CC(CNc1ccc(cc1[N+](=O)[O-])C(F)(F)F)OC(=O)c2cc3ccccc3oc2=O BTB05481 CC(CNc1ccc(cc1[N+](=O)[O-])C(F)(F)F)OC(=O)c2ccc(o2)[N+](=O)[O-] BTB05482 Cc1cc(ccc1Cl)Oc2ccc(cn2)[N+](=O)[O-] BTB03838 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3cc(c(cc3Cl)Cl)Cl AW00580 Cc1cc(cc(c1Cl)C)Oc2ccc(cn2)N BTB03829 c1ccc(c(c1)Oc2ccc(cn2)[N+](=O)[O-])F BTB03840 c1ccc(cc1)NC(=O)Oc2cccc(c2OC(=O)Nc3ccccc3)F RH00408 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OC(=O)c3cccnc3Oc4ccccc4 RH00411 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)S(=O)(=O)c4ccc(s4)Cl KM09901 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3cccs3 KM09902 CCOC(=O)C1CCN(CC1)c2c(ccs2)[N+](=O)[O-] KM09899 CCOC(=O)c1cnc2c(c1N3CCC(CC3)C(=O)OCC)c(nn2C)C KM09907 c1ccnc(c1)CCNc2ccc(cc2NC(=S)Nc3cc(ccc3Cl)Cl)C(F)(F)F BTB01987 c1cc(cc(c1)C(F)(F)F)/C(=C/c2ccc(cc2Cl)Cl)/C#N AW00576 c1cnc(nc1C(F)(F)F)N2CCC(CC2)O AW00577 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CCS(=O)(=O)c4ccc(cc4)F KM09920 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3cccc4c3nsn4 KM09923 c1cc(oc1)CNC(=S)Nc2ccc3c(c2)C(=O)OC3 KM09928 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc4c(c3)COCO4 BTB01952 Cc1cccc(c1NC(=O)C(C)N2CCCC2)C AW00585 c1cc(cc(c1)C(F)(F)F)/C(=C/c2ccc(cc2)C(F)(F)F)/C#N AW00589 c1cc(ccc1NC(=S)Nc2ccc3c(c2)C(=O)OC3)Cl KM09930 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cccc3c2nsn3 KM09934 c1ccc(cc1)CCNc2ccc(cc2/N=C/c3cc(ccc3O)Br)C(F)(F)F BTB02016 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCOC(=O)c2ccc(o2)[N+](=O)[O-] BTB05488 c1ccc2c(c1)cc(c(=O)o2)C(=O)OCCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05489 c1ccc(c(c1)C(=O)N)N2CCCCC2 BTB03853 c1ccc(c(c1)C#N)NC(=O)CSc2ncccn2 NRB00253 c1cc(ccc1NC(=S)Nc2ccc3c(c2)C(=O)OC3)F KM09940 Cc1c2ccccc2sc1/C=C/C(=O)Nc3nccs3 MWP00720 Cc1c2ccccc2sc1/C=C/C(=O)Oc3ccc(cc3)C#N MWP00737 Cc1c2ccccc2sc1/C=C/C(=O)Oc3ccc(cc3)OC MWP00739 Cc1c2ccccc2sc1COC(=O)c3ccccc3 MWP00742 Cc1cc(nc(n1)SCC(=O)Nc2ccc(c(c2)Cl)F)C NRB00257 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(ccc3NCCc4ccc(c(c4)OC)OC)C(F)(F)F BTB01974 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc3c(c2)COCO3 BTB01953 COc1cc(cc(c1OC)OC)CNc2cccc(c2)F BTB01963 c1cc(cc(c1)F)NCc2ccc3c(c2)OCO3 BTB01964 Cc1c2ccccc2sc1COC(=O)c3ccc(cc3Cl)Cl MWP00743 c1c(cc(cc1C(F)(F)F)NC=C2C(=O)NC(=S)NC2=O)C(F)(F)F BTB01997 c1c(cc(cc1C(F)(F)F)NC=C2C(=O)NC(=O)NC2=O)C(F)(F)F BTB01998 Cc1c2ccccc2sc1COC(=O)Nc3ccc(cc3Cl)Cl MWP00750 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc(s3)Cl KM09914 c1ccc2c(c1)CCN2S(=O)(=O)c3cccc4c3nsn4 KM09942 CCOC(=O)c1cnc2c(c1O)cccc2F BTB02003 COc1ccc(cc1)C(=O)CC2(c3cc(ccc3N(C2=O)CN4CCOCC4)Br)O BTB02024 c1ccc(cc1)C(CN)c2ccc3c(c2)OCCO3.Cl RJC00488 CCCCCCCCCc1ccc(cc1)c2cnc(nc2)CCCCCC RJC00489 c1cc(ccc1S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl AW00591 Cc1c2ccccc2sc1/C=C/C(=O)Nc3ccc(cc3)F MWP00729 Cc1ccc(cc1)SC(=O)/C=C/c2c(c3ccccc3s2)C MWP00733 c1cc(ccc1NC(=O)CSCCSCC(=O)Nc2ccc(cc2)OC(F)(F)F)OC(F)(F)F NRB00259 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nc(cc(n2)C)C NRB00262 CCCCCCc1cnc(nc1)c2ccc(cc2)[N+](=O)[O-] RJC00493 Cc1c2ccccc2sc1/C=C/C(=O)Oc3c(cccc3Cl)Cl MWP00738 Cc1c2ccccc2sc1COC(=O)c3ccc(cc3)[N+](=O)[O-] MWP00744 c1cc(ccc1C(=O)CSCCSCC(=O)c2ccc(cc2)F)F NRB00250 CN(CCOC(=O)c1cc2ccccc2oc1=O)c3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05512 Cn1c(nnc1SCC(=O)Nc2ccccc2C#N)c3ccccc3 NRB00254 COc1cccc2c1nc(s2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05521 Cc1ccc2c(c1)sc(n2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05523 CC(=O)N[C@@H]1[C@H]([C@@H]([C@H](O[C@H]1n2ccc(nc2=O)OC)COC(=O)C)OC(=O)C)OC(=O)C RJC00436 CC(C)(CCO)Nc1ccc(cc1[N+](=O)[O-])C(F)(F)F BTB05498 c1cc(ncc1[N+](=O)[O-])NCCOC(=O)c2ccc(o2)[N+](=O)[O-] BTB05499 CC(C)(COC(=O)c1ccc(o1)[N+](=O)[O-])Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05491 COCCCNC(=S)NNC(=O)c1cc(c(c(c1[N+](=O)[O-])OC)OC)OC BTB05492 c1cc(ncc1[N+](=O)[O-])N2CCCN(CC2)C(=O)N3CCOCC3 AW00597 COc1ccc2c(c1)nc([nH]2)S RH00387 CCCN(C(=O)CC#N)C(=O)Nc1ccccc1C KM09915 COc1cc2c(c(c1OC)OC)nc(oc2=O)c3cccnc3Oc4ccccc4 BTB05494 c1ccc(cc1)c2cnc(sc2=O)c3ccccc3 BTB05518 Cc1cc(ccc1Br)NC(=O)CSCCSCC(=O)Nc2ccc(c(c2)C)Br NRB00249 c1ccc2c(c1)cccc2SCC(=O)O RJC00448 c1ccc(cc1)CNc2ccc(cc2N)C(F)(F)F BTB01955 CC(C)(C)C1=NN(C(=O)C1)C BTB07041 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)F BTB07050 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3ccc(cc3)CC#N BTB07048 Cc1ccsc1/C=C/c2ccnc(n2)SCC(=O)Nc3ccc(cc3)C(C)C MWP00691 COc1ccc(cc1)NC(=S)Nc2ccc3c(c2)C(=O)OC3 KM09917 CCCn1c(=O)cc(n(c1=O)c2ccccc2C)N KM09919 c1ccc2c(c1)Cc3nc(cn3C2)c4ccc(cc4)F.Br BTB02012 CCOC(=O)C(=CNc1ccc2c(c1)[nH]nn2)C(=O)OCC BTB02015 COc1cc2c(c(c1OC)OC)[nH]c(=S)n(c2=O)CC=C BTB05474 c1ccc2c(c1)ccc(n2)c3ccc(cc3)F BTB05480 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc4c(cc(c(c4OC)OC)OC)c(=O)o3 BTB05495 c1cc(ncc1[N+](=O)[O-])NCCO BTB05497 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)S(=O)(=O)c4cccs4 KM09903 CCOC(=O)C1CCN(CC1)c2cc(nc3c2cccc3Cl)C(F)(F)F KM09905 Cc1ccc2c(c1)c(=O)oc(n2)c3ccc(o3)[N+](=O)[O-] BTB05486 CC(C)(COC(=O)c1cc2ccccc2oc1=O)Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05490 COc1ccc(cc1OC)CCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB01959 CCOC(=O)C(=CNc1ccccc1F)C(=O)OCC BTB01960 c1cc(c(c(c1)Cl)COc2ccc(cc2)CC#N)F BTB07033 Cc1c2ccccc2sc1COS(=O)(=O)c3ccc(cc3Cl)Cl MWP00759 CCOC(=O)c1c[nH]c2c(cc(cc2c1=O)Cl)C BTB02004 Cc1ccc2c(c1)c(=O)[nH]c(n2)NC(=O)c3ccc(cc3)[N+](=O)[O-] BTB02009 c1cnc(nc1)SCC(=O)Nc2ccc(cc2C(F)(F)F)F NRB00251 Cc1c(nc(s1)c2c(cccc2F)F)O NRB00252 Cc1c2ccccc2sc1C(=S)Nc3ccc(cc3)C(C)C MWP00774 c1ccc2cc(ccc2c1)C(=O)CC3(c4cc(ccc4N(C3=O)CN5CCOCC5)Br)O BTB02023 c1cc(cnc1)c2nc(cs2)C(=O)NCc3ccc(cc3)Cl MWP00710 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3cccs3 KM09908 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl KM09911 Cc1ccc(cc1)COc2ccc(cc2)CC#N BTB07031 c1cc(ccc1CC#N)OCc2ccc(c(c2)Cl)Cl BTB07032 C/C=C(\C)/c1nc2c(cc(cc2Br)Br)c(=O)o1 BTB01928 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)c4ccc(cn4)C(F)(F)F KM09909 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)c4c(cccn4)C(F)(F)F KM09910 c1cc(ccc1CC#N)OCc2ccc(cc2)Cl BTB07034 Cc1ccsc1/C=C/c2ccnc(n2)SCc3c(cccc3Cl)Cl MWP00686 c1ccc2c(c1)cc(c(=O)o2)C(=O)OCCNc3ccc(cn3)[N+](=O)[O-] BTB05500 COc1ccc(cc1OC)CCNc2ccc(cc2N)C(F)(F)F BTB01965 c1ccc(cc1)CCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB01967 CC(c1ccccc1)Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB01970 CC(C)(C)C1=NN(C(=O)C1)c2ccccc2 BTB07042 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)CC#N BTB07046 Cc1c2ccccc2sc1/C=N/Nc3nc(cs3)c4ccccc4Cl MWP00708 c1cc2c(cc1[N+](=O)[O-])sc(n2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05524 c1cc(c(cc1NC(=O)CSc2ccc(cn2)C(F)(F)F)Cl)F NRB00260 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3ccc4c(c3)COCO4 BTB01951 c1ccc2c(c1)c(c(s2)C(=O)Nc3c(cc(cc3Br)Br)C(=O)O)Cl BTB01929 Cc1ccsc1/C=C/c2ccnc(n2)Sc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] MWP00698 Cc1c2ccccc2sc1/C=N/NC(=S)N MWP00703 Cc1ccsc1/C=C/c2ccnc(n2)SCC(=O)Nc3ccccc3 MWP00689 Cc1ccsc1/C=C/c2ccnc(n2)Sc3ncc(s3)[N+](=O)[O-] MWP00697 Cc1ccsc1/C=C/c2ccnc(n2)SCc3cccc(c3)Cl MWP00687 c1ccc(cc1)CNC(=O)c2csc(n2)c3cccnc3 MWP00709 Cc1c2ccccc2sc1/C=N/Nc3nc(cs3)c4ccccc4 MWP00707 Cn1cnnc1SCC(=O)Nc2ccc(c(c2)Cl)F NRB00261 c1cc(sc1)C(=O)O/N=C(/c2ccc(cc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)\N BTB05527 CCOC(=O)c1c[nH]c2cc3c(cc2c1=O)OCO3 BTB02006 Cc1cccc(c1)C(=O)Nc2[nH]c(=O)c3cc(ccc3n2)C BTB02008 CCOC(=O)C(=CNc1ccc(cc1C)Cl)C(=O)OCC BTB01990 Cc1c2ccccc2sc1/C=N/NC(=S)Nc3ccc(cc3)Cl MWP00705 COc1cc(c(c(c1OC)OC)NC(=O)c2cccs2)C(=O)OC BTB05532 CC(=O)OC[C@H]1[C@@H]([C@H]([C@@H](C(O1)OC[C@@H]2[C@H]([C@@H]([C@H]([C@@H](O2)OC(C#N)c3ccccc3)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00434 CCOC(=O)C(=CNc1cccc(c1Cl)Cl)C(=O)OCC BTB01991 Cc1ccc(cc1)SCCC(=O)c2cccs2 MWP00747 CCOC(=O)CNC(=O)CSc1ncccn1 NRB00255 CC(=O)C.c1c(cc(cc1Cl)Cl)n2c(=N)n(sc2=N)c3cc(cc(c3)Cl)Cl.c1c(cc(cc1Cl)Cl)n2c(=N)n(sc2=N)c3cc(cc(c3)Cl)Cl NRB00248 CCOC(=O)C(=CNc1cc(ccc1Cl)C(F)(F)F)C(=O)OCC BTB01993 CCOC(=O)C(=CNc1cc(ccc1[N+](=O)[O-])C)C(=O)OCC BTB01995 Cc1ccc2c(c1)c(=O)[nH]c(n2)NC(=O)c3ccccc3Cl BTB02010 c1ccc2c(c1)c(c(s2)C(=O)Oc3ccc(cc3)CC#N)Cl BTB07049 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(c(c3)Cl)F BTB07051 c1cc(c(c(c1)Cl)C(=O)NC(=O)Oc2c(cccc2Cl)Cl)Cl BTB07055 c1ccc(c(c1)C#N)NC(=O)CSCCSCC(=O)Nc2ccccc2C#N NRB00263 CC(C)(CCOC(=O)c1cc2ccccc2oc1=O)Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05502 COc1ccc(cc1OC)CCNc2ccc(cc2/N=C/c3cc(cc(c3O)Cl)Cl)C(F)(F)F BTB01978 CCOC(=O)C(=CNc1ccc2c(c1)OCO2)C(=O)OCC BTB01992 CC(C)(CCOC(=O)c1ccc(o1)[N+](=O)[O-])Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05503 CCOC(=O)c1cnc2c(c1O)cc(cc2Cl)Br BTB01996 c1cc(c(c(c1)F)C(=O)NC(=O)Nc2ccc(cc2)C(F)(F)F)F RH00400 c1cc(c(c(c1)Cl)/C=N/c2ccc(c(c2)Cl)F)F BTB03727 CC(=Cc1nc2cccc(c2c(=O)o1)F)C BTB03729 CCOC(=O)/C(=C/Nc1cccc(c1C#N)F)/C#N BTB03737 CC(=O)C(=CNc1cccc(c1C#N)F)C(=O)C BTB03738 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cccc(c3C(=O)Nc4ccc(cc4)F)F BTB03742 c1cc(cc(c1)C(F)(F)F)c2nc3cccc(c3c(=O)o2)F BTB03734 c1cc(c(cc1C(=O)NC(=O)Nc2ccc(c(c2)Cl)F)Cl)F BTB03711 CC(C)(C)C(=O)Nc1cccc(c1C(=O)O)F BTB03735 CCOC(=O)C(=CNc1cccc(c1C#N)F)C(=O)OCC BTB03736 c1cc(c(c(c1)F)C(=O)NCc2cccs2)NC(=O)c3cccs3 BTB03743 c1ccc(cc1)CCNc2ccc(cc2NC(=S)Nc3cc(ccc3Cl)Cl)C(F)(F)F BTB01986 CCOC(=O)C(=CNc1cc(ccc1NCCc2ccccn2)C(F)(F)F)C(=O)OCC BTB01988 CCOC(=O)C(=CNc1cc(ccc1NCCc2ccc(c(c2)OC)OC)C(F)(F)F)C(=O)OCC BTB01966 c1ccnc(c1)CCNc2ccc(cc2N)C(F)(F)F BTB01972 c1ccc(cc1)OC(=O)NC(=O)c2ccc(cc2)Cl BTB07057 c1cc2c(c(c1)F)c(=O)oc(n2)c3cccs3 BTB03732 c1cc(sc1)C(=O)CCC(=O)c2cccs2 RJC00463 c1cc(oc1)CNC(=S)NCCNc2nccc(n2)C(F)(F)F AW00554 c1cc(c(cc1OCC(CNCCNc2nccc(n2)C(F)(F)F)O)Cl)Cl AW00555 c1cc(ccc1C2CC2(Br)Br)[N+](=O)[O-] RJC00452 c1ccc(cc1)C(=O)NC(=O)Oc2ccc(cc2)Cl BTB07058 c1cc(c(cc1C(=O)NC(=O)Nc2ccc(cc2F)F)Cl)F BTB03713 CCOC(=O)/C(=C/Nc1ccc(c(c1)Cl)F)/C#N BTB03723 c1cc(c(c(c1)F)OC(=O)NC(=O)c2c(cccc2Cl)Cl)F BTB07062 CCOC(=O)C(=CNc1ccc(cc1F)F)C(=O)OCC BTB03740 CC1CC(CN(C1)c2cc(c(cc2F)[N+](=O)[O-])NC(=O)C)C BTB03705 c1ccc(cc1)C(c2nc3cccc(c3c(=O)o2)F)C4CCCC4 BTB03731 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nc4cccc(c4c(=O)o3)F BTB03733 CC1CN(CC(O1)C)C(=O)NC(=O)c2ccc(c(c2)Cl)F BTB03712 CCOC(=O)C(=CNc1cccc(c1)C(=O)OC)C(=O)OCC BTB01994 c1c(cc(cc1C(F)(F)F)NC=C(C#N)C#N)C(F)(F)F BTB02000 CCOc1ccc2c(c1)sc(n2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05522 c1ccc2c(c1)nc(s2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05525 CC(=O)c1ccc(cc1)C2CC2(Cl)Cl RJC00459 CN1CCC(=NOC(=O)Nc2ccc(cc2)Cl)CC1 KM09888 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccc(c2C(=O)NCCc3ccncc3)F BTB03744 c1ccc(cc1)C(C2CCCC2)C(=O)Nc3cccc(c3C(=O)NCc4cccs4)F BTB03746 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCC3CC3 AW00563 c1cc(ccc1OCC(CNCCNc2nccc(n2)C(F)(F)F)O)OC(F)(F)F AW00556 c1ccc(cc1)c2nc(sn2)S AW00582 CC(C)c1csc2c1c(=O)[nH]cn2 AW00583 c1cc(c(c(c1)Cl)CN2CCN(CC2)c3nccc(n3)C(F)(F)F)F AW00560 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc(s3)Br KM09895 c1cc(cc(c1)Cl)/C(=C\c2nccn2C(=O)c3cccc(c3)Cl)/OC(=O)c4cccc(c4)Cl KM09944 CCOC(=O)c1c[nH]c2c(c1=O)cc(cc2F)F BTB03756 c1cc(c(c(c1)F)OC(=O)Nc2cc(cc(c2)Cl)Cl)OC(=O)Nc3cc(cc(c3)Cl)Cl RH00414 Cc1cccc(c1NC(=O)NCc2ccccc2)C KM09927 Cc1ccc(cc1)NS(=O)(=O)N(C)C KM09932 CC(C)(C)NC(=S)N/N=C/c1ccc(c(c1)OC)OCc2ccccc2 BTB03763 CCCNC(=O)Nc1ccccc1C KM09906 c1ccc(cc1)N/N=C(/Cc2ccccc2[N+](=O)[O-])\C(=O)O RJC00479 COc1c(cc(cc1[N+](=O)[O-])S(=O)(=O)N2CCOCC2)[N+](=O)[O-] KM09886 c1ccc(cc1)N2CCN(CC2)c3cc(nc4c3cccc4Cl)C(F)(F)F KM09891 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)Br KM09893 CCOC(=O)C(=CNc1ccc(cc1Cl)Br)C(=O)OCC BTB01989 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)S(=O)(=O)c4ccc(s4)Br KM09896 c1ccc(cc1)Nc2cc(nc3c2cccc3Cl)C(F)(F)F KM09892 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4cc(nc5c4cccc5Cl)C(F)(F)F KM09894 CCOC(=O)C1CCN(CC1)c2cc(nc3c2cc(cc3)Br)C(F)(F)F KM09898 CCOC(=O)C(=CNc1cc(ccc1NCCc2ccccc2)C(F)(F)F)C(=O)OCC BTB01976 CC(C)(C)c1cc(c(c(c1)C(C)(C)C)O)C(=O)/C=C/N(C)C RH00413 CC(C)(C)NC(=S)N/N=C/c1cc(cc(c1O)OC)Br BTB03759 COc1ccc(cc1OC)/C=N/CCNc2nccc(n2)C(F)(F)F AW00562 c1cc(cc(c1)C(F)(F)F)CSCC(=O)Nc2cc(cc(c2)Cl)Cl BTB03767 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCO BTB05475 CC(C)(CO)Nc1ccc(cc1[N+](=O)[O-])C(F)(F)F BTB05476 c1ccc(cc1)CCNc2ccc(cc2NC(=O)c3c(c4ccccc4s3)Cl)C(F)(F)F BTB01980 Cc1c2ccccc2sc1/C=C/C(=O)Sc3c(cccc3Cl)Cl MWP00735 c1ccc(cc1)c2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-] BTB03825 Cc1c(cccc1Cl)NC(=O)N2CCC(CC2)O AW00587 c1cc(cc(c1)NC(=S)N2CCC(CC2)O)C(F)(F)F AW00588 CN1CCC(=NOC(=O)Nc2cccc(c2)C(F)(F)F)CC1 KM09913 Cc1ccc(cc1)C(=O)CSC(=S)SC(C)(C)C BTB03854 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)Cl KM09900 COc1cc2c(c(c1OC)OC)nc(oc2=O)c3cccc(c3)C(F)(F)F BTB05477 c1cc(c(c(c1)Cl)Oc2ccc(cn2)N)Cl BTB03828 c1ccc(cc1)Cc2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-] BTB03824 c1cc(c(c(c1)F)C(=O)NC(=O)Nc2ccc(cc2)Br)F RH00401 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OC(=O)c3cccs3 RH00402 CC(=O)Nc1c(cc(c(c1OC)OC)OC)C(=O)O BTB05479 CCCn1c(=O)c(cn(c1=O)c2ccccc2C)Br KM10020 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3nnc(s3)Sc4ccnc5c4ccc(c5)Cl RH00428 CN(C)/C=N/c1nnc(s1)Sc2ccnc3c2ccc(c3)Cl RH00432 CC(=O)N1CCc2c1ccc(c2)[N+](=O)[O-] RH00434 Cc1c(cco1)c2cc(n(n2)c3cccc(c3Cl)Cl)N KM10021 CCOC(=O)N/N=C(\C)/c1c(c2cc(ccc2s1)Cl)C MWP00794 c1ccc(cc1)Cn2c(=O)c(cn(c2=O)C3CC3)C#N KM10025 CCCn1c(=O)c(cn(c1=O)C2CC2)C(=O)N KM10026 c1cc2c(cc1[N+](=O)[O-])CCN2C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RH00435 c1cc(c(cc1C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-])Cl)F BTB05636 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)CC(CN4CCCC4=O)O AW00640 Cc1c2ccccc2sc1C(=S)Nc3ccccc3 MWP00776 CN1C(=O)C(=CNc2ccccc2)C(=O)N(C1=O)C KM10001 C/C(=N\NC1=NCCCN1)/c2ccc(cc2)OC RH00423 c1cc(c(c(c1)Cl)Oc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N)Cl BTB03918 c1cc(c(c(c1)Cl)Oc2ccc(c(c2Cl)Oc3c(cccc3Cl)Cl)[N+](=O)[O-])Cl BTB03920 Cc1ccc(cc1)NC(=N)c2ccccc2.I NRB00293 CC(=O)N1CCc2c1c(ccc2)N RH00439 CCOC(=O)/C(=C/Nc1ccc2c(c1)CCN2C(=O)C)/C#N RH00444 CC(C)(C)CNC(=S)NN BTB03868 c1cc(ccc1/C=C\2/C(=O)NC(=S)S2)C#N BTB05555 CC(C=C)N1C(=O)c2ccccc2C1=O BTB03942 CN(C)c1cc(c(cc1[N+](=O)[O-])F)N2CCCC2 BTB03945 CCCn1c(=O)c(cn(c1=O)c2ccccc2C)C#N KM09997 Cc1ccccc1NC(=O)NCc2ccc(cc2)C(=O)OC KM09998 CCCCOc1cc(ccc1OC)C(=O)N KM09999 CC(=CC(=O)Nc1nnc(s1)Sc2ccnc3c2ccc(c3)Cl)C RH00418 CC(=O)N1CCc2c1ccc(c2)NC(=S)NCc3cccs3 RH00446 CN1C(=O)C(=CNc2cccc(c2)C(F)(F)F)C(=O)N(C1=O)C KM10007 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3nnc(s3)Sc4ccnc5c4ccc(c5)Cl RH00422 CN1C(=O)C(=CNc2ccc(cc2F)F)C(=O)N(C1=O)C KM10008 CCCn1c(=O)ccn(c1=O)c2ccccc2C KM10010 Cc1cc(ccc1Cl)C(=O)CSC(=S)SC(C)(C)C BTB03874 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc(cc2)Cl)N3CCCCC3 BTB03881 CC(C)c1nnc(s1)NCC(C)(C)C BTB03877 c1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00598 CC(C)(C)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00601 c1cc(c(c(c1)Cl)Oc2ccc(cc2[N+](=O)[O-])Cl)Cl BTB03903 c1cc(c(c(c1)Cl)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl BTB03904 CC1CCCN(C1)c2cc(c(cc2F)[N+](=O)[O-])N(C)C BTB03946 c1ccc(c(c1)NC(=O)Nc2cccc(c2)C(F)(F)F)SCc3ccc(cc3)Cl NRB00311 c1cc(ncc1C(F)(F)F)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB00316 Cc1ccc(c(c1)C)NC(=S)N2CCC(CC2)O AW00604 Cc1cccc(c1NC(=S)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl AW00606 CC(C)(C)SC(=S)SCC(=O)c1ccc(c(c1)Cl)Cl BTB03861 CC(C)(C)SC(=S)SCC(=O)c1cc2cc(ccc2o1)Br BTB03867 CC(=O)N1CCc2c1ccc(c2)NC(=S)NCCSC(C)(C)C RH00447 CCOC(=O)N/N=C/c1c(c2ccccc2s1)C MWP00795 CCOC(=O)N/N=C/c1c(c2cc(ccc2s1)Cl)C MWP00796 c1cc(c(cc1NC(=S)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl)Cl AW00592 c1cc(c(c(c1)Cl)C=C2C(=O)NC(=S)NC2=O)F BTB02088 Cn1c2ccc(cc2c(=O)nc1c3ccc(cc3)C#N)Cl BTB05606 c1cc(cc(c1)NC(=S)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)C(F)(F)F AW00602 c1cc(ccc1F)SCC(CN2CCN(CC2)c3nc4ccc(cc4s3)Cl)O AW00629 c1cc(c(cc1F)OC(F)(F)F)NC(=O)N2CCC(CC2)O AW00631 COc1ccc(cc1NC(=S)N2CCCN(CC2)Cc3ccc(cc3)F)Cl AW00633 CC1CC(CN(C1)c2cc(c(cc2F)[N+](=O)[O-])N(C)C)C BTB03948 Cc1cccc(c1)NC(=S)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-] AW00617 c1cc(c(nc1)N2CCCN(CC2)C(=S)Nc3ccc(cc3)Cl)[N+](=O)[O-] AW00618 CC(C)(C)OC(=O)NCCNC(=O)Nc1cccc(c1Cl)Cl AW00634 c1ccc2c(c1)ccn2CC(CN3CCN(CC3)c4nc5ccc(cc5s4)Cl)O AW00637 COc1ccc(cc1NC(=S)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-])Cl AW00616 c1cc(ccc1CN2CCCN(CC2)C(=S)NC3CCCCC3)F AW00620 c1cc(c(cc1NC(=O)N2CCC(CC2)O)Cl)Cl AW00622 c1cc(ccc1NC(=O)N2CCC(CC2)O)OC(F)(F)F AW00623 Cc1c(cccc1Cl)NC(=S)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00607 CC(=O)C(C)(C)OC(=O)NCCc1ccccn1 BTB05611 CC(=O)C(C)(C)OC(=O)NCCc1ccc(cc1)Cl BTB05613 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)CC(CN4CCCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl)O AW00625 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)NC(=S)Nc3ccccc3 KM09952 c1ccc(cc1)CCNC2(CCN(CC2)Cc3ccccc3)C#N KM09962 CC(C)(C)c1ccc(c(c1)C(C)(C)C)OCC(=O)NN RH00467 c1ccc(c(c1)C(=O)Nc2c(cc(cc2Br)F)F)F BTB03961 COc1ccc(cc1OC)S(=O)(=O)Nc2c(cc(cc2Br)F)F BTB03965 C1CCCC(CCC1)NC(=S)N2CCC(CC2)O AW00610 c1cc(c(nc1)N2CCCN(CC2)C(=S)Nc3ccc(cc3F)F)[N+](=O)[O-] AW00614 COc1ccccc1NC(=S)N2CCCN(CC2)Cc3ccc(cc3)F AW00621 Cc1c2ccccc2sc1/C=N/c3ccc(cc3)OC(=O)Nc4ccccc4 MWP00818 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)NC(=S)Nc3ccccc3Cl KM09953 COc1ccc(cc1)NC(=S)NC(=O)c2cc(cnc2)C#Cc3ccccc3 KM09954 Cc1c(ccc(c1O)c2cc[nH]n2)OCc3ccc(c(c3)Cl)Cl RH00458 Cc1c2ccccc2sc1CNC(=O)Nc3cccc(c3)Cl MWP00829 Cc1c2ccccc2sc1CNC(=S)Nc3ccc(cc3Cl)Cl MWP00833 Cc1cc(c(cc1Cl)C)SCC(=O)NN RH00470 CCOC(=O)c1cnn(c1N)C(=O)COc2ccc(cc2C(C)(C)C)C(C)(C)C RH00468 c1cc(sc1)C(=O)NNC(=O)CCCC(=O)NNC(=O)c2cccs2 NRB00350 c1cc(oc1)C(=O)NNC(=O)CCCCCCCCC(=O)NNC(=O)c2ccco2 NRB00351 Cc1ccccc1n2cc(c(=O)[nH]c2=O)C#N KM09986 Cc1c(c(n(n1)S(=O)(=O)c2ccccc2)C)Cc3csc4c3cc(cc4)Cl MWP00810 CCOC(=O)C(=CNc1ccc2c(c1)CCN2C(=O)C)C(=O)OCC RH00445 CC(C)(C)NC(=S)N(CCC#N)N BTB03968 Cc1c2ccccc2sc1CNC(=S)Nc3ccc(cc3)F MWP00835 c1c(csc1/C=C/2\C(=O)NC(=S)S2)Br BTB05559 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C(=N\O)/C(=O)Nc2ccccc2 BTB05562 CC(C)(C)C(=O)N1CCCN(CC1)c2ccc(cn2)[N+](=O)[O-] AW00632 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCN(CC2)C(=S)Nc3ccc(cc3Cl)Cl AW00638 CCCCOc1cc(ccc1OC)C(=O)O KM09976 CCCOc1cc(ccc1OC)C(=O)N KM09978 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OCc3ccccc3 RH00415 c1ccnc(c1)SCC(=O)O BTB05540 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2c(cc(cc2Cl)S(=O)(=O)N)Cl BTB03984 c1cc(ccc1C(=O)NNC(=O)CC(=O)NNC(=O)c2ccc(cc2)F)F NRB00348 c1cc(ncc1[N+](=O)[O-])N2CCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl AW00595 c1cc(c(cc1OCC(CN2CCN(CC2)c3nc4ccc(cc4s3)Cl)O)Cl)Cl AW00624 Cc1ccc(cc1S(=O)(=O)Oc2cccc3c2nc(cc3)C)[N+](=O)[O-] BTB05566 CN1C(=O)C(=CNc2ccc(cc2)OC)C(=O)N(C1=O)C KM10006 CCCn1c(=O)c(cn(c1=O)C2CC2)C#N KM10024 CN(C)c1ccc(cc1)C2CC(=O)c3ccccc3N2 NRB00361 Cc1ccc2cccc(c2n1)OS(=O)(=O)c3ccc(cc3F)F BTB05563 c1ccc2c(c1)C=CC3=NC(CN23)c4ccc(cc4)F.Br BTB02027 c1ccc2cc(ccc2c1)C3CN4c5ccccc5C=CC4=N3.Br BTB02032 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)/N=C/c3ccccc3O BTB02028 c1cc(c(cc1C(F)(F)F)/N=C/c2cc(ccc2O)Br)Cl BTB02039 c1cc(ccc1/C(=N/OC(=O)c2ccc(o2)[N+](=O)[O-])/N)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05541 c1ccc(cc1)c2cn(cnc2=O)Cc3ccccn3 BTB05544 Cc1c(cc(c(c1/N=C/c2cc(ccc2O)Br)OC)C(C)(C)C)/N=C/c3cc(ccc3O)Br BTB02047 CCC(c1ccccc1)C(=O)Nc2cc(c(cc2OC)Cl)OC BTB02051 c1ccc(cc1)c2csc(n2)CSc3ccccc3 KM10027 c1cc(c(cc1F)F)NC(=O)N KM10031 CC(=O)N1CCc2c1ccc(c2)NC=C(C#N)C#N RH00443 CN1c2ccccc2C(=O)NC1c3cc(cs3)Br BTB05574 CC(=O)N1CCc2c1ccc(c2)NC(=S)NC3CCCCCC3 RH00449 Cc1c(ccc(c1O)C(=O)C)OCc2ccc(c(c2)Cl)Cl RH00450 Cc1c(cccc1Cl)NC(=S)Nc2cc3c(c(c2C)[N+](=O)[O-])C(CC3(C)C)(C)C BTB02043 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)Nc3ccc(cc3)OC(F)(F)F KM09993 Cc1cc(cnc1)C(=O)NN KM10013 CCC(c1ccccc1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02057 CN1C(=O)C(=CNc2ccc(cc2)Cl)C(=O)N(C1=O)C KM10005 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2nc(cc(n2)c3cc(c(c(c3)OC)OC)OC)c4ccc(cc4OC)OC NRB00359 c1ccc2c(c1)C(=O)NC(N2)c3ccc(cc3)C#N BTB05578 c1ccc(cc1)c2cc(nc(n2)NS(=O)(=O)c3ccc(cc3)N)c4ccccc4 NRB00372 COc1ccc(cc1)c2cc(nc(n2)NS(=O)(=O)c3ccc(cc3)N)c4ccccc4 NRB00373 Cc1c2ccccc2sc1CNC(=O)Nc3ccccc3 MWP00831 Cc1c2ccccc2sc1CNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F MWP00836 c1cc(sc1/C=C\2/C(=O)NC(=S)S2)[N+](=O)[O-] BTB02102 c1ccc(cc1)C2=N/C(=C/c3ccc(s3)[N+](=O)[O-])/C(=O)O2 BTB02103 COc1ccc(c(c1)OC)/C=C\2/C(=O)OC(=N2)c3ccccc3 NRB00331 c1cc(ccc1C(=O)NNC(=O)CCC(=O)NNC(=O)c2ccc(cc2)F)F NRB00349 c1ccc(c(c1)C(=O)NCc2cccs2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05602 Cc1ccc(cc1)S(=O)(=O)NN2C(Nc3ccccc3C2=O)c4cccc(c4O)OC BTB02076 Cc1c(cc(c(c1/N=C/c2cc(cc(c2O)Cl)Cl)OC)C(C)(C)C)/N=C/c3cc(cc(c3O)Cl)Cl BTB02046 c1cc(ccc1SCC(=N)NS(=O)(=O)c2cc(cc(c2)Cl)Cl)Cl BTB05596 CC(=O)C(C)(C)OC(=O)N1CCOCC1 BTB05604 Cc1cccc2c1Nc3c(c(=O)c3=O)N2 MWP00865 c1ccc2c(c1)C(=O)NC(N2)c3cc(cs3)Br BTB05579 CCCCCC(=O)c1cc(c(cc1NC(=O)C)C)C BTB05584 Cc1ccc2cccc(c2n1)OS(=O)(=O)c3ccc(cc3)C(C)C BTB05564 Cn1c2ccc(cc2c(=O)nc1c3cc(cs3)Br)Cl BTB05594 c1cc(c(c(c1)Cl)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl BTB05598 c1ccc(c(c1)C(=O)NCCCN2CCCCC2)N BTB05600 CCOC(=O)c1ccc(cc1)S(=O)(=O)NNC(=O)c2ccccc2N BTB02069 c1cc(ccc1SCC(=N)NS(=O)(=O)c2ccc(cc2F)F)Cl BTB05589 CC(C)c1ccc(cc1)S(=O)(=O)NC(=N)CSc2ccc(cc2)Cl BTB05590 c1ccc(cc1)C2=N/C(=C\c3cc(cs3)Br)/C(=O)O2 BTB05595 CCC(c1ccccc1)C(=O)NNC(=O)c2ccc(cc2)OC BTB02041 c1ccc2c(c1)CCN(C2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB02053 Cc1c(cc(c(c1/N=C/c2ccccc2O)OC)C(C)(C)C)/N=C/c3ccccc3O BTB02052 Cc1c(c(n(n1)C(=O)Nc2cccc(c2)Cl)C)Cc3csc4c3cc(cc4)Cl MWP00823 Cc1c2cc(ccc2sc1C(=O)CC3C(=C(C(=O)O3)Cl)Cl)Cl MWP00824 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc(cc3)C#N)Cl MWP00825 c1ccc(cc1)CCN(CCc2ccccn2)C(=S)Nc3cc(ccc3Cl)Cl.Cl BTB02080 Cc1ccc(c(c1)NC(=S)N(CCc2ccccc2)CCc3ccccn3)C.Cl BTB02082 COc1cc(cc(c1OC)OC)CN(c2cccc(c2)F)C(=O)c3cccc(c3)[N+](=O)[O-] BTB02058 c1ccc(c(c1)C(F)(F)F)NC(=S)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00593 Cc1c(cccc1Cl)NC(=S)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00594 CC(C)(C)SC(=S)SCC(=O)c1ccc(cc1)F BTB03862 CC(C)(C)SC(=S)SCC(=O)c1cc2ccccc2o1 BTB03865 C/C=C(\C)/c1nnc(s1)NCC(C)(C)C BTB03875 c1ccc2c(c1)C=CC3=NC(CN23)c4ccc(cc4)Cl.Br BTB02045 CC(C)c1ccc(cc1)NC2=NNC(=O)C2 MWP00815 Cc1c2ccccc2sc1/C=N/c3ccc(cc3)OC(=O)Nc4cccc(c4)Cl MWP00817 Cc1c(c(n(n1)C(=O)Nc2ccccc2)C)Cc3csc4c3cc(cc4)Cl MWP00822 Cc1nc2ccc(cc2c(=O)o1)Br BTB02093 CCOC(=O)CCN1C(=O)c2ccccc2C1=O BTB02095 c1cc(sc1C=C2C(=O)NC(=S)NC2=O)[N+](=O)[O-] BTB02101 c1cc(sc1)CNC(=S)C(=O)Nc2ccc(cc2F)F NRB00310 c1ccc(c(c1)/N=C/c2cccs2)SCc3ccc(cc3)Cl NRB00312 Cc1ccccc1NC(=O)NCc2ccc(cc2)OC KM09961 CC(=O)C(C)(C)OC(=O)N1CCSCC1 BTB05605 c1ccc2c(c1)c(c[nH]2)CCc3ccccn3 BTB02066 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2ccccc2N BTB02067 Cc1c2cc(ccc2sc1/C(=N\Nc3c(cc(cc3Cl)Cl)Cl)/C)Cl MWP00798 Cc1c(c(n(n1)S(=O)(=O)c2ccccc2Cl)C)Cc3csc4c3cc(cc4)Cl MWP00811 Cc1ccc(cc1)S(=O)(=O)NN2C(Nc3ccccc3C2=O)c4cc(ccc4O)Br BTB02075 CC(C)c1ccc(c(c1)NC(=S)Nc2cc(ccc2Cl)Cl)C(C)C BTB02077 c1ccc(cc1)CCN(CCc2ccccn2)C(=S)Nc3cccc(c3)C(F)(F)F BTB02081 Cc1c(c(n(n1)C(=O)c2ccc(cc2)[N+](=O)[O-])C)Cc3csc4c3cc(cc4)Cl MWP00804 c1cc(ccc1/C(=C\c2nccn2C(=O)c3ccc(cc3)Cl)/OC(=O)c4ccc(cc4)Cl)Cl KM09950 c1ccc2c(c1)c(cc(n2)C(F)(F)F)Nc3ccc(cc3)Cl KM09965 Cc1cc(on1)Nc2cc(nc3c2cccc3Cl)C(F)(F)F KM09966 CC(C)(C)c1ccc(cc1)NC(=O)CSc2ccc(cn2)C(F)(F)F NRB00313 c1cc(ccc1NC(=O)/C(=C/c2cc(cs2)Br)/C#N)F BTB05549 Cc1cc(c(cc1C)NC(=S)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])C AW00608 COCCCNC(=S)N1CCN(CC1)c2ccc(cn2)[N+](=O)[O-] AW00609 c1cc2c(cc1NC(=O)CSc3ccc(cn3)C(F)(F)F)OCCO2 NRB00314 c1ccc(c(c1)C#N)NC(=O)CSc2nnc(s2)SCC(=O)Nc3ccccc3C#N NRB00264 Cc1ccc(cc1Cl)NC(=S)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-] AW00613 CCOC(=O)/C(=C\c1ccc(o1)[N+](=O)[O-])/C#N NRB00307 c1ccc(cc1)Oc2c(cccn2)c3nc(no3)c4ccc(cc4)Oc5ccc(cc5[N+](=O)[O-])C(F)(F)F BTB05547 c1ccc(c(c1)c2nc(no2)c3ccc(cc3)Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F)F BTB05548 c1cc2c(cc1[N+](=O)[O-])CCN2 RH00433 c1cc(c(cc1NC(=O)/C(=C/c2cc(cs2)Br)/C#N)Cl)F BTB05554 c1cc(c(c(c1)Cl)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F BTB05620 c1cc(c(cc1C(F)(F)F)NC(=O)CSc2ccc(cn2)C(F)(F)F)Cl NRB00315 c1cc(c(c(c1)Cl)C=C2C(=O)NC(=O)NC2=O)F BTB02083 c1ccc(cc1)Nc2nc(nc(n2)O)Nc3ccccc3 RH00424 Cc1ccccc1n2c(cc(=O)n(c2=O)Cc3ccc(cc3)OC)N KM09980 c1cc2c(ccnc2cc1Cl)Sc3nnc(s3)NC(=O)C4CC4 RH00420 c1ccc(c(c1)C(=O)O/N=C(/c2ccc(cc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)\N)F BTB05543 COc1ccc(cc1)/C(=C/c2cc(cs2)Br)/C#N BTB05550 Cc1ccc(cc1Cl)NC(=O)/C(=C/c2cc(cs2)Br)/C#N BTB05553 Cc1c2ccccc2sc1CNC(=O)c3ccc(cc3)C(F)(F)F MWP00839 c1ccc(c(c1)C(=O)NCCc2ccc(cc2)Cl)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05616 c1ccc(c(c1)C(=O)NCc2ccccn2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05618 C/C(=N\NC(=S)N)/C(OC)OC BTB05629 c1cc(c(cc1C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl)Cl BTB05624 c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00600 Cc1c(cccc1Cl)NC(=S)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F AW00603 c1ccc(cc1)CCNC(=S)N2CCC(CC2)O AW00605 c1ccc(c(c1)C#N)N2CCCCC2 BTB03852 c1ccc2c(c1)cc(c(=O)o2)C(=O)N3CCc4c3ccc(c4)[N+](=O)[O-] RH00437 CC(=O)N1CCc2c1ccc(c2)NC(=S)Nc3ccccc3Cl RH00441 CC(C)(C)SC(=S)SCC(=O)c1ccc(cc1)Cl BTB03856 Cc1nnc(s1)NCC(C)(C)C BTB03876 c1cc(ccc1SCC(=N)NS(=O)(=O)c2ccc(c(c2)Cl)F)Cl BTB05588 c1cc(ccc1C(=O)CC2(c3cc(ccc3N(C2=O)CN4CCCCC4)Br)O)Cl BTB02037 c1cc(ccc1C(=O)CC2(c3cc(ccc3N(C2=O)CN4CCOCC4)Br)O)Cl BTB02026 Cc1c2ccccc2sc1C(=S)NC MWP00780 Cc1ccc(c(c1)C)NC(=S)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F AW00599 Cc1cc(c(c(c1)C)NC(=O)CSCC(=O)c2ccc(cc2)Cl)C BTB04075 COc1c(c(c2c(n1)-c3ccccc3C2)c4ccccc4)C#N RH00520 CCCCn1c2ccccc2c3c(c1=O)c(cc(=O)o3)O RH00521 c1ccc(c(c1)C(=O)NCC(=O)c2ccc(cc2)Br)F BTB04142 c1cc(ccc1C(=O)CNC(=O)c2ccc(cc2)Cl)Cl BTB04144 CSc1c(c(nc(c1C#N)SCC(=O)c2cccc(c2)[N+](=O)[O-])N)C#N RH00573 Cc1c(ccc(n1)C(F)(F)F)NC(=O)/C=C\C(=O)O AW00670 CC(C)(C)c1ccc(cc1)C(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00673 CCCCc1ccc(c(c1)C)NC(=O)CSc2nnc(s2)N RH00525 CCCCc1ccc(c(c1)C)NC(=O)c2c(nn(n2)c3ccccc3)C RH00527 c1cc(nc(c1)NC(=O)c2ccc(cc2)[N+](=O)[O-])NC=C(C#N)C#N BTB04092 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2c(cc(cc2Cl)S(=O)(=O)N3CCOCC3)Cl BTB04095 CCC(C)NC(=S)NNC(=O)OCC BTB04017 CCCCc1ccc(c(c1)C)N/C=N/O RH00511 CCCCc1ccc(c(c1)C)NC(=O)NC(=O)c2ccccc2Cl RH00512 Cc1ccc(cc1)C(=O)c2ccccc2[N+](=O)[O-] RH00540 CSc1c(c(nc2c1c(c(s2)C(=O)c3ccc(cc3)OC(F)F)N)N)C#N RH00574 CCCCc1ccc(c(c1)C)NC=C(C(=O)OCC)C(=O)OCC RH00517 CCCCc1cc(c2c(c1)c(c(cn2)C(=O)O)O)C RH00522 c1cc(cc(c1)S(=O)(=O)N2CCOCC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB04072 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2c(cc(cc2Cl)S(=O)(=O)Nc3ccc(cc3F)F)Cl BTB04098 c1c(cc(c2c1nc(o2)S)Cl)Cl BTB04150 c1ccc(c(c1)C(=O)Nc2ccccc2N)O BTB04153 CC(C(=O)O)NCc1cc(cc(c1O)OC)Cl RH00578 CCCCc1ccc(c(c1)C)NC(=O)c2c(onc2c3ccccc3)C RH00526 c1cc(c(cc1NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl)Cl)F BTB04097 c1cc(c(c(c1)Cl)C(=O)Oc2ccc(cc2)F)Cl BTB04117 COc1ccc(cc1)NC(=S)NNC(=O)c2ccccc2[N+](=O)[O-] BLT00027 c1cc(ccc1[N+](=O)[O-])Oc2c(cc(cc2Cl)S(=O)(=O)N3CCCC3)Cl BTB04089 Cc1c(ccc(n1)C(F)(F)F)C(=O)O AW00680 c1cc([nH]c(=O)c1C(=O)N)C(F)(F)F AW00682 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCC(=O)c3ccc(cc3)Cl AW00683 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2c(cc(cc2Cl)S(=O)(=O)N3CCCCC3)Cl BTB04105 c1cc(ccc1C(=O)CN)Cl.Cl BTB04099 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2c(cc(cc2Cl)S(=O)(=O)N3CCCC3)Cl BTB04106 c1cc(cc(c1)[N+](=O)[O-])C(=O)CN.Cl BTB04110 c1cc(ccc1[N+](=O)[O-])Oc2c(cc(cc2Cl)S(=O)(=O)N3CCCCC3)Cl BTB04088 CCOC(=O)c1cc(c(nc1SCC(=O)OC)C)C(=O)OC AW00672 CC(C(=O)O)Sc1c(ccc(n1)OC)[N+](=O)[O-] RH00552 c1cc(ccc1C(=O)CN)Br.Cl BTB04111 c1ccc(c(c1)N)Sc2ccc(cc2[N+](=O)[O-])c3cnc4ccccc4n3 BLT00147 Cc1ccc(c(c1)[N+](=O)[O-])c2ccc(cc2[N+](=O)[O-])C MB00042 CCCCCc1ccc(cc1)C(=O)Nc2cc(cc(c2)Cl)Cl BR00004 c1cc(cc(c1)NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl)C(F)(F)F BTB04129 c1ccc2c(c1)ncc(n2)c3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl BLT00149 Cc1cc(ccc1NC(=O)NCc2ccc(cc2)C(=O)OC)C(=O)OC KM10094 c1ccc2c(c1)nnn2C3CCNCC3.Cl KM10095 Cc1cc(ccc1NC(=O)N(Cc2ccc(cc2)C(=O)OC)C(=O)C)C(=O)OC KM10102 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCC(=O)c3ccc(cc3)Br BTB04143 CC(C/N=C(\C)/c1cc(ccc1O)Cl)O BLT00231 c1ccc(cc1)NC(=O)c2ccc3c(c2)cccn3 KM10112 c1ccc(c(c1)C(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F)[N+](=O)[O-] BLT00023 CC(C)(C)c1ccc(c(c1)C(C)(C)C)OC(=O)c2ccc(cc2)[N+](=O)[O-] BTB04113 c1ccc(c(c1)C(=O)Oc2ccc(cc2)F)Cl BTB04116 COC(=O)c1ccc(o1)CSc2ccccc2N BLT00259 CCCCc1ccc(c(c1)C)NC(=O)CSc2cccc(c2Cl)Cl RH00530 c1cc(ccc1[N+](=O)[O-])Oc2c(cc(cc2Cl)S(=O)(=O)N3CCOCC3)Cl BTB04087 CCCCCCCc1ccc(cc1)NC(=O)Nc2ccccc2C(F)(F)F BR00015 CSc1ccccc1CNC(=O)NC23CC4CC(C2)CC(C4)C3 KM10103 c1ccc2c(c1)ncc(n2)c3ccc(c(c3)[N+](=O)[O-])Sc4ccccn4 BLT00150 c1ccc(c(c1)C(=O)Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F)O BTB04149 c1cc(ccc1OCC(CN2CCN(CC2)c3nc4ccc(cc4s3)Cl)O)SC(F)(F)F AW00641 c1cc(cc(c1)Cl)NC(=S)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00642 c1cc(sc1)C(=O)CCNc2ccc(cc2)Cl MWP00895 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccccc2F AW00653 Cc1c(ccc(n1)C(F)(F)F)C(=O)NNC(=O)c2cccs2 AW00654 CCOC(=O)C(C)(C(=O)OCC)Sc1c(c(c(c(n1)N)C#N)SC)C#N RH00559 c1cc(ccc1NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl)F BTB04114 CCCCCCCc1ccc(cc1)NC(=O)NNc2ccccc2C(F)(F)F BR00023 Cc1cc(c(c(c1CSc2ccccc2NC(=O)C(F)(F)F)C)CSc3ccccc3NC(=O)C(F)(F)F)C BLT00133 CCCCCc1ccc(cc1)C(=O)O/N=C/c2c(cccc2Cl)Cl BR00009 CC1CN(CC(O1)C)S(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3)[N+](=O)[O-])Cl BTB04090 c1cc(cc(c1)Cl)C(=O)Nc2cccc(n2)NC=C(C#N)C#N BTB04093 CCOC(=O)c1cc(c(nc1N2CCCN(CC2)Cc3ccc(cc3)F)C)C(=O)OC AW00650 CCCCc1ccc(c(c1)C)NC(=O)CSc2nnc(s2)NC(=O)c3ccc(c(c3)[N+](=O)[O-])N4CCCCC4 RH00546 c1cc(cc(c1)Cl)C(=O)NCC(=O)c2ccc(cc2)Cl BTB04100 CSc1c(c([nH]c(=S)c1C#N)N)C#N RH00551 CCCCCc1ccc(cc1)NC(=O)NNc2cc(cc(c2)C(F)(F)F)C(F)(F)F BR00026 CSc1c(c(nc(c1C#N)SCc2ccc(c(c2)F)F)N)C#N RH00560 CCCCCc1ccc(cc1)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl BR00028 CCCCc1ccc(c(c1)C)NC(=O)CSc2nnnn2c3ccccc3 RH00534 CCCCCc1ccc(cc1)C(=O)Nc2cccnc2 BR00007 c1ccc(cc1)n2cccc2c3nc(nc(n3)N4CC4)N5CC5 MB00046 c1ccc(c(c1)C(=O)NCC(=O)c2ccc(cc2)Cl)F BTB04146 c1ccc(c(c1)C(=O)Nc2ccccc2[N+](=O)[O-])O BTB04147 c1ccc(cc1)n2cc(c3c2cccc3)c4nc(nc(n4)N5CC5)N6CC6 MB00064 COC(=O)c1ccc(o1)CSc2ccccc2NC(=S)Nc3cccc(c3)C(F)(F)F BLT00262 CC(C(=O)O)NCc1ccc(c(c1)[N+](=O)[O-])Sc2ccc(cc2)Br RH00580 CCCCCCCc1ccc(cc1)NC(=O)NCc2ccccn2 BR00014 CCCCCCCc1ccc(cc1)C(=O)O/N=C/c2c(cccc2Cl)Cl BR00030 CCCCCc1ccc(cc1)C(=O)NC2=NCCS2 BR00038 c1cc(ccc1C(=O)NCC(=O)c2ccc(cc2)Br)Cl BTB04134 CN1c2ccccc2C(=O)NC1c3ccc(s3)[N+](=O)[O-] BTB02134 CC(=O)Nc1c(cccc1[N+](=O)[O-])C(=O)O RH00541 COC(=O)c1ccccc1CSc2ccccc2C(=O)O RH00537 COC(=O)c1cccc(c1)CSc2c(cccn2)C(=O)O RH00539 c1cc(c(nc1)SCc2csc3c2cc(cc3)Cl)[N+](=O)[O-] MWP00878 c1cc(=O)[nH]nc1c2ccncc2 RH00550 CC(C(=O)O)Sc1c(cccn1)[N+](=O)[O-] RH00553 Cn1c(nc(n1)/N=C/N(C)C)Sc2ccc(cn2)[N+](=O)[O-] RH00557 Cc1ccccc1C(=O)NCC(=O)c2ccc(cc2)Cl BTB04152 CCCCCCCc1ccc(cc1)C(=O)Nc2ccc(cc2)Cl BR00012 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02135 CC(=O)Nc1c(cccc1[N+](=O)[O-])C(=O)OC RH00481 CC(=O)c1cc(ccc1OCc2ccccc2)F RH00586 CC(C)c1ccc(cc1)NC(=O)CSCc2csc3c2cc(cc3)Cl MWP00884 c1cc(c(c(c1)Cl)C(=O)NC(=O)O/N=C\2/CCCc3c2cco3)Cl MWP00903 c1cc(c(cc1Cl)Cl)OCC(=O)NC2=NCCS2 BR00053 Cc1ccccc1C(=O)NCC(=O)c2ccc(cc2)Br BTB04133 c1ccc2cnc(cc2c1)C(=O)O CC04701 c1ccc(cc1)NCCC(=O)c2cccs2 MWP00890 Cc1ccc(c2c1c3ccccc3[nH]2)C RH00490 CCOC(=O)C1(C(=O)Nc2ccc(cc2O1)Cl)C RH00492 c1cc(c(c(c1)F)C#N)OCC(F)(F)F MWP00905 Cc1ccc(cc1[N+](=O)[O-])N2C(=O)CC(C2=O)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB02132 CSc1c(c(nc(c1C#N)SCC(=O)c2ccc(c(c2)Cl)Cl)N)C#N RH00570 Cc1ccccc1Oc2ccc(c(c2)Oc3ccccc3C)NC(=O)c4ccc(cc4)[N+](=O)[O-] BTB04141 CC1(CC2=C(C(C3=C(O2)CC(CC3=O)(C)C)c4ccc(s4)[N+](=O)[O-])C(=O)C1)C BTB02114 c1ccc2c(c1)C(=O)NC(N2)c3ccc(s3)[N+](=O)[O-] BTB02117 c1cc2c(cc1Cl)C(=O)NC(N2)c3ccc(s3)[N+](=O)[O-] BTB02123 CN1c2ccc(cc2C(=O)NC1c3ccc(s3)[N+](=O)[O-])Cl BTB02126 c1ccc(cc1)C(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00643 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3ccc4c(c3)CCN4C(=O)C RH00448 CC(=O)N1CCc2c1ccc(c2)NC(=O)c3c(c4ccccc4s3)Cl RH00451 Cc1ccc(cc1)S(=O)(=O)/C=C/c2ccc(o2)[N+](=O)[O-] NRB00390 c1ccc(cc1)CN2CCC(CC2)NCC(CSc3ccc(cc3)F)O AW00648 c1cc(c(cc1C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl)Cl BTB05625 c1cc(c(cc1Cl)Cl)C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05626 c1ccc(c(c1)C(=O)NCCCN2CCCCC2)NC(=O)c3ccc(cc3)[N+](=O)[O-] BTB05607 Cc1ccccc1n2ccc(=O)[nH]c2=O KM10067 Cc1cc(cc(c1O)C)CN2CC(CC(C2)C)C.Cl BTB04023 CC(=O)C(C)(C)OC(=O)NCCc1ccc(c(c1)OC)OC BTB05614 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])SCc2csc3c2cc(cc3)Cl MWP00879 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])SCc2csc3c2cc(cc3)Cl MWP00880 c1cc(c(c(c1)Cl)C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])F BTB05621 c1cc(ccc1C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl BTB05622 c1cc(c(c(c1)Cl)CN2CNC(=NC2)SCc3c(cccc3Cl)F)F.Br BTB03987 COc1ccccc1NC(=O)CSc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB02124 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc4c(c3)N(CC4)C(=O)C RH00455 Cc1cc2c(cc1C)CN(C2)c3ccccc3 MB00072 c1ccc(cc1)/C=C/2\CCCC3C2(OC4=C(C3c5ccccc5)CCCC4)N6CCCC6 RH00505 CCCCc1ccc(c(c1)C)N/C=N/OC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RH00513 c1cc2c(cc1Cl)c(=O)nc([nH]2)c3cc(cs3)Br BTB05608 c1cc(c(c(c1)Cl)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-])F BTB05627 c1ccc(c(c1)C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])F BTB05631 c1ccc(c(c1)C(=O)NCCc2ccncc2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05617 COc1cc(c(c(c1OC)OC)NS(=O)(=O)c2ccc(cc2)Cl)C(=O)OC BTB05619 c1cc(c(cc1S(=O)(=O)Nc2c(cc(cc2Br)F)F)Cl)Cl BTB03964 c1cc(cc(c1)Cl)NC(=O)O/N=C\2/CCCc3c2cco3 MWP00898 c1cc(c(c(c1)F)C(=O)NC(=O)O/N=C/2\CCCc3c2cco3)F MWP00902 c1ccnc(c1)Sc2c(cccn2)[N+](=O)[O-] BTB04043 c1cc(c(cc1F)F)NC(=O)NC(=O)CC#N KM10036 c1ccc(cc1)Sc2c(cccn2)[N+](=O)[O-] BTB04050 c1ccc(cc1)/C=C/2\CCCC3=C2OC4(CCCCC4C3c5ccccc5)N6CCCC6 RH00504 c1ccc(cc1)/C=C/2\CCCC3=C2OC(=C(C3c4ccccc4)C#N)N RH00506 c1cc(sc1)C(=O)Nc2c(cc(cc2Br)F)F BTB03963 Cc1ccc(cc1)C(=O)CC2(c3cc(ccc3N(C2=O)CN4CCCCC4)Br)O BTB02038 CCC(c1ccccc1)C(=O)NNC(=O)c2ccc(cc2)N(C)C BTB02040 CC(=O)Oc1cc(=O)n(c2c1cccc2)c3ccccc3 RH00514 CC1(CC(=O)C(C(=O)C1)C(c2ccc(s2)[N+](=O)[O-])C3=C(CC(CC3=O)(C)C)O)C BTB02113 Cc1ccc(cc1)S(=O)(=O)N/N=C(/CC(=O)OC)\C(=O)OC BTB04040 Cc1ccc(cc1[N+](=O)[O-])c2ccc(c(c2)[N+](=O)[O-])C MB00041 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F AW00645 CC(=O)OC(c1ccc(o1)[N+](=O)[O-])OC(=O)C RH00475 CCOC(=O)c1cnn(c1NC(=S)NC2CCCCC2)C(=O)COc3ccc(cc3C(C)(C)C)C(C)(C)C RH00477 Cc1c(ccc(n1)C(F)(F)F)C(=O)Oc2ccc3c(c2)OCO3 AW00651 CC(=O)Nc1ccc(cc1C(=O)OC)[N+](=O)[O-] RH00482 c1ccc(cc1)/C=N/C(c2ccccc2)c3c4ccccc4ccc3O RH00483 CC1CN(CC(O1)C)S(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl BTB04102 c1ccc(cc1)COc2ccc(cc2)C(F)(F)F BTB04014 COc1ccc(c(c1)[N+](=O)[O-])NC(=O)c2ccccc2O BTB04062 Cc1ccc(cc1)CC(=O)O MB00106 COc1ccc(cc1)NC(=O)NC(=O)CC#N KM10035 COc1ccc(cc1)n2c(cc(=O)[nH]c2=O)N KM10037 c1cc(c(cc1F)F)n2c(cc(=O)[nH]c2=O)N KM10039 Cc1cc(cc(c1O)C)CN2CCc3cc(c(cc3C2C)OC)OC.Cl BTB04037 c1ccc(cc1)CN2CCN(CC2)CCN3C(=O)c4ccccc4C3=O KM10043 Cc1ccccc1N2C(=O)CC(=O)NC2=O KM10050 c1ccc(cc1)CN2CCC(CC2)Nc3ccccc3[N+](=O)[O-] KM10051 c1cc(c(nc1)Sc2ncccn2)[N+](=O)[O-] BTB04045 c1cc(c(nc1)Sc2cc(ccc2Cl)Cl)[N+](=O)[O-] BTB04047 c1cc(nc(c1)NC=C(C#N)C#N)N BTB04071 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCN(CC2)C(=O)Nc3ccc(cc3F)F AW00652 CC(C)N1CCC(CC1)n2c3ccccc3nn2 KM10078 Cc1cccc(c1NC(=O)C(C)N2CCCCC2)C AW00661 CC1CC(CN(C1)Cc2cc(c(c(c2)Cl)O)Cl)C.Cl BTB04041 CCc1ccccc1n2c(=O)c3ccccc3nc2S AW00674 CC(C)(C)c1ccc(c(c1)C(C)(C)C)OC(=O)NC(=O)c2c(cccc2Cl)F BTB04121 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2c(cc(cc2Cl)S(=O)(=O)Nc3cc(cc(c3)Cl)Cl)Cl BTB04128 CC1CC(CN(C1)S(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl)C BTB04104 c1ccc(cc1)CN2CCC(CC2)Nc3ccccc3N KM10052 Cc1cc(nc2n1nc(c2NC(=O)C)C(C)(C)C)C(F)(F)F KM10065 COc1ccc(cc1)C(=O)c2ccc(cc2)[N+](=O)[O-] KM10068 CC1=NCCc2c1cc(c(c2)OC)OC BTB04055 c1cc(c(cc1F)F)NC(=O)CSc2ccc(cc2[N+](=O)[O-])Cl BTB04069 Cc1ccccc1n2cc(c(=O)[nH]c2=O)Br KM10080 COC(=O)c1ccc(o1)CSc2ccccc2NC(=S)Nc3cccc(c3)SC BLT00263 CC(=O)c1cc(cc(c1OC(=O)c2ccccc2Cl)Cl)Cl BLT00270 Cc1cc2c3c(c1)c4c(c(cc(=O)o4)O)c(=O)n3CCC2 RH00501 Cc1ccc(cc1)Sc2c(cccn2)[N+](=O)[O-] BTB04048 c1cc(c(nc1)Sc2ccc(cc2)Cl)[N+](=O)[O-] BTB04049 CCCCc1ccc(c(c1)C)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C RH00528 CC(=O)C(C(=O)C)Sc1nccc(n1)c2cccnc2 MWP01021 Cc1c(c(n[nH]1)C)Sc2nccc(n2)c3cccnc3 MWP01022 Cc1c(c(n(n1)S(=O)(=O)c2cccc(c2)C(F)(F)F)C)Sc3nccc(n3)c4cccnc4 MWP01024 Cc1c(c(n2c(n1)cc(n2)c3ccccc3)C)Sc4nccc(n4)c5cccnc5 MWP01028 c1cc(oc1)c2c(c(oc2c3ccco3)N)C#N NRB00495 c1ccc(cc1)S(=O)(=O)Cc2ccc(cc2)[N+](=O)[O-] NRB00498 c1cc(ccc1[N+](=O)[O-])OS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP00958 Cc1ccc(cc1)N/N=C\2/C(=NN(C2=O)C)Nc3ccccc3Cl MWP01011 CS(=O)(=O)NNc1nccc(n1)c2cccnc2 MWP01014 c1ccc(c(c1)S(=O)(=O)NNc2nccc(n2)c3cccnc3)Cl MWP01016 c1ccc2c(c1)nc(s2)SCc3ccc(cc3)[N+](=O)[O-] NRB00500 Cc1c(c(n(n1)C)C)Sc2nccc(n2)c3cccnc3 MWP01025 c1cc(ccc1/C=C/c2ccc(o2)[N+](=O)[O-])[N+](=O)[O-] NRB00506 c1ccc(cc1)C(C(=O)O)NC(=O)c2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-] NRB00430 COc1cccc(c1)NC(=O)C(c2ccccc2)C(=O)Nc3cccc(c3)OC RH00567 C=CCNC(=S)NNc1nccc(n1)c2cccnc2 MWP01032 CCc1nnc(s1)NC(=O)c2c(nn(n2)c3ccccc3)C BTB05752 CSc1c(c(nc(c1C#N)SCC(=O)c2ccc(cc2)OC(F)F)N)C#N RH00571 CC(C(=O)O)NCc1ccccc1O RH00576 CCOc1ccc(cc1)/C=N/NS(=O)(=O)c2ccc(cc2)C MB00159 CC(C(=O)O)NCc1cc2ccccc2cc1O RH00579 CSc1nn(c[n+]1c2ccccc2)c3ccccc3.