F)(F)F)C(F)(F)F TS-00825 CCOC(=O)c1c(c(sc1N)C(=O)OCC)C TS-00826 c1cc(ccc1c2ccnc(c2)Cl)C(F)(F)F TS-00829 CCOC(=O)c1ccc(cc1)Oc2cncc(n2)C TS-00830 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCCO TS-00831 CC(C)(C)OC(=O)N1CCN[C@H](C1)CC(=O)OC TS-00832 CCOc1c(cc(cn1)Br)C(=O)OC TS-00833 COC(=O)COc1c(cc(cc1F)F)C(=O)OC TS-00834 CCOC(=O)c1c(n(nn1)Cc2cccc(c2)N)C TS-00835 CCOC(=O)Cc1ccc(c(c1)F)Br TS-00836 Cc1c(oc(n1)C)C(=O)/C=C/c2ccc(cc2)Cl TS-00838 Cc1cc(cc(c1)c2cccc(n2)Br)C TS-00839 CCOC(=O)c1nc(on1)Cc2cccc(c2)OC TS-00840 COc1cc(c(cc1OC)OC)C(=O)n2ccnc2 TS-00841 Cc1nc2cc(ccc2o1)CNC(=O)OC(C)(C)C TS-00842 CC(=O)N1CCN(CC1)c2ccc(cc2)C(=O)OC TS-00843 COC(=O)CCN1CCN(CC1)Cc2ccccc2 TS-00844 Cc1cc(c(cc1NC(=O)C)Cl)S(=O)(=O)N TS-00845 c1cnn(c1C(F)(F)F)c2nc(cs2)C(=O)O TS-00846 CCOC(=O)CNc1ccc(cc1)OC(F)(F)F TS-00847 COc1cccc(c1)Cc2nc(cs2)CC(=O)O TS-00848 CCOC(=O)c1ccc(c(c1)Cl)Br TS-00849 c1cc(cc(c1)C(=O)O)COc2ccc(cc2F)F TS-00850 CCN(CC)c1ccc(cc1)C(=O)NCCC(=O)O TS-00851 c1c(cnc(c1Cl)NC2CCCC2)C(F)(F)F TS-00852 c1c(cc(nc1N2CCCCC2)Cl)C(F)(F)F TS-00853 COC(=O)[C@@H]1COC(=O)N1C2CCNCC2.Cl TS-00854 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O TS-00855 COC(=O)c1ccc(nc1)Oc2ccc(cc2F)F TS-00856 CC(=O)c1ccc(nc1)c2ccc(cc2)C(F)(F)F TS-00857 CC(=O)c1ccc(nc1)c2cccc(c2)C(F)(F)F TS-00858 c1ccc(cc1)c2ccc(cc2F)c3ccnc(n3)N TS-00859 CCOC(=O)C1CCCC1NCc2ccc(cc2)F TS-00860 c1nc2c(n1[C@H]3C[C@H](C=C3)CO)nc(nc2Cl)N TS-00861 c1cc(ccc1N)S(=O)(=O)Nc2ccc(cc2)F TS-00862 c1cc(cc(c1)F)NS(=O)(=O)c2ccc(cc2)N TS-00863 CC(C)c1ccc(cc1)/C=C/C(=O)c2ccccc2O TS-00864 CC(C)(C)OC(=O)N1CCC(CC1)n2cc(cn2)N TS-00865 CC[C@H]1CCCCN1C(=O)c2ccc(nc2Cl)C TS-00866 CC1(CCC(c2c1ccc(c2)Br)(C)C)C TS-00867 CC(C)(C)OC(=O)Nc1cc(ccc1OC)C(=O)O TS-00868 c1ccc(cc1)COc2ccc3c(c2)cc([nH]3)C(=O)O TS-00869 CCOC(=O)c1c(c([nH]c1C)C(=O)OC(C)(C)C)C TS-00870 COC(=O)[C@H]1CC(=O)N(C1)Cc2cccc(c2)Cl TS-00871 Cc1cccc(c1Br)C(=O)N2CCCC2 TS-00874 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C#CCO TS-00875 c1cc(c(c2c1cc(cc2)C(=O)O)S(=O)(=O)O)O TS-00876 c1ccc(c(c1)C(=O)/C=C/c2ccc3c(c2)OCO3)O TS-00877 c1cc(ccc1/C=C/c2ccc(cc2)C(=O)O)C(=O)O TS-00878 CCCc1nc(c(n1C)C(=O)OCC)C(=O)OCC TS-00879 CCCCCc1ccc(cc1)c2ccc(cc2)[C@H](C)O TS-00880 c1cc(ccc1c2cc(cnc2)Br)Cl TS-00881 CCOC(=O)[C@H](Cc1c[nH]c2c1cccc2)N.Cl TS-00882 CCOC(=O)C(c1ccc(cn1)C(F)(F)F)(F)F TS-00885 CCOC(=O)C(c1c(cccn1)C(F)(F)F)(F)F TS-00886 c1cc(c(nc1)Oc2ccc(cc2)CO)C(F)(F)F TS-00887 c1cc(ccc1CO)Oc2ccc(cn2)C(F)(F)F TS-00888 c1cc(nc(c1)Oc2ccc(cc2)CO)C(F)(F)F TS-00889 COC(=O)[C@H]1CC(=O)N(C1)Cc2ccc(c(c2)F)F TS-00890 c1ccc(c(c1)C(=O)O)S(=O)(=O)N2CCCCC2 TS-00891 CCOC(=O)c1cn2cc(ncc2n1)Br TS-00892 c1cc(ccc1CO)Oc2nccc(n2)C(F)(F)F TS-00893 c1cc(cc(c1)Oc2nccc(n2)C(F)(F)F)CO TS-00894 c1cc(ccc1CO)Oc2ccnc(n2)C(F)(F)F TS-00895 c1cc(cc(c1)Oc2ccnc(n2)C(F)(F)F)CO TS-00896 c1cc(ccc1c2cc(=O)c3c(cc(cc3o2)O)O)O TS-00897 c1cc(ccc1/C=C/C(=O)c2ccc(cc2)C(=O)O)F TS-00898 c1ccc(cc1)C(=O)Oc2ccccc2CCC(=O)O TS-00899 COC(=O)c1ccc(cc1)c2ccc(cc2)C(=O)OC TS-00900 c1ccc(c(c1)C(=O)O)S(=O)(=O)N2CCNCC2 TS-00901 Cc1c(snn1)N2CCCN2C(=O)OC(C)(C)C TS-00902 CC(C)(C)OC(=O)N1CCN(CC1)C2CCOCC2 TS-00903 CC1(Cc2c(c(sc2C(=O)O)SC)C(=O)C1)C TS-00904 CCOc1ccc(cc1/C=C/C(=O)O)Br TS-00905 c1cc(c(cc1Cl)Sc2ccc(cn2)N)Cl TS-00907 c1cc(cc(c1)OC(F)F)N2C[C@H](CC2=O)C(=O)O TS-00908 c1ccc(c(c1)C(=O)O)S(=O)(=O)N2CCOCC2 TS-00909 COC(=O)C(c1ccccc1)N2CCOCC2.Cl TS-00911 Cc1c(nnn1c2ccc(cc2Cl)Cl)C(=O)O TS-00912 CC(=O)OC[C@@H]1[C@H]([C@@H](C=CO1)OC(=O)C)OC(=O)C TS-00913 CC(C)(C)OC(=O)N[C@H]1CCCN(C1=O)CC(=O)O TS-00914 C#CCN1CCN(CC1=O)C(=O)OCc2ccccc2 TS-00915 CC(C)(C)OC(=O)N[C@@H](Cc1cscn1)C(=O)O TS-00916 COc1ccc2c(c1)c(c(cn2)Cl)Br TS-00917 COc1ccc(c(c1)CN2CCNCC2)OC.Cl TS-00918 CCOC(=O)c1cc2cc(ccc2[nH]1)OC(F)(F)F TS-00919 c1cc(ccc1CN2CC[C@@H](C2)C(=O)O)C(F)(F)F TS-00920 c1cc(cc(c1)C(F)(F)F)CN2CC[C@@H](C2)C(=O)O TS-00921 Cn1cc(nc1)S(=O)(=O)N2CCC(CC2)C(=O)O TS-00922 COC(=O)c1cc(c(nc1Cl)N2CCNCC2)F TS-00924 COc1cc2c(cc1OC)CN[C@@H](C2)C(=O)O.Cl TS-00925 c1cc(ccc1C#N)Oc2ccc(cc2)Br TS-00926 CCOC(=O)c1cc2c(cccc2s1)C(F)(F)F TS-00927 CCOC(=O)c1cc2ccc(cc2s1)C(F)(F)F TS-00928 CCOC(=O)c1cc2cccc(c2s1)C(F)(F)F TS-00929 c1cc(ccc1C(F)(F)F)Oc2ccnc(n2)Cl TS-00930 c1cc(cc(c1)Oc2ccnc(n2)Cl)C(F)(F)F TS-00931 COC(=O)c1cc(c(nc1Cl)N2CCOCC2)F TS-00932 CCC(=O)c1ccc(c(c1)Cl)OCc2ccccc2 TS-00933 CCc1ccc(cc1)CNC(=O)c2ccc(nc2)Cl TS-00934 c1cc(ccc1N2CC[C@@H](C2)C(=O)O)OC(F)(F)F TS-00935 c1cc(nnc1C(F)(F)F)N2CCC(CC2)C(=O)O TS-00936 c1cc(ncc1C(F)(F)F)N2CCN(CC2)CCO TS-00937 c1cc(ncc1C(F)(F)F)OCCN2CCNCC2 TS-00938 c1ccc2c(c1)nc(n2CC(=O)O)CN3CCOCC3 TS-00939 c1ccc(cc1)S(=O)(=O)n2ccc(c2)C(=O)C3CC3 TS-00940 c1ccc2c(c1)c(c(cn2)C(F)(F)F)Br TS-00941 c1ccc2c(c1)c(cc(n2)Br)C(F)(F)F TS-00942 COc1ccc2cc(ccc2c1CC#N)Br TS-00943 CCOC(=O)C(c1nnc(s1)C(F)(F)F)(F)F TS-00944 Cc1cc(c2c(c(sc2n1)C(=O)O)N)C(F)(F)F TS-00945 C[C@@H](C(=O)c1ccc(cc1F)F)OCc2ccccc2 TS-00946 c1ccc(cc1)S(=O)(=O)Cc2ccc(cc2)C(=O)O TS-00947 c1ccc(cc1)S(=O)(=O)Cc2cccc(c2)C(=O)O TS-00948 CC(C)(C)OC(=O)N1CCNCC1Cc2ccccc2 TS-00949 CC(C)(C)OC(=O)N1CCN[C@H](C1)Cc2ccccc2 TS-00950 CSc1nc(nc(n1)N)C23CC4CC(C2)CC(C4)C3 TS-00951 COc1c(csc1c2n[nH]c(=O)o2)Br TS-00952 c1ccc(cc1)/C=C/C(=O)c2cc(cc(c2)Cl)Cl TS-00953 CC(C)(C)OC(=O)N1CC[C@](C1)(CO)c2ccccc2 TS-00956 CC(C)(C)C(=O)Nc1cccc(n1)NC(=O)C(C)(C)C TS-00957 COC(=O)c1cccc(c1)COc2ccc(cc2F)F TS-00958 c1ccc(cc1)CC(=O)Cc2cccc(c2)C(F)(F)F TS-00959 COc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)N TS-00960 COc1cccc(c1)NS(=O)(=O)c2ccc(cc2)N TS-00961 CC(C)S(=O)(=O)c1cnc(nc1N)c2cccnc2 TS-00962 CC(C)(C)OC(=O)N1CCN(CC1)c2c(cccn2)N TS-00963 CC(C)(C)OC(=O)N1CCCN(CC1)c2cnccn2 TS-00964 c1c(cnc(c1Cl)NC2CCCCC2)C(F)(F)F TS-00965 c1cc(ccc1C(=O)C(=O)c2ccc(cc2)Cl)Cl TS-00966 c1ccc(cc1)SCc2ccc(cc2)Br TS-00967 CCOC(=O)[C@@H]1Cc2cc(ccc2CN1C(=O)OC)O TS-00968 c1ccc(cc1)C(c2ccccc2)N3CC(C3)(C4CC4)O TS-00971 c1c(cnc(c1Cl)OC2CCCCC2)C(F)(F)F TS-00972 CCOC(=O)C(c1c(cccn1)Br)(F)F TS-00973 c1cc(ccc1Oc2cc(ccn2)C#N)OC(F)(F)F TS-00974 CCCc1c(ccc(c1O)C(=O)C)SC(=O)C(C)C TS-00975 c1ccc(cc1)CNc2c(cc(c(n2)Cl)C(=O)O)F TS-00976 COC(=O)c1cc2cc(ccc2[nH]1)OCc3ccccc3 TS-00977 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)F TS-00979 c1cc(ccc1C(=O)C[C@@H](C(=O)O)N2CCCC2)Cl TS-00980 c1ccc(c(c1)CN)Sc2ccccc2CO.Cl TS-00981 Cc1cccc(c1Br)C(=O)N2CCCCC2 TS-00982 c1cc(cc(c1)Nc2cc(ccn2)C(=O)O)C(F)(F)F TS-00983 COc1ccc(cc1)/C=C/C(=O)c2ccc(cc2)C(=O)O TS-00984 CCOC(=O)Cc1c(c(sc1C(=O)OCC)N)C#N TS-00985 Cc1ccc(cc1)C(=O)/C=C/c2ccc(c(c2)OC)OC TS-00986 CC(C)C[C@@H](C(=O)O)NC(=O)c1cccnc1SC TS-00987 c1ccc(cc1)CN2CCN(CC2)c3cc(ccn3)CN TS-00988 COc1ccc(c(c1OC)Cl)/C=C/c2n[nH]c(=O)o2 TS-00989 CC(=O)N1CCN(CC1)c2c(cc(c(n2)Cl)C#N)F TS-00990 c1cc(ccc1N)S(=O)(=O)Nc2ccc(cc2)Cl TS-00991 c1cc(cc(c1)Cl)NS(=O)(=O)c2ccc(cc2)N TS-00992 COC(=O)c1cccc(c1Br)C(F)(F)F TS-00993 CCOC(=O)Cc1cnc2n1cc(cc2)Br TS-00996 c1cc(c(nc1)Oc2ccc(cc2)C(=O)O)C(F)(F)F TS-00997 c1cc(nc(c1)Oc2ccc(cc2)C(=O)O)C(F)(F)F TS-00998 c1cc(cc(c1)Oc2cccc(n2)C(F)(F)F)C(=O)O TS-00999 c1cc(c(nc1)c2ccc(cc2)OC(F)(F)F)C(=O)O TS-01000 c1cc(cc(c1)OC(F)(F)F)c2c(cccn2)C(=O)O TS-01001 c1cc(ccc1c2ccc(cn2)C(=O)O)OC(F)(F)F TS-01002 c1cc(cc(c1)OC(F)(F)F)c2ccc(cn2)C(=O)O TS-01003 c1cc(ccc1C(=O)O)Nc2nccc(n2)C(F)(F)F TS-01004 c1cc(cc(c1)Nc2nccc(n2)C(F)(F)F)C(=O)O TS-01005 c1cc(ccc1C(=O)O)Nc2ccnc(n2)C(F)(F)F TS-01006 c1cc(cc(c1)Nc2ccnc(n2)C(F)(F)F)C(=O)O TS-01007 COC(=O)CS(=O)(=O)c1ccc(cn1)C(F)(F)F TS-01008 CNCc1ccc(cc1)Oc2ccnc(n2)C(F)(F)F TS-01009 CCOC(=O)c1c(nc(s1)c2ccccc2Cl)O TS-01010 CCOC(=O)c1c(nc(s1)c2cccc(c2)Cl)O TS-01011 CCOC(=O)c1c(nc(s1)c2ccc(cc2)Cl)O TS-01012 COC(=O)C1CN(CCC1=O)Cc2ccccc2.Cl TS-01013 CCOC(=O)C(c1ccccc1)C2CCCCN2.Cl TS-01014 c1cc(ccc1C(=O)O)Oc2ccnc(n2)C(F)(F)F TS-01015 c1cc(cc(c1)Oc2ccnc(n2)C(F)(F)F)C(=O)O TS-01016 c1cc(cc(c1)Oc2nccc(n2)C(F)(F)F)C(=O)O TS-01017 c1cc(ccc1OCCN2CCCCC2)Br TS-01018 c1cc(cc(c1)Br)OCCN2CCCCC2 TS-01019 c1ccc(c(c1)OCCN2CCCCC2)Br TS-01020 COc1ccc(cc1OC)/C=C/C(=O)c2ccccc2O TS-01021 CC(C)(C)OC(=O)N1CCC(CC1)N2CCCOC2=O TS-01022 c1ccc(cc1)Sc2ccc(cc2)c3csc(n3)N TS-01023 c1ccc2c(c1)OC[C@H](O2)C(=O)N3CCNCC3.Cl TS-01024 COC(=O)C[C@H]1CN(CCN1)Cc2ccccc2.Cl TS-01025 CCOC(=O)c1cc2ccc(cc2s1)Br TS-01026 CCOC(=O)[C@@H]1CCN(CCC1=O)C(=O)OC(C)(C)C TS-01027 COc1ccc(cc1)CNCc2ccccc2C(=O)OC TS-01028 c1c(cnc(c1Cl)SCCC(=O)O)C(F)(F)F TS-01029 c1cc(ccc1OCCN2CCOCC2)Br TS-01030 c1cc(cc(c1)Br)OCCN2CCOCC2 TS-01031 c1ccc(c(c1)OCCN2CCOCC2)Br TS-01032 Cc1ccc(cc1)S(=O)(=O)N[C@@H](CC(=N)O)C(=O)O TS-01033 CCOC(=O)COc1ccc(cc1)OCc2ccccc2 TS-01034 c1ccc(cc1)CNc2cc(cc(n2)Cl)C(F)(F)F TS-01035 COC(=O)c1ccc(o1)Oc2cc(cc(c2)Cl)Cl TS-01036 c1c(cnc(c1Br)N2CCOCC2)C(=O)O TS-01037 c1cc(cc(c1)C(F)(F)F)CN2C[C@H](CC2=O)C(=O)O TS-01039 c1cc(ccc1CN2CCC(CC2)C(=O)O)C(F)(F)F TS-01040 COc1cc2c(cc1OC)CN[C@@H](C2)C(=O)OC.Cl TS-01041 COc1cc(cc(c1C(=O)O)C(F)(F)F)C(F)(F)F TS-01042 c1ccc(cc1)CN2CCC(C2)N3CC(CC3=O)C(=O)O TS-01043 CCOC(=O)c1cc(c(nc1N2CCCNCC2)C)C#N TS-01044 c1cc(ccc1N2C[C@H](CC2=O)C(=O)O)OC(F)(F)F TS-01046 COc1ccc2c(c1)cc([nH]2)c3nn(c(=O)o3)CC(=O)O TS-01047 CCOC(=O)c1c(c2cc(ccc2s1)C(F)(F)F)N TS-01048 CC(=O)c1c(ccs1)NC(=O)c2ccccc2C(=O)O TS-01049 CC(C)(C)OC(=O)N[C@H](c1c[nH]c2c1cccc2)C(=O)O TS-01052 CC(C)(C)OC(=O)N[C@@H](Cc1cccc(c1)C#N)C(=O)O TS-01053 c1cc(cc(c1)Cl)c2cc(c(o2)C(F)(F)F)C(=O)O TS-01054 Cc1ccc(cc1)/C=C/C(=O)c2cc(cc(c2)Cl)Cl TS-01055 c1cc(cc(c1)N)C(=O)/C=C/c2ccc(cc2)C(F)(F)F TS-01056 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccncc2 TS-01057 