[I-] NRB00426 CCCCc1ccc(c(c1)C)NC(=O)CSc2nnc(s2)NC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RH00569 COc1ccccc1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB04157 c1ccc(cc1)C(=O)CC2C(=C(C(=O)O2)Cl)Cl NRB00415 COc1cc(cc(c1OC)OC)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] BTB02136 CN(C)c1ccc(cc1)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] BTB02137 c1c(cc(cc1Cl)Cl)S(=O)(=O)NC(=N)CN2CCCCC2 BTB05645 CSc1c(c(nc2c1c(c(s2)C(=O)c3ccc(c(c3)F)F)N)N)C#N RH00572 Cc1ccc(cc1)C(=O)NC(c2ccccc2)C(=O)O NRB00431 Cc1c(c(c(cn1)CSCC(=O)Nc2ccccc2OC)CO)O BTB02141 COc1cc(c(c(c1OC)OC)NS(=O)(=O)c2cc(cc(c2)Cl)Cl)C(=O)OC BTB05657 c1cc(cc(c1)Cl)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05661 c1ccc2c(c1)c(=O)nc([nH]2)c3cc(cs3)Br BTB05667 Cc1ccccc1C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05641 CCOC(=O)COc1cccc2c1oc(=O)cc2C RH00584 c1cc(cc(c1)[N+](=O)[O-])C(=O)CNC(=O)c2ccc(cc2)Cl BTB04155 C1CSCCN1C(=O)CC#N BTB05671 CCOC(=O)c1cnn(c1NC(=O)c2cccc(c2)F)C(=O)COc3ccc(c4c3CCC4)C RH00608 Cc1c(c(c(cn1)CSCC(=O)Nc2cc(ccc2Cl)C(F)(F)F)CO)O BTB02142 Cc1c(c(c(cn1)CSCC(=O)Nc2ccccc2F)CO)O BTB02143 c1ccc(cc1)CC(C(=O)O)NCc2ccccc2O RH00596 CC(=CC(C(=O)O)NCc1ccccc1O)C RH00598 Cn1c2ccccc2c(=O)nc1c3cc(cs3)Br BTB05646 c1ccnc(c1)CCNc2ccc(cc2/N=C/c3ccc(s3)[N+](=O)[O-])C(F)(F)F BTB02153 c1cc(c(cc1C(F)(F)F)/N=C/c2ccc(s2)[N+](=O)[O-])N3CCCC3 BTB02154 COc1ccc(cc1OC)CCNc2ccc(cc2/N=C/c3ccc(s3)[N+](=O)[O-])C(F)(F)F BTB02155 Cc1cc(cc(c1Cl)C)Oc2nc(nc(n2)Oc3cc(c(c(c3)C)Cl)C)NCCSC(C)(C)C BTB05677 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3nnc(s3)C BTB05751 CCOC(=O)C(=CNNS(=O)(=O)c1ccc(cc1)C)C(=O)OCC BTB02212 Cc1ccc2c(c1)OC(N2)c3ccc(s3)[N+](=O)[O-] BTB02215 c1cc(c(c(c1OCC(F)(F)F)C#N)OCC(F)(F)F)S(=O)(=O)N2CCCC2 MWP00995 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc3c(c2)OCO3 BTB02165 c1cc(oc1)C(=O)NC2=NCCS2 BR00047 c1cc(c(cc1Cl)Cl)NCCC(=O)c2ccc(s2)Cl MWP00899 CC(C)c1ccc(cc1)NCCC(=O)c2ccc(s2)Cl MWP00901 c1cc(c(c(c1)OCC(F)(F)F)C#N)OCC(F)(F)F MWP00904 CC(=O)/C(=C/c1cccs1)/C#N NRB00397 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)Cl BTB05701 c1cc(cc(c1)Cl)NC(=O)OC2CCCCc3c2nccc3 MWP00940 c1cc(c(c(c1)Cl)C(=O)NC(=O)OCc2ccc(cc2Cl)Cl)F BTB04194 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)OCc3ccc(cc3Cl)Cl BTB04199 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccc(cc4)C(C)C)S RH00605 c1ccc(cc1)C(=O)O/N=C\2/CCCc3c2cco3 MWP00913 CCCCCc1ccc(cc1)NC(=O)NNc2ccc(c(c2)Cl)F BR00032 CC(C(=O)NC1=NCCS1)Oc2ccc(cc2Cl)Cl BR00054 CC1C(=NN(C1=O)c2ccccc2)C NRB00435 Cc1cc(no1)NC=C(C(=O)C)C(=O)C BTB05689 c1ccc(c(c1)c2csc(n2)N/N=C\3/CCCc4c3cco4)Cl MWP00931 CC(C)(C)c1ccc(cc1)Oc2nc(nc(n2)Oc3ccc(cc3)C(C)(C)C)NCCSC(C)(C)C BTB05680 Cc1cccc(c1Oc2nc(nc(n2)Oc3c(cccc3Cl)C)NCCSC(C)(C)C)Cl BTB05681 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3nncs3 BTB05748 CC1CN(CC(O1)C)C(=O)CC#N BTB05670 COc1ccc(c(c1)S(=O)(=O)Nc2c(cc(c(c2OC)OC)OC)C(=O)OC)OC BTB05674 c1cc(ccc1C(=O)O/N=C\2/CCCc3c2cco3)[N+](=O)[O-] MWP00915 c1cc(c(c(c1)Cl)Sc2c(=O)c(=O)c2Sc3c(cccc3Cl)Cl)Cl MWP00919 Cc1cc(nc2c1c(=O)n([nH]2)c3ccccc3)C NRB00461 c1ccc(cc1)NC(=O)O/N=C\2/CCCc3c2cco3 MWP00896 c1coc2c1/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/CCC2 MWP00920 CCOc1c(c(=O)c1=O)Nc2ccc(cc2)C(C)C MWP00924 CC(C)c1ccc(cc1)Nc2c(c(=O)c2=O)Nc3ccc(cc3)C(C)C MWP00926 COc1cccc(c1)Nc2c(c(=O)c2=O)Nc3cccc(c3)OC MWP00927 c1ccc(cc1)NC(=O)OC2CCCCc3c2nccc3 MWP00936 Cc1cc(no1)/N=C/N(C)C BTB05695 CC(=O)Nc1ccc(cc1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br BTB02195 Cc1cc(nc2c1C(=O)CC(C2)(C)C)C NRB00456 CCCCn1c(cc(c(c1=O)C#N)C)O RH00599 Cc1ccc(c2c1CCC2)OCc3nnc(n3C4CCCCC4)S RH00600 c1cc(c(cc1Cl)Cl)C(=O)O/N=C\2/CCCc3c2cco3 MWP00914 CN(C)C(=O)C(=O)c1c[nH]c2c1cccc2 MB00122 c1cocc1C=C2C(=O)OC3(CCCC3)OC2=O NRB00395 c1cc(ccc1N2CCCCC2)[N+](=O)[O-] BTB02173 CC\1=NOC(=O)/C1=C\c2ccccc2 NRB00441 c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccccc3 NRB00449 CCOC(=O)/C(=C/Nc1cc(on1)C)/C#N BTB05690 CC(C)(C)SCCNc1nc(nc(n1)Oc2cc(cc(c2)Cl)Cl)Oc3cc(cc(c3)Cl)Cl BTB05682 c1cc(c(c(c1)F)C(=O)Nc2nnc(s2)C(F)(F)F)F BTB02182 Cc1ccc(c(n1)C)C(=O)Nc2ccccc2 NRB00454 Cc1cc(n(c-2nn(c(=O)c12)c3ccccc3)c4ccccc4)C NRB00460 COc1cc(c(c(c1OC)OC)NC(=O)c2cc3ccccc3oc2=O)C(=O)OC BTB05660 COc1cc(c(c(c1OC)OC)NC(=O)c2ccc(o2)[N+](=O)[O-])C(=O)OC BTB05666 CC(=C1C(=O)NN(C1=O)c2ccccc2)C NRB00438 c1ccc(cc1)N/C=C\2/C(=NN(C2=O)c3ccccc3)Nc4ccccc4 NRB00436 c1ccc2c(c1)c(=O)nc3n2nc(s3)C(=O)c4ccc(c(c4)Cl)Cl BTB05707 CC(C)(C)SCCNc1nc(nc(n1)Oc2ccc(cc2)F)Oc3ccc(cc3)F BTB05679 Cc1cc(no1)NC=C(C#N)C#N BTB05691 c1ccc(c(c1)N2CCOCC2)[N+](=O)[O-] BTB02206 CCOC(=O)C(=CNNC(=O)C1C2CC(C1C(=O)O)C=C2)C(=O)OCC BTB02202 c1ccc(cc1)NC(=O)Nc2ccc(cc2)c3ccnc(n3)N MWP00950 c1cc(ccc1Nc2c(c(=O)c2=O)Nc3ccc(cc3)OC(F)(F)F)OC(F)(F)F MWP00928 c1ccc(cc1)CN2CCC3CCCCN3C2c4ccc(cc4)[N+](=O)[O-] BTB02191 CC(=C)n1c2ccccc2n(c1=O)c3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05647 COc1cc(c(c(c1OC)OC)NC(=O)c2cccc(c2)F)C(=O)OC BTB05658 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)Cl BTB02166 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(c(c2)Cl)Cl BTB02167 CN(C)c1ccc(cc1)CC(C#N)c2ccc(cc2)N BTB02170 CC(C)(C)SCCNc1nc(nc(n1)Oc2ccc(cc2)Cl)Oc3ccc(cc3)Cl BTB05676 c1cc(ccc1N/N=C/2\CCCc3c2cco3)[N+](=O)[O-] MWP00921 c1ccc(cc1)C2C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] NRB00446 c1cc2cccc3c2c(c1)NC(N3)c4cc(cc(c4O)Cl)Cl BTB02172 Cc1cc(c(c(c1)C)NC(=O)CSCc2cnc(c(c2CO)O)C)C BTB02139 Cc1c(c(c(cn1)CSCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)CO)O BTB02140 c1ccc(cc1)c2csc(n2)N/N=C/3\CCCc4c3cco4 MWP00930 COc1cccc(c1C(=O)Nc2nnc(s2)C(F)(F)F)OC BTB02181 CCOC(=O)N(/N=C/c1c(c2ccccc2s1)C)SC(Cl)(Cl)Cl MWP00981 Cc1ccc(cc1)/C=N/NS(=O)(=O)c2ccc(cc2)C BTB02158 c1cc2c(cc1Cl)NC(O2)c3ccc(s3)[N+](=O)[O-] BTB02163 c1cc(c(cc1C(F)(F)F)/N=C/c2ccc(s2)[N+](=O)[O-])N3CCOCC3 BTB02152 c1ccc2c(c1)NC(O2)c3ccc(s3)[N+](=O)[O-] BTB02161 c1ccc2c(c1)NC(N2)c3cc(cs3)[N+](=O)[O-] BTB02162 c1cc2c(nc1)C(CCCC2)OC(=O)c3ccc(cc3)Cl MWP00942 c1ccc(cc1)/C=C\2/C(=NOC2=O)c3ccc(cc3)[N+](=O)[O-] NRB00442 CC\1=NOC(=O)/C1=C\Nc2ccccc2 NRB00444 CC(=O)/C(=C/c1ccoc1)/C#N NRB00473 c1ccc(c(c1)CSC#N)[N+](=O)[O-] NRB00472 CC(=O)/C(=C/c1ccsc1)/C#N NRB00474 CCc1cc(c(s1)NC(=O)C(F)(F)F)C(=O)OCC BTB05736 CCCS(=O)(=O)c1ccc(cc1)NS(=O)(=O)c2c(c3cc(ccc3s2)Cl)C MWP00965 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc(c(c3)Cl)Cl)Cl MWP00968 COc1cccc(c1C#N)OCc2ccc(cc2)Cl MWP00986 CCOc1cccc(c1C#N)OCC(F)(F)F MWP00991 CC1(OC(=O)C(=Cc2ccc(o2)Br)C(=O)O1)C NRB00482 COc1ccccc1NC(=O)/C=N/O BTB05719 COc1cccc(c1C#N)OCc2ccccc2 MWP00985 c1cc(ccc1c2nc(cs2)CSC(=N)N)Br.Cl NRB00464 CC1(OC(=O)C(=Cc2ccoc2)C(=O)O1)C NRB00485 CCc1cc(c(s1)NC(=O)c2ccc(o2)[N+](=O)[O-])C(=O)OCC BTB05727 CCc1cc(c(s1)NC(=O)C(Cl)Cl)C(=O)OCC BTB05737 CCc1cc(c(s1)NC(=O)C(Cl)(Cl)Cl)C(=O)OCC BTB05738 CCc1cc(c(s1)NC(=O)c2cccc(c2)C(F)(F)F)C(=O)OCC BTB05729 c1ccc2c(c1)c(c(s2)C(=O)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl BTB02225 CCc1cc(c(s1)NC(=O)c2ccccc2F)C(=O)OCC BTB05730 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3nnc(s3)C4CC4 BTB05746 Cc1c(c(no1)NC=C(C(=O)C)C(=O)C)Br BTB05717 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCCCCO BTB05718 CCOC(=O)C(=CNNC(=O)CCc1ccc(cc1)O)C(=O)OCC BTB02230 Cc1ccc(c(c1)n2c(nc3ccc(cc3c2=O)Br)C)n4cccc4 BTB02237 CCOC(=O)C(=CNNC(=O)c1cccs1)C(=O)OCC BTB02211 Cc1ccc2c(c1)NC(O2)c3ccc(s3)[N+](=O)[O-] BTB02214 c1cc(ccc1Oc2nc(nc(n2)Oc3ccc(cc3)F)N4CCSCC4)F BTB05723 c1cc(ccc1Oc2nc(nc(n2)Oc3ccc(cc3)Cl)N4CCSCC4)Cl BTB05724 CC(C)(C)c1ccc(cc1)Oc2nc(nc(n2)Oc3ccc(cc3)C(C)(C)C)N4CCSCC4 BTB05725 c1cc(c(c(c1)Cl)C(=O)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl BTB02221 COc1ccc2c(c1)NC(N2)c3ccc(s3)[N+](=O)[O-] BTB02223 CCc1c(cc(s1)NC(=O)c2cc3ccccc3oc2=O)C(=O)OCC BTB05726 c1cc(c(cc1NC(=O)c2ccc(o2)[N+](=O)[O-])Cl)F BR00079 Cc1cc(no1)NS(=O)(=O)c2ccc(c(c2)Cl)F BTB05703 c1cc(c(cc1C(=O)CSC#N)Cl)Cl BTB05706 c1cc(cc(c1)OS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F)C(F)(F)F MWP00959 CCOC(=O)C(=CNNS(=O)(=O)c1ccc(cc1)Cl)C(=O)OCC BTB02241 c1cc(c(c(c1OCC(F)(F)F)C#N)OCC(F)(F)F)S(=O)(=O)N2CCOCC2 MWP00994 c1c(cc(c2c1[nH]c(n2)S)Br)C(F)(F)F BTB05749 Cc1c(c(no1)NC(=O)c2ccc(o2)[N+](=O)[O-])Br BTB05715 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=O)c3cccc(c3)F RH00606 Cc1cccc(c1)N2C(=O)CSC2=S MB00228 Cc1ccccc1N2C(=O)CSC2=S MB00230 CCc1cc(c(s1)NC(=O)c2cccnc2Oc3ccccc3)C(=O)OCC BTB05728 Cc1cc(cc(c1O)C)CN2CC(OC(C2)C)C.Cl BTB04022 c1ccc(c(c1)c2[nH]c3ccccc3n2)O BTB04025 c1ccc2c(c1)c(c[nH]2)/C=N/NC(=S)NC3CC3 BTB04026 Cc1nc2ccc(cc2c(=O)n1c3cc(ccc3N4CCOCC4)C(F)(F)F)Br BTB02235 c1ccc(cc1)c2nc(cs2)C3CC(=NN3c4ccccc4)c5ccc(cc5)Cl NRB00463 c1ccc(c(c1)N2CCCCC2)[N+](=O)[O-] BTB02207 CCOC(=O)CNC(=S)Nc1ccccc1N NRB00491 Cc1ccc(c2c1CCC2)OCc3nnc(n3Cc4ccccc4)S RH00590 Cc1ccc(c(c1)[N+](=O)[O-])NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02186 COc1ccc(c(c1)[N+](=O)[O-])NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02187 CN(C)c1ccc(cc1)C2N(CCC3N2CCCC3)Cc4ccccc4 BTB02192 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc(cc3)S(=O)(=O)C)Cl MWP00983 CN1C(=O)/C(=N/Nc2cccc(c2)Cl)/C(=N1)Nc3ccccc3Cl MWP01010 c1ccc(c(c1)NC(=O)CSCc2csc3c2cc(cc3)Cl)Cl MWP00881 COc1cccc(c1C#N)OCC(F)(F)F MWP00990 c1ccc(cc1)CN2CCC3CCCCN3C2c4ccc(c(c4)Cl)Cl BTB02205 CC(C)Oc1cccc(c1C#N)OCC(F)(F)F MWP00992 c1cc(cc(c1)Cl)NC(=O)Nc2ccc(cc2)c3ccnc(n3)N MWP00952 c1ccc(c(c1)C(=O)NC(=O)OCc2ccc(cc2Cl)Cl)Cl BTB04182 c1ccc(c(c1)C(=O)NC(=O)OCc2ccc(cc2Cl)Cl)F BTB04177 c1cc(c(c(c1)Cl)CSCC(=O)Nc2ccc(c(c2)Cl)F)F BTB04181 c1ccc(c(c1)C(=O)NNC(=S)N)Cl BTB04186 c1cc(oc1/C=C/C(=O)NCCCN2CCOCC2)[N+](=O)[O-] NRB00489 CCc1cccc(c1NC(=O)c2ccco2)C NRB00492 c1ccc(c(c1)c2ncc(o2)c3ccc(cc3)Br)F BTB04161 c1ccc2c(c1)cc(s2)C(=O)NN BTB04184 c1cc(c(cc1CS(=O)(=O)CC(=O)Nc2ccc(c(c2)Cl)F)Cl)Cl BTB04187 Cc1c(c(no1)c2c(cccc2Cl)F)c3ncc(o3)c4ccc(cc4)Br BTB04159 c1cc(ccc1c2ncc(o2)c3ccc(cc3)Br)Cl BTB04163 CCc1cccc(c1NC(=O)/C=C/c2ccco2)C NRB00494 Cc1ccccc1c2ncc(o2)c3ccc(cc3)Br BTB04158 c1ccc(c(c1)c2ncc(o2)c3ccc(cc3)Cl)F BTB04164 c1cc(ccc1c2cnc(o2)c3ccc(cc3)Cl)Cl BTB04165 c1cc(sc1)C(=O)OCc2ccc(cc2Cl)Cl BTB04171 c1cc(c(cc1CSCC(=O)Nc2ccc(c(c2)Cl)F)Cl)Cl BTB04176 c1cc(ccc1C(=O)OCc2ccc(cc2Cl)Cl)[N+](=O)[O-] BTB04173 c1cc(sc1)CNC(=O)c2ccc(o2)[N+](=O)[O-] BR00068 c1cc(oc1)CNC(=O)c2ccc(o2)[N+](=O)[O-] BR00069 c1cc(oc1C(=O)N2CCOCC2)[N+](=O)[O-] BR00070 c1cc(cc(c1)NC(=O)c2ccc(o2)[N+](=O)[O-])C(F)(F)F BR00086 COc1ccccc1NC(=O)c2ccc(o2)[N+](=O)[O-] BR00084 CCOC(=O)c1ccc(cc1)NC(=O)c2ccc(o2)[N+](=O)[O-] BR00076 c1cc(c(cc1C(F)(F)F)NC(=O)c2ccc(o2)[N+](=O)[O-])Cl BR00087 CC(=O)Nc1cccc(c1)OC MB00202 CC(=O)Nc1cccc(c1)Cl MB00204 c1cc(ccc1c2ncc(o2)c3ccc(cc3)Cl)[N+](=O)[O-] BTB04170 c1ccc(cc1)CC(=O)NC2=NCCS2 BR00064 c1cc(cnc1)CNC(=O)c2ccc(o2)[N+](=O)[O-] BR00067 c1cc(ccc1NC(=O)c2ccc(o2)[N+](=O)[O-])[N+](=O)[O-] BR00071 c1ccc(cc1)CNC(=O)c2ccc(o2)[N+](=O)[O-] BR00072 Cc1c(c(c(c(c1C)C)CSCC(=O)Nc2ccc(c(c2)Cl)F)C)C BTB04175 c1ccc(c(c1)NC(=O)c2ccc(o2)[N+](=O)[O-])F BR00073 c1cc(ccc1NC(=O)c2ccc(o2)[N+](=O)[O-])F BR00074 Cc1cc(no1)NC(=O)c2ccc(o2)[N+](=O)[O-] BR00078 COc1ccc(cc1)N2C(=O)CC(C2=O)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB02238 c1ccc(cc1)NC(=S)NNc2nccc(n2)c3cccnc3 MWP01031 CC(=O)Nc1cccc(c1)[N+](=O)[O-] MB00206 COc1cc(c(cc1Br)OC)Br MB00208 CC1=NN(C(=O)C1)c2ccc(cc2)Cl NRB00432 CN1C(=O)/C(=N/Nc2ccccc2)/C(=N1)Nc3ccccc3Cl MWP01004 c1cc(cnc1)c2ccnc(n2)NNC(=O)Nc3ccc(cc3)SC(F)(F)F MWP01009 c1ccc(c(c1)C(=O)O)I BTB05694 Cc1cc(no1)NS(=O)(=O)c2cc(cc(c2)Cl)Cl BTB05700 c1cc(ccc1c2ccnc(n2)N)NC(=O)Nc3ccc(cc3)OC(F)(F)F MWP00953 c1cc(cc(c1)S(=O)(=O)Nc2ccc(cc2)c3ccnc(n3)N)C(F)(F)F MWP00956 c1cc2c(cc1F)NC(N2)c3ccc(s3)[N+](=O)[O-] BTB02227 Cc1nc2ccc(cc2c(=O)n1c3ccccc3N4CCCCC4)Br BTB02229 Cc1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccc(cc4OCc5ccc(cc5)F)OCc6ccccc6 RH00643 CC(C)c1ccc(cc1)NC2(CCCCC2)C(=O)N BTB00068 CC(=O)Nc1cccc(c1C(=O)O)F BTB04253 COc1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)c3ncon3)OC BTB04259 COc1ccc(cc1)C2c3c4ccccc4ccc3OC25c6ccccc6C=CC5=O BTB04248 COc1ccc(c(c1c2cc[nH]n2)OCc3ccccc3)OC RH00646 c1cc(cc(c1)NC(=O)Oc2ccc(cc2Cl)F)C(F)(F)F BTB04231 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=O)CSc3nc(c(o3)c4ccccc4)c5ccccc5 RH00649 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Oc3ccc(cc3Cl)F BTB04233 Cc1cc2c3c(c1)c(cc(=O)n3CCC2)O RH00662 CCCCCCCC1N[C@@H](CS1)C(=O)O RH00665 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CC4)O RH00671 c1ccc2cc(ccc2c1)C(=O)CC3(c4cc(ccc4NC3=O)Br)O BTB00081 CC(=O)N1c2ccccc2C=Cc3c1cccc3 RH00650 Cc1ccc2c(c1)CCCN2C(=O)CC(=O)N3CCCc4c3ccc(c4)C RH00658 c1ccc(cc1)C(C(=O)N2CCc3c2cccc3)C(=O)N4CCc5c4cccc5 RH00659 CCCCCCCCCCC1N[C@@H](CS1)C(=O)O RH00666 CC(C)(C)C1N[C@@H](CS1)C(=O)O RH00667 CCC1(C(=C)S/C(=N\c2ccc(cc2)C(C)(C)C)/N1)CC BTB04289 CCC1(C(=C)S/C(=N\c2ccc(c(c2)Cl)F)/N1)CC BTB04291 c1ccc(c(c1)C(=O)O)Sc2ccc(cc2)[N+](=O)[O-] NRB00552 COc1ccc(cc1)Sc2ccccc2C(=O)O NRB00553 c1ccc(c(c1)C(=O)O)Sc2cc(c(cc2C(=O)O)Sc3ccccc3C(=O)O)C(=O)O NRB00556 Cc1c2ccccc2sc1/C=N/NC(=O)NCc3ccccc3 MWP01087 COc1ccc2ccccc2c1Br RH00653 C=CCSc1ccc(c(c1OCC(F)(F)F)C#N)OCC(F)(F)F MWP01081 Cc1ccc(cc1[N+](=O)[O-])C(=O)NCC(=O)O RH00657 c1ccc(cc1)C(C(=O)Nc2ccccc2)C(=O)Nc3ccccc3 RH00661 Cc1c(nn(n1)c2ccccc2)C(=O)N3CCCN=C3SC BTB05765 CCCCCCCc1ccc(cc1)C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05768 C1CC1NC(=O)C(Cl)Cl BTB04284 C1CC1NC(=O)C(Cl)(Cl)Cl BTB04285 CCOC(=O)c1c(c2ccccc2n(c1=O)C)O BTB05773 CSC(=S)Nc1ccc(cc1F)F BTB05775 c1ccc(cc1)C(=N)Nc2ccc(c(c2)Cl)Cl BTB04299 CCCCCCCCCCCC1N[C@@H](CS1)C(=O)O RH00669 c1ccc(cc1)CC/N=C/c2ccccc2 RH00673 c1ccc(cc1)CSc2nc3ccccc3s2 NRB00501 CC(=O)CSc1ccc(c(c1OCC(F)(F)F)C#N)OCC(F)(F)F MWP01082 Cc1cc(ccc1[N+](=O)[O-])C(=O)NN RH00675 CCOC(=O)C1=C(NC(=C(C1)C(=O)OCC)C)C NRB00518 c1cnc(nc1)Sc2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01068 c1cc(ncc1C(F)(F)F)Sc2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01070 c1cc(ccc1N2CCOCC2)[N+](=O)[O-] BTB05771 CN1c2ccccc2C(=O)NC1C3CCC=CC3 BTB02254 c1cc2c(cc1[N+](=O)[O-])C(=O)NC(N2)C3CCC=CC3 BTB02255 CC(C)(C)NC(=S)NC1CC1 BTB04286 CCC1(C(=C)S/C(=N\c2cc(cc(c2)Cl)Cl)/N1)CC BTB04290 CCC1(C(=C)S/C(=N\c2ccc(cc2F)F)/N1)CC BTB04293 Cc1cc(n(n1)c2ccccc2)OC(=O)c3c(nn(n3)c4ccccc4)C BTB05791 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(cc1)F BTB05793 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(c(c1)F)F BTB05794 Cc1ccc(cc1Cl)NC(=O)/C(=C/N(C)C)/C#N BTB05795 c1ccc(c(c1)C(=O)NC(=O)NC2CC2)Cl BTB04268 COc1ccc(c(c1)S(=O)(=O)NC2CC2)OC BTB04270 CCc1cc(c(s1)NC(=S)Nc2ccccc2F)C(=O)OCC BTB05753 Cc1ccc(c(c1)C)C(=O)CC2(c3cc(ccc3NC2=O)Br)O BTB00089 CCc1cc(c(s1)NC(=S)Nc2ccccc2C(F)(F)F)C(=O)OCC BTB05754 CCc1cc(c(s1)NC(=S)Nc2cccc(c2)Cl)C(=O)OCC BTB05755 CCCCCCCc1ccc(cc1)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05767 CCCCCCCc1ccc(cc1)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-] BTB05769 CCOC(=O)C(=CNNC(=O)c1ccc(cc1)OC)C(=O)OCC BTB02243 CCOC(=O)CCc1ccc2c(c1)NC(O2)c3ccc(cc3)N(C)C BTB02246 c1ccc(cc1)/C=N/Nc2nccc(n2)c3cccnc3 MWP01035 c1cc(cnc1)c2ccnc(n2)N/N=C/c3ccc(cc3)[N+](=O)[O-] MWP01036 Cc1cc(n(n1)c2ccccc2)OC(=O)c3cccnc3Oc4ccccc4 BTB05800 CCOC(=O)CCc1ccc2c(c1)NC(O2)c3cccc(c3)[N+](=O)[O-] BTB02245 CCOC(=O)C(=CNNc1cccc(c1)Cl)C(=O)OCC BTB02250 CCC(c1ccccc1)C(=O)NNC(=O)c2ccccc2N BTB02251 CN1c2ccc(cc2C(=O)NC1C3CCC=CC3)Cl BTB02256 Cc1ccc(cc1)NC(=O)c2ccccc2N BTB02268 Cc1cc(n(n1)c2ccccc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05798 Cc1cc(n(n1)c2ccccc2)OC(=O)c3c(onc3c4ccccc4)C BTB05801 CCOC(=O)C(=CNNS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)OCC BTB02242 COc1ccc(cc1OC)CCNC(=O)c2ccccc2N BTB02272 Cc1cc(c(cc1Cl)C)S/C(=C/N(C)C)/C(=O)OC BTB05848 Cc1ccc(cc1)Sc2cccc(c2C#N)F MWP01124 Cc1cc(n(n1)c2ccccc2)OS(=O)(=O)c3ccc(cc3)Cl BTB05856 Cc1cc(n(n1)c2ccccc2)OS(=O)(=O)c3ccc(c(c3)Cl)F BTB05859 CN(C)/C=N/c1nnc(s1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05862 c1ccc(cc1)CSc2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01076 c1ccc(c(c1)CSc2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F)Cl MWP01078 COC(=O)c1ccc(o1)CS(=O)(=O)C(Cl)(Cl)Cl NRB00517 Cn1c2ccc(cc2c(=O)s1)S(=O)(=O)NC3CC3 BTB04272 COc1cc(cc(c1OC)OC)C2Nc3c(c4c(s3)CCCC4)C(=O)N2 BTB02257 CN(C)c1ccc(cc1)C2Nc3c(c4c(s3)CCCC4)C(=O)N2 BTB02258 c1cc2c(cc1C3Nc4c(c5c(s4)CCCC5)C(=O)N3)OCO2 BTB02259 c1cc(ccc1C2Nc3c(c4c(s3)CCCC4)C(=O)N2)Cl BTB02271 Cc1ccc(cc1)c2cnc(sc2=O)c3ccccc3 BTB05845 c1c(cc(c2c1[nH]c(n2)S)Cl)C(F)(F)F BTB05757 c1cc(cc(c1)C(F)(F)F)C(=O)NC2CC2 BTB04273 c1c(cc(cc1Cl)Cl)C(=O)NC2CC2 BTB04274 Cc1c(nn(n1)c2ccccc2)C(=O)N3CCN=C3SC BTB05759 CCCCCc1ccc(cc1)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-] BTB05763 Cc1nnc(s1)/N=C/N(C)C BTB05812 Cc1cc(c(cc1Cl)Cl)SCC(=O)OC BTB05823 c1cc(c(cc1C(F)(F)F)N)N2CCCC2 BTB05831 c1cc(c(cc1NC(=O)Cc2n[nH]nn2)Cl)F BTB05818 Cc1cc(c(cc1Cl)Cl)S/C(=C\N(C)C)/C(=O)OC BTB05846 Cc1cc(c(cc1Cl)C)S(=O)(=O)CC(=O)OC BTB05847 Cc1ccc(cc1)Oc2cccc(c2C#N)F MWP01110 c1cc2c(c(c1)Oc3ccc(cc3)F)c(nc(n2)N)N MWP01114 CC1COC(N1)c2cccc(c2)[N+](=O)[O-] BTB02247 c1ccc(cc1)NC(=O)c2ccccc2N BTB02274 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)N BTB02266 Cc1ccc(c(c1)C)NC(=O)c2ccccc2N BTB02269 c1ccc(cc1)n2cc(c(n2)N)C#N BTB02273 c1cc(cnc1)c2ccnc(n2)N/N=C/c3ccc(cc3Cl)Cl MWP01034 c1ccc(cc1)n2c(c(c(n2)CC#N)C#N)/N=C/c3cc(cc(c3O)Cl)Cl BTB02284 c1ccc(cc1)C(c2ccccc2)(C(=O)NN)O BTB02286 c1cc(cc(c1)Cl)CNC(=O)N/N=C/c2cccs2 MWP01092 c1ccc(c(c1)c2c(c(ns2)N3CCOCC3)C#N)Cl MWP01097 CC(C)(C)NC(=S)N/N=C\1/CCCc2c1cco2 MWP01100 c1cc(ccc1C(=O)N/N=C\2/CCCc3c2cco3)[N+](=O)[O-] MWP01101 Cc1cc(c(cc1Cl)C)SCC(=O)OC BTB05824 CC(c1ccccc1)NC(=O)c2ccccc2N BTB02285 Cc1cc(c(c(c1)C)NC(=O)CSc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C BTB05826 COc1cccc2c1nc(s2)NC=C(C#N)C#N BTB05808 Cc1cc(c(c(c1)C)NC(=O)CS(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(F)(F)F)C BTB05827 c1cc(c(c(c1)Sc2ccc(cc2)Cl)C#N)F MWP01125 CCc1nnc(s1)N/C=N/O BTB05809 c1cc(c(cc1F)F)NC(=O)Cc2n[nH]nn2 BTB05819 c1cc(ccc1NC(=O)Cc2n[nH]nn2)F BTB05821 Cc1ccc(c2c1CCC2)OCC(=O)NNS(=O)(=O)c3ccc(cc3C)[N+](=O)[O-] RH00633 CC(=O)c1c(ccc(c1OCc2ccccc2)OC)OC RH00634 c1cc(sc1)C(=O)O/N=C(/c2ccc(cc2)[N+](=O)[O-])\N BTB04193 c1ccc(cc1)Oc2cccc(c2C#N)F MWP01102 C1CN2CCC1C(C2)(C#N)O.Cl MWP01104 c1cc(c(c(c1)F)C#N)OCc2ccc(cc2)Cl MWP01122 Cc1ccc(cc1)n2nc(nn2)c3ccc(cc3)Cl BTB02294 c1cc(cc(c1)Cl)n2c(c(cn2)C#N)N BTB02305 Cn1c(c(c(n1)CC#N)C#N)N BTB02279 c1ccc(cc1)/C=C\2/C(=NOC2=O)CSc3ccccc3 MWP00909 Cc1ccc(c2c1CCC2)OCC(=O)N/N=C/c3ccccc3Cl RH00613 CSCCC(C(=O)O)NCc1ccccc1O RH00618 CN(C)/C=N/c1nnc(s1)Sc2ccc(cn2)[N+](=O)[O-] BTB05864 CN(C)/C=N/c1nnc(s1)Sc2c(cccn2)[N+](=O)[O-] BTB05865 CN(C)/C=N/c1nnc(s1)SCC(=O)c2ccc(cc2)F BTB05866 c1ccc2c(c1)cccc2Sc3cccc4c3cccc4 NRB00548 c1cc2c(c(c1)OCc3ccc(cc3)C(F)(F)F)c(nc(n2)N)N MWP01126 c1ccc(c(c1)CSc2ccccc2C(=O)O)C(=O)O NRB00557 c1cc2cccc(c2c(c1)C(=O)O)SCCC(=O)O NRB00559 Cc1c2ccccc2sc1/C=N/NC(=O)NCc3ccc(cc3)Cl MWP01089 c1ccc(c(c1)c2c(c(ns2)N3CCSCC3)C#N)Cl MWP01098 c1ccc(cc1)n2c(c(cn2)C(=O)N)N BTB02287 c1ccc(c(c1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] BTB02288 c1ccc(cc1)n2c(c(cn2)C#N)n3cccc3 BTB02289 c1ccc(cc1)n2c(c(c(n2)CC#N)C#N)n3cccc3 BTB02290 Cc1c(c(n[nH]1)C)c2ccc(cc2C(=O)O)OC BTB04228 c1cc(c(c(c1)Cl)NC(=O)Oc2ccc(cc2Cl)F)Cl BTB04230 Cc1c(c(c(c(c1C)C)CS(=O)(=O)CC(=O)Nc2ccc(c(c2)Cl)F)C)C BTB04189 COc1ccc(cc1OC)CCNC(=O)c2cccc(c2)Cl MB00248 c1cc(c(c(c1)Cl)CS(=O)(=O)CC(=O)Nc2ccc(c(c2)Cl)F)F BTB04191 CCOC(=O)C1C(CC(=CC1=O)c2ccc(cc2)C)c3ccccc3 BTB00009 c1ccc2c(c1)cccc2/C=C/c3ccc(cc3)F BTB00016 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=S)N BTB04202 c1cc(oc1)C(=O)NNC(=S)N BTB04204 CC1CN(CC(O1)C)c2ccc(cc2)[N+](=O)[O-] BTB04206 CC(C)(C)C(=O)Nc1ccc(cc1[N+](=O)[O-])F BTB04214 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=O)CSc3cc(cc(c3)C)C RH00648 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=O)Cc3ccccc3 RH00627 Cc1ccc(c2c1CCC2)OCC(=O)N/N=C/c3cccc(c3)C(F)(F)F RH00611 Cc1c(c(n(n1)C)C)c2ccc(cc2C(=O)O)OC BTB04229 C1CCCCCC(=O)C(CCCC1)CN2CCOCC2.Cl BTB00006 COc1cc2c(cc1OC)C(=NCC2)c3ccc(cc3)Cl MB00252 c1ccc(c(c1)NC(=S)NCc2ccco2)Cl BTB00025 c1cc(cc(c1)NC(=S)NCc2ccco2)C(F)(F)F BTB00026 Cc1ccccc1NC(=S)NCc2ccco2 BTB00030 c1cc(ccc1/C(=N/OC(=O)c2ccc(cc2)Cl)/N)[N+](=O)[O-] BTB04198 CC(C)(C)C(=O)Nc1ccc(cc1)F BTB04212 COc1cccc(c1)NC(=S)NCc2ccco2 BTB00027 Cc1cccc(c1)NC(=S)NCc2ccco2 BTB00028 c1ccc2c(c1)cc(s2)C(=O)N3CCOCC3 BTB04217 CC1CCN(CC1)C(=O)c2cc3ccccc3s2 BTB04219 CC(=O)C(=CNc1ccc(cc1)Br)C(=O)C BTB04226 Cc1ccc(c2c1CCC2)OCC(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F RH00630 COc1ccc(cc1OC)CCNC(=O)c2ccc(cc2)Cl MB00249 Cc1cc(cc(c1)N2C(CC(=N2)c3cc(ccc3OCc4ccccc4)F)c5cccc(c5)C(F)(F)F)C RH00632 COc1ccc(cc1)N(Cc2ccccc2)Cc3ccccc3 RH00629 c1ccc(cc1)C(=O)CSc2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01077 COc1ccccc1NC(=S)NCc2ccco2 BTB00033 Cc1cccc(c1NC(=S)NCc2ccco2)C BTB00035 CC(c1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccc(cc3)C(C)C)/CCC2)C BTB00039 C/C(=N\O)/c1cc2ccccc2o1 BTB04227 c1ccc2c(c1)cccc2NC(=S)NCc3ccco3 BTB00034 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])NN=C(C2CC2)C3CC3 BTB00042 c1ccc(cc1)COc2ccc(cc2C3=NN(C(C3)c4cccc(c4)C(F)(F)F)c5ccccc5)F RH00628 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3Cl)F BTB04235 c1ccc2c(c1)c(c(s2)C(=O)Oc3ccc(cc3Cl)F)Cl BTB04237 c1ccc2c(c1)cc(s2)C(=O)Oc3ccc(cc3Cl)F BTB04238 C1CC1N2CNC(=S)NC2 BTB04258 c1ccc(cc1)COc2ccc(cc2C3=NN(C(C3)c4cccc(c4)C(F)(F)F)c5ccc(cc5Cl)Cl)F RH00631 Cc1ccc(c2c1CCC2)OCC(=O)NNS(=O)(=O)c3ccc(cc3)C(C)C RH00635 Cc1ccc(c2c1CCC2)OCC(=O)NNS(=O)(=O)c3ccc(c(c3)OC)OC RH00636 COc1c(cc(c(c1C(=O)O)OC)[N+](=O)[O-])[N+](=O)[O-] RH00642 c1cc(cc(c1)S(=O)(=O)NNc2nccc(n2)c3cccnc3)C(F)(F)F MWP01013 Cc1c(c(no1)c2ccccc2Cl)C(=O)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB02220 CC\1CC(C/C1=N\Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])(C)C BTB00043 CC(=O)Nc1cc(ccc1OC)Cl RH00651 c1ccc(c(c1)C(=O)NC(=O)NC2CC2)F BTB04267 CCOc1ccccc1NC(=O)Oc2ccc(cc2Cl)F BTB04234 C1CCC(CC1)NC2(CCCCC2)C(=O)N BTB00070 Cc1c(c(n(n1)c2ccccc2)C)c3ccc(cc3C(=O)O)OC BTB04246 CCOC(=O)CCc1ccc2c(c1)NC(O2)c3ccc(s3)[N+](=O)[O-] BTB02226 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=O)CSc3cc(ccc3Cl)Cl RH00641 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])S(=O)(=O)CC(=O)Nc2ccc(cc2F)F BTB04243 c1cc(c(cc1CSC2=NCN(CN2)C3CC3)Cl)Cl.Br BTB04278 CCOc1c(c(c(c(n1)N)C#N)c2ccccc2)C#N RH00654 c1cc(c(c(c1)Cl)CSC2=NCN(CN2)C3CC3)F.Br BTB04280 c1cc(cc(c1)C#N)CSC2=NCN(CN2)C3CC3.Br BTB04281 c1cc(ccc1C(=O)/C=C/c2ccc3c(c2)OCO3)[N+](=O)[O-] BTB00062 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3ccc[nH]3)/C#N)C#N)n4cccc4 BTB02402 CC(=O)Nc1ccc(cc1C(=O)C(=O)Nc2cccc(c2)OC)Br BTB00245 c1ccc(cc1)C(=O)Oc2c(cc(cc2Cl)Cl)/C=N/c3ccc(cc3)Cl BTB00251 c1c(c(cc(c1[N+](=O)[O-])N2CCCCC2)N3CCCCC3)C(F)(F)F BTB02411 c1ccc(c(c1)n2c(nnc2S)CCc3nc(no3)c4ccc(cc4)Cl)F BTB02336 CC(C)NS(=O)(=O)c1ccccc1I NRB00630 CCCCNS(=O)(=O)c1ccccc1I NRB00631 CC(C)(C)c1cc(c(c(c1)[N+](=O)[O-])OC(=O)c2ccc(cc2Cl)Cl)C(C)(C)C BTB04319 CC(C)(C)c1cc(c(c(c1)[N+](=O)[O-])OC(=O)c2cccnc2Oc3ccccc3)C(C)(C)C BTB04322 Cc1cc(c(cc1)/C(=N/N=C(/c2c(cc(cc2)C)C)\C)/C)C BTB00224 C/C(=N\N=C(\c1cc(ccc1)[N+](=O)[O-])/C)/c2cc(ccc2)[N+](=O)[O-] BTB00229 C/C(=N\N=C(\c1ccc(cc1)[N+](=O)[O-])/C)/c2ccc(cc2)[N+](=O)[O-] BTB00232 CCOC(=O)C1=C(N=C2N(C1c3ccccc3)CCS2)C.Br RH00700 CCc1c(cc2c(c1)C(CCC2(C)C)(C)C)/C(=N/N=C(/c3c(cc4c(c3)C(CCC4(C)C)(C)C)CC)\C)/C BTB00233 CCOC(=O)c1cnc(nc1N)Sc2ccc(cn2)[N+](=O)[O-] BTB04333 C/C(=N\N=C(\c1ccc(cc1)O)/C)/c2ccc(cc2)O BTB00236 c1ccc(c(c1)/C=N/c2cccc(c2)C(F)(F)F)O BTB00240 c1c(cc(c(c1C(=O)O)c2c(cc(cc2Cl)Cl)C(=O)O)Cl)Cl NRB00622 c1ccc(cc1)CNS(=O)(=O)c2ccccc2I NRB00635 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)c5c4cccc5)O RH00679 c1cc2c(cc1Cl)C(=O)C(=O)N2 RH00683 CCOC(=O)C1=C(NC(=S)NC1c2ccccc2)C RH00687 Cc1cc(n(n1)c2ccccc2)OC(=O)c3cccc(c3)F BTB05857 CCOC(=O)c1cnc(nc1N)Sc2c(cc(cc2[N+](=O)[O-])[N+](=O)[O-])C BTB04332 CC(C)(C)c1ccc(s1)C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F MBE00191 c1ccc(cc1)S(=O)(=O)/N=C(/NCCc2ccccn2)\Nc3cccc(c3)Cl NH00011 c1ccc(cc1)S(=O)(=O)/N=C(/Nc2cccc(c2)Cl)\SCC(=O)O NH00052 CC(=O)c1ccc(c(c1)CS/C(=N\S(=O)(=O)c2ccccc2)/Nc3cccc(c3Cl)Cl)OC NH00042 CCOc1ccc(cc1)NC(=O)C(=O)c2cc(ccc2NC(=O)C)Br BTB00244 c1cc(ccc1CCc2nnc(n2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)S)O BTB02381 CN1CCC(=N1)/C=C/c2cccs2.Cl MWP01209 Cc1cc2c3c(c1)c(c(c(=O)n3CCC2)c4ccccc4)OCc5c(cccc5Cl)Cl RH00694 Cc1ccc(c(c1)COc2c3cc(cc4c3n(c(=O)c2c5ccccc5)CCC4)C)C RH00696 Cc1ccc(cc1)COc2c3cc(cc4c3n(c(=O)c2c5ccccc5)CCC4)C RH00698 CCCCCc1ccc(cc1)C(=O)NN RH00701 c1ccc(c(c1)C(=O)NCCCn2ccnc2)N BTB04308 c1ccc(c(c1)C(=O)NCCCn2ccnc2)NS(=O)(=O)c3ccc(cc3)Cl BTB04309 c1ccc(c(c1)C(=O)NCCCn2ccnc2)NC(=O)c3ccc(cc3)[N+](=O)[O-] BTB04310 CCc1ccc(cc1)c2ccc(cc2)OC(=O)c3c(cc(cc3Br)C(F)(F)F)[N+](=O)[O-] BTB05867 c1cc(c(c(c1)Cl)C(=O)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl)Cl BTB02325 Cc1ccc(cc1)NS(=O)(=O)c2ccccc2I NRB00637 CCCCc1cc(c2c(c1)c(cc(n2)c3ccc(c(c3)OC)OC)C(=O)O)C RH00682 c1ccc(cc1)CNC(=S)NNC(=O)c2ccccc2 RH00686 CCOC(=O)C(=CNNC(=O)c1ccccc1n2cccc2)C(=O)OCC BTB02389 c1cc(ccc1c2ccc(s2)C(=O)Oc3ccc(cc3Cl)Cl)Cl MBE00090 c1cc(oc1)COC(=O)c2ccc(s2)c3ccc(cc3)Cl MBE00105 CCCCC(C(=O)O)C(=O)O RH00690 CC(=O)Nc1ccc(cc1)NS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01147 Cc1cc(c(cc1Cl)C)S(=O)(=O)/C(=C/N(C)C)/C(=O)OC BTB05851 Cc1cc(n(n1)c2ccccc2)OS(=O)(=O)c3ccc(c(c3)Cl)Cl BTB05852 c1cc(ccc1NC(=O)CSc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F BTB05855 c1ccc(cc1)c2nnc(o2)c3csc(n3)c4cccnc4 MWP01171 c1cc2cccc(c2c(c1)C(=O)O)I NRB00572 COc1cc(c(cc1SCC(=O)NNC(=O)c2cccc(c2)[N+](=O)[O-])OC)[N+](=O)[O-] BTB02342 c1ccc(cc1)Oc2c(cccn2)C(=O)NCC3CC3 BTB05869 c1cc(ccc1c2ccc(s2)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl MBE00085 Cc1cc(no1)NC(=O)NC(=O)c2c(cccc2Cl)Cl BTB05837 Cc1cc(no1)NC(=O)NC(=O)c2c(cccc2Cl)F BTB05838 CCOC(=O)/C(=C/N(C)c1ccc(cc1)O)/C#N BTB05840 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])n2c(c(cn2)C#N)N BTB02343 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)CC(=O)OC BTB05844 CC(C)(C)c1ccc(cc1)OC(=O)c2ccc(s2)C(C)(C)C MBE00155 Cc1c(c(no1)NC(=O)NC(=O)c2c(cccc2Cl)F)Br BTB05841 Cc1c(c(no1)NC(=O)NC(=O)c2ccccc2F)Br BTB05842 Cc1c(c(no1)NC(=O)NC(=O)c2c(cccc2Cl)Cl)Br BTB05843 c1cc(c(cc1Cl)S(=O)(=O)N)Cl NRB00580 c1ccc(cc1)CS(=O)c2ccccc2 NRB00581 CS(=O)c1ccc(cc1)[N+](=O)[O-] NRB00582 COc1cc(c(cc1Cl)OC)n2c(nnc2S)CCc3nc(no3)c4ccc(cc4)Cl BTB02340 Cc1cccc(c1)C(=O)NNC(=O)CSc2cc(c(cc2OC)[N+](=O)[O-])OC BTB02341 CCOC(=O)c1c(c(sc1Nc2ccccc2C(F)(F)F)C(=O)c3ccc(cc3)Cl)N MBE00252 c1ccc2c(c1)cccc2Sc3cccc4c3c(ccc4)C(=O)O NRB00561 c1cc2c(cc1NC(=O)N)cn[nH]2 BTB05835 Cc1ccc(cc1)NC(=S)NNC(=O)CSc2cc(c(cc2OC)[N+](=O)[O-])OC BTB02332 Cc1c(cccc1Cl)n2c(nnc2S)CSc3cc(c(cc3OC)[N+](=O)[O-])OC BTB02348 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2csc(n2)c3cccnc3 MWP01172 Cc1c(cccc1Cl)NC(=S)NNC(=O)CSc2cc(c(cc2OC)[N+](=O)[O-])OC BTB02328 COc1cc(c(cc1SCC(=O)NNC(=S)Nc2ccc(cc2)F)OC)[N+](=O)[O-] BTB02329 Cc1ccc(c(c1)C)NC(=S)NNC(=O)CSc2cc(c(cc2OC)[N+](=O)[O-])OC BTB02331 COc1ccc(cc1)NS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01135 c1ccc2c(c1)C(=O)c3cccc(c3C2=O)Sc4cccc5c4C(=O)c6ccccc6C5=O NRB00567 CN(C)S(=O)(=O)c1ccccc1[N+](=O)[O-] NRB00574 COc1cc(c(cc1SCC(=O)NNC(=S)Nc2cc(ccc2Cl)C(F)(F)F)OC)[N+](=O)[O-] BTB02334 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C/3\C(NN(C(=S)S3)C)c4ccccc4 MBE00211 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4cc(cc(c4)C(F)(F)F)C(F)(F)F NH00129 c1ccc(cc1)S(=O)Cc2ccccc2C(=O)O NRB00603 CCc1ccc(cc1)c2ccc(cc2)C(=O)NC(CC)(CC)C#C BTB05913 COc1cc(c(cc1SCc2nnc(o2)c3cccc(c3)[N+](=O)[O-])OC)[N+](=O)[O-] BTB02378 COc1cc(c(cc1SCC(=O)NNC(=S)Nc2ccc(c(c2)Cl)Cl)OC)[N+](=O)[O-] BTB02333 Cc1c(nn(n1)c2ccccc2)C(=O)NCC3CC3 BTB05875 c1cc(sc1)C(=O)NCC2CC2 BTB05876 c1cc(c(c(c1)Cl)C(=O)NC(=O)NCC2CC2)F BTB05879 c1cc(cc(c1)NS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F)C(F)(F)F MWP01137 c1cc(ccc1c2nc(on2)CCc3nnc(n3c4cc(cc(c4)C(F)(F)F)C(F)(F)F)S)Cl BTB02335 CN(C)c1ccc(cc1)/C=N/c2ccc(cc2)S(=O)(=O)N BTB00185 Cn1c(nc(n1)c2ccc(cc2)OC)O NH00121 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl BTB02326 COc1cc(c(cc1SCC(=O)NNC(=S)Nc2cccc(c2)Cl)OC)[N+](=O)[O-] BTB02330 c1cc(ccc1NC(=S)NNC(=O)C2(CN3CCC2CC3)O)Cl MWP01232 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NNc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB02344 COc1cc(c(cc1SCc2nnc(n2c3ccc(cc3)F)S)OC)[N+](=O)[O-] BTB02349 c1ccc2c(c1)c(nn(c2=O)CCO)c3cc(cc(c3)C(F)(F)F)C(F)(F)F NH00131 CCOC(=O)c1c(c(sc1Nc2ccccc2C(F)(F)F)C(=O)OCC)N MBE00251 c1cc(ccc1C(=O)O)NS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01138 CCNS(=O)(=O)c1ccccc1I NRB00628 Cc1cc2c3c(c1)c(c(c(=O)n3CCC2)c4ccccc4)OS(=O)(=O)c5ccc(cc5)C(C)C RH00710 CC(=O)NS(=O)(=O)c1ccc(cc1)/N=C/c2ccc3c(c2)OCO3 BTB00192 CC(=O)NS(=O)(=O)c1ccc(cc1)/N=C/c2cc(cc(c2O)Cl)Cl BTB00193 CCc1ccc(cc1)c2ccc(cc2)OC(=O)c3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05868 c1ccc(cc1)C(c2ccccc2)(c3nnc(n3c4ccc(cc4)F)S)O BTB02319 COc1ccc(cc1)S(=O)c2ccccc2C(=O)O NRB00593 C1CC1CN2CNC(=S)NC2 BTB05889 c1cc(c(cc1S(=O)(=O)NCC2CC2)Cl)F BTB05890 Cc1c(cccc1Cl)n2c(nnc2S)CCc3nc(no3)c4ccc(cc4)Cl BTB02339 Cc1ccccc1S(=O)c2ccccc2C(=O)O NRB00596 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)NCC2CC2 BTB05891 Cc1ccc(c(c1)C)n2c(nnc2S)CSc3cc(c(cc3OC)[N+](=O)[O-])OC BTB02351 CCCNS(=O)(=O)c1ccccc1I NRB00629 CN1CCC(=N1)c2ccc(s2)Cl MWP01192 c1ccc(c(c1)C(=O)NC(=O)NCC2CC2)F BTB05870 c1ccc(cc1)CN2CCC(=N2)c3cccs3 MWP01198 c1cc(c(c(c1)Cl)C(=O)NC(=O)NCC2CC2)Cl BTB05878 c1c(cc(cc1Cl)Cl)S(=O)(=O)NCC2CC2 BTB05881 CC(=O)C(=CNc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)C BTB02372 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)NC(=O)c3ccccc3F BTB05909 CN1CCC(=N1)c2cccs2.Cl.Cl MWP01199 CCc1ccc(cc1)c2ccc(cc2)C(=O)NC(C)(C)C#C BTB05912 c1cc2c(cc1Cl)c(c(s2)Br)/C=N/Nc3c(cc(cc3Cl)Cl)Cl MWP01146 CCc1ccc(cc1)c2ccc(cc2)C(=O)NC3(CCCCC3)C#C BTB05914 COc1ccc(c(c1C(=O)NCC2CC2)OC)[N+](=O)[O-] BTB05874 c1cc2cccc(c2c(c1)C(=O)O)S(=O)c3cccc4c3c(ccc4)C(=O)O NRB00607 COc1cc(c(cc1SCC(=O)NNC(=O)c2c(cccc2F)F)OC)[N+](=O)[O-] BTB02359 COc1cccc(c1C(=O)NNC(=O)CSc2cc(c(cc2OC)[N+](=O)[O-])OC)OC BTB02360 COc1cc(c(cc1SCC(=O)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)OC)[N+](=O)[O-] BTB02363 COc1cc(c(cc1SCC(=O)NNS(=O)(=O)c2ccc(cc2)Cl)OC)[N+](=O)[O-] BTB02364 c1cc(ccc1CCC(=O)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)O BTB02365 CC1CN(CC(O1)C)c2ccc(c(c2)O)[N+](=O)[O-] BTB05901 c1cc(oc1)C(=O)CCSc2ccc(cc2)C(F)(F)F MWP01152 CCOC(=O)/C(=C/NCC1CC1)/C#N BTB05894 Cc1cc(c(cc1Cl)C)S(=O)(=O)N BTB05895 c1cc(c(c(c1)Cl)SCCC(=O)c2ccco2)Cl MWP01153 c1cc2cccc3c2c(c1)C(=O)S3 NRB00573 CC(C)(C)c1nnc(s1)/N=C/N(C)C BTB05811 Cn1c(c(cn1)C#N)n2cccc2 BTB02308 c1ccn(c1)c2c(cnn2c3cccc(c3)Cl)C#N BTB02310 Cc1cccc(c1)C(=O)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl BTB02318 c1cc(ccc1Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])Cl NRB00613 c1ccc2cc(ccc2c1)Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] NRB00616 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3ccccc3C(=O)NCC4CC4 BTB05919 c1ccc(cc1)CN2CCC(=N2)c3ccc(s3)Cl MWP01194 c1ccc(cc1)CCn2c(nnc2S)CCc3ccc(cc3)O BTB02383 c1ccc(cc1)S(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3OCC(F)(F)F)C#N)OCC(F)(F)F MWP01140 c1ccc(cc1)C(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3OCC(F)(F)F)C#N)OCC(F)(F)F MWP01141 Cc1cc(c(cc1Cl)C)S(=O)(=O)NCC2CC2 BTB05882 c1cc(sc1)C(=O)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02374 c1ccc(cc1)C(c2ccccc2)(C(=O)NNC(=S)Nc3cc(ccc3Cl)Cl)O BTB02298 Cc1cc(ccc1NC(=S)NNC(=O)C(c2ccccc2)(c3ccccc3)O)Cl BTB02301 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)c3cccs3 BTB05920 Cc1cc(c(cc1Cl)C)S(=O)(=O)/N=C/N(C)C BTB05923 c1cc(c(c(c1OCC(F)(F)F)C#N)OCC(F)(F)F)Br MWP01165 COc1cc(c(cc1SCc2nnc(n2c3ccc(c(c3)Cl)Cl)S)OC)[N+](=O)[O-] BTB02353 c1ccc(c(c1)C(F)(F)F)N/N=C/c2c3cc(ccc3sc2Br)Cl MWP01145 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)CSc2cc(c(cc2OC)[N+](=O)[O-])OC BTB02361 CC(=O)Oc1ccc(c2c1[C@@H]3CC[C@H]2C=C3)OC(=O)C NRB00571 CC(=O)C(=CNc1ccccc1SCCC#N)C(=O)C BTB02371 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2ccccc2C(=O)NCC3CC3 BTB05911 c1ccc(c(c1)C(=O)NCC2CC2)NS(=O)(=O)c3ccc(cc3F)F BTB05915 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3ccccc3C(=O)NCC4CC4 BTB05917 CC1(CCC(N=C(N1)SCc2cccc(c2)C(F)(F)F)(C)C)C.Cl BTB02423 c1cc(ccc1C(F)(F)F)S(=O)(=O)NNC(=O)C2(CN3CCC2CC3)O.Cl MWP01235 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)c4ccccc4 BTB02312 Cc1cc(c2cc(ccc2n1)Br)C(=O)NN BTB00115 c1cc(ccc1Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])Br NRB00612 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])NC2CCCCC2 NRB00614 COc1cc(c(cc1SCC(=O)NNC(=O)c2c(cccc2Cl)Cl)OC)[N+](=O)[O-] BTB02358 COc1ccc(c(c1)C(=O)O)Sc2ccc(cc2C(=O)O)OC NRB00566 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)/N=C/c3cc(c(c(c3)OC)OC)OC)C BTB00187 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)N BTB05897 c1cc(c(cc1N2CCOCC2)O)[N+](=O)[O-] BTB05900 CC1CCN(CC1)c2ccc(c(c2)O)[N+](=O)[O-] BTB05905 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)NC(=O)c3c(cccc3Cl)F BTB05908 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Nc2ccccc2C(=O)NCC3CC3 BTB05910 c1ccc2c(c1)c(=O)n(c(n2)S)NC(=O)c3cccnc3 BTB02399 c1ccc(cc1)/C=N/c2ccc(cc2)S(=O)(=O)N BTB00181 CN(C)c1ccc(cc1)/C=C(\C#N)/c2c(c(n(n2)c3ccccc3)n4cccc4)C#N BTB02391 c1ccc(c(c1)C(=O)NNC(=O)c2ccccc2Cl)N BTB02393 c1cc(c(c(c1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OCC(F)(F)F)C#N)OCC(F)(F)F MWP01215 c1cc(ccc1c2cc(cs2)C(=O)N3CCCCC3)Cl MBE00086 COc1ccc(c(c1C(=O)Nc2ccccc2C(=O)NCC3CC3)OC)[N+](=O)[O-] BTB05918 CC(=O)NS(=O)(=O)c1ccc(cc1)/N=C/c2ccccc2O BTB00190 c1cc(ccc1c2ccc(s2)C(=O)Nc3ccc(cc3F)F)Cl MBE00087 CC(c1ccccc1)n2c(nnc2S)CCc3ccc(cc3)O BTB02385 COc1ccc(cc1OC)CC2c3cc(c(cc3CCN2C=C(C#N)C#N)OC)OC BTB02410 c1ccc(c(c1)C(=O)NNC=C(C#N)C#N)n2cccc2 BTB02388 CC1c2cc(c(cc2CCN1C=C(C#N)C#N)OC)OC BTB04342 CCOC(=O)c1cc(nc2c1cc(cc2)Br)C BTB00099 c1ccc(cc1)COC(=O)c2ccc(cc2)Sc3ccc(cc3)C(=O)OCc4ccccc4 NRB00606 COc1ccc(cc1)Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] NRB00610 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)/N=C/N(C)C BTB05922 CSc1cccc(c1)N/C(=N/S(=O)(=O)c2ccccc2)/SC NH00006 CC(=O)c1ccc(c(c1)CS/C(=N/S(=O)(=O)c2ccccc2)/Nc3cccc(c3)F)OC NH00045 c1cc(c(cc1CO)[N+](=O)[O-])N2CCOCC2.Cl BTB02380 CSc1cccc(c1)n2c(nnc2S)CCc3ccc(cc3)O BTB02382 Cc1cccc(n1)NC(=O)NC(=O)c2ccc(s2)C(C)(C)C