CC(C)(C)OC(=O)N1CC[C@@](C1)(c2ccccc2)C(=O)O TS-01058 CC(=O)N[C@H]1CCc2c(sc(n2)N)C1.Br TS-01059 Cc1cncc(n1)N2CCCN(CC2)C(=O)OC(C)(C)C TS-01060 C=CCSc1c(cccn1)c2nn(c(=O)o2)CC(=O)O TS-01061 COC(=O)CNS(=O)(=O)c1ccsc1C(=O)OC TS-01062 Cc1ccc(cc1)C[C@H](CC(=O)O)NC(=O)OC(C)(C)C TS-01063 CC(C)(C)OC(=O)N1CCC(CC1)Oc2ccc(cn2)N TS-01064 CC(C)(C)OC(=O)N1CCN(CC1)c2cc(cnc2)OC TS-01065 c1ccc(c(c1)OCc2nc(on2)c3n[nH]c(=O)o3)Cl TS-01066 c1ccc2c(c1)c3ccccc3n2c4ccc(cc4)N.Cl TS-01067 c1cc2c(ccnc2cc1Cl)Sc3nnc(s3)N TS-01068 c1c(c(c(nc1Br)Br)N)C(=O)N TS-01069 c1cc(ccc1C(=O)O)Oc2ncc(cn2)Br TS-01070 c1cc(ccc1/C=C/C(=O)c2cc(cc(c2)Cl)Cl)F TS-01072 CC(C)(C)OC(=O)N1CCN(CC1)CCn2cc(cn2)N TS-01073 c1cc(ccc1C(=O)C[C@@H](C(=O)O)N2CCCCC2)Cl TS-01074 c1cc(ccc1c2cnc(o2)CCC(=O)O)Br TS-01075 CC(C)(C)OC(=O)n1ccc2c1ccc(c2)Br TS-01076 c1ccc(cc1)[C@H](C(=O)c2ccccc2)OCCCC(=O)O TS-01077 CC(C)(C)OC(=O)N1CCc2c(sc(c2C(=O)O)N)C1 TS-01078 CC(C)(C)OC(=O)N1CCC(CC1)N2CCC[C@H]2C(=O)O TS-01079 CC(C)(C)OC(=O)N1CCCC(C1)N2CCCC2C(=O)O TS-01080 CC(C)(C)OC(=O)N1CCC(CC1)N2CCC(CC2)CO TS-01081 c1cc(c(c(c1)OCC(F)(F)F)C#N)OCC(F)(F)F TS-01082 c1cc(ccc1Oc2cc(ccn2)C(=O)O)OC(F)(F)F TS-01083 COC(=O)CCSc1c(cc(cn1)C(F)(F)F)Cl TS-01084 Cc1nc(cs1)c2cccs2 TS-01426 CNCc1ccccc1c2ccco2 TS-01427 c1cc(oc1)c2ccnc(c2)C(=O)O TS-01428 c1cc(ccc1C2(CCC2)C(=O)O)C(F)(F)F TS-01429 C1CC1(CC#N)CO TS-01430 COC(=O)C1(CC1)O TS-01431 Cc1ccncc1CN TS-01432 Cc1cccnc1CN TS-01433 Cc1ccc(nc1)CN TS-01434 c1cc(ncc1CN)N TS-01437 Cc1c(ocn1)C(=O)O TS-01439 CN1CCNCCC1=O TS-01440 COc1c(ccs1)N TS-01441 C1COCCC1(CN)O TS-01442 C#CCOc1ccccc1 TS-01443 c1cc2c(nc1)CCC2=O TS-01444 c1ccc2c(c1)C[C@@H]2CN TS-01445 Cc1cccnc1CNC TS-01446 COc1ccc(cn1)CN TS-01447 COc1cc(ccn1)CN TS-01448 CCOc1c(ccs1)N TS-01449 c1cc2c(cc[nH]2)nc1CN TS-01450 CCOc1ccc(cn1)CN TS-01451 CCOc1cc(ccn1)CN TS-01452 c1c(cc(cc1O)Cl)CN TS-01453 c1cc2c(cc1C#N)[nH]c(=O)[nH]2 TS-01454 Cc1ccc(cc1)C2(CC2)CN TS-01455 Cc1cc2c(cc1C)[nH]c(=O)[nH]2 TS-01456 Cc1ccc2c(c1C)[nH]c(=O)[nH]2 TS-01457 c1cc(cnc1)[C@@H]2CCCCN2 TS-01458 CNCc1ccc(cc1)N(C)C TS-01459 CC(C)(c1ccc(cc1)OC)N TS-01460 COc1ccc(cc1OC)CN TS-01461 C1CCN(CC1)C2CCNCC2 TS-01462 CC(C)(C)[C@H]1C(=O)NCC(=O)N1 TS-01463 c1c(n[nH]c1Cl)C(F)(F)F TS-01464 c1cc2c(cc1F)[nH]c(n2)Cl TS-01465 COc1cc(cc(c1)Cl)CN TS-01466 c1cc(oc1)c2ccc(cc2)CN TS-01467 c1cc2cc(ccc2cc1CN)O TS-01468 c1cc(ncc1CN)n2ccnc2 TS-01469 c1cnc(cc1CN)n2ccnc2 TS-01470 c1cncc(c1C(F)(F)F)CN TS-01471 COc1cccc(c1)C2(CC2)CN TS-01472 c1cc2c(cc1C#N)[nH]c(n2)Cl TS-01473 c1ccc2c(c1)C[C@@H](CO2)C(=O)O TS-01474 Cc1c(nc(o1)c2ccoc2)CN TS-01475 Cc1c(nc(o1)c2ccco2)CN TS-01476 c1cc(c(c(c1)F)C2(CC2)CN)F TS-01478 CC(C)(CN)c1c(cccc1F)F TS-01479 CC(=O)[C@@H](c1ccccc1)N.Cl TS-01480 c1c2c(cc(c1F)Cl)[nH]c(=O)[nH]2 TS-01481 c1cc(ccc1CN)Cn2ccnc2 TS-01482 c1cc(cc(c1)Cn2ccnc2)CN TS-01483 c1cc(cc(c1)C(=O)O)c2c[nH]cn2 TS-01484 Cc1c(nc(o1)c2ccncc2)CN TS-01485 Cc1c(nc(o1)c2cccnc2)CN TS-01486 CC[C@]1(Nc2ccccc2C(=O)N1)C TS-01487 CNc1ccccc1OC(F)(F)F TS-01488 c1ccc(cc1)Oc2c(ccs2)N TS-01489 COc1cccc(c1)C2(CCC2)CN TS-01490 c1cc(ncc1CN)N2CCCCC2 TS-01491 c1cnc(cc1CN)N2CCNCC2 TS-01492 c1cc(ncc1CN)N2CCOCC2 TS-01493 c1cncc(c1CN)N.Cl.Cl TS-01494 c1cc(c(c(c1)F)C2(CCC2)CN)F TS-01495 Cc1nc2cc(ccc2o1)CN.Cl TS-01496 c1cc(cc(c1)C(=O)O)c2ncccn2 TS-01497 COc1ccc2cccc(c2c1)CCN TS-01498 c1cc2c(cc1C(F)(F)F)[nH]c(=O)[nH]2 TS-01499 c1c2c(cc(c1Cl)Cl)[nH]c(=O)[nH]2 TS-01500 c1cc(cc(c1)CN2CCCCC2)CN TS-01501 Cc1cc(c(c(n1)Cl)C(=O)O)Cl TS-01502 c1cnc(cc1CN)OC2CCCCC2 TS-01503 c1cc(ncc1CN)OC2CCCCC2 TS-01504 CN1CCN(CC1)c2cc(ccn2)CN TS-01505 c1cnc(cc1CN)OC2CCOCC2 TS-01506 c1cc(ncc1CN)OC2CCOCC2 TS-01507 c1cc(ccc1C2(CC2)C#N)C(F)(F)F TS-01508 Cc1c2c(c3ccccc3n1)C(=O)NC2=O TS-01509 CN1CCN(CC1)Cc2ccc(cc2)CN TS-01513 c1ccc(cc1)Oc2cc(sc2)C(=O)O TS-01514 c1cc2c(cc1C(F)(F)F)[nH]c(n2)Cl TS-01515 c1ccc(cc1)[C@@H](c2ccccn2)N.Cl TS-01516 CNCc1ccc(o1)c2ccc(cc2)Cl TS-01517 CNCc1c([nH]c(n1)c2ccccc2)Cl TS-01518 COc1ccc2c(c1)cc(c(n2)Cl)CO TS-01519 CC1(CC(=O)CC(=C1)NCc2ccccc2)C TS-01520 CC(c1ccccc1)N2C[C@H](CC2=O)C(=O)O TS-01521 c1cc(cc(c1)Br)C(=N)N.Cl TS-01522 c1cc(ccc1C(=N)N)Br.Cl TS-01523 c1cc(nc(c1)n2ccnc2)CN.Cl.Cl TS-01524 Cc1nccc(n1)c2cccc(c2)Br TS-01525 C#Cc1ccncc1 TS-01527 c1cncnc1C#N TS-01528 Cn1cc(cn1)C#N TS-01529 c1ccn(c1)C2CC2 TS-01530 c1[nH]c(c(n1)C#N)N TS-01531 c1cnccc1CN TS-01532 Cc1ccc(nc1)O TS-01533 c1cnc(cc1O)N TS-01534 c1cnc(cc1N)O TS-01535 c1cc(c(nc1)O)N TS-01536 c1cncc(c1N)O TS-01537 c1cncnc1CO TS-01538 c1cnc(nc1)CO TS-01539 CC(=O)c1c[nH]cn1 TS-01540 Cc1cc(=O)[nH]nc1 TS-01541 CC(C)c1cc[nH]n1 TS-01542 CCc1[nH]cc(n1)C TS-01543 c1c(ncnc1O)N TS-01544 c1c(nc[nH]1)C(=O)N TS-01545 CNCc1ccoc1 TS-01546 Cc1cc([nH]c1)CO TS-01547 CC1=C(C(=O)NC1)C TS-01548 c1ccn(c1)CCO TS-01549 C1COCCC1C#N TS-01550 C=C1CC(C1)C(=O)N TS-01551 CCn1ccc(n1)N TS-01552 CCn1cc(cn1)N TS-01553 CNCc1c[nH]cn1 TS-01554 CNCc1[nH]ccn1 TS-01555 C1CC(C1)NC2CC2 TS-01556 c1c(nc[nH]1)C(=O)O TS-01557 c1cnc(cc1F)N TS-01558 C1CC(=CC(=O)O)C1 TS-01559 Cc1ccoc1CO TS-01560 CC1C(=O)C=C(O1)C TS-01561 Cc1c(c[nH]n1)CO TS-01562 c1c(nc[nH]1)CCO TS-01563 C1C[C@@H](CC=C1)CO TS-01564 c1c(con1)C(=O)O TS-01565 c1conc1C(=O)O TS-01566 C1C=C[C@H](N1)C(=O)O TS-01567 Cc1c(ocn1)CO TS-01568 COc1c[nH]nc1N TS-01569 C[C@H]1CCCNC1=O TS-01570 C1[C@H](C=C[C@H]1N)CO TS-01571 C[C@H]1CC(=O)N(C1)C TS-01573 CC1(C[C@@H]1C(=O)N)C TS-01574 C1CCC(CC1)CN TS-01576 CC[C@H]1CCCCN1 TS-01577 CC1(C[C@@H]1C(=O)O)C TS-01578 C1C[C@H](NC1)C(=O)N TS-01579 C1CNCC(=O)NC1 TS-01580 Cc1cnc(s1)N TS-01581 c1csc(n1)CN TS-01582 C1CCC(CC1)CO TS-01583 CN[C@H]1CCN(C1)C TS-01584 C1CNCCC1CN TS-01585 CCN1CCNCC1 TS-01586 CN1CCCNCC1 TS-01587 c1cnc(cc1F)F TS-01588 C1[C@H](NC1=O)C(=O)O TS-01589 C1C[C@@H](NC1)C(=O)O TS-01590 C1CC(C1)(C(=O)O)N TS-01591 C1CC1[C@@H](C(=O)O)N TS-01592 COC(=O)C1(CC1)N TS-01593 C1C[C@H](OC1)C(=O)N TS-01594 CNC[C@H]1CCOC1 TS-01595 C1CNCCC1CO TS-01596 CN1CC[C@@H](C1)CO TS-01597 CCN1CC[C@@H](C1)O TS-01598 COC[C@H]1CCCN1 TS-01599 C1CC(OC1)C(=O)O TS-01601 C1C(CC1O)C(=O)O TS-01602 C1CC(C1)(C(=O)O)O TS-01603 C1CCO[C@H](C1)CO TS-01604 Cc1c(cccn1)C#N TS-01606 Cc1cccc(n1)C#N TS-01607 Cc1cccnc1C#N TS-01608 Cc1cc(ccn1)C#N TS-01609 c1cc(ncc1N)C#N TS-01610 c1cnc(cc1N)C#N TS-01611 c1ccc2c(c1)CNC2 TS-01612 c1c2cn[nH]c2ncn1 TS-01613 c1c(c(ncn1)N)C#N TS-01614 C1CNCC1=O.Cl TS-01616 c1cncc(c1C#N)F TS-01617 Cn1cc(c(n1)N)C#N TS-01618 CCc1cccnc1N TS-01619 CCc1ccnc(c1)N TS-01620 CNCc1ccncc1 TS-01621 CNCc1ccccn1 TS-01622 c1ccnc(c1)CCN TS-01623 C[C@@H](c1ccncc1)N TS-01624 C1CC(NC1)N.Cl TS-01625 c1cnc(cn1)C(=O)N TS-01626 c1cncnc1C(=O)N TS-01627 Cc1cccc(c1N)O TS-01628 C1C=CCC2C1C(=O)N2 TS-01629 Cc1ccncc1CO TS-01630 C[C@@H](c1ccncc1)O TS-01631 c1c(n[nH]c1N)C2CC2 TS-01632 Cc1cnc(cn1)CN TS-01633 Cc1ccsc1C#N TS-01634 Cc1cc(c(nc1)O)N TS-01635 c1cncc(c1N)CO TS-01636 Cc1ncc(cn1)CO TS-01637 COC(=O)n1cccc1 TS-01638 Cc1cc([nH]c1)C(=O)O TS-01639 COc1c(nccn1)N TS-01640 CC(=O)Nc1ccn[nH]1 TS-01641 CNc1ccc(cc1)F TS-01642 C1C[C@@H](CC=C1)C(=O)N TS-01643 CC(C)c1cc(n[nH]1)N TS-01644 CNCc1ccn(n1)C TS-01645 Cc1c(c[nH]n1)CNC TS-01646 Cc1[nH]cc(n1)CNC TS-01647 CNCc1nccn1C TS-01648 c1nc2c(s1)CCC2 TS-01649 Cc1ccoc1C(=O)O TS-01650 COC(=O)c1cc[nH]n1 TS-01651 Cc1c(c[nH]n1)C(=O)O TS-01652 Cn1cc(nc1)C(=O)O TS-01653 c1c(nc[nH]1)CC(=O)O TS-01654 COC(=O)c1c[nH]nc1 TS-01655 Cc1cc(no1)C(=O)N TS-01656 Cc1nc(co1)C(=O)N TS-01657 Cc1c(ccc(n1)N)F TS-01658 C=CCC1(CC1)C(=O)O TS-01659 C1CCC(=CC(=O)O)C1 TS-01660 C1CC(CC=C1)C(=O)O TS-01661 C1CCC(=CC1)C(=O)O TS-01662 Cc1nc(co1)C(=O)O TS-01663 Cc1ncc(o1)C(=O)O TS-01664 C1COCCC1(C#N)O TS-01665 C1C[C@H](C(=O)C1)C(=O)N TS-01666 C1CCC(C1)CC(=O)N TS-01667 CNCc1cccs1 TS-01668 CNCc1ccsc1 TS-01669 CCCc1nccs1 TS-01670 C1CSCCC1C#N TS-01671 CCC1CCC(CC1)N TS-01672 CCN1CCCCCC1 TS-01673 Cc1ccc(nc1)Cl TS-01674 Cc1c(cccn1)Cl TS-01675 c1cc(c(cc1O)O)F TS-01676 CC(=O)[C@@H]1CCC(=O)O1 TS-01677 COC(=O)C1CC(=O)C1 TS-01679 c1cc(oc1CO)CO TS-01680 CC(=O)C1CCOCC1 TS-01682 C1CNCCC1C(=O)N TS-01685 C1C[C@@H](CNC1)C(=O)N TS-01686 CCN1CCCNCC1 TS-01688 c1c(cncc1Cl)N TS-01689 c1cc(c(nc1)N)Cl TS-01690 C1[C@@H](CNC1=O)C(=O)O TS-01691 CC(=O)O[C@H]1CC(=O)N1 TS-01692 CO[C@H]1CCCNC1=O TS-01693 CN1CC[C@@H](C1)C(=O)O TS-01694 CCOC(=O)C1(CC1)N TS-01695 c1ccc2c(c1)CC2C#N TS-01696 CCc1nc(sn1)N TS-01697 CN1CCC(CC1)CO TS-01698 COC[C@H]1CCCNC1 TS-01699 CN1CCC[C@@H]1CCO TS-01700 C1C(CN1)(F)F.Cl TS-01701 c1c(c(cnn1)Cl)N TS-01702 C1CCO[C@@H](C1)C(=O)O TS-01703 CC1(COC(=O)[C@H]1O)C TS-01704 c1cc2cnccc2nc1 TS-01705 C1CC(CCC1CO)O TS-01706 CC1CC(CC(O1)C)O TS-01707 CCc1[nH]c(cn1)Cl TS-01708 C1COC(=O)N1CCO TS-01709 Cc1ccc(cc1C)C#N TS-01710 Cc1coc2c1cccc2 TS-01711 C#Cc1ccc(cc1)CO TS-01712 Cc1[nH]c2ccccc2n1 TS-01713 Cc1cn2ccccc2n1 TS-01714 Cc1ccc(s1)Cl TS-01715 c1ccc(cc1)[C@@H](C#N)O TS-01716 Cc1cc(cc(c1)O)C#N TS-01717 c1ccc2c(c1)[nH]c(n2)N TS-01718 c1cc2c(cc1N)cn[nH]2 TS-01719 c1ccn2c(c1)ncc2N TS-01720 c1cc2nccn2cc1N TS-01721 Cc1c(ccc(n1)N)C#N TS-01722 Cc1cc(cnc1N)C#N TS-01723 c1ccc2c(c1)CC[C@@H]2N TS-01724 c1ccc(cc1)C2(CC2)N TS-01725 c1ccc2c(c1)CCNC2 TS-01726 c1ccc2c(c1)CCCN2 TS-01727 c1c(cn[nH]1)CN.Cl TS-01728 c1cc(c2ccoc2c1)O TS-01729 COc1ccc(cn1)C#N TS-01730 c1cc(ncc1CO)C#N TS-01731 c1ccn2c(c1)nnc2N TS-01732 c1cc2c(ncnn2c1)N TS-01733 Cc1cnc(c(n1)C#N)N TS-01734 c1c(cnc2c1CCC2)N TS-01735 C=CCNc1cccnc1 TS-01736 c1cc2c([nH]c(=O)[nH]2)nc1 TS-01737 c1cc2c(nc1)CC[C@@H]2O TS-01738 Cc1cccnc1C(=O)C TS-01739 Cc1ccnc(c1)C(=O)C TS-01740 CC(=O)Cc1ccncc1 TS-01741 Cc1ccc(cn1)C(=O)C TS-01742 Cc1ccncc1C(=O)C TS-01743 Cc1cccc(n1)C(=O)C TS-01744 Cc1cccnc1C(=N)N TS-01745 c1cc2c(cc1F)nc[nH]2 TS-01746 c1cc2c(cn[nH]2)c(c1)F TS-01747 c1[nH]c2c(c(=O)n1)CCC2 TS-01748 Cc1c(cccn1)C(=O)N TS-01749 Cc1cccnc1C(=O)N TS-01750 Cc1ccnc(c1)C(=O)N TS-01751 Cc1ccncc1C(=O)N TS-01752 Cc1ccc(cn1)C(=O)N TS-01753 c1c(cn[nH]1)C#CCCO TS-01754 Cc1c(nccn1)C(=O)C TS-01755 c1cc2c(nc1)scn2 TS-01756 CCCc1ccccc1O TS-01757 Cc1cccc(c1C)CO TS-01758 Cc1cccc(c1)CCO TS-01759 CCCc1ccc(cc1)O TS-01760 CC(C)c1ccc(cn1)N TS-01761 Cc1ccnc(c1)CNC TS-01762 CNCCc1ccncc1 TS-01763 CNCCc1cccnc1 TS-01764 CCNCc1ccncc1 TS-01765 Cc1cccc(n1)CNC TS-01766 Cc1ccncc1C(=O)O TS-01767 CC(=O)c1ccnc(n1)N TS-01768 c1cc(sc1)C(=O)C#N TS-01769 Cc1c(cccc1OC)N TS-01770 Cc1c(cccc1N)CO TS-01771 Cc1cc(c(cc1C)O)N TS-01772 Cc1ccc(cc1N)CO TS-01773 c1cc(cc(c1)CO)CN TS-01774 Cc1ccc(c(n1)C)CO TS-01775 Cc1cc(cc(n1)C)CO TS-01776 CNc1ccc(cc1)OC TS-01777 C1CC(CNC1)O.Cl TS-01778 C1Cc2c(non2)C(=O)C1 TS-01779 c1cc(nc(c1)O)C(=O)N TS-01780 Cc1ccc(c(c1)O)OC TS-01781 Cc1cc(cc(c1)OC)O TS-01782 Cc1cc(ccc1O)OC TS-01783 c1c(n2c(n1)CCC2)CO TS-01784 CCOc1cc(ccn1)N TS-01785 CCOc1ccc(cn1)N TS-01786 CCOc1ccnc(c1)N TS-01787 CNc1cccc(n1)OC TS-01788 Cc1ccc(c(n1)OC)N TS-01789 CCOc1ccncc1N TS-01790 CNc1c(cccn1)CO TS-01791 Cc1c(cnc(n1)C)CO TS-01792 c1cnccc1OCCN TS-01793 C#CCN1CCNCC1=O TS-01794 Cc1csc(n1)CC#N TS-01795 c1cnc(cc1C(=O)O)O TS-01796 COc1cc(ccc1O)N TS-01797 Cc1cc(c([nH]1)C)C(=O)O TS-01798 Cn1cccc1CC(=O)O TS-01799 Cc1cc([nH]c1)C(=O)OC TS-01800 Cc1ccc(c(n1)O)CO TS-01801 Cc1c(c(=O)cc[nH]1)OC TS-01802 Cc1cc(nc(n1)N)OC TS-01803 CCOc1cnc(nc1)N TS-01804 Cc1c(cnc(n1)N)CO TS-01805 Cc1cc(nn1C)C(=O)N TS-01806 Cc1cc(cc(c1F)C)N TS-01807 CNCc1ccc(cc1)F TS-01808 c1cc(ccc1CCN)F TS-01809 Cc1c(c(n(n1)C)C)CN TS-01810 Cc1nc(cs1)C2CC2 TS-01811 Cc1nc2c(s1)CCC2 TS-01812 c1csc2c1CNCC2 TS-01813 C1CCC(CC1)NC2CC2 TS-01814 C1CCC2C(C1)CCCN2 TS-01815 C1CC[C@H]2CNCC[C@H]2C1 TS-01816 C1CCC2CNCCC2C1 TS-01817 C1CC(C1)(C(F)(F)F)O TS-01818 c1cc(c(nc1)F)C(=O)N TS-01819 CC(=O)OCc1ccco1 TS-01820 Cc1cc(c(o1)C)C(=O)O TS-01821 Cc1ccoc1C(=O)OC TS-01822 CCOC(=O)c1ccoc1 TS-01823 Cc1cc(c(c(=O)o1)C)O TS-01824 Cn1cc(cn1)C(=O)OC TS-01825 COCc1[nH]c(=O)ccn1 TS-01826 CCc1cc(ccc1O)F TS-01827 c1cc(cc(c1)F)CCO TS-01828 c1ccc(c(c1)CCO)F TS-01829 CNCc1c(cccn1)F TS-01830 CCc1[nH]c(c(n1)C)CO TS-01831 c1c(nc(s1)N)C2CC2 TS-01832 C1Cc2c(sc(n2)N)C1 TS-01833 C1CCN(CC1)C2CNC2 TS-01834 Cc1c(cno1)C(=O)OC TS-01835 Cc1cc(on1)CC(=O)O TS-01836 Cc1cnoc1C(=O)OC TS-01837 CCOC(=O)c1ccon1 TS-01838 CNCc1ccc(o1)CO TS-01839 CC(C)(C)c1nnc(o1)N TS-01840 C1Cc2c(sc(=O)[nH]2)C1 TS-01841 C1CC1c2nnc(s2)N TS-01842 C1CCCC(CC1)C(=O)N TS-01843 C1CCC(C1)CCC(=O)N TS-01844 Cc1ccc(s1)CNC TS-01845 Cc1ccc(cc1Cl)N TS-01846 CC1CCC(CC1)C(=O)O TS-01847 CN1CCC(CC1)C(=O)N TS-01848 CNC(=O)C1CCNCC1 TS-01849 CC(=O)N1CCCNCC1 TS-01850 Cc1c(scn1)CNC TS-01851 CCCC1CCC(CC1)O TS-01852 CN(C)CC1CCNCC1 TS-01853 Cc1ccc(c(c1)Cl)O TS-01854 Cc1ccc(c(n1)Cl)N TS-01855 Cc1cc(ncc1Cl)N TS-01856 Cc1cnc(cc1N)Cl TS-01857 c1cc(ncc1CN)Cl TS-01858 COC(=O)c1cncs1 TS-01859 C1CNCCC1CC(=O)O TS-01860 CN1CCCCC1C(=O)O TS-01861 COC(=O)C[C@H]1CCNC1 TS-01862 C1CC(=O)N(C1)CCCO TS-01863 C1CC(CCC1C(=O)N)O TS-01864 Cc1cccc2c1nccc2 TS-01865 c1ccc(cc1)C2(CC2)C#N TS-01866 Cc1c2ccccc2ccn1 TS-01867 c1cc2c(cc1C#N)CCC2 TS-01868 Cc1c(sc(n1)C)CO TS-01869 CC(=O)C1=CSCCN1 TS-01870 CN1CCC(CC1)CCO TS-01871 CC(C)(C1CCNCC1)O TS-01872 C1CNCCC1CCCO TS-01873 C1CCCN(CC1)CCO TS-01874 c1cc(c(c(c1)Cl)N)O TS-01875 c1cc(c(c(c1)O)Cl)N TS-01876 C1CC(C1)(C(=O)O)C(=O)O TS-01877 Cc1cnc(c(n1)C#N)C#N TS-01878 C[C@H](C(=O)O)C1(CCC1)O TS-01879 C1CC(CCC1C(=O)O)O TS-01880 c1ccc2c(c1)cc(cn2)N TS-01881 Cc1cccc2c1nccn2 TS-01882 c1ccc2c(c1)ccnc2N TS-01883 c1ccnc(c1)C2(CC2)C#N TS-01884 c1cnc(cc1C#N)C2CC2 TS-01885 Cc1ccc2c(c1)nccn2 TS-01886 COc1ccsc1CO TS-01887 C1CNCCN(C1)CCO TS-01889 C1COCCC1(C(=O)O)N TS-01890 C1COC(CN1)CC(=O)O TS-01891 COC(=O)[C@@H]1CNCCO1 TS-01893 COC(=O)[C@@H]1COCCN1 TS-01894 c1ccc(cc1)C(=O)CC#N TS-01896 CC(C)c1ccc(cc1)C#N TS-01897 c1ccc2c(c1)ncc(n2)O TS-01898 C1[C@H](C(=O)CS1)C(=O)O TS-01899 Cc1cccc2c1CCC2=O TS-01900 Cc1ccc2c(c1)CCC2=O TS-01901 CC(C)(C#N)c1ccccn1 TS-01902 CC(C)c1ccnc(c1)C#N TS-01907 C1CSCCC1C(=O)O TS-01908 C1CC(CNC1)C#N.Cl TS-01909 c1cc(oc1)Br TS-01910 c1c[nH]nc1Br TS-01911 c1c([nH]cn1)Br TS-01912 c1ccnc(c1)C(F)(F)F TS-01913 c1cc2c(cc1C#N)OCO2 TS-01914 c1cc(cc(c1)C(=O)O)C#N TS-01915 c1ccc(c(c1)C#N)C(=O)O TS-01916 c1ccc2c(c1)c(ccn2)F TS-01917 c1cc2cc(ccc2nc1)F TS-01918 c1cc(ccc1CCO)C#N TS-01919 CN1c2ccccc2CC1=O TS-01920 Cc1cc(ccc1OC)C#N TS-01921 c1cc(ccc1CCC#N)O TS-01922 CCOc1ccc(cc1)C#N TS-01923 c1ccc(cc1)OCCC#N TS-01924 Cc1cc(cc(c1)OC)C#N TS-01925 Cc1ccc2c(c1)nc([nH]2)N TS-01926 Cc1cc(n2ccnc2n1)C TS-01927 Cc1cn2cc(ccc2n1)N TS-01928 C1CS[C@@H](CN1)C(=O)O TS-01930 C1CSCN[C@@H]1C(=O)O TS-01931 c1cc2c(c(c1)N)CCCC2 TS-01932 c1ccc(cc1)[C@H](C2CC2)N TS-01933 c1ccc(cc1)C2(CC2)CN TS-01934 c1cncnc1C(F)(F)F TS-01937 c1cc2c(cc1F)nccn2 TS-01938 c1ccc2c(c1)C[C@H]2C(=O)O TS-01939 COc1ccc2c(c1)cco2 TS-01940 Cc1cccc2c1COC2=O TS-01941 Cc1cccc2c1C(=O)OC2 TS-01942 Cc1cccc2c1[nH]c(=O)[nH]2 TS-01943 CCOc1ccc(cn1)C#N TS-01944 CCOc1cc(ccn1)C#N TS-01945 Cc1ccc(c2c1CCC2)O TS-01946 c1ccc2c(c1)CCC[C@@H]2O TS-01947 c1cc2c(c(c1)N)CCNC2 TS-01948 c1cc(cnc1)C2CCNC2 TS-01949 c1cc(ccc1C(=O)C#N)F TS-01950 Cc1cccc2c1[nH]c(=O)o2 TS-01951 Cc1c(cco1)C(=O)CC#N TS-01953 Cc1cc(=O)n2c([nH]1)ccn2 TS-01954 Cc1ccc(cc1F)CC#N TS-01955 c1cc(cc(c1)F)CCC#N TS-01956 c1ccc2c(c1)CC(C2N)O TS-01957 c1ccc2c(c1)[C@H](CCO2)N TS-01958 Cc1cccc(c1C(=O)N)C TS-01959 Cc1ccc(cc1C)C(=O)N TS-01960 CCC(=O)c1cccc(n1)C TS-01961 c1cc(ncc1N)N2CCC2 TS-01962 c1c(c([nH]n1)N)C2=CCCC2 TS-01963 c1cc(sc1)C2(CC2)C#N TS-01964 Cc1ccc(cc1)CCNC TS-01965 Cc1cc(c(c(c1)C)CN)C TS-01966 Cc1ccccc1CCNC TS-01967 Cc1cccc(c1)CCNC TS-01968 Cc1ccc(cc1)C(C)(C)N TS-01969 Cn1ccc(n1)C(F)(F)F TS-01970 COc1ccc2c(c1)non2 TS-01972 c1cc2c(cc1F)C(=O)CC2 TS-01973 c1ccc2c(c1)C(CC2O)O TS-01974 C[C@H](c1ccccc1)C(=O)O TS-01975 Cc1ccc(c(c1)O)C(=O)C TS-01976 Cc1ccc(cc1N)C(=O)N TS-01977 Cc1ccc(c(c1)N)C(=O)N TS-01978 CNC(=O)Cc1ccncc1 TS-01981 CNC(=O)Cc1cccnc1 TS-01982 Cc1c(cccn1)C(=O)NC TS-01983 CCN(C)c1ccc(cc1)N TS-01984 Cc1cc(sn1)N.Cl TS-01985 c1csc(n1)CN.Cl TS-01986 Cc1cc(ccc1C(=O)O)N TS-01987 c1cc2c(cc1N)COCO2 TS-01988 CC(=O)c1cc(ccc1O)N TS-01989 Cc1ccc(cc1C(=O)O)N TS-01990 c1cc(cc(c1)C(=O)O)CN TS-01991 Cc1c(cccn1)CC(=O)O TS-01992 COC(=O)c1ccc(cc1)N TS-01993 COC(=O)Cc1ccccn1 TS-01994 COC(=O)Cc1cccnc1 TS-01995 c1cc2c(cc1F)CCCN2 TS-01996 c1ccn(c1)c2nncs2 TS-01997 c1cc(c2c(c1)nsn2)N TS-01998 c1ccc(cc1)C[C@@H](CO)N TS-01999 CNCC(c1ccccc1)O TS-02000 COc1cccc(c1)CCN TS-02001 CC(c1ccc(cc1)OC)N TS-02002 CC(C)(C#N)c1cccs1 TS-02003 COC(=O)C1CNC1.Cl TS-02004 CNC1CCOCC1.Cl TS-02005 COC[C@H]1CCCN1.Cl TS-02006 c1c(oc(n1)N)C(F)(F)F TS-02007 c1(nc([nH]n1)N)C(F)(F)F TS-02008 c1cc(sc1)C(F)(F)F TS-02009 COC(=O)c1ccccc1O TS-02010 c1cc(ccc1CO)C(=O)O TS-02011 c1cc(cc(c1)C(=O)O)CO TS-02012 c1c(c(=O)[nH]c(=O)[nH]1)C2CC2 TS-02014 C1Cc2c(nc(nc2O)O)C1 TS-02015 CNc1cc(ccn1)C(=O)O TS-02016 Cc1c(ccc(n1)N)C(=O)O TS-02017 Cc1c(cnc(n1)C)C(=O)O TS-02018 Cc1cnc(cn1)C(=O)OC TS-02019 CCOC(=O)c1ccncn1 TS-02020 CCOC(=O)c1ncccn1 TS-02021 c1cc(nc(c1)C(=O)N)CO TS-02022 COc1cccc(n1)C(=O)N TS-02023 c1cc2c(cc1O)nsn2 TS-02024 CCCc1c(cccc1O)O TS-02025 CCCc1ccc(cc1O)O TS-02026 COCCc1ccc(cc1)O TS-02027 CCOc1cc(ccc1O)C TS-02028 c1c(n2c(n1)CCCC2)CO TS-02029 COc1cccc(n1)C(=O)O TS-02030 c1cc(nc(c1)C(=O)O)CO TS-02031 c1cc(ncc1C(=O)O)CO TS-02032 COC(=O)c1cnccc1O TS-02034 c1ccc(c(c1)CC(=O)N)F TS-02036 c1ccc(c(c1)C(=O)CN)F TS-02037 COc1ccc(c(c1)CO)N TS-02038 CCOC(=O)C1(CCC1)C#N TS-02039 Cn1cccc1CC(=O)OC TS-02040 CNCCc1ccc(cc1)F TS-02041 Cc1cc(ccc1CNC)F TS-02042 Cc1cccc(c1F)CNC TS-02043 Cc1ccc(c(c1)F)CNC TS-02044 Cc1ccc(c(c1)CNC)F TS-02045 Cc1cc(cc(c1CN)C)F TS-02046 C1CCC2C(C1)C(=O)CCN2 TS-02047 c1cc(c(cc1O)Cl)C#N TS-02048 c1c2c(cnc1Cl)cn[nH]2 TS-02049 c1c(c(nc(c1F)O)O)C#N TS-02050 c1cc(c(c(c1N)F)C#N)F TS-02051 c1cc(c(cc1F)N)C(=O)N TS-02052 COc1cccc(c1OC)O TS-02053 COc1ccc(cc1OC)O TS-02054 Cc1cc(nn1C)C(=O)OC TS-02055 CCCc1[nH]cc(n1)C(=O)O TS-02056 CCCc1[nH]c(cn1)C(=O)O TS-02057 CCOc1[nH]c(=O)cc(n1)C TS-02058 c1ccc2c(c1)cc(cn2)C#N TS-02059 c1ccc2cnc(cc2c1)C#N TS-02060 c1cscc1/C=C/C(=O)O TS-02061 c1cc2c(cc1Cl)non2 TS-02062 c1cncc2c1nc(o2)Cl TS-02063 COC(=O)c1cccnc1F TS-02064 COC(=O)c1ccc(cn1)F TS-02065 Cc1cc(on1)CC(=O)OC TS-02066 CCOC(=O)c1c(ocn1)C TS-02067 C1CC2=C(C1)SCC(=O)N2 TS-02068 Cc1ccc(cc1)[S@](=O)N TS-02069 c1ccnc(c1)SCCO TS-02070 C1CC(C1)N2CCC(CC2)O TS-02071 Cc1nc(cs1)C(C)(C)C TS-02072 C1COCC(=O)N1C2CNC2 TS-02073 Cc1cc(c(s1)C)C(=O)O TS-02074 C1CCC(CC1)CCC(=O)O TS-02075 CC(=O)N1CCC(CC1)NC TS-02076 CCCCC1(CCCCC1)O TS-02077 c1cncc(c1Cl)C(=O)N TS-02078 c1cc(nc(c1)Cl)C(=O)N TS-02079 c1c(cncc1Cl)C(=O)N TS-02080 Cc1cc(c(cc1C)Cl)O TS-02081 c1cc(cc(c1)Cl)CCO TS-02082 Cc1ccc(cc1Cl)OC TS-02083 CCc1cc(ccc1Cl)O TS-02084 CC(c1cccc(c1)N)(F)F TS-02085 CC(c1ccc(cc1)N)(F)F TS-02086 CC(c1ccccc1N)(F)F TS-02087 CNCc1cc(cc(c1)F)F TS-02088 CCc1nc(cs1)C(=O)O TS-02089 C1CC(CCC1CN)C(=O)O TS-02090 C[C@@H](C1CCNCC1)C(=O)O TS-02091 CCOC(=O)C1CCNCC1 TS-02094 CN1CCC(CC1)C(=O)OC TS-02095 CCOC(=O)[C@H]1CCN(C1)C TS-02096 Cc1ccc(cc1)C2(CC2)C#N TS-02097 c1cc(ccc1CC#N)C2CC2 TS-02098 c1cc(ccc1CO)C(F)F TS-02099 Cc1nc2cc(ccc2o1)C#N TS-02100 C1CC2(C1)OCC(CO2)CO TS-02101 COC1CCC(CC1)C(=O)O TS-02102 COC(=O)C1CCC(CC1)O TS-02103 CCOC(=O)C1CCCC1O TS-02104 