MBE00195 CC(C)(C)c1ccc(s1)C(=O)NC(=O)Nc2cccnc2 MBE00196 c1ccc(cc1)S(=O)(=O)/N=C(\Nc2cccc(c2)C(F)(F)F)/SCC(=O)O NH00053 CSc1cccc(c1)N/C(=N\S(=O)(=O)c2ccccc2)/SCC(=O)O NH00057 CCOC(=O)c1cnc(nc1N)S BTB04316 CC1c2cc(c(cc2CCN1C(=O)Nc3cccc(c3)C(F)(F)F)OC)OC BTB04344 CC1c2cc(c(cc2CCN1S(=O)(=O)C)OC)OC BTB04345 Cc1ccc(cc1)/C(=N/N=C(/c2ccc(cc2)C)\C)/C BTB00221 c1ccc(c(c1)/C=N/c2ccc(cc2)S(=O)(=O)N)O BTB00183 CCOC(=O)NC(=S)c1ccc(cc1)OC NH00120 c1ccc(c(c1)C(=O)NNC(=O)CCc2ccc(cc2)O)N BTB02394 CN(C)c1ccc(c(c1)Cl)/C=C(\C#N)/c2c(c(n(n2)c3ccccc3)n4cccc4)C#N BTB02396 COc1ccc(cc1)c2[nH]c(=O)[nH]n2 NH00116 c1ccc(cc1)CN2CCC(=N2)/C=C/c3ccco3.Cl MWP01231 COc1ccc(cc1)NC(=S)NNC(=O)C2(CN3CCC2CC3)O MWP01233 COc1ccc(c(c1)C(=O)O)S(=O)c2ccccc2C(=O)O NRB00599 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3c(cccc3Cl)Cl)/C#N)C#N)n4cccc4 BTB02398 c1ccc(c(c1)C(=O)O)S(=O)c2cc(c(cc2C(=O)O)S(=O)c3ccccc3C(=O)O)C(=O)O NRB00601 c1ccc2cc(ccc2c1)S(=O)c3ccccc3C(=O)O NRB00602 c1ccc(cc1)S(=O)c2cccc3c2c(ccc3)C(=O)O NRB00604 c1ccc2c(c1)cccc2S(=O)c3cccc4c3c(ccc4)C(=O)O NRB00605 CC(C)(C)c1cc(c(c(c1)[N+](=O)[O-])OC(=O)c2cccc(c2)C(F)(F)F)C(C)(C)C BTB04320 c1ccc(cc1)CCN/C(=N/S(=O)(=O)c2ccccc2)/Nc3cccc(c3)Cl NH00009 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3c(cccc3Cl)F)/C#N)C#N)n4cccc4 BTB02397 c1ccc(c(c1)C(=O)NCCCn2ccnc2)NC(=O)Nc3c(cccc3Cl)Cl BTB04318 CCCCCCCCCCCC1N([C@@H](CS1)C(=O)O)C(=O)C RH00689 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3ccccn3)/C#N)C#N)n4cccc4 BTB02403 CCOC(=O)c1cnc(nc1N)SCC(=O)c2ccc(cc2)Br BTB04327 CCOC(=O)c1cnc(nc1N)SCC(=O)c2cccc(c2)[N+](=O)[O-] BTB04328 CC1(NN2C(=N1)C(=CN=C2SC)C#N)c3cc(cc(c3)Cl)Cl RH00697 CCOC(=O)c1cnc(nc1N)SCC(=O)c2ccc(cc2)c3ccccc3 BTB04330 CCOC(=O)c1cnc(nc1N)Sc2c(cccn2)[N+](=O)[O-] BTB04331 CCOC(=O)c1cnc(nc1N)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB04334 Cc1cc2c3c(c1)c(c(c(=O)n3CCC2)c4ccccc4)OS(=O)(=O)c5cccc(c5)C(F)(F)F RH00707 c1ccc(cc1)S(=O)(=O)c2ccccc2C(F)(F)F BTB02466 COc1ccccc1Oc2ccc(cc2NC(=O)c3cc4ccccc4oc3=O)C(F)(F)F BTB04409 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc(ccc3Oc4ccccc4OC)C(F)(F)F BTB04412 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CN3CCOCC3 RH00754 COc1ccccc1Oc2ccc(cc2NC(=O)NC(=O)c3ccccc3Cl)C(F)(F)F BTB04418 COc1ccccc1Oc2ccc(cc2NC(=O)NC(=O)c3c(cccc3Cl)Cl)C(F)(F)F BTB04420 c1cc(ccc1c2nc(on2)CCC(=O)Nc3ccc(cc3)C(F)(F)F)Cl BTB02445 COc1ccccc1Oc2ccc(cc2NC(=O)c3ccc(cc3Cl)Cl)C(F)(F)F BTB04410 CCCc1ccc(cc1)c2ccc(cc2)C(=O)N BTB05924 c1cc(c(cc1Br)I)S(=O)(=O)N NRB00662 COc1ccccc1Oc2ccc(cc2NC(=O)c3c(c4ccccc4s3)Cl)C(F)(F)F BTB04414 c1cc(c(c(c1)Cl)C(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl BTB05951 c1cc(cc2c1cc[nH]2)Br RH00739 Cc1cc(n(n1)c2ccccc2)OC(=O)c3c(onc3c4c(cccc4Cl)Cl)C RH00740 CCCc1ccc(cc1)c2ccc(cc2)C(=O)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05931 CN(c1ccccc1[N+](=O)[O-])NC(=O)NC(=O)c2ccc(c(c2)Cl)F BTB05933 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl BTB05958 COc1ccccc1Oc2ccc(cc2NC(=O)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F BTB04413 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(c3cc(ccc3[nH]2)[N+](=O)[O-])c4ccccc4 RH00759 c1cc2c(cc[nH]2)cc1Br RH00766 Cc1c(nn(n1)c2ccccc2)C(=O)NC(=O)N3CCCC3 BTB05936 COc1ccccc1Oc2ccc(cc2NC(=O)C(c3ccccc3)C4CCCC4)C(F)(F)F BTB04411 CCC(CC)(C#C)NC(=O)NC(=O)c1ccc(c(c1)Cl)F BTB05940 COc1ccc(c(c1)S(=O)(=O)Nc2cccc(c2)C#N)OC NH00231 COc1ccc(c(c1)S(=O)(=O)Nc2cccc(c2)[N+](=O)[O-])OC NH00233 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])F BTB05952 CC1CN(CC(O1)C)c2ccc(cc2N)C(=O)C BTB02449 Cc1ccc(cc1)S(=O)(=O)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl BTB02458 CC(=NNC(=O)c1cccnc1)C BTB00357 c1cc(cnc1)C(=O)N/N=C/c2cccs2 BTB00365 c1cc(sc1)c2nc3c(cc(cc3Br)Br)c(=O)o2 BTB02534 Cc1nc2c(cc(cc2Br)Br)c(=O)n1c3cccc(c3)C(F)(F)F BTB02536 c1cc(oc1)CNS(=O)(=O)c2ccc(c(c2)Cl)Cl NH00314 CNS(=O)(=O)c1cc(ccc1Cl)C(F)(F)F NRB00671 C/C(=N\N=C1NCCN1)/c2ccc(cc2)Br BTB02539 COc1ccccc1NC(=O)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02511 CNS(=O)(=O)c1ccc(cc1Br)[N+](=O)[O-] NRB00655 Cc1cc(c(cc1C)I)S(=O)(=O)NC NRB00657 Cc1ccc(c(c1)I)S(=O)(=O)N NRB00658 Cc1ccc(c(c1)I)S(=O)(=O)NC NRB00659 COc1ccc(c(c1)S(=O)(=O)Nc2cccc(c2)Cl)OC NH00227 CNS(=O)(=O)c1ccc(cc1I)Br NRB00663 CNS(=O)(=O)c1ccc(cc1I)Cl NRB00665 COc1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)Cl)OC NH00234 CCOC(=O)NC(=S)N1CCCC1 NH00192 COc1ccc(cc1OC)S(=O)(=O)Nc2ccccc2[N+](=O)[O-] NH00249 COc1ccc(c(c1)S(=O)(=O)N2CCOCC2)OC NH00210 COc1ccc(c(c1)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC NH00207 COc1ccc(c(c1)S(=O)(=O)N2CCCC2)OC NH00211 COc1ccc(c(c1)S(=O)(=O)NCc2ccco2)OC NH00214 CCOC(=O)/C(=C/N1CCN(CC1)c2ccc(cn2)[N+](=O)[O-])/C#N BTB05944 c1cc(ccc1c2nc(on2)CCC(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl BTB02460 c1cc(ccc1c2nc(on2)CCC(=O)NNS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)Cl BTB02461 c1ccc2c(c1)cccc2/C=N/NC(=O)c3cccnc3 BTB00373 CCCNS(=O)(=O)c1ccc(cc1I)Cl NRB00642 CC(C)NS(=O)(=O)c1ccc(cc1I)Cl NRB00643 COc1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)C#N)OC NH00252 Cc1c(nn(n1)c2ccccc2)C(=O)NC(=O)N3CCSCC3 BTB05927 CCCc1ccc(cc1)c2ccc(cc2)C(=O)Oc3c(cc(cc3Br)C(F)(F)F)[N+](=O)[O-] BTB05929 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC(=O)NC(=O)c2ccc(c(c2)Cl)F BTB05932 CN(c1ccc(cc1[N+](=O)[O-])C#N)NC(=O)NC(=O)c2ccc(c(c2)Cl)F BTB05934 c1ccc2c(c1)c(c[nH]2)C3=NCCO3 NH00204 CC(C)(C)CNC(=O)NC(=O)c1ccc(c(c1)Cl)F BTB05941 c1cc(c(c(c1)F)C(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])F BTB05943 c1cc(ccc1c2nc(on2)CCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl BTB02446 Cc1cc(c(cc1Cl)C)S(=O)(=O)n2cccc2 BTB05948 c1ccc(c(c1)C(=O)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl)n4cccc4 BTB02456 CN(C)c1ccc(cc1)C(=O)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl BTB02457 Cc1ccc(cc1)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02463 c1cc(c(cc1Cl)S(=O)(=O)N)I NRB00666 c1cc(c(cc1F)F)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] BTB05956 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] BTB05950 CC1(CCC(N=C(N1)SC)(C)C)C.I BTB02424 CC(C)CNC(=S)N1CCCC1 NH00219 COc1ccc(c(c1)S(=O)(=O)/N=C(\Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/SC)OC NH00221 C1CCN(CC1)C=C(C#N)C#N BTB02428 Cc1c(cnn1c2ccccc2)/C(=N/C(=O)NN)/C BTB02436 c1cc(c(c(c1)F)NC(=O)CCc2nc(no2)c3ccc(cc3)Cl)F BTB02443 CC(C)CN/C(=N/S(=O)(=O)c1cc(ccc1OC)OC)/SC NH00222 c1cc(c(cc1Cl)I)S(=O)(=O)NC2CCCCC2 NRB00647 Cc1ccc(cc1)NS(=O)(=O)c2ccc(cc2I)Cl NRB00650 Cc1cc(c(cc1C)I)S(=O)(=O)N NRB00656 c1cc(ccc1c2nc(on2)CCC(=O)Nc3ccc(cc3)F)Cl BTB02444 CC(C)(C)NS(=O)(=O)c1cc(ccc1OC)OC NH00212 c1ccc(cc1)S(=O)(=O)C/C(=N/O)/N BTB05990 CC(=O)c1ccc(c(c1)NC(=S)Nc2cc(ccc2Cl)Cl)N3CCCCC3 BTB02472 COc1ccc(cc1OC)S(=O)(=O)Nc2cccc(c2)[N+](=O)[O-] NH00241 COc1ccc(cc1OC)S(=O)(=O)Nc2ccc(cc2)[N+](=O)[O-] NH00242 CCOC(=O)NC(=S)NN(C)C NH00457 Cc1ccc(cc1S(=O)(=O)Oc2ccsc2C(=O)OC)[N+](=O)[O-] BTB06011 CC(C)CNC(=S)NCc1ccco1 NH00220 COc1ccc(c(c1)S(=O)(=O)Nc2ccccc2Cl)OC NH00226 CC(=O)C(=CNc1ccc(c(c1)Cl)Cl)C(=O)C BTB02485 c1cc(cc(c1)N2CCNC2=S)C(F)(F)F BTB02493 c1ccc2c(c1)c(=O)oc(n2)c3ccco3 BTB02494 Cc1ccc(cc1)S(=O)(=O)c2ccccc2C(F)(F)F BTB02464 c1cc(ccc1S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl BTB02467 c1cc(ncc1[N+](=O)[O-])N2CCN(CC2)C(=O)C(Cl)(Cl)Cl BTB05963 COC(=O)c1c(ccs1)OC(=O)c2cccnc2Oc3ccccc3 BTB05965 c1ccc(cc1)S(=O)(=O)/N=C(/Nc2cccc(c2)Cl)\NN NH00190 CSc1cccc(c1)N/C(=N\S(=O)(=O)c2ccccc2)/NN NH00176 COc1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)[N+](=O)[O-])OC NH00232 CC(C)(C)c1cc(c(cc1OC)C(C)(C)C)OC NRB00680 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3ccsc3C(=O)OC BTB05967 c1cc(ncc1[N+](=O)[O-])N2CCN(CC2)C(=O)C(Cl)Cl BTB05968 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])S(=O)(=O)NN BTB05973 COc1ccc(cc1OC)S(=O)(=O)Nc2ccc(cc2)C#N NH00250 CNS(=O)(=O)c1cc(ccc1I)Cl NRB00667 c1cc(c(cc1Br)S(=O)(=O)N)I NRB00668 CNS(=O)(=O)c1cc(ccc1I)Br NRB00669 COc1ccc(cc1OC)S(=O)(=O)Nc2cccc(c2)Br NH00251 c1cc(c(c(c1)Cl)C(=O)NC(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl BTB05953 COc1ccccc1Oc2ccc(cc2NC(=O)NC(=O)c3ccccc3F)C(F)(F)F BTB04417 COc1ccccc1Oc2ccc(cc2NC(=O)NC(=O)c3c(cccc3Cl)F)C(F)(F)F BTB04421 c1ccn2c(c1)cnc2Sc3c(cccn3)[N+](=O)[O-] BTB04422 c1cc(c(c(c1)F)C(=O)NCC(=O)O)F BTB02520 CCOC(=O)NC(=S)NCc1cccs1 NH00419 CNC(=O)c1ccccc1Sc2ccccc2C(=O)NC NRB00687 CNC(=O)c1ccccc1S(=O)c2ccccc2CO NRB00690 CC(=O)OCc1ccccc1S(=O)c2ccccc2C(=O)NC NRB00694 CNC(=S)N(C)NC(=S)Nc1ccc(c(c1)OC)OC NH00449 c1cc(c(c(c1)Cl)Cl)NC(=O)CCc2nc(no2)c3ccc(cc3)Cl BTB02447 COc1ccc(cc1)NS(=O)(=O)c2ccc(cc2I)Cl NRB00651 c1cc(ccc1NS(=O)(=O)c2ccc(cc2I)Cl)Cl NRB00652 CCOC(=O)NC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F NH00191 Cc1cc(n(n1)c2ccc(nn2)Sc3ccc(cc3)Cl)C BTB05992 CCc1cccc(c1NC(=O)C)CC NRB00682 c1ccc2c(c1)c3ccccc3[nH]c2=O NRB00684 c1ccc(c(c1)C(=O)O)S(=O)(=O)c2ccccc2C(=O)O NRB00686 COc1ccc(c(c1)S(=O)(=O)Nc2cccc(c2)Br)OC NH00253 c1cc(c(c(c1)F)NS(=O)(=O)c2ccc(c(c2)Cl)Cl)F NH00308 c1ccc(c(c1)C(=O)NC(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])F BTB05954 c1cc(c(cc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl)F BTB05957 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] BTB05959 c1ccc(c(c1)S(=O)(=O)NC2CCCCC2)I NRB00634 c1cc(c(cc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl)Cl BTB05960 c1cc(c(cc1S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl)Cl NH00309 CC(C)(C)NS(=O)(=O)c1ccc(c(c1)Cl)Cl NH00312 CNS(=O)(=O)c1c2ccccc2ccc1I NRB00673 COC(=O)c1c(ccs1)OC(=O)c2cc3ccccc3oc2=O BTB05964 c1cc2cccc(c2c(c1)C(=O)N)I NRB00698 CC(C)(C)C(=O)NC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl NH00472 Cc1cc(c(c(c1)Br)NC(=S)NNc2ccccc2)Br NH00578 CNC(=O)c1cccc2c1c(ccc2)Br NRB00700 COC(=O)c1c(ccs1)OC(=O)c2c(cccc2F)F BTB05966 Cc1cc(n(n1)c2ccc(nn2)N3CCOCC3)C BTB05982 COC(=O)c1c(ccs1)OS(=O)(=O)c2ccc(cc2)Cl BTB06012 c1ccc(c(c1)NC(=O)CS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)F BTB02515 c1ccc2c(c1)cc(c(=O)o2)C(=O)N3CCCCC3 BTB04386 CCc1ccc(cc1)c2ccc(cc2)C(=O)Nc3nnc(s3)C(C)(C)C BTB05985 CNC(=O)c1ccccc1Sc2ccccc2CO NRB00689 CNC(=O)c1ccccc1[S+]2c3ccccc3C(=O)N2C.[Cl-] NRB00691 Cc1cc(c(cc1Cl)C)S(=O)(=O)NN BTB05988 COC(=O)c1cc(ccc1n2cccc2)[N+](=O)[O-] BTB02475 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])N BTB05997 c1ccc(cc1)N(Cc2c(cccc2Cl)F)NC(=O)NC(=O)c3c(cccc3Cl)F BTB06000 CCOC(=O)C(=CNCCNc1ccc(cc1[N+](=O)[O-])C(F)(F)F)C(=O)OCC BTB02487 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCNC=C(C#N)C#N BTB02488 c1ccc(cc1)S(=O)(=O)C/C(=N/OS(=O)(=O)c2cc(cc(c2)Cl)Cl)/N BTB06005 c1ccc(cc1)S(=O)(=O)C/C(=N/OS(=O)(=O)c2ccc(cc2)Cl)/N BTB06010 Cc1cccnc1N2C(=O)C3C4CC(C3C2=O)C=C4 BTB02497 Cc1cccc(n1)N2C(=O)C3C4CC(C3C2=O)C=C4 BTB02498 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3ccc(c(c3)Cl)F BTB04380 C/C(=N\NC1=NCCCN1)/c2ccccc2 BTB02529 COC(=O)c1c(c2cccnc2s1)O RH00712 CC1CN(CC(O1)C)C2=NCCN2.Br BTB04351 COc1cc(c(c(c1O)Br)Br)C2Nc3cccc(c3C(=O)N2)F BTB04355 c1ccn(c1)c2cccc(c2)C#N BTB02480 c1ccc(cc1)N(Cc2c(cccc2Cl)F)NC(=O)C(Cl)(Cl)Cl BTB06019 c1ccc(cc1)N(Cc2c(cccc2Cl)F)NC(=O)CSC3=NCCCN3.Cl BTB06020 COc1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)Br)OC NH00229 c1ccc(cc1)CN2CCN=C2SCC(=O)NN(Cc3c(cccc3Cl)F)c4ccccc4.Cl BTB06022 c1c2c(cc(c1Cl)Cl)nc([nH]2)S BTB02521 COc1ccccc1CCC(=O)O BTB02522 COC(=O)c1c(c2ccccc2s1)Cl BTB00312 COc1cc(c(cc1SCc2nnc(n2c3cccc(c3)Cl)S)OC)[N+](=O)[O-] BTB02350 Cc1ccc(cc1)n2c(nnc2S)CSc3cc(c(cc3OC)[N+](=O)[O-])OC BTB02352 Cc1ccccc1c2nnc(o2)CSc3cc(c(cc3OC)[N+](=O)[O-])OC BTB02379 c1cc(c(cc1Cl)C(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])N BTB05996 COC(=O)c1c(ccs1)OS(=O)(=O)c2cc(cc(c2)Cl)Cl BTB06003 CCOC(=O)NC(=S)Nc1ccc(cc1)N2CC(OC(C2)C)C NH00585 c1cc2cccc(c2c(c1)C(=O)N)Br NRB00701 CCOC(=O)c1c(c(sc1Nc2ccccc2F)C(=O)c3ccc(cc3)Cl)N MBE00259 C/C(=N\N=C1NCCN1)/c2ccc(cc2)[N+](=O)[O-] BTB02541 C/C(=N\N=C1NCCN1)/c2ccc(cc2)F BTB02544 c1ccc(cc1)NC(=S)NCc2ccccn2 BTB04371 CC1CN(CC(O1)C)C2=NCCN2S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB04379 COc1ccc(cc1)NS(=O)(=O)c2ccccc2I NRB00638 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)/N=C/c3ccccc3O)C BTB00198 C/C(=N\N=C(\c1ccc(cc1)OC)/C)/c2ccc(cc2)OC BTB00226 CC1=N/C(=C\c2ccccc2)/C(=O)O1 RH00721 C/C(=N\N=C(\c1ccc(cc1)F)/C)/c2ccc(cc2)F BTB00237 COc1cc(cc(c1OC)OC)/C=N/N BTB00238 CCOc1ccc(cc1)/N=C/c2ccccc2O BTB00242 c1cc2c(cc[nH]2)cc1I RH00726 CCCCCOc1ccc(cc1)C(=O)NN RH00731 c1ccc-2c(c1)CCc3c2[nH]c4c3cccc4 RH00733 c1ccc2c(c1)c3c([nH]2)CCCCCC3 RH00736 Cc1ccc(cc1S(=O)(=O)Oc2c3cc(cc4c3n(c(=O)c2c5ccccc5)CCC4)C)[N+](=O)[O-] RH00711 CCCCn1c2ccccc2c(c(c1=O)C)C RH00713 c1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)Cl)I NRB00639 CC1c2cc(c(cc2CCN1C(=O)c3ccc(cc3Cl)Cl)OC)OC BTB04343 CC1c2cc(c(cc2CCN1S(=O)(=O)c3cc(ccc3OC)OC)OC)OC BTB04346 c1ccc(cc1)c2c3cc(ccc3[nH]c2C(=O)O)[N+](=O)[O-] RH00720 c1ccc(cc1)N2CCCC2=O RH00722 CCCCc1cc(c2c(c1)c(cc(=O)[nH]2)C)C RH00725 c1ccc2c(c1)cc(c(=O)o2)C(=O)NC3CC3 BTB04385 CC(C)(C)c1ccc(s1)C(=O)O/N=C(/c2ccc(cc2)Cl)\N MBE00168 Cc1ccccc1/C(=N/OC(=O)c2ccc(s2)C(C)(C)C)/N MBE00173 Cc1cc(no1)NC(=O)NC(=O)c2ccc(s2)C(C)(C)C MBE00198 c1cc(ccc1c2ccc(s2)C(=O)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl MBE00201 Cc1c(nn(n1)c2ccccc2)C(=O)NC(=O)N3CC(OC(C3)C)C BTB05928 COC(=O)c1c(c2cc(ccc2[nH]1)[N+](=O)[O-])c3ccccc3 RH00749 Cc1ccc(cc1Cl)/N=C/c2ccccc2O BTB00243 CC(=O)Nc1ccc(cc1C(=O)C(=O)Nc2ccc3c(c2)OCO3)Br BTB00246 c1ccc(cc1)C(=O)Oc2c(cc(cc2Cl)Cl)/C=N/c3cccc(c3)C(F)(F)F BTB00256 CC1c2cc(c(cc2CCN1C(=S)Nc3cc(ccc3Cl)Cl)OC)OC BTB04349 CC(=O)CC(=O)Nc1ccc(cc1F)F BTB04360 c1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)[N+](=O)[O-])I NRB00640 c1ccc(cc1)NC(=S)NNC(=O)c2cccnc2 BTB00335 Cc1ccc(cc1)/C=C/2\C(=O)OC(=N2)C RH00730 c1ccc2c(c1)c3c([nH]2)C(=O)CCC3 RH00732 CC1c2cc(c(cc2CCN1S(=O)(=O)c3ccc(cc3)Cl)OC)OC BTB04347 c1ccc(cc1)CNS(=O)(=O)c2ccc(cc2I)Cl NRB00648 c1ccc(cc1)NS(=O)(=O)c2ccc(cc2I)Cl NRB00649 c1cc(ccc1NS(=O)(=O)c2ccc(cc2I)Cl)[N+](=O)[O-] NRB00653 c1ccc(c(c1)C(=O)Nc2ccc3c(c2)OCCO3)NC(=O)c4ccco4 BTB02506 c1ccc(c(c1)NC(=O)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F BTB02510 c1cc2c(c(c1)F)c(=O)oc(n2)c3ccc(c(c3)Cl)F BTB04375 Cc1ccc(cc1Cl)/N=C/c2ccc(c(c2)OC)OC(=O)c3ccccc3 BTB00281 C/C(=N\N=C\c1cc(c(c(c1)OC)OC)OC)/c2ccc(cc2)OC BTB00285 c1cc(ccc1c2nnc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl MBE00286 COC(=O)CSc1c(cccn1)C(=O)OC RH00714 c1ccc2c(c1)C(=O)CCCCC(=O)N2 RH00729 c1ccc2c(c1)c(c(s2)C(=O)NN)Cl BTB00313 c1cc(c(cc1C(=O)NC(=O)NC2CC2)Cl)F BTB05938 C#CC1(CCCCC1)NC(=O)NC(=O)c2ccc(c(c2)Cl)F BTB05939 CC1CN(CC(O1)C)C2=NCCN2S(=O)(=O)c3ccc(cc3)Cl BTB04406 CCOC(=O)C1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(=O)C BTB02442 c1cc(ncc1[N+](=O)[O-])N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl BTB05945 CCOC(=O)C(C)c1c(=O)[nH]c2ccccc2n1 MGH00029 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3cc(cc(c3)Cl)Cl BTB04382 CC(C)(C)NC(=O)c1cc2ccccc2oc1=O BTB04384 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)COc3ccc4c(c3)OCO4 RH00746 CC(C)(C)c1ccc(cc1)c2nc3cccc(c3c(=O)o2)F BTB04388 CSC1=NCCN1CC(=O)c2ccc(cc2)Cl.Br BTB04401 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)c2ccc(cc2)Cl BTB02465 CN(c1ccc(cn1)[N+](=O)[O-])NC(=O)NC(=O)c2ccc(c(c2)Cl)F BTB05935 c1ccc2c(c1)c(nnc2O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F NH00130 Cn1c(=O)c2ccccc2c(n1)c3cc(cc(c3)C(F)(F)F)C(F)(F)F NH00132 c1ccc(c(c1)C(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)N3CCOCC3 NH00135 CCCCCCC(C)OC(=O)c1ccccc1C(=O)O NRB00621 CC(=O)NS(=O)(=O)c1ccc(cc1)/N=C/c2ccco2 BTB00196 Cc1ccc(c2c1nc(cc2Oc3c(cccn3)[N+](=O)[O-])C)Cl BTB04451 COc1cccc(c1)n2c(n[nH]c2=S)c3cccnc3 BTB00337 CCOC(=O)C1CCN(CC1)c2ccc(cc2N)C(=O)C BTB02448 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3nnc(s3)N RH00753 c1ccc2c(c1)c3c([nH]2)CCCCCCCCCC3 RH00737 c1ccc2c(c1)c(c(s2)C(=O)N/N=C/c3cccs3)Cl BTB00327 CC(=N)c1c(c2ccccc2n(c1=O)C)O RH00764 COc1cccc(c1)NC(=S)NNC(=O)c2cccnc2 BTB00332 c1cc(cc(c1)Cl)NC(=S)NNC(=O)c2cccnc2 BTB00333 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)/N=C/c3cc(cc(c3O)Cl)Cl)C BTB00197 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CN3CCCCC3 RH00752 COc1cc(ccc1OC(=O)c2ccccc2)/C=N/c3ccc(cc3)Cl BTB00280 Cc1ccc(cc1C)/N=C/c2cc(cc(c2OC(=O)c3ccccc3)Cl)Cl BTB00284 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)COc3cc(c(c(c3)C)Cl)C RH00755 c1ccc2c(c1)c(c(s2)C(=O)N(CCC#N)C3CCCCC3)Cl BTB00317 CCC(CC)(C#C)NC(=O)c1c(c2ccccc2s1)Cl BTB00320 COc1cccc(c1)NC(=S)NNC(=O)c2c(c3ccccc3s2)Cl BTB00328 c1ccc2c(c1)c3c([nH]2)CCC3 RH00738 CCNS(=O)(=O)c1ccc(cc1I)Cl NRB00641 CCCCNS(=O)(=O)c1ccc(cc1I)Cl NRB00644 c1ccc(cc1)NC(=S)NC(=O)/C=C/c2cccs2 MGH00166 c1cc(sc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2)Cl MGH00168 c1ccc(cc1)CNC(=S)NC(=O)/C=C/c2cccs2 MGH00169 c1cc(c(c(c1)Cl)CNC(=S)NC(=O)/C=C/c2cccs2)Cl MGH00170 CC(=O)NCc1ccccc1Br NRB00715 c1ccc(c(c1)C(=O)O)N/C=C/[N+](=O)[O-] RH00839 CSC1=NCCN1CC(=O)c2ccc(cc2)F.Br BTB04554 CC(=O)Nc1ccc(cc1NC(=O)c2ccc(cc2Cl)Cl)OC BTB00534 CC(=O)Nc1ccc(cc1NC(=O)c2c(c3ccccc3s2)Cl)OC BTB00535 CC(=O)N1C(OC(=N1)c2cccnc2)c3ccccc3Cl BTB00376 c1cc(cnc1)C(=N)NNC(=O)c2cccnc2 BTB00379 CC(=O)N1C(OC(=N1)c2cccnc2)(C)C BTB00356 c1ccc2c(c1)c(c(s2)c3nc4cc(ccc4c(=O)o3)Cl)Cl BTB00475 CCNc1c(cc(cc1[N+](=O)[O-])Cl)[N+](=O)[O-] MGH00105 Cc1ccc2c(c1)c(=O)oc(n2)c3c(c4ccccc4s3)Cl BTB00476 COC(=O)c1c(c(c([nH]1)C(=O)OC)O)O RH00825 CC1CN(CC(O1)C)c2ccc(cc2)NC(=S)NN NH00595 CC1CN(CC(O1)C)c2ccc(cc2)NC(=S)NNCCC#N NH00596 c1ccc(c(c1)C(=O)O)Sc2c(cc(cc2[N+](=O)[O-])[N+](=O)[O-])C(=O)O RH00860 CC(=O)Nc1ccc(c(c1)C(=O)O)Sc2ccccc2C(=O)O NRB00733 CSc1ccc(cc1)Br BTB04532 CC(=O)OCc1ccccc1Sc2ccccc2C(=O)NC NRB00735 c1ccc2c(c1)c(c(cn2)[N+](=O)[O-])O RH00840 COc1cc(cc(c1OC)OC)CCC(=O)NNC(=S)Nc2cc(ccc2Cl)Cl BTB02579 c1ccc(c(c1)C(=O)O)Sc2ccc(cc2C(=O)O)C(=O)O NRB00726 Cc1cc(n(n1)c2cccc(c2)Cl)Nc3ccccc3C(=O)O RH00841 Cc1cc(n(n1)c2c(cccc2Cl)Cl)Nc3ccccc3C(=O)O RH00842 Cc1cc(n(n1)c2ccc(cc2)[N+](=O)[O-])Nc3ccccc3C(=O)O RH00843 c1ccc(c(c1)C(=O)O)Sc2ccc(cc2C(=O)O)[N+](=O)[O-] NRB00730 c1cc(c(cc1N)C(=O)O)Sc2ccc(cc2C(=O)O)N NRB00732 CC1(c2c(c3ccccc3[nH]2)CC(N1)C(=O)O)C RH00846 CSc1[nH]c(=O)c(c(n1)c2ccccc2)C#N RH00853 Cc1cc(=O)oc2c1c(nn2C)C BTB06049 c1ccc(c(c1)/C=C/2\CS/C(=C/c3ccccc3Cl)/C2=O)Cl BTB06054 Cc1c2c(cc(=O)oc2n(n1)C)C(F)(F)F BTB06056 CC(C)(C)NC(=S)N(C)N NH00425 CCOC(=O)NC(=S)NCCc1ccccn1 NH00431 CNC(=S)N(C)NC(=S)Nc1cc(cc(c1)Cl)Cl NH00445 c1c(cc2c(c1)OCO2)/C=N/CC/N=C/c3cc4c(cc3)OCO4 BTB00398 COc1cc(cc(c1OC)OC)CCC(=O)NNC(=S)Nc2ccc(cc2)F BTB02580 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCC2CC2 BTB06031 CNC(=S)N(C)NC(=S)Nc1ccc(c(c1)Cl)F NH00446 Cc1nc2c(cc(cc2Br)Br)c(=O)n1c3ccc(c(c3)Cl)Cl BTB02537 CSc1nc(cnn1)c2ccc(cc2)Cl BTB06034 Cc1c(c(c2cc(cc(c2n1)F)F)O)I BTB06039 Cc1ccc(cc1)/C(=N/N=C2NCCN2)/C BTB02540 c1cc(c(nc1)N2CCSCC2)[N+](=O)[O-] BTB04481 C/C(=N\NC1=NCCN1Cc2ccccc2)/c3ccc(cc3)F BTB02545 Cc1cc(=O)oc2c1c(nn2c3ccccc3)C BTB06045 Cc1ccc(cc1)/C(=N/NC2=NCCN2Cc3ccccc3)/C BTB02548 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccccc3Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB04431 c1ccc(c(c1)CC(=O)O)I NRB00709 c1cc(c(cc1F)F)NC(=S)NCCCn2ccnc2 NH00523 c1cc(c(cc1Cl)[N+](=O)[O-])N2CCSCC2 BTB04484 Cc1cc2c(cc1C)CSC(SC2)(C)c3ccc(cc3)F BTB00441 Cc1cc2c(cc1C)CSC3(CCCCC3C)SC2 BTB00451 c1ccc(c(c1)C(=O)O)N2CCCCC2 BTB04438 c1cn(cn1)CCCN2CNC(=S)NC2 BTB04450 c1cc(cc(c1)Cl)n2c(n[nH]c2=S)c3cccnc3 BTB00339 c1cc(ncc1[N+](=O)[O-])N2CCSCC2 BTB04482 CCOC(=O)NC(=S)NCCCn1ccnc1 NH00526 Cc1cc(c(c(c1)Br)NC(=S)NN)Br NH00575 c1ccc2c(c1)c(c(c(=O)o2)[N+](=O)[O-])O MGH00113 Cc1cc(c2cc(ccc2n1)F)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB04490 Cc1ccc(cc1)/C(=C/c2cccs2)/C#N BTB02569 c1cc2cccc(c2c(c1)CO)Br NRB00702 COc1c2ccccc2oc(=O)c1[N+](=O)[O-] MGH00123 Cc1ccc(cc1)C(=O)CN2CCN=C2SC.Br BTB04553 CN(C)c1ccc(cc1)C2Nc3cccc4c3c(ccc4)N2 BTB00551 c1cc(c(c(c1)F)C(=O)Nc2ccc(c(c2)Cl)F)NC(=O)c3cccs3 BTB04558 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccc(cc2C)C BTB00561 Cc1ccc(cc1NC(=O)C)/N=C/c2cc(c(c(c2)OC)OC)OC BTB00564 CC1(C(=C)S/C(=N\c2ccc(cc2OC)OC)/N1)C BTB04568 Cc1ccc(cc1[N+](=O)[O-])NC(=O)C BTB00569 c1cc(sc1)/C=C/C(=O)NC(=S)N2CCOCC2 MGH00181 Cc1ccc(cc1)/C(=N/NC2=NCCCN2)/C BTB02528 Cc1cc(c2cccc(c2n1)Cl)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB04488 c1cc(cnc1)C(=O)N/N=C/c2ccc3c(c2)OCO3 BTB00362 c1cc(cnc1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl BTB00363 COc1cccc(c1OC)/C=N/NC(=O)c2ccncc2 BTB00388 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=O)CCc2cc(c(c(c2)OC)OC)OC BTB02592 c1ccc(c(c1)C(=O)N2CCSCC2)NC(=O)C(Cl)(Cl)Cl BTB04545 c1ccc(cc1)N(Cc2c(cccc2Cl)F)NC(=O)c3cccc(c3)C(F)(F)F BTB06016 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCCn2ccnc2 BTB06030 c1cc(c(cc1N)C(=O)O)Sc2ccc(cc2C(=O)O)N.Cl.Cl NRB00720 Cc1cc(cc(c1N2CCSCC2)[N+](=O)[O-])[N+](=O)[O-] BTB04483 Cc1cc(ccc1Cl)C(=O)CN2C(=O)c3ccccc3C2=O BTB04524 Cc1cc2c(cc1C)CSC(SC2)c3ccco3 BTB00421 Cc1cc2c(cc1C)CSC(SC2)(C)c3ccc(c(c3)OC)O BTB00442 c1cc(sc1)/C=C/C(=O)NC(=S)N2CCCCC2 MGH00182 c1cc2c(c(c1)Cl)c(=O)oc(n2)c3cccs3 BTB04573 c1cc(sc1)/C=C/C(=O)NC(=O)Nc2ccc(cc2)Cl MGH00187 c1ccc(cc1)S(=O)(=O)C/C(=N/OS(=O)(=O)c2ccc(cc2F)F)/N BTB06006 Cc1ccc(cc1S(=O)(=O)O/N=C(/CS(=O)(=O)c2ccccc2)\N)[N+](=O)[O-] BTB06009 c1ccc(cc1)N(Cc2c(cccc2Cl)F)NC(=O)NC(=O)c3ccc(c(c3)Cl)F BTB06014 CC(=O)Nc1ccccc1I NRB00707 Cc1cc2c(cc1C)CSC(SC2)c3cc(cc(c3O)Cl)Cl BTB00417 COc1cc(cc(c1O)/C=N/c2cccc(c2)C#C)Br BTB04462 C#Cc1cccc(c1)/N=C/c2cc(cc(c2O)Br)Cl BTB04463 C#Cc1cccc(c1)/N=C/c2cc(ccc2O)[N+](=O)[O-] BTB04464 C#Cc1cccc(c1)/N=C/c2cc(cc(c2O)Cl)Cl BTB04466 c1ccc(c(c1)/C=N/NC(=O)c2cccnc2)Cl BTB00374 COC(=O)CNCC(=O)OC.Cl RH00802 c1cc(c(c(c1)Cl)CCO)[N+](=O)[O-] RH00808 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccc(c2C(=O)Nc3ccc(c(c3)Cl)F)F BTB04564 CCOC(=O)c1c(c2cccnc2s1)N MGH00198 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3ccccc3N4CCOCC4 BTB04485 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3nnc(s3)NC(=O)C=C(C)C RH00799 Cc1cc(c2cc(ccc2n1)Cl)Oc3c(cccn3)[N+](=O)[O-] BTB04492 CCc1c(nc2ccccc2n1)N(C)/N=C/c3ccc(cc3Cl)Cl MGH00094 COc1ccc(c(c1)S(=O)(=O)N2CCC(CC2)CCCC3CCN(CC3)S(=O)(=O)c4cc(ccc4OC)OC)OC BTB04453 C#Cc1cccc(c1)NC(=O)NC(=O)c2c(cccc2Cl)Cl BTB04457 C#Cc1cccc(c1)NC(=O)NC(=O)c2c(cccc2F)F BTB04458 c1ccc(c(c1)C(=O)NC(=O)N2CCSCC2)Cl BTB04459 c1cc(c(c(c1)F)C#N)n2c(c(cn2)C#N)N BTB04517 c1cc2c(cc1Br)c3c([nH]2)CCC3 RH00801 Cc1cc2c(cc1C)CSC(SC2)c3cc(c(c(c3)OC)OC)OC BTB00418 Cc1cc2c(cc1C)CSC(SC2)c3ccc4c(c3)OCO4 BTB00419 Cc1cc2c(cc1C)CSC(SC2)c3cccs3 BTB00420 Cc1cc(c(c(c1)C)NC(=O)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C BTB02562 Cc1cc(c2cc(cc(c2n1)F)F)O BTB06033 C/C(=N\NC1=NCCCN1)/c2ccc(cc2)F BTB02530 Cc1cc(cc(c1O)/C=N/c2cccc(c2)C#C)Cl BTB04467 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3nnc(s3)NC(=O)c4ccc(cc4)C(C)(C)C RH00821 Cc1cc(c2ccccc2n1)Oc3c(cccn3)[N+](=O)[O-] BTB04494 Cc1cc(c(c(c1)C)/N=C\2/N(C3(CCCCC3)C(=C)S2)C(=O)c4c5ccccc5sc4Cl)C BTB00478 Cc1cccc(c1/N=C\2/N(C3(CCCCC3)C(=C)S2)C(=O)c4c(c5ccccc5s4)Cl)Cl BTB00480 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC(=O)NC(=O)c2c(cccc2Cl)Cl BTB04503 COc1c(c(cc(c1)/C=N/CC/N=C/c2cc(c(c(c2)OC)OC)OC)OC)OC BTB00397 Cc1cc2c(cc1C)CSC(SC2)c3ccc(c(c3)OC)O BTB00416 C/C(=N\NC1=NCCN1Cc2ccccc2)/c3ccccc3 BTB02549 Cc1cccc(c1/N=C/2\NC3(CCCCC3)C(=C)S2)C BTB00489 COc1cccc2c1oc(=N)c(c2)C#N BTB00493 c1cc(c(c(c1)Cl)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])F BTB02564 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3ccccc3C(=O)O BTB00384 Cc1cc2c(cc1C)CSC(SC2)(C)c3ccc(cc3)[N+](=O)[O-] BTB00440 Cc1ccc(cc1)/C(=C/c2c(cccc2Cl)F)/C#N BTB02567 COc1cc(cc(c1OC)OC)CCC(=O)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02578 CCSc1c(nc2ccccc2n1)SCC MGH00069 Cc1cc2c(cc1C)CSC3(CC(CC3C)(C)C)SC2 BTB00450 CC(=O)c1cc(c(cc1CC(=O)OC)OC)OC RH00822 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNC(=O)CCc3cc(c(c(c3)OC)OC)OC BTB02585 c1ccnc(c1)C(=N)NNC(=O)c2cccnc2 BTB00378 c1cc(cnc1)C(=O)NNC(=N)c2ccncc2 BTB00380 c1ccnc(c1)c2[nH]c(nn2)c3cccnc3 BTB00381 CC(C)c1ccc(cc1)/C=N/NC(=O)c2ccncc2 BTB00390 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3nnc(s3)NC(=O)c4ccc(c(c4)Cl)F RH00817 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)C(F)(F)F RH00781 Cc1cc(ccc1[N+](=O)[O-])C(=O)NNC(=O)C(F)(F)F RH00780 Cc1ccc(c2c1c3ccccc3n2C)C RH00793 C/C(=N\NC1=NCCCN1)/c2ccc(cc2)Br BTB02531 Cc1nc2c(cc(cc2Br)Br)c(=O)o1 BTB02532 COc1ccc(cc1OC)S(=O)(=O)Nc2ccccc2Cl NH00246 Cc1cccc(c1NC(=S)NNC(=O)c2cccnc2)C BTB00334 c1ccc(cc1)Sc2c(nc3ccccc3n2)Sc4ccccc4 MGH00071 c1ccc2c(c1)nc(c(n2)Sc3ccc(cc3)Cl)Sc4ccc(cc4)Cl MGH00072 Cc1cc(c[nH]c1=O)[N+](=O)[O-] RH00776 c1cc2c3c(ccc(c3c1)Br)CC2 RH00779 CS(=O)(=O)c1ccc(cc1)[N+](=O)[O-] RH00770 CCC1(C(=C)S/C(=N\c2ccc(cc2C)C)/N1)CC BTB04519 CC1CC(CN(C1)c2ccc(cc2[N+](=O)[O-])S(=O)(=O)N)C BTB04523 Cc1c2c(nn(c2oc(=O)c1Cl)c3ccccc3)C BTB06048 Cc1ccc2c(c1)c3c([nH]2)CCCC3 RH00819 Cc1cccc(c1/N=C/2\NC3(CCCCC3)C(=C)S2)Cl BTB00487 Cc1c2cc(c(cc2cc(n1)O)OC)OC RH00826 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NCC(=O)O BTB02581 CCOC(=O)/C(=C/NN(C)c1cccc(c1C#N)F)/C#N BTB04499 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCc4ccccc4C3 BTB00512 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)S(=O)(=O)Nc4ncccn4)Cl BTB00522 CCOC(=O)C1CCN(CC1)C(=S)Nc2c(cccc2C)C BTB00528 Cc1ccc2cc(ccc2n1)F BTB02593 CN(c1ccc(cc1[N+](=O)[O-])Cl)NC(=O)NC(=O)c2c(cccc2Cl)Cl BTB04506 COc1cc(cc(c1OC)OC)C(C#N)N(Cc2ccccc2)C(=O)c3c(c4ccccc4s3)Cl BTB00505 c1ccc(cc1)CN(C(C#N)c2ccc3c(c2)OCO3)C(=O)c4c(c5ccccc5s4)Cl BTB00506 c1cc(cc(c1)Cl)/C(=C/c2c(cccc2Cl)F)/C#N BTB02565 c1ccc(cc1)N(Cc2c(cccc2Cl)F)/N=C/c3cc(cs3)Br BTB06051 c1cc(sc1)/C=C/2\CS/C(=C/c3cccs3)/C2=O BTB06057 Cc1c(c(c2cc(ccc2n1)F)O)I BTB06058 c1ccc(c(c1)NC(=O)N/C=C/c2cccs2)Cl MGH00161 c1cc(sc1)/C=C/NC(=O)NCc2ccc(cc2)C(F)(F)F MGH00165 c1ccc(c(c1)NC(=S)NC(=O)/C=C/c2cccs2)Cl MGH00167 COc1cccc2c1nc(s2)NS(=O)(=O)CS(=O)(=O)Nc3nc4c(cccc4s3)OC BTB06060 c1cc(c(cc1N2CCCCC2)Oc3nc4c(s3)cc(cc4Cl)Cl)[N+](=O)[O-] BTB06063 C/C(=N\Nc1ccccc1)/c2cc3cc(ccc3oc2=O)Br RH00829 Cc1c2cc(c(cc2c(c(n1)O)[N+](=O)[O-])OC)OC RH00831 c1ccc(cc1)CSc2nc3c(c4cc(ccc4[nH]3)Br)nn2 BTB00500 C1CC2CCC1CN(C2)C(=S)NCCCN3CCOCC3 BTB02561 CC/C=N/Nc1ccc(cc1)[N+](=O)[O-] RH00837 c1ccc(c(c1)NCCC(=O)O)Cl RH00850 c1cc2c(cc(c(c2nc1)OC(=O)c3cccs3)Cl)Cl RH00852 c1cc(c(cc1[N+](=O)[O-])C(=O)O)Sc2ccc(cc2C(=O)O)[N+](=O)[O-] RH00854 CN(c1ccccc1[N+](=O)[O-])NC=C(C#N)C#N BTB04497 CCOC(=O)/C(=C/NN(C)c1ccccc1[N+](=O)[O-])/C#N BTB04498 c1c(cc(c(c1[N+](=O)[O-])N2CCCC2)[N+](=O)[O-])Cl MGH00106 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3c(c4ccccc4s3)Cl)C BTB00521 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)S(=O)(=O)Nc4nccs4)Cl BTB00523 COc1cc(cc(c1OC)OC)CCC(=O)NNC(=O)c2c(cccc2Cl)Cl BTB02584 COc1ccc2c(c1)CCCN2C(=O)NC(=O)c3c(cccc3Cl)F BTB04536 COc1ccccc1NC(=S)Nc2ccc(c(c2)OC)OC BTB00541 Cc1cccc(c1NC(=S)Nc2ccc(c(c2)OC)OC)C BTB00542 COc1ccc(cc1)/C=N/NC(=O)c2ccncc2 BTB00389 CC(C)(C)c1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S BTB04361 c1ccc(c(c1)C(=O)NCCCn2ccnc2)NC=C(C#N)C#N BTB04369 CN(c1cccc(c1C#N)Cl)NC(=O)NC(=O)c2c(cccc2Cl)Cl BTB04501 c1cc(ccc1C2CC(=O)NC(=O)C2)Cl RH00814 CC1(C(=C)S/C(=N\c2ccccc2Cl)/N1C(=O)c3c(c4ccccc4s3)Cl)C BTB00479 c1ccc2c(c1)c(c(c(=O)o2)[N+](=O)[O-])N MGH00120 CN(c1cccc(c1C#N)F)NC(=O)NC(=O)c2c(cccc2Cl)Cl BTB04502 CN(c1ccccc1[N+](=O)[O-])NC(=O)NC(=O)c2c(cccc2Cl)Cl BTB04505 CCOC(=O)/C(=C/NN(C)c1ccc(cc1[N+](=O)[O-])C(F)(F)F)/C#N BTB04509 c1cc(c(cc1Sc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N)Cl)Cl BTB04513 Cc1ccc(cc1)/N=C\2/NC(C(=C)S2)(C)C BTB04520 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3ccc(c(c3)Cl)Cl BTB04525 CC1CN(CC(O1)C)c2ccc(cc2[N+](=O)[O-])S(=O)(=O)N BTB04527 CCC1(C(=C)S/C(=N/c2ccccc2Cl)/N1)CC BTB00485 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N2CC3CCC(C2)CC3 BTB02573 Cc1cc(c(c(c1)Br)NC(=S)OC)Br NH00605 Cc1c(c(c2cc(ccc2n1)Cl)O)I BTB06059 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)NCC(=O)O BTB02588 c1cc(cc(c1)Oc2nc3cc(ccc3s2)Cl)N4CCOCC4 BTB06069 c1cc(ccc1c2nc3c(cc(cc3Br)Br)c(=O)o2)[N+](=O)[O-] BTB02533 CC1CN(CC(O1)C)c2ccc(cc2)NC(=S)Nc3ccc(cc3)N4CC(OC(C4)C)C NH00586 c1cc(ccc1C(=O)Nc2c(cc(cc2Br)Br)C(=O)Nc3ccc(cc3)F)[N+](=O)[O-] BTB02543 c1ccc(cc1)Nc2c(cc(cc2[N+](=O)[O-])Cl)[N+](=O)[O-] MGH00152 CC1CN(CC(O1)C)c2ccc(cc2)NC(=S)OC NH00597 CCOC(=O)NC(=S)N1C(CCCC1C)C NH00603 C/C(=C\C(=O)Nc1ccc(cc1)F)/Nc2ccc(cc2)F BTB06046 Cc1cc(no1)N2C(=O)C=CC2=O BTB06065 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2nnc(s2)N BTB06066 COC(=O)COc1c(cc(cc1Br)Br)C(=O)OC RH00856 c1cc(c(cc1S(=O)(=O)N)[N+](=O)[O-])N2CCOCC2 BTB04537 c1cc(ccc1C2=NNC(=O)CC2)Cl BTB04540 c1ccc(c(c1)NC(=O)c2cc(cc(c2NC(=O)c3cccs3)Br)Br)Cl BTB02551 c1ccc(cc1)C(=O)Nc2c(cc(cc2Br)Br)C(=O)Nc3ccc(cc3)F BTB02552 Cc1c2c(=O)c3ccccc3[nH]c2n(n1)c4ccccc4 RH00836 Cc1cc(c(c(c1)Br)NC(=S)NNCCC#N)Br NH00577 CN1CCCN(CC1)C(=S)NCCCN2CCOCC2 BTB02557 C1CCC(CC1)NC(=S)N2CC3CCC(C2)CC3 BTB02558 COc1ccc(cc1)/C(=C/c2cccs2)/C#N BTB02566 COc1ccc2c(c1)CCCN2C(=O)c3c(cccc3F)F BTB04535 CC(=O)Nc1ccccc1Br NRB00708 c1ccn2c(c1)cnc2Sc3ccc(cn3)[N+](=O)[O-] BTB04423 c1ccn2c(c1)cnc2Sc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB04424 CCOC(=O)/C(=C(/C)\Nc1ccc(cc1)F)/C2CC(=O)N(C2=O)c3cc(on3)C BTB06074 c1c(cc(c2c1sc(n2)Sc3nnc(s3)N)Cl)Cl BTB06075 c1cc(cc(c1)Oc2ccc(cn2)[N+](=O)[O-])N3CCN(CC3)c4cccc(c4)Oc5ccc(cn5)[N+](=O)[O-] BTB06117 CCC(c1ccccc1)N(C)C(=S)Nc2ccccc2 NRB00809 Cc1cc(c2c(c1)c(cc(n2)C)O)C BTB06136 Cc1ccc(cc1)S(=O)(=O)O/N=C(/CS(=O)(=O)c2ccccc2)\N BTB06137 Cc1cc(c2ccccc2n1)Sc3nnc(s3)N BTB06085 CN(C)/C=N/c1nnc(s1)Sc2nc3cc(ccc3s2)Cl BTB06083 c1cc(cc(c1)Oc2nc3c(s2)cc(cc3Cl)Cl)N4CCOCC4 BTB06078 CN(c1ccccc1C(=O)NC2CCCCC2)C(=O)CSc3ccc(cc3)Cl BTB02630 CCN(CC)C(=S)Oc1c(cc(cc1C)C)C BTB02626 CSc1ccccc1C(=O)N2CCSCC2 NH00822 CSc1ccccc1C(=O)c2ccccc2C(=O)O NH00855 CC1CCN(CC1)c2ccc(c(c2)Oc3nc4c(s3)cc(cc4Cl)Cl)[N+](=O)[O-] BTB06102 c1ccc2c(c1)c(=O)n3c4cc(ccc4sc3n2)Cl BTB06129 Cc1cc(ccc1Cl)OS(=O)(=O)c2cccc(c2)S(=O)(=O)Oc3ccc(c(c3)C)Cl BTB06132 CCO/C=C(\C#N)/C(=O)Nc1ccc(c(c1)Cl)F BTB06122 CCOC(=O)CNC(=O)c1c(cccc1OC)OC BTB02598 c1cc2c(cc1C(=O)NN)OCO2 BTB02600 c1c(c(cc(c1N2CCCCC2)Cl)[N+](=O)[O-])N3CCCCC3 BTB02640 Cc1cc(n(n1)c2ccc(nn2)SCC(=O)Nc3ccc(cc3)Cl)C BTB06112 c1cc(ccc1S(=O)(=O)C/C(=N/O)/N)Cl BTB06126 c1ccc(cc1)n2c(=O)ccc(=O)[nH]2 BTB02614 CCOC(=O)CNC(=O)CCc1cc(c(c(c1)OC)OC)OC BTB02602 COc1cc(cc(c1OC)OC)CCC(=O)NCC(=O)O BTB02605 c1cc(cnc1)C(=O)OCC#CCOC(=O)c2cccnc2 NRB00754 c1cc(cnc1)C(=O)OCC#CC#CCOC(=O)c2cccnc2 NRB00756 Cn1ccnc1SCC(=O)Nc2ccc(cc2)I NRB00039 CC1CN(CC(O1)C)c2ccc(c(c2)[N+](=O)[O-])Oc3nc4c(s3)cc(cc4Cl)Cl BTB06107 CCOC(=O)NC(=S)N1CCSCC1 NH00662 CCOC(=O)NC(=S)c1ccc[nH]1 NH00704 CCN1CCCC1CN2CNC(=S)NC2 BTB02634 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)C#N NRB00021 c1c(c(cc(c1N2CCOCC2)Cl)[N+](=O)[O-])N3CCOCC3 BTB02641 C1CCCC(CC1)NC(=S)NCCO NH00767 c1cc(ccc1C(=O)CSc2ccc(cc2)Cl)F NRB00005 Cc1ccc(cc1)SCC(=O)c2ccc(cc2)Br NRB00010 c1ccc(c(c1)C(=O)NCC(=O)NN)[N+](=O)[O-] BTB02609 CC(=O)Nc1ccc(cc1NC=C(C#N)C#N)F BTB02611 CCOC(=O)C(=CNNC(C)(C)C)C(=O)OCC BTB02668 c1cc(ccc1C(=O)CSc2ccc(cc2)Cl)Br NRB00012 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)O/N=C(/CS(=O)(=O)c2ccccc2)\N BTB06140 c1cc(ccc1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB04608 c1cc(ccc1C(=O)NC(=O)N2CCSCC2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB04610 CCC(C)(C#C)OC(=O)NC(=O)c1c(cccc1Cl)Cl BTB04615 CCC(C)(C#C)OC(=O)NC(=O)c1c(cccc1Cl)F BTB04619 COc1nc(nc(n1)OC)Nc2ccc(cc2)F BTB00588 Cc1ccc(cc1Cl)Nc2nc(nc(n2)OC)OC BTB00589 c1cc(ccc1NC(=O)CN2CCCC2)I NRB00029 c1ccc(cc1)CC2C(=O)N(C(=O)N2)c3ccccc3 NRB00811 CCC(C)(C#C)OCC(CS(=O)(=O)[O-])O.[Na+] NRB00796 Cc1cc(n(n1)c2nc3ccccc3s2)C NRB00802 c1ccc(cc1)C(=O)OCCCCOC(=O)c2ccccc2 NRB00807 CC(C)(C)c1ccc(cc1)NC(=O)CSCC(=O)NN NRB00013 c1cc(ccc1NC(=O)CN2CCCCC2)I NRB00033 C1CCC(CC1)NC(=S)C(=S)NC2CCCCC2 NRB00036 c1cc2c(c(c1)F)c(=O)n3c4cc(ccc4sc3n2)Cl BTB06139 CCCCCCN1C(=O)C(NC1=O)c2ccccc2 NRB00812 COc1cc2c(cc1OC)CN(CC2)C(=S)Nc3ccc(cc3)[N+](=O)[O-] BTB02653 CC(C)(C)NNC(=O)c1ccccc1N BTB02696 c1cc2cccnc2c(c1)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl BTB02678 c1cc(c(cc1Cl)NC(=S)Nn2cnnc2)Cl BTB02679 c1cc(cc(c1)Oc2nc3c(s2)cc(cc3Cl)Cl)N4CCN(CC4)c5cccc(c5)Oc6nc7c(s6)cc(cc7Cl)Cl BTB06116 Cc1cc(=O)oc2c1c(nn2c3ccc(cc3)[N+](=O)[O-])C BTB06104 c1cc(ccc1C(=O)Nc2ccc(cc2)Cl)Cl BTB06174 c1cc(c(cc1NC(=O)/C(=C/N2CCOCC2)/C#N)Cl)F BTB06124 Cc1cc(c2cc(ccc2n1)Cl)Oc3nc4c(s3)cc(cc4Cl)Cl BTB06108 CC\1=NN(C(=O)/C1=C/N(C)C)C BTB06158 COC(=O)/C=C\1/C(=O)Nc2ccccc2N1 BTB06159 CC1=NN(C(=O)CC1)c2cc(cc(c2)Cl)Cl BTB06160 c1cc(ccc1c2cn3c(n2)sc(n3)C(F)(F)F)[N+](=O)[O-].Br BTB02686 c1cc(c(cc1C(F)(F)F)C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl BTB02671 c1c(c(cc(c1Cl)N2CCOCC2)N3CCOCC3)N BTB02645 COc1cc2c(cc1OC)CN(CC2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB02654 CCOC(=O)C(=CNc1ccccc1[N+](=O)[O-])C(=O)OCC BTB02656 Cc1ccc2c(c1)c(nc(n2)NC(=O)C(C)(C)C)O BTB02658 CCOC(=O)c1c[nH]c2c(c1=O)cccc2[N+](=O)[O-] BTB02661 CN(CCC#N)c1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB02638 CCOC(=O)C(=CNc1ccc(cc1[N+](=O)[O-])OC)C(=O)OCC BTB02657 CCOC(=O)C(=CNc1ccccc1N2CCOCC2)C(=O)OCC BTB02660 c1ccc(cc1)c2csc(=N)n2c3cc(ccc3N4CCOCC4)C(F)(F)F.Cl BTB02681 c1ccc(cc1)C(C2CCCC2)C(=O)N BTB02684 COc1ccc(cc1OC)CCNC(=O)c2ccccc2 BTB02643 COC(=O)C1C2CC(C1C(=O)Nc3ccccc3)C=C2 NRB00037 c1cc2c(cc[nH]2)cc1NC(=S)NC3CC4CC3C=C4 RH00906 c1cc(oc1)CNC(=S)Nc2ccc3c(c2)cc[nH]3 RH00910 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2F)F NRB00056 COc1cc(cc(c1OC)OC)C(SCC(=O)O)SCC(=O)O BTB00637 C#CCOCCCS(=O)(=O)[O-].