CN(C)C(=O)[C@@H]1CNCCO1 TS-02105 Cc1ccc2cc(ccc2n1)N TS-02106 c1cc(ccc1C2(CC2)C#N)N TS-02107 c1ccnc(c1)C2(CCC2)C#N TS-02108 Cc1[nH]cc(n1)c2ccccc2 TS-02109 c1cnc(c(n1)C(=O)O)Cl TS-02110 C1CNC[C@H]1N.Cl.Cl TS-02111 CCOC(=O)[C@@H]1CNCCO1 TS-02112 COC(=O)C[C@H]1CNCCO1 TS-02113 c1cc2ccc(cc2c(c1)N)O TS-02114 c1cc(oc1)c2ccc(cc2)N TS-02115 c1ccc(c(c1)c2ccco2)N TS-02116 Cc1cc(c2ccccc2n1)O TS-02117 Cc1ccc2cc(ccc2n1)O TS-02118 c1ccc(cc1)CN2CC=CC2 TS-02119 COc1ccc(c(c1F)F)O TS-02120 Cc1ccc(cc1)C(F)(F)F TS-02121 C.C1C[C@@H]([C@H]1C(=O)O)C(=O)O TS-02122 c1ccc(cc1)Oc2ccoc2 TS-02123 Cc1ccc2ccc(=O)oc2c1 TS-02124 c1cc2cc[nH]c2c(c1)C(=O)N TS-02126 c1cc(cc(c1)n2cncn2)N TS-02127 c1cc(ncc1N)n2ccnc2 TS-02128 c1cc(cnc1)c2cc([nH]n2)N TS-02129 CC(C)(C#N)c1ccc(cc1)N TS-02131 CNCc1c[nH]c2c1cccc2 TS-02132 CNCc1ccc2c(c1)cc[nH]2 TS-02133 Cn1c(cc(n1)C(=O)O)Cl TS-02134 c1cc(c(cc1F)Cl)CO TS-02135 C1CCC(CC1)(C#N)N.Cl TS-02136 Cn1c(ccn1)Br TS-02137 Cc1ccnc(c1)C(F)(F)F TS-02138 c1ccc2c(c1)cc(c(=O)o2)N TS-02139 c1ccc2c(c1)cc(o2)C(=O)N TS-02140 c1ccc2c(c1)c(cc(=O)[nH]2)O TS-02141 COC(=O)c1ccc(cc1)C#N TS-02142 C#CCOC(=O)c1cccnc1 TS-02143 c1ccc2c(c1)c(n[nH]2)C(=O)N TS-02144 c1ccc(cc1)c2nc(no2)N TS-02145 c1cc2c(c[nH]c2nc1)C(=O)N TS-02146 Cc1ccc2c(c1)[nH]cc2CO TS-02147 Cc1cc(c(cc1OC)C)C#N TS-02148 Cc1cc(ccc1CC#N)OC TS-02149 Cn1c2ccccc2nc1CN TS-02151 COC(=O)[C@@H]1CSCCN1 TS-02152 c1ccc(cc1)C2(CCC2)CN TS-02153 c1c(c(n[nH]1)N)Br TS-02154 c1cc2c(c(c1)N)C(=O)NC2=O TS-02155 c1cc(c2nccn2c1)C(=O)O TS-02156 Cc1c(cc(cn1)C(=O)O)C#N TS-02157 COC(=O)c1ccc(cn1)C#N TS-02158 c1ccn(c1)c2cc(ccn2)F TS-02159 c1ccn(c1)c2ccc(cn2)F TS-02160 CC1(c2ccccc2C(=O)O1)C TS-02162 c1cc2c(c(c1)O)CC(=O)CC2 TS-02163 CCc1nc2c(cccc2o1)N TS-02164 Cn1ccc2c1ccnc2OC TS-02165 Cc1nnc(o1)Br TS-02166 c1cc2c(cc1C(=O)O)ocn2 TS-02167 c1cc(ncc1F)n2ccnc2 TS-02168 Cc1cccc2c1NC(=O)CO2 TS-02169 COc1ccccc1OCC#N TS-02170 COc1ccc(cc1)OCC#N TS-02171 c1cnc(cc1C(=O)O)C2CC2 TS-02172 Cc1nc2cccc(c2o1)CO TS-02173 COc1ccc(cc1OC)C#N TS-02174 COc1ccc2c(c1)nc([nH]2)N TS-02175 Cc1cc(=O)n2c([nH]1)cc(n2)C TS-02176 c1ccc(c(c1)N2CCCC2)O TS-02177 CC(=O)c1ccc(cc1)CCN TS-02178 CC(C)c1ccc(cc1)C(=O)N TS-02179 c1cc(ncc1N)N2CCCC2 TS-02180 c1cc(c(nc1)N2CCCC2)N TS-02181 c1c(c([nH]n1)N)C2=CCCCC2 TS-02182 c1cc(sc1)C2(CCC2)C#N TS-02183 Cc1cc(c(c(c1)C)CNC)C TS-02184 Cc1cc(nn1C)C(F)(F)F TS-02185 c1cc(oc1)c2cc(no2)CN TS-02187 Cc1cc(=O)oc2c1c(n[nH]2)C TS-02188 Cc1cc(cc2c1CCC2=O)F TS-02191 CC1(Cc2cccc(c2O1)O)C TS-02192 c1cc2c(cc1CCO)CCO2 TS-02193 Cc1ccccc1CCC(=O)O TS-02195 Cc1cccc(c1C)C(=O)OC TS-02196 c1cc(c(nc1)OC2CCC2)N TS-02197 c1ccc2c(c1)NC[C@@H](O2)CN TS-02198 CN(C)c1ccc(cc1)C(=O)N TS-02199 Cc1nc2ccc(cc2s1)N TS-02200 c1c(nc(s1)CC#N)C2CC2 TS-02201 CC(C)(C)c1cccc(c1)CO TS-02202 c1cncc(c1C(F)(F)F)F TS-02203 c1cc2c(cc1C(=O)N)OCO2 TS-02204 c1cc2c(cc1F)CCC(=O)N2 TS-02205 c1ccc(c(c1)OCCC#N)F TS-02206 Cc1ccc(cc1)C(=O)NOC TS-02207 Cc1ccc(c(c1)C(=O)OC)N TS-02208 Cc1cc(ccc1C(=O)OC)N TS-02209 Cc1ccc(cc1N)C(=O)OC TS-02210 c1cc2c(cc1N)OCCCO2 TS-02211 c1c2c(c([nH]1)C(=O)O)CCCC2 TS-02212 CN(C)c1cccc(c1)C(=O)O TS-02213 Cc1cccc(c1)[C@H](C(=O)O)N TS-02214 C[C@H](c1cccc(c1)N)C(=O)O TS-02215 CC(C)(c1ccccn1)C(=O)O TS-02216 CC(C)c1ccnc(c1)C(=O)O TS-02217 COC(=O)Cc1cccc(c1)N TS-02218 Cc1ccc(c(c1)NC(=O)C)O TS-02219 C[C@H]1CCc2cc(ccc2N1)F TS-02220 c1ccc(c(c1)CNC2CC2)F TS-02221 Cc1ccc2c(c1)[nH]c(=S)o2 TS-02222 Cc1cc(cc(c1O)C)CNC TS-02223 c1c(cn(n1)C2CCCCC2)N TS-02224 c1cnc2c(n1)cc(cn2)Cl TS-02225 C1CNCCC1C(=O)O.Cl TS-02226 c1cc2c(c(c1)F)OCCC2=O TS-02228 Cc1ccc(c(c1C)O)C(=O)O TS-02229 COc1ccccc1CC(=O)O TS-02230 c1cc(cc(c1)Cl)[C@H](C(=O)O)O TS-02231 Cc1ccc(c(c1)C(=O)O)OC TS-02232 COCc1cccc(c1)C(=O)O TS-02233 CN1CCN(c2c1c(=O)c2=O)C TS-02234 c1c(n2c(n1)CCCC2)C(=O)O TS-02235 c1cnccc1C(=O)NCCO TS-02236 c1ccc(c(c1)[C@H](C2CC2)O)F TS-02237 c1cc(ncc1F)N2CCCC2 TS-02238 COc1ccc2c(c1)nsn2 TS-02239 Cc1cc(=O)n2ccsc2n1 TS-02240 CC(C)(c1ccc(cc1)OC)O TS-02241 Cc1cn2ccc(cc2n1)Cl TS-02242 Cc1cn2cc(ccc2n1)Cl TS-02243 Cn1c2cccc(c2cn1)Cl TS-02244 CC(c1ccccc1C#N)(F)F TS-02245 CC(c1cccc(c1)C#N)(F)F TS-02246 CC(c1ccc(cc1)C#N)(F)F TS-02247 CCOc1cccc(n1)C(=O)O TS-02248 CCOc1cnccc1C(=O)O TS-02249 CCOc1ccc(cn1)C(=O)O TS-02250 CCOc1cc(ccn1)C(=O)O TS-02251 COc1cccc(c1CN)OC TS-02252 CCOC(=O)c1c(c(c[nH]1)C)C TS-02255 Cc1cc(c(n1C)C)C(=O)OC TS-02256 c1ccc2cc(ccc2c1)CC#N TS-02257 c1c(cn(n1)C2CCOCC2)N TS-02258 CC1(CC(CC(C1)(C)C#N)O)C TS-02259 CNCc1ccc(cc1)SC TS-02260 C[C@@H](c1ccc(cc1)SC)N TS-02261 C1COC(CN1)C(=O)O.Cl TS-02262 COc1cc(cc(c1)Cl)C#N TS-02263 c1cc2c(cc1N)c(n[nH]2)Cl TS-02264 c1cc2c(cc1N)[nH]nc2Cl TS-02265 Cc1cc(n2c(n1)ccn2)Cl TS-02266 Cc1cnc2n1nc(cc2)Cl TS-02267 c1cc(ccc1C2(CC2)N)Cl TS-02268 COC(=O)C1(CC1)C(F)(F)F TS-02269 c1c(csc1C(F)(F)F)O TS-02270 Cc1cc(=O)oc(c1C(=O)O)C TS-02271 COC(=O)c1c(cccc1O)O TS-02272 COC(=O)c1ccc(c(c1)O)O TS-02273 C1CC(CCC1C(F)(F)F)O TS-02274 COCC(=O)c1ccc(cc1)F TS-02275 CCOC(=O)c1cc(oc1C)C TS-02276 CCCc1ncc(n1C)C(=O)O TS-02277 CC(C)(C)c1c(c[nH]n1)C(=O)O TS-02278 CCCc1nc(cn1C)C(=O)O TS-02279 CCc1cc(nc(n1)COC)O TS-02280 c1ccn(c1)c2cccc(c2)C#N TS-02281 c1cc(sc1)C2(CC2)C(=O)O TS-02282 c1ccc(cc1)SCC(=O)O TS-02283 C[C@H]1CCc2c(sc(n2)N)C1 TS-02284 c1cc2c(cc1Cl)C(=O)OC2 TS-02285 c1cc2c(cc1Cl)nc(o2)N TS-02286 c1cc(ccc1CN)C#N.Cl TS-02287 c1cc(ccc1CC#N)N.Cl TS-02288 COC(=O)c1c(cccc1F)N TS-02289 CCOC(=O)c1cc(cnc1)F TS-02290 COc1ccc(c(c1)F)C(=O)N TS-02292 CC(C)(C)c1c(con1)C(=O)O TS-02293 CCOC(=O)c1c(oc(n1)C)C TS-02294 c1cc(cc(c1)c2ccco2)C#N TS-02295 c1cc(cc(c1)n2ccnc2)C#N TS-02296 CNCc1cc(ccc1OC)F TS-02297 CNCc1cccc(c1F)OC TS-02298 CNCc1ccc(cc1F)OC TS-02299 c1c(nc(s1)C2CC2)C(=O)O TS-02300 c1c(nc(s1)C(=O)O)C2CC2 TS-02301 CC(=O)C1CCN(CC1)C(=O)C TS-02302 c1cc2c(cc1Cl)onc2O TS-02303 c1cnc2ccsc2c1Cl TS-02304 c1cnc(c2c1scc2)Cl TS-02305 CNCCc1ccc(cc1)Cl TS-02306 c1ccc2c(c1)CC[C@H]2N.Cl TS-02307 CNCCc1ccccc1Cl TS-02308 CNCCc1cccc(c1)Cl TS-02309 c1cnc([nH]1)CN.Cl.Cl TS-02310 c1c(cc(c2c1C(=O)CO2)F)F TS-02311 COc1cc(cc(c1O)OC)O TS-02312 c1cc(oc1)c2cc(ccn2)C#N TS-02313 c1cc(ncc1C#N)n2ccnc2 TS-02314 CC(C)(c1cccs1)C(=O)O TS-02315 CNC1COCC1N2CCCC2 TS-02316 C1CC(OC1)CN2CCNCC2 TS-02317 c1cc(c(cc1C(=O)N)N)Cl TS-02318 c1cc(c(cc1Cl)N)C(=O)N TS-02319 CNC(=O)c1ccnc(c1)Cl TS-02320 c1ccc(cc1)CC(=N)N.Cl TS-02321 c1c(sc(n1)N)Cl.Cl TS-02322 c1cc(cc(c1)N)c2cncnc2 TS-02323 c1cc(cc(c1)N)c2ncccn2 TS-02324 c1cc(cnc1)c2ccnc(c2)N TS-02325 c1cnccc1c2ccnc(c2)N TS-02326 Cc1ccccc1S(=O)(=O)N TS-02327 CCOC(=O)c1c(scn1)C TS-02328 CCOC(=O)c1csnc1C TS-02329 CC(C)(C)CN1CC(C1)C(=O)O TS-02330 COC(=O)C1CCC(CC1)CN TS-02331 CCc1ccccc1n2cccc2 TS-02332 c1cc(c(c(c1)N)Cl)C(=O)O TS-02333 Cc1cc(cc(n1)Cl)C(=O)O TS-02334 Cc1cc(c(nc1)Cl)C(=O)O TS-02335 Cc1cc(nc(c1)Cl)C(=O)O TS-02336 c1cc(c(cc1Cl)O)C(=O)N TS-02339 CC(C)(c1ccc(nc1)Cl)O TS-02340 c1cc2cc(ccc2nc1)C(=O)N TS-02341 c1ccc2c(c1)ccc(n2)C(=O)N TS-02342 CCOc1ccsc1C(=O)O TS-02343 CC1CC(CC(O1)C)CC(=O)O TS-02344 CNCc1ccc2c(c1)cccn2 TS-02347 Cc1ccc(c(c1)C)c2cc[nH]n2 TS-02348 c1ccn(c1)c2cccc(c2)CN TS-02349 CNCc1cc2ccccc2nc1 TS-02350 CNCc1ccc2ccccc2n1 TS-02351 c1cc(cc(c1)N2CCCC2)C#N TS-02352 c1cc(ccc1C2(CCC2)C#N)N TS-02353 c1c(cc(cc1O)Cl)C(=O)O TS-02354 c1c(cnc(c1C(=O)O)Cl)N TS-02355 c1c(cnc(c1Cl)N)C(=O)O TS-02356 c1cc(nc(c1N)C(=O)O)Cl TS-02357 COC(=O)c1c(nccn1)Cl TS-02358 c1cc(ncc1C(=O)NO)Cl TS-02359 c1cncc(c1Br)N TS-02360 Cc1cnc(cn1)Br TS-02361 Cc1c(cncn1)Br TS-02362 C1CC(CNC1)N.Cl.Cl TS-02363 c1cc(c(c(c1N)F)C(=O)O)F TS-02364 c1c(c(cc(c1F)N)F)C(=O)O TS-02365 c1cc(c(c(c1N)C(=O)O)F)F TS-02366 c1ccnc(c1)C(C(=O)O)(F)F TS-02367 c1ccc2c(c1)c(ccn2)C(=O)O TS-02368 c1cc2c(cc1C(=O)N)nccn2 TS-02369 c1ccc2c(c1)ncc(n2)C(=O)N TS-02370 COc1cccc(c1)C2(CC2)C#N TS-02371 c1ccn(c1)c2ccc(cc2)CO TS-02372 COc1ccc(cc1)C2(CC2)C#N TS-02373 c1cc(cc(c1)[C@H](C2CC2)O)C#N TS-02374 Cc1cccc(c1n2cccc2)O TS-02375 Cc1ccnc2c1ccc(c2)OC TS-02376 Cc1ccnc(c1N)n2cccc2 TS-02377 c1ccc(cc1)Cn2ccc(n2)N TS-02378 CNCc1cnc2ccccc2n1 TS-02379 c1cc(ncc1C#N)N2CCCC2 TS-02380 c1cc(ncc1C#N)NC2CCC2 TS-02381 c1cnc(cc1C#N)NC2CCC2 TS-02382 c1cc(c(nc1)NC2CCC2)C#N TS-02383 c1cnc(cc1C#N)N2CCCC2 TS-02384 Cc1cnc(cn1)Cn2cccc2 TS-02385 Cc1cc(nc(n1)n2cccc2)C TS-02386 Cc1c(sc(n1)COC)CO TS-02387 c1c(cnc(c1Cl)O)C(=O)O TS-02388 Cc1ccncc1C(=O)O.Cl TS-02389 c1ccnc(c1)CC(=O)O.Cl TS-02390 COc1c(ccnc1CO)Cl TS-02391 c1cc2c(cc1F)CNC2.Cl TS-02392 CNCc1c(cccc1Cl)F TS-02393 c1cc(cc(c1)O)CCN.Cl TS-02394 c1ccc(cc1)[C@H](CN)O.Cl TS-02395 c1cnc(cc1Br)O TS-02396 c1cc(ncc1Br)O TS-02397 c1cnc(cc1O)Br TS-02398 C#CCn1ccc(n1)C(F)(F)F TS-02399 CC1=C(Cc2c1cccc2)C(=O)O TS-02400 c1cc2cc(ccc2cc1CO)O TS-02401 c1ccn(c1)c2c(cccc2O)N TS-02402 c1cc(cc(c1)n2cccn2)CO TS-02403 Cc1nc(co1)c2ccc(cc2)N TS-02404 c1cc(ccc1CN)c2cnco2 TS-02405 c1cc(ccc1CO)c2c[nH]cn2 TS-02406 c1cnc(cc1C#N)OCC2CC2 TS-02407 c1cc(ncc1C#N)OCC2CC2 TS-02408 c1cc(nc(c1)OCC2CC2)C#N TS-02409 c1cc(ccc1Cn2cncn2)N TS-02410 Cc1ccnc(c1N)n2ccnc2 TS-02411 Cn1c(cc(n1)c2cccnc2)N TS-02412 Cc1c(c2ccccc2[nH]1)CNC TS-02413 c1cnccc1OCCN.Cl TS-02414 c1cc(ccc1CC(F)(F)F)N TS-02415 CNc1ccccc1C(F)(F)F TS-02416 Cc1c[nH]c2c1cc(cc2)C(=O)O TS-02417 Cc1cc2ccc(cn2c1)C(=O)O TS-02418 Cc1ccc(c(c1)c2ccno2)O TS-02419 CC(=O)c1ccc2c(c1)CC(=O)N2 TS-02420 CNn1cnc2ccccc2c1=O TS-02421 CC(=O)Nc1ccc(cc1C#N)N TS-02422 c1ccc(cc1)N2C(=O)CC(=N2)N TS-02423 c1cc(ccc1C2(CCC2)C#N)F TS-02424 Cc1ccc(c(c1)N)C(=O)C2CC2 TS-02425 CC(C)(C#N)c1ccc(cc1)OC TS-02426 c1ccc(cc1)C2(CCC2)C(=O)N TS-02427 Cc1ccc(cc1)C2(CC2)C(=O)N TS-02428 Cc1c(n2ccccc2n1)CNC