[Na+] NRB00792 CC1=NN(C(=O)CC1)c2ccccc2 BTB06145 c1ccc2c(c1)nc(o2)SCC(=O)Nc3ccc(cc3)F NRB00024 c1cc(ccc1NCC(=O)NN)F NRB00025 c1cc(ccc1NC(=O)CSc2ccc(cc2)Cl)F NRB00022 Cn1ccnc1SCC(=O)Nc2ccc(cc2)F NRB00023 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)I NRB00028 c1ccc(cc1)CNCC(=O)Nc2ccc(cc2)I NRB00031 Cc1c2ccccc2oc1c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F RH00896 Cn1cc(c(n1)N)C(=O)Nc2ccc(c(c2)Cl)F BTB06147 Cn1cnnc1SCC(=O)Nc2ccc(cc2F)F NRB00053 c1cc(cc(c1)S(=O)(=O)Oc2cc(cc(c2)Cl)Cl)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl BTB06131 c1cc(c(cc1I)Cl)Cl BTB06155 CC\1=NN(C(=O)/C1=C/N(C)C)c2ccccc2 BTB06156 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)Cl BTB06165 Cn1cnnc1SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F NRB00062 c1cc(c(cc1C(F)(F)F)NC(=O)CSc2nnc(s2)SCC(=O)Nc3cc(ccc3Cl)C(F)(F)F)Cl NRB00063 c1cc(ccc1C(=O)CSc2ccc(cc2)Cl)Cl NRB00006 c1ccnc(c1)SCC(=O)c2ccc(cc2)Cl NRB00007 Cc1c2ccccc2oc1c3nc(no3)c4ccc(cc4)OS(=O)(=O)N(C)C RH00897 CCC(CN(CC)/C=C(\C#N)/C(=O)OCC)O BTB04626 Cc1cc(ccc1Cl)C(=O)CC(c2c(cccc2Cl)F)Sc3ccccc3N BTB04642 c1ccc(c(c1)n2c(csc2=N)c3ccc(cc3)Cl)N4CCOCC4.Cl BTB02647 c1cc(cc(c1)[N+](=O)[O-])NCC(=O)NN NRB00015 c1ccc(c(c1)NC(=S)NC(=O)c2ccc(cc2F)F)Cl MGH00227 c1cc(ccc1NC(=S)NC(=O)c2ccc(cc2F)F)Cl MGH00228 c1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2F)F)\N MGH00232 CCCCc1ccc(c(c1)C)NC(=O)CC RH00867 Cc1c(c(n(n1)c2ccccc2)O)/C=C\3/C(=NN(C3=O)c4ccccc4)C BTB06157 CC\1=NN(C(=O)/C1=C/c2c(cccc2Cl)Cl)c3ccccc3 BTB06175 COc1cc2c(cc1OC)C(=NCC2)c3ccccc3 BTB02676 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(ccc3NC(=O)C)OC BTB00533 COc1cccc(c1)NC(=S)Nc2ccc(c(c2)OC)OC BTB00540 COc1cccc(c1)Nc2nc3ccccc3s2 BTB00596 Cc1ccc(cc1Cl)Nc2nc3ccccc3s2 BTB00598 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc4c3nccc4 BTB02677 CC(C)(C)NNC(=S)Nc1cc(ccc1Cl)Cl BTB02683 C/C=C(\C)/C(=O)Nc1nncs1 BTB02685 c1cc2c3c(c(ncn3)N4CCOCC4)sc2nc1 MGH00211 c1cc2c(cc1C(SCC(=O)O)SCC(=O)O)OCO2 BTB00639 c1cc(ccc1C(=O)CCSc2ccc(cc2)Br)Cl NRB00057 c1cc2c(cc1/N=C/c3cc(cc(c3O)Cl)Cl)nc[nH]2 BTB00625 COc1cc(cc(c1OC)OC)/C=N/c2ccc3c(c2)ccc(=O)o3 BTB00626 c1cc(ccc1C(=O)Nn2cnnc2)[N+](=O)[O-] BTB02692 c1cc(sc1)C(=O)Nn2cnnc2.Br BTB02693 c1cc(ccc1CCN2CCOCC2)[N+](=O)[O-].Cl BTB02694 c1ccc(c(c1)NC(=S)Nc2ccc3c(c2)cc[nH]3)N4CCOCC4 RH00908 c1ccc(cc1)COc2ccc(cc2)NC(=S)Nc3ccc4c(c3)cc[nH]4 RH00909 Cc1cc2c(c(c1)Br)nc(oc2=O)c3cccc(c3)C(F)(F)F BTB04580 CC(C)N(C(C)C)C(=O)NC(=O)c1ccc(cc1F)F MGH00235 Cc1ccc(cc1NC(=O)C)[N+](=O)[O-] BTB00550 COc1cc2c(cc1OC)C(NCC2)c3ccccc3 BTB02690 c1cc(c(cc1F)F)C(=O)NC(=S)N2CCOCC2 MGH00238 c1ccc(cc1)c2csc(n2)c3ccncc3.Br ML00033 Cc1c2ccccc2oc1c3nc(no3)c4ccc(cc4)OC(F)(F)F RH00895 CS/C(=C/C(=O)c1cccs1)/Nc2ccccc2Cl MGH00199 CS(=O)(=O)c1ncc(cn1)Cl RH00798 CS(=O)(=O)c1ncc(c(n1)C(=O)O)Cl RH00789 c1cc(c(c(c1)F)C(=O)NC(=O)N2CCSCC2)F BTB04461 c1cc2c(c(c1)F)C(=O)NC(N2)c3cc(ccc3O)[N+](=O)[O-] BTB04585 c1cc(ncc1[N+](=O)[O-])Sc2[nH]c(nn2)C(F)(F)F BTB04588 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2[nH]nc(n2)C(F)(F)F BTB04589 Cc1ccc(c(c1)/N=C/c2ccc3c(c2)OCO3)NC(=O)C BTB00591 c1cc(ccc1C(=O)CSc2ccc(cc2)Br)Cl NRB00002 CC(=O)OCCCCN1C(=O)c2ccccc2C1=O RH00923 COc1ccc(cc1)c2csc(n2)c3ccncc3.Br ML00032 CCOC(=O)Cc1ccccc1[N+](=O)[O-] RH00894 COc1c2c(c3cccnc3s2)ncn1 MGH00210 c1ccc(cc1)CC(=O)Nc2ccccc2NC(=O)Cc3ccccc3 RH00927 CC1=C(C(CC(=O)N1)c2ccc(cc2)OC)C(=O)OC RH00928 c1ccc(cc1)CN2C(=O)c3cccc4c3c(ccc4Cl)C2=O RH00900 Cc1ccc(c2c1nc(cc2Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)C)Cl BTB04452 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F RH00794 CCOC(=O)C1CCN(CC1)C(=S)Nc2cccc(c2)OC BTB00562 c1ccc(cc1)CNC(=S)C(=O)Nc2cc(ccc2Cl)C(F)(F)F NRB00064 c1cc(c(cc1Br)C(F)(F)F)NC(=O)C(F)(F)F BTB02702 CCC(C)(C#C)OC(=O)NC(=O)c1c(cccc1F)F BTB04621 CCC(C)(C#C)OC(=O)NC(=O)c1ccccc1Cl BTB04622 CCC(C)(C#C)OC(=O)NC(=O)c1ccccc1F BTB04623 c1ccnc(c1)SCCC(=O)c2ccc(cc2)Cl NRB00044 Cc1ccc(c(c1)/N=C/c2ccncc2)NC(=O)C BTB00592 c1ccc(cc1)N/N=C/C=C(\C#N)/c2c(c(n(n2)c3ccccc3)n4cccc4)C#N BTB04594 c1ccc2c(c1)c(c(s2)C(=O)N/N=C/c3c(cccc3Cl)Cl)Cl BTB04598 CCOC(=O)CNC(=O)c1c(cccc1F)F BTB04601 c1ccc(c(c1)NC(=O)NC(=O)c2ccc(cc2F)F)Cl MGH00224 Cc1cc(c2cc(ccc2n1)Cl)Oc3nc4cc(ccc4s3)Cl BTB06081 CN(C)/C=N/c1nnc(s1)Sc2nc3c(s2)cc(cc3Cl)Cl BTB06084 c1cc(ccc1NC(=O)NC(=O)c2ccc(cc2F)F)Cl MGH00225 CS/C(=C\C(=O)c1ccccc1)/Nc2ccccc2Cl MGH00174 COc1cc(c(cc1OC)Br)/C=C(\C#N)/C(=O)O RH00874 Cc1cc(c2ccccc2n1)Sc3nnc(s3)/N=C/N(C)C BTB06091 Cc1cc(=O)oc2c1c(n[nH]2)C BTB06100 COc1ccc(cc1OC)NC(=S)Nc2ccccc2Cl BTB00543 CS/C(=C/C(=O)c1ccco1)/Nc2ccccc2Cl MGH00200 c1cc2c3c(c(=O)[nH]cn3)sc2nc1 MGH00205 CC(=O)O/N=C(/c1ccc(cc1F)F)\N MGH00231 COc1cc(cc(c1OC)OC)C2Nc3cccc4c3c(ccc4)N2 BTB00554 c1cc2cccc3c2c(c1)NC(N3)c4ccc5c(c4)OCO5 BTB00555 CCc1cc2c(cc1C(=O)CSc3c(cccn3)C(=O)O)C(CCC2(C)C)(C)C RH00866 c1cc(cc(c1)C(F)(F)F)c2nc3c(cc(c(c3c(=O)o2)F)Br)Br BTB04578 Cc1ccc(cc1/N=C/c2ccc(c(c2)Cl)Cl)NC(=O)C BTB00579 CN(CC(=O)O)c1ccc(cc1C(=O)O)OC RH00871 Cc1ccccc1NC(=O)C(c2ccccc2)C(=O)Nc3ccccc3C RH00873 Cn1c(nnc1Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C(F)(F)F RH01402 c1ccc2c(c1)ccnc2NC(=O)c3cccs3 BTB02631 c1ccc(c(c1)NC(=O)c2cccs2)N3CCOCC3 BTB02633 Cc1c2ccccc2oc1C(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N RH00885 c1cc(c(cc1N2CCSCC2)Oc3nc4cc(ccc4s3)Cl)[N+](=O)[O-] BTB06092 Cc1cc(n(n1)c2ccc(nn2)N3CCC(CC3)C)C BTB06094 Cc1cc(n(n1)c2ccc(nn2)N3CC(OC(C3)C)C)C BTB06096 CCOC(=O)CNC(=O)c1ccc(cc1)[N+](=O)[O-] BTB02596 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)N3CCOCC3 BTB06071 c1cc2c(cc1Cl)nc(s2)Sc3nnc(s3)N BTB06076 c1ccc(cc1)Sc2c3c(c4cccnc4s3)ncn2 MGH00215 Cc1c2ccccc2oc1C(=O)O/N=C(/c3ccc(cc3)OS(=O)(=O)N(C)C)\N RH00886 Cc1c2ccccc2oc1C(=O)O/N=C(/c3ccc(cc3Cl)Cl)\N RH00887 c1cc(cc(c1)C(F)(F)F)c2nc3c(cc(c(c3c(=O)o2)Cl)Br)Br BTB04579 c1cc(cc(c1)C(F)(F)F)c2nc3cccc(c3c(=O)o2)Cl BTB04581 c1cc(c(cc1Br)Br)OCC(=O)NN NRB00014 C1CCC(C1)NC(=S)NCCO NH00764 c1ccc2c(c1)n3cnnc3s2 NRB00804 c1cc(ccc1C(=O)OCC#CCOC(=O)c2ccc(cc2)[N+](=O)[O-])[N+](=O)[O-] NRB00805 COC(=O)NC(=O)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB04611 c1cc(c(c(c1)F)C(=O)Nn2cnnc2)F BTB02691 Cc1c2ccccc2sc1C(=O)CSc3c(cccn3)C(=O)O RH00877 Cc1c2ccccc2oc1C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N RH00888 C1CCN(C1)CCN2CNC(=S)NC2 BTB02635 CCOC(=O)NC(=S)Nc1ccc(cc1F)F NH00664 C1CSCCN1c2[nH]c(=O)[nH]n2 NH00668 c1ccc(cc1)N/N=C/C=C2C(=O)NC(=O)NC2=O BTB04596 COC(=O)c1c2ccccc2[nH]c1C(=O)OC RH00889 c1cc(=O)oc2c1cc(cc2)/N=C/c3cc(cc(c3O)Cl)Cl BTB00628 Cc1ccc(c(c1)/N=C/c2cc(c(c(c2)OC)OC)OC)NC(=O)C BTB00590 Cc1cc(n(n1)c2ccc(nn2)SCc3ccc(cc3)Cl)C BTB06110 Cc1cc(c2cc(cc(c2n1)F)F)Oc3nc4c(s3)cc(cc4Cl)Cl BTB06087 Cc1cc(n(n1)c2ccc(nn2)Sc3ccccn3)C BTB06111 c1cc(cc(c1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)N3CCN(CC3)c4cccc(c4)Oc5ccc(cc5[N+](=O)[O-])C(F)(F)F BTB06115 CC(C)(C)NC(=S)N(C)NC(=O)c1c(cccc1Cl)Cl NH00607 c1cc(sc1)/C=C/NC(=O)Nc2ccc(cc2)Cl MGH00162 c1cc(c(c(c1)Cl)CNC(=O)N/C=C/c2cccs2)Cl MGH00164 c1ccc(cc1)C(=O)OCC#CCOC(=O)c2ccccc2 NRB00806 C/C(=N\Nc1ccccc1)/C=N/O BTB04603 Cc1cc(n(n1)c2ccc(nn2)N3CCSCC3)C BTB06093 c1cc(c(cc1N2CCSCC2)Oc3nc4c(s3)cc(cc4Cl)Cl)[N+](=O)[O-] BTB06099 Cc1ccc2c(c1)c(=O)n3c4cc(ccc4sc3n2)Cl BTB06128 c1cc(cc(c1)S(=O)(=O)Oc2ccc(cc2F)F)S(=O)(=O)Oc3ccc(cc3F)F BTB06133 CCN(CC)C(=S)Oc1c(cc(cc1Br)Br)Br BTB02625 c1ccc(cc1)N2C(=O)CCC(=O)N2 BTB02624 Cc1cc(c(cc1Cl)C)SCCNC(=O)C BTB06267 CCC(=O)N1CC(C(=O)N(c2c1cccc2)C(=O)CC)C NRB00836 CN(C)c1ccc(cc1N)c2c3ccccc3c(=O)[nH]n2 BTB02780 c1cc2cccc(c2c(c1)S(=O)(=O)O)Cl BTB06262 CCOc1ccc(cc1)/C=N/NC(=O)N/N=C/c2ccc(cc2)OCC ML00129 c1cc(ccc1NC(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl BTB06281 Cc1c2c(cc(=O)oc2n(n1)c3ccccc3)c4ccccc4 BTB06211 Cc1cccc(c1NC(=O)CSc2c(cccc2Cl)[N+](=O)[O-])C BTB02786 COc1c2c(c(c(c1Br)Br)Br)OCCO2 NRB00875 COc1c(cc(cc1)/C=N/NC(=O)N/N=C/c2cc(c(cc2)OC)OC)OC ML00130 COc1cc(cc2c1OCO2)[N+](=O)[O-] NRB00891 CC(=O)Oc1cccc2c1OCCO2 NRB00881 CCCCCCNC(=O)NC(CC(=O)O)c1ccccc1 NRB00827 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2ccc(cc2)C(C)(C)C RH00985 CC(C(=O)O)Sc1ccc(cc1[N+](=O)[O-])C(F)(F)F RH00992 Cc1cc(c(c2c1CCC2)OC)/C(=N/O)/N RH00993 c1ccc(cc1)C2C(=C(C(=O)O2)Cl)Cl RH00994 Cc1cccc(c1NC(=O)CSc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C BTB02785 c1ccc(cc1)Oc2c(cccc2Cl)[N+](=O)[O-] BTB02772 Cc1c2c(=O)c3ccccc3[nH]c2n(n1)c4ccc(cc4)[N+](=O)[O-] RH00975 C[C@H]1C(=O)Nc2cc(ccc2S1)C(F)(F)F RH00997 c1ccc(cc1)Oc2c(cccn2)C(=O)NNc3c(cc(cc3Cl)Cl)Cl BTB04684 COc1ccc(cc1OC)S(=O)(=O)NNc2c(cc(cc2Cl)Cl)Cl BTB04686 c1cc(c(c(c1)F)C(=O)NC(=O)NNc2c(cc(cc2Cl)Cl)Cl)F BTB04689 CSc1c(cccn1)C(=O)O BTB06287 CC(C)(C)SCCNc1nc(nc(n1)Sc2ccc(cc2)Cl)NCCSC(C)(C)C BTB06285 CC(C)(C)SCCNc1nc(nc(n1)Sc2ccc(cc2)Cl)N3CCSCC3 BTB06286 c1ccc(cc1)/C=N/NC(=O)c2ccccc2O RH00976 Cc1c2c(c3ccccc3nc2n(n1)c4ccccc4)N5CCOCC5 RH00981 c1c(cc(c2c1c3c([nH]2)CCCC3)Cl)Cl RH00977 Cc1cc(c(cc1Cl)C)S(=O)(=O)CC#N BTB06288 c1cc(ccc1/C(=N/OS(=O)(=O)c2ccc(cc2)Cl)/N)C(F)(F)F BTB06291 Cc1cc(c(cc1Cl)Cl)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB06238 Cc1cc(c(cc1Cl)Cl)Sc2ccc(cn2)[N+](=O)[O-] BTB06240 c1ccc(c(c1)Nc2nc(cs2)c3ccc(cc3)Br)Cl.Br ML00088 c1ccc(c(c1)Nc2nc(cs2)c3cccc(c3)[N+](=O)[O-])Cl.Br ML00090 CCc1cc2c(cc1c3csc(n3)Nc4ccccc4Cl)C(CCC2(C)C)(C)C.Br ML00093 CC(=O)Nc1ccc(cc1[N+](=O)[O-])OC RH00991 CCN(CC)S(=O)(=O)c1ccc(s1)c2csc(n2)C AW00029 COc1ccc(c(c1)/C=N/NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3)OC ML00100 c1cc(sc1)c2cc[nH]n2 AW00038 CC(=O)CC(=O)Nc1ccc(cc1)OC BTB04711 CCCN(C)S(=O)(=O)c1cccc2c1cccc2N NRB00868 c1cc(c(c(c1)Cl)C(=O)NC(=O)NNc2c(cc(cc2Cl)Cl)Cl)Cl BTB04691 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)C=C(C#N)C#N BTB04697 CSc1[nH]c2ccccc2n1 RH00984 Cn1cnnc1SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB00091 c1cc(cc(c1)NC(=O)C(Cl)Cl)C#N BTB02750 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB02747 c1cc(c(c(c1)Cl)C(=O)Nc2ccc(cc2)C#N)Cl BTB02753 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cccc(c3)C#N BTB02756 c1cc(ccc1N/C=C/C=C/C=N/c2ccc(cc2)F)F.Cl NRB00096 c1ccc(cc1)C(c2c3ccccc3ccc2O)N4CCCCC4 NRB00097 c1ccnc(c1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB00092 c1cc(ccc1C(=O)CCSc2ccc(cc2)Cl)Cl NRB00042 c1cc(cc(c1)Cl)C(=O)Nc2cccc(c2)F BTB06196 CCN(C1CCCCC1)S(=O)(=O)c2cccc3c2cccc3N NRB00869 CCCCN(C)S(=O)(=O)c1cccc2c1cccc2N NRB00870 COc1c(cc(c2c1OCCO2)Br)Br NRB00873 c1cc(c(cc1F)F)NC(=O)CN2CCCCC2 NRB00058 Cc1c2c(n[nH]c2oc(=O)c1Cl)C BTB06212 COc1cccc(c1OC)/C=N/NC(=S)NCCc2ccccc2 ML00114 COC(=O)c1ccccc1NC(=O)c2ccccc2 BTB00740 CCCCCCNC(=O)NCCCC(=O)O NRB00826 c1cc(ccc1NC(=O)C(=S)NC2CCCCC2)F NRB00089 c1ccc(cc1)CNC(=S)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB00090 c1cc(oc1)CNC(=S)C(=O)Nc2cc(ccc2Cl)C(F)(F)F NRB00065 CCOC(=O)C(Cc1ccccc1)NC(=O)Nc2ccccc2 NRB00829 c1ccc(cc1)C2=NN(C(=O)C2)c3ccccc3 BTB06198 CC(=O)N1CCC(=O)Nc2c1cccc2 NRB00838 CC\1=NN(C(=O)/C1=C\c2ccc(cc2)Cl)c3ccccc3 BTB06177 Cc1c2c(cc(=O)oc2n(n1)C)c3ccccc3 BTB06205 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)F NRB00078 c1ccc2c(c1)c(c(s2)C(=O)NCC3CCC(CC3)C#N)Cl BTB02714 CN(c1ccc(cc1[N+](=O)[O-])Cl)/N=C/C=N/Nc2ccccc2 BTB04613 CN(c1ccccc1[N+](=O)[O-])/N=C/C=N/Nc2ccccc2 BTB04614 c1cc(c(c(c1)Cl)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F BTB02708 c1cc(c(cc1S(=O)(=O)NNc2c(cc(cc2Cl)Cl)Cl)Cl)Cl BTB04685 COc1ccc(c(c1)OC)/C=N/N2CCC(=O)Nc3c2cccc3 NRB00831 CC(=O)N1CCC(=O)N(c2c1cccc2)Cc3ccccc3 NRB00832 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(cc2F)F NRB00070 Cc1c2c(nn(c2oc(=O)c1Cl)C)C BTB06220 c1cc(c(c(c1)F)NC(=O)c2c(cccc2Cl)F)F BTB02709 CC1CC(=O)Nc2ccccc2N1C(=O)NC NRB00833 c1cc(cc(c1)F)NC(=O)c2ccc(cc2)Cl BTB06195 COc1ccc(cc1NC(=O)C(=S)NCc2ccco2)Cl NRB00080 c1cc(c(c(c1)Cl)C(=O)Nc2cc(ccc2Cl)Cl)F BTB02710 c1ccc2c(c1)c(c(s2)C(=O)NCCSCCO)Cl BTB02715 c1cc2cccnc2c(c1)NC(=O)CN3CCOCC3 BTB02726 Cc1ccc(c(c1)C)n2c(nnn2)c3ccc(c(c3)Cl)Cl BTB06215 Cc1c2c(n[nH]c2oc(=O)c1[N+](=O)[O-])C BTB06217 c1cc(c(cc1Br)C(F)(F)F)NC(=O)C(Cl)(Cl)Cl BTB02704 c1ccc(c(c1)C#N)NC(=O)CSc2ccccn2 NRB00060 Cc1ccc(cc1)SCC(=O)Nc2ccccc2C#N NRB00061 c1ccc(cc1)NC(=O)NCCC(=O)O NRB00823 CCCCCCNC(=O)NCCC(=O)O NRB00824 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2ccc(cc2Cl)Cl BTB02737 c1cc(ccc1NC(=O)c2ccc(c(c2)Cl)Cl)Cl BTB06187 Cc1ccc(c(c1)C)NC(=O)c2ccc(c(c2)Cl)Cl BTB06188 c1ccc(cc1)NC(=O)c2ccc(c(c2)Cl)Cl BTB06189 Cc1ccc(c(c1)C(=O)Nc2ccc(cc2)F)NC(=O)c3c(cccc3Cl)F BTB02719 CCCc1ccc(cc1)NC(=O)C BTB04635 CC(=O)Nc1ccc(cc1)C2CCCCC2 BTB04636 c1cc(c(c(c1)Cl)C(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)F BTB02711 Cc1ccc2c(c1)c(=O)oc(n2)c3c(cccc3Cl)F BTB02712 c1cc2cccnc2c(c1)NC(=O)C(Cl)(Cl)Cl BTB02713 c1cc(c(cc1C(=O)Nc2ccc(c(c2)Cl)Cl)Cl)Cl BTB06190 COc1cccc(c1O)/C=N/c2ccccc2C(=O)Nc3ccc(cc3)F BTB00724 CS(=O)(=O)NNc1c(cc(cc1Cl)Cl)Cl BTB04683 Cc1ccc(cc1)SCC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB04706 c1cc(ccc1SCC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl BTB04707 c1cc(c(cc1Br)C(F)(F)F)NC(=O)C(Cl)Cl BTB02729 CC1CC(=O)Nc2ccccc2N1C(=O)c3c(c4ccccc4s3)Cl BTB00662 c1cc(c(cc1F)F)NC(=O)C(=S)NC2CCCCC2 NRB00046 c1ccc(cc1)C\2=NOC(=O)/C2=C\c3ccc(cc3)C#N BTB06179 c1cc(c(cc1C(F)(F)F)NC(=O)C(=S)N2CCOCC2)Cl NRB00084 c1cc(ccc1Oc2ccc(c(c2)C(F)(F)F)[N+](=O)[O-])Cl BTB02720 Cc1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)NC(=O)c3c(cccc3Cl)F BTB02724 Cc1cc2c(cc1C)NC(=O)CC(N2)C BTB00743 COc1ccc(cc1OC)S(=O)(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB04693 COc1cc(cc(c1OC)OC)/C=N/NC(=S)NCCc2ccccc2 ML00118 COc1ccc(cc1)/C=N/NC(=O)N/N=C/c2ccc(cc2)OC ML00127 CCOc1c(cccc1)/C=N/NC(=O)N/N=C/c2c(cccc2)OCC ML00128 COc1cc(c(cc1)OC)/C=N/NC(=O)N/N=C/c2c(ccc(c2)OC)OC ML00131 c1cc(c(cc1C(F)(F)F)NC(=O)C(=S)NC2CCCCC2)Cl NRB00066 CC(=O)Nc1ccc(cc1NCc2cc(c(c(c2)OC)OC)OC)OC BTB00656 Cc1ccc(cc1)SCCC(=O)c2ccc(cc2)Cl NRB00050 CCCCCCNC(=O)NC(Cc1ccccc1)C(=O)O NRB00816 c1ccc(cc1)c2ccc(cc2)c3csc(n3)c4cccnc4.Br ML00058 COc1ccc(cc1NC(=O)CSCc2ccc(cc2)Cl)Cl NRB00079 c1ccc(c(c1)C(=O)NC(=O)NNc2c(cc(cc2Cl)Cl)Cl)Cl BTB04687 c1ccc(c(c1)C(=O)NC(=O)NNc2c(cc(cc2Cl)Cl)Cl)F BTB04688 c1cc(c(c(c1)Cl)C(=O)NC(=O)NNc2c(cc(cc2Cl)Cl)Cl)F BTB04690 CC(=O)Nc1ccc(cc1[N+](=O)[O-])C(F)(F)F BTB00736 c1cc(ccc1N2C(=O)C=CC2=O)F BTB00665 c1cc(ccc1C2=CN(C(=CO2)O)c3ccc(cc3)Cl)[N+](=O)[O-] NRB00059 COC(=O)c1ccccc1NC(=O)c2ccc(cc2Cl)Cl BTB00764 c1ccc(cc1)CNC(=S)C(=O)Nc2cc(cc(c2)Cl)Cl NRB00072 c1cc(ccc1c2csc(n2)c3ccncc3)[N+](=O)[O-].Br.Br ML00038 CN1CCN(CC1)CC(=O)Nc2ccc(cc2F)F NRB00068 c1cc(oc1)CNC(=S)C(=O)Nc2ccc(cc2F)F NRB00071 CC1CN(c2ccccc2N(C1=O)C)C.Cl NRB00841 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(cc2)F NRB00082 COc1cc(cc(c1OC)OC)C2=NCCc3c2cc(c(c3)OC)OC RH00960 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2ccc(cc2F)F BTB06225 CC(C)CNS(=O)(=O)c1cccc2c1cccc2N NRB00853 COc1ccc(cc1NC(=O)C(=S)NC2CCCCC2)Cl NRB00086 c1cc(c(c(c1)F)C(=O)NNc2c(cc(cc2Cl)Cl)Cl)F BTB04680 CCOC(=O)Cc1csc(n1)NC(=O)C(Cl)(Cl)Cl BTB06245 Cc1ccc(c(c1)C)c2csc(n2)c3cccnc3.Br ML00080 CSc1cccc(c1)NC(=O)C(=S)NCc2ccccc2 NRB00074 Cc1ccc(cc1)SCC(=O)Nc2cccc(c2)SC NRB00077 COc1ccc(cc1)Oc2ccc(cc2N)C(F)(F)F RH00953 CC(C)(C)NS(=O)(=O)c1cccc2c1cccc2N NRB00854 CCCCCNS(=O)(=O)c1cccc2c1cccc2N NRB00855 c1cc(oc1)CNC(=S)C(=O)Nc2ccc(cc2)F NRB00083 Cc1ccccc1C2CC(=O)NC(=C2C(=O)OC)C RH00958 c1cc2c(cccc2S(=O)(=O)N3CCCCC3)c(c1)N NRB00865 CCCCNS(=O)(=O)c1cccc2c1cccc2N NRB00852 c1cc2c(cccc2S(=O)(=O)NC3CCCCC3)c(c1)N NRB00860 CN(C)S(=O)(=O)c1cccc2c1cccc2N NRB00861 CCCN(CCC)S(=O)(=O)c1cccc2c1cccc2N NRB00862 CCOC(=O)Cc1csc(n1)N/C=N/O BTB06230 Cc1ccc2cc(ccc2n1)[N+](=O)[O-] BTB06234 CC1CC(=O)Nc2ccccc2N1C(=O)c3ccc(cc3Cl)Cl BTB00663 c1ccc(cc1)Nc2c3c(c4cccnc4s3)ncn2 MGH00214 c1cc(c(cc1F)F)/C(=N/O)/N MGH00219 c1ccc(cc1)NC(=O)NC(=O)c2ccc(cc2F)F MGH00223 CCOC(=O)C1CCN(CC1)C(=S)Nc2cccc(c2)C BTB00560 CC(=O)NNc1c2c(c3cccnc3s2)ncn1 MGH00245 CCN1c2ccccc2N(CCC1=O)C.Cl NRB00843 c1ccc(cc1)CNS(=O)(=O)c2cccc3c2cccc3N NRB00858 CN1c2ccccc2NC(CC1=O)c3ccccc3.Cl NRB00844 CCNS(=O)(=O)c1cccc2c1cccc2N NRB00849 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])CO BTB02725 CC(=O)Nc1ccc(cc1/N=C/c2cc(c(c(c2)OC)OC)OC)OC BTB00655 COc1cc(cc(c1OC)OC)/N=C/c2cc(cc(c2O)Cl)Cl BTB00658 c1cc(ccc1c2nnnn2c3ccc(cc3)Cl)Cl BTB06246 Cc1cc(c(cc1Cl)Cl)SCc2c(cccc2Cl)Cl BTB06250 CCc1cc2c(cc1c3csc(n3)c4cccnc4)C(CCC2(C)C)(C)C.Br ML00060 c1cc2c(cc[nH]2)cc1NC(=S)NC3CCCCC3 RH00905 c1cc(ccc1C(=O)CCC(=O)O)Br RH00893 c1cc(oc1)C(=O)NCC(=O)NN BTB04605 c1cc(c(c(c1)F)C(=O)NCC(=O)NN)F BTB04606 CC(C)(C)NC(=O)NC(=O)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB04607 Cc1cc(c(cc1Cl)Cl)Sc2c(cccn2)[N+](=O)[O-] BTB06236 Cc1cc(c(cc1Cl)Cl)SCc2cccc(c2)F BTB06258 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Cc2c(cccc2Cl)F BTB06259 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Cc2cccc(c2)F BTB06261 c1cc(ccc1CC#N)/N=C/c2cc(ccc2O)Br BTB00681 Cc1cc(ccc1Cl)C(=O)CC(c2c(cccc2Cl)Cl)Sc3ccccc3N BTB04643 CCOC(=O)C1CCN(CC1)CC(=O)Nc2cccc3c2nccc3 BTB02727 CCc1cc2c(cc1c3csc(n3)c4ccncc4)C(CCC2(C)C)(C)C.Br ML00042 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)c3ccncc3.Br ML00037 c1cc(ccc1c2csc(n2)c3ccncc3)F.Br ML00040 CCOC(=O)c1ccc(cc1)NC(=S)NN ML00050 COc1ccccc1Nc2nnns2 ML00056 COc1ccc(cc1)c2csc(n2)c3cccnc3.Br ML00059 Cc1ccc(cc1)SCC(=O)Nc2cccc(c2)C#N BTB02777 Cc1cc(ccc1Cl)C2=Nc3ccccc3SC(C2)c4c(cccc4Cl)Cl BTB04645 c1ccc(cc1)c2c3cc(ccc3n4c2c(=O)[nH]nc4)[N+](=O)[O-] RH00916 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2cccnc2)Cl BTB04604 CC1=C(C(CC(=O)N1)c2ccccc2)C(=O)OC RH00946 CC1=C(C(CC(=O)N1)c2ccccc2[N+](=O)[O-])C(=O)OC RH00947 c1ccn(c1)c2c(cc(cc2Cl)Br)Cl BTB04649 CCOC(=O)c1ccc(cc1)N2C(=O)CC(C2=O)SCC(=O)Nc3ccc(cc3)F BTB00686 Cc1ccc(cc1)c2csc(n2)c3ccncc3.Br ML00035 c1cc(ccc1CC#N)/N=C/c2cc(cc(c2O)Cl)Cl BTB00680 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)Cl)C#N BTB02757 c1ccn(c1)c2c(cc(cc2Br)F)Br BTB04656 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)Br BTB04654 c1ccc(cc1)c2ccc(cc2)c3cnc(s3)c4ccncc4.Br ML00039 Cc1ccc(c(c1)C)Nc2nnns2 ML00052 CN(C)c1ccc(cc1[N+](=O)[O-])c2c3ccccc3c(=O)[nH]n2 BTB02768 c1ccnc(c1)C(=N)NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl BTB04667 c1ccnc(c1)C(=N)NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3)[N+](=O)[O-])Cl BTB04673 CC(=N)NS(=O)(=O)c1cc(c(c(c1)Cl)Oc2ccc(cc2)[N+](=O)[O-])Cl BTB04674 c1cc(ccc1C(=N)NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3)[N+](=O)[O-])Cl)Cl BTB04675 c1ccc(c(c1)c2nnnn2c3cccc(c3)F)Cl BTB06269 Cc1ccc(cc1)c2csc(n2)Nc3ccccc3Cl.Br ML00084 Cc1cc(c(c(c1Cl)Br)n2cccc2)Br BTB04650 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)Br BTB04651 c1cc(ccc1NC(=O)CSc2ccc(cc2)Cl)Br BTB04652 c1cnc(nc1)SCC(=O)Nc2ccc(cc2)Br BTB04655 CC(=O)Nc1cc(ccc1C(=O)O)Cl BTB00691 c1ccn(c1)c2c(cc(c(c2Br)Cl)F)Br BTB04657 c1cc(cnc1)C(=N)NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl BTB04665 COc1ccc(cc1OC)CCNC(=O)c2cc(c(c(c2)OC)OC)OC RH00955 CN(C)CCC(=O)c1ccc2c(c1)OCCO2.Cl NRB00886 Cc1ccc(cc1Cl)n2c(nc3cc(ccc3c2=O)Cl)C BTB00698 CCCc1cc(c(c(c1)Br)n2cccc2)Br BTB04647 c1cc(ccc1[N+](=O)[O-])Oc2c(cc(cc2Cl)S(=O)(=O)NC(=N)c3ccncc3)Cl BTB04672 CC(=O)Nc1ccc2c(c1)OCCO2 NRB00893 Cc1cccc(c1NC(=S)N(Cc2ccccc2)Cc3ccc(c(c3)OC)OC)C BTB00727 c1ccc(cc1)c2csc(n2)Nc3ccccc3Cl.Br ML00091 COc1cc(ccc1O)/C=N/Cc2ccccc2 BTB00697 Cc1nc2cc(ccc2c(=O)n1c3ccc(cc3)Cl)Cl BTB00701 Cc1ccc(cc1)SCC(=O)c2ccc(cc2)F BTB00718 CCOc1ccc(cc1)/C=N/NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 ML00098 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Cc2c(cccc2Cl)Cl BTB06260 c1cc(ccc1C(=N)NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl)Cl BTB04664 Cc1cc(c(cc1Cl)C)SCC#N BTB06283 CCOC(=O)c1ccc(cc1)NC(=S)N/N=C/c2ccccc2Cl ML00101 CCOC(=O)c1ccc(cc1)NC(=S)N/N=C/c2cc(ccc2OC)OC ML00103 CCOc1ccc(cc1)/C=N/NC(=S)N ML00109 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2c(cc(cc2Cl)S(=O)(=O)NC(=N)c3ccncc3)Cl BTB04669 Cc1ccc(cc1)S(=O)(=O)NNc2c(cc(cc2Cl)Cl)Cl BTB04681 Cc1cccc(c1NC(=S)N(Cc2ccccc2)Cc3ccc4c(c3)OCO4)C BTB00713 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccc(cc3)C(C)(C)C RH00988 COc1ccc(c(c1)N/C(=C/C(=O)OC)/C(=O)OC)OC RH00989 COc1cc(c(cc1Cl)OC)/N=C/c2ccc3c(c2)OCO3 BTB00730 c1ccc(cc1)C/N=C/c2ccc3c(c2)OCO3 BTB00692 c1ccc(cc1)C/N=C/c2cc(cc(c2O)Cl)Cl BTB00693 COc1ccc(cc1OC)/C=N/Cc2ccccc2 BTB00696 Cc1ccc(c(c1)C)Nc2nc3ccccc3s2 BTB00595 c1c(cc(c(c1[N+](=O)[O-])Sc2[nH]nc(n2)C(F)(F)F)[N+](=O)[O-])C(F)(F)F BTB04590 COCCCNC(=S)Nc1cccc(c1)C#N BTB02760 CCOC(=O)C(=CNc1cccc(c1)C#N)C(=O)OCC BTB02761 c1cc(cc(c1)NC(=O)C(Cl)(Cl)Cl)C#N BTB02749 c1cc(cc(c1)NC(=O)CN2CCCCC2)C#N BTB02774 C/C(=C\c1ccccc1)/[N+](=O)[O-] S06879 Cc1ccc(cc1)SCC(=O)c2cccc(c2)[N+](=O)[O-] BTB00726 c1ccc(c(c1)/C=N/c2ccccc2C(=O)Nc3ccc(cc3)F)O BTB00720 c1cc(cc(c1)NC(=O)c2c(cccc2F)F)C#N BTB02754 COc1ccc(cc1)c2csc(n2)Nc3ccccc3Cl.Br ML00083 CCCNC(=O)NNC(=O)c1cccs1 RH00990 c1cc(ccc1C(=O)NC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB04702 c1ccc(c(c1)C(=O)NC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl BTB04703 CS(=O)(=O)N(c1cccc(c1)C#N)S(=O)(=O)C BTB02758 c1ccc(cc1)N/N=C/C=C2C(=O)NC(=S)NC2=O BTB04595 c1ccc(cc1)N/N=C/C=N/NC(=O)c2c(c3ccccc3s2)Cl BTB04597 c1ccc(cc1)c2ccc(cc2)c3csc(n3)Nc4ccccc4Cl.Br ML00087 c1ccn(c1)c2cccc(c2)/C(=N/O)/N BTB02771 c1cc(cc(c1)[N+](=O)[O-])/C(=N/O)/N BTB02770 c1cc(cc(c1)NC(=O)CN2CCOCC2)C#N BTB02775 Cc1ccc(cn1)CC(=S)N2CCOCC2 RH00942 c1ccc2c(c1)/C(=N/N)/C(=O)N2 RH00963 c1ccn(c1)c2c(cc(cc2Br)C3CCCCC3)Br BTB04648 Cc1cc(ccc1Cl)C2=Nc3ccccc3SC(C2)c4c(cccc4Cl)F BTB04644 Cc1cc(ccc1NC(=O)c2cccs2)c3nnc(o3)C(F)(F)F RH00933 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCCCC4 BTB02767 CCOC(=O)C(=CNc1ccc(cc1C)c2nnc(o2)C(F)(F)F)C(=O)OCC RH00944 c1ccnc(c1)SCC(=O)Nc2ccc3c(c2)OCCO3 NRB00094 c1cc(cc(c1)NC(=O)CSc2ccc(cc2)Cl)C#N BTB02776 CCOC(=O)/C(=C\Nc1ccc(cc1C)c2nnc(o2)C(F)(F)F)/C#N RH00951 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCc3ccco3 AW00032 c1cc(ccc1NC(=O)CC#N)Cl BTB06264 c1ccc(cc1)NC(=O)CC#N BTB06265 Cc1cc2c(cc1C)CSC(SC2)(C)C RH00970 c1ccc(cc1)Nc2nc(cs2)CN3CCCCC3 RH00972 c1ccc(cc1)c2c(n3c(n2)SCC3=O)c4ccccc4 NRB00945 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)c3ccc(cc3)[N+](=O)[O-] BTB02820 COc1cc(cc(c1Oc2ccc(cn2)[N+](=O)[O-])Br)C3SCCS3 BTB06326 COc1cc(cc(c1Oc2c(cccn2)[N+](=O)[O-])Br)C3SCCS3 BTB06328 Cc1ccc(cc1S(=O)(=O)Nc2c(cc(cc2C)C)C)[N+](=O)[O-] BTB00855 c1cc(c(cc1[N+](=O)[O-])Cl)N2CCCCC2 BTB02815 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)CCCC(=O)O BTB02809 c1ccc2c(c1)c(c(s2)C(=O)O/N=C(/c3cccc(c3)[N+](=O)[O-])\N)Cl BTB02811 c1cc(cc(c1)[N+](=O)[O-])/C(=N/OC(=O)c2ccc(cc2)[N+](=O)[O-])/N BTB02813 CC1CCN(CC(C1)(C)C)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB02868 CC1(CC2CC(C1)(CN2c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C)C BTB02870 CCOC(=O)C(=CNc1cc(ccc1F)C(F)(F)F)C(=O)OCC AW00114 Cc1cccc(c1NC(=O)CSC(=O)c2ccc(cc2)[N+](=O)[O-])C BTB02789 Cn1cc(c(n1)/N=C/N(C)C)C(=O)Nc2ccc(c(c2)Cl)F BTB06358 CC1CCC(CN(C1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F)(C)C BTB02867 CC1(CC2CC(C1)(CN2c3ccc(cc3[N+](=O)[O-])C(F)(F)F)C)C BTB02869 c1cc2c(cc1NC(=O)CN3CCOCC3)OCCO2 NRB00104 Cc1cc(c(c(c1Cl)C)Cl)OC(=O)c2ccc(cc2)[N+](=O)[O-] BTB02854 Cc1cc(c(c(c1Cl)C)Cl)OC(=O)C(c2ccccc2)C3CCCC3 BTB02857 Cc1cc(c(c(c1Cl)C)Cl)Oc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] BTB02858 c1ccc(cc1)C(=O)CC(C[N+](=O)[O-])c2ccc(cc2)Cl NRB00105 c1cc(cc(c1)[N+](=O)[O-])c2ncon2 BTB02807 Cc1cc(c(c(c1Cl)C)Cl)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB02859 c1cc(ccc1CN2CCN(CC2)CCO)[N+](=O)[O-] AW00111 Cc1cc(c(cc1Cl)C)SCC2=NNC(=O)C2 BTB06359 c1ccnc(c1)SCC2=NNC(=O)C2 BTB06361 c1ccc(cc1)C(C(=O)c2ccccc2)Sc3ccc(cc3)Cl BTB02890 CCCCCCCCCCCCNC(=N)NC(=S)NC(=S)NCCCCCCCCCCCC NRB00936 c1cc2ccc(nc2c(c1)C(F)(F)F)C(F)(F)F NRB00901 c1ccc2c(c1)ccc(c2C(c3cccs3)N4CCCCC4)O NRB00102 C=CCSc1[nH]c(c(n1)c2ccccc2)c3ccccc3 NRB00949 Cc1cc(n(n1)S(=O)(=O)c2cc(ccc2OC)c3csnn3)C NRB00956 CC1(C/C(=N\NC(=O)N)/c2ccc(cc2O1)OCc3ccccc3)C NRB00913 c1cc(cnc1)NC(=S)N2CCN(CC2)c3nccc(n3)C(F)(F)F AW00137 COc1ccc(cc1S(=O)(=O)Nc2ccccc2)c3csnn3 NRB00957 CNC(=S)NNC(=O)c1ccccn1 NRB00959 CC(C)(C#C)N1CNC(=S)NC1 BTB02903 c1ccn(c1)c2cccc(c2)/C(=N/OC(=O)c3ccc(cc3)[N+](=O)[O-])/N BTB02906 c1ccn(c1)c2cccc(c2)/C(=N/OC(=O)c3cccs3)/N BTB02907 CC(C)NC(=S)NC(=N)Nc1ccc(c(c1)Cl)Cl.C(=C\C(=O)O)\C(=O)O NRB00937 C=CCn1c(n[nH]c1=S)c2ccccc2O NRB00966 c1cc(c(cc1C(F)(F)F)NC(=O)c2ccncc2)N3CCCCC3 BTB02865 Cc1cc(=O)oc2c1c(n[nH]2)CSc3ccc(cc3)Cl BTB06367 C=CCSc1c(cccn1)C(=O)O BTB06373 c1cc(ccc1N2C(=O)CCC2=O)S(=O)(=O)N3CCN(CC3)c4nccc(n4)C(F)(F)F AW00136 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C/C(=N/Nc3c(cc(cc3Cl)Cl)Cl)/C BTB04743 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC#N BTB06378 c1cc(c(cc1F)F)NC(=S)N2CCN(CC2)c3nccc(n3)C(F)(F)F AW00138 c1ccc(cc1)c2c(nc([nH]2)Sc3ccc(cc3)[N+](=O)[O-])c4ccccc4 NRB00947 c1cc(c(cc1NC(=S)N2CCN(CC2)c3nccc(n3)C(F)(F)F)Cl)F AW00139 CN(C)/C=C/1\C(=NNC1=O)CSc2ccccn2 BTB06385 Cc1cc(c(cc1Cl)Cl)SCC\2=NNC(=O)/C2=C/N(C)C BTB06386 Cc1cc(c(cc1Cl)Cl)SCc2c3c(cc(=O)oc3[nH]n2)C BTB06387 CCCCCCCCCCCCCCCC(=O)Nc1nc(=S)ss1 NRB00933 c1ccc(cc1)c2cnns2 NRB00953 CCOC(=O)CC1=CSC2=NCCN12.Cl BTB06353 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)c3cccs3 BTB02821 c1ccc(cc1)c2csc(n2)N/N=C/c3ccc(cc3)F.Cl ML00184 C=CCNC(=S)NNC(=O)c1ccccn1 NRB00961 CC(C)C(C)(C#N)NC(=O)c1cccnc1SC BTB06360 Cc1cc(c(cc1Cl)Cl)SCC2=NNC(=O)C2 BTB06362 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])Cl BTB02871 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C=N/OCC#Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB04752 Cc1c(nc(s1)c2ccccc2)c3ccc(cc3)CC(C)C RH01018 Cc1cccc2c1N(CCC2)c3nc(nc(n3)OC)OC BTB00839 Cc1ccc(cc1S(=O)(=O)Nc2cccc(c2)C(F)(F)F)[N+](=O)[O-] BTB00853 Cc1ccc(cc1S(=O)(=O)Nc2cc(c(cc2OC)Cl)OC)[N+](=O)[O-] BTB00854 c1cc(oc1)CNC(=S)C(=O)Nc2ccc3c(c2)OCCO3 NRB00113 c1cc(c(cc1/C=N/NC(=O)CNc2ccc(cc2F)F)[N+](=O)[O-])N3CCCC3 NRB00115 CCOC(=O)N/N=C/c1cccc2c1cccc2 ML00214 CC(=O)CN1C(=O)c2ccccc2S1(=O)=O BTB06380 Cc1cc(=O)oc2c1c(nn2c3ccccc3)c4ccccc4 BTB06383 CCCSc1c(cccn1)C(=O)N BTB06388 c1ccn(c1)c2ccc(cc2C#N)[N+](=O)[O-] BTB02905 c1ccc(c(c1)C(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccccc3N)C(=O)O BTB02887 Cc1cc(cc2c1ncc(c2O)C(=O)O)Cl BTB02846 CCOC(=O)N/N=C/c1ccc2c(c1)OCO2 ML00197 CCCSc1c(cccn1)C(=O)O BTB06368 CCCCCSc1c(cccn1)C(=O)O BTB06369 c1ccc(c(c1)C(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl)C(=O)O BTB02885 c1cc2c(cc1C(F)(F)F)n(nn2)O AW00118 Cc1cc(c(c(c1Cl)C)Cl)Oc2ccc(cc2)[N+](=O)[O-] BTB02866 CCOC(=O)N/N=C/c1ccc(c(c1)OC)OC ML00209 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)CCO AW00120 c1cc(ccc1C(=O)Nc2ccc(cc2)n3c(ccn3)C(F)(F)F)Cl AW00169 c1cc(c(cc1F)F)N2C(=O)CCC2=O NRB00133 Cc1cc(ccc1NC(=S)NNC(=O)c2c(c3ccccc3s2)Cl)Cl BTB00805 c1cc(ccc1N2C(SCC2=O)c3ccc(c(c3)Cl)Cl)F BTB00828 c1cc(ccc1NC(=O)CSc2ccc(cn2)C(F)(F)F)F NRB00124 CCN(CC)c1ccc(cc1)/C=C/c2cc[n+](cc2)Cc3ccc(cc3)F.[I-] NRB00128 c1ccnc(c1)SCC(=O)Nc2cccc(c2)[N+](=O)[O-] NRB00129 Cn1c(n[nH]c1=S)c2ccccc2O NRB00968 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)c3ccccc3C(=O)O BTB02886 CC(C(=O)O)Sc1[nH]c(c(n1)c2ccccc2)c3ccccc3 NRB00946 COc1ccc(cc1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl BTB02915 c1ccc2c(c1)CCN2Cn3c4ccccc4nn3 NRB00119 c1cc(ccc1C#N)Oc2ccc(cc2N)C(F)(F)F BTB02963 c1cc(c(cc1F)F)NC(=O)CSc2ccc(cn2)C(F)(F)F NRB00122 Cn1cc(c(n1)C(F)(F)F)S(=O)(=O)NCc2ccc3c(c2)OCO3 AW00155 C=CCNC(=S)NNC(=O)c1ccccc1 NRB00960 Cc1ccc(cc1S(=O)(=O)Nc2ccc3c(c2)OCO3)[N+](=O)[O-] BTB00856 Cc1ccc(cc1NC(=O)CSc2ccc(cn2)C(F)(F)F)F NRB00112 C=CCn1c(n[nH]c1=S)c2ccc(cc2)O NRB00969 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C=N/OCc2c(cccc2Cl)F BTB04751 c1cc(ccc1SCC2=NNC(=O)C2)Cl BTB06365 CCCCCC[n+]1ccccc1/C=C/c2ccc(cc2)N(C)C.[I-] NRB00125 COc1ccc(cc1NC(=O)CSc2ccc(cc2)Cl)Cl NRB00126 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C=N/OC(=O)c2ccc(cc2)F BTB04747 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C=N/OCc2c(cccc2Cl)Cl BTB04749 CCOC(=O)C1CCN(CC1)c2nc(nc(n2)OC)OC BTB00784 CCNS(=O)(=O)c1ccc(cc1)c2c(c3ccc(cc3o2)S(=O)(=O)NCC)Cl NRB00942 COc1ccc(cc1NC(=O)CSc2ccc(cn2)C(F)(F)F)Cl NRB00130 Cc1ccc2c(c1)CCCN2C(=O)c3c(c4ccccc4s3)Cl BTB00792 C/C(=N\NC(=O)OC)/c1ccc(cc1)c2ccccc2 NRB00985 C/C(=N\NC(=O)O)/c1ccc(cc1)Oc2ccccc2 NRB00986 c1cc(oc1)CNC(=S)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB00114 CNC(=S)NNC(=O)c1ccc(cc1)O NRB00963 Cc1c(c(nc(n1)c2ccccn2)N3CCN(CC3)CCO)Cl AW00143 COc1ccc(cc1)N2C(SCC2=O)c3ccccc3 BTB00804 c1cc2c(c(ccc2)/C=N/NC(=O)N/N=C/c3c4c(ccc3)cccc4)cc1 ML00190 c1cc(cc(c1)/C=N/NC(=O)N/N=C/c2cc(ccc2)O)O ML00192 CCOC(=O)N/N=C/c1ccc(cc1)OC ML00207 c1ccc(cc1)C(=O)COc2ccc(cc2Cl)S(=O)(=O)Nc3ccccc3 NRB00990 c1ccn(c1)c2cccc(c2)c3nc(on3)c4ccc(cc4)[N+](=O)[O-] BTB02909 c1ccc(cc1)c2c(nc([nH]2)SCC(=O)O)c3ccccc3 NRB00944 Cc1ccc(cc1S(=O)(=O)Nc2ccc(cc2)F)[N+](=O)[O-] BTB00798 Cc1ccc(cc1Cl)N2C(SCC2=O)c3ccc(c(c3)Cl)Cl BTB00803 c1c(ccnc1)/C=N/NC(=O)N/N=C/c2ccncc2 ML00187 c1csc(c1)/C=N/NC(=O)N/N=C/c2sccc2 ML00188 COc1c(ccc(c1)/C=N/NC(=O)N/N=C/c2cc(c(cc2)O)OC)O ML00191 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)O/N=C(/Cc3nc4cccnc4n3C5CC5)\N RH01024 CCSc1c(cccn1)C(=O)O BTB06379 CCOC(=O)N/N=C/c1ccccc1Cl ML00210 CCOc1c(cc(cc1)/C=N/NC(=O)N/N=C/c2cc(c(cc2)OCC)OC)OC ML00193 c1cc2c(c(c(cc2)O)/C=N/NC(=O)N/N=C/c3c(ccc4c3cccc4)O)cc1 ML00202 Cc1ccc(cc1)S(=O)(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N BTB06292 c1cc(ccc1NC(=S)Nc2ccc(cc2)Cl)Cl BTB04719 c1ccn(c1)c2cccc(c2)/C(=N/OC(=O)c3c(cccc3F)F)/N BTB02908 c1ccn(c1)c2cccc(c2)c3nc(on3)c4c(cccc4F)F BTB02911 c1ccc(c(c1)C2Nc3ccccc3C(=O)N2c4ccc(cc4)F)O BTB00759 c1cc(ccc1N2C(SCC2=O)c3ccc4c(c3)OCO4)F BTB00769 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C=N/OC(=O)c2cccs2 BTB04745 CCOC(=O)NNC(=S)Nc1ccccc1Cl ML00206 CCOC(=O)NNC(=S)Nc1cccc(c1)C(F)(F)F ML00208 COc1cc(c(cc1Cl)OC)/N=C/c2cc(cc(c2O)Cl)Cl BTB00767 CCOC(=O)/C(=C/N1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F)/C#N BTB04698 c1ccc(cc1)C2N(C(=O)CS2)c3ccccc3 BTB00768 CCOC(=O)NNC(=S)Nc1c(cccc1C)C ML00211 CCOC(=O)N/N=C/c1ccc(c(c1)Cl)Cl ML00212 Cc1ccc(cc1S(=O)(=O)N)[N+](=O)[O-] BTB00779 CC(=O)Nc1ccc(cc1C#N)N BTB00738 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2C(=O)OC BTB00741 c1cc(ccc1C(=O)Oc2ccc(cc2Sc3cc(ccc3OC(=O)c4ccc(cc4)[N+](=O)[O-])Cl)Cl)[N+](=O)[O-] BTB02957 c1cc2c(cccc2S(=O)(=O)N3CCCCCC3)c(c1)N NRB00866 c1cc(ccc1n2c(nnn2)c3ccc(c(c3)Cl)Cl)Cl BTB06249 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB06256 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2cc(c(cc2C)Cl)C BTB06224 CC1CC(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)[N+](=O)[O-] BTB00667 c1cc(c(nc1)N2CCN(CC2)CCO)[N+](=O)[O-] AW00142 c1c(c(c(cc1Br)Br)O)/C=N/NC(=O)N/N=C/c2c(c(cc(c2)Br)Br)O ML00150 c1ccc(cc1)/C=C/C=N/NC(=O)N/N=C/C=C/c2ccccc2 ML00152 c1ccc(cc1)Nc2nc3c(s2)CCCC3.Cl ML00161 COc1ccc(cc1)/C=N/Nc2nc(cs2)c3ccccc3.Cl ML00165 Cc1ccc(c(c1)C)n2c(nnn2)SCc3nc(no3)c4cccc(c4)[N+](=O)[O-] BTB02953 COc1ccc(cc1)NC(=S)NCCSc2ccc(cc2)Cl BTB02955 COc1ccc(cc1)/N=C/c2ccccc2 BTB00778 c1cc(oc1)C/N=C/c2ccc3c(c2)OCO3 BTB00780 c1cc(sc1)C(=O)Oc2ccc(cc2Sc3cc(ccc3OC(=O)c4cccs4)Cl)Cl BTB02958 c1c(ccc(c1)F)/C=N/NC(=O)N/N=C/c2ccc(cc2)F ML00137 c1cc(c(c(c1)Cl)/C=N/NC(=O)N/N=C/c2c(cccc2Cl)Cl)Cl ML00138 Cc1ccc(cc1)NC(=O)CSc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] BTB00676 c1cc(ccc1NC(=O)CSc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])F BTB00678 Cc1ccc(cc1)Sc2cc(ccc2[N+](=O)[O-])C(=O)c3ccccc3C(=O)O BTB02769 c1cc(c(cc1Oc2ccc(cc2Cl)Cl)C(F)(F)F)[N+](=O)[O-] BTB02741 Cc1cc(c(cc1Cl)Cl)Sc2nc(nc(n2)Sc3cc(c(cc3Cl)Cl)C)NC(C)(C#N)C(C)C BTB06346 CC(C)(C)SCCN/C(=N\c1ccc(cc1)Cl)/c2ccccc2Cl BTB06319 c1cc(ccc1C(=O)N2CCNCC2)[N+](=O)[O-] BTB06396 CCOC(=O)NNC(=S)Nc1cccc(c1)C ML00215 c1cc(ccc1NC(=S)NCCCn2ccnc2)Cl BTB04721 c1cc(c(cc1Cl)NC(=S)NCCCn2ccnc2)Cl BTB04722 CCOC(=O)CNc1ccc(c(c1)Cl)Cl RH01000 CCOc1ccc(cc1)/C=N/Nc2nc(cs2)c3ccccc3.Cl ML00168 Cc1ccc(cc1C)/N=C\2/N(C(=O)/C(=C/C(=O)OC)/S2)c3ccc(c(c3)C)C BTB04729 COC(=O)/C=C\1/C(=O)N(/C(=N/c2cccc(c2)SC)/S1)c3cccc(c3)SC BTB04731 CCOC(=O)CC(=O)NCC(=O)OCC RH01001 c1c(cc(c2c1nc(cc2O)O)Cl)Cl RH01004 C1C2CC3CC1CC(C2)(C3)C(=O)NN RH01025 Cc1ccc(cc1)Nc2nnns2 ML00062 c1cc(cnc1)c2nc(cs2)c3ccc(cc3)F.Br ML00064 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)c3cccnc3.Br ML00065 CC1=C(C(CC(=O)N1)c2ccc(cc2)F)C(=O)OC RH00945 COc1cccc(c1O)C2Nc3ccccc3C(=O)N2c4ccc(cc4)F BTB00758 c1cc(sc1)c2nnc(n2N)S RH01029 c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB02779 c1ccnc(c1)NC(=S)Nc2ccc(cc2Cl)Cl BTB04736 Cc1ccc(cc1Cl)/N=C/c2ccc(c(c2)Cl)Cl BTB00775 COc1ccc2c(c1)CCCN2C(=O)c3c(c4ccccc4s3)Cl BTB00793 c1cc(ccc1NCCC(=O)O)Cl RH01022 Cc1cc(c(cc1Cl)Cl)SCC#N BTB06266 c1cc2c(nc1)n(c(n2)C/C(=N/OC(=O)c3ccc(cc3)OC(F)(F)F)/N)C4CC4 RH01023 COC(=O)c1cc(=O)n2c3ccccc3nc2s1 BTB04713 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)c3c(cccc3F)F BTB02819 c1c(c(c(cc1Cl)Cl)O)/C=N/NC(=O)N/N=C/c2c(c(cc(c2)Cl)Cl)O ML00146 c1cc(cc(c1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F NRB00100 c1c(cc(c(c1)O)/C=N/NC(=O)N/N=C/c2c(ccc(c2)Br)O)Br ML00149 COc1c(cc(cc1)/C=N/NC(=O)N/N=C/c2cc(c(cc2)OC)Br)Br ML00151 c1ccc(cc1)/C=N/Nc2nc(cs2)c3ccccc3.Cl ML00162 c1cc(cc(c1)SCC(=O)Nc2ccc(cc2F)F)C(F)(F)F NRB00101 c1ccc(cc1)C(=O)N/N=C/c2cc(ccc2N3CCCCC3)[N+](=O)[O-] NRB00103 c1ccc(c(c1)C(=O)NC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)F BTB04705 c1ccc(cc1)/C=N/c2cccc(c2)C(F)(F)F BTB00776 Cc1cccc(c1NC(=O)CSC(=O)c2c(c3ccccc3s2)Cl)C BTB02788 c1cc(c(cc1)Cl)/C=N/NC(=O)N/N=C/c2c(cccc2)Cl ML00135 CC(c1ccc(cc1)/C=N/NC(=O)N/N=C/c2ccc(cc2)C(C)C)C ML00136 c1cc(cc(c1)[N+](=O)[O-])/C(=N/OC(=O)c2c(cccc2F)F)/N BTB02812 c1cc(cc(c1)[N+](=O)[O-])/C(=N/OC(=O)c2cccs2)/N BTB02814 CN(c1ccc(cc1)/C=N/NC(=O)N/N=C/c2ccc(cc2)N(C)C)C ML00140 Cc1c(n2ccccc2n1)C(=O)NN RH01013 Cc1c(nc(s1)N)c2ccc(cc2)CC(C)C.Br RH01015 c1cc(ccc1CN2CCN(CC2)CCO)F AW00107 COc1ccc(cc1/C=N/NC(=O)CNc2ccccc2)Br NRB00109 COc1cc(cc(c1Oc2nc3c(s2)cc(cc3Cl)Cl)Br)C4SCCS4 BTB06327 CC1(CC(=O)c2cc(c(cc2O1)O)Cl)C NRB00918 Cn1c(n[nH]c1=S)COc2ccccc2 NRB00977 Cc1ccc(cc1[N+](=O)[O-])NS(=O)(=O)c2cc(ccc2C)[N+](=O)[O-] BTB00852 COc1ccc(cc1OC)/C=N/NC(=S)N ML00173 c1cc(ncc1C(F)(F)F)SCC(=O)N RH01002 COC(=O)/C=C\1/C(=O)N(/C(=N/c2ccc(cc2)Cl)/S1)c3ccc(cc3)Cl BTB04730 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(cc2)C3CCCCC3 RH01010 c1cc(cc(c1)/C=N/NC(=O)N/N=C/c2cc(ccc2)[N+](=O)[O-])[N+](=O)[O-] ML00143 c1c(cnc(c1Cl)N2CCN(CC2)CCO)C(F)(F)F AW00100 CC(C)(C)c1ccc(cc1)/N=C\2/N(C(=O)/C(=C/C(=O)OC)/S2)c3ccc(cc3)C(C)(C)C BTB04732 COc1cc(cc(c1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Br)C3SCCS3 BTB06312 Cc1ccc(cc1C)NC(=S)Nc2ccc(c(c2)C)C BTB04720 c1ccc(cc1)c2csc(n2)N/N=C/c3ccccc3Cl.Cl ML00176 c1cc(c(cc1/C=N/NC(=S)N)Cl)Cl ML00179 CSc1cccc(c1)NC(=S)Nc2ccccn2 BTB04738 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C=N/OC(=O)c2c(cccc2F)F BTB04744 Cc1cccc2c1nc(cc2O)C NRB00906 c1ccc(cc1)c2nnc(o2)S NRB00926 c1ccc(cc1)CC(=O)N2CCOCC2 NRB00927 COc1cc(cc(c1O)Br)C2SCCS2 BTB06307 Cc1cc2c(cc1C)CSC(SC2)/C=C/c3ccccc3 RH00969 Cc1c(ccc2c1OC(CC2=O)(C)C)OC NRB00915 CC1(CC(=O)c2cc(c(cc2O1)OC)OC)C NRB00916 CC(C)(C)SCCN/C(=N\c1cccc(c1)F)/c2ccccc2Cl BTB06320 c1cc2c(c(c1)F)ncc(c2O)C(=O)O BTB02847 COC(=O)/C=C\1/C(=O)N(/C(=N/c2cccc(c2)C(F)(F)F)/S1)c3cccc(c3)C(F)(F)F BTB04734 Cc1cc(c(c(c1Cl)C)Cl)OC(=O)c2cccs2 BTB02855 Cc1cc(c(c(c1Cl)C)Cl)OC(=O)c2c(cccc2Cl)Cl BTB02856 c1c(cnc(c1C(F)(F)F)N2CCN(CC2)CCO)Cl AW00098 Cc1cccc(c1)c2nc3cc(ccc3c(=O)o2)Cl NRB00165 CCOC(=O)c1c(csc1N)c2ccc(cc2)F AW00215 CCOc1ccc(cc1)/C=N/NC(=O)OCC ML00218 CC(C)(C)c1ccc(cc1)NC(=O)CCC(=O)N(Cc2ccccc2)Cc3ccccc3 NRB00168 CCOC(=O)N/N=C/c1cc(cc(c1O)Br)Br ML00221 CCOC(=O)N/N=C/c1cc(ccc1O)Br ML00222 CC(=O)Nc1cc2cc(ccc2oc1=O)NC(=O)c3c(cccc3F)F BTB04783 CC(=O)Nc1cc2cc(ccc2oc1=O)NS(=O)(=O)c3ccc(c(c3)OC)OC BTB04791 COC(=O)c1cccc(c1C(=O)OC)/N=C/c2cc(cc(c2O)Cl)Cl BTB00873 c1ccc(cc1)C(=O)NNC(=O)NC(=O)c2ccccc2Cl RH01053 c1ccc(c(c1)C(=O)NC(=O)NNC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl RH01054 CC(C)(C)NC(=S)Nc1cc(ccc1Cl)C(F)(F)F BTB02977 c1c(cc2c(c1F)nc(s2)N)F BTB04754 COc1ccc(cc1)c2nnc(n2c3cccc(c3)OC)S BTB00881 COc1ccc(cc1)c2nnc(n2c3ccccc3Cl)S BTB00885 Cc1nnc2n1N=C(C(S2)C)c3ccc(cc3)CC(C)C.Br RH01057 CC(=O)c1ccc(c(c1)CSc2nccc(n2)O)OC BTB04760 CC(C)(C)NC(=S)Nc1c(cc(cc1Cl)Cl)Cl BTB02985 Cc1cc(c(c(c1)C)NC(=S)NC(C)(C)C)C BTB02986 Cc1c(c(c(cn1)CSc2nccc(n2)O)CO)O BTB04763 Cc1ccc(c(c1)C)NC(=S)N BTB04770 Cc1ccc(cc1C)N2C(=O)CC(=O)N(C2=S)c3ccc(c(c3)C)C BTB04776 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2Sc3cc(ccc3OS(=O)(=O)c4ccc(cc4)C)Cl)Cl BTB02998 CN(C)/C=N/C(=S)Nc1cccc(c1)Cl BTB04782 Cc1cc(ccc1Cl)C2=CSC3=NCCN23.Br BTB03010 Cc1cc(ccc1Cl)C2=CSC3=NCCCN23.Br BTB03011 c1ccc(cc1)COc2ccc(cc2)/C(=N/O)/N BTB03013 Cc1ccc(cc1)c2nnn(n2)CC(=O)Nc3ccc(cc3F)F NRB00134 c1cc(ccc1n2c(ccn2)C(F)(F)F)[N+](=O)[O-] AW00166 c1ccc(c(c1)C(=O)NC(=O)NNC(=O)c2ccco2)Cl RH01055 c1cc(ccc1NC(=O)CSc2nnc(s2)SCC(=O)Nc3ccc(cc3)F)F NRB00131 c1ccc(c(c1)C(=O)Nc2ccc(cc2)n3c(ccn3)C(F)(F)F)C(=O)O AW00168 c1cc(ccc1SCC/N=C/c2ccc(s2)[N+](=O)[O-])Cl BTB02990 c1cc(ccc1SCC/N=C/c2cc(cc(c2O)Cl)Cl)Cl BTB02991 c1cc(c(c(c1)Cl)CSc2nccc(n2)O)Cl BTB04761 C=CCNC(=S)NNC(=O)Cc1ccc(cc1)[N+](=O)[O-] NRB00964 c1cc(ccc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)n3c(ccn3)C(F)(F)F AW00179 CN(C)/C=N/C(=S)Nc1cccc(c1)F BTB04781 C=CCn1c(n[nH]c1=S)c2ccccc2 NRB00974 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2SCc3ccccc3)Cl NRB00142 c1cc-2c(cc1S(=O)(=O)N3CCCCC3)C(=O)c4c2ccc(c4)S(=O)(=O)N5CCCCC5 NRB00991 CCCC(=O)c1cc2cc(ccc2oc1=O)[N+](=O)[O-] BTB06397 CCOC(=O)c1ccc(cc1)NC(=O)CSc2ccccn2 NRB00132 C/C(=N\O)/c1ccc2c(c1)CCC2 NRB01001 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)CCOC(=O)CCC(=O)O AW00180 c1ccc(cc1)CSc2cc(ccc2NC(=O)Nc3ccccc3)Cl NRB00141 Cn1c(n[nH]c1=S)c2ccccn2.CN(C)C=O NRB00971 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=O)c3cccc(c3)C(F)(F)F BTB03075 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3ccc4c(c3)cc(c(=O)o4)NC(=O)C BTB04775 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)CCOC(=O)CSCC(=O)O AW00184 CC(=O)Nc1cc(c(cc1N=Nc2c(cc(cc2Cl)[N+](=O)[O-])[N+](=O)[O-])OC)N(CCC#N)CCO NRB01101 CCOC(=O)c1c(n(c2c1cc(cc2)OC(=O)c3cccnc3SCC)c4ccccc4)C RH01064 CCOC(=O)c1c(n(c2c1cc(cc2)OC(=O)c3cccs3)c4ccccc4)C RH01065 COc1ccc(cc1OC)CCNC(=N)N.OS(=O)(=O)O RH01066 c1ccc(c(c1)C(=O)NC2CCCCNC2=O)N BTB06496 Cc1ccc2cc(ccc2c1)F RH01072 c1ccc2c(c1)C(C(=O)N2)(Cc3ccncc3)O RH01085 CCCC(=O)c1cc2cc(cc(c2oc1=O)Br)Br BTB06398 c1cc2c(cc1Br)C(C(=O)N2)(Cc3ccncc3)O RH01087 CC(=O)Nc1cc2cc(ccc2oc1=O)NS(=O)(=O)c3ccc(c(c3)Cl)Cl BTB04793 Cc1c(cccc1Cl)NC(=S)/N=C/N(C)C BTB04784 CN(C)/C=N/C(=S)Nc1cccc(c1)SC BTB04785 CC(C)(C#C)N1CNC(=NC1)SC.I BTB03080 CC(=O)COc1ccc(cc1Cl)Cl BTB03082 CCCC(=O)c1cc2cc(ccc2oc1=O)Br BTB06399 CCCc1cc(=O)oc2c1c(n[nH]2)C BTB06405 COc1ccccc1c2nnc(n2c3ccccc3)S RH01070 COc1cc(cc(c1O)Br)/C=C(\C#N)/C(=O)Nc2ccc(c(c2)Cl)F BTB06406 CCCc1cc(=O)oc2c1c(nn2c3ccccc3)C BTB06409 c1ccc2c(c1)c(c(s2)C(=O)NNC(=O)NC(=O)c3ccccc3Cl)Cl RH01047 CCOC(=O)c1c(n(c2c1cc(cc2)OC)c3ccccc3)C RH01048 COc1cccc(c1)CC(=O)NNC(=O)NC(=O)c2ccccc2Cl RH01052 c1ccc(cc1)NC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW00194 CC(=O)Nc1ccc2c(c1)CCCC2=O NRB00998 c1ccc(cc1)Oc2c(cccn2)C(=O)NN BTB03059 c1ccc(cc1)Oc2c(cccn2)C(=O)Oc3ccccc3 BTB03060 CCOC(=O)CC1=Nn2c(nnc2SC1)c3cccs3 RH01033 c1ccc(c(c1)C(=O)NC(=O)NNC(=O)c2cccs2)Cl RH01039 c1ccc(c(c1)C(=O)NC(=O)NNC(=O)c2ccc(cc2)C(F)(F)F)Cl RH01045 c1ccc(cc1)CSc2cc(ccc2NC(=O)c3ccccc3Cl)Cl NRB00139 CCOC(=O)c1c(n(c2c1cc(cc2)O)C3CC3)C RH01050 c1cc-2c(cc1S(=O)(=O)N3CCOCC3)C(=O)c4c2ccc(c4)S(=O)(=O)N5CCOCC5 NRB00992 c1cc-2c(cc1S(=O)(=O)N)C(=O)c3c2ccc(c3)S(=O)(=O)N NRB00993 c1cc(ccc1NC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl AW00193 c1ccc2c(c1)c(c[nH]2)/C=C(\C#N)/c3[nH]c4ccccc4n3 BTB04758 CC(C)(C)NC(=S)Nc1cccc(c1Cl)Cl BTB02973 CSc1c(cccn1)C(=O)N BTB06434 Cc1ccc(cc1NC(=S)Nc2ccc(cc2)n3c(ccn3)C(F)(F)F)Cl AW00178 CC(C)NC(=S)NNC(=O)C1CC2CCC1O2 AW00196 c1cc(sc1)c2nc3cc(ccc3c(=O)o2)Cl NRB00146 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)C3CCCCC3 NRB00155 CCOC(=O)C(=CNCCNc1c(cccn1)C(F)(F)F)C(=O)OCC AW00203 CCC(=O)N1CCCc2c1cccc2 NRB01032 CC(=O)OC(c1ccc(cc1)S(=O)(=O)C)OC(=O)C NRB01028 CCOC(=O)/C(=C/NC1CCCCNC1=O)/C#N BTB06498 c1ccc(c(c1)C(=O)NC(=O)NNC(=O)c2cc(cc(c2)Cl)Cl)Cl RH01051 CCCc1cc(=O)oc2c1c(nn2c3cccc(c3)Cl)C BTB06410 Cc1cccc(c1)NC(=S)NCc2ccccn2 BTB06413 c1cc(ccc1C(=O)N2CCN(CC2)C(=O)c3ccc(cc3)Cl)Cl BTB06415 CN(C)c1ccc(cc1)C(=O)c2ccccc2 NRB01050 CCOC(=O)c1ccccc1C(=O)c2ccc(cc2)N(C)C NRB01052 c1cc(ccc1S(=O)(=O)c2ccc(c(c2)O)[N+](=O)[O-])Cl BTB06435 CCOC(=O)CSc1cc(c(cc1C)Cl)C BTB06438 CN(C)c1ccc(cc1)C(=O)N2CCCc3c2cccc3 NRB01012 Cc1c2ccccc2c(c3c1cccc3)C(=O)OC NRB01020 CC(C)c1ccc(c(c1)Br)NC(=O)C NRB01031 CCOc1cc(c(cc1N(CCOC(=O)C)CCOC(=O)C)NC(=O)C)/N=N/c2c(cc(cc2Br)[N+](=O)[O-])[N+](=O)[O-] NRB01098 CCCC\1=NN(C(=O)/C1=C/c2ccc(cc2)Cl)c3ccccc3 BTB06418 CC(C)(C)c1ccc(cc1[N+](=O)[O-])C(=O)O NRB01030 c1cc(ccc1Sc2ccc(c(c2)O)[N+](=O)[O-])Cl BTB06427 c1ccc(cc1)Sc2ccc(c(c2)O)[N+](=O)[O-] BTB06428 CC\1=NN(C(=O)/C1=C\c2cc(cs2)Br)c3cccc(c3)Cl BTB06420 c1cc-2c(cc1Br)CCc3c2ccc(c3)Br NRB01048 Cc1cc(c(cc1Cl)C)Sc2ccc(c(c2)O)[N+](=O)[O-] BTB06429 CC(=O)C(=CNc1c(cn(n1)C)C(=O)Nc2ccc(c(c2)Cl)F)C(=O)C BTB06424 c1ccc(cc1)S(=O)(=O)c2ccc(c(c2)O)[N+](=O)[O-] BTB06430 c1ccc2c(c1)cc(s2)C(=O)Oc3cc(ccc3[N+](=O)[O-])S(=O)(=O)c4ccc(cc4)Cl BTB06436 CSc1c(cccn1)C#N BTB06444 Cc1ccc(c(c1)C)NC(=S)NC(C)(C)C BTB02987 c1ccc(cc1)Oc2c(cccn2)C(=O)O BTB02988 c1cc(sc1)c2nnc3n2N=C(CS3)c4ccc(cc4)OC(F)(F)F.Br RH01061 CC(=O)Nc1cc(c(cc1/N=N\c2c(cc(cc2Br)[N+](=O)[O-])[N+](=O)[O-])OC)N(CCOC(=O)C)CCOC(=O)C NRB01100 CC(=O)Nc1ccc(cc1Cl)[N+](=O)[O-] BTB06452 Cc1cc(ccc1Cl)c2cnc3ccc(cc3n2)OC BTB03032 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccc(cc3)F BTB03047 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3cc(ccc3N4CCOCC4)C(F)(F)F BTB03050 c1cc(ccc1NC(=O)/C=C/C(=O)O)n2c(ccn2)C(F)(F)F AW00170 CC(C)(C)NC(=S)Nc1ccccc1C(F)(F)F BTB02981 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)CCOC(=O)/C=C/C(=O)O AW00174 CC(C)(C)CC(C)(C)NC(=O)c1cccnc1Oc2ccccc2 BTB03051 CC(C)(C#C)NC(=O)c1cccnc1Oc2ccccc2 BTB03052 Cc1ccc(cc1)SC(=O)c2cccnc2Oc3ccccc3 BTB03055 C/C(=N\O)/COc1ccc(cc1Cl)Cl BTB03087 C/C(=N\OC(=O)c1c(cccc1Cl)F)/COc2ccc(cc2Cl)Cl BTB03088 C/C(=N\OC(=O)c1c(cccc1F)F)/COc2ccc(cc2Cl)Cl BTB03089 c1cc(ccc1C2=NCCO2)NC(=O)Nc3ccc(cc3)OC(F)(F)F AW00201 CC(=O)Nc1ccc(cc1)[N+](=O)[O-] BTB06454 c1cc(ccc1C(=O)N)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB03016 c1cc(ccc1C2CCCCC2)NC(=O)CSCC(=O)NN NRB00159 COC(=O)c1ccccc1c2ccccc2C(=O)OC NRB01044 CCOC(=O)N/N=C/c1cccc(c1)[N+](=O)[O-] ML00216 Cc1ccc2c(c1)c(=O)n(c(n2)C)c3ccc(cc3)F BTB00749 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)C3CCCCC3 NRB00156 CC(=O)Nc1ccc(cc1)/N=N/c2ccccc2 BTB06462 Cc1c(c(no1)c2ccccc2)C(=O)O/N=C(\C)/COc3ccc(cc3Cl)Cl BTB03090 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc(ccc2N)[N+](=O)[O-] BTB03095 c1ccc2c(c1)c(c(s2)C(=O)NNC(=O)c3ccccc3N)Cl BTB03097 CCc1c(c2cc(ccc2n1Cc3ccccc3)O)C(=O)OC RH01056 COc1cc(cc(c1OS(=O)(=O)c2ccc(cc2)Cl)Br)C3SCCS3 BTB06477 COc1cc(cc(c1OC(=O)c2cc3ccccc3s2)Br)C4SCCS4 BTB06483 c1ccc2c(c1)[nH]c(n2)/C(=C/c3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)/C#N BTB04757 CCOC(=O)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl NRB00127 c1cc(ccc1C#N)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB02962 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)C(=S)NCc4ccccc4 RH01011 CC(=O)Nc1ccc(cc1)/C=N/NC(=O)N/N=C/c2ccc(cc2)NC(=O)C ML00142 c1c(ccc(c1)O)/C=N/NC(=O)N/N=C/c2ccc(cc2)O ML00144 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=O)NC(=O)c3ccccc3Cl RH01040 c1ccc(c(c1)C(=O)NC(=O)NNC(=O)c2cccnc2)Cl RH01041 CN(C)/C=N/C(=S)Nc1cccc(c1)C(F)(F)F BTB04779 CC(=O)Nc1cc2cc(ccc2oc1=O)NC(=O)c3ccc(cc3)[N+](=O)[O-] BTB04771 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc4c(c3)cc(c(=O)o4)NC(=O)C BTB04772 c1ccc(cc1)Sc2c(cccn2)C#N BTB06464 c1ccc(cc1)COc2ccc(cc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB06473 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)NC(=O)c3ccccc3Cl RH01043 COc1cccc(c1)C(=O)NNC(=O)NC(=O)c2ccccc2Cl RH01044 c1ccc(c(c1)C(=O)NC(=O)NNC(=O)COc2ccc(cc2)SC(F)(F)F)Cl RH01046 c1ccc(cc1)n2c3c(cn2)c(nc(n3)c4ccncc4)N BTB03038 Cc1cc(ccc1NC(=O)C)[N+](=O)[O-] BTB06461 CC(=O)Nc1ccc(cc1Cl)/N=N/c2ccccc2 BTB06463 COc1cc(cc(c1OC)OC)/C=C(\C#N)/c2c(c(n(n2)c3ccccc3)n4cccc4)C#N BTB03039 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3ccc(c(c3)Cl)Cl)/C#N)C#N)n4cccc4 BTB03040 Cc1ccc(cc1Cl)/N=C\2/N(C(=O)/C(=C/C(=O)OC)/S2)c3ccc(c(c3)Cl)C BTB04733 c1ccnc(c1)NC(=S)Nc2cccc(c2)C(F)(F)F BTB04737 CCOC(=O)c1c(nc2n1cccc2)C RH01008 CCCCc1ccc(c(c1)C)NC(=O)C(=S)NCc2ccccc2 RH01012 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=O)c3ccc(cc3)[N+](=O)[O-] BTB03073 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=O)c3cccnc3Oc4ccccc4 BTB03074 c1ccc(cc1)Oc2c(cccn2)C(=O)N3CCOCC3 BTB03053 c1ccc(cc1)COc2ccc(cc2)Oc3c(cccn3)[N+](=O)[O-] BTB06474 c1ccc(cc1)COc2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-] BTB06475 c1ccc(cc1)COc2ccc(cc2)Oc3ccc(cc3)[N+](=O)[O-] BTB06476 c1ccc2c(c1)c(cc3c2cc(cc3)[N+](=O)[O-])C#N NRB01061 c1ccc2c(c1)CN(C2)c3cccc(c3)Cl NRB01073 c1cc(ccc1C2SCCS2)Oc3ccc(cc3)[N+](=O)[O-] BTB06455 c1cc(ccc1c2ncon2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB03017 CCOC(=O)c1ccc(c(c1)Cl)OC(=O)c2cccnc2Oc3ccccc3 BTB03063 c1cc(c(cc1NC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl AW00191 CCOC(=O)c1ccc(cc1)NC(=O)C(=S)NCc2ccccc2 NRB00148 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3c(cc(cc3Br)C4SCCS4)OC BTB06482 CCOC(=O)NNC(=S)Nc1ccccc1OC ML00226 CCOC(=O)N/N=C/c1ccco1 ML00228 CCOC(=O)N/N=C/c1cccs1 ML00229 Cc1cc(ccc1NC(=S)NNC(=O)c2ccc(cc2)OC)Cl BTB00862 c1ccc(cc1)Oc2c(cccn2)C(=O)Sc3ccccc3 BTB03054 CCOC(=O)CSC(=O)c1cccnc1Oc2ccccc2 BTB03058 COc1ccc(cc1)C(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F BTB00869 CCOC(=O)N/N=C/c1ccc(c(c1)O)OC ML00230 CCOC(=O)N/N=C/c1c2ccccc2ccc1O ML00231 CCOC(=O)N/N=C/c1c[nH]c2c1cccc2 ML00232 c1ccc(cc1)Oc2c(cccn2)C(=O)Oc3ccc(cc3)[N+](=O)[O-] BTB03061 COc1ccc(cc1)OC(=O)c2cccnc2Oc3ccccc3 BTB03062 COc1cc(cc(c1OC(=O)c2cccs2)Br)C3SCCS3 BTB06478 Cc1cc(c(cc1Cl)C)S(=O)(=O)Oc2c(cc(cc2Br)C3SCCS3)OC BTB06479 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2Br)C3SCCS3)OC BTB06480 COc1cc(cc(c1OS(=O)(=O)c2cc(cc(c2)Cl)Cl)Br)C3SCCS3 BTB06481 COc1ccc(cc1NC(=O)CSCc2ccco2)Cl NRB00169 CCOc1ccccc1/C=N/NC(=O)OCC ML00217 CCOC(=O)N/N=C/c1cc(cc(c1O)Cl)Cl ML00220 CCOC(=O)N/N=C/c1ccc(cc1)O ML00223 CCOC(=O)CSC(=O)c1c(onc1c2c(cccc2Cl)Cl)C BTB00867 CCOC(=O)N/N=C/c1ccc(cc1)Cl ML00225 Cc1cc(cc(c1)N2Cc3ccccc3C2)C NRB01076 c1cc(c(cc1[N+](=O)[O-])C(F)(F)F)N2CCCCC2 NRB01083 CCOC(=O)N/N=C/c1ccccc1O ML00227 Cc1cc(ccc1n2c(nnc2S)c3ccc(cc3)OC)Cl BTB00884 c1ccc(cc1)NNC(=S)Nc2ccccc2Cl ML00240 c1ccc2c(c1)CCCN2C(=O)C(F)(F)F NRB01103 COc1cccc(c1)NC(=S)NNc2ccccc2 ML00238 c1ccc(c(c1)/C=N/c2nccs2)O ML00246 c1ccc(cc1)NC(=S)NNc2cccc(c2)C(F)(F)F ML00239 COc1ccc(cc1)c2nnc(n2c3cc(ccc3Cl)Cl)S BTB00886 CCOC(=O)c1c(onc1c2c(cccc2Cl)Cl)C BTB00888 CNc1ccc(cc1C(F)(F)F)[N+](=O)[O-] NRB01081 CC(C)(C)c1cn2c(n1)sc(n2)C(C)(C)C BTB06488 CCOC(=O)N/N=C/c1cccc(c1)O ML00235 Cc1cc(cc(c1Cl)C)Oc2c(cccn2)C(=O)O BTB06497 C1CCNC(=O)C(C1)N2CNC(=S)NC2 BTB06499 Cc1cc(ccc1NC(=O)C)/N=N/c2ccccc2 BTB06500 Cc1ccc(cc1)C(=O)CSC2=NCCCCC2.Br ML00242 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSC2=NCCCCC2.Br ML00244 CCCC(=O)c1cc2ccccc2oc1=O BTB06400 CCCc1cc(=O)oc2c1c(nn2C)C BTB06404 CCCC1=NN(C(=O)C1)c2ccccc2 BTB06411 COc1cc(ccc1O)/C=N/c2nccs2 ML00248 Cc1nnc2n1N=C(CS2)c3ccc(cc3)Br.Br RH01058 c1ccn2c(c1)ncc2[N+](=O)[O-] NRB01107 CCN(CCOCCOCC)c1ccc(c(c1)NC(=O)C)N=Nc2c(cc(cc2C#N)[N+](=O)[O-])C#N NRB01104 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=O)c3cc(ccc3N)Cl BTB03098 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=O)c3cc(ccc3N)[N+](=O)[O-] BTB03099 CC(C)(C)c1ccc(cc1)c2nc3cc(ccc3c(=O)o2)Cl NRB00160 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)cc(c(=O)o3)NC(=O)C BTB04792 COc1ccc(cc1)C(=O)NN BTB00865 Cn1ccnc1SCC(=O)Nc2ccc(cc2)C3CCCCC3 NRB00161 CC(C)c1ccc(cc1)NC(=S)NNC(=O)c2ccc(cc2)OC BTB00871 COc1cc(c(cc1Cl)OC)N2C(SCC2=O)c3ccccc3 BTB00872 CCOC(=O)CSC(=O)c1c(c2ccccc2s1)Cl BTB00876 c1cc(ccc1NC(=O)CCC(=O)N2CCCC2)F NRB00164 CCOC(=O)c1c(csc1N)c2ccc(cn2)C AW00213 COc1ccc(cc1)C(=O)c2ccc(cc2OC)OC NRB01079 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2cccs2 BTB03084 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2cc(c(c(c2)OC)OC)OC BTB03086 CC(=O)Nc1cc(=O)oc2c1cc(cc2)NC(=O)c3ccc(cc3)F BTB04787 CC(=O)Nc1cc2cc(ccc2oc1=O)NS(=O)(=O)c3cc(ccc3OC)OC BTB04790 c1cc(ccc1NC(=O)CSc2nccc(n2)C(F)(F)F)Br AW00238 c1cc2c(cc1NC(=O)CSCc3ccc(cc3Cl)Cl)OCO2 NRB00180 Cc1cc(cc(c1OC)[N+](=O)[O-])[N+](=O)[O-] BTB03138 c1ccc(c(c1)C(=O)NC2CCCCNC2=O)NC(=O)c3ccc(cc3)Cl BTB06526 Cc1c(c(c(c(c1C)C)CSCC(=O)Nc2ccc(cc2F)F)C)C NRB00178 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=O)c3ccccc3N BTB03108 CCOC(=O)c1ccc(cc1)NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F AW00222 c1ccc(c(c1)C#N)NC(=O)CSc2ccc(cn2)C(F)(F)F NRB00171 CC1=C(C(=O)c2ccccc2C1=O)C NRB01132 c1ccc(cc1)C2=C(C(=O)OC2)C#N NRB01134 COc1ccccc1c2nnc(n2c3ccccc3)Sc4ccc(cc4[N+](=O)[O-])C(F)(F)F RH01122 c1cc(c(c(c1)Cl)C(=O)NC(=O)Oc2ccc(cc2F)F)Cl BTB04836 COc1ccc(c(c1C(=O)Nc2ccc(c(c2)Cl)F)OC)[N+](=O)[O-] BTB04839 COc1ccc(cc1NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F)Cl AW00234 Cc1cccc(c1OC(=O)c2cc(cc(c2)Cl)F)OC BTB03162 CC(=O)c1cc2cc(ccc2o1)[N+](=O)[O-] BTB03194 c1cc(ccc1C#N)N2CCOCC2 NRB01111 COc1cc(ccc1[N+](=O)[O-])Sc2ccc(cc2)Cl BTB06532 Cc1cccc(c1NC(=S)N2CCCc3c2c(ccc3)C)C BTB01014 Cc1cccc(c1NC(=S)N2CCCc3c2cccc3)C BTB01015 c1c(c(sc1[N+](=O)[O-])N)[N+](=O)[O-] NRB01126 Cn1ccnc1SCC(=O)Nc2ccc3c(c2)OCO3 NRB00172 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)c3ccc(cc3)Cl BTB06538 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)c3ccc(cc3)[N+](=O)[O-] BTB06540 CC(=O)Oc1cc(ccc1[N+](=O)[O-])Sc2ccccc2 BTB06535 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)c3ccccc3N BTB06534 CCOC(=O)c1c(n(c2c1cc(cc2)OC)C3CC3)C RH01103 Cc1cc(n(n1)c2ccc(cc2)[N+](=O)[O-])OC(=O)c3c(nn(n3)c4ccccc4)C BTB06553 c1cc(c(cc1[N+](=O)[O-])C2SCCS2)Oc3nc4cc(ccc4s3)Cl BTB06558 COc1ccc(c(c1C(=O)NCCCn2ccnc2)OC)[N+](=O)[O-] BTB04844 c1cc(oc1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F AW00242 c1cc(ccc1NC(=O)/C=C/C(=O)O)Oc2ccc(cc2)OC(F)(F)F AW00243 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc(cc2)OC(F)(F)F NRB00185 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)c3ccccc3 BTB06539 c1ccc(cc1)n2ncc(n2)C(=O)NNC(=O)c3ccc(c(c3)Cl)Cl BTB06541 CC(=O)c1cc(c(s1)NC(=O)C)C(=O)[O-].[Na+] NRB01125 Cc1cc(n(c(=O)c1C#N)CCO)O NRB01130 Cc1ccc2c(c1)CCCN2C(=S)Nc3cccc(c3)C(F)(F)F BTB01016 c1ccc2c(c1)CCN(C2)C(=S)Nc3cccc(c3)C(F)(F)F BTB01017 c1ccc2c(c1)CCN(C2)C(=S)Nc3ccccc3Cl BTB01021 Cc1ccc2c(c1)CCCN2C(=S)Nc3cccc(c3)Cl BTB01024 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)Cl)Oc3ccc(cc3Cl)Cl BTB04863 CC(c1cccc(c1)[N+](=O)[O-])(SCC(=O)O)SCC(=O)O BTB00982 Cc1cc(c(cc1C)[N+](=O)[O-])NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C BTB04832 c1cc(c(c(c1)Cl)C(=O)NC(=O)Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl BTB04838 Cc1cc(c(cc1C)[N+](=O)[O-])NS(=O)(=O)c2ccc(c(c2)Cl)Cl BTB04841 c1cc(c(c(c1)Cl)C(=O)NC(=O)Oc2ccc(cc2)C(F)(F)F)Cl BTB04846 c1cc(c(c(c1)Cl)C(=O)NC(=O)Oc2ccc(cc2Cl)F)Cl BTB04847 CC(=O)Oc1cc(ccc1[N+](=O)[O-])Sc2ccc(cc2)Cl BTB06536 c1cc(ccc1Sc2ccc(c(c2)OCC#N)[N+](=O)[O-])Cl BTB06537 Cc1c(nn(n1)c2ccccc2)c3nnc(o3)c4ccccc4 BTB06548 c1cc(ccc1C2=Nn3c(nnc3SC2)c4cc(cc(c4)Cl)Cl)Br.Br RH01108 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccccc3Oc4ccc(cc4Cl)Cl BTB04853 Cc1cc(c(cc1C)[N+](=O)[O-])NS(=O)(=O)c2ccc(c(c2)OC)OC BTB04856 c1ccc(c(c1)NC(=O)c2cccs2)Oc3ccc(cc3Cl)Cl BTB04857 c1ccc(c(c1)NC(=O)CC#N)F BTB06552 c1cc(ccc1NC(=O)c2ccc(c(c2)Cl)Cl)Oc3ccc(cc3)OC(F)(F)F AW00247 Cc1c(c(n(n1)c2ccccc2)O)C(=O)c3c(nn(n3)c4ccccc4)C BTB06543 c1ccc2c(c1)c(=O)c3cccnc3o2 BTB03140 C(CCC(=O)NCC(=O)O)CC(=O)NCC(=O)O RH01099 c1ccc(c(c1)NC(=O)c2c(cccc2F)F)Oc3ccc(cc3Cl)Cl BTB04859 COc1ccc(c(c1C(=O)Nc2ccc(cc2F)F)OC)[N+](=O)[O-] BTB04843 COc1c(c(c(c(=O)[nH]1)C#N)c2ccc(cc2)Cl)C#N BTB03160 CC(=O)c1c(c(c(c(=O)[nH]1)C#N)c2ccc(cc2)OC)C#N BTB03161 C#CC1(CCCCC1)NC(=O)c2cc(cc(c2)Cl)Cl BTB03174 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F)F AW00244 c1cc(oc1)CSCC(=O)Nc2c(c(c(c(c2F)F)F)F)F NRB00186 Cc1ccc(cc1)C2=Nn3c(nnc3SC2)c4cc(cc(c4)Cl)Cl.Br RH01111 Cc1c(nn(n1)c2ccccc2)c3nnc(o3)c4ccc(c(c4)Cl)Cl BTB06550 Cc1c2cc(c(cc2cc(n1)OCc3c(cccc3Cl)F)OC)OC RH01114 COc1ccccc1c2nnc(n2c3ccccc3)Sc4c(cccn4)[N+](=O)[O-] RH01119 c1ccc(cc1)Oc2c(cccn2)C(=O)N BTB03139 CCOC(=O)/C(=C/c1cc(c(c(c1)OC)OC)OC)/C#N BTB03155 Cc1cc(cc(c1S(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-])[N+](=O)[O-] BTB03156 c1cc(ccc1NC(=O)C2CC2)Oc3ccc(cc3)OC(F)(F)F AW00241 CC(C)(C)c1ccc(cc1)CSCC(=O)Nc2ccccc2C#N NRB00182 Cc1ccc(cc1NC(=O)CSc2ccccn2)F NRB00183 Cc1ccc(cc1NC(=O)CSc2nccn2C)F NRB00184 Cc1cc(=O)cc(n1NC(=O)c2ccc(cc2)OC)C BTB03176 Cc1cc(=O)cc(n1NC(=O)c2cccnc2)C BTB03177 Cc1cc(c2c(c1)c(=O)oc(n2)c3ccc(cc3)C(C)(C)C)C NRB00192 CCOC(=O)N/N=C/c1cc(ccc1O)Cl ML00286 c1ccc(c(c1)NC(=O)c2ccc(cc2)F)Oc3ccc(cc3Cl)Cl BTB04850 CCOC(=S)SCc1ccc(cc1)C(=O)Oc2ccc(cc2Cl)F BTB04851 c1cc(ccc1C(=O)CNc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl BTB03170 c1cc(c(c(c1)Cl)/C=N/NC(=S)NC2CC3CC2C=C3)Cl ML00281 c1ccnc(c1)SCC(=O)Nc2ccc(cc2)OC(F)(F)F NRB00181 CCOC(=S)SCc1ccc(cc1)C(=O)Oc2ccc(cc2F)F BTB04852 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccccc3Oc4ccc(cc4Cl)Cl BTB04855 COc1ccc(cc1OC)S(=O)(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl BTB04862 c1ccc(cc1)Oc2c(cccn2)C#N BTB03141 c1ccc(cc1)S(=O)(=O)c2ccc(c(c2)OS(=O)(=O)c3ccc(cc3F)F)[N+](=O)[O-] BTB06579 c1cc(cc(c1)Sc2c(cccn2)C(=O)Nc3ccc(c(c3)Cl)Cl)C(F)(F)F BTB06581 c1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4ccc(c(c4)Cl)F RH01139 Cc1ccc(cc1)C(C)(SCC(=O)O)SCC(=O)O BTB00980 CCCC(C)(SCC(=O)O)SCC(=O)O BTB00992 CCCCCCC(C)(SCC(=O)O)SCC(=O)O BTB00996 Cc1c(c(no1)c2ccccc2)C(=O)NC(=S)Nc3ccc(cc3)Cl BTB01010 Cc1ccc2c(c1)CCCN2C(=S)Nc3c(cccc3C)C BTB01012 Cc1cccc2c1N(CCC2)C(=S)Nc3cccc(c3)C(F)(F)F BTB01018 CCCc1cc(nc(n1)SCC(=O)Nc2ccc(c(c2)Cl)F)O BTB06514 CCOC(=O)c1ccc(cc1)NC(=S)NC(C)(C)CO BTB00948 Cc1c(c(ccc1C(c2ccc(cc2)N(C)C)c3ccc(cc3)N(C)C)OC)C NRB01148 Cn1c2ccccc2c(=O)s1 BTB03211 c1cc(cc(c1)Cl)Sc2c(cccn2)C(=O)Nc3ccc(cc3Cl)Cl BTB06569 c1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)Oc3ccc(cc3Cl)Cl BTB04860 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl BTB04861 COc1ccc(cc1[N+](=O)[O-])C(F)(F)F BTB03145 COc1ccccc1c2nnc(n2c3ccccc3)Sc4c(ccs4)[N+](=O)[O-] RH01120 Cc1c2cc(c(cc2cc(n1)OC(=O)c3ccc(cc3)[N+](=O)[O-])OC)OC RH01123 c1cc(ccc1NC(=O)CSc2ccc(cn2)C(F)(F)F)OC(F)(F)F NRB00187 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F)O AW00248 CCN(CC)c1ccc(cc1)/N=N/c2c(cc(cc2Cl)C#N)Cl NRB01158 c1cc(ncc1)/C=N/NC(=O)N/N=C/c2ncccc2 ML00307 CNC(=S)N/N=C/c1cc(ccc1O)Br ML00311 CNC(=S)N/N=C/c1cccc2c1cccc2 ML00312 CNC(=S)N/N=C/c1ccc2c(c1)OCO2 ML00310 c1ccc(cc1)C(=O)CSC2=NCCCCC2.Br ML00319 CCOC(=O)C(Cc1ccc(cc1)F)(C(=O)OCC)NC(=O)C RH01127 CCN1c2cc(c(cc2C(CC1(C)C)C)N=Nc3ccc(cc3)[N+](=O)[O-])NC(=O)C NRB01150 Cc1cc(c2c(c1)c(=O)oc(n2)c3ccc(cc3)C(F)(F)F)C NRB00188 c1ccc2c(c1)CCCN2C(=S)Nc3cccc(c3)C(F)(F)F BTB01019 CCN(CC)c1ccc(cc1)N=Nc2ccc3c(c2)OCCO3 NRB01155 COc1cc(c(cc1Cl)OC)/N=C/c2cccs2 BTB00979 Cc1c2cc(c(cc2cc(n1)OS(=O)(=O)c3ccc(cc3)C(C)C)OC)OC RH01129 Cc1ccc(cc1)S(=O)(=O)Oc2cc3cc(c(cc3c(n2)C)OC)OC RH01135 Cc1ccc(cc1S(=O)(=O)Oc2cc3cc(c(cc3c(n2)C)OC)OC)[N+](=O)[O-] RH01136 c1ccc2c(c1)CCCN2C(=S)Nc3ccccc3Cl BTB01023 CCOC(=O)c1cc(ccc1C#N)OC BTB03181 c1ccc(c(c1)C(=O)Nc2cc(ccc2Cl)C(F)(F)F)C(=O)O BTB03213 c1c(cc(cc1C(F)(F)F)NC(=O)CCC(=O)O)C(F)(F)F BTB03214 C#CC1(CCCCC1)NC(=O)c2ccccc2C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB03219 C1CCC(CC1)NC(=NC#N)NC2CCCCC2 NRB01171 c1ccc(cc1)S(=O)(=O)c2ccc(c(c2)OS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] BTB06576 Cc1cccc2c1N(CCC2)C(=S)Nc3ccccc3Cl BTB01022 CNC(=S)N/N=C/c1cccc(c1)[N+](=O)[O-] ML00314 CNC(=S)N/N=C/c1ccc(c(c1)OC)OC ML00315 c1c(cc(c(c1)O)/C=N/NC(=O)N/N=C/c2c(ccc(c2)Cl)O)Cl ML00285 c1cc(c(cc1/C=N/NC(=S)NC2CC3CC2C=C3)Cl)Cl ML00292 c1cc(ccc1NC(=O)CSCC(=O)O)Oc2ccc(cc2)OC(F)(F)F AW00252 Cc1cc(c(cc1OC)C)C(c2ccc(cc2)N(C)C)c3ccc(cc3)N(C)C NRB01149 c1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4ccco4 RH01141 c1ccc-2c(c1)Cc3c2nc(s3)NC(=O)c4ccco4 RH01142 CC(C)CC(C)(SCC(=O)O)SCC(=O)O BTB00999 c1cncc(c1)/C=N/NC(=O)N/N=C/c2cnccc2 ML00301 Cc1ccc(cc1)/C(=N/NC(=O)N/N=C(/c2ccc(cc2)C)\C)/C ML00302 Cc1ccc(cc1)S(=O)(=O)Oc2cc(ccc2[N+](=O)[O-])S(=O)(=O)c3ccccc3 BTB06578 Cc1ccc(cc1)NC(=O)c2cccnc2Sc3cccc(c3)C(F)(F)F BTB06582 COCCCNC(=O)c1ccccc1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB03222 CCC(C)NC(=O)c1c(ccc(c1OC)[N+](=O)[O-])OC BTB03230 CNC(=S)N/N=C/c1cc(cc(c1O)Br)Br ML00317 C1CCC(CC1)(SCC(=O)O)SCC(=O)O BTB00990 CCN(CC)c1ccc(cc1)N=Nc2c(cc(cc2Cl)C(F)(F)F)Cl NRB01159 CCN(CC)c1ccc(cc1)N=Nc2c(cc(cc2Br)C(F)(F)F)Br NRB01160 CN(C)c1ccc(cc1)C(c2ccc(cc2)N(C)C)c3ccc(cc3)OC(F)(F)F NRB01162 c1cc(cc(c1)Cl)NC(=O)CC#N BTB06560 c1ccc(cc1)Oc2c(cccn2)C(=O)Sc3ccc(cc3)Cl BTB03056 CSc1cccc(c1)NC(=O)CSc2ccccn2 NRB00162 c1c(c(n(n1)CCC#N)N)C#N BTB03241 c1cc(cc(c1)Sc2c(cccn2)C(=O)Nc3ccc(cc3Cl)Cl)C(F)(F)F BTB06583 c1ccc(cc1)S(=O)(=O)c2ccc(c(c2)OC(=O)c3ccc(cc3)Cl)[N+](=O)[O-] BTB06584 c1cc2c(cc1F)C(C(=O)N2)(Cc3ccncc3)O RH01076 C1CCCC(CC1)(SCC(=O)O)SCC(=O)O BTB00991 c1cc(ccc1C(=O)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F)C(F)(F)F AW00240 CCCc1cc(nc(n1)SCC(=O)Nc2cc(cc(c2)Cl)Cl)O BTB06519 c1ccc(c(c1)C(=O)NC2CCCCNC2=O)NC(=O)c3cccs3 BTB06524 CNc1ccccc1C(=O)NNC(=O)c2cccnc2Oc3ccccc3 BTB03109 c1ccc(c(c1)/C=N/NC(=S)NC2CC3CCC2C3)Cl ML00264 c1cc(c(cc1Br)/C=N/NC(=S)NC2CC3CCC2C3)O ML00267 COc1cc(cc(c1OC)OC)/C=N/NC(=S)NC2CC3CCC2C3 ML00268 Cc1ccc(cc1)n2nc(nn2)c3cc(c(c(c3)OC)OC)OC BTB03115 Cc1cccc(c1)C(=O)O/N=C(\C)/COc2ccc(cc2Cl)Cl BTB03116 c1cc(c(c(c1)F)NC(=O)CN2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)F AW00211 CCOC(=O)/C=C(/Nc1c(c(ccc1)N/C(=C/C(=O)OCC)/C)C)\C RH01034 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=S)Nc3ccc(c(c3)Cl)Cl BTB03066 Cc1cc(ccc1Br)NC(=S)NNC(=O)c2cccnc2Oc3ccccc3 BTB03067 Cc1cc(c(cc1C)[N+](=O)[O-])NC(=O)c2cccs2 BTB04824 CC(C(OC)OC)NC(=O)NC(=O)c1ccccc1Cl BTB04828 COc1c(c(cc(c1)/C=N/CCCC/N=C/c2cc(c(c(c2)OC)OC)OC)OC)OC BTB00950 Cc1c2cc(cc(c2oc1C(=O)c3ccc(cc3)Cl)Cl)Cl BTB03100 COc1ccc2c(c1)sc(n2)N BTB04799 CCOC(=O)C(=CNc1nc2ccc(cc2s1)C)C(=O)OCC BTB04802 CCOC(=O)c1cc(ccc1NC(=O)c2ccc(cc2)Cl)C BTB00919 CCOC(=O)CSc1nnc(n1c2ccccc2)c3ccccc3OC RH01079 CC1C(=Nn2c(nnc2S1)c3cccs3)c4ccc(cc4)CC(C)C.Br RH01059 CCOC(=O)c1c(n(c2c1cc(cc2)OC(=O)c3ccc(cc3)C)c4ccccc4)C RH01060 CCOC(=O)/C(=C/Nc1nc2ccc(cc2s1)C)/C#N BTB04812 CCOC(=O)c1c(n(c2c1cc(cc2)OC(=O)C(c3ccccc3)C4CCCC4)c5ccccc5)C RH01062 c1ccc(cc1)COc2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl BTB06468 Cc1cc(c(cc1Cl)C)S(=O)(=O)Oc2ccc(cc2)OCc3ccccc3 BTB06469 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)OCc3ccccc3 BTB06470 c1ccc(cc1)COc2ccc(cc2)OS(=O)(=O)c3cc(cc(c3)Cl)Cl BTB06471 CC(c1ccccc1)(SCC(=O)O)SCC(=O)O BTB00969 CC(C(OC)OC)NC(=O)NC(=O)c1c(cccc1F)F BTB04826 Cc1cc(c(cc1C)[N+](=O)[O-])NC(=O)c2ccc(cc2)F BTB04831 c1ccc(cc1)CN2CCc3c(c4cc(ccc4[nH]3)F)C2.Cl RH01104 c1ccc2c(c1)C(C(=O)N2)(Cc3ccccn3)O RH01084 c1ccnc(c1)CC2(c3cc(ccc3NC2=O)Br)O RH01086 c1ccc(c(c1)C(=O)Nc2nccs2)Cl ML00251 c1cc(ccc1C(=O)Nc2nccs2)[N+](=O)[O-] ML00252 CCOC(=O)c1cc(ccc1NC(=O)c2cc(ccc2[N+](=O)[O-])C)C BTB00930 c1cc2c(cc1Cl)sc(n2)N BTB04800 CCOC(=O)C(=CNc1nc2ccc(cc2s1)F)C(=O)OCC BTB04801 CCOC(=O)c1cc(ccc1NC(=O)c2c(c3ccccc3s2)Cl)C BTB00931 CCOC(=O)c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)C BTB00932 C1CN(CCN1CCNC=C(C#N)C#N)C=C(C#N)C#N BTB03048 c1ccc(cc1)Oc2c(cccn2)c3nnc(n3c4ccc(c(c4)Cl)Cl)S BTB03070 Cc1cc(ccc1Br)n2c(nnc2S)c3cccnc3Oc4ccccc4 BTB03071 CCCCCC[n+]1ccccc1/C=C\c2cccs2.[I-] NRB00150 c1cc(ccc1CSCC(=O)Nc2ccc(cc2F)F)Cl NRB00151 CN(C)c1ccc(cc1)C(c2ccc(cc2)N(C)C)c3ccc(cc3Cl)Cl NRB01142 CN(C)c1ccc(cc1)C(c2ccc(cc2)N(C)C)c3ccc(c(c3)Cl)Cl NRB01143 Cc1cccc(c1)COc2cc3cc(c(cc3c(n2)C)OC)OC RH01110 c1ccc(cc1)Oc2c(cccn2)C(=O)Nn3c(=O)c4cc(ccc4nc3S)Cl BTB03122 c1ccn(c1)c2ccc(cc2C#N)N BTB03126 c1cc(cc(c1)Cl)C(=O)Nc2nccs2 ML00253 c1cc(ccc1C(=O)Nc2nccs2)Cl ML00254 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2nccs2 ML00257 CCOC(=O)N/N=C/c1cc(c(c(c1)OC)OC)OC ML00258 c1cc(ccc1F)S(=O)(=O)NN BTB00968 CC(=O)C(=CNC1CCCCNC1=O)C(=O)C BTB06522 COc1c(c(cc(c1)/C=N/NC(=O)N/N=C/c2cc(c(c(c2)OC)OC)OC)OC)OC ML00259 CCOC(=O)c1cc(ccc1/N=C/c2cc(cc(c2O)Cl)Cl)C BTB00920 Cc1ccc(c(c1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)[N+](=O)[O-] BTB00921 Cc1ccc(c(c1)c2nc3ccccc3c(=O)o2)[N+](=O)[O-] BTB00923 C/C=C/C=N/NC(=O)N/N=C/C=C/C ML00260 CCOC(=O)N/N=C/C=C/C ML00261 Cn1ccnc1SCC(=O)Nc2cc(ccc2OC)Cl NRB00153 CC1(CNc2ccccc2C(=O)N1)OC BTB03112 c1cc(ccc1NC(=S)Nc2ccc(c(c2)Cl)F)Oc3ccc(cc3)OC(F)(F)F AW00227 c1cc(cnc1)C(=O)CSc2nccc(n2)C(F)(F)F AW00230 CCOC(=O)NNC(=S)Nc1cccc(c1)OC ML00274 Cc1cccc(c1)NC(=S)NNC(=O)NNC(=S)Nc2cccc(c2)C ML00276 Cc1cccc(c1NC(=S)NNC(=O)NNC(=S)Nc2c(cccc2C)C)C ML00280 c1ccc2c(c1)c(=O)s[nH]2 BTB03127 c1ccc(cc1)Oc2c(cccn2)C(=O)Nn3c(=O)c4ccccc4nc3S BTB03123 CC(C)(C)SCC(=O)Nc1cc(ccc1Oc2ccc(cc2)C#N)C(F)(F)F BTB03124 Cc1ccccc1C(=O)Nc2nccs2 ML00255 CCOC(=O)N/N=C/c1ccc(c(c1)Br)OC ML00263 Cc1c(c(no1)c2ccccc2Cl)NC(=O)NNC(=S)NC(C)(C)C BTB03101 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)NN BTB03129 c1cc(ccc1NC(=S)Nc2cc(ccc2Cl)Cl)Oc3ccc(cc3)OC(F)(F)F AW00221 c1cc(c(cc1C2=Nn3c(nnc3SC2)c4cc(cc(c4)Cl)Cl)F)F.Br RH01117 COc1ccccc1c2nnc(n2c3ccccc3)SC RH01121 c1ccc2c(c1)cc(s2)C(=O)Nc3ccccc3C(=O)NC4CCCCNC4=O BTB06525 c1ccc(c(c1)C(=O)NC2CCCCNC2=O)NC(=O)c3cccc(c3)C(F)(F)F BTB06527 Cc1ccc(cc1)n2nc(nn2)c3ccc(c(c3)Cl)Cl BTB03114 c1cc(ccc1C#N)Oc2ccc(cc2NC(=O)c3ccc(cc3)F)C(F)(F)F BTB03118 c1cc(ccc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)Oc3ccc(cc3)OC(F)(F)F AW00226 c1cc(c(nc1)N2CCNC2=S)C(F)(F)F AW00231 c1cc(ccc1NC(=O)Nc2ccc(cc2F)F)Oc3ccc(cc3)OC(F)(F)F AW00233 CCCCc1ccc(cc1)NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F AW00235 Cc1c(c(c(c(c1C)C)CSCC(=O)Nc2cccc(c2)SC)C)C NRB00177 Cc1cc(ccc1n2cccc2)c3nnc(o3)C(F)(F)F RH01097 c1cc(sc1)c2nnc3n2N=C(CS3)CC(=O)O RH01098 Cc1nc2ccccc2c(=O)n1c3ccc(cc3F)F NRB00170 Cc1cc(cc(c1Sc2ccc(cc2)Cl)[N+](=O)[O-])[N+](=O)[O-] BTB03134 Cc1cc(ccc1Br)Nc2nnc(s2)c3cccnc3Oc4ccccc4 BTB03136 c1cc(ccc1NC(=S)NC2CCCCCCC2)Oc3ccc(cc3)OC(F)(F)F AW00223 c1ccc(c(c1)C(F)(F)F)NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F AW00225 Cc1nc2ccccc2c(=O)n1c3ccc(c(c3)Cl)F NRB00173 c1c(cc(cc1Cl)Br)Cl BTB03107 c1cc(c(cc1NC2=C(C(=O)C(=C(C2=O)Cl)Nc3ccc(c(c3)S(=O)(=O)[O-])N)Cl)S(=O)(=O)[O-])N.[Na+].[Na+] NRB01127 C1CCC(CC1)NC(=O)CC#N BTB06546 Cc1cc(n(c(=O)c1C#N)CCCOC)O NRB01131 c1cc2c(cc1Br)/C(=N\NC(=O)c3ccncc3)/C(=O)N2 ML00388 c1cnccc1C(=O)NNC(=S)NC2CCCCC2 ML00393 CCOC(=O)C(=CNNCCC#N)C(=O)OCC BTB03238 CC(=O)c1cc2cc(cc(c2oc1=O)Cl)Cl BTB01084 CCCCNC(=S)NNC(=O)c1ccncc1 ML00398 c1cc(ccc1CCc2nnc(n2c3ccc(cc3)F)S)O BTB01090 Cc1c(cccc1Cl)n2c(nnc2S)CCc3ccc(cc3)O BTB01091 c1cc(cc(c1)n2c(nnc2S)CCc3ccc(cc3)O)C(F)(F)F BTB01094 c1ccc(cc1)Cn2c(c(c3c(c2=O)cccn3)C#N)N RH01162 c1cc(ccc1CCC(=O)NNC(=S)Nc2ccc(cc2)F)O BTB01087 c1ccc(c(c1)NC(=O)NC(=O)c2c(cccc2Cl)F)Oc3ccc(cc3Cl)Cl BTB04878 CCCCCCCNC(=S)NNC(=O)c1ccncc1 ML00401 CCCCn1c(n[nH]c1=S)c2ccncc2 ML00402 c1cc(ccc1CCc2nnc(n2c3ccc(cc3)Cl)S)O BTB01093 c1cc(ccc1NC(=S)NNC(=O)c2ccncc2)S(=O)(=O)N3CCCCC3 ML00385 CC(C)NC(=O)N1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB03274 COc1ccc(cc1)NC(=S)NNC(=O)c2ccncc2 ML00374 Cc1cc(no1)C(=O)Nc2nc-3c(s2)CCc4c3ccc(c4)OC RH01158 C[C@H](C(=O)O)O[C@@H]1[C@H]([C@H](O[C@H]2[C@H]1OC(OC2)c3ccccc3)OCc4ccccc4)NC(=O)C RH01183 CCCCCCCn1c(n[nH]c1=S)c2ccncc2 ML00403 CCCCCCCCCC(=O)Nc1nc-2c(s1)Cc3c2cccc3 RH01165 COc1ccc(cc1OC2CCCC2)C3CC(=O)NN3 RH01187 c1cnccc1CN2CNC(=S)NC2 ML00419 c1ccc(cc1)CCN2CNC(=S)NC2 ML00422 CCOC(=O)N/N=C(\C)/c1cccc(c1)[N+](=O)[O-] ML00404 Cn1c2ccc(cc2c(=O)s1)S(=O)(=O)Oc3ccc(cc3Cl)Cl BTB03260 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNC(=O)c3cc(c(c(c3)OC)OC)OC BTB01095 Cc1c(c(no1)c2ccccc2)C(=O)NNC(=O)Nc3c(onc3c4ccccc4Cl)C BTB01101 c1cc(cc(c1)OC(C(F)F)(F)F)NC(=O)CSc2ccc(cc2)Br NRB00202 C/C(=N\OC(=O)Nc1ccccc1)/c2cc3cc(ccc3o2)[N+](=O)[O-] BTB03278 CCOC(=O)c1ccccc1NC(=O)CSc2ncccn2 RH01177 CN(C)/C=N/c1nc-2c(s1)CCc3c2cccc3 RH01179 c1cc(cc(c1)Cl)n2c(n[nH]c2=S)c3ccncc3 ML00387 CC1CC(CC(C1)(C)C)N2CNC(=S)NC2 ML00406 C1CC(OC1)CN2CNC(=S)NC2 ML00407 CN1CCCCC(C1=O)c2cccc(c2)OC RH01185 COc1ccc(cc1)NC(=S)NNC(=O)CSc2nnc(n2c3ccccc3)c4ccccc4OC RH01156 CC(C)(C)c1csc(n1)Nc2cccc(c2)SC BTB04902 Cc1cccc(c1)/N=C/2\NC(C(=C)S2)(C)C BTB04871 c1ccc(c(c1)C(=O)NC(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl)Cl BTB04873 CCCCCCCCC(=O)Nc1nc-2c(s1)Cc3c2cccc3 RH01172 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)CN3CCOCC3)Cl RH01131 CCOC(=O)CC1=Nn2c(nnc2SC1)c3cc(cc(c3)Cl)Cl RH01133 CC(=O)c1ccccc1NC(=O)CN2CCOCC2 RH01138 C=CCNC(=S)NNC(=O)c1ccncc1 ML00392 COc1cc(cc(c1OC)OC)C(=O)N/N=C/2\c3cc(ccc3NC2=O)Br ML00394 CN(C)/C=N/c1nc-2c(s1)CCc3c2ccc(c3)OC RH01180 CC(C)NC(=NC#N)NC(C)C NRB01188 COC(=O)Cc1c(nnn1c2ccc(cc2)Cl)C(=O)OC NRB01197 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2nccs2 NRB01199 COCc1c(nns1)C(=O)OC NRB01210 CS(=O)(=O)Nc1ccccc1Oc2ccc(cc2Cl)Cl BTB04865 c1ccn(c1)c2c(cnn2CCC#N)C#N BTB03242 CC(C)(C)NC(=S)Nc1ccc(c(c1)OC)OC BTB03246 c1cc(c(cc1Cl)Cl)NC(=O)CC#N BTB06601 c1ccc(cc1)CNC(=S)C(=O)Nc2ccc3c(c2)OCO3 NRB00195 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F AW00256 Cc1ccc2cccc(c2n1)OC(=O)c3cccnc3Oc4ccccc4 BTB03253 Cc1cc(cc(c1O)C)C=C2C(=O)NC(=S)NC2=O BTB03258 c1ccc(cc1)c2c3cc(ccc3[nH]c(=O)c2N4CCOCC4)Cl RH01134 c1ccc-2c(c1)Cc3c2nc(s3)NC(=O)c4ccc(c(c4)Cl)F RH01140 c1ccc(c(c1)NC=C(C#N)C#N)Oc2ccc(cc2Cl)Cl BTB04881 c1ccc2c(c1)cc(c(=O)o2)[N+](=O)[O-] BTB06587 CN(C)/C=C(\C#N)/C(=O)NC1CCCCC1 BTB06588 c1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4ccc(cc4)[N+](=O)[O-] RH01145 Cc1c(c2cc(ccc2n1C3CC3)OC)C(=O)ON4C(=O)CCC4=O RH01150 CC(C)(C)NC(=S)Nc1ccccc1[N+](=O)[O-] BTB03233 CN(C)/C=C(\C#N)/C(=O)Nc1ccccc1F BTB06589 CCOC(=O)/C=C(\C)/Nc1ccc(cc1)Cl BTB01150 Cc1ccc(c2c1nc(cc2O)C)Cl BTB01151 COc1cccc(c1)NC(=S)Nc2cccc(c2)OC ML00441 CC1(CC(=O)c2ccc(cc2O1)OCC(=O)Nc3ccccc3)C RH01211 c1cc(ccc1NC(=O)CSCc2ccc(cc2Cl)Cl)OC(F)(F)F NRB00200 c1ccc2c(c1)cc(n2CC(CNCc3ccc(cc3Cl)Cl)O)c4ccc(cc4)F AW00264 COc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCCC2 RH01125 Cc1ccc(cc1)CNC(=O)c2cccnc2Sc3cccc(c3)C(F)(F)F BTB06630 c1cc(ccc1NC(=O)CCC(=O)O)Oc2ccc(cc2)OC(F)(F)F AW00257 Cc1ccc(cc1NC(=O)C(=S)NCc2ccccc2)F NRB00197 COc1ccc(cc1OC)CCNCC(Cn2ccc3c2cccc3)O AW00265 CN(C)/C=C(\C#N)/C(=O)NCC=C BTB06593 CC(=O)Nc1cc2cc(ccc2oc1=O)[N+](=O)[O-] BTB03237 COc1ccccc1c2nnc(n2c3ccccc3)SCC(=O)NNC(=O)C(F)(F)F RH01148 CC(C)c1cc(c(cc1C(C)C)/N=C/c2cc(cc(c2O)Cl)Cl)C(C)C BTB01055 CS(=O)(=O)N1CCCc2c1cccc2 BTB01058 COc1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4cccs4 RH01196 c1ccc-2c(c1)Cc3c2nc(s3)NC(=O)c4cccc(c4)F RH01198 CNC(=S)N/N=C/c1ccccc1O ML00321 Cc1cccc(c1n2c(nnn2)SCc3cc(cc(c3)F)F)C AW00258 c1cc(cc(c1)Sc2c(cccn2)C(=O)NCc3ccc(cc3Cl)Cl)C(F)(F)F BTB06629 c1cc(ccc1SCC(=O)Nc2cc(c(cc2F)F)F)Br NRB00213 CC(C)(C)c1ccc(cc1)CSCC(=O)Nc2cc(c(cc2F)F)F NRB00214 COC(=O)c1c(c2ccccc2s1)O BTB04875 c1ccc(c(c1)NC(=O)NC(=O)c2c(cccc2Cl)Cl)Oc3ccc(cc3Cl)Cl BTB04876 Cc1ccc2cccc(c2n1)OC(=O)c3c(cccc3Cl)F BTB03262 c1ccc(c(c1)NC(=O)NC(=O)c2c(cccc2F)F)Oc3ccc(cc3Cl)Cl BTB04877 c1ccc(cc1)C(CC(=O)c2cccs2)C(=O)O RH01213 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2cc(ccc2O)Br BTB04928 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)Nc2ccccc2Cl ML00356 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F ML00367 CC(=O)c1cc2cc(ccc2oc1=O)Br BTB01061 c1ccc(cc1)S(=O)(=O)c2ccc(c(c2)OC(=O)c3ccc(c(c3)Cl)Cl)[N+](=O)[O-] BTB06585 CCOC(=O)C(=CNNc1ccnc2c1ccc(c2)Cl)C(=O)OCC BTB03195 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2cc(ccc2Cl)Cl AW00260 CNC(=S)N/N=C/c1c2ccccc2ccc1O ML00322 CNC(=S)N/N=C/c1ccc(cc1)Cl ML00323 CNC(=S)N/N=C/c1ccc(cc1)OC ML00325 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(cc1Cl)Cl BTB06614 Cc1cc(ccc1NC(=O)/C(=C/N(C)C)/C#N)Cl BTB06615 CNC(=O)/C(=C/N(C)C)/C#N BTB06616 Cc1nc2ccccc2c(=O)n1c3ccc(cc3C(F)(F)F)Br NRB00211 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)N/N=C\3/c4cc(ccc4NC3=O)Br.Br ML00448 c1ccc(cc1)c2ccc(cc2)c3csc(n3)N/N=C\4/c5cc(ccc5NC4=O)Br.Cl ML00449 CCOC(=O)N/N=C(\C)/c1ccc(cc1)OC ML00451 c1ccc(cc1)Cn2c3ccccc3c4c2CCCC4=O RH01202 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2cc(cc(c2O)Cl)F BTB04929 Cc1cc(ccc1NC(=O)CC#N)Cl BTB06605 CC(=O)Nc1cc2cc(ccc2oc1=O)N BTB03243 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCNCC2 BTB03244 c1cc(cc(c1)Cl)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F AW00255 c1cc(ccc1NC(=O)CSc2ccc(cc2)Br)OC(F)(F)F NRB00196 CC(C)(C)c1ccc(cc1)OS(=O)(=O)c2ccc3c(c2)c(=O)sn3C BTB03261 COc1ccc(cc1/C=C/C(=O)Nc2ccc(cc2F)F)Br NRB00209 c1ccc2c(c1)cc([nH]2)c3cccs3 AW00283 c1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4cccc(c4)F RH01128 C/C(=N\O)/c1cc2cc(ccc2o1)[N+](=O)[O-] BTB03264 C/C(=N\OS(=O)(=O)C)/c1cc2cc(ccc2o1)[N+](=O)[O-] BTB03267 c1cc(cc(c1)Sc2c(cccn2)C(=O)NCc3ccc(c(c3)Cl)Cl)C(F)(F)F BTB06628 c1cc(c(c(c1)Cl)C(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl BTB03273 c1ccnc(c1)CNC(=O)CC#N BTB06613 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(cc1OC)OC BTB06617 c1cc2c(cc[nH]2)c(c1)[N+](=O)[O-] RH01152 Cc1cc(c2c(n1)ccc3c2[nH]nc3)O RH01155 CC1(C(=C)S/C(=N/c2cccc(c2)Cl)/N1)C BTB04869 Cc1c(cccc1Cl)Nc2nc(cs2)C(C)(C)C BTB04901 CCCNC(=O)O/N=C(\C)/c1cc2cc(ccc2o1)[N+](=O)[O-] BTB03280 c1cc(ccc1C(C#N)N2CCOCC2)Cl BTB03301 c1c(cnc(c1[N+](=O)[O-])N)Br BTB03307 c1ccc(cc1)CNc2nnc(s2)c3ccccc3 NRB01179 c1ccc-2c(c1)Cc3c2nc(s3)NC(=O)c4ccc(cc4)[N+](=O)[O-] RH01151 CCCCCCCC(=O)Nc1nc-2c(s1)CCc3c2ccc(c3)OC RH01173 c1ccc(c(c1)C(=O)NC(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl)F BTB04879 c1cc(c(cc1Cl)Cl)CSCC(=O)Nc2cc(c(cc2F)F)F NRB00215 COc1cc(cc(c1OC)OC)C(C#N)N2CCOCC2 BTB03302 c1ccc(c(c1)NS(=O)(=O)c2ccc(c(c2)Cl)Cl)Oc3ccc(cc3Cl)Cl BTB04864 CCN(Cc1ccc(cc1)CN(CC)C(=S)Nc2cccc(c2)C(F)(F)F)C(=S)Nc3cccc(c3)C(F)(F)F BTB01141 c1cc(ncc1Br)N BTB03304 c1ccc(cc1)c2c(n(nn2)c3ccc(cc3)Br)N NRB01228 Cc1cc2c(cc1N=Nc3ccc(cc3)C(=O)C)C(CC(N2CCO)(C)C)C NRB01151 CCN(CC)c1ccc(cc1)N=Nc2ccc(c(c2)C(F)(F)F)C#N NRB01157 c1cc(ccc1NC(=O)CC#N)[N+](=O)[O-] BTB06565 COC(COc1cc(ccc1[N+](=O)[O-])Sc2ccc(cc2)Cl)OC BTB06563 CN(C)c1ccc(cc1)C(c2ccc(cc2)N(C)C)c3ccc(cc3)OC(F)F NRB01164 CCOC(=O)C(=CNc1ccccc1Oc2ccc(cc2Cl)Cl)C(=O)OCC BTB04883 c1cc(cnc1)CN2CNC(=S)NC2 ML00408 c1ccnc(c1)CCN2CNC(=S)NC2 ML00418 COc1ccc(cc1OC)CCN2CNC(=S)NC2 ML00423 Cc1nc2ccccc2c(=O)n1c3cc(c(cc3F)F)F NRB00210 CN(C)/C=C(\C#N)/C(=O)Nc1cccc(c1)Cl BTB06590 CN(C)/C=C(\C#N)/C(=O)Nc1ccccc1 BTB06591 c1cc(cc(c1)NC(=S)NNC(=O)c2ccncc2)C(F)(F)F ML00378 CCOC(=O)/C(=C/Nc1ccccc1Oc2ccc(cc2Cl)Cl)/C#N BTB04882 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)Cl)/C(=O)O2 BTB04888 CC1=NN(C(=O)C1N=Nc2ccc(cc2)[N+](=O)[O-])c3ccccc3 NRB01167 Cc1ccc(cc1)NC(=O)c2cccnc2Sc3cccc(c3)Cl BTB06571 c1cc(ccc1C#N)Oc2ccc(cc2/N=C/c3cc(cc(c3O)Cl)Cl)C(F)(F)F BTB03119 CCOC(=O)NNC(=S)Nc1ccc(cc1)Cl ML00270 COc1ccccc1NC(=S)NNC(=O)NNC(=S)Nc2ccccc2OC ML00272 c1ccc(cc1)CN2C(=O)CSC2=S NRB01201 c1cc(oc1)CNC(=S)Nc2ccc(cc2)C3=NCCO3 AW00281 COc1ccc(cc1)C(=O)CSC2=NCCCC2.Br ML00351 c1cc(cc(c1)Cl)Sc2c(cccn2)C(=O)NCc3ccc(c(c3)Cl)Cl BTB06633 CCOC(=O)c1cn(nn1)c2ccc(cc2)Cl NRB01217 COC(=O)Cc1c(nnn1c2ccc(cc2)Br)C(=O)OC NRB01220 c1cc(ncc1C(F)(F)F)SCC(=O)Nc2cc(c(cc2F)F)F NRB00212 CCOC(=O)/C(=C/NCCc1ccc(cc1)Cl)/C#N BTB04889 Cc1cccc(c1)NC(=S)N RH01166 CCCCCCCCC(=O)Nc1nc-2c(s1)CCc3c2ccc(c3)OC RH01164 Cc1ccc(c(c1)C)Nc2nc(cs2)C(C)(C)C BTB04905 c1ccc(c(c1)C(=O)Nc2ccc(cc2)F)NC(=S)Nc3cccc(c3)C(F)(F)F BTB01043 c1ccc(c(c1)C(=O)Nc2ccc(cc2)F)NC(=S)Nc3ccccc3Cl BTB01045 CCOC(=O)N/N=C/1\c2cc(ccc2NC1=O)Br ML00273 c1cc(ccc1C#N)Oc2ccc(cc2NC(=O)C(F)(F)F)C(F)(F)F BTB03121 COc1ccccc1C(=O)NNC(=S)Nc2ccccc2 RH01069 c1ccnc(c1)CC2(c3cc(ccc3NC2=O)F)O RH01073 COc1ccc(cc1)NC(=S)NNC(=O)c2cc(c(c(c2)OC)OC)OC ML00365 Cc1ccc(c(c1)C)NC(=S)N2CCCc3c2c(ccc3)C BTB01029 c1cc(ccc1CCC(=O)N/N=C/c2ccc(c(c2)Cl)Cl)O BTB01033 COc1cc(cc(c1OC)OC)/C=N/NC(=O)CCc2ccc(cc2)O BTB01034 COc1cc(cc(c1OC)OC)c2nnc(n2c3cccc(c3)C(F)(F)F)SC(c4ccccc4)C(=O)c5ccc(cc5)Cl.Br ML00372 Cc1cccc(c1NC(=S)NNC(=O)c2ccncc2)C ML00375 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=O)CCc2ccc(cc2)O BTB01036 c1cc(cc(c1)NC(=S)N(Cc2ccc3c(c2)OCO3)c4ccc(cc4)F)C(F)(F)F BTB01038 c1ccc(c(c1)C(=O)Nc2ccc(cc2)F)NC(=S)Nc3ccc(c(c3)Cl)Cl BTB01048 CCCNC(=S)NNC(=O)c1ccncc1 ML00395 c1ccc2c(c1)CCN(C2)C(=S)Nc3cccc(c3)Cl BTB01025 Cc1ccc(c(c1)C)NC(=S)N2CCc3ccccc3C2 BTB01028 Cc1ccc(c(c1)C)NC(=S)N2CCCc3c2cccc3 BTB01030 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2nc3cc(ccc3s2)Cl)Cl BTB04820 COc1ccc2c(c1)nc(s2)NC(=O)NC(=O)c3c(cccc3Cl)Cl BTB04821 c1cc(ccc1CCC(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)O BTB00938 CCOC(=O)C(=CNc1nc2ccc(cc2s1)OC)C(=O)OCC BTB04803 CCOC(=O)C(=CNc1nc2ccc(cc2s1)Cl)C(=O)OCC BTB04804 CCCCCC(=O)Nc1nc-2c(s1)CCc3c2ccc(c3)OC RH01175 CC(=O)Nc1cc2ccccc2oc1=O BTB01088 CNC(=S)N/N=C/C=C/c1ccccc1 ML00331 COc1ccc(cc1)C(=O)CS/C/2=N/CCCCCC2.Br ML00349 c1ccc2c(c1)cc(c(=O)o2)C(=O)NCCc3ccc(cc3)Cl BTB04897 CC1(C(=C)S/C(=N\c2cc(cc(c2)OC)OC)/N1)C BTB04884 COC(=O)/C=C(/C(=O)OC)\Nc1ccccc1Oc2ccc(cc2Cl)Cl BTB04885 CN(C)/C=C(/c1ccccc1)\C(=S)c2ccccc2 NRB01274 COc1ccc(cc1)C(=S)/C=C\Nc2ccc(cc2)OC NRB01275 Cc1ccc(c(c1)Cl)NC(=S)NNC(=O)CCc2ccc(cc2)O BTB01053 CCOC(=O)/C(=C/Nc1nc2c(cccc2s1)OC)/C#N BTB04810 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2nc3cc(ccc3s2)F)Cl BTB04822 COc1ccc(cc1OC)/C=N/NC(=S)NC2CC3CCC2C3 ML00265 CCOC(=O)c1cc(ccc1NC(=S)Nc2cccc(c2)Cl)C BTB00928 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSC2=NCCCC2.Br ML00350 Cc1ccccc1NC(=S)Nc2ccccc2C(=O)Nc3ccc(cc3)F BTB01046 c1cc(ccc1CCNC=C(C#N)C#N)Cl BTB04890 c1ccc(cc1)n2c(n[nH]c2=O)CSc3ccc(cc3)Cl NRB00216 CNC(=S)N/N=C/c1cc(c(c(c1)OC)OC)OC ML00334 Cc1cc(no1)C(=O)Nc2nc-3c(s2)Cc4c3cccc4 RH01206 CCOC(=O)c1cc(ccc1NC(=S)Nc2ccc(cc2C)Cl)C BTB00933 CCOC(=O)c1cc(ccc1NC(=S)Nc2cc(ccc2Cl)Cl)C BTB00934 c1cc(ccc1CCC(=O)NN)O BTB00937 COc1ccc-2c(c1)CCc3c2nc(s3)N/C=N/O RH01189 Cc1ccc(c(c1)Cl)NC(=S)Nc2ccccc2C(=O)Nc3ccc(cc3)F BTB01047 c1cc(cc(c1)NC(=S)NNC(=O)CCc2ccc(cc2)O)C(F)(F)F BTB01049 c1ccc(c(c1)C(F)(F)F)Nc2nnc(s2)c3ccc(cc3)NC(=O)c4cccs4 RH01194 c1ccc-2c(c1)Cc3c2nc(s3)NC(=O)c4cccs4 RH01195 Cc1cccc(c1NC(=S)NNC(=O)CCc2ccc(cc2)O)C BTB01050 c1ccc(c(c1)NC(=S)NNC(=O)CCc2ccc(cc2)O)Cl BTB01051 CC(=O)Nc1cc2cc(ccc2oc1=O)NC(=O)C(F)(F)F BTB04925 CC(=O)Nc1nc-2c(s1)CCc3c2ccc(c3)OC RH01203 CS(=O)(=O)N(Cc1ccccc1)Cc2ccc3c(c2)OCO3 BTB01067 C=CCn1c(n[nH]c1=S)c2ccncc2 ML00397 c1ccc-2c(c1)CCc3c2nc(s3)N/C=N/O RH01190 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc4cc(ccc4oc3=O)[N+](=O)[O-] BTB04916 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3c(cc(cc3Cl)F)C(=O)C BTB04934 CN(c1ccc(cc1)/C=N/CCC/N=C/c2ccc(cc2)N(C)C)C BTB01085 c1c(cc(c(c1)Cl)Cl)/C=N/CCC/N=C/c2cc(c(cc2)Cl)Cl BTB01086 CC(=O)Nc1cc2cc(ccc2oc1=O)N/C(=C\C(=O)OC)/C(=O)OC BTB04920 CC(=O)Nc1cc2cc(ccc2oc1=O)NC(=O)C(Cl)(Cl)Cl BTB04921 CCOc1c(cc(cc1Br)Br)/C=C/2\C(=O)NC(=S)S2 BTB04946 c1cc(cc(c1)C#N)CSc2[nH]c3ccc(cc3n2)C(F)(F)F.Br BTB04953 Cc1ccc(c(c1)C)n2c(nnc2S)CCc3ccc(cc3)O BTB01092 COc1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4ccc(cc4)[N+](=O)[O-] RH01204 Cc1cc(ccc1NC(=O)CCC(=O)O)F RH01205 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2cc(cc(c2O)Cl)Cl BTB04927 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2F)F BTB04957 Cc1ccc(cc1Cl)/N=c\2/n(c(cs2)C(C)(C)C)c3ccc(c(c3)Cl)C BTB04958 C/C(=C(/C#N)\C(=O)Nc1ccc(cc1F)F)/N(C)C BTB06649 c1ccn(c1)c2ccc(cn2)C#N BTB03310 Cc1c(nn(n1)c2ccccc2)C(=O)O CC16201 Cc1cc(ccc1Cl)Oc2ccnc3c2ccc(c3)Cl BTB04979 c1cc(c(cc1F)F)CNC(=O)CC#N BTB06676 CN(C)/C=C(\C#N)/C(=O)NCc1ccc(cc1F)F BTB06682 CCOC(=O)c1csc(n1)NC(=O)CN2CCCCC2 RH01242 c1ccc(cc1)c2ccc(cc2)C(CCN3CCCCC3)O BTB03321 CC(C)(C)c1cs/c(=N/c2ccccn2)/n1c3ccc(cc3Cl)Cl BTB04973 CN(C)/C=N/c1nnc(s1)C(F)(F)F BTB04984 Cc1ccc(cc1/N=C/c2ccc(cc2)N(C)C)NS(=O)(=O)C BTB01180 