TS-02429 Cc1ccc(cc1C(F)(F)F)O TS-02431 COc1ccc2c(c1)ccc(=O)o2 TS-02433 Cc1[nH]c2ccc(cc2n1)C(=O)O TS-02434 Cc1cn2cc(ccc2n1)C(=O)O TS-02436 Cc1nc2cc(ccc2o1)C(=O)N TS-02437 c1ccc2c(c1)c(no2)CC(=O)N TS-02438 Cc1ccc(cc1)C2(CC2)C(=O)O TS-02439 COc1ccc(cc1)C(=O)C2CC2 TS-02440 CC(C)n1c2ccccc2[nH]c1=O TS-02441 c1ccc(cc1)Oc2ccsc2 TS-02443 c1cc(sc1)c2ccnc(c2)N TS-02444 C[C@H]1CNCCN1c2ccccc2 TS-02446 c1c(onc1Br)CN TS-02447 Cc1cscc1Br TS-02448 Cc1nc2cc(ccc2o1)C(=O)O TS-02449 COC(=O)c1cccc2c1ocn2 TS-02450 c1cc(ccc1c2cc(n[nH]2)N)F TS-02451 c1ccnc(c1)C2(CCC2)C(=O)O TS-02455 c1ccc2c(c1)[C@@H](CCN2)C(=O)O TS-02456 c1ccc2c(c1)CNC[C@H]2C(=O)O TS-02459 c1cc2c(cc1CC(=O)N)CCO2 TS-02461 c1ccc2c(c1)CC[C@H](O2)C(=O)N TS-02462 c1ccc2c(c1)cc(s2)C(=O)N TS-02463 CC(C)(C)c1cccc(c1)C(=O)N TS-02464 c1ccc(cc1)N2CC[C@@H](C2)CO TS-02465 CCCc1ccc(cc1)NC(=O)C TS-02466 CC(C)c1ccccc1NC(=O)C TS-02467 c1cc(ccc1N)N2CCNCC2 TS-02468 c1ccc(c(c1)N)N2CCNCC2 TS-02469 c1cnc(cc1N2CCCCC2)N TS-02470 c1cc(ncc1N)N2CCCCC2 TS-02471 c1cnc(cc1CN)N2CCCC2 TS-02472 CN1CCC=C(C1)C(=O)O.Cl TS-02473 c1ccc(c(c1)n2cccc2)Cl TS-02474 Cc1cc(c2ccccc2n1)Cl TS-02475 Cc1ccc(s1)CNC.Cl TS-02476 c1cc(c(cc1F)c2cc[nH]n2)O TS-02477 c1ccc2c(c1)CC[C@H](O2)C(=O)O TS-02478 c1ccc2c(c1)NCC(O2)C(=O)N TS-02479 CNCc1c[nH]c2c1cc(cc2)F TS-02480 CC(C)(C)c1cccc(c1)C(=O)O TS-02481 Cc1cc(c(c(c1)C)CC(=O)O)C TS-02482 CCOC(=O)c1c(cccc1C)C TS-02483 c1cc(ncc1N)OCC2CCC2 TS-02484 c1cc(c(nc1)OCC2CCC2)N TS-02485 c1cc(ncc1N2CCCC2)CO TS-02486 CC(C)(C)C(=O)Nc1ccncc1 TS-02487 Cc1ccnc(n1)N2CCNCC2 TS-02488 c1cnc(cc1N2CCNCC2)N TS-02489 c1c(cnc(n1)N2CCCCC2)N TS-02490 c1cnc(cn1)N2CCCNCC2 TS-02491 c1c(sc(n1)N)Br TS-02492 c1cc2n(c1)[C@@H](CCC2=O)C(=O)O TS-02493 CC(=O)c1cc2c(cc1N)OCO2 TS-02494 COc1cc(cc(c1O)OC)C#N TS-02495 c1csc2c1ncc(c2)C(=O)O TS-02496 CCOC(=O)c1c(cccc1N)C TS-02497 CC(C)(c1cccc(c1)N)C(=O)O TS-02498 C[C@H](c1cccc(c1)N)C(=O)OC TS-02499 CN(C)c1ccc(cc1)CC(=O)O TS-02500 c1cnc(cc1N2CCOCC2)N TS-02501 CS(=O)(=O)N1CCC(CC1)O TS-02502 Cc1cc(c(cc1OC)C)CNC TS-02503 CC(C)(CN)c1cccc(c1)OC TS-02504 c1cc(ccc1c2cnco2)Cl TS-02505 c1ccc2c(c1)c(cnc2Cl)O TS-02506 CN1CCC[C@@H](C1)C(=O)O.Cl TS-02507 COC(=O)C1CCNCC1.Cl TS-02508 c1cc(c(cc1O)Cl)N.Cl TS-02509 c1c(c(n[nH]1)C(F)(F)F)C(=O)O TS-02510 c1cc(c(c(c1)F)O)C(F)(F)F TS-02511 CCN1C(=O)CC(=N1)C(F)(F)F TS-02512 COC(=O)c1ccccc1C(=O)O TS-02513 CC(=O)c1ccc(c(c1)C(=O)O)O TS-02514 c1cc(ccc1C2(CC2)C(=O)O)F TS-02515 Cc1ccc(c(c1)C)OCC(=O)O TS-02516 Cc1cc(ccc1CC(=O)O)OC TS-02517 Cc1cc(cc(c1)OC)C(=O)OC TS-02518 Cc1cc(ccc1C(=O)OC)OC TS-02519 c1c(n2c(n1)CCCCC2)C(=O)O TS-02520 CCOC(=O)c1cnc(nc1C)C TS-02521 COc1cccc(c1)C/C(=N/O)/N TS-02522 Cc1ccc(cc1)OC/C(=N/O)/N TS-02523 c1ccc(cc1)c2ccnc(c2)C#N TS-02524 c1ccc(c(c1)[C@@H]2CNCCN2)F TS-02526 c1cc(ncc1F)N2CCCCC2 TS-02527 c1c(c(no1)C(F)(F)F)C(=O)O TS-02528 CC(C)(C#N)c1cccc(c1F)F TS-02529 CCOC(=O)c1ccc(c(c1)O)N TS-02530 COc1ccc(cc1N)C(=O)OC TS-02531 COc1ccc(cc1C(=O)OC)N TS-02532 c1cc(ncc1F)N2CCNCC2 TS-02533 C1CC(N(C1)C2CCC=C2)C(=O)O TS-02534 c1cc2c(cc1Cl)C(=O)CCN2 TS-02535 Cn1c2cccc(c2c(n1)N)Cl TS-02536 CCOC(=O)c1cccc(c1O)O TS-02537 C[C@@H](C(=O)O)Oc1ccc(cc1)O TS-02538 c1cc(ncc1F)N2CCOCC2 TS-02539 c1ccnc(c1)S(=O)(=O)CC#N TS-02540 CC(C)(C)OC(=O)N1CC(C1)C#N TS-02541 Cc1ccc(c(c1)n2cccc2)C#N TS-02542 c1cc(sc1)C2(CCC2)C(=O)O TS-02543 CCSc1ccc(cc1)C(=O)O TS-02544 Cc1nc2cc(c(cc2o1)N)Cl TS-02545 Cc1c(c(nc(c1Cl)C)O)C#N TS-02546 CCOC(=O)c1c(cccc1F)N TS-02547 CCOC(=O)c1ccc(c(c1)N)F TS-02548 CCOC(=O)c1ccc(cc1N)F TS-02549 c1cc(c(c(c1)F)CNC2CC2)F TS-02550 COc1ccc2ccccc2c1C#N TS-02551 c1cnn(c1)Cc2ccc(cc2)C#N TS-02552 Cc1nc2c(s1)CC[C@H]2C(=O)O TS-02553 CCSc1c(cccn1)C(=O)O TS-02554 CC(C)(C)OC(=O)NC1CC(=C)C1 TS-02555 CCOC1=CC[C@H](CC1)NC(=O)C TS-02556 CC(C)(C)OC(=O)N1CCC=CC1 TS-02557 c1ccc(cc1)Cc2ccc(cc2)N TS-02558 c1cc(nn2c1ncc2CO)Cl TS-02559 Cc1ccc(cc1NC(=O)C)Cl TS-02560 c1c(nc(cn1)Cl)N2CCCC2 TS-02561 c1cnc(c(n1)C#N)Br TS-02562 CCOC(=O)c1ccc(cc1O)F TS-02563 COC(=O)[C@@H](c1ccc(cc1)F)O TS-02564 C1C(CC12CC(C2)C(=O)O)C(=O)O TS-02566 COC(=O)C1CC=CCC1C(=O)O TS-02567 c1cc(ccc1Cn2cncn2)C#N TS-02568 c1ccc(cc1)n2cc(c(n2)N)C#N TS-02569 C[C@]1(CC(=O)CC(C1)(C)C)C(=O)O TS-02570 CCN(CC)C(=O)[C@H]1CCCNC1 TS-02572 CC(c1ccc(cc1)Cl)C(=O)O TS-02573 CCC(=O)c1ccc(cc1O)Cl TS-02574 CCC(=O)c1ccc(c(c1)Cl)O TS-02575 c1cc(cnc1)C(=O)c2cnccn2 TS-02576 c1ccnc(c1)c2cccc(c2)CO TS-02577 CC1(C=Cc2cc(ccc2O1)C#N)C TS-02578 Cc1cc(nc(n1)N)c2ccccc2 TS-02579 CC(C)(C)c1nc(cs1)C(=O)O TS-02580 CCOC(=O)c1c(nc(s1)C)C TS-02581 CC(C)NC(=O)CN1CCNCC1 TS-02582 c1c2c(cc(c1Cl)F)nc([nH]2)N TS-02583 CC(=O)Nc1ccc(cc1O)Cl TS-02584 Cc1cc(c(nc1)Cl)C(=O)OC TS-02586 CCOC(=O)c1ccnc(c1)Cl TS-02587 CCOC(=O)c1cnccc1Cl TS-02588 c1cc(cc(c1)Cl)OCC(=O)N TS-02589 CNCc1ccc(c(c1)Cl)OC TS-02590 CCc1cc(cnc1)Br TS-02591 c1cc(c2cn[nH]c2c1)C(F)(F)F TS-02592 c1cc2cn[nH]c2c(c1)C(F)(F)F TS-02593 CC(c1ccccc1C(=O)O)(F)F TS-02594 CC(c1cccc(c1)C(=O)O)(F)F TS-02595 CC(c1ccc(cc1)C(=O)O)(F)F TS-02596 CCOC(=O)c1c(cccc1F)F TS-02597 COC(=O)c1ccc(cc1)C(F)F TS-02598 c1cc(c(c(c1)F)C/C(=N/O)/N)F TS-02599 Cc1ccc(c2c1cccc2)C(=O)O TS-02600 c1ccc(cc1)Oc2c(cccn2)N TS-02601 c1cc(cc(c1)c2cncnc2)CO TS-02602 c1cc(ncc1C#N)OC2CC=CC2 TS-02603 c1cc(nc(c1)OC2CC=CC2)C#N TS-02604 c1cnc(cc1C#N)OC2CC=CC2 TS-02605 Cc1cc(nc(n1)N)c2cccnc2 TS-02606 Cc1cc(nc(n1)N)c2ccncc2 TS-02607 c1cc(sc1)c2cc(ccn2)C#N TS-02608 c1cc(sc1)c2ccc(cn2)C#N TS-02609 CC(C)(C)OC(=O)N1CCC(C1)N TS-02610 CC(C)(C)OC(=O)N1CCC[C@H]1N TS-02611 CN(C)C(=O)COC1CCNCC1 TS-02613 c1cc(cc(c1)N2CCCCC2)C#N TS-02614 c1cc(cc(c1)Cl)OCC(=O)O TS-02615 COC(=O)c1ccc(cc1O)Cl TS-02616 COC(=O)c1cc(cnc1N)Cl TS-02617 Cc1cc(ncc1N)Br TS-02618 c1cc(ncc1CN)Br TS-02619 C1CC(CNC1)CN.Cl.Cl TS-02620 Cc1cccnc1C(C(=O)O)(F)F TS-02621 Cc1ccc(nc1)C(C(=O)O)(F)F TS-02622 Cc1cccc(n1)C(C(=O)O)(F)F TS-02623 COC(=O)c1ccc(c(c1N)F)F TS-02624 COC(=O)c1cc(c(cc1N)F)F TS-02625 c1cc2c(cc1C(F)(F)F)NCC2 TS-02626 c1ccc(cc1)c2c[nH]cc2C(=O)O TS-02628 c1ccc2c(c1)ccc(n2)CC(=O)O TS-02629 COC(=O)c1cccc2c1cccn2 TS-02630 COC(=O)c1cc2ccccc2nc1 TS-02631 COC(=O)c1ccc2ccccc2n1 TS-02632 c1cc(cnc1)Oc2ccc(cn2)N TS-02633 c1cnn(c1)c2ccc(cc2)C(=O)N TS-02634 CC(C)(C)OC(=O)NC1CC(C1)O TS-02635 COc1cccc(c1)C2(CCC2)C#N TS-02637 CC(=O)CCc1c[nH]c2c1cccc2 TS-02638 COc1c(cc(cn1)C(=O)O)Cl TS-02639 COc1ccnc(c1C(=O)O)Cl TS-02640 c1cc2c(cc1F)CNCC2.Cl TS-02641 c1cnc(cc1CO)Br TS-02642 COC(=O)c1cc(cc(c1O)F)F TS-02643 c1cc(cc(c1)C(=O)O)c2ccn[nH]2 TS-02644 c1ccc(c(c1)C(=O)O)n2cccn2 TS-02645 c1cc(ccc1c2c[nH]nc2)C(=O)O TS-02646 c1cc(cnc1)c2c[nH]cc2C(=O)O TS-02647 c1ccc2c(c1)n(c(=O)o2)CCC#N TS-02648 COc1ccc2ccccc2c1CO TS-02649 CNCc1cc(on1)c2ccccc2 TS-02650 c1cnc(cc1C#N)OCC2CCC2 TS-02651 c1cc(ncc1C#N)OCC2CCC2 TS-02652 c1cc(nc(c1)OCC2CCC2)C#N TS-02653 c1cc(c(nc1)OCC2CCC2)C#N TS-02654 c1cc(nc(c1N)C#N)N2CCCC2 TS-02655 CNCc1ccc(nc1)n2ccnc2 TS-02656 c1cnc(cc1C#N)N2CCNCC2 TS-02657 CCOC(=O)[C@@H]1CSCCC1=O TS-02658 c1cc(c(cc1F)Cl)CC(=O)O TS-02659 c1cc(c(cc1F)CC(=O)O)Cl TS-02660 c1ccc2c(c1)cc(c(n2)Cl)C#N TS-02661 CC(=O)c1ccc(o1)Br TS-02662 c1cc(cc(c1)C(=O)O)c2cnco2 TS-02663 c1cc(nc(c1)C(=O)O)c2ccco2 TS-02664 c1cc(oc1)c2cc(ccn2)C(=O)O TS-02665 c1cc(oc1)c2cc(cnc2)C(=O)O TS-02666 c1cnc(cc1c2ccoc2)C(=O)O TS-02667 c1cc2ccc(nc2c(c1)O)C(=O)O TS-02668 CNCc1ccccc1C(F)(F)F TS-02669 Cn1ccc2c1ccc(c2)C(=O)OC TS-02670 CC(=O)c1ccc2c(c1)CC(=O)N2C TS-02671 c1ccc(c(c1)C2(CCCC2)C#N)F TS-02672 C[C@@H](Cc1ccc(cc1)F)N.Cl TS-02673 c1cc(ncc1Cl)SCCO TS-02674 CNCc1ccc(o1)Br TS-02675 Cc1c(cccc1C(F)(F)F)CO TS-02676 CNCc1ccc(nc1)C(F)(F)F TS-02677 c1ccc(cc1)C(=O)C2(CC2)C(=O)O TS-02678 COc1ccc2cc([nH]c2c1)C(=O)N TS-02679 c1ccc2c(c1)[nH]c(n2)CCC(=O)O TS-02680 CCOC(=O)c1cc(c(nc1)C)C#N TS-02681 COc1ccc2c(c1)c(c[nH]2)CCN TS-02682 CC(=O)N1CCNc2ccccc2C1 TS-02683 c1ccc(cc1)[C@H](C2CCCCC2)O TS-02684 CC(c1ccccc1)N2CCNCC2 TS-02685 COc1ccc(c(n1)OC)N.Cl TS-02688 C1CC1C(=O)N2CCNCC2.Cl TS-02689 c1c(cnc(c1N)Br)F TS-02690 c1c(cnc2c1C(=O)CCC2)C(=O)O TS-02691 Cc1nc2cccc(c2o1)C(=O)OC TS-02692 c1cc(c(c(c1)F)C#N)OC2CCC2 TS-02693 c1cc(cc(c1)N2CCCC2)C(=O)O TS-02694 c1ccc(cc1)N2CC[C@@H](C2)C(=O)O TS-02695 CN1CCc2c1ccc(c2)C(=O)OC TS-02696 COC(=O)c1cccc2c1CCCN2 TS-02697 COC(=O)c1ccc2c(c1)CCCN2 TS-02698 c1ccc(cc1)N2CC(CC2=O)CO TS-02699 c1cc2c(cc1N)N3CCN=C3S2 TS-02700 c1ccc(cc1)N2CCC(CC2)CO TS-02701 c1ccc(cc1)CN2CC[C@@H](C2)CO TS-02702 c1ccc(cc1)CN2CCC[C@@H](C2)O TS-02703 C[C@@]1(CCN(C1)Cc2ccccc2)O TS-02704 Cc1ccnc(c1N)N2CCCCC2 TS-02705 c1cnc(cc1CN)N2CCCCC2 TS-02706 c1c(onc1Br)C(=O)O TS-02707 Cc1c(c2ccc(cc2o1)O)C(=O)O TS-02708 COc1cccc(c1)C2(CC2)C(=O)O TS-02709 COc1ccc(cc1)C2(CC2)C(=O)O TS-02710 COC(=O)Cc1ccc2c(c1)CCO2 TS-02711 COC(=O)[C@@H]1CCc2ccccc2O1 TS-02712 CC(=O)c1ccc(c(c1O)CC=C)O TS-02713 c1cnc(cc1C(=O)O)N2CCCC2 TS-02714 c1cc(c(nc1)N2CCCC2)C(=O)O TS-02715 c1cc(ncc1C(=O)O)NC2CCC2 TS-02716 c1cnc(cc1C(=O)O)NC2CCC2 TS-02717 c1cc(c(nc1)NC2CCC2)C(=O)O TS-02718 c1cnc(cc1N2CCCC2)C(=O)O TS-02719 c1cc(cnc1)N2CC[C@@H](C2)C(=O)O TS-02721 CC(=O)Nc1ccccc1NC(=O)C TS-02722 c1cc2c(cc1F)CC[C@@]2(C3CC3)O TS-02723 c1ccc(cc1)Cc2c(nsn2)O TS-02724 CC1(CCc2cc(ccc2O1)CO)C TS-02725 c1cc(ncc1N)OC2CCCCC2 TS-02726 c1cc(c(nc1)OC2CCCCC2)N TS-02727 c1cc(c(nc1)N2CCCCC2)CO TS-02728 CC[C@H](C)NC(=O)c1ccccc1N TS-02729 Cc1cncc(n1)N2CCCNCC2 TS-02730 CNC1CCN(CC1)S(=O)(=O)C TS-02731 c1cc(c(cc1F)F)C(=N)N.Cl TS-02732 c1ccn(c1)Cc2ccc(c(c2)F)F TS-02733 c1cc(c(c(c1)F)C2(CCC2)C#N)F TS-02734 CC(=O)c1ccc(cc1O)NC(=O)C TS-02735 CC(=O)c1cc(ccc1O)NC(=O)C TS-02736 Cc1ccc2c(c1)O[C@@H](CN2)C(=O)O