Cc1ccc(cc1NC(=S)Nc2cccc(c2)Cl)NS(=O)(=O)C BTB01183 C/C(=N/NCCC#N)/C(=N\OC(=O)c1ccc(cc1)[N+](=O)[O-])/C(=O)Nc2ccccc2 BTB03344 Cc1cc(cc(c1Cl)C)Oc2ccnc3c2ccc(c3)Cl BTB04962 C1CCC(C1)(CC(=O)O)C(=O)O AW00301 Cc1nc2ccccc2c(=O)n1c3ccc(cc3)C(C)(C)C NRB00223 Cc1ccc(cc1C)/N=c\2/n(c(cs2)C(C)(C)C)c3ccc(c(c3)C)C BTB04964 CC(C)(C)c1ccc(cc1)n\2c(cs/c2=N/c3ccccn3)C(C)(C)C BTB04967 Cc1ccc(cc1C)n\2c(cs/c2=N/c3ccccn3)C(C)(C)C BTB04971 c1cc(c(cc1[N+](=O)[O-])Cl)/N=C/c2cc(cc(c2O)Cl)Cl BTB01167 c1cc(ccc1/C=N/NC(=S)Nc2cc(ccc2Cl)Cl)Oc3nccc(n3)C(F)(F)F AW00304 c1cc(ncc1C(F)(F)F)N2CCCN(CC2)C(=S)NC3CCCCCCC3 AW00293 c1cc(ncc1C(F)(F)F)N2CCCN(CC2)C(=S)Nc3cc(cc(c3)Cl)Cl AW00294 c1ccc(cc1)CNC(=S)C(=O)Nc2cc(c(cc2F)F)F NRB00218 Cc1c(c(c(cn1)CSc2[nH]c3ccc(cc3n2)C(F)(F)F)CO)O.Cl BTB04976 c1ccc(cc1)SCC(CN2CCN(CC2)c3nccc(n3)C(F)(F)F)O AW00308 c1cc2c(cc1N)S(=O)(=O)C=C2 MWP00044 c1ccc(cc1)COC(=O)Cc2csc3c2cc(cc3)Cl MWP00090 COC(=O)Cc1csc2c1cc(cc2)Cl MWP00091 c1cc(c(c(c1)F)C(=O)NC(=O)Nc2ccc(cc2F)Br)F BTB06672 CN(c1ccc(cc1F)F)C(=O)CSc2ccc(cc2)Cl BTB06688 c1cc(c(cc1Cl)Cl)OCc2csc3c2cc(cc3)Cl MWP00101 CCOC(=O)/C(=C(/C)\Nc1ccc(cc1)F)/C2CC(=O)N(C2=O)c3ccc(cc3)OC BTB01163 CC(C)(C)c1csc(n1)Cc2ccc(cc2)Cl.Br BTB05045 c1ccc(c(c1)NC(=S)N2CCN(CC2)c3nccc(n3)C(F)(F)F)N4CCOCC4 AW00305 CCOC(=O)CNC(=O)CSc1ccc(cc1)Cl NRB00226 c1cc(sc1)CN2CNC(=S)NC2 BTB03367 Cc1ccc(cc1/N=C/c2cc(ccc2O)Br)NS(=O)(=O)C BTB01179 Cc1nc2c(cc(cc2Br)Br)c(=O)n1Cc3cccs3 BTB03375 Cc1ccc(cc1[N+](=O)[O-])NS(=O)(=O)C BTB01159 CCOC(=O)/C(=C(/C)\Nc1ccc(cc1)F)/C2CC(=O)N(C2=O)c3ccc(cc3)F BTB01162 COC(=O)/C=C\1/C(=O)N(/C(=N/c2ccccn2)/S1)c3cccc(c3)SC BTB04994 Cc1ccc(cc1C)N\2C(=O)/C(=C/C(=O)OC)/S/C2=N\c3ccccn3 BTB04995 c1ccc2c(c1)c3ccccc3c4c2nc5nnc(n5n4)S RJC00047 Cc1c(c(no1)c2ccccc2)C(=O)On3c(=O)c4ccccc4nc3c5ccccc5 BTB05047 c1cc(c(c(c1)Cl)CSc2[nH]c3ccc(cc3n2)C(F)(F)F)Cl.Cl BTB04975 Cc1n[nH]c(=S)n1/N=C\c2cc(c(c(c2)OC)OC)OC RJC00021 c1cc(c(cc1C2(CSc3n2c4ccc(cc4n3)C(F)(F)F)O)Cl)Cl.Br BTB04980 c1ccc(cc1)C(=O)CNc2ccccc2C(=O)O BTB03377 c1ccnc(c1)NC(=S)Nc2ccccn2 RJC00024 c1ccc(cc1)N2C(=O)/C(=C\c3cccs3)/SC2=S RJC00026 CN(C)/C=N/c1nc2c(cccc2s1)OC BTB04989 CN(C)/C=N/c1nc2ccc(cc2s1)F BTB04988 COC(=O)/C=C\1/C(=O)N(/C(=N/c2ccccn2)/S1)c3ccc(cc3)Cl BTB04996 Cc1ccc(c(c1)C)NC(=S)NCCCOC BTB01196 Cc1ccccc1NC(=S)Nc2cc(ccc2C)NS(=O)(=O)C BTB01182 CCOC(=O)c1ccc(cc1)N2C(=O)CC(C2=O)/C(=C(\C)/N)/C(=O)OCC BTB01185 Cc1nc2ccc(cc2o1)NS(=O)(=O)c3ccccc3Cl MWP00040 CC1=NN(C(=O)C1)c2ccc(cc2)/N=C/c3ccc(c(c3)OC)O BTB01204 c1cc(ccc1C2(CSc3n2c4ccc(cc4n3)C(F)(F)F)O)Cl.Br BTB04978 COc1cc(cc(c1OC)OC)/C=N\n2cn[nH]c2=S RJC00018 Cc1ccc(cc1NS(=O)(=O)C)/N=C/c2cc(cc(c2O)Cl)Cl BTB01166 Cc1ccc(cc1NC(=S)Nc2cccc(c2C)Cl)NS(=O)(=O)C BTB01168 c1cc(ccc1C2NC(CS2)C(=O)O)Cl BTB04985 c1ccc(cc1)c2nnc(s2)N RJC00031 CSc1ccccc1NC=C(C#N)C#N BTB05003 Cc1ccc(cc1NC(=S)Nc2ccc(cc2)F)NS(=O)(=O)C BTB01171 Cc1ccc(cc1/N=C/c2ccccc2O)NS(=O)(=O)C BTB01173 c1ccc2c(c1)CCCN2c3nc(nc(n3)N4CCOCC4)N5CCCC5 BTB01188 Cc1c(cccc1Cl)NC(=S)NCCCOC BTB01193 Cc1ccccc1NC(=S)NCCCOC BTB01194 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)Cc4ccncc4)Cl BTB01219 CC1=NN(C(=O)C1)c2ccc(cc2)/N=C/c3ccc(c(c3)Cl)Cl BTB01205 Cc1cc(n(n1)c2ccc(cc2)NC(=O)c3cc(c(c(c3)OC)OC)OC)OC(=O)c4cc(c(c(c4)OC)OC)OC BTB01223 c1cnc(nc1)NC(=O)c2ccc(cc2)Cl BTB06689 CN(C)C(=O)Cc1c2ccccc2sc1Cl MWP00108 c1ccc(cc1)COC(=O)Cc2c3ccccc3sc2Cl MWP00109 COC(=O)c1c(nn[nH]1)C(=O)OC RJC00007 Cc1ccc(cc1NC(=S)Nc2cccc(c2)C(F)(F)F)NS(=O)(=O)C BTB01169 CC(C)(C)NCC(=O)Nc1cc(cc(c1)Cl)Cl BTB05001 c1c(cc(cc1Cl)Cl)NC(=O)CNC2CCCCC2 BTB05002 c1ccc2c(c1)C=CS2(=O)=O MWP00042 c1cc2c(cc1[N+](=O)[O-])S(=O)(=O)C=C2 MWP00043 CCOC(=O)/C(=C/Nc1ccccc1SC)/C#N BTB05004 Cc1cc(c2ccccc2n1)Oc3ccc(cc3)Cl BTB05006 CC(=O)c1ccc(cc1Cl)[N+](=O)[O-] MWP00070 c1ccc(c(c1)C(=O)NNC(=S)Nc2cccc(c2)Cl)Cl BTB01237 c1ccc(c(c1)C(=O)NNC(=S)Nc2cc(ccc2Cl)Cl)Cl BTB01241 Cc1c(nn(n1)c2ccccc2)C(=O)ONC(=O)c3ccccc3 BTB03353 Cc1ccc(cc1)Oc2cc(nc3c2cccc3)C BTB05016 Cc1ccc(cc1C)Oc2cc(nc3c2cccc3)C BTB05017 c1cc(c(c(c1)Cl)C(=O)NC(=O)NCc2cccs2)Cl BTB03351 c1ccc(c(c1)C(=O)NCc2cccs2)NC(=O)c3ccccc3Cl BTB03383 c1ccc(c(c1)c2nc(no2)c3cccc(c3)[N+](=O)[O-])N BTB03386 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl BTB03390 Cc1cccc(c1NC(=S)NCCCOC)C BTB01208 CCOC(=O)C1=C(N(C(=O)C1CC(=O)Nc2ccc(cc2)F)c3ccc(cc3)F)C BTB01215 CCOC(=O)C1=C(C(=O)N(C1C)c2ccc(cc2)F)CC(=O)Nc3ccc(cc3)OC BTB01216 c1cc2c(cc1Cl)c(cs2)CC(=O)O MWP00086 CCOC(=O)c1ccc(cc1)NC(=O)CC2C(=C(N(C2=O)c3ccc(cc3)F)C)C(=O)OCC BTB01217 CCOC(=O)c1ccc(cc1)NC(=O)CC2C(=C(NC2=O)C)C(=O)OCC BTB01218 CCOC(=O)C1=C(NC(=O)C1CC(=O)Nc2ccccc2)C BTB01227 Cc1cccc(c1NC(=S)NNC(=O)c2ccccc2Cl)C BTB01232 CCSC([C@H]([C@@H]([C@@H]([C@H](CO)O)O)O)O)SCC RJC00051 CCOC(=O)/C(=C(/C)\Nc1ccc(cc1)F)/C2CC(=O)N(C2=O)c3ccccc3 BTB01155 CN(C)/C=N/c1nc2ccc(cc2s1)Cl BTB04990 COC(=O)/C=C\1/C(=O)N(/C(=N/c2ccccn2)/S1)c3cccc(c3)C(F)(F)F BTB04993 Cc1ccc(cc1/N=C/c2cccs2)NS(=O)(=O)C BTB01175 Cc1ccc(cc1/N=C/c2ccc(c(c2)Cl)Cl)NS(=O)(=O)C BTB01177 c1cc(cc(c1)Cl)N2C(=O)/C(=C\c3cccs3)/SC2=S RJC00032 CC(=O)c1ccc(c(c1)COn2c(=O)c3ccccc3nc2c4ccccc4)OC BTB05018 CCOC(=O)/C(=C(/C)\N)/C1CC(=O)N(C1=O)c2ccccc2 BTB01186 c1ccc2c(c1)cc3ccccc3c2/C=C(\C#N)/c4ccc(cc4)[N+](=O)[O-] NRB01280 Cc1cc(ccc1Cl)Oc2cc(nc3c2cccc3)C BTB05005 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB03392 c1ccc2c(c1)cc(c(=O)o2)C(=O)O BTB01252 CCOC(=O)C(=CNc1c(cccc1Cl)F)C(=O)OCC BTB03350 COC(=O)C/C(=N\NC(=O)c1ccccc1N)/C(=O)OC BTB05012 Cc1ccc(cc1)COn2c(=O)c3ccccc3nc2c4ccccc4 BTB05013 Cn1c(nnn1)SCC(=O)Nc2ccccc2C#N NRB00230 Cc1c2ccccc2sc1COc3ccc(cc3Cl)Cl MWP00102 CNC(=O)Cc1c2ccccc2sc1Cl MWP00107 CC(=O)C(=CNc1c(cccc1Cl)F)C(=O)C BTB03352 c1ccc(c(c1)C(=O)NNC(=S)Nc2ccc(cc2)F)Cl BTB01235 COCCCNC(=S)Nc1ccc(cc1)Cl BTB01191 c1cc(ccc1C#N)OCc2c3cc(ccc3sc2Cl)Cl MWP00127 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccccc3Cl)Cl MWP00154 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc(cc3)Cl)Cl MWP00155 C([C@@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)NN=C(N)N)O)O)O)O.Cl RJC00041 c1cnc(nc1C(F)(F)F)N2CCN(CC2)C(=O)/C=C/C(=O)O AW00309 c1ccc(cc1)c2nc3ccccc3c(=O)n2OCc4c(cccc4Cl)Cl BTB05009 Cc1cccc(c1Oc2cc(nc3c2cccc3)C)C BTB05010 COCCCNC(=S)Nc1cccc(c1)Cl BTB01192 Cn1c(nnn1)SCC(=O)Nc2ccc(cc2)OC(F)(F)F NRB00231 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nnnn2C NRB00232 Cc1cc(ccc1Oc2cc(nc3c2cccc3)C)Cl BTB05015 COCCCNC(=S)Nc1ccc(cc1)F BTB01207 CC(C)CCCC(C)C1CCC2[C@@]1(CCC3C2CC=C4[C@@]3(CC[C@@H](C4)OC(=O)C)C)C BTB01201 COCCCNC(=S)Nc1ccccc1OC BTB01209 c1cc(ccc1N2C(=O)CC3(C2=O)CCCC3)OC(F)(F)F AW00313 Cc1c2ccccc2sc1CC(=S)N3CCOCC3 MWP00119 Cc1c2ccccc2sc1CC(=O)O MWP00120 Cc1cc(n(n1)c2ccc(cc2)NC(=O)c3c(c4ccccc4s3)Cl)OC(=O)c5c(c6ccccc6s5)Cl BTB01222 COC(=O)c1ccc(cc1NC(=O)c2ccc(cc2)F)Cl BTB05036 c1ccc(cc1)c2nc3ccccc3c(=O)n2OC(=O)c4cccc(c4)C(F)(F)F BTB05037 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3cc(ccc3C(=O)OC)Cl BTB05039 C([C@@H]([C@@H]([C@H]([C@@H](C(=O)NN)O)O)O)O)O RJC00044 COCCCn1c(=O)c2ccccc2[nH]c1=S BTB01195 CC1=NN(C(=O)C1)c2ccc(cc2)/N=C/c3ccc(cc3)N(C)C BTB01200 Cc1c2cc(ccc2sc1S(=O)(=O)Oc3ccccc3Cl)Cl MWP00160 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccccc3OC)Cl MWP00157 c1cc(ccc1Cc2ccncc2)N BTB01214 c1ccc(cc1)c2nc3ccccc3c(=O)n2OC(=O)c4ccccc4Cl BTB05024 c1ccc(c(c1)C(F)(F)F)NC(=S)Nc2ccc3c(c2)S(=O)(=O)C=C3 MWP00167 COc1cc2c(cc1OC)C3c4ccccc4NC(=O)CN3CC2 NRB01259 C=C1[C@H]([C@@H]([C@H]([C@@H](O1)OCc2ccccc2)OCc3ccccc3)OCc4ccccc4)OCc5ccccc5 RJC00043 CC(C)(C)c1csc(n1)Cc2ccc(cc2)OC.Br BTB05040 c1cc(sc1)CNC(=O)c2cc(ccc2N)Cl BTB03368 CNc1ccccc1C(=O)NCc2cccs2 BTB03370 CCOC(=O)CCc1cc(c(c(c1)/N=C/c2cc(c(cc2)Cl)Cl)O)/N=C/c3cc(c(cc3)Cl)Cl BTB01258 Cc1c(nc(s1)c2ccccc2)CC(=O)NN RH01226 Cc1c2cc(ccc2sc1S(=O)(=O)Oc3ccc(cc3)OC)Cl MWP00158 C1[C@@H]([C@@H]([C@H]([C@@H](O1)NNC(=S)N)O)O)O RJC00053 c1ccc(cc1)c2nc3ccccc3c(=O)n2OCc4cc(cc5c4OCOC5)Cl BTB05022 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)On3c(=O)c4ccccc4nc3c5ccccc5 BTB05025 c1ccc(cc1)c2nc3ccccc3c(=O)n2OC(=O)c4ccc(cc4)F BTB05032 c1cc(oc1c2nnc(o2)S)[N+](=O)[O-] RJC00001 c1ccc(c(c1)C(=O)NCCc2ccc(cc2)Cl)N BTB04891 c1cc(ccc1CCNC(=O)c2cc(ccc2N)Cl)Cl BTB04892 CCCCCCCCC(=O)Nc1nc-2c(s1)CCc3c2cccc3 RH01171 CCOC(=O)CCc1cc(c(c(c1)/N=C/c2c(ccc(c2)Br)O)O)/N=C/c3c(ccc(c3)Br)O BTB01259 c1cc(sc1)CNC(=O)c2cc(ccc2NC(=O)CSc3ccc(cc3)Cl)Cl BTB03381 CCOC(=O)c1csc(n1)NC(=O)CSc2cc(ccc2OC)OC RH01241 CCOc1ccc(cc1/C=C\2/C(=O)NC(=S)S2)Br BTB04949 COc1cc(cc(c1OC(=O)NC(=O)c2c(cccc2Cl)Cl)Br)C3SCCS3 BTB06691 Cc1c(nn(n1)c2ccccc2)C(=O)ONC(=O)c3ccco3 BTB03354 CCOC(CNC(=S)NC12CC3CC(C1)CC(C3)C2)OCC RJC00009 COc1ccc(cc1)/C=N/NC(=S)NN RJC00011 C(=C/C(=O)O)\C(=O)NNC(=N)N RJC00013 Cc1c2ccccc2sc1C(=O)C MWP00008 Cc1nc2ccc(cc2o1)NC(=O)C(Cl)Cl MWP00020 CCOC(=O)C(C(=O)OCC)NC(=O)c1c(nn(n1)c2ccccc2)C BTB06652 Cc1n[nH]c(=S)n1/N=C\c2ccco2 RJC00004 Cc1nc2ccc(cc2o1)NC(=O)c3ccccc3Cl MWP00028 c1cc(ccc1C/N=C/c2cc(cc(c2O)Cl)Cl)Cl BTB01083 CCOC(=O)/C(=C/Nc1ccc2c(c1)cc(c(=O)o2)NC(=O)C)/C#N BTB04914 CCOc1ccccc1/C=N/NC(=S)NC ML00326 CC(C)c1ccc(cc1)/C=N/NC(=S)NC ML00328 CNC(=S)N/N=C/c1ccc(c(c1)Br)OC ML00329 CC(C)(C)c1cs/c(=N\c2cccc(c2)C(F)(F)F)/n1c3cccc(c3)C(F)(F)F BTB04956 Cc1cc(c2cc(ccc2n1)F)O BTB01148 Cc1nc2ccc(cc2o1)NC(=O)Nc3ccccc3 MWP00022 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2cc(ccc2O)F BTB04930 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2cc(ccc2O)Cl BTB04931 c1ccc(cc1)NNC(=O)c2cc(ccc2NC(=O)c3cccnc3Oc4ccccc4)Cl BTB04932 c1ccc(cc1)S(=O)(=O)c2ccc(c(c2)Oc3ccc(cn3)[N+](=O)[O-])[N+](=O)[O-] BTB06638 Cc1cc(ccc1NC(=O)C)/N=N/c2cccc(c2)C(F)(F)F BTB06648 Cc1nc2ccc(cc2o1)NS(=O)(=O)c3ccc(c(c3)Cl)F MWP00038 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3C(=O)C)Cl BTB04933 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3C(=O)C)Br BTB04935 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cn3)Br BTB03311 COc1cc(cc(c1OC)OC)C2c3cc(c(cc3CCN2)OC)OC NRB01256 c1ccc(cc1)/C=C/C=N/NC(=O)CCc2ccc(cc2)O BTB01035 Cc1ccccc1NC(=S)N(Cc2ccc3c(c2)OCO3)c4ccc(cc4)F BTB01041 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl BTB03349 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc3c(c2)S(=O)(=O)C=C3)Cl MWP00045 Cc1cc(c2cc(ccc2n1)Cl)O BTB01152 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cn3)Br)Cl BTB03317 CC(C)(C)NC(=S)Nc1ccc(cc1[N+](=O)[O-])OC BTB03325 c1cc(c(cc1C(=O)Nc2nnc(s2)Sc3nc4cc(ccc4s3)Cl)Cl)Cl BTB06625 c1cc(cc(c1)Cl)Sc2c(cccn2)C(=O)NCc3ccc(cc3Cl)Cl BTB06632 COc1ccc(cc1)n2c(n[nH]c2=S)c3ccco3 ML00345 CC(C)(C)c1cs/c(=N/c2ccccn2)/n1c3ccc(cc3)Cl BTB04968 Cc1ccc(c(c1)C(C(=O)O)O)C BTB06663 CCOC(=O)N/N=C(\C)/c1ccc(cc1)C ML00452 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)c3csc(n3)C AW00295 COC(=O)C(C(C(=O)OC)N1CCOCC1)N2CCOCC2 NRB00220 COc1ccc(cc1OC)CC/N=C/c2ccc(cc2)Oc3nccc(n3)C(F)(F)F AW00298 c1cc(c2cc[nH]c2c1)C(=O)O CC28701 c1ccc(cc1)NC2=C(C(=O)N(C2=O)c3ccccc3)Cl RH01249 Cc1nc2ccc(cc2o1)NC(=O)NC MWP00023 c1ccc(cc1)CNC(=S)C(=O)Nc2cccc(c2)C(F)(F)F NRB00221 COc1ccc(cc1)n2c(nnc2SCc3ccc(cc3)C#N)c4ccco4.Br ML00347 CC(=O)Nc1cc2cc(ccc2oc1=O)NS(=O)(=O)c3ccc(cc3)Cl BTB03336 CCOC(=O)CCC(C#N)(c1cc(c(c(c1)OC)OC)OC)N2CCOCC2 BTB03337 CCOC(=O)c1csc(n1)NC(=O)CSc2cc(ccc2Cl)Cl RH01243 c1ccc(cc1)c2cc(=O)[nH]c(=O)[nH]2 RH01244 CC(C)(C)c1cs/c(=N/c2ccccn2)/n1c3cccc(c3)C(F)(F)F BTB04969 c1cc2c(cc1C(F)(F)F)nc([nH]2)S RH01250 CC(=O)/C(=N\O)/C(=O)Nc1ccccc1 BTB03338 CC(C)CC(C)N(c1ccc(cc1)OC)C(=S)Nc2cc(ccc2Cl)Cl BTB03341 c1ccc(c(c1)N)NC=C(C#N)C#N BTB03342 c1ccc(cc1)S(=O)(=O)C2CC2(Cl)Cl NRB01292 Cc1ccc(cc1)NC(=S)NNC(=O)Cc2c(sc(n2)c3ccccc3)C RH01254 CC(C)(C)c1cs/c(=N/c2ccccn2)/n1c3cccc(c3)SC BTB04970 c1cc2c(cc1Cl)c(cs2)CC#N MWP00085 Cc1cc(n(n1)c2ccc(cc2)S(=O)(=O)N)C BTB06658 c1ccc(cc1)Oc2ccc(cc2)C(=O)CCN3CCOCC3 BTB03314 CCC(=O)c1ccc(cc1)c2ccccc2 BTB03320 Cc1cc(ccc1Cl)C2(CSc3n2c4ccc(cc4n3)C(F)(F)F)O.Br BTB04977 CCCn1c(n[nH]c1=O)c2cccs2 NRB00219 c1cc(ccc1CC(=O)NCCNC(=S)Nc2ccc(cc2F)F)O AW00299 c1cc(c(cc1F)F)NC(=O)CSCc2ccc(cc2Cl)Cl NRB00222 c1ccc(cc1)c2ccc(cc2)c3csc(n3)c4ccc(cc4)Cl MWP00291 CC(=O)Nc1ccc(cc1F)F BTB03441 CC(=O)C(c1ccc(cc1C(=O)O)OC)C(=O)C BTB03450 c1ccc(cc1)c2ccc(cc2)c3csc(n3)c4ccncc4.Br MWP00293 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)O BTB06756 c1cc(ccc1C(=O)COC(=O)c2cc(cc(c2I)Cl)Cl)Br RJC00113 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3nnc(s3)C4CC4 BTB05060 c1cc(cc(c1)Br)C(=O)OCC(=O)c2ccc(cc2)Br RJC00109 c1cc(c(cc1C(=O)NCCc2ccncc2)Cl)Cl BTB03433 c1ccc(c(c1)N/C=N/O)Sc2nc3c(s2)cc(cc3Cl)Cl BTB06769 CN(C)/C=N/c1nnc(s1)SCC(=O)Nc2ccc(cc2F)F BTB06770 Cc1cc(ccc1NC(=O)CSc2nnc(s2)/N=C/N(C)C)Cl BTB06771 c1ccc(cc1)SCC(=O)NCc2cccs2 BTB03458 c1cc(sc1)CNC(=O)CSc2ccc(cc2)Cl BTB03460 CS(=O)(=O)NCCc1ccncc1 BTB03439 Cc1ccc(cc1)S(=O)(=O)NCCc2ccncc2 BTB03437 c1cnccc1CCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB03438 Cc1c2cc(ccc2sc1C(=O)CCSc3ccc(cc3)Cl)Cl MWP00282 c1cc(cc(c1)NC(=O)c2ccc(cc2)Cl)C(F)(F)F BTB01249 c1cnccc1CCNC=C(C#N)C#N BTB03430 COc1ccc(c(c1)C(=O)OCC(=O)c2ccc(cc2)Br)Br RJC00104 c1ccc(cc1)C(/C=C/C(c2ccccc2)c3ccccc3)c4ccccc4 NRB01345 CCN(CC)c1ccc(cc1)C#N NRB00242 c1ccc(cc1)C(COCC(c2ccccc2)(c3ccccc3)O)(c4ccccc4)O NRB01349 CN(C)/C=N/c1ccccc1Sc2nc3c(s2)cc(cc3Cl)Cl BTB06767 c1ccc(cc1)CN(C2CC3CCC2C3)C(=O)NC(=O)c4c(cccc4Cl)Cl BTB05080 c1ccc2c(c1)cc(c(=O)o2)C#N BTB01247 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)c2cccs2 AW00328 c1cc2c(cc1Br)cc(c(=O)o2)C(=O)O BTB01253 Cc1cc(ccc1Nc2nnc(s2)c3ccccc3Cl)Cl BTB01255 Cc1c2cc(ccc2sc1CC(=O)Oc3ccc(cc3)[N+](=O)[O-])Cl MWP00253 c1ccc(cc1)C(Cc2cccc(c2)[N+](=O)[O-])(C#N)c3ccccc3 NRB01334 c1cc(cc(c1)NC(=S)NN=C2CCCCCC2)C(F)(F)F BTB05122 c1cc(c(cc1C(F)(F)F)NC(=S)NN=C2CCCCCC2)Cl BTB05123 Cc1ccc(c(c1)C)NC(=S)NN=C2CCCCCC2 BTB05125 Cc1cc(c2cc(ccc2n1)Cl)OCc3c(cccc3Cl)Cl BTB01324 Cn1c(nnn1)SCC(=O)Nc2cccc(c2)SC NRB00233 c1ccc(cc1)Sc2ccccc2C(=O)OCC(=O)c3ccc(cc3)Br RJC00074 c1ccc2c(c1)cccc2Sc3ccccc3C(=O)OCC(=O)c4ccc(cc4)Br RJC00075 c1cc2cccc(c2c(c1)C(=O)OCC(=O)c3ccc(cc3)Br)I RJC00078 c1cnc(nc1)SCC(=O)Nc2ccc(cc2)OC(F)(F)F NRB00246 Cc1ccc(c(c1)C)NC(=S)NN=C(C)C BTB05103 c1cc(c(cc1F)F)NC(=O)CC#N BTB05104 c1cc(c(cc1NC(=O)CC#N)Cl)F BTB05106 Cc1ccc(cc1)CSc2nc(c3n2cccc3)C(=O)C(F)(F)F BTB05120 c1ccc(cc1)CC(C#N)(c2ccccc2)c3ccc(cc3)[N+](=O)[O-] NRB01335 c1ccc(c(c1)c2nc(no2)c3ccc(cc3)Cl)N BTB03385 c1ccc(c(c1)CC(=O)OCC(=O)c2ccc(cc2)Br)Br RJC00068 c1ccc(c(c1)CC(=O)OCC(=O)c2ccc(cc2)Br)I RJC00072 c1cc(ccc1Oc2ccnc3c2ccc(c3)Cl)F BTB05019 c1cc(ccc1Oc2ccnc3c2ccc(c3)Cl)Cl BTB05020 CC(C)(C)c1csc(n1)Cc2ccccc2Cl.Br BTB05044 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(ccc3C(=O)OC)Cl BTB05046 Cc1c(c(c(cn1)COn2c(=O)c3ccccc3nc2c4ccccc4)CO)O BTB05021 c1ccc(cc1)c2nc3ccccc3c(=O)n2OCc4ccc(cc4)Br BTB05023 Cc1c(cccc1Cl)NC(=S)NNC(=O)c2ccccc2Cl BTB01233 CC(C)c1cccc(c1OC(=O)NC(=O)c2c(cccc2F)F)C(C)C BTB05065 c1cc(ccc1OCOc2ccc(cc2)Cl)Cl BTB05077 COc1cc(cc(c1OC)OC)C(=O)Nc2ccc3c(c2)nn[nH]3 BTB01311 c1ccc(cc1)CNC(=O)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB00237 Cc1c2cc(ccc2sc1c3csc(n3)C)Cl MWP00222 c1cc(ccc1NC(=O)CSCc2ccc(c(c2)Cl)Cl)OC(F)(F)F NRB00238 COC(=O)c1ccc(cc1NC(=O)c2ccccc2Cl)Cl BTB05027 CC(=O)OC[C@@H]([C@H]([C@H]([C@@H](C(=O)O)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00061 Cc1ccc(cc1)Cc2nc(cs2)C(C)(C)C.Br BTB05042 CCOC(=O)/C=C(\C)/Nc1ccc(cc1)OC BTB01229 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3nnc(s3)C4CC4 BTB05058 Cc1cc(n(n1)c2ccc(cc2)NC(=O)c3ccc(c(c3)Cl)Cl)OC(=O)c4ccc(c(c4)Cl)Cl BTB01288 c1ccc2c(c1)[nH]c(n2)c3ccc(cc3)CSc4ccc(cc4)Cl BTB03449 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2c(cc(cc2Br)F)F)Cl BTB03461 Cn1c(nnn1)SCC(=O)Nc2cc(ccc2OC)Cl NRB00234 c1cc(c(cc1F)F)NC(=S)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F AW00315 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)S(=O)(=O)c3ccc(cc3)Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB05048 COC(=O)c1ccc(cc1NC(=O)c2cccnc2Oc3ccccc3)Cl BTB05031 COc1cccc(c1)NC(=S)NNC(=O)c2ccccc2Cl BTB01239 c1ccn2c(c1)cnc2SCc3c(cccc3Cl)Cl BTB05051 CCOC(=O)c1cc2ccccc2oc1=O BTB05052 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Oc3ccccc3Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB05053 c1ccc(cc1)/C(=N/N=C/c2ccc3c(c2)OCO3)/C(=O)c4ccccc4 BTB01278 CCOC(=O)/C(=C/Nc1ccccc1N)/C#N BTB03406 c1cc(c(cc1Br)Cl)N/C=C/C(=O)C(F)(F)F AW00350 Cc1c2ccccc2sc1C(=O)COC(=O)c3ccccc3Cl MWP00204 COC(=O)/C=C\1/C(=O)N=C(S1)Cc2ccc(cc2)[N+](=O)[O-] BTB05070 c1cc2c(cc1/N=C/c3cc(cc(c3O)Cl)Cl)nn[nH]2 BTB01314 Cc1c2cc(ccc2sc1CC(=O)Nc3ccccc3)Cl MWP00240 Cc1c2cc(ccc2sc1CC(=O)Nc3cccc(c3)Cl)Cl MWP00242 C1CC1c2nnc(s2)NC(=O)C(F)(F)F BTB05084 c1ccn2c(c1)cnc2SCc3ccc(cc3)Cl BTB05093 Cc1c2cc(ccc2sc1CC(=O)Nc3ccc(cc3)Cl)Cl MWP00243 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(Cc3ccc(cc3)N(C)C)C(C)C BTB01317 c1cc(cc(c1)Cl)NC(=S)NN=C2CCCCCC2 BTB05119 CCOC(=O)/C(=C/Nc1c(cccn1)C)/C#N BTB03408 c1cc(c(cc1Cl)Cl)NC(=O)c2cnccn2 BTB06752 c1ccc(cc1)NC(=O)OC2c3cc(ccc3OC(=O)N2c4ccccc4)Cl BTB03511 c1ccc(cc1)Oc2c(cccn2)C(=O)NCCSC3=NCCN3.Br BTB03515 c1ccc(c(c1)c2n[nH]c(=S)n2c3cc(ccc3Cl)Cl)Cl BTB01270 Cc1ccccc1C(=O)OCC(=O)c2c(c3cc(ccc3s2)Cl)C MWP00209 Cc1c2cc(ccc2sc1C(=O)Cn3ccnc3)Cl MWP00210 c1cc(ccc1OCC(CN2CCN(CC2)c3nccc(n3)C(F)(F)F)O)F AW00311 Cc1c2ccccc2sc1CC(=O)Nc3ccc(cc3)Cl MWP00214 Cc1cc(n(n1)c2ccc(cc2)NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C)OC(=O)c5c(onc5c6c(cccc6Cl)Cl)C BTB01290 c1cnccc1CCN2CNC(=NC2)S BTB03466 c1cc(c(c(c1)Cl)Cl)S(=O)(=O)N2CCCN(CC2)C(=O)c3cccs3 AW00342 c1cc(cc(c1)F)NC(=S)NN=C2CCCCCC2 BTB05117 c1cc(c(cc1Cl)Cl)N/C=C/C(=O)C(F)(F)F AW00349 c1cc(ccc1Cc2ccncc2)/N=C/c3cc(cc(c3O)Cl)Cl BTB01309 c1ccc(cc1)CN(Cc2ccccc2)O NRB01310 Cc1ccc(cc1)SCc2c3ccccc3sc2Cl MWP00178 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc4c(c3)COCO4)Cl BTB01313 CN(c1ccc(cc1F)F)C(=O)CC#N BTB06692 c1cc(cnc1)NC(=O)c2ccc(cc2)Cl BTB06697 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3nnc(s3)C4CC4 BTB05059 c1cc(ccc1OCc2cc(cc3c2OCOC3)Cl)S(=O)(=O)c4ccc(cc4)OCc5cc(cc6c5OCOC6)Cl BTB05056 Cc1c2ccccc2sc1c3csc(n3)C.Br MWP00227 Cc1c2ccccc2sc1c3csc(n3)c4ccc(cc4)Cl MWP00228 Cc1ccc2c(c1)c(c(s2)C(=O)C)C MWP00218 c1cc(cc(c1)NC(=O)CSc2nnc(s2)N)C(F)(F)F NRB00236 c1cc(ccc1NC(=O)Nc2ccc(cc2)Cl)Cl RJC00062 c1cc(cnc1)C(=O)Nc2ccc(cc2)Cl BTB06718 c1cc(cnc1)C(=O)Nc2ccc(cc2Cl)Cl BTB06719 C/C(=N\c1nnc(s1)Sc2nc3cc(ccc3s2)Cl)/N(C)C BTB06729 c1ccc(cc1)Sc2cccc3c2c(ccc3)C(=O)OCC(=O)c4ccc(cc4)Br RJC00073 CC(C)(C)c1cc(ccc1Oc2c(cccn2)[N+](=O)[O-])Oc3c(cccn3)[N+](=O)[O-] BTB06731 CCC1(c2ccccc2N=C1N)c3ccccc3 NRB01318 c1cc2cccc(c2c(c1)C(=O)OCC(=O)c3ccc(cc3)Br)Br RJC00083 c1ccc(cc1)Oc2c(cccn2)C(=O)Oc3ccccc3Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB05054 CCOC(=O)CCc1ccc(c(c1)[N+](=O)[O-])OC(=O)c2c(onc2c3c(cccc3Cl)Cl)C BTB01320 Cc1c2ccccc2sc1c3csc(n3)c4ccncc4.Br MWP00229 c1ccc(cc1)C(=O)O/N=C(/Cc2csc3c2cc(cc3)Cl)\N MWP00232 CCOC(=O)NNC(=O)Nc1cccc(c1)C(F)(F)F NRB01351 c1ccc(cc1)/C(=N\N=C\c2cccs2)/C(=O)c3ccccc3 BTB01281 Cc1ccc(c(c1C)NC(=O)c2ccc(cc2)Cl)[N+](=O)[O-] BTB06733 Cc1cc(c2cc(ccc2n1)F)OC(=O)c3c(onc3c4ccccc4)C BTB01297 Cc1cc(c2cc(ccc2n1)F)OC(=O)c3c(c4ccccc4s3)Cl BTB01298 CCOC(=O)C1=CNc2ccccc2N=C1N BTB03402 Cc1c(c(no1)c2ccccc2Cl)C(=O)N(Cc3ccc(cc3)N(C)C)C(C)C BTB01319 c1ccc(cc1)NC(=O)O/N=C(/Cc2csc3c2cc(cc3)Cl)\N MWP00233 CNC(=O)O/N=C(/Cc1csc2c1cc(cc2)Cl)\N MWP00234 Cc1c2ccccc2sc1c3csc(n3)c4ccccc4 MWP00225 Cc1c2cc(ccc2sc1CC(=O)O)Cl MWP00226 c1ccc(cc1)/C(=N/N=C/c2ccc(cc2)Cl)/C(=O)c3ccccc3 BTB01282 c1ccc(c(c1)C(F)(F)F)NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F AW00341 Cc1ccc(c2c1nc(cc2OCc3c(c(c(c(c3C)C)C)C)C)C)Cl BTB01284 c1ccc(c(c1)c2nnc(s2)Nc3ccc(cc3)F)Cl BTB01256 c1ccc(cc1)SCc2c3ccccc3sc2Cl MWP00176 CC(C)N(Cc1ccc(cc1)N(C)C)S(=O)(=O)c2ccccc2[N+](=O)[O-] BTB01295 Cn1c(nnn1)SCC(=O)Nc2cccc(c2)C(F)(F)F NRB00235 COc1cc(cc(c1OC)OC)/C=N/N=C\2/NC(=O)CS2 RJC00037 c1cc(sc1)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)Br RJC00038 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc(ccc3C(=O)OC)Cl BTB05033 c1ccc(cc1)C(=O)O/N=C(/Cc2csc3c2cccc3)\N MWP00246 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc4c(c3)nn[nH]4)Cl BTB01310 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc4c(c3)nn[nH]4 BTB01312 CN(C)/C=C(\C#N)/c1cccc(c1)C(F)(F)F AW00343 CCN(Cc1cc(c(c(c1)OC)OC)OC)S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl BTB01272 CN(C)c1ccc(cc1)/C=N/N=C(/c2ccccc2)\C(=O)c3ccccc3 BTB01277 Cc1c(c(no1)c2ccccc2)C(=O)N(Cc3ccc(cc3)N(C)C)C(C)C BTB01315 c1ccc(c(c1)NC(=S)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)N4CCOCC4 AW00316 c1cc(cnc1)NC(=S)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F AW00319 Cc1c2cc(ccc2sc1c3csc(n3)c4ccccc4)Cl MWP00221 c1cc(c(cc1C(=O)Nc2cc3cc(ccc3oc2=O)[N+](=O)[O-])Cl)Cl BTB03414 Cc1ccc(cc1NC(=O)CSc2ncccn2)F NRB00247 c1cc(c(c(c1)Cl)n2cc[nH]c2=S)Cl RJC00035 COC(=O)C/C(=N/NC(=O)c1cc(ccc1N)[N+](=O)[O-])/C(=O)OC BTB05035 c1cc(ccc1CSc2[nH]c3ccc(cc3n2)C(F)(F)F)Br.Br BTB04959 Cc1ccccc1C(=O)OCC(=O)c2c(c3ccccc3s2)C MWP00205 Cc1c2cc(ccc2sc1C(=O)COC(=O)c3ccc(cc3Cl)Cl)Cl MWP00207 c1cc(c(c(c1)C(=O)OCC(=O)c2ccc(cc2)Br)Br)C(=O)OCC(=O)c3ccc(cc3)Br RJC00102 c1cc(ccc1C(=O)NCCc2ccncc2)[N+](=O)[O-] BTB03432 c1ccc(cc1)c2nccc(n2)C(F)(F)F AW00322 CC(C)N(Cc1ccc(cc1)N(C)C)C(=O)c2c(c3ccccc3s2)Cl BTB01318 Cc1c2cc(ccc2sc1C(=O)COC(=O)c3ccccc3Cl)Cl MWP00208 Cc1c2ccccc2sc1CC(=O)Nc3ccccc3F MWP00211 Cc1c2ccccc2sc1CC(=O)Nc3ccccc3 MWP00213 CC(=O)Nc1ccc(cc1)CC(C#N)C#N BTB03407 c1cc2c(cc1Cl)sc(n2)N3CCCNCC3 AW00326 CCCCCc1ccc(cc1)C(=O)Oc2ccc(cc2)C#N NRB01329 c1ccc(cc1)C(Cc2ccccc2[N+](=O)[O-])(C#N)c3ccccc3 NRB01330 CCC(C#N)(c1ccccc1)c2ccc(cc2Cl)[N+](=O)[O-] NRB01331 CCOC(=O)C12CCC(CC1)(CC2)OS(=O)(=O)c3ccc(cc3)C NRB01359 CCOC(=O)C(C(=O)OCC)NC(=O)c1cc2ccccc2s1 BTB06653 CCOC(=O)C(C(=O)OCC)NC(=O)c1cccnc1SC BTB06654 c1cc2c(cc1C(F)(F)F)nc([nH]2)SCc3cc(cc4c3OCOC4)Cl.Cl BTB04965 CC(=O)c1ccc(c(c1)CSc2[nH]c3ccc(cc3n2)C(F)(F)F)OC.Cl BTB04966 COc1ccc-2c(c1)CCc3c2nc(s3)/N=C/c4ccc(cc4)C(F)(F)F RH01220 CC(=O)Nc1cc(ccc1Sc2ccccc2N)[N+](=O)[O-] AW00323 c1ccc(cc1)C(C#N)N2CCSCC2 NRB01313 c1cc2c(cc1Cl)sc(n2)N3CCCN(CC3)C(=S)NC4CCCCCCC4 AW00338 CCOC(CC(c1ccccc1)(c2ccccc2)C(=O)N(C)C)OCC NRB01321 CC(C)(C)c1cc(ccc1Oc2ccc(cn2)[N+](=O)[O-])Oc3ccc(cn3)[N+](=O)[O-] BTB06727 c1ccc(cc1)c2ccc(cc2)c3csc(n3)c4cccnc4 MWP00294 CCCCCC(=O)Nc1nc-2c(s1)CCc3c2cccc3 RH01223 COc1ccc(cc1Br)/C=C\2/C(=O)NC(=S)S2 BTB04947 c1cc2c(=O)c3cc(ccc3oc2nc1)[N+](=O)[O-] BTB04948 CC(C)(C)NC(=S)Nc1ccc(cc1Cl)[N+](=O)[O-] BTB03327 Cc1cccc(c1NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)Cl AW00339 COC(=O)c1ccc(cc1NS(=O)(=O)C)Cl BTB06700 c1ccnc(c1)NC(=O)CC#N BTB06714 CCCC1=NN(C(=O)C1)c2ccc(cc2)S(=O)(=O)N BTB06720 CC(C)(C)c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB06723 CN(C)/C=C(\C#N)/C(=O)Nc1ccccn1 BTB06724 CC(=O)O/N=C(/Cc1csc2c1cc(cc2)Cl)\N MWP00235 CC(=O)Nc1ccc(cc1C(=O)OCC(=O)c2ccc(cc2)Br)Cl RJC00091 c1ccc(c(c1)C(=O)NCCc2ccncc2)N BTB03423 c1cc2c(cc1[N+](=O)[O-])cc(c(=O)o2)N BTB03328 Cc1ccc(c(c1)[N+](=O)[O-])NC(=S)NC(C)(C)C BTB03332 CC(C)(C)NC(=S)Nc1ccc(cc1[N+](=O)[O-])C(F)(F)F BTB03333 Cc1nc2ccc(cc2o1)NC(=O)c3ccccc3C(F)(F)F MWP00030 CC(=C1CCCCC1)C(=O)O NRB01376 Cc1c(c(no1)c2ccccc2)NC(=O)N3c4ccc(cc4CCC3C)F BTB03395 c1cc(c(cc1Cl)NC(=S)NCCc2ccncc2)Cl BTB03436 c1ccc(cc1)NC(=O)O/N=C(/Cc2csc3c2cccc3)\N MWP00248 CCOC(=O)/C(=C/Nc1ccncc1)/C#N BTB03405 c1cc(cnc1)NC(=O)c2ccc(cc2Cl)Cl BTB06742 Cc1ccc(c(c1)C(=O)OCC(=O)c2ccc(cc2)Br)I RJC00105 c1cc(c(cc1C(F)(F)F)NC(=S)NN)Cl BTB05098 c1ccn2c(c1)c(nc2SCc3cccc(c3)F)C(=O)C(F)(F)F BTB05101 c1cc(c(cc1[N+](=O)[O-])C(=O)NCCc2ccncc2)N BTB03424 CCOC(=O)c1ccc(cc1)N2CC3CCCCN3C2c4ccccc4 BTB01365 Cc1nc2ccc(cc2o1)NS(=O)(=O)c3ccc(cc3F)F MWP00039 CCc1c([nH]c2c1cc(cc2)[N+](=O)[O-])C RH01219 Cc1ccc(c(c1)C)NC(=S)N2CCN(CC2)c3nccc(n3)C(F)(F)F AW00306 Cc1nc2cc(ccc2c(=O)n1c3ccncc3)Cl BTB01327 Cn1c(=O)n2n(c1=O)C3CC2C=C3 NRB01366 Cc1c(c(no1)c2ccccc2Cl)NC(=O)NCc3cccs3 BTB03403 CCOC(=O)/C(=C/NC1CCN(CC1)Cc2ccccc2)/C#N BTB03404 c1cc(ccc1C(=O)Nc2cnccn2)Cl BTB06748 c1cc(ccc1NC(=O)c2cnccn2)Cl BTB06753 CNc1ccccc1C(=O)NCCc2ccncc2 BTB03422 CN(C)c1ccc(c(c1)Cl)/C=C\2/C(=O)OC(=N2)c3ccccc3 BTB01352 c1ccc(c(c1)N)Sc2nc3cc(ccc3s2)Cl BTB06768 c1cnccc1CCNC(=O)C(F)(F)F BTB03453 Cc1ccc(c(c1)O)NC(=O)c2ccc(cc2)CSc3ccc(cc3)Cl BTB03456 c1ccc(c(c1)N)Sc2nc3c(s2)cc(cc3Cl)Cl BTB06743 Cc1nc2cc(ccc2c(=O)n1Cc3ccncc3)Cl BTB01330 COc1cc(cc(c1OC)OC)/C=N/N=C/c2cc(cc(c2O)Cl)Cl BTB01337 c1cc(cnc1)c2nnnn2c3ccc(cc3Cl)Cl BTB06744 CCOC(=O)c1ccc(cc1)/N=C/c2cc(cc(c2O)Cl)Cl BTB01345 CN(c1ccc(cc1F)F)C(=O)CSc2cc(ccc2Cl)Cl BTB06755 Cc1c2cc(ccc2sc1C(=O)CCSc3ccccc3)Cl MWP00281 CC(C)NC(=S)NCCc1ccncc1 BTB03435 Cc1cc(c(cc1Cl)C)Sc2ccc(cc2[N+](=O)[O-])C(=O)O BTB06757 c1cc(ccc1S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(=O)O)Cl BTB06759 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(=O)O BTB06760 Cc1c(c(c(c(c1C)C)CSc2nnc(n2c3ccccc3OC)c4ccccc4Cl)C)C BTB01361 Cc1cc(c(cc1Cl)C)SCCC(=O)c2c(c3cc(ccc3s2)Cl)C MWP00284 Cc1ccc(cc1Cl)NC(=O)CC#N BTB05181 CC(C)(C)c1csc(n1)N/N=C/c2cccs2.Br BTB05182 C/C(=N\N=C(/N=C/N(C)C)\SC)/c1ccc(c(c1)Cl)Cl BTB05184 c1cc(c(cc1Cl)Cl)OCOc2ccc(cc2Cl)Cl BTB05155 CSc1ccc(cc1)OCOc2ccc(cc2)SC BTB05158 CCOC(=O)/C(=C/N/C(=N\N=C(/C)\c1ccc(cc1)Br)/SC)/C#N BTB05190 CN(C)/C=N/C(=N\N=C\c1c(cccc1Cl)Cl)/SC BTB05174 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2[N+](=O)[O-])OC BTB01442 Cc1c2ccccc2sc1/C(=N/OC(=O)Nc3ccccc3)/C MWP00348 Cc1c2ccccc2sc1/C(=N/OC(=O)c3ccccc3)/C MWP00355 COC(=O)/C=c\1/c(=O)n2c3cc(c(cc3nc2s1)Cl)Cl BTB05164 Cc1cc(ccc1NC(=O)c2c(cccc2Cl)Cl)NC(=O)C BTB01415 Cc1cc2c(cc1C)CSC(SC2)c3cccc(c3O)OC BTB01410 COc1ccc(c(c1)[N+](=O)[O-])NC(=S)NC(=O)c2ccccc2 BTB01427 CS/C(=N/N=C/c1c(cccc1Cl)Cl)/N BTB05171 Cc1cc(ccc1NS(=O)(=O)c2ccc(cc2)Cl)NC(=O)C BTB01425 c1ccc2c(c1)nc(s2)N(c3cccc(c3)Cl)C(=S)Nc4ccc(cc4)F BTB01430 c1ccc2c(c1)nc(s2)N(c3cccc(c3)Cl)C(=S)Nc4ccc(cc4Cl)Cl BTB01431 CN(C)c1ccc(cc1)/C=N/NC(=S)N BTB05176 Cc1cc2c(cc1C)CSC(SC2)(C)c3cccc(c3)[N+](=O)[O-] BTB01437 Cn1c(nnc1Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)c3csc4c3cc(cc4)Cl MWP00385 c1ccc2c(c1)nc(s2)Nc3cccc(c3)Cl BTB01433 Cc1ccc(cc1)C2(SCc3cc(c(cc3CS2)C)C)C BTB01439 CC1(C(=C)S/C(=N\c2ccccc2OC)/N1)C BTB01441 c1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)SCCC(=O)O RJC00171 CCC(C)(C)c1ccc(c(c1)C(C)(C)CC)OCC(=O)Nc2ccc(c(c2)N)Cl NRB01437 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)Cl)/CO2 RJC00143 c1ccc2c(c1)C(=O)/C(=C/c3ccncc3)/CO2 RJC00144 c1ccc2c(c1)c(c[nH]2)/C=C/3\COc4ccccc4C3=O RJC00146 Cc1c2ccccc2sc1/C(=N/OC(=O)c3ccccc3Cl)/C MWP00356 Cc1c2ccccc2sc1/C(=N/OC(=O)c3ccc(cc3)C(F)(F)F)/C MWP00357 Cc1cc(ccc1NC(=S)N(c2cccc(c2)Cl)c3nc4ccccc4s3)Cl BTB01432 Cc1c(c(n(n1)c2ccccc2)C)/N=N/c3ccc(cc3F)F BTB03536 Cc1c2cc(ccc2sc1CC(=O)NNC(=O)Nc3ccccc3)Cl MWP00370 Cc1c2cc(ccc2sc1CC(=O)NNC(=O)c3ccccc3)Cl MWP00390 c1ccc(c(c1)NC(=S)NNS(=O)(=O)c2ccc(cc2)Cl)F AW00376 CC(C)(C)OC(=O)NCCNC(=O)c1ccccc1Cl AW00377 Cc1c2c(cc(=O)oc2n(n1)c3cccc(c3)Cl)C(F)(F)F BTB06791 c1ccc(cc1)NC(=O)NNC(=O)c2csc(n2)Cc3ccsc3 MWP00379 c1ccc2cc(ccc2c1)/C=C/3\COc4ccccc4C3=O RJC00147 c1cc(ccc1c2nnnn2c3cnccn3)Cl BTB06803 CC(C)(C)OC(=O)NCCNC(=S)Nc1ccc(cc1OC)OC AW00378 Cc1cc(ccc1NC(=O)c2ccc(cc2)[N+](=O)[O-])NC(=O)C BTB01413 Cc1ccc(c(c1)C(=O)Nc2ccc(cc2C)NC(=O)C)[N+](=O)[O-] BTB01414 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)SCC(=O)O RJC00174 COc1ccc(cc1OC)/C=C/2\Cc3ccccc3C2=O RJC00130 c1ccc2cc(ccc2c1)/C=C/3\CCc4ccccc4C3=O RJC00140 Cc1ccc(c(c1)C)N(CC=C)C2=NC(C(=C)S2)(C)C BTB05237 c1cc(c(cc1C(F)(F)F)NC(=O)CC#N)Cl BTB05180 c1ccc(cc1)/C=C/2\CSc3ccccc3C2=O RJC00148 c1ccc2cc(ccc2c1)/C=C/3\CSc4ccccc4C3=O RJC00153 CSC(=NS(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)SC BTB06825 CCO/C(=N\Nc1ccccc1[N+](=O)[O-])/CC(=O)OCC NRB01449 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCc3ccncc3 BTB03471 Cc1c2cc(ccc2sc1CC(=O)NNC(=O)C)Cl MWP00389 c1ccc(cc1)C2/C(=C/c3cccs3)/C(=O)c4ccccc4O2 RJC00163 CCCCCCCCCCCCCCCCCCOc1ccccc1C(=O)CC(=O)OCC NRB01433 CCOC(=O)c1c(cccc1OC)OC NRB01434 Cc1ccc(cc1)S(=O)(=O)N2CCCN(CC2)C(=O)OC(C)(C)C AW00383 CC(C)(C)OC(=O)N1CCCN(CC1)C(=S)Nc2ccc(cc2F)F AW00384 Cc1cc(=O)oc2c1c(nn2c3ccccc3)C(F)(F)F BTB06806 CC(C)NC(=O)NCCNC(=O)OC(C)(C)C AW00393 CCOC(=O)CNC(=O)c1c(onc1c2c(cccc2Cl)Cl)C BTB03475 c1ccc(cc1)Oc2c(cccn2)C(=O)NCC(=O)NN BTB03490 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2[N+](=O)[O-])C BTB01434 CC1(C(=C)S/C(=N/c2cccc(c2)C(F)(F)F)/N1)C BTB01435 CC1(CC(=O)c2ccc(cc2O1)OCc3cccc(c3)F)C RJC00182 CC1(CC(=O)c2cc(c(cc2O1)OCc3ccc(cc3)[N+](=O)[O-])OCc4ccc(cc4)[N+](=O)[O-])C RJC00190 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)c4ccc(cc4)OC(=O)c5c(onc5c6c(cccc6Cl)Cl)C BTB05210 Cc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2C)[N+](=O)[O-] BTB01443 CC(C)(C)OC(=O)NCCNC(=O)c1ccc(cc1)OC(F)(F)F AW00397 CCOC(=O)/C(=C/N/C(=N\N=C\c1c(cccc1Cl)Cl)/SC)/C#N BTB05191 C/C(=N\Nc1nc(cs1)C(C)(C)C)/c2ccc(cc2)F.Br BTB05193 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)[N+](=O)[O-])C BTB01444 Cc1ccc(cc1)S(=O)(=O)N(c2cccc(c2)Cl)c3nc4ccccc4s3 BTB01445 CC(=O)C(=NNc1ccc(cc1F)F)C(=O)C BTB03507 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Br)SCC(=O)O RJC00175 c1cc(ccc1c2ccc(cc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB05195 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)c2ccc(cc2)Cl AW00386 CC1(CC(=O)c2ccc(cc2O1)OCc3ccc(cc3)F)C RJC00183 Cc1cc(cc2c1C(=O)CC(O2)(C)C)OCc3ccc(cc3)Br RJC00187 CN(C)c1ccc(cc1)C2NN3C(=N2)C(=CN=C3SC)C#N BTB05201 CC(C)(C)OC(=O)NCCNC(=O)Nc1ccccc1C(F)(F)F AW00395 CC(C)(C)OC(=O)NCCNC(=S)NCc1ccccc1 AW00396 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCC(=O)NN BTB03504 CCc1ccc(cc1)NC(=S)Nc2ccc(cc2C(=O)c3ccccc3)Cl BTB01343 Cc1ccc(c(c1)C)NC(=S)N2CCCN(CC2)C(=O)OC(C)(C)C AW00381 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)c2ccc(cc2)[N+](=O)[O-] AW00388 CC(C)CNC(=S)NCCNC(=O)OC(C)(C)C AW00387 Cc1nc(cs1)c2ccc(cc2)NC(=O)C AW00392 CS/C(=N/N=C/c1c(cccc1Cl)F)/N BTB05197 Cc1c2cc(ccc2sc1/C(=N/OC(=O)Nc3ccc(cc3)Cl)/C)Cl MWP00319 C/C(=N\N=C(\N)/SC)/c1ccc(cc1)F BTB05214 Cc1c(c(n(n1)c2ccccc2)c3ccccc3[N+](=O)[O-])C(=O)O NRB01451 CN(C)/C=C(\C#N)/C(=O)Nc1ccccc1Oc2ccc(cc2Cl)Cl BTB06826 c1ccc(cc1)CN2c3ccccc3C(=O)CS2(=O)=O BTB06829 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)Nc2ccc(cc2F)F)Cl BTB05131 Cc1ccc(cc1)S(=O)(=O)CCNC(=O)c2c(onc2c3c(cccc3Cl)Cl)C BTB03498 CCOC(=O)CCC(C#N)(c1cccs1)N2CCOCC2 BTB03502 CC(C)(C)OC(=O)NCCNS(=O)(=O)c1ccc(cc1)Cl AW00382 C[C@H]1c2c(c(c(c(c2)[C@H](c3c(c(c(c(c3)[C@H](c4c(c(c(c(c4)[C@H](c5c(c(c(c1c5)O)Br)O)C)O)Br)O)C)O)Br)O)C)O)Br)O NRB01439 CCOC(=O)c1ccc(cc1)N2CC3CCCCN3C2c4cccc(c4O)OC BTB01363 c1cc(cnc1)c2nc(cs2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F MWP00341 c1ccc(cc1)C2/C(=C/c3c[nH]c4c3cccc4)/C(=O)c5ccccc5O2 RJC00164 c1cc(sc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)N)C(F)(F)F BTB06812 C/C(=N\N=C(/N)\SC)/c1ccc(c(c1)Cl)Cl BTB05137 CC(CO)(CO)NCC(COc1ccc(cc1)OC(F)(F)F)O AW00358 c1ccc(c(c1)NC(=O)CC#N)Oc2cc(ccc2Cl)Cl BTB06815 CN(C)C(=O)c1cccnc1SC BTB06828 c1ccc(cc1)CS(=O)(=O)CC(COc2ccc(cc2)OC(F)(F)F)O AW00365 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2ccc(cc2)Cl AW00367 Cc1cc(c2cc(ccc2n1)Cl)OCc3cc(ccc3OC)C(=O)C BTB01322 c1ccc(cc1)C(=O)c2cc(ccc2NC(=S)Nc3cccc(c3)Cl)Cl BTB01325 CCOC(=O)COc1ccc2c(c1)OC(CC2=O)(C)C RJC00177 c1cc2c(cc1/N=C/c3cc(ccc3O)Br)nn[nH]2 BTB01340 CC(C)(C)OC(=O)NCCNC(=S)NC1CCCCCCC1 AW00375 Cc1cccc(c1)NC(=S)N2CCOC2c3ccsc3 MWP00287 c1ccc(c(c1)N/C=N/O)Sc2nc3cc(ccc3s2)Cl BTB06776 c1cc(ccc1OCC(CN2CCN(CC2)c3nccc(n3)C(F)(F)F)O)OC(F)(F)F AW00359 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])C(=O)O BTB06783 CCOC(=O)/C(=C/N(C)c1ccc(cc1F)F)/C#N BTB06784 CN1C(=O)CC(=N1)C(F)(F)F BTB06790 CN(C)/C=N/c1nnc(s1)SCc2ccc(cc2)C(=O)Oc3c(cccc3F)F BTB06794 CN(C)/C=N/c1nnc(s1)SCc2ccc(cc2)C(=O)Oc3ccc(cc3F)F BTB06795 COc1cccc(c1)/C=C/2\Cc3ccccc3C2=O RJC00125 c1ccc(cc1)Sc2cccc3c2c(ccc3)C(=O)N RJC00126 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCSC3=NCCN3.Br BTB03514 Cc1cc(c(cc1Cl)C)SCCC(=O)c2c(c3ccccc3s2)C MWP00278 CN(C)/C=N/c1nnc(s1)SCC(=O)c2ccc(cc2)[N+](=O)[O-] BTB06779 c1ccc(cc1)C2=CC=C(C2)c3ccccc3 NRB01379 Cc1c(c(n(n1)c2ccccc2)c3ccccc3[N+](=O)[O-])C(=O)C NRB01406 c1cc(sc1)C(C#N)N2CCOCC2 BTB03488 c1ccc2c(c1)c(c(s2)Cl)CSc3ccc(cc3)Cl MWP00177 Cc1c2cc(ccc2sc1CC(=S)N3CCOCC3)Cl MWP00201 c1cc(c(cc1CSCC(=O)Nc2ccc(cc2F)F)Cl)Cl NRB00239 CCOc1ccc(cc1)NC(=O)C(=O)Nc2ccccc2 NRB00240 CN(C)c1ccc(cc1)/C=C/2\Cc3ccccc3C2=O RJC00127 COc1cc(ccc1O)/C=C/2\Cc3ccccc3C2=O RJC00129 c1cc(ccc1CSc2[nH]c(=O)cc(n2)N)C(=O)Oc3ccc(cc3F)F BTB06821 CCCc1cc(=O)[nH]c(n1)SCc2ccc(cc2)C(=O)Oc3ccc(cc3F)F BTB06822 CC1(CC(=O)c2ccc(cc2O1)OCC(=O)O)C RJC00176 c1ccc(cc1)N2C(=O)CC(=N2)C(F)(F)F BTB06798 Cc1cc(=O)oc2c1c(nn2C)C(F)(F)F BTB06800 CN(C)/C=C/1\C(=NN(C1=O)c2ccccc2)C(F)(F)F BTB06808 CC\1=NN(C(=O)/C1=C/2\C(=NN(C2=O)c3ccccc3)C)c4ccccc4 NRB01407 Cc1c2ccccc2sc1C(=O)c3ccccc3C(=O)O MWP00297 C/C(=N\N=C(/N)\SCc1c(cccc1Cl)Cl)/c2ccc(c(c2)Cl)Cl BTB05136 Cc1cc(n(n1)C2=NCCN2C=C(C#N)C#N)C BTB05139 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)Nc2ccc(c(c2)Cl)F)Cl BTB05160 CO[C@@H]1[C@H]([C@H](C2[C@H](O1)COC(O2)c3ccccc3)O)O RJC00065 c1ccc(c(c1)C(F)(F)F)NC(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00334 c1ccc(c(c1)C(F)(F)F)NC(=O)N2CCCN(CC2)c3c(cccn3)C(F)(F)F AW00336 CCC(c1ccccc1)(c2ccc(cc2)[N+](=O)[O-])C(=O)N NRB01333 CC1(NN2C(=N1)C(=CN=C2SC)C#N)c3ccc(c(c3)Cl)Cl BTB05143 c1ccc2c(c1)C/C(=C\c3ccccc3Cl)/C2=O RJC00122 CCN(CC)c1ccc(cc1)N/N=C\2/C(=NN(C2=O)c3ccccc3)C NRB01416 c1ccc(cc1)NC(=O)c2csc3c2cc(cc3)Cl MWP00268 Cc1ccc(cc1NS(=O)(=O)C)NC(=S)Nc2ccccc2Cl BTB01391 COC(=O)c1ccccc1NS(=O)(=O)C BTB06819 CN(C)/C=N/S(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3 BTB06824 Cc1nc2cc(ccc2c(=O)n1c3cccnc3)Cl BTB01328 COc1cc(cc(c1OC)OC)/C=N/N=C/c2cc(ccc2O)Br BTB01338 CS(=O)(=O)NNC(=O)c1csc(n1)c2cccnc2 MWP00342 c1cc(ccc1C#N)OCOc2ccc(cc2)C#N BTB05159 COc1ccc(cc1)/C=C/2\CCc3ccc(cc3C2=O)OC RJC00138 COc1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)Cl)/CC2 RJC00139 CC(C)NC(=O)c1cccc2c1c(ccc2)Sc3ccccc3 RJC00141 Cc1cc(c(cc1Cl)C)SCC(=O)N(C)c2ccc(cc2F)F BTB06693 CN(C)/C=C(\C#N)/C(=O)N(C)c1ccc(cc1F)F BTB06695 Cc1ccc(c(c1C)NC(=O)c2c(nn(n2)c3ccccc3)C)[N+](=O)[O-] BTB06734 Cc1ccc(c(c1C)NC(=O)NC(=O)c2c(cccc2Cl)Cl)[N+](=O)[O-] BTB06735 Cc1ccc(c(c1C)NC(=O)NC(=O)c2c(cccc2F)F)[N+](=O)[O-] BTB06736 Cc1ccc(cc1NS(=O)(=O)C)NC(=S)Nc2ccc(cc2)OC BTB01392 Cc1ccc(cc1NS(=O)(=O)C)NC(=S)Nc2cccc(c2)Cl BTB01390 Cc1ccc(cc1NS(=O)(=O)C)NC(=S)Nc2cccc(c2)C(F)(F)F BTB01393 Cc1ccc(cc1NS(=O)(=O)C)NC(=S)Nc2ccccc2OC BTB01394 C/C(=N\NC(=S)N)/c1cc2cc(ccc2o1)Cl BTB05148 c1cc(ccc1S(=O)(=O)O/N=C(/CC(=O)Nc2ccc(cc2F)F)\N)Cl BTB05151 COc1cc(cc(c1OC)OC)/C=C/2\Cc3ccccc3C2=O RJC00131 c1ccc2c(c1)cccc2/C=C/3\Cc4ccccc4C3=O RJC00132 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2ccc(cc2F)F)Cl BTB05129 c1ccc(cc1)c2ccc(cc2)c3csc(n3)c4ccccc4 MWP00290 Cc1c2cc(ccc2sc1/C(=N/O)/C)Cl MWP00315 c1ccc(cc1)NC(=O)NNC(=O)c2csc(n2)c3cccnc3 MWP00334 c1cc(cnc1)c2nc(cs2)C(=O)NNC(=O)Nc3ccc(cc3)Cl MWP00335 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCS(=O)(=O)c3ccc(cc3)Cl BTB03497 COc1cc(cc(c1OC)OC)C2=NNC(=O)CC2 BTB03505 Cc1ccc(cc1[N+](=O)[O-])C2=N/C(=C\c3cccs3)/C(=O)O2 BTB01399 Cc1ccc(cc1[N+](=O)[O-])C2=N/C(=C\c3ccc(cc3)N(C)C)/C(=O)O2 BTB01400 Cc1ccc(cc1)C2SCc3cc(c(cc3CS2)C)C BTB01407 Cc1ccc(cc1NS(=O)(=O)C)NC(=S)NCc2ccccc2 BTB01395 c1ccc(cc1)C(=O)c2cc(ccc2NC(=S)Nc3ccc(cc3)F)Cl BTB01397 Cc1cccc(c1)NC(=S)Nc2ccc(c(c2)NS(=O)(=O)C)C BTB01379 c1cc(cnc1)c2nc(cs2)C(=O)NNS(=O)(=O)c3ccc(cc3F)F MWP00345 CC1(C(=C)S/C(=N\c2ccccc2Cl)/N1)C BTB01403 Cc1cc2c(cc1C)CSC(SC2)c3ccccc3Cl BTB01406 Cc1cc2c(cc1C)CSC(SC2)c3ccc(c(c3)Cl)Cl BTB01408 c1ccc(cc1)/C=C/2\COc3ccccc3C2=O RJC00142 c1ccc(c(c1)C(=O)OCC(=O)c2ccc(cc2)Br)Sc3ccccc3C(=O)OCC(=O)c4ccc(cc4)Br RJC00100 c1ccn2c(c1)cnc2SCc3cccc(c3)F.Br BTB05097 Cc1c(c(no1)c2ccccc2Cl)NC(=O)NCCc3ccncc3 BTB03426 c1cc(c(c(c1)Cl)C(=O)NC(=O)NCCc2ccncc2)Cl BTB03428 c1cc(c(c(c1)F)C(=O)NC(=O)NCCc2ccncc2)F BTB03429 c1ccn2c(c1)cnc2SCc3ccc(cc3)[N+](=O)[O-].Br BTB05109 Cc1c2cc(ccc2sc1CC(=O)NNC(=O)NC(C)C)Cl MWP00369 C[n+]1cccc(c1)c2[nH]c(nn2)c3ccccc3.