TS-02737 CC(=O)N[C@H](c1ccccc1)C(=O)O TS-02738 c1ccn(c1)c2c(ccs2)C(=O)O TS-02739 COC(=O)c1cc2c(ccs2)nc1 TS-02740 CC(C)(C)c1ccc(c(c1)N)C(=O)O TS-02741 CCOC(=O)c1c2c(c[nH]1)CCCC2 TS-02742 CCOC(=O)c1c2c(c([nH]1)C)CCC2 TS-02743 CC(C)(c1cccc(c1)N)C(=O)OC TS-02744 Cc1ccnc(c1N)N2CCOCC2 TS-02745 c1cc(nc(c1)N2CCOCC2)CN TS-02746 c1cc(nn2c1nc(c2)C3CC3)Cl TS-02747 c1ccc(cc1)c2c(c([nH]n2)N)Cl TS-02748 c1ccc(cc1)n2c(c(cn2)N)Cl TS-02749 CCOC(=O)[C@H]1CCCNC1.Cl TS-02750 CCOC(=O)[C@@H]1CCCCN1.Cl TS-02751 c1c(sc(n1)CO)Br TS-02752 Cc1cccc(c1C(=O)O)OC(=O)C TS-02753 COC(=O)c1cccc2c1OCCO2 TS-02754 Cc1cccc(c1OC(=O)C)C(=O)O TS-02755 CC(=O)c1ccc(c(c1)C(=O)OC)O TS-02756 c1cc(ccc1C2(CCC2)C(=O)O)F TS-02757 CCCc1cc(c(cc1O)O)C(=O)C TS-02758 c1cc(ncc1N)OC2CCOCC2 TS-02759 c1cc(c(nc1)OC2CCOCC2)N TS-02760 CC(C)(C)OC(=O)Nc1ccccn1 TS-02761 CC(C)(C)OC(=O)Nc1ccncc1 TS-02762 CC(C)(C)C(=O)Nc1ccncc1O TS-02763 Cc1ccc(cc1)c2ccnc(c2)C#N TS-02764 CNCc1ccc(o1)N2CCCCC2 TS-02765 c1cc(ncc1Cl)n2cc(cn2)N TS-02766 CNCc1c2ccccc2[nH]c1Cl TS-02767 c1ccc(c(c1)c2nnc(s2)N)F TS-02768 C1C[C@@H](C=C1)N2CCC(CC2)C(=O)O TS-02769 c1cc(ccc1c2nnc(o2)N)Cl TS-02770 CCOC(=O)[C@@H]1C[C@H](CN1)O.Cl TS-02771 c1ccc(c(c1)CC#N)Br TS-02772 CCOC(=O)c1c(cc(cc1O)O)C TS-02774 c1ccnc(c1)Oc2ccc(cc2)C#N TS-02775 c1ccc(cc1)Oc2cc(ccn2)C#N TS-02776 c1ccc(cc1)Oc2c(cccn2)C#N TS-02777 c1cc(ccc1C#N)Nc2cncnc2 TS-02778 CNCc1ccc(o1)N2CCOCC2 TS-02779 CC(C)(C)OC(=O)N1CCCC1C#N TS-02780 c1cc(c(cc1O)Cl)C(F)(F)F TS-02781 c1cn2cc(nc2cc1Cl)C(=O)O TS-02783 c1cc(ccc1C2CC2C(=O)O)Cl TS-02784 c1cc(ccc1C2(CC2)C(=O)O)Cl TS-02785 c1cc(cc(c1)Cl)C2(CC2)C(=O)O TS-02786 c1cnc(cc1Cl)N2CCCCC2 TS-02787 c1cc(ncc1Cl)N2CCCCC2 TS-02788 C(#N)c1c(nc([nH]1)Br)C#N TS-02789 c1nc(c(s1)C(F)(F)F)C(=O)O TS-02790 CC(=O)c1ccc(nc1)c2ccccc2 TS-02791 COc1ccc2cccc(c2c1)CC#N TS-02792 Cc1c(c(n(n1)c2ccccc2)C)C#N TS-02793 C1CCC(C1)N2CCC(CC2)C(=O)O TS-02794 C1CCC(CC1)N2CCC[C@H]2C(=O)O TS-02795 C1CCC(C1)NC2CCCC2C(=O)O TS-02796 c1cnc(cc1Cl)N2CCNCC2 TS-02797 c1c(nc(cn1)Cl)N2CCCCC2 TS-02798 c1cc2c(cc1C(F)(F)F)nccn2 TS-02799 c1cc(c(c(c1)F)C2(CC2)C(=O)O)F TS-02800 COC(=O)C1CC2(C1)CC(C2)C(=O)O TS-02801 c1ccc(cc1)c2ccccc2C(=O)O TS-02802 CC(=O)c1ccc(nc1)c2cccnc2 TS-02803 CC(=O)c1ccc(nc1)c2ccncc2 TS-02804 COc1cc(ccc1C(=O)O)SC TS-02805 C1CNCCC1C(=O)N2CCOCC2 TS-02806 Cc1cccc(n1)NCc2ccccc2 TS-02807 Cc1ccnc(c1)NCc2ccccc2 TS-02808 CCn1c(cc(n1)C(F)(F)F)Cl TS-02809 c1cc(cc(c1)Cl)C(=O)CC(=O)O TS-02810 CCC(=O)c1ccc(c(c1)Cl)OC TS-02811 c1cnc(cc1Cl)N2CCOCC2 TS-02812 c1cc(c(nc1)N2CCOCC2)Cl TS-02813 c1ccc(cc1)c2cc(cnc2)C(=O)O TS-02814 c1ccc(cc1)c2cnccc2C(=O)O TS-02815 C1C[C@H](N(C1)C2CCOCC2)C(=O)O TS-02816 CC(C)(C)N1C[C@H](CC1=O)C(=O)OC TS-02817 c1ccc(cc1)CNc2ccc(cc2)O TS-02818 C1CN(CCC1CO)C2CCOCC2 TS-02819 COC(=O)[C@@H](c1ccccc1Cl)N TS-02820 c1ccnc(c1)N2CCNCC2.Cl TS-02821 CC(c1ccc(cc1)Br)N TS-02822 c1ccc(c(c1)CCN)Br TS-02823 CC(C)(c1c(cccc1F)F)C(=O)O TS-02824 CC(C)(c1cccc(c1F)F)C(=O)O TS-02825 c1cc(ccc1c2cncnc2)C(=O)O TS-02826 c1cc(cc(c1)C(=O)O)c2cncnc2 TS-02827 c1cc(ccc1c2cnccn2)C(=O)O TS-02828 c1cc(cc(c1)C(=O)O)c2cnccn2 TS-02829 c1ccnc(c1)c2ccc(cn2)C(=O)O TS-02830 c1ccnc(c1)c2cc(ccn2)C(=O)O TS-02831 c1ccnc(c1)c2cccc(n2)C(=O)O TS-02832 c1cc(nc(c1)C(=O)O)c2cccnc2 TS-02833 c1cc(nc(c1)C(=O)O)c2ccncc2 TS-02834 c1ccnc(c1)c2c(cccn2)C(=O)O TS-02835 c1ccnc(c1)c2ccc(nc2)C(=O)O TS-02836 c1ccc(cc1)COc2ccc(cn2)N TS-02837 Cc1nc(cs1)c2ccc(cc2)C#N TS-02838 Cc1c(sc(n1)c2ccccc2)C#N TS-02839 CC(C)(C)OC(=O)N1CCCC(C1)N TS-02840 CC(C)(C)OC(=O)N(C)[C@H]1CCNC1 TS-02841 c1ccc(c(c1)C#N)NC2CCCCC2 TS-02843 CCOC(=O)c1ccc(c(c1)O)Cl TS-02844 CCOC(=O)c1cc(cnc1N)Cl TS-02845 c1ccc(c(c1)OC/C(=N/O)/N)Cl TS-02846 c1cc(cc(c1)Cl)OC/C(=N/O)/N TS-02847 Cc1cc(cc(c1Cl)C)OCCO TS-02848 c1cnc(cc1Br)C(=O)N TS-02850 CC(=O)c1ncc(cn1)Br TS-02851 Cc1cc(c(cc1C)Br)O TS-02852 Cc1cccc(c1Br)CO TS-02853 c1cc(cc(c1)Br)CCO TS-02854 Cc1ccc(cc1CO)Br TS-02855 Cc1cc(nc(c1N)C)Br TS-02856 CN1CCC(CC1)CN.Cl.Cl TS-02857 c1cc(cc(c1)[C@H](C(F)(F)F)O)C#N TS-02858 c1ccn(c1)c2ccc(cc2)CC(=O)O TS-02859 Cc1ccc(cc1)c2c[nH]cc2C(=O)O TS-02860 Cc1ccc2cc(ccc2n1)C(=O)OC TS-02861 CC(C)(C)OC(=O)N1CC[C@@H](C1)CO TS-02862 c1cc(ccc1CC#N)N2CCNCC2 TS-02864 CN1CCN(CC1)c2cccc(c2)C#N TS-02865 c1cc(cc(c1)F)[C@H]2CCNC2.Cl TS-02866 c1cc(c2nnc(n2c1)C(F)(F)F)N TS-02867 CC(=O)Cc1cccc(c1)C(F)(F)F TS-02868 COC(=O)c1ccccc1c2ccco2 TS-02869 COc1cc2ccccc2cc1C(=O)O TS-02870 COC(=O)c1ccc2cc(ccc2c1)O TS-02871 c1cnn(c1)c2ccc(cc2)CC(=O)O TS-02872 c1cc(ccc1C#N)N2CC(C2)C(=O)O TS-02873 COC(=O)Cc1ccc2c(c1)nccn2 TS-02874 c1ccc(c(c1)CN2CCOCC2)C#N TS-02876 c1cnc(cc1C#N)OC2CCCCC2 TS-02877 c1cc(nc(c1N)C#N)N2CCCCC2 TS-02878 CN1CCN(CC1)c2cc(ccn2)C#N TS-02879 CN1CCN(CC1)c2cccc(n2)C#N TS-02880 CN1CCN(CC1)c2ccc(cn2)C#N TS-02881 c1c(cnc(n1)C(=O)O)Br TS-02882 COc1cc(ccc1Br)O TS-02883 c1cc([nH]c1C(F)(F)F)C(F)(F)F TS-02884 COc1cccc(n1)C(C(=O)O)(F)F TS-02885 c1cc2c(cc1C(F)(F)F)OCCN2 TS-02886 Cc1c(nc(o1)c2ccccc2)C(=O)O TS-02887 Cc1nc(c(o1)C(=O)O)c2ccccc2 TS-02888 Cc1c(c(c2ccccc2n1)C(=O)O)O TS-02889 CC(C)(c1ccc(cc1)C(F)(F)F)N TS-02890 COc1cc(cc(c1)OC)n2cccc2 TS-02891 c1cc2c(nc1)n(c(=O)[nH]2)C3CCCC3 TS-02892 C.CC(OC(=O)N[C@H]1C[C@@H](C1)O)(C)C TS-02893 c1cc2c(c(c1)F)OCC[C@@H]2N.Cl TS-02895 COc1ccc(c(c1)OC)CN.Cl TS-02896 c1cc(ccc1CC(F)(F)F)C(=O)O TS-02897 c1ccc(cc1)Oc2cc(oc2)C(=O)O TS-02898 c1cc(cc(c1)F)Oc2c(cccn2)N TS-02899 c1cnc(cc1C#N)OC2CCOCC2 TS-02900 c1cc(ccc1c2ccsc2)C(=O)O TS-02901 Cc1ccc(cc1)C2(CCCC2)C(=O)O TS-02902 c1ccc(cc1)C2(CCCCC2)C(=O)O TS-02903 CC(=O)c1ccc(cc1)N2CCNCC2 TS-02904 CN1CCN(CC1)c2ccccc2C=O TS-02905 CNCc1ccc(s1)c2ccccn2 TS-02906 Cc1c(sc(n1)c2ccccc2)CN TS-02907 c1cc(c(cc1F)Cl)OCC(=O)O TS-02908 c1c(nc(s1)N2CCOCC2)Cl TS-02909 CC(C)C(C#N)N1CCOCC1.Cl TS-02910 Cc1cc(cc(c1C(=O)O)Cl)Cl TS-02913 c1cc(c(cc1C(=O)O)N)C(F)(F)F TS-02914 COC(=O)c1cc(cnc1)C(F)(F)F TS-02915 Cc1ccc(cc1CN)OC(F)(F)F TS-02916 c1cnc(cc1C(=O)O)OC2CC=CC2 TS-02917 c1cc(ncc1C(=O)O)OC2CC=CC2 TS-02918 c1cc(nc(c1)OC2CC=CC2)C(=O)O TS-02919 COc1cc2cc[nH]c(=O)c2cc1OC TS-02920 CC[C@H]1C(=O)NC(=O)c2ccccc2O1 TS-02921 CC(C)(C(=O)O)Oc1ccc(cc1)C#N TS-02922 Cc1ccc(cc1)NC(=O)/C=C/C(=O)O TS-02923 CNCc1c(c[nH]n1)c2ccc(cc2)F TS-02924 c1cc(sc1)c2cc(cnc2)C(=O)O TS-02925 c1cc(nc(c1)C(=O)O)c2cccs2 TS-02926 c1cc(sc1)c2cc(ccn2)C(=O)O TS-02927 c1cc(cnc1)c2ccc(s2)C(=O)O TS-02928 c1cc(sc1c2ccncc2)C(=O)O TS-02929 c1ccc(cc1)c2c(ncs2)C(=O)O TS-02931 c1cc(cc(c1)C(=O)O)CN2CCCC2 TS-02932 c1ccc(c(c1)CN2CCCC2)C(=O)O TS-02933 c1ccc(cc1)CN2CC[C@@H](C2)C(=O)O TS-02936 c1ccc(cc1)NC2CCCC2C(=O)O TS-02937 c1ccc(cc1)CN2C[C@H](CC2=O)CO TS-02938 CC1(CCc2cc(ccc2O1)CNC)C TS-02939 CN1CCN(CC1)c2cccc(c2)CN TS-02940 CNCc1ccnc(c1)N2CCCCC2 TS-02941 CCOC(=O)c1c(nc(s1)Cl)C TS-02942 C1COCCN1c2c(nsn2)Cl TS-02943 C1CC2(CCCN2C1)CC(=O)O.Cl TS-02944 c1c(cc(c(c1Cl)O)Cl)C(=O)N TS-02945 CNCc1c(ccs1)Br TS-02946 CNCc1cc(cs1)Br TS-02947 c1cc(cc(c1)F)c2c(c[nH]n2)C(=O)O TS-02948 Cc1ccc(c2c1CCC2)OCC(=O)O TS-02949 COc1cccc(c1)C2(CCC2)C(=O)O TS-02950 c1cnc(cc1N2CCCCC2)C(=O)O TS-02951 c1cc(cnc1)N2CCC(CC2)C(=O)O TS-02952 c1cc(cnc1)CN2CC[C@@H](C2)C(=O)O TS-02953 Cc1c(ccc(n1)Br)Cl TS-02955 Cc1cc(c(nc1)Br)Cl TS-02956 c1cc(c(c(c1)Br)N)Cl TS-02957 COc1ccc(cc1N)OC(F)(F)F TS-02958 CCOC(=O)[C@@H]1CCC(=O)c2n1ccc2 TS-02959 CN1CCN(CC1)c2c(cccn2)CO TS-02960 c1cc(sc1)Sc2ccc(cc2)N TS-02961 c1c(c(c(cn1)Br)Cl)N TS-02962 c1c(cnc(c1N)Br)Cl TS-02963 c1c(cnc(c1Cl)N)Br TS-02964 c1ccc2c(c1)c(cc(n2)Cl)C(=O)O TS-02965 Cc1c(c(nn1C)C(=O)O)C(F)(F)F TS-02966 c1cc(cc(c1)F)C2(CCCC2)C(=O)O TS-02968 c1cc(ncc1N)OCC2CCOCC2 TS-02969 c1cc(ncc1N)OC[C@H]2CCCCO2 TS-02970 c1cc(c(nc1)OC[C@H]2CCCCO2)N TS-02971 c1cc(c(nc1)OCC2CCOCC2)N TS-02972 CC(=O)N[C@H]1CCC(=CC1)N2CCCC2 TS-02973 c1c(cnc(c1Br)O)Cl TS-02974 c1c(cnc(c1Cl)O)Br TS-02975 CC(C)(C)OC(=O)NC1CNC1.Cl TS-02976 c1cc2cncc(c2nc1)Br TS-02977 c1c(cnc(c1F)C(=O)O)C(F)(F)F TS-02978 c1cc(c(cc1OC(F)(F)F)CN)F TS-02979 c1c(cc(cc1OC(F)(F)F)F)CN TS-02980 c1cc(ccc1NC(=O)/C=C/C(=O)O)F TS-02981 c1cc(ccc1N2CC[C@@H](C2)C(=O)O)F TS-02982 c1cc2cnccc2c(c1)S(=O)(=O)O TS-02984 c1cc(oc1)CN2CCC(CC2)C(=O)O TS-02985 c1cocc1CN2CCC(CC2)C(=O)O TS-02986 c1cc(ccc1CCC#N)Br TS-02987 Cc1cc(cc(c1Br)C)C#N TS-02988 c1cc(c(c(c1)F)C(=O)O)OC2CCC2 TS-02989 COC(=O)C1CCc2cc(ccc2O1)F TS-02990 CC(C)(C)OC(=O)N1CCCCC1C#N TS-02991 C1CCCN(CC1)C(=O)[C@H]2CCCNC2 TS-02993 c1cc(c(c(c1)C(F)(F)F)Cl)CO TS-02994 Cc1c(n2c(n1)cccc2Cl)C(=O)O TS-02996 c1cn2cc(nc2cc1Cl)CC(=O)O TS-02997 c1cc2nc(cn2c(c1)Cl)CC(=O)O TS-02998 c1cnc(cc1Cl)C(=O)N2CCCC2 TS-02999 c1cc(ccc1C2(CCCC2)CO)Cl TS-03000 Cc1ccc2c(c1)[nH]cc2CCN.Cl TS-03001 c1cc(cc(c1)Cl)CN2CCNCC2 TS-03002 c1cc(c(cc1CC#N)Br)N TS-03003 Cc1cn2cc(ccc2n1)Br TS-03004 Cc1ccn2c(c1)ncc2Br TS-03005 c1c(nc(s1)C(F)(F)F)CC(=O)O TS-03006 c1ccc(cc1)S(=O)(=O)[C@H]2CC(=O)N2 TS-03007 Cc1ccc(cc1)c2ccc(cn2)C(=O)C TS-03010 Cc1cccc(c1)c2ccc(cn2)C(=O)C TS-03011 CS(=O)(=O)Nc1ccc2c(c1)CCC2 TS-03012 CCOC(=O)[C@@H]1CCc2c1nc(s2)C TS-03013 C1CCC(CC1)N2CCC(CC2)C(=O)O TS-03015 C1CCC(CC1)NC2CCCC2C(=O)O TS-03016 C1CCN(CC1)C2(CCNCC2)C(=O)N TS-03017 c1cc(cc(c1)Cl)N2CC[C@@H](C2)CO TS-03018 c1cc(ncc1Cl)N2CCCNCC2 TS-03019 Cc1ccccc1C2CCNCC2.Cl TS-03020 c1cc2c(cc1N)c(n[nH]2)Br TS-03021 c1cc2ncc(n2cc1Br)N TS-03022 c1cc2c(c(c1)Br)c(n[nH]2)N TS-03023 c1cc(sc1)C2(CCOCC2)C(=O)O TS-03025 C[C@@]1(c2ccsc2CCO1)CC(=O)O TS-03026 CN1CCC(CC1)N2CCC[C@H]2C(=O)O TS-03027 C1CC(CNC1)C(=O)N2CCC(CC2)O TS-03028 c1ccc(cc1)CN2CCNCC2.Cl TS-03029 c1ccc(cc1)c2ccc(c(c2)N)C(=O)O TS-03030 Cc1ccc(cc1)c2cccc(n2)C(=O)O TS-03031 Cc1cccc(c1)c2cccc(n2)C(=O)O TS-03032 Cc1ccccc1c2cccc(n2)C(=O)O TS-03033 Cc1ccc(cc1)c2cc(ccn2)C(=O)O TS-03034 Cc1cccc(c1)c2cc(ccn2)C(=O)O TS-03035 Cc1ccccc1c2cc(ccn2)C(=O)O TS-03036 Cc1ccc(cc1)c2ccnc(c2)C(=O)O TS-03037 Cc1cccc(c1)c2ccnc(c2)C(=O)O TS-03038 Cc1ccccc1c2ccnc(c2)C(=O)O TS-03039 Cc1ccc(cc1)c2ccc(cn2)C(=O)O TS-03040 Cc1cccc(c1)c2ccc(cn2)C(=O)O TS-03041 Cc1ccccc1c2ccc(cn2)C(=O)O TS-03042 Cc1cc(n(n1)C)Oc2ccc(cc2)C#N TS-03043 C1CN(CCC1C(=O)O)C2CCOCC2 TS-03045 C1C[C@H](N(C1)C2CCC(CC2)O)C(=O)O TS-03046 c1ccc2c(c1)CCC[C@@H]2Nc3c[nH]nc3 TS-03048 c1ccc2c(c1)CCN[C@H]2C(=O)O.Cl TS-03050 c1cc(ccc1C2=CCNCC2)F.Cl TS-03052 c1cc2n[nH]c(=O)n2cc1Br TS-03053 CC(=O)c1ccc(c(c1)Br)N TS-03054 c1cc(ccc1CC(=O)N)Br TS-03055 Cc1cccc(c1Br)C(=O)N TS-03056 CNCCc1ccc(cc1)Br TS-03057 Cc1cccc(c1Br)CNC TS-03058 CNCCc1cccc(c1)Br TS-03059 c1ccc(cc1)Oc2cccc(c2)C(=O)O TS-03060 c1ccc(cc1)Oc2c(cccn2)C(=O)N TS-03061 CC(C)(C)OC(=O)N(C)[C@H]1CCCNC1 TS-03062 CC(C)(C)OC(=O)N1CCCC[C@@H]1CN TS-03063 CC[C@H]1CN(CCN1)C(=O)OC(C)(C)C TS-03065 Cc1cc(ccc1OC(C)C(=O)O)Cl TS-03067 c1cc2c(c(c1)Br)nsn2 TS-03068 Cn1c2ccc(cc2c(n1)N)C(F)(F)F TS-03069 c1ccc(cc1)Oc2cc(ccn2)C(=O)O TS-03070 c1cc(ccc1C2(CC2)CN)C(F)(F)F TS-03071 CC(=O)c1ccc(nc1)c2ccc(cc2)F TS-03072 CC(=O)c1ccc(nc1)c2cccc(c2)F TS-03073 CN1CCC(CC1)Nc2ccccc2C#N TS-03074 c1cnc(cc1C#N)NCC2CCCCC2 TS-03075 c1cc(ncc1C#N)NCC2CCCCC2 TS-03076 c1cc(nc(c1)NCC2CCCCC2)C#N TS-03077 c1cc(c(nc1)NCC2CCCCC2)C#N TS-03078 COc1ccc(c(c1OC)Cl)C(=O)N TS-03079 c1cc(c(c(c1)N)Br)C(=O)O TS-03080 c1cc(c(cc1C(=O)O)Br)N TS-03081 c1cc(c(cc1C(=O)O)N)Br TS-03082 c1c(cnc2c1nsn2)Br TS-03083 COc1ccc2cccc(c2c1)CC(=O)O TS-03084 CCOc1ccc2ccccc2c1C(=O)O TS-03085 CCOC(=O)c1ccc2cc(ccc2c1)O TS-03086 COc1ccc2cc(ccc2c1)C(=O)OC TS-03087 COC(=O)C1CN(C1)c2ccc(cc2)C#N TS-03088 c1ccc(cc1)CN2CCC(CC2)(C#N)O TS-03089 C[C@H]1CN(N(C1=O)CC=C)c2ccccc2 TS-03090 COc1ccc(c(c1OC)Cl)C(=O)O TS-03091 COc1cc(c(cc1OC)Cl)C(=O)O TS-03092 c1c(c(c(cn1)Br)C(=O)O)N TS-03094 COC(=O)c1c(nccn1)Br TS-03095 c1cc(nnc1C(F)(F)F)N2CCCC2 TS-03097 c1cc(nc(c1)C(=O)O)c2ccc(cc2)F TS-03098 c1cc(cc(c1)F)c2cccc(n2)C(=O)O TS-03099 c1ccc(c(c1)c2cccc(n2)C(=O)O)F TS-03100 c1cc(ccc1c2cc(ccn2)C(=O)O)F TS-03101 c1cc(cc(c1)F)c2cc(ccn2)C(=O)O TS-03102 c1ccc(c(c1)c2cc(ccn2)C(=O)O)F TS-03103 c1cc(ccc1c2ccnc(c2)C(=O)O)F TS-03104 c1cc(cc(c1)F)c2ccnc(c2)C(=O)O TS-03105 c1ccc(c(c1)c2ccnc(c2)C(=O)O)F TS-03106 c1cc(ccc1c2ccc(cn2)C(=O)O)F TS-03107 c1cc(cc(c1)F)c2ccc(cn2)C(=O)O TS-03108 c1ccc(c(c1)c2ccc(cn2)C(=O)O)F TS-03109 Cc1c(c(on1)C)c2ccc(cc2)C(=O)O TS-03110 Cc1c(nc(o1)c2ccccc2)C(=O)OC TS-03111 Cc1c(c(c2ccccc2n1)C(=O)OC)O TS-03112 CC(C)(CN)c1ccc(cc1)C(F)(F)F TS-03113 CC(=O)c1c(cc(s1)c2ccccc2)N TS-03114 CC(=O)c1ccc(cc1)N2CCCCCC2 TS-03115 CNC(=O)COc1ccc(cc1Cl)F TS-03116 c1c(cc(cc1F)Br)C(=O)N TS-03117 Cc1c(c([nH]c1C(=O)O)C)Br TS-03118 CNCc1c(cccc1Br)F TS-03119 CNCc1cccc(c1F)Br TS-03120 Cc1cc(cc(c1NC(=O)C)Cl)Cl TS-03121 c1cc(ccc1C/C(=N/O)/N)C(F)(F)F TS-03122 COc1ccc(cc1)c2ccc(o2)C(=O)O TS-03123 c1cc(ccc1C(=O)O)O[C@H]2CCCC=C2 TS-03124 COc1ccc(c(c1)C#N)N2CCOCC2 TS-03125 c1cnc(cc1C#N)OC[C@H]2CCCCO2 TS-03126 c1cc(ncc1C#N)OC[C@H]2CCCCO2 TS-03127 c1cc(nc(c1)OC[C@H]2CCCCO2)C#N TS-03128 CC(C)(C)c1cc(nc(n1)N)C(F)(F)F TS-03129 Cc1c(c2cc(ccc2[nH]1)OC)CC(=O)O TS-03131 CC(=O)N1Cc2ccccc2C[C@H]1C(=O)O TS-03132 c1ccc(cc1)N2[C@H](CCC2=O)CC(=O)O TS-03133 CC1(Cc2c(cc(cn2)C(=O)O)C(=O)C1)C TS-03134 COC(=O)[C@H]1CC(=O)N(C1)c2ccccc2 TS-03135 COC(=O)[C@@H]1CCC(=O)N1c2ccccc2 TS-03136 CCOC(=O)c1cc2c(nc1)CCCC2=O TS-03137 Cc1nc(cs1)c2ccccc2C(=O)O TS-03138 c1ccc(cc1)c2csc(n2)CC(=O)O TS-03139 COC(=O)c1csc(n1)c2ccccc2 TS-03140 c1cc(ccc1CN2CCCCC2)C(=O)O TS-03141 c1cc(cc(c1)C(=O)O)CN2CCCCC2 TS-03142 c1ccc(c(c1)C(=O)O)NC2CCCCC2 TS-03143 c1ccc(c(c1)CN2CCCCC2)C(=O)O TS-03144 CN1CCN(CC1)c2ccc(cc2)C(=O)N TS-03145 c1ccc(cc1)CNc2cncc(n2)Cl TS-03146 c1ccc2c(c1)[nH]c(n2)CN.Cl.Cl TS-03147 c1ccc(cc1)COC(=O)N2CC[C@@H](C2)N TS-03148 c1cc(ccc1CN2CCNCC2)C(=O)O TS-03149 c1ccnc(c1)CN2CCC(CC2)C(=O)O TS-03150 c1cc(cnc1)CN2CCC(CC2)C(=O)O TS-03151 c1ccc(cc1)CN2CC[C@](C2)(C(=O)O)N TS-03152 COC(=O)c1cc(ccn1)N2CCCCC2 TS-03153 c1c(cc(c2c1[nH]cn2)Cl)C(F)(F)F TS-03154 CS(=O)(=O)c1ccc(c(c1)Cl)CO TS-03155 COC(=O)c1cc(c(c(c1)Cl)O)Cl TS-03156 c1c2c(c(s1)Br)OCCO2 TS-03157 C[C@@H](CO)Oc1ccc(cc1Cl)Cl TS-03158 c1cc(ccc1OCC(=N)N)Cl.Cl TS-03159 c1ccc(c(c1)OCC(=N)N)Cl.Cl TS-03160 c1cc(c(c(c1)OC(F)(F)F)C(=O)O)N TS-03161 c1cc(ccc1CC(=O)O)N2CCOCC2 TS-03162 c1cc(cc(c1)C(=O)O)CN2CCOCC2 TS-03163 c1ccc(cc1)[C@H](C(=O)O)N2CCOCC2 TS-03164 c1ccc(c(c1)CN2CCOCC2)C(=O)O TS-03165 c1cnc(cc1C(=O)O)OC2CCCCC2 TS-03166 c1cc(ncc1C(=O)O)OC2CCCCC2 TS-03167 c1cc(nc(c1)OC2CCCCC2)C(=O)O TS-03168 c1cc(c(nc1)OC2CCCCC2)C(=O)O TS-03169 c1ccc(cc1)CN2CCOC(C2)C(=O)O TS-03170 COc1ccc(cc1)N2CC[C@@H](C2)C(=O)O TS-03171 COc1cccc(c1)N2CC[C@@H](C2)C(=O)O TS-03172 c1cc(c(cc1Br)CO)Cl TS-03173 c1cc(nn2c1nc(c2)C(F)(F)F)Cl TS-03174 c1cc(ccc1C2(CC2)C#N)Br TS-03176 c1cc(cc(c1)Br)C2(CC2)C#N TS-03177 c1ccn(c1)c2cccc(c2)S(=O)(=O)N TS-03178 c1ccc(c(c1)CN)Br.Cl TS-03179 COC(=O)c1ccc2c(c1)c(ncn2)Cl TS-03180 COC(=O)c1ccc2c(c1)ncnc2Cl TS-03181 c1cc(c2ccncc2c1N)Br TS-03182 c1cc(cc(c1)Br)c2c[nH]nc2 TS-03183 c1cc(cc(c1)Br)c2ccn[nH]2 TS-03184 c1ccc(cc1)c2cc([nH]n2)Br TS-03185 Cc1cc2c(cc1Br)nccn2 TS-03186 c1ccc2c(c1)[nH]c(=O)c(n2)c3ccccn3 TS-03190 c1cc(ccc1CN2CC[C@@H](C2)C(=O)O)F TS-03191 c1cc(cc(c1)F)CN2CC[C@@H](C2)C(=O)O TS-03192 c1ccc(c(c1)CN2CC[C@@H](C2)C(=O)O)F TS-03193 c1ccc(cc1)/C=C/C(=O)c2cccc(c2)N TS-03194 c1cn2ccnc2nc1C(F)(F)F.Cl TS-03195 c1cc(cc(c1)Br)c2ncco2 TS-03196 c1cnc(cc1Br)n2ccnc2 TS-03197 c1ccn(c1)c2cnc(cn2)Br TS-03198 c1cc2c(c(c1N)Br)nccn2 TS-03199 c1cc(ccc1CN2CCOC[C@@H]2CN)F TS-03200 CC(C)(C)c1csc(n1)C2CCNCC2 TS-03201 c1cc(c(cc1C(F)(F)F)Cl)C(=O)O TS-03202 CCOC(=O)c1cn2c(n1)cccc2Cl TS-03203 CCOC(=O)c1cn2ccc(cc2n1)Cl TS-03204 c1cc(ccc1C2(CCCC2)C(=O)O)Cl TS-03205 c1cc(ccc1CN2CCCNCC2)Cl TS-03206 c1cc(cc(c1)Cl)CN2CCCNCC2 TS-03207 Cc1nc(c(s1)C(=O)OC)C(F)(F)F TS-03208 c1cc(ccc1C2(CCC2)C#N)C(F)(F)F TS-03209 c1ccc(cc1)Oc2cccc3c2c(n[nH]3)N TS-03210 COC(=O)[C@H]1CC(=O)N(C1)C2CCCCC2 TS-03211 c1cc(sc1)CN2CCC(CC2)C(=O)O TS-03212 c1cscc1CN2CCC(CC2)C(=O)O TS-03213 c1ccc(cc1)CN2CCS(=O)(=O)CC2 TS-03214 c1c(c(cnc1C(F)(F)F)Cl)C(=O)O TS-03215 c1cc(ccc1N2CC[C@@H](C2)C(=O)O)Cl TS-03216 c1cc(cc(c1)Cl)N2CC[C@@H](C2)C(=O)O TS-03217 CN1c2ccc(cc2CC1=O)Br TS-03218 c1cc(nc(c1)Br)C(=O)C2CC2 TS-03219 Cc1cc(n2c(cnc2n1)Br)C TS-03220 c1ccc2c(c1)nc(s2)c3ccc(cc3)N TS-03221 CN1CCC(CC1)N2CCC(CC2)C(=O)O TS-03222 CC1CN(CCC1N2CCCC2C(=O)O)C TS-03223 c1ccc(cc1)CN2CC[C@@H](C2)n3cccc3 TS-03224 COc1ccc2c(c1)c(c[nH]2)CCN.Cl TS-03225 c1cc2nc(cn2cc1Br)CO TS-03226 c1cc(ccc1[C@H](C2CC2)O)Br TS-03227 c1cnc(cc1Br)N2CCCC2 TS-03228 c1cc(nc(c1)Br)N2CCCC2 TS-03229 CC(=O)c1ccc(nc1)c2ccc(cc2)OC TS-03230 CC(=O)c1ccc(nc1)c2cccc(c2)OC TS-03231 C1CC(CCC1N2CCC(CC2)C(=O)O)O TS-03232 CC[C@H]1CC(=O)CCN1C(=O)OC(C)(C)C TS-03233 CC(C)(C)OC(=O)c1cc(ccc1Cl)N TS-03236 Cn1c(cc(n1)C(=O)N2CCCCC2)Cl TS-03237 c1c(cnc2c1nc([nH]2)CO)Br TS-03238 Cc1cc(cc(c1N(C)C)C)Br TS-03239 Cc1c(cnc(n1)Cc2ccccc2)C(=O)O TS-03240 c1ccc2c(c1)[nH]c(=O)c(n2)c3cccs3 TS-03241 CC[C@@]1(CCCN(C1)C(=O)OC(C)(C)C)N TS-03242 CC(C)[C@@H]1CNCCN1C(=O)OC(C)(C)C TS-03243 Cn1cc(c(n1)C(F)(F)F)Br TS-03244 Cc1ccc(cc1CC(=O)O)Br TS-03245 Cc1cc(cc(c1Br)C)C(=O)O TS-03247 Cc1cc(cc(c1C(=O)O)C)Br TS-03248 Cc1cccc(c1Br)C(=O)OC TS-03249 Cc1ccc(cc1C(=O)OC)Br TS-03250 COCC(=O)c1ccc(cc1)Br TS-03251 Cc1cc(ccc1Br)CC(=O)O TS-03252 c1ccc(c(c1)C/C(=N/O)/N)Br TS-03253 c1cc2c(cc1C(F)(F)F)cc([nH]2)C(=O)O TS-03255 c1cc(cc(c1)Oc2ccc(cc2)N)C(=O)O TS-03256 COc1ccc(cc1)c2cccc(n2)C(=O)O TS-03257 COc1cccc(c1)c2cccc(n2)C(=O)O TS-03258 COc1ccccc1c2cccc(n2)C(=O)O TS-03259 COc1ccc(cc1)c2cc(ccn2)C(=O)O TS-03260 COc1cccc(c1)c2cc(ccn2)C(=O)O TS-03261 COc1ccccc1c2cc(ccn2)C(=O)O TS-03262 COc1ccc(cc1)c2ccnc(c2)C(=O)O TS-03263 COc1cccc(c1)c2ccnc(c2)C(=O)O TS-03264 COc1ccc(cc1)c2ccc(cn2)C(=O)O TS-03266 COc1cccc(c1)c2ccc(cn2)C(=O)O TS-03267 COc1ccccc1c2ccc(cn2)C(=O)O TS-03268 CC(=O)N1CCN(CC1)c2cccc(c2)C#N TS-03270 CC(=O)N1CCN(CC1)c2ccc(cc2)C#N TS-03271 c1cc(c(cc1F)OCC#N)Br TS-03272 COC(=O)c1ccc(c(c1)N)Br TS-03273 CCOC(=O)c1ccnc(c1)Br TS-03274 C[C@](CO)(c1cccc(c1)Br)N TS-03275 c1cc(ccc1C2(CC2)C(=O)O)C(F)(F)F TS-03276 c1cc(cc(c1)C(F)(F)F)C2(CC2)C(=O)O TS-03277 CC(=O)Oc1ccc2cc(ccc2c1)C(=O)O TS-03278 c1cc(ncc1C(F)(F)F)N2CCCCC2 TS-03279 c1cc(cc(c1)N2CCNCC2)C(F)(F)F TS-03280 CN1CCC(CC1)(C#N)c2cccc(c2)OC TS-03283 c1cc(c(cc1CC#N)Cl)Br TS-03284 Cc1cc(c(cc1Cl)C)SCC(=O)O TS-03285 COc1ccc(cc1Br)C(=O)O TS-03286 COc1c(cc(cn1)Br)C(=O)N TS-03287 c1c(cn(n1)C2CCOCC2)Br TS-03288 COC(=O)C[C@H]1CNCCN1.Cl.Cl TS-03289 c1cc(nnc1C(F)(F)F)N2CCCCC2 TS-03290 c1ccc(cc1)Sc2c(cccn2)C(=O)O TS-03291 c1ccc(cc1)Sc2ccc(cn2)C(=O)O TS-03292 CC(=O)c1ccc(nc1)c2ccc(cc2)Cl TS-03293 CC(=O)c1ccc(nc1)c2cccc(c2)Cl TS-03294 COc1ccc(nc1Br)C(=O)O TS-03295 CNCCc1ccc(cc1F)Br TS-03296 CC(C)(c1ccc(cc1)C(F)(F)F)C(=O)O TS-03297 c1cnc(cc1C(F)(F)F)N2CCOCC2 TS-03298 Cc1cc(c(c2c1C(=O)C(C2)(C)C)C(=O)O)C TS-03299 C.C[C@@H]1CN(C[C@@H](O1)C)c2ccc(cc2)C#N TS-03300 CC[C@H]1CCCCN1C(=O)c2ccc(nc2)C TS-03301 CC(C)(C)c1ccc(cc1)CN2CCNCC2 TS-03302 c1cc(c(cc1CC(=O)O)F)Br TS-03303 CC(=O)Nc1ccc2c(c1)C(=O)CC(O2)(C)C TS-03305 c1ccc(cc1)CN2CCC(=O)[C@@H](C2)C(=O)O TS-03306 Cc1nc(cs1)c2cccc(c2)C(=O)OC TS-03308 COc1ccc(cc1)C2(CCCCC2)C(=O)O TS-03309 CN1CCC(CC1)Nc2ccccc2C(=O)O TS-03310 c1cc(ccc1c2cncc(n2)Cl)C(=O)O TS-03311 c1cnc(nc1)c2ccc(cc2)Br TS-03312 