[I-] NRB01444 c1ccc2c(c1)C/C(=C\c3cccc(c3)Cl)/C2=O RJC00123 COc1ccc(cc1O)/C=C/2\Cc3ccccc3C2=O RJC00128 c1cc(c(c(c1)Cl)/C=N/NC(=S)N)Cl BTB05146 c1cc(c(c(c1)Cl)/C=N/NC(=S)N)F BTB05147 Cc1ccc(cc1NS(=O)(=O)C)NC(=S)NC(=O)c2ccccc2 BTB01398 CC(C)NC(=O)NNC(=O)c1csc(n1)c2cccnc2 MWP00337 c1ccc(cc1)C(=O)NNC(=O)c2csc(n2)c3cccnc3 MWP00339 c1cc(c(nc1)Oc2ccc(cc2)c3ccc(cc3)Oc4c(cccn4)[N+](=O)[O-])[N+](=O)[O-] BTB05229 c1ccc2c(c1)CCNC2=S MWP00430 c1ccc2c(c1)C(=O)/C(=C/c3cccs3)/CO2 RJC00145 Cc1ccc(cc1)/C=C/2\CSc3ccccc3C2=O RJC00149 c1ccc(cc1)S(=O)(=O)NNC(=O)c2csc(n2)c3cccnc3 MWP00343 CC(C)NC(=O)NNC(=O)c1csc(n1)Cc2ccsc2 MWP00377 c1ccc(cc1)NC(=S)NN=C2CCCCCC2 BTB05115 Cc1ccc(cc1)S(=O)(=O)O/N=C(/CC(=O)Nc2ccc(cc2F)F)\N BTB05132 C/C(=N\NC(=S)N)/c1ccc(c(c1)Cl)Cl BTB05133 C/C(=N\Nc1nc(cs1)C(C)(C)C)/c2cc3cc(ccc3o2)Cl.Br BTB05169 c1cc2c(cc1/C=N/NC(=S)N)OCO2 BTB05177 C/C(=N\Nc1nc(cs1)C(C)(C)C)/c2ccc(c(c2)Cl)Cl.Br BTB05144 CCOC(=O)/C(=C/N/C(=N\N=C(/C)\c1ccc(c(c1)Cl)Cl)/SC)/C#N BTB05145 c1cc(ccc1NC(=O)CC#N)F BTB05238 CCc1c(nc2c(n1)cc(cc2Cl)C(F)(F)F)CC BTB05244 c1ccc(cc1)C2(CC2(c3ccccc3)c4ccccc4)c5ccccc5 RJC00226 c1ccc2cc(ccc2c1)/C=C/3\Cc4ccccc4C3=O RJC00133 COc1ccc2c(c1)C(=O)/C(=C/c3ccccc3)/CC2 RJC00137 Cc1c(c(n(n1)c2ccccc2)C)/N=N/c3cc(cc(c3)Cl)Cl BTB03537 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCNC(=O)OC(C)(C)C AW00374 c1cc(ccc1/N=C/c2cc(cc(c2O)Cl)Cl)N3CCOCC3 BTB01376 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)c3ccc(cc3)OS(=O)(=O)c4ccc(cc4)C BTB05187 Cc1cc(ccc1NC(=O)c2c(onc2c3ccccc3Cl)C)NC(=O)C BTB01411 Cc1cc(ccc1NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C)NC(=O)C BTB01412 CC(C)(C)c1csc(n1)N/N=C/c2ccc(cc2)Cl.Br BTB05178 C/C(=N\N=C(/N)\SC)/c1ccc(cc1)Br BTB05186 Cc1cc2c(cc1C)CSC(SC2)c3ccc(cc3)N(C)C BTB01409 CCOC(=O)c1ccc(cc1)NC(=O)CSc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB01464 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCc3cccnc3 AW00423 CC(C)(C)OC(=O)NCCN1C(=O)CC2(C1=O)CCCC2 AW00424 c1ccc(c(c1)C(=O)CC#N)[N+](=O)[O-] NRB01454 CCOC(=O)/C(=C/Nc1cc(ccc1C)C(=O)OC)/C#N BTB03649 Cc1ccc(cc1)S(=O)(=O)n2c3ccc(cc3nc2Sc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-])C BTB01480 C(CC(=O)O)c1c(=O)[nH]c(=O)[nH]n1 NRB01467 CC\1=NN(C(=O)/C1=C(/c2ccccc2)\Nc3ccc(cc3)OC)c4ccccc4 NRB01461 CC1=NN(C(=O)C1)c2c(cc(cc2Cl)Cl)Cl NRB01471 c1ccc(cc1)n2c(=O)n3n(c2=O)C4CCC3C4 RJC00231 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)Cc4ccccc4 AW00407 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3ccc(cc3Cl)Cl AW00414 Cc1ccc(c(c1)[N+](=O)[O-])C(=O)N(c2cccc(c2)Cl)c3nc4ccccc4s3 BTB01455 Cc1c2cc(ccc2sc1CC(=O)NNS(=O)(=O)c3ccccc3C(F)(F)F)Cl MWP00396 CCO.Cc1c2c([nH]n1)NC(C3=C2CC(CC3=O)(C)C)c4ccc(cc4)OC NRB01475 Cc1ccc(c(c1)C)NS(=O)(=O)c2ccc(s2)c3csc(n3)C AW00421 COc1ccc(c(c1)[N+](=O)[O-])NS(=O)(=O)c2ccc(cc2)Cl BTB01460 CCCCCCCCCCCCCCCCCC(=O)Nc1ccc2c(c1)C(=O)C(C2)Sc3nnnn3c4ccccc4 NRB01517 CCOC(=O)C(=CNc1cc(ccc1C)C(=O)OC)C(=O)OCC BTB03651 c1ccc(cc1)c2nc(sn2)N3CCCN(CC3)C(=O)Nc4ccccc4Cl AW00459 Cc1cc(cc(c1)NC(=O)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-])C AW00460 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2ccccc2N BTB06854 Cc1c2ccccc2sc1c3ccnn3C(=O)Nc4ccccc4 MWP00408 COc1ccc(cc1)C(=O)Sc2ccccc2 RJC00234 c1cc(c(cc1OCC(CN2CCCN(CC2)c3nc4ccc(cc4s3)Cl)O)Cl)Cl AW00462 Cc1c(cccc1Cl)NC(=O)N2CCCN(CC2)c3nc(ns3)c4ccccc4 AW00466 CS/C(=N/N=C/c1ccc(cc1)Cl)/N BTB05196 CCCC(C(c1ccccc1)NC(=O)c2ccccc2)O NRB01482 Cc1c2c(n(n1)c3ccccc3)NC(C4=C2CC(CC4=O)(C)C)c5ccc(cc5)N(C)C NRB01474 Cc1c2c([nH]n1)NC(C3=C2CCCC3=O)c4ccc(cc4)N(C)C NRB01476 c1cc(ccc1C(COc2ccc(cc2)F)(c3ccc(cc3)Cl)O)Cl RJC00245 c1ccc(cc1)COC(=O)NCCC(C(=O)O)O NRB01485 CCOC(=O)/C(=C/N/C(=N\N=C\c1ccc2c(c1)OCO2)/SC)/C#N BTB05226 CCOC(=O)/C(=C/N/C(=N\N=C\c1cccs1)/SC)/C#N BTB05227 CC1(CC(=O)c2ccc(cc2O1)OCc3ccccc3F)C RJC00181 Cc1cc(cc2c1C(=O)CC(O2)(C)C)OCc3ccccc3 RJC00185 CC1(NN2C(=N1)C(=CN=C2SC)C#N)c3ccc(cc3)Br BTB05192 c1ccc(c(c1)C(=O)Oc2ccc(cc2)c3ccc(cc3)OC(=O)c4ccccc4Cl)Cl BTB05194 CS/C(=N/S(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)/N/N=C/c4ccc(cc4)Cl BTB06880 c1ccc(c(c1)CN2CCOCC2)C(=O)Nc3cc(ccc3O)Cl BTB03610 CN(C)c1ccc(cc1)/C=N/N=C(\N)/SC BTB05198 c1cc(c(c(c1)F)C(=O)Oc2ccc(cc2)c3ccc(cc3)OC(=O)c4c(cccc4F)F)F BTB05199 COc1ccc(c(c1)C(=O)NN)Br BTB06852 Cc1c(c(n[nH]1)C)/N=N/c2ccc(cc2F)F BTB03540 Cc1ccc(cc1C)n2c(nnc2S)c3c(nn(n3)c4ccccc4)C BTB03587 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl AW00431 Cc1cc(cc(c1)NC(=S)NCCCNC(=O)OC(C)(C)C)C AW00473 c1ccc2c(c1)nc(s2)c3ccc(cc3)CSc4ccc(cc4)Cl BTB03572 c1ccn(c1)c2c(cc(cc2Cl)C(=O)Nc3cc(c(cc3Cl)Cl)Cl)Cl BTB03573 c1cc(sc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)NC(=S)Nc4ccc(cc4)Cl)C(F)(F)F BTB06832 Cc1ccc(cc1)SCc2ccc(cc2)c3nc4ccccc4s3 BTB03595 CC(C)(C)OC(=O)NCCNC(=O)/C=C/C(=O)O AW00406 Cc1ccc(c(c1)C)OS(=O)(=O)c2ccc(s2)c3csc(n3)C AW00432 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCN(CC3)C(=O)OC(C)(C)C AW00408 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCCNC(=O)OC(C)(C)C AW00409 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Oc3ccc(cc3Cl)Cl AW00434 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCCc3ccc(c(c3)OC)OC AW00411 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F AW00412 CC(C)(C)OC(=O)NCC/N=C/c1ccc(cc1Cl)Cl AW00417 c1ccc(cc1)Oc2nc(nc(n2)Oc3ccccc3)Oc4ccccc4 NRB01501 c1ccn(c1)c2c(cc(cc2Cl)C(=O)Nc3ccc(cc3F)F)Cl BTB03574 Cc1ccc(c(c1)N)NS(=O)(=O)c2ccc(cc2)Cl BTB01463 CC(C)(C)OC(=O)N1CCCN(CC1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F AW00439 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Oc3ccc(cc3)Cl AW00443 Cc1c(nn(n1)c2ccccc2)C(=O)OC BTB03578 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Oc3ccccc3Cl AW00450 c1ccc(c(c1)C(F)(F)F)NC(=O)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-] AW00451 COc1ccc(cc1)/C=N/c2[nH]c3ccccc3n2 NRB01493 CCOC(=O)C(C#N)C1(C(=NN(C1=O)c2ccccc2)C)c3c(nn(c3O)c4ccccc4)C NRB01459 c1c(c(sc1Cl)Cl)S(=O)(=O)N BTB06837 c1ccc2c(c1)C(=O)CS(=O)(=O)N2Cc3c(cccc3Cl)F BTB06841 COc1ccc(c(c1)C(=O)NNC(=O)c2ccccc2N)Br BTB06870 COc1cccc(c1)C(=O)NNC(=O)c2ccccc2N BTB06871 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3ccc4c(c3)cn[nH]4 BTB03568 c1cc(c(nc1)N2CCCNCC2)[N+](=O)[O-] AW00446 CC(C)(C)OC(=O)NCC/N=C/c1ccc(cc1)O AW00418 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCc3ccccn3 AW00422 c1cc2c(cc1S(=O)(=O)N)NN(O2)N NRB01507 C/C(=N\N=C(\N=C\N(C)C)/SC)/c1cc2ccccc2o1 BTB05218 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-] AW00454 CC(C)(C)OC(=O)NCC/N=C/c1cccc(c1)[N+](=O)[O-] AW00425 c1cc2c(cc1/C=C/C=C/C(=O)N3CCCCC3)OCO2 NRB01456 C/C(=C\c1cccc(c1)[N+](=O)[O-])/C(=N/O)/C NRB01490 C/C(=N\OC(=O)c1ccc(c(c1)Cl)Cl)/c2ccc(c(c2)F)F BTB06856 C/C(=N\OC(=O)c1ccc(cc1)F)/c2ccc(c(c2)F)F BTB06860 C/C(=N\OC(=O)c1ccccc1F)/c2ccc(c(c2)F)F BTB06861 C/C(=N\OC(=O)c1ccc(cc1)[N+](=O)[O-])/c2ccc(c(c2)F)F BTB06857 c1c(cc(c(c1Cl)N)Cl)C(=O)Nc2cc(cc(c2)Cl)Cl BTB03563 Cc1c2ccccc2sc1c3ccnn3S(=O)(=O)C MWP00417 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)F)c4cccnc4 AW00447 Cc1c2ccccc2sc1c3ccnn3S(=O)(=O)c4ccccc4F MWP00420 CCCCOc1cc(c(cc1[N+](=O)[O-])OCCCC)N2CCOCC2 NRB01523 C/C(=N\OCc1c(cccc1Cl)F)/c2ccc(c(c2)F)F BTB06875 COC(=O)c1ccc(cc1N(Cc2c(cccc2Cl)F)S(=O)(=O)C)Cl BTB06844 COC(=O)c1ccccc1N(Cc2ccc(c(c2)Cl)Cl)S(=O)(=O)C BTB06847 CC(C)c1ccc(cc1)N(CCc2ccccn2)C(=O)C(C)(C)C BTB01676 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2ccc(cc2F)F BTB05283 Cc1cccc(c1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C BTB05297 Cc1c(c(on1)C)/N=N/c2cc(cc(c2)Cl)Cl BTB03545 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3nnc(s3)C(F)(F)F BTB03566 Cc1c(nn(n1)c2ccccc2)C(=O)N BTB03582 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=S)Nc3ccc(cc3)Cl BTB03586 Cc1ccc(cc1C)NC(=S)NNC(=O)c2c(nn(n2)c3ccccc3)C BTB03585 COC(=O)c1ccc(cc1N(Cc2ccccc2)S(=O)(=O)C)Cl BTB06849 C/C(=N\OCc1ccc(cc1)Br)/c2ccc(c(c2)F)F BTB06876 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NS(=O)(=O)c3ccc(cc3)F)C BTB01467 c1ccc(c(c1)CSc2ccc(cc2)Cl)C(=O)Nc3cc(ccc3O)Cl BTB03608 Cc1ccc(cc1)SCc2ccccc2C(=O)Nc3cc(ccc3O)Cl BTB03609 CC1=NN=C(C1=NNc2cc(cc(c2)Cl)Cl)C BTB03547 CC(C)(C)NC(=O)NC(=O)c1c(cccc1Cl)F BTB03559 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NS(=O)(=O)c3ccc(cc3)Cl)C BTB01472 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3ccccc3C(F)(F)F BTB01484 Cc1c2cc(ccc2sc1CC(=O)NNS(=O)(=O)c3ccccc3)Cl MWP00395 c1ccc(cc1)c2nc(cs2)c3cccs3 AW00436 Cc1c(nn(n1)c2ccccc2)C(=O)NN BTB03569 Cc1ccc(c(c1)O)NC(=O)c2ccc(cc2)CSC BTB03571 Cc1c(cccc1Cl)n2c(nnc2S)c3c(nn(n3)c4ccccc4)C BTB03588 c1cc(c(c(c1)F)C(=O)NC(=O)N2CCSC2)F BTB03592 c1ccc2c(c1)cc(s2)C(=O)O CC12201 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)c3nc(ns3)c4ccccc4 AW00428 Cc1c2cc(ccc2sc1C(=O)/C=C/N(C)C)Cl MWP00428 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCc3c(cccc3Cl)F AW00448 Cc1cc(c(c(c1)C)n2c(nnn2)SCc3c(cccc3Cl)F)C AW00449 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3ccc(cc3Cl)Br AW00430 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3ccc(cc3OC)OC AW00433 CC(C)(C)OC(=O)NCCNc1ccc(cc1[N+](=O)[O-])C(F)(F)F AW00435 Cc1ccc(cc1)S(=O)(=O)Oc2cc3c(cc2OS(=O)(=O)c4ccc(cc4)C)OC(CC3=O)(C)C RJC00193 c1cc(ccc1c2coc3cc(cc(c3c2=O)O)O)OC4[C@@H]([C@H]([C@@H]([C@H](O4)CO)O)O)O RJC00214 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2ccc(c(c2)F)F BTB06858 CS/C(=N/S(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)/NNC(=O)Nc4ccccc4 BTB06882 CS/C(=N/S(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)/NNC(=O)Nc4ccc(cc4)Cl BTB06883 Cc1c2cc(ccc2sc1c3ccnn3S(=O)(=O)C)Cl MWP00449 C/C(=N\OC(=O)c1ccc(cc1)C(C)(C)C)/c2ccc(c(c2)F)F BTB06859 CC(C)(C)OC(=O)NCCNc1ccc(cc1N)C(F)(F)F AW00453 CC1(CC(=O)c2c(cc(cc2OS(=O)(=O)c3ccccc3)OS(=O)(=O)c4ccccc4)O1)C RJC00194 c1ccc2c(c1)cc(o2)C(=O)c3ccc(c(c3)F)F BTB06889 CCOC(=O)/C(=C/N/C(=N\N=C(/C)\c1cc2ccccc2o1)/SC)/C#N BTB05224 C/C(=C\c1ccc(cc1)Cl)/C(=N/O)/C NRB01489 c1ccc2c(c1)[nH]c(n2)S(=O)(=O)O NRB01502 c1cc(ccc1NC(=O)NNC(=O)c2csc(n2)Cc3ccsc3)Cl MWP00399 c1cc(ccc1NC(=O)Nc2csc(n2)Cc3ccsc3)[N+](=O)[O-] MWP00403 CCCCCCCCCCCC(=O)Nc1ccc2c(c1)C(=O)C(C2)Sc3nnnn3c4ccccc4 NRB01518 CCC(C)(C)c1ccc(c(c1)C(C)(C)CC)OCCCC(=O)Nc2ccc3c(c2)C(=O)C(C3)Sc4nnnn4c5ccccc5 NRB01519 CCCc1c(nc2cc(c(cc2n1)Cl)Cl)C BTB05247 CCCc1c(nc2cc(c(cc2n1)C)C)C BTB05248 Cc1c(nn(n1)c2ccccc2)c3nnc(n3c4ccc(cc4)Cl)S BTB03589 c1ccc2c(c1)[nH]c(n2)CC#N BTB06788 CCOC(=O)N1CCN(CC1)CC(COc2ccc(cc2)OC(F)(F)F)O AW00361 CCOC(=O)CCC(C#N)(c1ccc(cc1)Cl)N2CCOCC2 BTB03489 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCS(=O)(=O)c3ccccc3 BTB03496 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)Cl)N BTB06865 Cc1ccc(cc1)S(=O)(=O)O/N=C(\C)/c2ccc(c(c2)F)F BTB06869 Cc1c2ccccc2sc1C(=O)/C=C/N(C)C MWP00405 COc1ccc(cc1)C(=O)/C(=N\O)/c2ccccc2 NRB01484 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)Cl)[N+](=O)[O-] BTB06909 c1ccc(c(c1)C(=O)NC(=O)N2CCSC2)Cl BTB03590 c1cc(c(c(c1)Cl)C(=O)NC(=O)N2CCSC2)Cl BTB03591 CN(C)/C=C/1\C(=O)c2ccc(cc2N(S1(=O)=O)Cc3c(cccc3Cl)F)Cl BTB06912 c1ccc2c(c1)CCN=C2SCC(=O)c3ccc(cc3)Cl.Br MWP00441 COc1ccccc1/C=C/2\Cc3ccccc3C2=O RJC00121 COc1ccc(cc1)/C=C/2\CSc3ccccc3C2=O RJC00150 Cc1c(s/c(=N\c2ccccc2)/n1c3ccccc3)C BTB05140 Cc1cs/c(=N\c2ccccc2)/n1c3ccccc3 BTB05141 Cc1cc(c(c(c1)C)/N=C\2/N(C3(CCCCC3)C(=C)S2)C(=O)c4c(cccc4F)F)C BTB01544 Cc1cc(c2ccccc2n1)Oc3ccc(cc3)OC BTB05231 CCOC(=O)/C(=C/N/C(=N\N=C(/C)\c1ccc(cc1)F)/SC)/C#N BTB05225 Cc1c(cccc1Cl)NC(=S)NNC(=O)c2c(nn(n2)c3ccccc3)C BTB03584 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2ccccc2[N+](=O)[O-] BTB06910 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)F)F BTB01526 CCC(CC)(C#C)NC(=O)NC(=O)c1ccccc1Cl BTB05251 CCOC(=O)c1c([nH]c2c1cc(cc2)O)C BTB01488 c1ccc(cc1)c2c3cc(ccc3nc(c2C#N)N)Cl BTB01516 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)Nc2ccc(c(c2)Cl)F)F BTB05161 Cc1cc(ccc1Cl)OCOc2ccc(c(c2)C)Cl BTB05165 CC(C)(C)c1csc(n1)N/N=C/c2c(cccc2Cl)Cl.Br BTB05167 CCOC(=O)c1ccc(cc1)N2CC3CCCCN3C2c4ccc(cc4)Cl BTB01350 c1cc(c(c(c1)Cl)Oc2ccc(cc2)c3ccc(cc3)Oc4c(cccc4Cl)[N+](=O)[O-])[N+](=O)[O-] BTB05232 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2F)F)F BTB01527 CCc1ccc(cc1C)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05235 CCc1ccc(cc1CC)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05236 CCc1c(nc2cc(c(cc2n1)Cl)Cl)CC BTB05243 COc1cccc(c1)/N=C\2/N(C3(CCCCC3)C(=C)S2)C(=O)c4c(cccc4F)F BTB01543 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN=C3SC BTB03622 c1ccc(cc1)c2ccc(cc2)C(=O)CSC3=NCCc4c3cccc4.Br MWP00444 Cc1c2cc(ccc2sc1c3ccnn3C(=O)C)Cl MWP00445 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NC(=S)NCCCOC)C BTB01478 Cn1c(nnc1SCc2ccccc2Cl)c3csc(n3)c4cccnc4 MWP00432 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)N4CCOCC4)Cl BTB01386 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)N4CCOCC4 BTB01387 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)Nc2ccc(cc2F)F)F BTB05130 c1cc(ccc1S(=O)(=O)Nc2ccc(cc2Cl)[N+](=O)[O-])Cl BTB01383 Cc1c2cc(ccc2sc1/C(=N/OC(=O)C)/C)Cl MWP00320 Cc1c2cc(ccc2sc1/C(=N/OC(=O)c3ccccc3)/C)Cl MWP00321 C=C1C2(CCCCC2)N(/C(=N/c3ccccc3Cl)/S1)C(=O)c4c(cccc4F)F BTB01541 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CCC(=O)O BTB03643 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccccc3N BTB03645 CN(C)/C=C/C(=O)c1ccc(cc1Cl)[N+](=O)[O-] MWP00465 Cc1ccccc1NC(=O)COc2ccc3c(c2)OC(CC3=O)(C)C RJC00195 CC1(CC(=O)c2ccc(cc2O1)OCC(=O)Nc3ccc(cc3)Br)C RJC00196 CC(C)(C)C1OC(C(O1)C(c2ccccc2)(c3ccccc3)O)C(c4ccccc4)(c5ccccc5)O RJC00228 COc1ccc(cc1)c2c(=O)c3ccc(cc3oc2c4ccccc4)O RJC00212 Cc1c2cc(ccc2sc1/C(=N/OC(=O)c3ccccc3Cl)/C)Cl MWP00322 Cc1c2cc(ccc2sc1/C(=N/OC(=O)c3ccc(cc3)C(F)(F)F)/C)Cl MWP00323 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)N4CCOCC4 BTB01388 Cc1c2cc(ccc2sc1/C(=N/OC(=O)Nc3ccccc3)/C)Cl MWP00318 c1cc(cc(c1)Cl)C(=O)Nc2ccc3c(c2)nn[nH]3 BTB01509 COc1cc(cc(c1OC)OC)COc2ccc(cc2)[N+](=O)[O-] BTB01513 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)NC(=S)S2 BTB01514 Cc1c2ccccc2sc1c3ccnn3C(=O)c4ccc(cc4)C(F)(F)F MWP00414 Cc1ccc(cc1C)NC(=O)C BTB05228 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05281 CSc1ncc(c2n1nc(n2)c3ccc(cc3)Cl)C#N BTB05282 Cc1ccc2c(c1)c(=O)n(c(n2)c3c(c4ccccc4s3)Cl)c5cc(cc(c5)C(F)(F)F)C(F)(F)F BTB01535 c1ccc(cc1)c2c(=O)c3c(cc(cc3oc2c4ccccc4)O)O RJC00213 c1cc(ccc1c2ccc(cc2)OS(=O)(=O)c3ccc(c(c3)Cl)Cl)OS(=O)(=O)c4ccc(c(c4)Cl)Cl BTB05211 CC(C)c1ccc(cc1)/C=C/2\CSc3ccccc3C2=O RJC00151 c1ccc2c(c1)c(c[nH]2)/C=C/3\CSc4ccccc4C3=O RJC00155 CSC1=NC=C(C2=NC(NN21)c3ccc(cc3)Cl)C#N BTB05200 CCOC(=O)/C(=C/N/C(=N\N=C\c1c(cccc1Cl)F)/SC)/C#N BTB05203 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Oc2ccc(c(c2)O)C(=O)Cc3ccccc3)OC(=O)C)OC(=O)C)OC(=O)C RJC00204 c1ccc(c(c1)NC(=O)NC(=O)c2c(cccc2Cl)Cl)N3CCCCC3 BTB03549 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3cc(cc(c3)Cl)Cl BTB03565 Cc1c(nn(n1)c2ccccc2)C(=O)Sc3ccc(cc3)Cl BTB03567 c1ccc(cc1)c2coc3cc(ccc3c2=O)O RJC00206 COC(=O)c1ccccc1N(Cc2c(cccc2Cl)F)S(=O)(=O)C BTB06833 c1ccn(c1)c2c(cc(cc2Cl)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl BTB03575 CC(C)(C)OC(=O)NCCNC(=O)Nc1ccccc1 AW00399 CC(C)(C)OC(=O)NCCNC(=S)NC1CCCCC1 AW00400 Cc1cccc(c1NC(=S)NCCNC(=O)OC(C)(C)C)Cl AW00404 CS/C(=N/N=C/c1ccc2c(c1)OCO2)/N BTB05213 CS/C(=N/N=C/c1cccs1)/N BTB05216 Cc1ccc(cc1)S(=O)(=O)n2c3ccc(cc3[nH]c2=S)C BTB01479 CCOC(=O)/C(=C/N/C(=N\N=C\c1ccc(cc1)Cl)/SC)/C#N BTB05204 Cc1c(c(on1)C)/N=N/c2ccc(cc2F)F BTB03544 c1cc(c(c(c1)Cl)C(=O)NC(=O)N2CCSC2)F BTB03593 C/C(=N\N=C(\N)/SC)/c1cc2ccccc2o1 BTB05217 c1ccc2c(c1)c(c(s2)C(=O)N(c3cccc(c3)Cl)c4nc5ccccc5s4)Cl BTB01454 CC(C)(C)OC(=O)NCC/N=C/c1ccc(cc1)Cl AW00405 CN(C)/C=N/C(=N\N=C\c1c(cccc1Cl)F)/SC BTB05207 c1ccc2c(c1)nc(s2)N(c3cccc(c3)Cl)C(=O)c4ccc(cc4)[N+](=O)[O-] BTB01458 CC1CN(CC(O1)C)C(C#N)c2c(cccc2Cl)F BTB03577 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3c(cccc3Cl)Cl BTB03579 c1ccc2c(c1)cc(s2)C(=O)Oc3ccc(cc3)c4ccc(cc4)OC(=O)c5cc6ccccc6s5 BTB05209 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3ccc(cc3)Cl BTB03580 Cc1ccc(cc1NC(=O)c2ccccc2Cl)NC(=O)C BTB01568 Cc1ccc(c(c1)N)NC(=O)c2ccccc2N BTB01591 c1cc(ccc1C(=O)CSCC(=O)c2ccc(cc2)Br)Br BTB03676 c1cc(ccc1Oc2ccc(cn2)[N+](=O)[O-])Cl BTB03685 c1ccc(c(c1)C(=O)Nc2ccc(cc2[N+](=O)[O-])Cl)[N+](=O)[O-] BTB01602 Cc1c2cc(ccc2sc1c3ccnc(n3)SCc4ccc(cc4)F)Cl MWP00475 CS/C(=C(\C#N)/C(=O)N)/N(CC=C)CC=C RJC00273 CC(C)NC(=O)c1ccccc1Sc2ccccc2 RJC00285 Cc1ccc(cc1)OCC(=O)O RJC00256 c1cc2c(=O)c3cc(ccc3oc2nc1)NC(=O)c4ccc(cc4)[N+](=O)[O-] BTB05308 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3Cl)[N+](=O)[O-] BTB03658 c1cc(cnc1)c2nc(cs2)C(=O)O CC13701 Cc1ccc(cc1)NC(=O)c2csc(n2)c3cccnc3 MWP00504 Cc1ccc(cc1Cl)NC(=O)Cc2ncon2 BTB05291 c1c(cc(cc1Cl)Cl)NC(=O)Cc2ncon2 BTB05294 c1cc(cnc1)c2nc(cs2)C(=O)Nc3ccc(cc3Cl)Cl MWP00505 c1ccc(cc1)OC(=O)c2csc(n2)c3cccnc3 MWP00508 c1cc(cc(c1)C(F)(F)F)C(=O)C=C2SCCS2 RJC00312 CSc1ccc(cc1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05299 CC(C)C(C(c1ccccc1)(c2ccccc2)O)N RJC00278 c1c2c(cc(c1F)Cl)nc([nH]2)S BTB03700 c1cc(sc1)C(=O)O/N=C(/CC(=O)Nc2ccc(c(c2)Cl)F)\N BTB05310 C1CCN(CC1)CCC2CCCCN2.Cl.Cl BTB01616 c1c(cc(cc1C(F)(F)F)NC(=S)N2CCCCC2CCN3CCOCC3)C(F)(F)F BTB01736 c1cc(c(cc1Cl)NC(=S)N2CCCCC2CCN3CCOCC3)Cl BTB01737 CC1(C(=C)S/C(=N\c2cccc(c2)OC)/N1C(=O)C(c3ccccc3)C4CCCC4)C BTB01585 c1cc(c(cc1F)F)NC(=O)Cc2ncon2 BTB05295 c1ccc(cc1)C(=O)Cc2nc(cs2)O BTB05321 Cc1c(cccc1Cl)NC(=O)N2CCCN(CC2)Cc3c(cccc3Cl)F AW00528 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)Cc3ccc(cc3Cl)Cl AW00533 Cc1ccc(c(c1)C2=NN(C(O2)c3ccc(cc3)N(C)C)C(=O)C)[N+](=O)[O-] BTB01705 Cc1ccc(cc1)S(=O)(=O)N2CN3CCN(C3)C2 BTB01773 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3cccc(c3)[N+](=O)[O-])Cl MWP00545 Cc1ccc(cc1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05303 COc1ccccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05304 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SC AW00534 c1ccc2c(c1)cc(c3c(c2=O)ccs3)Br NRB01587 Cc1ccc(cc1)S(=O)(=O)NNC(=S)NCc2ccccc2 BTB01723 c1ccc(cc1)SC(=O)c2csc(n2)c3cccnc3 MWP00510 Cc1c2cc(ccc2sc1C(=O)CSc3ccc(cc3)Cl)Cl MWP00513 c1ccc2c(c1)c(c(s2)C(=O)NCCc3ccccn3)Cl BTB01610 CC1C(Sc2ccccc2NC1=O)C RJC00306 Cc1c2cc(ccc2sc1c3ccnc(n3)SCc4ccccc4Cl)Cl MWP00473 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCCNC(=O)OC(C)(C)C AW00472 Cc1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)NC(=O)c3ccccc3/N=C/c4cc(cc(c4O)Cl)Cl BTB01594 CC(C)(C)C(=O)Nc1c(c(cc(c1Cl)Cl)Cl)Cl BTB01595 Cc1ccc(c(c1)C)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05302 c1ccc(cc1)CC(C#N)Sc2ccccc2 NRB01568 c1ccc(cc1)[S+](CC#N)[O-] NRB01569 CCc1cc(c(c(c1)CC)NC(=O)C(C)(C)C)CC BTB01598 Cc1c2cc(ccc2sc1S(=O)(=O)N(C)c3ccccc3)Cl MWP00549 Cc1ccc(cc1)CSc2nccc(n2)c3c(c4cc(ccc4s3)Cl)C MWP00474 Cc1c2cc(ccc2sc1c3ccnc(n3)SCC#C)Cl MWP00476 c1ccc(cc1)/C=C/2\CCCC(C2=O)CN3CCOCC3.Cl NRB01540 CS/C(=C(\C#N)/C(=O)N)/NCC=C RJC00272 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)c(=O)c4cccnc4o3 BTB05317 Cc1cc(c(cc1Cl)C)SCC(=O)c2c(c3cc(ccc3s2)Cl)C MWP00516 c1cc(oc1)c2ccnc(n2)SCC(=O)Nc3cc(cc(c3)Cl)Cl MWP00524 CC(C)(C)OC(=O)NCCC/N=C/c1ccc(cc1)C(F)(F)F AW00474 c1ccc2c(c1)c(=O)c(co2)C3CC(=O)Nc4ccccc4S3 RJC00309 Cc1c2cc(ccc2sc1c3ccnc(n3)SCC=C)Cl MWP00477 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2c(c(cc(c2Cl)Cl)Cl)Cl BTB01600 c1ccc(c(c1)C(=O)Nc2ccc(cc2N)Cl)N BTB01603 c1cc(c(nc1)Sc2nccc(n2)c3ccco3)[N+](=O)[O-] MWP00528 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCC=C AW00477 CC1CC(=O)N(c2ccccc2S1(=O)=O)C RJC00325 c1cc(cnc1)c2nc(cs2)C(=O)Sc3ccc(cc3)Cl MWP00509 c1ccc(cc1)C(=O)N/N=C\2/c3ccccc3NC2=O RJC00255 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN=C3SC BTB03623 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN=C3SC BTB03624 c1ccc(cc1)CCC(CCN2CCCCC2)(c3ccccc3)O.Cl RJC00262 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCCN=C3SC BTB03626 c1cc(ccc1NC(=S)N2CCCCC2CCN3CCOCC3)F BTB01739 CSC1=NC=C(C2=NC(NN21)c3ccc4c(c3)OCO4)C#N BTB05287 CS(=O)(=O)Nc1ccc2c(c1)c(=O)c3cccnc3o2 BTB05324 CSc1cc(=O)c2ccccc2s1 RJC00282 c1ccc(cc1)CN2c3cc(ccc3C(=O)CS2(=O)=O)Cl BTB06908 Cc1cccc(c1)C(=O)Nc2ccccc2c3nnc(o3)c4ccc(c(c4)Cl)Cl BTB06944 c1cc(ccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl BTB05288 Cc1cc(ccc1Cl)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05289 c1ccc(c(c1)NC(=O)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-])Cl AW00461 c1cc2c(cc1F)C(=O)C(=O)N2 BTB01627 c1cc(sc1)/C=C(\C#N)/c2csc3c2cc(cc3)Cl BTB01633 CCOC(=O)C1=C(/C(=N\O)/NC1=O)SC RJC00284 Cc1ccc2c(c1)nc-3c(n2)C(=O)c4c3cccc4 BTB05340 COC(=O)C/C(=N\NC(=O)c1cccs1)/C(=O)OC BTB03640 Cc1ccc(c(c1)C2=NN(C(O2)c3cc(c(c(c3)OC)OC)OC)C(=O)C)[N+](=O)[O-] BTB01706 c1ccnc(c1)CCN/N=C/c2cc(cc(c2O)Cl)Cl BTB01718 CCOC(=O)COc1c(cc(cc1Br)/C=N/NC(=S)Nc2cc(ccc2Cl)Cl)Br AW00484 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCc3cc(cc(c3)F)F AW00476 Cn1c(nnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)c3csc(n3)Cc4ccsc4 MWP00533 c1ccc2c(c1)c(c(s2)C(=O)NCC(=O)O)Cl BTB01608 CC1CC(=O)Nc2ccccc2S1 RJC00303 c1ccc(cc1)C(=O)n2c(ccn2)c3ccc(cc3Cl)[N+](=O)[O-] MWP00469 Cc1c2cc(ccc2sc1c3cc(n(n3)C)NC(=O)c4ccccc4)Cl MWP00567 c1ccc(cc1)/C=C/2\CCCC(C2=O)CN3CCCCC3.Cl NRB01539 Cc1ccc(cc1Cl)NC(=O)C/C(=N/O)/N BTB05273 c1cc(c(cc1C(F)(F)F)NC(=O)C/C(=N/O)/N)Cl BTB05274 COC(=O)c1c(c2ccccc2s1)OC(=O)c3ccccc3Cl BTB05263 c1ccc(cc1)C(Sc2ccc(cc2)Cl)Sc3ccc(cc3)Cl NRB01560 COc1ccc(cc1OC)S(=O)(=O)Oc2c3ccccc3sc2C(=O)OC BTB05278 COc1ccc(cc1)C(COc2ccc(cc2)Br)(c3ccc(cc3)OC)O RJC00250 CN(C)C(=S)SCC#N NRB01563 c1ccc(cc1)C(Sc2ccccc2)Sc3ccccc3 NRB01562 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCC#C AW00479 Cc1cccc(c1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl BTB05255 C/C(=C\1/C(=O)NC(=S)S1)/c2cccc(c2)[N+](=O)[O-] BTB01730 CSC1=NC=C(C2=NC(NN21)c3c(cccc3Cl)F)C#N BTB05285 Cc1cccc(c1NC(=O)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-])Cl AW00456 COC(=O)c1c(c2ccccc2s1)OS(=O)(=O)c3ccc(cc3)Cl BTB05276 CN1c2ccccc2C(C1=O)(Cc3ccccc3)c4ccccc4 NRB01543 Cc1cccc(c1)C(=O)Nc2ccccc2c3nnc(o3)c4ccc(cc4)C(C)(C)C BTB06921 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCCN=C3SC BTB03628 c1ccc(cc1)C(COc2ccc(cc2)F)(c3ccccc3)O RJC00252 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SC(=O)c3ccc(cc3)Cl AW00475 COc1ccc(c(c1)c2nnc(o2)c3ccccc3N)Br BTB06952 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)NC(=O)c4ccc(cc4)Cl BTB06905 c1c(cc(c2c1[nH]cn2)Br)C(F)(F)F BTB05258 Cc1cc(ccc1Cl)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05262 Cc1cccc(c1)C(=O)Nc2ccccc2c3nnc(o3)c4cc(ccc4Br)OC BTB06955 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3[N+](=O)[O-] BTB06915 Cc1ccc(cc1)S(=O)(=O)Oc2c3ccccc3sc2C(=O)OC BTB05268 Cc1nc(c(o1)c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3)S(=O)(=O)N/N=C/c4ccco4 NRB01533 c1c(cc(cc1Cl)Cl)NC(=O)C/C(=N/O)/N BTB05272 Cc1nc(c(o1)c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3)S(=O)(=O)NN NRB01536 COc1cccc(c1)C(=O)NNC(=O)c2ccccc2[N+](=O)[O-] BTB06940 CCCCc1ccc(c(c1)C)NC(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00483 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCCCN AW00509 c1ccc(cc1)c2nc(sn2)N3CCCN(CC3)C(=O)Nc4ccc(cc4F)F AW00464 CN(C)/C=C/1\C(=O)c2ccccc2N(S1(=O)=O)Cc3ccc(c(c3)Cl)Cl BTB06907 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)NC(=O)c4ccc(cc4)C(F)(F)F BTB06924 c1cc(ncc1Br)NC(=O)CCC(=O)O BTB03647 c1ccc(c(c1)c2nnc(o2)c3ccc(c(c3)Cl)Cl)NC(=O)c4ccc(cc4)Cl BTB06942 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)[N+](=O)[O-] BTB06916 CCCCCC(=O)Nc1ccccc1c2nnc(o2)c3ccc(cc3)C(C)(C)C BTB06919 CN(C)/C=C/1\C(=O)c2ccccc2N(S1(=O)=O)Cc3c(cccc3Cl)F BTB06913 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)NC(=O)Nc4ccc(cc4)Cl BTB06931 Cc1ccc(cc1NC(=O)c2ccncc2)C(=O)OC BTB03650 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2ccc(c(c2)F)F BTB06862 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccc(c(c2)F)F BTB06863 COc1cccc(c1)C(=O)NN BTB06864 C#CC1(CCCCC1)NC(=O)NC(=O)c2ccccc2Cl BTB05252 Cc1ccc(c(c1)O)NC(=O)c2ccc(cc2)CSc3ccccn3 BTB03596 CN1c2ccccc2C(C1=O)(Cc3ccccc3)Cc4ccccc4 NRB01544 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3ccc(c(c3)C(F)(F)F)Br AW00482 Cc1c(c(nc(n1)SCC(=O)c2cccs2)O)CC=C AW00486 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)c3cccs3)C AW00487 c1cc(c(cc1Br)/C=C\2/C(=O)NC(=S)S2)O BTB01745 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccccc3CC4c5ccccc5CCN4C BTB01767 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-] AW00455 c1c(cc(cc1F)F)NC(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW00491 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F AW00489 COc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05265 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(c3cccc(c3)Cl)c4nc5ccccc5s4 BTB01452 Cc1ccc(cc1)SCc2ccc(cc2)C(=O)Nc3ccc(cc3O)C BTB03597 Cc1ccc(c(c1)[N+](=O)[O-])NS(=O)(=O)c2ccc(cc2)Cl BTB01456 c1cc(c(c(c1)F)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F BTB01524 CCOC(=O)C(=CNc1ccccc1c2nnc(o2)c3ccc(cc3)Cl)C(=O)OCC BTB06946 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)NC(=O)CCC(=O)O BTB06949 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)NC(=O)c4ccccc4Cl BTB06923 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)Nc4ccccc4 BTB06968 c1cc(c(cc1C(F)(F)F)NC(=O)Cc2ncon2)Cl BTB05292 c1cc(ccc1NC(=O)Cc2ncon2)F BTB05293 CN(C)C(=S)SCC(=O)OC NRB01564 COc1ccc(c(c1)c2nnc(o2)c3ccccc3NC(=O)c4ccc(cc4)C(F)(F)F)Br BTB06953 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3c4ccccc4sc3C(=O)OC BTB05267 COC(=O)c1c(c2ccccc2s1)OC(=O)c3cccnc3Oc4ccccc4 BTB05269 CN(C)c1ccc(cc1)c2nc3c(cnc(n3n2)SC)C#N BTB05284 CC(C)C(c1c2ccccc2ccn1)OC(=O)c3ccccc3 NRB01552 c1cc(cc(c1)NC(=O)c2c(cccc2F)F)C(F)(F)F BTB01525 Cc1c(c(no1)c2ccccc2)C(=O)N3CCCN=C3SC BTB03627 CC1CC(CN(C1)/C(=N/S(=O)(=O)c2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4)/SC)C BTB06970 c1cnccc1C(=O)Nc2nncs2 BTB03653 c1cnccc1C(=O)Nc2nccs2 BTB03655 Cc1ccc(cc1)C(c2c3ccccc3ccn2)O NRB01550 COc1cccc(c1)c2nnc(o2)c3ccccc3[N+](=O)[O-] BTB06945 CCc1nnc(s1)NC(=O)c2ccncc2 BTB03654 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3N BTB06917 CC(=O)Nc1ccccc1c2nnc(o2)c3ccc(cc3)C(C)(C)C BTB06922 COc1ccc(c(c1)c2nnc(o2)c3ccccc3NC(=O)Nc4ccc(cc4)Cl)Br BTB06957 c1ccc(c(c1)c2nnc(o2)c3ccc(c(c3)Cl)Cl)[N+](=O)[O-] BTB06934 c1cc(ccc1C(=O)CSCC(=O)c2ccc(cc2)[N+](=O)[O-])[N+](=O)[O-] BTB03680 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCCN=C3C BTB03629 COC(=O)C/C(=N\NC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C(=O)OC BTB03638 Cc1c2cc(ccc2sc1CC(=O)NNC(=O)c3ccc(cc3)C(F)(F)F)Cl MWP00392 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F BTB05253 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCC(=O)c3cccs3 AW00485 Cc1cc(=O)[nH]c(n1)SCC#C RJC00290 CCOC(=O)C(=CNc1ccc(cn1)Br)C(=O)OCC BTB03659 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(c(c2)Cl)Cl)[N+](=O)[O-] BTB06933 c1cc(ccc1NC(=S)N2CCCN(CC2)Cc3ccc(cc3Cl)Cl)F AW00519 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)[N+](=O)[O-] BTB03687 c1cc(c(c(c1)Cl)Oc2ccc(cn2)[N+](=O)[O-])Cl BTB03688 Cc1cc(cc(c1Cl)C)Oc2ccc(cn2)[N+](=O)[O-] BTB03689 Cc1ccc(c(c1)C)NC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW00494 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3ccc(cc3)F BTB01486 CCOC(=O)C1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] BTB01503 c1cc(c(c(c1)Cl)Cl)n2ccnc2SCc3c(cccc3Cl)F AW00467 Cc1c(cccc1Cl)/N=C\2/N(C3(CCCCC3)C(=C)S2)C(=O)c4c(cccc4F)F BTB01540 COC(=O)c1c(c2ccccc2s1)OS(=O)(=O)c3ccc(c(c3)Cl)Cl BTB05279 Cc1cc(cc(c1Cl)C)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05280 c1cc(ccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])F BTB05290 Cc1ccc(cc1NC(=S)Nc2ccc(c(c2)Cl)Cl)NC(=O)C BTB01563 c1ccc(cc1)C(=C2C=CC=C2)c3ccccc3 RJC00230 CC(C)(C)OC(=O)N1CCCN(CC1)C(=S)Nc2cccc(c2)C(F)(F)F AW00490 c1cc(c(cc1Cl)Cl)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05296 C1CC2(CCC1C(C2C(=O)O)C(=O)O)Br NRB01684 c1ccc(cc1)n2c(=O)n3n(c2=O)C4CC3C=C4 RJC00239 c1ccc2c(c1)c(=O)n(c(n2)SCC(=O)c3cccs3)c4cccnc4 AW00497 Cc1ccccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05300 c1cc(cc(c1)[N+](=O)[O-])/C=C\2/C(=O)NC(=S)S2 BTB01682 Cc1ccc(c(c1)C(=O)N/N=C/c2ccc(cc2)N(C)C)[N+](=O)[O-] BTB01688 c1cc2c(cc1CO)OCO2 CC01609 Cc1cc(cc(c1C)C)/N=C\2/N(C(C(=C)S2)(C)C)C(=O)c3c(cccc3F)F BTB01542 Cc1c(c(n[nH]1)C)/N=N/c2ccc(cc2Cl)Cl BTB03541 CS/C(=N\S(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)/N4CCCCC4 BTB06962 Cc1ccc(cc1NC(=S)Nc2ccc(cc2C)Cl)NC(=O)C BTB01565 Cc1ccc(cc1NS(=O)(=O)c2cc(ccc2Cl)Cl)NC(=O)C BTB01566 c1ccc2c(c1)nc(s2)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB01592 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)Nc4ccc(cc4)Cl BTB06969 C[C@H]1CC[C@H](CC1)NC(=O)C NRB01687 c1ccc(c(c1)C2=Nc3ccccc3SC(C2)c4ccc(cc4)[N+](=O)[O-])O RJC00354 Cc1c2ccccc2sc1/C=C/c3ccnc(n3)SC MWP00648 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)NC(=O)/C=C/C(=O)O BTB06947 COc1ccc(c(c1)c2nnc(o2)c3ccccc3NC(=O)c4ccc(cc4)Cl)Br BTB06956 Cc1ccc(c(c1)C(=O)NNC(=N)c2ccccn2)[N+](=O)[O-] BTB01692 Cc1ccc(cc1NS(=O)(=O)c2cccc(c2)C(F)(F)F)NC(=O)C BTB01569 c1ccc2c(c1)cc(s2)C(=O)Nc3ccc4c(c3)c(=O)c5cccnc5o4 BTB05307 c1ccc(cc1)c2ccc(cc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB05309 COc1ccc(c(c1)c2nnc(o2)c3ccccc3NC(=O)NC(=O)c4ccccc4Cl)Br BTB06958 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2ccccc2c3nnc(o3)c4ccc(cc4)C(C)(C)C BTB06966 c1ccc2c(c1)CCN=C2SC(=O)c3ccc(cc3)Cl MWP00479 CC(=O)N1c2ccccc2SC(CC1=O)c3ccccc3 RJC00315 c1ccc(cc1)n2c(=O)cc(c3c2CCCCC3)O NRB01624 c1cc(ccc1CN2CCCN(CC2)C(=S)Nc3ccc(cc3)Cl)F AW00521 c1cc(ccc1CN2CCCN(CC2)C(=S)Nc3ccc(cc3)F)F AW00522 c1ccc(cc1)C2C3CSc4ccccc4C3=Nc5ccccc5S2 RJC00334 C1[C@H](C2CC1C[C@H]2O)C(=O)O NRB01951 c1ccc2c(c1)NC(=O)CC(S2)c3cccc(c3)Br RJC00310 c1cc(c(c(c1)Cl)CN2CCCN(CC2)C(=S)NC3CCCCCCC3)F AW00525 Cc1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccccc4 RJC00339 Cc1c2ccccc2sc1/C=C/c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(C)C MWP00649 CCC(=O)N1c2ccccc2N=C(CC1c3ccccc3)c4ccccc4 RJC00381 CC(CC(=O)O)Oc1ccccc1[N+](=O)[O-] RJC00383 COc1ccc(cc1OC)S(=O)(=O)Nc2ccc3c(c2)c(=O)c4cccnc4o3 BTB05325 CC1CCN(CC1)/C(=N/S(=O)(=O)c2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4)/SC BTB06971 c1ccc(cc1)C2CC(=Nc3ccccc3N2)c4ccc(cc4)OCC(=O)Nc5ccccc5 RJC00378 Cc1cc2c(cc1C)nc3c(n2)-c4ccccc4C3=O BTB05331 Cc1ccc(cc1)S(=O)(=O)O/N=C(/CC(=O)Nc2cc(ccc2Cl)C(F)(F)F)\N BTB05316 CCNC(=S)NNC(=O)c1c(nc2n1cccc2)C NRB01598 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccccc2c3nnc(o3)c4cccc(c4)OC BTB06978 Cc1ccc(c(c1)C)n2c(nnn2)SCc3c(cccc3Cl)F AW00538 Cc1ccc(cc1)Cc2c(nc(nc2O)SCc3c(cccc3Cl)F)C AW00541 Cc1ccc(=O)n(n1)Cc2ccccc2 BTB06988 Cc1ccc(=O)n(n1)Cc2ccc(cc2)F BTB06987 c1cc(cnc1)c2ccnc(n2)Sc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] MWP00601 c1cc(cnc1)c2ccnc(n2)SCc3ccc(cc3)C(F)(F)F MWP00582 c1ccc(cc1)CSc2nccc(n2)c3cccnc3 MWP00583 c1cc(c(c(c1)Cl)CSc2nccc(n2)c3cccnc3)Cl MWP00584 c1cc(cc(c1)NC(=S)N2CCCCC2CCN3CCOCC3)C(F)(F)F BTB01738 CSc1cccc(c1)NC(=S)N2CCCCC2CCN3CCOCC3 BTB01740 c1cc(sc1)/C=C\2/C(=O)NC(=S)S2 BTB01742 c1ccc2c(c1)-c3c(nc4ccc(cc4n3)C(F)(F)F)C2=O BTB05333 c1ccc(cc1)C2C3COc4ccccc4C3=Nc5ccccc5S2 RJC00333 c1ccc(cc1)C2=Nc3ccccc3SC(C2)c4ccc(cc4Cl)Cl RJC00337 c1cc(cc(c1)F)/N=C/c2ccc3c(c2)OCO3 BTB01763 CN(C)/C=N/S(=O)(=O)c1cc(c(c(c1)Cl)Oc2ccc(cc2)[N+](=O)[O-])Cl BTB05374 COc1ccc(c2c1nc-3c(n2)C(=O)c4c3cccc4)OC BTB05336 C/C(=N\Nc1nc[nH]n1)/c2ccc(c(c2)Cl)Cl BTB05338 Cc1c2cc(ccc2sc1c3cc(n(n3)C)N4C(=O)c5ccccc5C4=O)Cl MWP00575 Cc1ccc(c(c1)c2nnc(n2c3cccc(c3)Cl)S)[N+](=O)[O-] BTB01712 CC1CC(=S)Nc2ccccc2S1 RJC00328 c1ccc(cc1)C2CC(=S)Nc3ccccc3S2 RJC00330 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2ccc(cc2)F)C#N BTB05362 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2cc(cc(c2)Cl)Cl)C#N BTB05364 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2ccc(c(c2)Cl)F)C#N BTB05366 c1ccc(cc1)C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 NRB01627 c1ccc(cc1)C2C3CCc4ccccc4C3=Nc5ccccc5S2 RJC00332 C1C2CC3(CC1CC(C2)(C3)Cl)C(=O)O NRB01947 c1cc(ccc1C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])F BTB05344 Cc1ccc(cc1)S(=O)(=O)NNC(=S)NCCCOC BTB01724 CN(C)CCS(=O)(=O)C.Br NRB01954 CCCCCCCCCCCCCCCC#CCO NRB01971 c1cc(cc(c1)C(F)(F)F)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05357 CN(C)C(=O)/C=C/c1ccccc1 NRB01986 c1cc(c(c(c1)Cl)CSc2nnc(o2)c3cn4cc(cc(c4n3)Cl)C(F)(F)F)F AW00543 c1cc(c(c(c1)Cl)CSc2nccn2c3cccnc3)F AW00545 CCOC(=O)c1c2c(sc1N)CN(CC2)Cc3ccccc3 AW00552 c1cc(sc1)C(=O)O/N=C(/CC(=O)Nc2ccc(cc2)F)\N BTB05334 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)CCC(=O)O BTB06974 COc1cccc(c1)c2nnc(o2)c3ccccc3N BTB06976 c1cc(sc1)C(=O)O/N=C(/CC(=O)Nc2cc(ccc2Cl)C(F)(F)F)\N BTB05335 c1ccc(cc1)Cn2c3ccccc3c4c(c2=O)c(cc(=O)o4)O NRB01639 c1ccc(cc1)C2=Nc3ccccc3SC(C2)c4ccccc4Cl RJC00336 COc1cc(cc(c1)NC(=O)C(c2ccccc2)C3CCCC3)C(F)(F)F BTB01788 c1ccc2c(c1)C(=O)NCC(=O)N2 BTB01794 c1cc(ccc1/C=N/Nc2nc[nH]n2)Cl BTB05359 c1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccc(cc4)O RJC00346 COc1ccc(cc1)C2=Nc3ccccc3SC(C2)c4ccccc4 RJC00347 Cc1cc(c2cc(ccc2n1)Br)C(=O)N/N=C/c3cccc(c3O)OC BTB01805 Cc1ccc(cc1[N+](=O)[O-])Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05329 c1cc(c(c(c1)Cl)Oc2ccc(cc2)S(=O)(=O)N)[N+](=O)[O-] BTB05330 Cc1ccc2c(c1)C(=O)C(C(=O)N2)(c3ccccc3)O NRB01609 Cc1ccc(cc1NC(=S)NCCNc2nccc(n2)C(F)(F)F)Cl AW00547 c1ccc2c(c1)c(c(s2)C(=O)N(c3cc(cc(c3)C(F)(F)F)C(F)(F)F)c4nc5ccccc5s4)Cl BTB01841 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCCC2 BTB01842 Cc1ccc(c(c1)C(=O)NNC(=S)Nc2cccc(c2)Cl)[N+](=O)[O-] BTB01708 CC1C/C(=N\NC(=O)N)/CC(C1)(C)C NRB01753 c1cc(ccc1c2cnc3cc(cc(c3n2)Br)C(F)(F)F)F BTB05455 c1cc(cc(c1)F)/N=C/c2ccc(c(c2)Cl)Cl BTB01760 Cc1ccc(cc1)S(=O)(=O)OC23CCC(CC2)C=C3 NRB01674 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)C(c4ccccc4)C5CCCC5 BTB01776 C/C=C(\C)/C(=O)NC(=S)NNC(=O)c1ccc(cc1)N(C)C BTB01782 CCOC(=O)C(=CNc1ccccc1c2nnc(o2)c3ccc(cc3)C(C)(C)C)C(=O)OCC BTB06973 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)NC(=O)c4ccccc4F BTB06975 COc1cccc(c1)c2nnc(o2)c3ccccc3NS(=O)(=O)c4ccc(cc4)Cl BTB06980 Cc1ccc(=O)n(n1)Cc2ccc(cc2)[N+](=O)[O-] BTB06984 Cc1ccc(c(c1)[N+](=O)[O-])c2[nH]c(nn2)c3ccncc3 BTB01709 c1ccc(c(c1)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl BTB05352 Cc1ccc(=O)n(n1)Cc2ccc(c(c2)Cl)Cl BTB06989 C1C(=NNC1=O)C(F)(F)F BTB07000 c1cc(c(cc1C2=CSC3=NCCCN23)F)F.Br BTB07003 COc1cccc(c1OC)/C=C\2/C(=O)NC(=S)S2 BTB01732 Cc1ccc(c(c1)C(=O)NN)N BTB01810 Cc1ccccc1C(=O)N(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3nc4ccccc4s3 BTB01839 c1cc(c(cc1c2csc(n2)Nc3ccc(cc3F)F)F)F BTB07002 Cc1ccc(cc1)NS(=O)(=O)c2c(c3cc(ccc3s2)Cl)C MWP00547 Cc1ccc(cc1)S(=O)(=O)N(CCC#N)CCC#N NRB01682 c1ccc2c(c1)c3cccc4c3n2c(=O)cc4O NRB01640 c1ccc(cc1)CN2CC3CCC2[C@@H](C3)O NRB01964 CC(C)(C1CCCC1N(C)C)OC(=O)c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-].Cl NRB01969 COc1cc(cc(c1OC)OC)C2CC(=Nc3ccccc3S2)c4ccccc4 RJC00342 Cc1cc(c2cc(ccc2n1)Br)C(=O)N/N=C/c3ccccc3O BTB01804 CN(C)/C=N/S(=O)(=O)c1ccc(cc1)Oc2c(cccc2Cl)[N+](=O)[O-] BTB05360 c1cc2c(cc1C3Nc4ccc(cc4C(=O)N3)[N+](=O)[O-])OCO2 BTB01828 c1cc(sc1)C2Nc3ccc(cc3C(=O)N2)[N+](=O)[O-] BTB01829 CC1Cc2c(nc(nc2N)N)CC1C BTB01820 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cccnc3 MWP00587 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCNc2nccc(n2)C(F)(F)F AW00549 CCOC(=O)C(=CNc1cc(ccc1N2CCCCC2)C(F)(F)F)C(=O)OCC BTB01846 Cc1c2cc(ccc2sc1c3cc([nH]n3)NC(=O)c4ccc(cc4)Cl)Cl MWP00594 Cc1c2cc(ccc2sc1c3cc([nH]n3)NC(=O)c4ccccc4)Cl MWP00595 C1CC2C=CC1C(C2C(=O)O)C(=O)O NRB02007 c1ccc(cc1)c2cc(nc(n2)SCc3c(cccc3Cl)F)O AW00539 Cc1cc(=O)n2c([nH]1)cc(n2)c3c(c4cc(ccc4s3)Cl)C MWP00593 c1ccc2c(c1)nc(s2)N(c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)c4ccc(cc4)[N+](=O)[O-] BTB01815 CCCCc1c(nc(nc1O)SCc2c(cccc2Cl)F)C AW00542 c1cc(cnc1)c2ccnc(n2)Sc3ncc(s3)[N+](=O)[O-] MWP00602 c1cc(ccc1CSC(=S)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)OC(F)(F)F AW00546 c1cc(cc(c1)NC(=S)NCCNc2nccc(n2)C(F)(F)F)C(F)(F)F AW00548 c1ccc(cc1)S(=O)(=O)n2cccc2 BTB07001 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)c4ccc(cc4)C(F)(F)F BTB06920 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2c3nnc(o3)c4ccc(cc4)Cl BTB06927 COc1ccc(cc1OC)S(=O)(=O)Nc2ccccc2c3nnc(o3)c4ccc(cc4)Cl BTB06928 c1cc(ccc1C(=O)CC(=S)C#N)Cl BTB06938 COc1ccc(c(c1)c2nnc(o2)c3ccccc3[N+](=O)[O-])Br BTB06939 CC(C)NC(=O)ONC(=O)c1csc(n1)c2cccnc2 MWP00600 c1cc(cnc1)c2ccnc(n2)Sc3c(cccn3)[N+](=O)[O-] MWP00603 c1cc2c(=O)c3cc(ccc3oc2nc1)NS(=O)(=O)c4ccc(c(c4)Cl)Cl BTB05323 Cc1c(n2ccccc2n1)C(=O)N/N=C/c3ccccc3O NRB01599 c1ccc(cc1)Cc2c(c3ccccc3n(c2=O)Cc4ccccc4)O NRB01601 Cc1ccccc1Cn2c(=O)ccc(n2)C BTB06983 c1ccc(c(c1)C2=Nc3ccccc3SC(C2)c4ccc(cc4)O)O RJC00357 c1ccc(cc1)c2cc3c(c(cc(=O)o3)O)c(=O)n2c4ccccc4 NRB01625 c1cc(ccc1[N+](=O)[O-])Oc2c(cc(cc2Cl)S(=O)(=O)N)Cl BTB05367 c1ccc2c(c1)cccc2NC(=O)N3CCCN(CC3)c4c(cccn4)[N+](=O)[O-] AW00457 Cc1cc(c(c(c1)C)n2c(nnn2)SCc3ccc(cc3)OC(F)(F)F)C AW00495 c1cc(cnc1)Nc2nc(cs2)c3cccs3 AW00498 c1ccc(cc1)C(=O)/C=C/2\C(=O)Oc3ccccc3N2 RJC00241 COc1ccc2c(c1)CCC(=O)C2 NRB01650 Cc1cccc(c1)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05353 c1cc(ccc1C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05354 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(ccc2NCCNC(=O)OC(C)(C)C)C(F)(F)F AW00537 Cc1ccc(cc1Cl)NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N BTB05363 c1ccc(cc1)C(C2CCCC2)C(=O)Nc3ccccc3SCCC#N BTB01774 