c1cc(cc(c1)Br)c2ncccn2 TS-03313 c1ccc(cc1)CN2CCC(CC2)(C(=O)O)O TS-03314 c1cc(c(cc1C(=O)O)Br)Cl TS-03315 c1cc(c(c(c1)Br)C(=O)O)Cl TS-03316 COc1ccc(cc1c2ccccc2)N.Cl TS-03317 c1cc(ccc1C2(CCC2)C#N)Br TS-03318 Cc1ccc2cc(ccc2n1)NS(=O)(=O)C TS-03319 c1ccc(c(c1)C#N)S(=O)(=O)N2CCCC2 TS-03320 Cc1c(cn(n1)c2ccc(cc2)Cl)C(=O)O TS-03321 COC(=O)c1c(c(cs1)Br)O TS-03322 Cn1ccnc1c2ccc(cc2)Br TS-03323 c1cc(c(cc1Cl)SCC(=O)O)Cl TS-03324 c1cc(nnc1)N2CCNCC2.Cl.Cl TS-03325 Cc1ccc(cc1)/C=C/C(=O)c2cccc(c2)N TS-03329 Cc1c(c(no1)c2ccccc2Cl)C(=O)O TS-03330 Cc1c(nc(o1)c2ccc(cc2)Cl)C(=O)O TS-03331 Cc1nc(co1)c2ccc(cc2)Br TS-03332 CC(=O)n1ccc2c1ccc(c2)Br TS-03333 Cn1c2ccc(cc2ccc1=O)Br TS-03334 c1cc(ccc1Cn2cncn2)Br TS-03335 c1cc(cc(c1)Br)Cn2cncn2 TS-03336 c1ccn(c1)c2cc(cnc2N)Br TS-03337 Cc1c(nc2c(n1)cc(cn2)Br)C TS-03338 c1cc(ccc1C2(CCCCC2)C(=O)O)Cl TS-03339 COC(=O)C1(CCCC1)c2ccc(cc2)Cl TS-03340 CC(=O)n1cc2cc(ccc2n1)Br TS-03341 Cn1c2cccc(c2c(n1)N)Oc3ccccc3 TS-03342 CC(=O)NC1CCC(CC1)N2CCN(CC2)C TS-03343 c1cc(ccc1CN2CC[C@@H](C2)C(=O)O)Cl TS-03346 c1cc(cc(c1)Cl)CN2CC[C@@H](C2)C(=O)O TS-03347 CC(=O)C1(CCNCC1)c2ccccc2.Cl TS-03348 c1c[nH]c2c1c(cc(c2)C(=O)O)Br TS-03349 c1ccc2c(c1)c(c(c(n2)O)Br)O TS-03350 C1CN=C(N[C@@H]1C(F)(F)F)N.Cl.Cl TS-03351 c1ccn(c1)c2ccc(c(c2)F)Br TS-03352 CC(C)(C)OC(=O)N1CCN(CC1)C2CCC2 TS-03354 c1ccc(cc1)CN2CCC(CC2)n3cccc3 TS-03355 c1cc2ncc(n2cc1Br)C(=O)O TS-03356 c1cn2cc(nc2cc1Br)C(=O)O TS-03358 c1cc(ccc1C2(CC2)C(=O)O)Br TS-03359 c1cc(cc(c1)Br)C2(CC2)C(=O)O TS-03360 CN1Cc2cc(ccc2NC1=O)Br TS-03361 c1cc(ncc1C(F)(F)F)C(C(=O)O)(F)F TS-03362 c1cc(c(nc1)C(C(=O)O)(F)F)C(F)(F)F TS-03363 c1cnc(cc1Br)N2CCCCC2 TS-03364 c1ccc2c(c1)c(cc(n2)C(F)(F)F)C(=O)O TS-03365 c1ccc2c(c1)cc(c(n2)C(=O)O)C(F)(F)F TS-03366 c1ccc2c(c1)c(c(cn2)C(F)(F)F)C(=O)O TS-03367 c1ccc2c(c1)c(cc(n2)C(=O)O)C(F)(F)F TS-03368 c1ccc2c(c1)c(c(cn2)C(=O)O)C(F)(F)F TS-03369 c1ccc2c(c1)cc(c(n2)C(F)(F)F)C(=O)O TS-03370 c1cc(cc(c1)N)C(=O)/C=C/c2ccc(cc2)F TS-03371 c1c(cnc(n1)N2CCCCC2)Br TS-03375 c1c(cc(c2c1CCO2)C(=O)O)Br TS-03376 CC(C)(c1ccc(cc1)Br)C(=O)O TS-03377 Cc1cc(cc(c1C(=O)OC)C)Br TS-03378 c1cnc(cc1Br)N2CCOCC2 TS-03379 COC(=O)c1cc2ccc(cc2[nH]1)C(F)(F)F TS-03380 C[C@@]1(c2cccn2-c3ccccc3CO1)C(=O)O TS-03381 CCOC(=O)C1CNc2ccccc2O1.Cl TS-03382 C[C@H]1c2cc(c(cc2CCN1)OC)OC.Cl TS-03383 COC(=O)c1ccc2c(c1)nc([nH]2)C(F)(F)F TS-03384 c1ccc(cc1)C(=O)c2ccc(cc2C(=O)O)F TS-03385 c1ccc(c(c1)C(=O)c2ccc(cc2)F)C(=O)O TS-03386 CCOC(=O)c1ccc(cc1O)Br TS-03387 CCOC(=O)c1c(cncc1Br)N TS-03388 c1cc(c(cc1[C@H](C2CC2)O)Br)F TS-03389 Cc1ccc(cc1)Sc2c(cccn2)C(=O)O TS-03390 c1cnc(cc1N2CCCC2)C(=O)N3CCCC3 TS-03391 CCOC(=O)c1c(c(c([nH]1)C)Br)C TS-03392 c1cc(nnc1C(F)(F)F)N2CCC(CC2)N TS-03393 CN1CCN(CC1)c2ccc(nn2)C(F)(F)F TS-03394 c1ccc(cc1)n2c(cc(n2)C(F)(F)F)Cl TS-03395 COC(=O)Cc1ccc(c(c1)F)Br TS-03396 CC(C)(C)OC(=O)n1cc(cn1)Br TS-03397 c1cc2c(cc1C(F)(F)F)O[C@@H](CN2)C(=O)O TS-03398 c1cc(nnc1C(F)(F)F)N2CCC(CC2)O TS-03399 CCOC(=O)c1cc2c(nc1)CC(CC2=O)(C)C TS-03400 c1ccc(cc1)S(=O)(=O)Cc2ccc(cc2)N TS-03401 c1ccc(cc1)S(=O)(=O)Cc2cccc(c2)N TS-03402 c1ccc2c(c1)cc(nc2N3CCNCC3)Cl TS-03403 C1CCC(CC1)N2CCC(CC2)C(=O)O.Cl TS-03404 COC(=O)Nc1ccc(c(c1)F)Br TS-03405 c1ccc(cc1)c2c(nnc(n2)N)c3ccccc3 TS-03406 c1cc(ccc1Nc2cc(ccn2)C(=O)O)Cl TS-03407 COC(=O)c1ccc(cc1Cl)S(=O)(=O)C TS-03408 c1ccc2c(c1)cc(nc2N3CCOCC3)Cl TS-03409 c1cc(c(cc1F)OCC(=O)O)Br TS-03410 CC(C)(C)OC(=O)NC1CC(c2c1cccc2)O TS-03411 CN1CCC(CC1)(c2cccc(c2)OC)C(=O)O TS-03412 c1csc2c1c(ncn2)N3CCC(CC3)CO TS-03413 c1ccc(c(c1)CC(=N)N)Br.Cl TS-03414 c1cc(ccc1CC(=N)N)Br.Cl TS-03415 c1ccc(c(c1)C#N)S(=O)(=O)N2CCCCC2 TS-03418 c1c(cc(c(c1C(=O)O)Cl)N)Br TS-03419 c1c(cn2c(c1F)nnc2N)F.Br TS-03420 COc1c(csc1C(=O)OC)Br TS-03421 c1cc(c(cc1F)F)Oc2ccc(cn2)C(=O)O TS-03422 Cn1c(cc(n1)C(F)(F)F)c2ccccc2C#N TS-03423 C.C[C@@H]1CN(C[C@@H](O1)C)c2ccc(cc2)C(=O)O TS-03424 c1c(cc(c(c1C(=O)O)O)Br)Cl TS-03425 c1cc(cc(c1)C(F)(F)F)C(=O)c2cnccn2 TS-03427 CC(C)(C)OC(=O)N1CCC(=CC1)N2CCCC2 TS-03428 CC(C)(C)OC(=O)N1CCC(=O)C2C1CCCC2 TS-03429 CCN1CCN(CC1)C2CCC(CC2)NC(=O)C TS-03430 c1cc(cc(c1)Cl)CN2C[C@H](CC2=O)C(=O)O TS-03432 COC(=O)[C@H]1CC(=O)N(C1)c2cccc(c2)Cl TS-03433 CCNC(=O)/C=C/c1cccc(c1)Br TS-03434 c1cc(c(nc1)Oc2ccc(cc2)N)C(F)(F)F TS-03435 c1cc(nc(c1)Oc2ccc(cc2)N)C(F)(F)F TS-03436 CC(C)(C)OC(=O)N1CCC(CC1)N2CCCC2 TS-03437 C[C@H]1CN(CCN1C2CCC2)C(=O)OC(C)(C)C TS-03438 CC(C)(C)OC(=O)N1CCCN(CC1)C2CCC2 TS-03439 CCn1c(nc(n1)Br)Br TS-03440 c1cc(cc(c1)Br)[C@H](C(F)(F)F)O TS-03441 c1cc2c(cc1Br)C=C(CO2)C(=O)O TS-03442 Cc1c(n2cc(ccc2n1)Br)C(=O)O TS-03444 c1cc2nc(cn2cc1Br)CC(=O)O TS-03447 c1cc(ccc1C2(CCC2)C(=O)O)Br TS-03450 c1cc(ccc1N)Oc2nccc(n2)C(F)(F)F TS-03451 c1cc(ccc1N)Oc2ccnc(n2)C(F)(F)F TS-03452 c1cc(cc(c1)Oc2nccc(n2)C(F)(F)F)N TS-03453 c1cc(cc(c1)Oc2ccnc(n2)C(F)(F)F)N TS-03454 c1cc(c(cc1CN2C[C@H](CC2=O)C(=O)O)F)F TS-03455 c1cc(ccc1c2nnc(s2)N)Br TS-03456 CN1CCN(CC1)c2cc(ccn2)Br TS-03457 c1cc(c(cc1C(F)(F)F)C#N)N2CCOCC2 TS-03458 c1cc(cc2c1cc(cc2)O)C(=O)N3CCNCC3 TS-03459 c1cc(c2c(c1)OCCO2)N3CCNCC3.Cl TS-03460 c1ccc(cc1)CN2CCN[C@@H](C2)C(=O)O.Cl TS-03461 Cc1c(c([nH]n1)N)Br.Br TS-03462 COC(=O)c1cc(cc2c1OCC2)Br TS-03463 c1cc2c(cc1C(F)(F)F)ncc(c2O)C(=O)O TS-03465 c1cc(ccc1c2c(nco2)C(=O)O)C(F)(F)F TS-03466 c1cc(cc2c1cc(cc2)O)C(=O)N3CCOCC3 TS-03467 c1ccc(cc1)S(=O)(=O)n2ccc3c2cccc3 TS-03468 c1ccc(cc1)C(=O)c2cnc3n2nc(cc3)Cl TS-03469 c1ccc(cc1)CN2CCOC(C2)C(=O)O.Cl TS-03470 COC(=O)c1cc(c(nc1Cl)N2CCCC2)F TS-03471 c1cc(ccc1C(F)(F)F)N2CC[C@@H](C2)C(=O)O TS-03472 c1cc(cc(c1)N2CC[C@@H](C2)C(=O)O)C(F)(F)F TS-03473 CCOC(=O)c1c(c(c(n1C)C)Br)C TS-03474 c1cc(ncc1C(F)(F)F)N2CCC(CC2)CO TS-03475 c1cc(nc(c1)N2CCC(CC2)CO)C(F)(F)F TS-03476 c1cnc(nc1C(F)(F)F)N2CCC(CC2)CO TS-03477 CC[C@H](C)[C@H]1COC(=O)N1C2CCNCC2.Cl TS-03480 COc1ccc(cc1N2CCNCC2)Cl.Cl TS-03481 c1ccc(cc1)CN2CCC(CC2)N.Cl.Cl TS-03482 COc1ccc(cc1)c2cc(cnc2)Br TS-03483 c1cc2c(cc1Br)nc([nH]2)C(F)(F)F TS-03484 c1cc2c(cc1C(F)(F)F)c(n[nH]2)Br TS-03485 c1cc(ccc1Oc2ccc(cn2)N)Br TS-03486 c1cc(cc(c1)Br)Oc2ccc(cn2)N TS-03487 Cc1cccc(c1Br)C(=O)n2ccnc2 TS-03488 COc1ccc(cc1)N2CCNCC2.Cl.Cl TS-03489 COC(=O)c1cc(cc(c1O)Br)Cl TS-03490 c1cn2c(cnc2nc1C(F)(F)F)Br TS-03491 c1cc(ncc1N)Oc2cc(cnc2)Br TS-03492 c1cc(cc(c1)Oc2ncc(cn2)Br)N TS-03493 c1cc(nc(c1)C(=O)O)c2ccc(cc2)C(F)(F)F TS-03496 c1cc(cc(c1)C(F)(F)F)c2cccc(n2)C(=O)O TS-03497 c1ccc(c(c1)c2cccc(n2)C(=O)O)C(F)(F)F TS-03498 c1cc(ccc1c2ccc(cn2)C(=O)O)C(F)(F)F TS-03499 c1cc(cc(c1)C(F)(F)F)c2ccc(cn2)C(=O)O TS-03500 c1ccc(c(c1)c2ccc(cn2)C(=O)O)C(F)(F)F TS-03501 c1cc(ccc1c2cc(ccn2)C(=O)O)C(F)(F)F TS-03502 c1cc(cc(c1)C(F)(F)F)c2cc(ccn2)C(=O)O TS-03503 c1ccc(c(c1)c2cc(ccn2)C(=O)O)C(F)(F)F TS-03504 c1cc(ccc1c2ccnc(c2)C(=O)O)C(F)(F)F TS-03505 c1cc(cc(c1)C(F)(F)F)c2ccnc(c2)C(=O)O TS-03506 c1ccc(c(c1)c2ccnc(c2)C(=O)O)C(F)(F)F TS-03507 c1ccc(cc1)c2cc(cnc2C(=O)O)C(F)(F)F TS-03508 c1cc(c(nc1)N2CCNCC2)C(F)(F)F.Cl TS-03509 c1cc(c(cc1C(=O)N)C(F)(F)F)Br TS-03510 c1ccc2c(c1)COc3ccc(cc3C2=O)CC(=O)O TS-03511 CC(C)(C)OC(=O)N1CCC(CC1)N2CCCCC2 TS-03512 CCOC(=O)c1cn2ccc(cc2n1)Br TS-03513 CCOC(=O)c1cn2cc(ccc2n1)Br TS-03514 CCOC(=O)c1ccc2ncc(n2c1)Br TS-03515 CCOC(=O)c1cnc2n1cc(cc2)Br TS-03516 Cc1c(n(c(c1S(=O)(=O)C)N)C2CCCCC2)C TS-03518 Cc1c(nc(o1)c2ccc(cc2)C(F)(F)F)C(=O)O TS-03521 c1cc(c(cc1CN2C[C@H](CC2=O)C(=O)O)F)Cl TS-03522 c1c(c2nc(cn2nc1Cl)C3CC3)Br TS-03523 COC(=O)c1cc(c(nc1Cl)N2CCCCC2)F TS-03524 COc1cc(cc(c1O)Br)/C=C/C(=O)O TS-03525 CC(C)(C)OC(=O)Nc1ccc(cn1)Br TS-03526 CC(C)(C)OC(=O)Nc1ccnc(c1)Br TS-03527 CC(C)(C)OC(=O)Nc1cccnc1Br TS-03528 CC(C)(C)OC(=O)Nc1cccc(n1)Br TS-03529 CC(C)(C)OC(=O)Nc1cc(ccn1)Br TS-03530 c1cc(ccc1C(C#N)N2CCOCC2)Cl.Cl TS-03531 c1cc(ccc1C(F)(F)F)N2C[C@H](CC2=O)C(=O)O TS-03532 c1cnc(cc1N2CCCCC2)C(=O)N3CCCCC3 TS-03534 c1cc2c(cc[nH]2)c(c1)N3CCNCC3.Cl.Cl TS-03535 c1cnc(cc1C(F)(F)F)N2CCC(CC2)C(=O)O TS-03536 c1cc(c(nc1)N2CCC(CC2)C(=O)O)C(F)(F)F TS-03537 c1cc(c(cc1C(F)(F)F)C(=O)O)N2CCOCC2 TS-03538 c1c(cn2cc(nc2c1Br)C(=O)O)Cl TS-03539 c1cnc2c(n1)cc(cc2Br)C(F)(F)F TS-03540 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)C#N TS-03541 c1ccc(cc1)n2c(c(c(n2)C3CC3)Br)N TS-03542 c1ccc(cc1)CN2CCN(CC2)c3cc(ccn3)C#N TS-03543 C[C@@](c1cccc(c1)Br)(C(=O)O)N.Cl TS-03544 c1c(cc(c2c1[nH]c(=O)[nH]2)Br)C(F)(F)F TS-03545 c1cc(c(nc1)Sc2ccc(cc2)Br)N TS-03546 c1c(cnc(c1Cl)OC2CCOCC2)C(F)(F)F TS-03547 c1cc(cc(c1)C(F)(F)F)C2(CCNCC2)O.Cl TS-03548 c1ccc(cc1)[C@@H]2COC(=O)N2C3CCNCC3.Cl TS-03549 CCOC(=O)c1c(nc2n1ccc(c2)Br)C TS-03550 c1cc(cnc1)CCN.Br.Br TS-03551 c1cc(ccc1N2C[C@H](CC2=O)C(=O)O)Br TS-03552 c1cc(ccc1c2nc(cs2)C(=O)O)Br TS-03553 c1cc(cc(c1)Br)c2nc(cs2)C(=O)O TS-03554 Cc1cccc(c1Br)C(=O)N2CCOCC2 TS-03555 c1cnc(nc1C(F)(F)F)n2cc(cn2)Br TS-03557 c1cc(ccc1Oc2ccc(cn2)C(=O)O)Br TS-03560 COc1ccc2cc(ccc2c1CC(=O)O)Br TS-03561 C[C@@H]1[C@@H](OC(=O)N1C2CCNCC2)c3ccccc3.Cl TS-03562 Cc1ccc(cc1)C#N TS-03564 Cc1ccc(c(c1)N)C TS-03565 c1cc(ncc1Cl)O TS-03566 CC(=O)c1ccncc1N TS-03567 COC(=O)c1cnccn1 TS-03568 COc1ccc(cc1)CC#N TS-03569 Cc1cccc(c1C)C(=O)O TS-03570 CC(=O)c1cccc(n1)C(=O)C TS-03571 Cc1ccc(cc1)[C@@H](C)C(=O)O TS-03572 c1ccc(cc1)c2ccncc2N TS-03573 CC(=O)Nc1ccc(cc1)Br TS-03575 COc1cccc(c1)c2c(cccn2)C(=O)O TS-03576 c1ccc(cc1)c2c(ccc(n2)Br)N TS-03577 c1cc(cnc1)C(=O)N.I TS-03578 CC(C)(C)OC(=O)N1CCN[C@@H](C1)c2ccccc2 TS-03580 c1cc(c(nc1)c2ccc(cc2)C(F)(F)F)C(=O)O TS-03581 C[C@H]1CN(CCC1=O)C TS-03582 c1ccc(c(c1)C(=O)O)O TS-03583 Cc1cc(cnc1N)Cl TS-03584 Cc1cc(cnc1O)Cl TS-03585 c1ccnc(c1)c2cccc(c2)N TS-03586 c1cc(c(nc1)Br)O TS-03587 c1ccnc(c1)c2cccc(c2)N.Cl.Cl TS-03589