c1ccc2c(c1)nc(s2)N(c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)c4c(cccc4F)F BTB01816 Cc1c2cc(ccc2sc1C(=O)CSc3nnc(s3)SCC#C)Cl MWP00537 Cc1c2cc(ccc2sc1C(=O)CSc3nnc(s3)SC)Cl MWP00538 c1ccc(cc1)C(C#N)(c2ccccc2)C3(CC3S(=O)(=O)c4ccccc4)C(C#N)(c5ccccc5)c6ccccc6 NRB01575 c1ccc(cc1)C(C2CCCC2)C(=O)O BTB01553 COc1cc(cc(c1OC)OC)/C=C/C(=O)O BTB01558 CC(=O)Nc1c(c(c(c(c1Cl)Cl)Cl)Cl)Cl BTB01573 Cc1ccc(c(c1)[N+](=O)[O-])NC(=O)c2ccccc2[N+](=O)[O-] BTB01586 CN1CCc2ccccc2C1Cc3ccccc3NS(=O)(=O)c4cc(c(cc4Cl)Cl)Cl BTB01791 CN1CCc2ccccc2C1Cc3ccccc3NS(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F BTB01796 c1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccc(cc4)Br RJC00344 c1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccc(cc4)Cl RJC00345 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2cc(ccc2Cl)C(F)(F)F)C#N BTB05365 Cc1cc(c2cc(ccc2n1)Br)C(=O)N/N=C\c3cc(cc(c3O)Cl)Cl BTB01807 COc1ccc(c(c1)O)C2=Nc3ccccc3SC(C2)c4ccccc4 RJC00350 COc1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccccc4O RJC00353 Cc1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccccc4O RJC00355 Cc1c2cc(ccc2sc1c3cnc(s3)NC(=O)c4ccccc4)Cl MWP00628 c1ccc(c(c1)/C=C/c2cccs2)C(=O)O NRB01585 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)c4ccc(cc4)Cl BTB06918 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2c3nnc(o3)c4ccc(cc4)C(C)(C)C BTB06963 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Nc2ccccc2c3nnc(o3)c4ccc(cc4)C(C)(C)C BTB06965 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NS(=O)(=O)c4ccc(cc4)Cl BTB06964 CCOC(=O)C(=CNc1cc(cc(c1)OC)C(F)(F)F)C(=O)OCC BTB01851 CCOC(=O)C(=CNc1ccc(cc1)N2CCOCC2)C(=O)OCC BTB01852 CCOC(=O)C(=CNc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)OCC BTB01853 Cc1c2cc(ccc2sc1c3cc([nH]n3)NC(=O)C)Cl MWP00596 c1cc(cnc1)NC(=S)N2CCCN(CC2)Cc3ccc(cc3Cl)Cl AW00524 CCOC(=O)C(=CNc1cc(ccc1n2cccc2)C)C(=O)OCC BTB01854 Cc1c2ccccc2sc1/C=C(\C#N)/S(=O)(=O)C(C)(C)C MWP00614 Cc1c2ccccc2sc1/C=N/Nc3c(cc(cc3Cl)Cl)Cl MWP00621 Cc1c2ccccc2sc1/C=N/Nc3ccccc3 MWP00623 Cc1c(cccc1Cl)NC(=S)N2CCCN(CC2)Cc3ccc(cc3)F AW00529 c1ccc(cc1)C2CC(=O)Nc3ccccc3S2(=O)=O RJC00324 c1cc2c(=O)c3cc(ccc3oc2nc1)NC=C(C#N)C#N BTB05343 c1cc(c(c(c1)F)C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])F BTB05348 Cc1cccc(c1)C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05349 CCCC(=O)N1c2ccccc2N=C(CC1c3ccccc3)c4ccccc4 RJC00382 Cc1ccc(c(c1)C)NC(=S)NCCCNC(=O)c2cccs2 AW00508 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SC(=O)c3ccc(nc3C)C(F)(F)F AW00480 C1C2CC3(CC1CC(C2)(C3)Br)C(=O)O NRB01917 COc1ccc(c(c1)O)C2=Nc3ccccc3SC(C2)c4ccc(c(c4)O)OC RJC00363 COc1ccc(c(c1)O)C2=Nc3ccccc3SC(C2)c4ccc5c(c4)OCO5 RJC00365 c1cc2c(=O)c3cc(ccc3oc2nc1)NS(=O)(=O)c4ccc(cc4)Cl BTB05318 c1ccc(c(c1)C2CC2)/N=C/c3cc(cc(c3O)Cl)Cl NRB01672 C[C@H]1CC[C@@H](CC1)NC(=O)C NRB01677 CSc1nccc(n1)c2cccnc2 MWP00604 Cc1ccc(c(c1)NC(=O)C(c2ccccc2)C3CCCC3)n4cccc4 BTB01775 CC1CC(CC(C1)(C)C)NC(=O)C(c2ccccc2)C3CCCC3 BTB01777 COc1cc(cc(c1OC)OC)CN2CCCN(C2c3cc(ccc3O)Br)Cc4cc(c(c(c4)OC)OC)OC BTB01697 CCOC(=O)/C(=C/C(=O)c1ccc(cc1)OC)/O RJC00246 Cc1cc(cc(c1)NC(=O)N2CCCN(CC2)Cc3c(cccc3Cl)F)C AW00502 COc1cc2ccccc2c(=O)c3c1scc3 NRB01588 c1ccc(c(c1)CSc2nccc(n2)c3ccco3)Cl MWP00519 c1cc(ccc1C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F BTB05355 c1ccnc(c1)CCN(c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl.Cl BTB01652 c1ccc(cc1)C2CC(=Nc3ccccc3N2)c4ccccc4 RJC00374 CCOC(=O)COc1ccc(cc1)C2=Nc3ccccc3NC(C2)c4ccccc4 RJC00376 CC(=O)N1c2ccccc2N=C(CC1c3ccccc3)c4ccccc4 RJC00380 Cc1ccc(c(c1)C(=O)N(CCc2ccccn2)c3ccccc3)[N+](=O)[O-] BTB01677 CCOC(=O)c1ccc(c(c1)C)[N+](=O)[O-] BTB01681 CN(CCC#N)c1ccc(cc1)/C=N/CCC/N=C\c2ccc(cc2)N(C)CCC#N BTB01696 Cc1ccc(c(c1)N)C(=O)Nc2ccc(cc2N)OC BTB01702 c1ccn(c1)c2ccc3c(c2)c(=O)c4cccnc4o3 BTB05341 CCOC(=O)/C(=C/Nc1ccc2c(c1)c(=O)c3cccnc3o2)/C#N BTB05342 COc1cc(cc(c1OC)OC)C2CC(=S)Nc3ccccc3S2 RJC00331 c1ccc(cc1)CSc2nccc(n2)c3ccco3 MWP00522 Cc1c2cc(ccc2sc1c3cc(n(n3)C)N)Cl MWP00566 Cc1ccc(cc1NC(=S)N2CCCN(CC2)Cc3ccc(cc3Cl)Cl)Cl AW00520 c1ccc(c(c1)NC(=O)CSc2nccc(n2)c3ccco3)Cl MWP00523 c1cc(oc1)c2ccnc(n2)SCC(=O)Nc3ccc(cc3F)F MWP00525 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3ccco3 MWP00526 Cc1c2cc(ccc2sc1c3cc(n(n3)C)NC(=O)c4cccc(c4)Cl)Cl MWP00569 COc1ccccc1C2CC(=Nc3ccccc3S2)c4ccccc4O RJC00352 c1ccc(cc1)n2c3ccccc3c(cc2=O)O NRB01611 CCOC(=O)/C(=C/Nc1cc(c(c(c1)Cl)O)C)/C#N BTB05449 c1cc(ccc1c2cnc3cc(cc(c3n2)Cl)C(F)(F)F)F BTB05454 c1cc(ccc1c2cnc3cc(cc(c3n2)Br)C(F)(F)F)Br BTB05458 COc1cc2c(c(c1OC)OC)[nH]c(=S)n(c2=O)c3ccccc3 BTB05464 CC(C)(C)SCCn1c(=O)c2cc(c(c(c2[nH]c1=S)OC)OC)OC BTB05471 c1cc(sc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)/N=C(\NN)/N4CCCC4)C(F)(F)F BTB07005 c1ccc(cc1)/N=c\2/n(cc(s2)c3ccc(c(c3)F)F)c4ccccc4.Br BTB07006 c1ccc2c(c1)c(c(s2)C(=O)Nc3cc(ccc3N4CCOCC4)C(F)(F)F)Cl BTB01903 c1cc(c(cc1C(F)(F)F)NC=C(C#N)C#N)N2CCCCC2 BTB01909 COc1ccc(cc1)COCC(CS(=O)(=O)c2ccc(c(c2)OC)OC)O RDR03130 Cc1cccc(c1)C2c3cc(c(cc3CCN2C(=O)c4c(c5ccccc5s4)Cl)OC)OC BTB01926 C1C2CC3CC1C(C(C2)C3=O)O NRB01688 CC(CNc1ccc(cc1[N+](=O)[O-])C(F)(F)F)O BTB05472 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)F)F)Cl BTB07011 Cc1nc(cs1)c2ccc(c(c2)F)F BTB07015 c1cc(sc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)/N=C(\NNS(=O)(=O)c4ccc(cc4)Cl)/N5CCCC5)C(F)(F)F BTB07017 CCN1c2cc(ccc2C(CC1(C)C)C)NC(=O)C NRB02093 c1ccc2c(c1)C(=O)N(C2=O)C(CCC(=O)O)C(=O)O BTB07024 Cc1cccc(c1)C(C)(C(C)(C)CN(C)C)O NRB01696 CC(C)N1CC(OC1=O)COc2ccc(cc2Cl)Cl RDR03102 CN(C)c1ccc2c(c1)Sc3cc(ccc3N2C(=O)c4ccccc4)N(C)C NRB02099 COc1cc2c(c(c1OC)OC)[nH]c(=S)n(c2=O)Cc3cccs3 BTB05465 c1c(cc(c-2c1C(=C(C#N)C#N)c3c2c(cc(c3)S(=O)(=O)N)[N+](=O)[O-])[N+](=O)[O-])S(=O)(=O)N.C1COCCO1 RJC00408 c1ccc(cc1)C2CC(=O)NC(=S)N2c3ccc(cc3Cl)Cl RDR03265 CCC(=O)Nc1ccc2c(c1)N(C(CC2C)(C)C)CC NRB02094 Cc1ccc(cc1)S(=O)(=O)O.Cc1ccc(cc1)S(=O)(=O)OC2CCC3(CN(CC[C@]3(C2)C)C)C NRB01750 CNC(=O)c1cc(ccc1Br)OC RJC00412 CNC(=O)c1cc(ccc1I)Cl RJC00416 CC(C)N1CC(OC1=O)COc2ccccc2Cl RDR03106 c1ccc(cc1)SCC(CNCc2ccc(cc2)Cl)O RDR03172 Cc1ccccc1C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-] BTB05425 c1ccc(c(c1)COC(=O)c2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-])I RJC00418 c1ccc(cc1)S(=O)(=O)CC(CS(=O)(=O)c2ccc(cc2)Br)O RDR03171 C1C(COCO1)([N+](=O)[O-])[N+](=O)[O-] NRB02075 c1ccc2c(c1)ccc3c2-c4cccc5c4c(ccc5)C3=O NRB02112 c1cc(ccc1N2CCC2)[N+](=O)[O-] NRB02115 CN1CCN(CC1)c2ccc(cc2)[N+](=O)[O-] NRB02117 c1cc(ccc1N=C2SCCS2)Cl RDR03123 COc1ccc(cc1)COCC(CS(=O)(=O)c2ccc(cc2)Cl)O RDR03126 Cc1ccc(cc1)S(=O)(=O)CC(COCc2ccc(cc2)OC)O RDR03128 CN(C)/C=N/C(=O)NCc1cccs1 BTB05407 c1c(cc(c(c1[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl)[N+](=O)[O-])C(F)(F)F BTB05412 COC(=O)/C(=C\C=C\c1ccccc1)/C#N NRB02091 CCN(CCN1C(=O)CCC1=O)c2cccc(c2)NC(=O)C NRB02092 Cc1cc(ccc1Cl)O/C=C/C(=O)c2ccc(cc2)Br NRB05012 CCCCn1c2ccccc2c(c(c1=O)Cc3ccccc3)O NRB02128 CC(C)(C)OC(=O)CC(C(=O)N)NC(=O)OCc1ccccc1 RJC00425 CC(=O)NC1=NN(C(N1C(=O)C)c2cc(c(c(c2)OC)OC)OC)C(=O)C RJC00426 c1ccc(cc1)COC(=O)NC(COC(=O)OCc2ccccc2)C(=O)O NRB01725 C1CCC2[C@H](CCCC2C1)O NRB01738 Cc1c2cc(ccc2sc1/C=N/Nc3ccc(cc3)[N+](=O)[O-])Cl MWP00673 COc1cc2c(cc1OC)C(=NCC2)c3c(c4ccccc4s3)Cl BTB01896 COc1ccc(cc1OC)CCNC(=O)c2cc3ccccc3oc2=O BTB01898 c1cc(ccc1C#N)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05416 Cc1c(c(no1)c2ccccc2)C(=O)NCCc3ccc(c(c3)OC)OC BTB01889 c1cc2cccc(c2c(c1)COC(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-])Br RJC00419 COC(=O)c1ccccc1Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] RJC00422 c1ccc(cc1)OCCCCC#N NRB02143 c1ccc(c(c1)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-])F BTB05426 COc1ccc(c(c1C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-])OC)[N+](=O)[O-] BTB05427 c1ccc(cc1)c2ccc(cc2)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05431 c1ccnc(c1)CNC(=O)N BTB05401 CNc1ccc(cc1C(=O)N)Cl BTB01822 CCC(C)/C(=N/O)/c1ccccc1 NRB02026 c1cc(c(cc1c2cnc3cc(cc(c3n2)Br)C(F)(F)F)Cl)Cl BTB05384 c1ccc(c(c1)C(=O)NNc2c(cc(cc2Cl)Cl)Cl)N BTB05410 c1cc(c(cc1F)F)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05413 Cc1cc2c(cc1C)nc(cn2)c3ccc(c(c3)Cl)Cl BTB05389 c1ccc(c(c1)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-])Cl BTB05423 Cc1c2ccccc2sc1/C=N/c3ccc(cc3)[N+](=O)[O-] MWP00617 Cc1c2ccccc2sc1/C=N/c3ccc(cc3)C(C)C MWP00618 CCOC(=O)C(=CNc1cc(ccc1N2CCc3ccccc3C2)C(F)(F)F)C(=O)OCC BTB01878 Cc1ccccc1C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05419 CCOC(=O)C(=CNc1cc(ccc1N2CCOCC2)C(F)(F)F)C(=O)OCC BTB01855 CCOC(=O)C1CCN(CC1)c2ccc(cc2NC=C(C(=O)OCC)C(=O)OCC)C(F)(F)F BTB01856 c1ccc(c(c1)C(=O)N(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3nc4ccccc4s3)Cl BTB01840 c1cc(c(c(c1)F)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-])F BTB05429 CCOC(=O)C(=CNc1ccc(cc1)F)C(=O)OCC BTB01847 c1cc(c(cc1C(F)(F)F)/N=C/c2cc(cc(c2O)Cl)Cl)N3CCOCC3 BTB01861 COc1ccc(cc1OC)CCNC(=O)c2ccccc2Cl BTB01869 Cc1ccc(c(c1)[N+](=O)[O-])NCCc2ccccn2 BTB01874 Cc1ccc(c(c1)C)NC(=S)NCCNc2nccc(n2)C(F)(F)F AW00551 c1cc(c(c(c1)Cl)/C=N/Nc2nc[nH]n2)Cl BTB05350 CCOC(=O)C(=CNc1cc(ccc1n2cccc2)OC)C(=O)OCC BTB01879 CC(C)c1ccc(cc1)C2CC(=O)Nc3ccccc3S2 MWP00674 Cc1c2cc(ccc2sc1C(=O)/C(=C/N(C)C)/C#N)Cl MWP00676 c1cc(c(cc1Cl)C(=O)N)I RJC00415 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCOCC2 BTB01843 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCc3ccc(c(c3)OC)OC BTB01890 Cc1c2ccccc2sc1/C=N/Nc3ccc(cc3)[N+](=O)[O-] MWP00620 Cc1ccsc1C2CC(=O)Nc3ccccc3S2 MWP00654 c1cc(c(cc1C(F)(F)F)/N=C/c2cc(cc(c2O)Cl)Cl)Cl BTB01848 Cc1c2cc(ccc2sc1c3csc(n3)NC(=O)c4ccc(cc4)Cl)Cl MWP00627 Cc1c2ccccc2sc1/C=C/c3ccnc(n3)SCc4ccccc4 MWP00640 Cc1c2ccccc2sc1/C=C/c3ccnc(n3)SCc4ccc(cc4)F MWP00642 c1ccc2c(c1)N=C(CC(S2)c3ccc(cc3)Cl)c4ccc(cc4)O RJC00360 c1ccc(cc1)C/N=C/c2c(c3ccccc3[nH]c2=O)O NRB01634 COC(=O)/C=C(\C(=O)OC)/Nc1ccc(cc1)Cl BTB05391 c1cc(c(cc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl)Cl BTB05417 c1ccc(c(c1)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F BTB05418 COc1cc(c(c(c1OC)OC)N)C(=O)OC BTB05442 Cc1ccc(cc1)S(=O)(=O)/C(=C\c2c(c3cc(ccc3s2)Cl)C)/C#N MWP00684 c1ccc2c(c1)cccc2Sc3ccccc3C(=O)N RJC00407 C=CCn1c(n[nH]c1=S)c2ccc(cc2)S(=O)(=O)N RJC00429 C1CC2C3CC1CC2OC3=O NRB01759 COc1cc(c(c(c1OC)OC)[N+](=O)[O-])C(=O)O BTB05392 CCOC(=O)C(=CNc1ccccc1SCCC#N)C(=O)OCC BTB01850 c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cccnc3 MWP00586 c1cc(sc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)/N=C(\NNC(=O)c4ccc(cc4)Cl)/N5CCCC5)C(F)(F)F BTB07018 c1ccc(c(c1)C(=O)NC(=O)NN/C(=N\S(=O)(=O)c2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4)/N5CCCC5)F BTB07019 c1cc(ccc1C(F)(F)F)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05433 COc1ccc(c(c1C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)OC)[N+](=O)[O-] BTB05420 Cc1cccc(c1)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-] BTB05424 c1cc(ccc1C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-])[N+](=O)[O-] BTB05428 c1ccc(c(c1)C(=O)NNc2c(cc(cc2Cl)Cl)Cl)NC(=O)c3cccs3 BTB05444 Cc1ccc(c(c1)C)Nc2nc(cs2)c3ccc(c(c3)F)F BTB07008 c1cc(cc(c1)C(F)(F)F)C(=O)Oc2c(cc(cc2Br)C(F)(F)F)[N+](=O)[O-] BTB05430 c1cc(c(cc1C(F)(F)F)N)N2CCCCC2 BTB01859 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc(cc3)Br)Cl MWP00541 COc1ccc(cc1OC)C2CC(=Nc3ccccc3S2)c4ccccc4O RJC00358 COc1ccc(c(c1)O)C2=Nc3ccccc3SC(C2)c4cccc(c4)O RJC00362 Cc1c2ccccc2sc1/C=C/c3ccnc(n3)SCc4cccc(c4)Cl MWP00641 c1ccc(c(c1)C2CC(=O)Nc3ccccc3S2)Cl MWP00658 CC(/C(=N/O)/c1ccccc1)SC NRB02030 COc1cc(c(c(c1OC)OC)N)C(=O)O BTB05448 Cc1cc(ccc1[N+](=O)[O-])C(=O)NCCc2ccc(c(c2)OC)OC BTB01871 COc1cc2c(cc1OC)C(=NCC2)c3ccc(cc3)[N+](=O)[O-] BTB01885 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCc3ccc(c(c3)OC)OC BTB01888 c1ccc(cc1)C2CC(=O)Nc3ccccc3S2 MWP00675 Cc1cccc(c1N=C2SCCS2)C RDR03089 CC(C)N1CC(OC1=O)COc2ccc(cc2)Br RDR03090 COc1ccc(cc1OC)CCNC(=O)c2c(c3ccccc3s2)Cl BTB01891 Cc1c(c(no1)c2ccccc2)C3=NCCc4c3cc(c(c4)OC)OC BTB01895 Cc1c2ccccc2sc1/C=C/c3ccnc(n3)SCC(=O)Nc4ccccc4 MWP00650 c1cc(sc1)C(=O)O/N=C(/CC(=O)Nc2ccc(cc2F)F)\N BTB05311 COc1ccc(c(c1)O)C2=Nc3ccccc3SC(C2)c4ccc(c(c4)OC)OC RJC00364 c1ccc(cc1)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05351 c1cc(sc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)/N=C(\NNC(=O)Nc4ccc(cc4)Cl)/N5CCCC5)C(F)(F)F BTB07022 CC(=C(c1ccccc1)NC(=O)C)C NRB02054 c1ccc(c(c1)C(=O)N)Sc2ccccc2[N+](=O)[O-] RJC00409 COc1ccc(cc1)/C=C(/C(=O)c2ccccc2OCc3ccccc3)\[N+](=O)[O-] NRB04942 C/C=C(\C)/C(=O)NC(=S)NNC(=O)c1c(onc1c2ccccc2)C BTB01785 c1ccc(cc1)C(C2CCCC2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB01787 c1ccc2c(c1)[nH]c(n2)c3c(cccc3Cl)Cl BTB05394 COc1cccc(c1)C2CC(=Nc3ccccc3S2)c4ccccc4 RJC00338 Cc1ccc(cc1)SCC(=O)c2c(c3cc(ccc3s2)Cl)C MWP00514 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccccc3C(=O)NNc4c(cc(cc4Cl)Cl)Cl BTB05443 CC1=C(CC(C(C1)C(=O)O)C(=O)O)C NRB01786 Cc1ccc2c(c1)c(=O)n(c(n2)S)c3cccnc3 RDR03318 CC1CCN(CC1)/C(=N/S(=O)(=O)c2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4)/NN BTB07025 c1ccc2c(c1)c(c(s2)C(=O)Nc3cc(ccc3N4CCCC4)C(F)(F)F)Cl BTB01899 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=O)c4c(c5ccccc5s4)Cl)C(F)(F)F BTB01900 CC(C)N1CC(OC1=O)COc2ccc(cc2)F RDR03105 c1ccc(c(c1)N=C2SCCS2)Cl RDR03110 c1cc(c(c(c1)Cl)Cl)/N=C/2\NCCN/C(=N/c3cccc(c3Cl)Cl)/SS2 RDR00654 c1cc(cc(c1)Cl)/N=C/2\NCCN/C(=N/c3cccc(c3)Cl)/SS2 RDR00655 CC12CCC3c4ccc(cc4CCC3C1CC[C@]2(C#C)O)Oc5ccc(cc5)[N+](=O)[O-] NRB03724 CC(C)CCCC(C)C1CCC2C1(CCC3C2CC[C@@]4(C3(CCC(C4)O)C)O)C NRB03746 CC1C(C2(CCC1CC2)CO)C NRB02140 COC(=O)CCCC/C=N/Nc1ccc(cc1)[N+](=O)[O-] NRB02142 c1cc(c(cc1/N=C/2\NCCN/C(=N/c3ccc(c(c3)Cl)Cl)/SS2)Cl)Cl RDR00647 CC12CCC3(C[C@@H]1CCC4C2CCC5(C4CCC5O)C)OCCO3 NRB03720 CCN(CC)OC(=O)c1c(onc1c2c(cccc2Cl)Cl)C RF01340 Cc1ccc2c(c1)c(no2)OC(=O)NC(C)(C)C RF01343 CC(C)NC(=O)Oc1c2ccccc2on1 RF01347 c1cc(c(c(c1)Cl)/C=N/Nc2c(cncc2Cl)Cl)Cl RF01354 c1ccc(cc1)CNC(=S)NCCNC(=O)Cc2ccc(cc2)O RDR03349 c1ccc(cc1)NC(=O)NNc2c(cncc2Cl)Cl RF01330 CCOC(=O)C12CCCC(CC1=O)(C(=O)C2)C(=O)OCC NRB01822 CC12CCC3C(C1CCC2O)CCC4=CC(=O)C(=C)CC34C NRB03737 C[C@@H]1CC2C3CCC4CC(=O)C=CC4(C3[C@@H](CC2([C@]1(C(=O)COC(=O)C)O)C)O)C NRB03740 Cc1ccc(cc1)/C(=C/C=C(C#N)C#N)/Nc2ccccc2 NRB05025 Cc1ccc(cc1)/C(=C/C=C(C#N)C#N)/Nc2ccc(cc2)C NRB05026 c1cc(ccc1C(=O)/C=C/Sc2nc3cc(ccc3s2)Cl)Br NRB05038 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC=C(C#N)C#N)C(F)(F)F BTB01907 CCOC(=O)C1CCN(CC1)c2ccc(cc2NC=C(C#N)C#N)C(F)(F)F BTB01908 c1ccc2c(c1)CCN(C2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB01912 CN(C)CCSC(=S)NC1CCCCCCC1.Cl RDR03166 COc1cc2c(cc1OC)C(N(CC2)C(=O)c3c(c4ccccc4s3)Cl)c5ccccc5Cl BTB01916 COc1cc2c(cc1OC)C(NCC2)c3ccc(cc3)N BTB01920 c1ccc(cc1)c2c(c3cc(ccc3[nH]c2=O)OC(F)(F)F)O NRB02258 CCOC(=O)C12CCC(CC1=O)(C(=O)C2)C(=O)OCC NRB02268 C1C2C3C2C(=O)C1C3C(=O)O NRB02153 c1ccc2c(c1)c(c(s2)C(=O)N/N=C/c3ccc(c(c3)Cl)O)Cl RH00226 CCOC(=O)C1CCN(CC1)c2ccc(cc2NC(=O)c3c(c4ccccc4s3)Cl)C(F)(F)F BTB01902 c1cc(c(cc1C(F)(F)F)NC=C(C#N)C#N)N2CCOCC2 BTB01905 c1cc(c(cc1C(F)(F)F)NC=C(C#N)C#N)N2CCCC2 BTB01906 c1ccc2c(c1)/C(=N\N=C(N)N)/C(=O)N2 RJC01505 c1ccc(cc1)c2cc(=O)c3ccccc3o2 RJC01511 Cc1ccc2c(c1)c(no2)OC(=O)NC(C)C RF01342 c1cc(ccc1C(=O)/C=C/Sc2nc3cc(ccc3s2)Cl)I NRB05040 Cc1ccnc(n1)S/C=C/C(=O)c2ccc(cc2)I NRB05041 CC(=O)N[C@H]([C@H]([C@@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)C(=S)N RJC01514 COc1ccc(cc1)C(=O)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB05046 CC(C)CCCC(C)C1CCC2C1(CCC3C2CC(C4(C3CCC(C4)OC(=O)C)C)OC(=O)C)C NRB03747 c1ccc(cc1)c2c(cnc(n2)N)c3nnnn3c4ccccc4 NRB05022 c1ccc(c(c1)/N=C\2/N(C(=O)CS2)c3ccccc3F)F RDR00662 CCN(CC)OC(=O)Nc1c(onc1c2c(cccc2Cl)Cl)C RF01339 c1cc(ccc1NC(=S)NNc2c(cncc2Cl)Cl)F RF01349 Cc1c(n2ccccc2n1)C(=O)N/N=C\c3ccc(cc3)Cl NRB05056 c1c(c(c(cn1)Cl)N/N=C/C2CC3CC2C=C3)Cl RF01358 Cc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2)C(=O)O NRB05051 c1cc(ccc1C(=O)/C=C/Oc2ccc(cc2)Cl)Br NRB05052 CC(C)CCCC(C)C1CCC2C1(CCC3C2CC([C@@]4(C3(CCC(C4)OC(=O)C)C)O)OC(=O)C)C NRB03753 c1cc(c(nc1)NC2CC2)[N+](=O)[O-] RH00271 c1ccc(cc1)c2c(cno2)c3nnnn3c4ccc(cc4)Br NRB05139 COc1ccc(cc1)n2c(nnn2)c3cnoc3c4ccccc4 NRB05140 Cc1c(c(=O)c2ccccc2s1)Cc3ccc(c(c3)Cl)Cl RDR03273 CC12CC/C(=N\O)/C=C1C=CC3C2CCC4(C3CCC45CCC(=O)O5)C NRB03749 CC(C)(C12CC3CC(C1)CC(C3)C2)O NRB01891 c1ccc(cc1)C(=O)/C=C/Sc2nc3cc(ccc3s2)Cl NRB05032 CCC(C)(C)/C(=N\Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/c2ccccc2 NRB02162 Cc1ccc(cc1)n2c(nnn2)c3cnn(c3c4ccccc4)c5ccccc5 NRB05142 COc1ccc2c(c1)[nH]c(=O)c(c2O)Cc3ccccc3 RJC01492 c1cc(c(cc1Cl)Cl)NC(=S)NNc2c(cncc2Cl)Cl RF01351 c1cc(cc(c1)[N+](=O)[O-])/C=N/Nc2c(cncc2Cl)Cl RF01353 CN(C)c1ccc(cc1)/C=N/Nc2c(cncc2Cl)Cl RF01355 CCOC(=O)c1ccc(cc1)NC(=S)N/N=C/c2c(cccc2Cl)Cl NRB05059 CCOC(=O)c1ccc(cc1)NC(=S)N/N=C/c2ccc(cc2)[N+](=O)[O-] NRB05060 CC(=O)/C(=C\Nc1ccc(cc1)O)/c2nnnn2c3ccccc3 NRB05016 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)OC23CCC(CC2)(CC3)C(=O)N NRB02209 CC(C)(CC1(CCCCC1)CO)O NRB02212 c1cc(ccc1C(=O)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br NRB05049 c1cc(ccc1C(=O)/C=C/Sc2nc3cc(ccc3s2)Cl)F NRB05035 CCCNC(=O)Oc1c2cc(ccc2on1)Cl RF01328 c1cc(ccc1NC(=O)NNc2c(cncc2Cl)Cl)Cl RF01331 CCc1ccc(cc1)C(=O)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB05045 CC(C)NC(=O)Oc1c2ccc(cc2on1)Cl RF01334 CC(C)NC(=O)Oc1c2cc(ccc2on1)Cl RF01335 CC(C)NC(=O)NNc1c(cncc1Cl)Cl RF01337 Cc1ccc(cc1)C(=O)/C=C/Oc2ccc(c(c2)C)Cl NRB05053 Cc1c(n2ccccc2n1)C(=O)NNC(=O)N NRB05055 COC(=O)C1C2CC3CC(C2)C(C1C3)OS(=O)(=O)c4ccc(cc4)[N+](=O)[O-] NRB02177 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)OC2C3CC4CC(C3)C(C2C4)C#N NRB02188 Cc1c(c(ccn1)O)OC(C)C(=O)N RF01407 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3c4ccccc4on3 RF01446 c1cc(ccc1C(=O)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F NRB05047 c1cc(ccc1C(=O)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl NRB05048 CCOC(=O)C(C(F)(F)F)(NCc1ccccc1)NC(=O)C RJC01532 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C(=N/OC(=O)C(C)(C)C)/N RF01378 CC(=O)OC12CC3CC(C1)C(C(C3)C2)O NRB01908 c1ccc2c(c1)c(cc(n2)c3ccco3)C(=O)O RDR03220 c1cc(sc1)CNC(=O)N BTB05399 CCOC(=O)C(=CNc1ccccc1n2cccc2)C(=O)OCC BTB01860 c1ccc(c(c1)/C=N/c2cc(ccc2Cl)C(F)(F)F)O BTB01849 Cc1c2ccccc2sc1/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl MWP00612 COc1ccc(cc1OC)CCNC(=O)c2ccc(cc2)[N+](=O)[O-] BTB01875 COc1ccc(cc1)C(=O)/C=C/Sc2nc3cc(ccc3s2)Cl NRB05034 c1cc(ccc1C(=O)/C=C/Sc2nc3cc(ccc3s2)Cl)Cl NRB05037 c1ccc2c(c1)c(=O)n(c(n2)S)c3cccnc3 RDR03317 Cc1ccc(cc1)S(=O)(=O)OCC2C3CCC(C3)C2O NRB01909 CC(=O)OC1CCC2C1(CCC3C2C=CC4=CC(=O)C=CC34C)C NRB03742 Cn1c(=N)nc2c(n1)c3ccccc3[nH]2 RJC01503 CC(C)CCCC(C)C1CCC2C1(CCC3=C4CCC(CC4(C(CC23)OC(=O)C)C)O)C NRB03760 COc1ccc(cc1OC)CCNC(=O)c2c(cccc2Cl)Cl BTB01876 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCC2 BTB01877 Cc1ccccc1CSc2nccc(n2)/C=C/c3c(c4ccccc4s3)C MWP00643 Cc1ccc(c(c1)[N+](=O)[O-])OC(C)CC(=O)O RJC00384 CC(CC(=O)O)Oc1ccc(cc1[N+](=O)[O-])Cl RJC00385 Cc1c2cc(ccc2sc1/C=N/Nc3ccccn3)Cl MWP00672 c1cc(sc1)CCC(=O)O RJC01494 CCOC(=O)C(C(F)(F)F)(NC(=O)NC(=O)C)O RJC01524 CCCCn1c2ccccc2c(c(c1=O)CC)O NRB02127 COc1ccc2c(c1)c(c(c(=O)[nH]2)c3ccccc3)O NRB02130 CC(C)(C)c1ccc(cc1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05434 Cc1cc(cc(c1O)Cl)NC=C(C(=O)C)C(=O)C BTB05438 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccccc3C(=O)NNc4c(cc(cc4Cl)Cl)Cl BTB05441 c1ccc(cc1)CCNC(=S)NN RDR00814 c1ccc(cc1)CCNC(=S)N/N=C/c2ccccc2O RDR00815 c1ccc(cc1)SC(C(=O)Nc2ccc(cc2)F)(F)F RDR03185 CCOC(=O)CNC(=O)[C@H]([C@@H]([C@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC01516 CCCCn1c2ccccc2c(c(c1=O)c3ccccc3)O NRB02122 COc1ccc(cc1)/N=C\2/N(C(=O)CS2)c3ccc(cc3)OC RDR00673 CC12CCC3C(C1CCC2O)CCC4=CCCCC34 NRB03722 c1cc(cnc1)c2nc(cs2)c3ccc(c(c3)F)F BTB07010 c1cc(c(cc1c2csc(n2)N)F)F BTB07014 c1cc(sc1)c2cc(nn2c3ccc(cc3)S(=O)(=O)/N=C(\N/N=C/c4ccc(cc4)Cl)/N5CCCC5)C(F)(F)F BTB07016 c1cc(c(cc1C2=NNC3=NCCN3C2)F)F BTB07021 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C)NC(=O)C RJC01540 c1cc(ccc1NC(=O)c2ccncc2)F BTB01927 CC12CCC(=O)C=C1C[C@H](C3C2CCC4(C3CC[C@@]45CCC(=O)O5)C)C(=O)OC6CCCC6 NRB03717 CSc1nc2ccccc2c(=O)n1c3cccnc3 RDR03320 CC(=O)[C@]1(CCC2C1(CC(C3(C2CCC4=CC(=O)CCC43C)F)O)C)OC(=O)C NRB03816 COc1ccc(cc1OC)CCNC(=O)c2ccccc2[N+](=O)[O-] BTB01870 C[C@@]12CCCCC1(CC[C@H](C2)O)C NRB01741 CC(C)CCCC(C)C1CCC2C1(CCC3C2CC[C@@]4(C3(CCC(C4)OC(=O)C)C)Cl)C NRB03718 Cc1cc(c(=O)[nH]n1)Cc2cccs2 RH00265 Cc1cc(c(=O)[nH]n1)Cc2ccc(cc2)C(F)(F)F RH00267 Cc1ccc(cc1)S(=O)(=O)O[C@@H]2CC3C[C@@H](C2C3)F NRB02231 COc1ccc(c(c1)S(=O)(=O)CC(CS(=O)(=O)c2ccccc2)O)OC RDR03170 Cc1ccc(c(c1)C(=O)N)I RJC00413 Cc1ccc(c(c1)C(=O)NC)I RJC00414 CC(=O)OC1CCC2=C3CCC4(CCCC4C3CC(C2(C1)C)OC(=O)C)C NRB03768 CC(C)CCCC(C)C1CCC2C1(CCC3C2CC[C@@]4(C3(CCC(C4)OC(=O)C)C)O)C NRB03775 Cc1ccc(cc1)S(=O)(=O)OCC2CC3CCC2C(C3)O NRB01793 CC1CC(CC2(C1)CC(=O)N(C2=O)c3ccc(cc3)Cl)(C)C RDR03388 CC1CC2(C(CC[C@]2(C#C)O)C3C1c4ccc(cc4CC3)OC)C NRB03794 CC12CCC3C(C1CCC2=O)CCC4=CCCCC34 NRB03735 c1cc(ccc1NC(=S)Nc2ccc3cn[nH]c3c2)F RDR00562 c1ccc(cc1)c2c(c3ccccc3[nH]c2=O)O NRB02133 CC(=O)NC(=N/N=C\1/c2ccccc2NC1=O)NC(=O)C RJC01513 CC(CCCO)C1CCC2C1(CCC3C2CCC4C3(CCCC4)C)C NRB03719 CCOC(=O)OC1CCC2C1(CCC3C2CCC4=CC(=O)C(=C)CC34C)C NRB03723 CC(=O)/C(=C\Nc1ccccc1O)/c2nnnn2c3ccccc3 NRB05017 CC(=O)OC1CCC23COC([C@]2(C1)Br)CC4C3CCC5(C4CCC5OC(=O)c6ccccc6)C NRB03725 CC(=O)[C@]1(CCC2C1(CC(=O)C3C2CC[C@@]4(C3(CCC(=O)C4)C)C)C)O NRB03728 Cc1ccc(cc1)N(/C=C/c2nnnn2c3ccccc3)C(=O)C NRB05019 Cc1ccc(cc1)C(=O)/C=C/Sc2ccccn2 NRB05009 CCOC(=O)c1c2csc(c2c(=O)n(n1)c3ccc(cc3)C(C)(C)C)N/C=C(\C#N)/C(=O)OCC RH00286 C1CC2(CC(=O)C1(CC2=O)C(=O)O)C(=O)O NRB02292 c1c(cc(c(c1/C=N/NC(=S)NCC2CCCO2)O)Cl)Cl RDR00929 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1)O RJC01548 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C)NC(=O)c2ccccc2 RJC01560 C[C@@]1(CCC2C1(CCC3C2CCC4=CC(=O)C(=C)CC34C)C)O NRB03837 COc1ccc(cc1)C(=O)/C=C\Nc2ccc(cc2)OC(F)(F)F NRB05122 c1cc(ccc1C(=O)/C=C\Nc2ccc(cc2)OC(F)(F)F)F NRB05123 CCc1c(c(=O)[nH]c(n1)S)C#N RH00268 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C(F)(F)F)NC(=O)c2ccccc2 RJC01572 CC(C)/C(=N/O)/c1ccccc1 NRB02327 CC(C1CCC2C1(CCC3C2CCC4=CC(=O)CCC34C)C)O NRB03833 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1)OC RJC01578 Cc1cc2c(cc1OC)CCC3C2CCC4(C3CCC4=O)C NRB03844 CC(=O)OC1CCC2C1(CCC3C2CC[C@@H]4C3(C/C(=C\c5ccccc5)/C(C4)OC(=O)C)C)C NRB03835 Cc1ccc2c(c1)nc([nH]2)S/C=C/C(=O)c3ccc(cc3)OC NRB05117 Cc1ccc(cc1)Cc2cc(n[nH]c2=O)C RH00270 c1cc(cnc1)c2[nH]nc(n2)c3cccnc3 NRB02384 c1cc(ccc1c2[nH]ncn2)[N+](=O)[O-] NRB02386 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)c2ccccc2 RJC01571 c1cc(oc1)Cn2c(cc(nc2=S)O)O RDR00877 CC12CCC3c4ccc(cc4CCC3C1CCC2=O)OCCCCCCN(C)C NRB03843 CC12CCC(=O)C=C1CCC3C2C(=O)CC4(C3CCC4=O)C NRB03820 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1)NC(=O)C RJC01520 CCNC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl RDR00909 CC(C)(C)c1ccc(c(c1)Br)NC(=O)C2CC2 RF01619 Cc1cc(cc2c1C3CCC4(C(C3CC2)CC[C@]4(C)O)C)OC NRB03848 c1ccc(cc1)c2c(cnn2c3ccccc3)c4nnnn4c5ccc(cc5)F NRB05144 Cc1ccc2c(c1)c(c(c(=O)[nH]2)c3ccccc3)O NRB02370 Cc1ccc(cc1)n2c(nnn2)c3cnn(c3C)c4ccccc4 NRB05149 CCOC(=O)C(C(F)(F)F)(Nc1cccc(n1)C)NC(=O)c2ccccc2 RJC01573 CCOC(=O)/C(=C/NNc1ccc(cc1)[N+](=O)[O-])/C#N RH00287 Cc1cc(cc(c1OC(=O)Nc2ccccc2)C)C(C)(C)c3cc(c(c(c3)C)OC(=O)Nc4ccccc4)C RH00294 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)Cl)NC(=O)c2ccccc2 RJC01567 CC(=O)O[C@H]([C@@H]([C@H](C(=O)Nc1ccccc1)OC(=O)C)OC(=O)C)[C@@H](C(=O)Nc2ccccc2)OC(=O)C RJC01519 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Oc2ccccc2)OC(=O)C)OC(=O)C)OC(=O)C NRB05173 CCOC(=O)c1c2csc(c2c(=O)n(n1)c3ccc(cc3)C(C)(C)C)NC=C(C(=O)OCC)C(=O)OCC RH00284 c1cc(ccc1CSCCC(=O)Nc2ccc(cc2)Cl)Cl RDR03417 c1cc(oc1)/C=N/NC(=S)NCC2CCCO2 RDR00928 CC12CCC3C(C1CCC2OC(=O)c4ccccc4)CC=C5C3(CCC(C5)O)CO NRB03823 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1OC)NC(=O)c2ccccc2 RJC01569 CCN(CC)C(=S)Oc1ccccc1[N+](=O)[O-] RDR00819 COCCCNc1nc(cs1)c2ccccc2.Br RDR00832 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C)NC(=O)C RJC01528 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C(F)(F)F)NC(=O)C RJC01533 CC1(c2ccccc2-n3c1cc4c(c3=O)c(cc(=O)o4)O)C NRB05091 CCOC(=O)NC(=S)Nc1ccc(cc1NC(=S)NC(=O)OCC)C(C)(C)C RF01585 CC(C)(C)C(=O)NC(=O)Nc1cc(ccc1Cl)C(F)(F)F RF01487 CCOC(=O)C(C(=O)C)Sc1[nH]nc(n1)c2ccc(cc2)Cl NRB05070 CN1CC[C@@]2(CCCC[C@@H]2C1)Cl.C(=O)(C(=O)O)O NRB02263 CC(C)(C)C1=CC(=O)C(=CC1=O)C(C)(C)C RF01571 CC(=O)Nc1cccc(c1)C(C)(C)C RF01579 CC(C)(C)c1ccc(c(c1)NC(=O)N(C)C)NC(=O)N(C)C RF01590 CC12CCC3c4ccc(cc4CCC3C1CC[C@]2(C#C)O)OC NRB03793 c1ccc(cc1)C(=O)/C(=C\N2CCCC2)/c3nnnn3c4ccccc4 NRB05127 CC(C)(C)NC(=S)N/N=C/c1cccnc1 RDR00898 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)S(=O)(=O)N)NC(=O)c2ccccc2 RJC01575 Cc1ccccc1COc2c3ccc(cc3ncn2)Cl RH00228 CC(C)CCCC(C)C1CCC2C1(CCC3=C4CCC(CC4(C(CC23)O)C)O)C NRB03754 Cc1ccc2c(c1)c(ncn2)Oc3c(cccn3)[N+](=O)[O-] RH00234 CC12CCC3c4ccc(cc4CCC3C1CCC2=O)OCCCC#N NRB03851 c1ccc(c(c1)C(=O)Nc2nc[nH]n2)O RDR00838 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)C RJC01534 CC12CCC3C(C1CCC2O)CCC4=CC5(CCC34C)OCCO5 NRB03811 c1ccc(cc1)C(=O)N/C(=C\c2ccc3c(c2)OCO3)/C(=O)O RDR00756 Cc1cc(cc(c1OC(=O)Nc2cc(cc(c2)Cl)Cl)C)C(C)(C)c3cc(c(c(c3)C)OC(=O)Nc4cc(cc(c4)Cl)Cl)C RH00291 CCN(CC)C(=S)Oc1ccc(cc1C(=O)Nc2ccc(cc2)F)Br RDR00839 CC(C)(C)c1ccc(c(c1)NC(=O)C(Cl)Cl)NC(=O)C(Cl)Cl RF01613 c1cc(ccc1S(=O)(=O)N/N=C/c2ccc3c(c2)OCO3)Cl RDR00710 CC1CC2(C(CCC2O)C3C1c4ccc(cc4CC3)O)C NRB03797 c1cc2c(cc1C(=O)CCN3CCOCC3)OCCCO2.Cl NRB05082 c1ccc2cc(ccc2c1)n3c(nnn3)/C=C/N4CCCC4 NRB05084 CCN(CC)C(=S)Oc1ccccc1C(=O)Nc2ccc(c(c2)Cl)Cl RDR00840 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C(F)(F)F)NC(=O)C RJC01535 C[C@@H]1CC2C3CCC4CC(CCC4(C3[C@@H](CC2([C@]1(C(=O)C)O)C)O)C)O NRB03745 CC1(CCC(CC1)C(C)(C)O)C NRB02318 CS(=O)(=O)N1CCN(CC1)CCOS(=O)(=O)C RH00272 c1cc(ccc1C(=O)/C=C\Nc2ccc(cc2)OC(F)(F)F)Cl NRB05124 c1ccc2c(c1)-c3ccccc3C2=NN NRB02256 C/C(=N\O)/C(=O)Nc1cccc(c1)C(F)(F)F NRB02323 CC(=O)Oc1ccc2c(c1)CCC3C2=CCC4(C3CCC4OC(=O)C)C NRB03799 c1cc(ccc1NC(=S)N/N=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)F RDR00731 CCOC(=O)C(C(F)(F)F)(NC(=O)c1c(cccc1F)F)O RJC01551 CCOC(=O)c1cnc2ccc(c(c2c1O)C#N)F RH00252 Cc1ccc2c(c1)c(=O)n(c(n2)SC)c3cccnc3 RDR03350 CC(=O)c1c(cc2n(c1=O)-c3ccccc3C2(C)C)O NRB05066 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1Cl)NC(=O)C RJC01538 c1cc(cnc1)/C=N/c2ccc(cc2Cl)Br RDR00848 c1cc2c(cc1/C=N/c3ccc(cc3Cl)Br)OCO2 RDR00850 CCN(CC)C(=S)Oc1c(cccc1Cl)Cl RDR00861 CCN(CC)C(=S)Oc1ccc(cc1)I RDR00866 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1F)F)NC(=O)C RJC01541 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C(=N/OC(=O)C3CC3)/N RF01377 Cc1ccc2c(c1)c(ncn2)Oc3c(cccn3)N RH00239 CC(=O)Nc1ccc(c(c1)C#N)F RH00243 Cc1ccc2c(c1)c(ncn2)O RH00231 CC1(c2cc(ccc2-n3c1cc(c(c3=O)c4ccccc4)O)Cl)C NRB05092 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1)NC(=O)c2ccccc2 RJC01559 c1ccc2c(c1)C(=O)C(C2=O)c3ccncc3 NRB05098 c1ccc2c(c1)/C(=N/N=C(N)N)/C(=O)N2 RJC01506 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)Cl)NC(=O)C RJC01536 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)Cl)NC(=O)C RJC01537 c1cc(ccc1/C(=C/C=C(C#N)C#N)/Sc2ccc(cc2)Cl)Cl NRB05107 Cc1cc(c(=O)[nH]n1)Cc2ccc(cc2)Cl RH00255 c1cc(cnc1)Nc2nnc(s2)C(F)(F)F RDR03354 c1cc(c(c(c1)Cl)C(=O)c2c(c3c(cc(nc3s2)c4cccs4)C(F)(F)F)N)Cl RF01515 Cc1ccc(cc1)S(=O)(=O)OCC23CCC(CC2)CC3 NRB02238 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)F)NC(=O)C RJC01529 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)F)NC(=O)C RJC01530 c1ccc(cc1)CCNC(=S)N/N=C/c2ccc(cc2)Cl RDR00817 CCOC(=O)C(C(F)(F)F)(NC(=O)Nc1ccccc1)O RJC01552 CC(NC(=S)N/N=C/C=N/NC(=S)NC(C)(C)C)(C)C RDR00920 c1cc(cnc1)/C=N/NC(=S)NCC2CCCO2 RDR00926 CN(C)CC1(CCCCC1)CC(c2cccc(c2)F)OC(=O)c3ccc(cc3)[N+](=O)[O-].Cl NRB02289 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)C RJC01539 CC(C)/C(=N\O)/c1ccc(cc1)[N+](=O)[O-] NRB02330 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1F)NC(=O)C RJC01531 c1ccc(c(c1)C(=O)c2cccs2)C(=O)O NRB02138 Cc1csc([n+]1C)NCc2cccnc2.[I-] RDR00575 c1cc(c(c(c1)Cl)Cl)NC(=S)Nc2ccc(cc2)S(=O)(=O)N RDR00592 CC1(CS/C(=N\c2cccnc2)/N1)CO RDR03315 CC12CC=C3c4ccc(cc4CCC3C1CCC2O)O NRB03796 CCOC(=O)NC(=S)Nc1cc(ccc1NC(=O)C)C(C)(C)C RF01563 CC(C)(C)c1ccc(cc1)c2ncc(s2)c3cccc(c3)[N+](=O)[O-] RH00250 CCOC(=O)c1c(n(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O RF01470 CN(C)/C=N/N=C/c1cc(cc(c1O)Cl)Cl RF01482 c1cc(ccc1C(=O)/C=C/S(=O)(=O)c2ccc(cc2)Br)Cl NRB05113 Cn1c2ccccc2c(c(c1=O)I)O NRB05093 Cc1ccc(cc1)C(=O)/C=C/Sc2[nH]c3ccc(cc3n2)C NRB05115 Cc1ccc2c(c1)nc([nH]2)S/C=C/C(=O)c3cccc(c3)Br NRB05118 CCc1ccc(cc1)C(=O)/C=C\Nc2ccc(cc2)OC(F)(F)F NRB05121 CC1\2CCC3C(C1CC/C2=N\NC(=O)N)CC=C4C3(CCC(C4)O)C NRB03731 CC(=O)C1CCC2C1(CCC3C2CC[C@@H]4[C@@]3(CCC(=O)C4)C)C NRB03854 CC(=O)c1ccc(cc1)OCC(=O)OC RH00257 Cc1cc(cc2c1C3CCC4(C(C3CC2)CCC4O)C)OC NRB03832 CC(=O)Nc1ccc(cc1)C(C)(C)C RF01502 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C)NC(=O)c2ccccc2 RJC01561 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)F)NC(=O)c2ccccc2 RJC01563 C/C=C(/c1ccccc1)\C(=N\O)\C NRB02305 CC(C)c1ccc(cc1)NCC(COc2ccc(c(c2)Cl)Cl)O RDR03298 c1ccc(cc1)c2cn3cc(cc(c3n2)Cl)C(F)(F)F RDR03299 c1ccc(cc1)C2OCC3(CO2)COC(OC3)c4ccccc4 NRB02254 c1ccc(cc1)C2=N/C(=C/c3ccc(o3)c4ccc(cc4Cl)Br)/C(=O)O2 RDR00724 Cc1c(c(=O)n(nc1C(=O)N/N=C/c2ccc(cc2)OC)c3ccc(cc3)C(C)(C)C)C#N RH00285 CC(c1ccccc1)NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)Cl RDR00913 c1ccc(cc1)CCNC(=S)N/N=C/c2ccc3c(c2)OCO3 RDR00818 Cc1c(c(ccn1)O)OCC(=O)OC.Cl RF01506 c1cc(ccc1/C(=C/C=C(C#N)C#N)/Sc2ccc(cc2)Cl)F NRB05106 c1cc(ccc1C2N[C@@H](CS2)C(=O)O)F NRB05175 Cc1c(c(no1)c2c(cccc2F)F)C(=O)ONC(=O)c3ccccc3 RF01536 c1cc(cnc1)/C=N/NC(=S)NCc2ccco2 RDR00921 c1cc(ccc1C(=O)/C=C/S(=O)(=O)c2ccc(cc2)Cl)F NRB05114 CCc1ccc(cc1)C(=O)/C=C/Sc2[nH]c3ccc(cc3n2)C NRB05116 c1c(cc(c(c1C(=O)O)N)Br)Br BTB01924 COc1ccc(cc1)/C=N/NC(=S)NCC2CCCO2 RDR00934 Cc1c(c(=O)n(nc1C(=O)NN)c2ccc(cc2)C(C)(C)C)C#N RH00282 c1cc(ccc1OCC(=O)O)OC(F)(F)F RDR03369 CC(C(=O)O)Oc1ccc(cc1)OC(F)(F)F RDR03370 c1cc(ccc1CS(=O)(=O)CC(COc2ccc(cc2)F)O)Cl RDR03437 c1ccc(cc1)n2c(n[nH]c2=S)c3cccc(c3)C(F)(F)F RDR03492 C([C@@H](C1[C@@H]([C@@H](C(=O)O1)O)O)O)O NRB05186 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1Cl)NC(=O)c2ccccc2 RJC01568 c1ccc(cc1)c2c(cnn2c3ccccc3)c4nnnn4c5ccc(cc5)I NRB05146 c1cc(oc1)Cn2c(cc(nc2=S)N)O RDR00859 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)Cl)NC(=O)c2ccccc2 RJC01566 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C)NC(=O)c2ccccc2 RJC01562 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)F)NC(=O)c2ccccc2 RJC01564 Cc1ccc(cc1)/C(=N/OC(=O)c2ccc(cc2)[N+](=O)[O-])/C(C)C NRB02324 COc1cccc(c1)NC(=O)CCC(=O)O RDR01043 Cc1cc(n(c(=O)c1C#N)NC(=S)NC2CCCCC2)C RH00308 C1CCC(C1)NC(=S)NNC(=O)CC#N RH00312 Cc1cc(nc(n1)SCC(=O)c2ccc(cc2)F)O RDR00941 COC(=O)C(C(F)(F)F)(NC(=O)c1cccc(c1)C(F)(F)F)O RJC01594 Cc1c(cnc(n1)N)c2nnnn2c3ccc(cc3)c4ccccc4 NRB05130 CC(C)CC(C(=O)O)NC(=O)CN RJC01625 COc1ccc(cc1)/C(=C/c2cc(c(c(c2)OC)OC)OC)/C#N RDR00954 c1ccc2c(c1)c3c(c(c2O)Cl)nc4ccccc4n3 RDR00966 Cc1cc(n(c(=O)c1C#N)NC(=S)NC2CCCC2)C RH00317 c1cc(cnc1)n2c(n[nH]c2=S)c3ccc(cc3Cl)Cl RDR03494 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)Cc4ccccc4Br RJC01634 CC(C)(C)c1ccc(c(c1)[N+](=O)[O-])NC(=O)c2ccccc2 RF01718 CC(C)(C)c1ccc(c(c1)[N+](=O)[O-])NC(=O)CN2CCOCC2 RF01719 Cc1cc(=O)n2c(csc2n1)c3ccc(cc3)Cl RDR00973 c1ccc(cc1)COc2ccc(cc2)C(=O)N RF01745 c1cc(c(c(c1)Cl)CN2CSCC2=O)Cl RDR03419 C(O)[C@@H](O)[C@@H](O)[C@H](O)CO NRB05167 C([C@H]([C@@H]([C@@H](C(=O)[O-])O)O)O)O.[K+] NRB05170 C[C@@]1(CCC2C1(CCC3C2CCC4=C3CCC(=O)C4)C)O NRB03856 Cc1cc(cc2c1C3CCC4(C(C3CC2)CC[C@]4(C#C)O)C)OC NRB03859 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)c2ccccc2 RJC01583 CC(=O)OC1CCC2(C3CCC4(C(C3CC([C@]2(C1)O)O)CCC4OC(=O)C)C)C NRB03863 Cc1cc(cc2c1C3CCC4(C(C3C=C2)CCC4=O)C)O NRB03864 c1cc(ccc1CC(=O)NCCNC(=S)Nc2ccc(cc2)Cl)O RDR03393 CC12CCC3c4ccc(cc4CCC3C1CCC2O)OC NRB03860 c1cc(sc1C#N)[N+](=O)[O-] RF01682 CC(=O)C1CCC2C1(CCC3C2CCC4[C@@]3(CCC(=O)C4)C)C NRB03874 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1)OC(C)C RJC01579 CCOC(=O)c1cnn(c1/N=C/N(C)C)c2ccc(cc2)[N+](=O)[O-] RH00296 Cc1cccn2c1nc(c2)c3ccccc3Cl.Br RDR01056 CC(=O)Nc1nc(cs1)c2ccc3ccccc3c2 RDR01058 C1CCC(CC1)NC(=S)NNC(=O)CC#N RH00307 CC(C)(C)NC(=S)N/N=C/c1cc(c(c(c1)Br)O)Br RDR01070 c1ccc(cc1)c2c(cn[nH]2)c3nnnn3c4ccc(cc4)Br NRB05151 CCOC(=O)c1cnn(c1N)c2ccc(cc2)[N+](=O)[O-] RH00289 c1cc(c(c(c1)Cl)S/C=C/C(=O)c2ccc(cc2)F)Cl NRB03908 Cc1cc(oc-2cc3ccccc3c12)c4ccccc4 NRB03911 c1cc(ccc1C(=O)/C=C/Sc2ccc(cc2)Cl)Cl NRB03903 c1cc(c(c(c1)Cl)S/C=C/C(=O)c2ccc(cc2)Cl)Cl NRB03904 COc1ccc(cc1)C(=O)O/C=C/C(=O)c2ccccc2 NRB03913 CC(=O)O[C@H]1[C@@H]([C@H](O[C@H]([C@@H]1OC(=O)C)OC(=O)C)C(=O)OC)OC(=O)C NRB05157 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)Cc4ccc(c(c4)Cl)Cl RJC01632 CN(C)c1ccc(cc1)/C=N/OC(=O)Nc2ccc(cc2)C(F)(F)F RF01644 Cc1c(c(=O)cco1)OCc2ccc(cc2)Cl RF01785 CC1=NC2N(C(=O)C1)C(=CS2)c3ccccc3Cl RDR00976 Cc1ccc(cc1C)NC(=O)/C=C/C(=O)O RDR01082 c1cc(ccc1C(F)(F)F)NC(=O)O/N=C/c2ccc(cc2Cl)Cl RF01639 c1cc(c(c(c1)Cl)/C=N/OC(=O)Nc2ccc(cc2)C(F)(F)F)Cl RF01640 CC(C1CCC2C1(CCC3C2CC[C@@]4(C3(CC(=C)CC4)C)C)C)O NRB03895 CCOC(=O)c1ccc(cc1)OCc2ccccc2 RF01741 c1ccc(cc1)O[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)CO)O)O)O NRB05164 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2cccc(c2)F RDR01072 CC(C)(C)OC(=O)N[C@@H](CCCNC(=N)N)C(=O)O.Cl RJC01690 c1cc(ccc1C(F)(F)F)NC(=O)O/N=C/c2ccc(c(c2)Cl)Cl RF01641 CC12CCC3c4ccc(cc4C=CC3C1CCC2=O)O NRB03890 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)Cc4ccc(cc4)[N+](=O)[O-] RJC01636 c1cc(ccc1c2cc3c(c(nnc3O)N)c(n2)O)Cl RF01704 CC(=O)OC1CCC2(C3CCC4(C(C3CC=C2C1)CCC4OC(=O)C)C)C NRB03882 c1cc(cc(c1)NC(=O)C(Cl)(Cl)Cl)c2cc(no2)c3c(cccc3Cl)Cl RF01973 Cc1ccc(cc1)n2c(nnn2)c3cnc(nc3c4ccccc4)N NRB05131 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3c(cccc3Cl)Cl)\[N+](=O)[O-] RF01707 Cc1c(cnn1c2ccccc2)c3nnnn3c4ccc(cc4)Cl NRB05147 C[C@@]1(CCC2C1(CCC3C2C=CC4=CC(=O)CCC34C)C)O NRB03899 COc1ccc(cc1)C(=O)C2=NNCC2c3c4ccccc4cc5c3cccc5 RJC01645 c1ccc2c(c1)cc3ccccc3c2C4CNN=C4C(=O)c5ccc(cc5)F RJC01646 c1cc(cc(c1)[N+](=O)[O-])/C=N/OC(=O)Nc2ccc(cc2)C(F)(F)F RF01643 c1ccc2c(c1)cc3ccccc3c2C4CNN=C4C(=O)c5cccc(c5)Br RJC01647 Cc1cc2c(cc1C)nc3c(n2)c4ccccc4c(c3Cl)O RDR01044 c1c(c(=O)c(cn1CCC#N)Cl)Cl RF01799 c1ccc(cc1)C2CNN=C2C(=O)c3ccc4c(c3)ccc5c4cccc5 RJC01658 c1ccc(cc1)C2CNN=C2C(=O)c3cc4ccccc4c5c3cccc5 RJC01661 CCOC(=O)Cn1cc(c(=O)c(c1)Cl)Cl RF01795 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)Cc4cccc(c4)Br RJC01635 c1ccc(c(c1)/C=N/c2nc[nH]n2)O RDR01052 Cc1ccc(cc1C)/N=C/c2cc(c(c(c2)OC)OC)OC RDR01062 Cc1ccc2c(c1)cc3c(n2)c4ccccc4oc3=O NRB03943 c1ccc2c(c1)cc3ccccc3c2C4CNN=C4C(=O)c5ccc(cc5)Br RJC01648 Cc1ccc(cc1)/C=N/NC(=S)Nc2ccc(cc2)OC RDR01066 c1cc(cc(c1)F)NC(=O)CCC(=O)O RDR01085 c1cc(ccc1n2c(c(cn2)C(=O)O)N)[N+](=O)[O-] RH00303 Cc1cc(cc(c1Br)C)CO RH00248 CC(=O)Nc1ccc(cc1)I RH00230 Cc1ccc(c2c1CCC2)OC(C)(C)C(=O)OC RH00233 Cc1cc(n(c(=O)c1C#N)NC(=S)NC2CCCCCC2)C RH00314 CN(C)c1ccc(cc1)/C=N/NC(=S)Nc2cccc(c2Cl)Cl RDR01019 C1CCCC(CC1)NC(=S)NNC(=O)CC#N RH00313 c1ccc(cc1)/C=C/C=C/c2ccccc2 NRB02401 CC(C)c1cc(c(c(c1)C(C)C)[N+](=O)[O-])C(C)C NRB02403 c1ccc(cc1)C2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)O2 RDR00751 c1cc(ccc1C(F)(F)F)N2CSCC2=O RDR03365 CC(=NOC(=O)Nc1ccc(cc1)C(F)(F)F)C RF01635 c1ccc(cc1)CS(=O)(=O)CC(COc2ccc(cc2)F)O RDR03438 c1cc(cc(c1)C(F)(F)F)CSCCNC(=O)N2CCSCC2 RDR03441 CC1CN(CC(O1)C)C(=O)NCCSCc2cccc(c2)C(F)(F)F RDR03442 COC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1F)O RJC01592 COC(=O)C(C(F)(F)F)(NC(=O)c1c(cccc1F)F)O RJC01593 Cc1c(c(nc(n1)C2CC2)O)Cl RF01712 CCNC(=S)N/N=C/c1cc(c(c(c1)OC)OC)OC RDR01094 c1cc(cnc1)/N=C/c2ccc(cc2)Cl RDR01095 CC(=O)Nc1ccc(c(c1)Cl)Cl RDR01104 c1cc(ccc1C(=O)/C=C/S(=O)(=O)c2ccc(cc2)Cl)Br NRB05104 CCOC(=O)c1c(c(c(=O)n(n1)c2ccc(cc2)C(C)(C)C)C#N)C RH00280 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C(/Cc3ccc(cc3)C(C)(C)C)\N RF01770 c1ccc(cc1)C23CC4CC(C2)CC(C4)C3 NRB02356 CCn1c2ccccc2c(c(c1=O)C)O NRB02368 CCn1c2ccccc2c(cc1=O)O NRB02371 CC12CCC3c4ccc(cc4CCC3C1CCC2=O)OC NRB03887 CCOC(=O)COc1cccc(c1)C(=O)C RH00263 CCN(CC)C(=S)Oc1ccc(cc1)[N+](=O)[O-] RDR00862 CCOC(=O)C(C(F)(F)F)(NC(=O)C)N1CCCCC1 RJC01542 c1cc2c(nc1)sc(n2)Sc3c(cccn3)[N+](=O)[O-] RH00335 c1cc2c(c(c1)F)c(=N)n(cn2)NC(=O)c3ccncc3 RH00336 CCOC(=O)c1c(c2c(cc(cc2o1)C)C)C RDR01030 CCOC(=O)c1ccc(cc1)Nc2nc(cs2)c3ccc4ccccc4c3 RDR01029 Cc1cc(cc2c1C3CCC4(C(C3C=C2)CCC4O)C)OC NRB03880 CC1=C(Sc2ccccc2N1)C(=O)Nn3cnc4cccc(c4c3=N)F RH00341 c1ccc(cc1)CC(C(=O)O)NC(=O)CN RJC01601 c1cc(cc(c1)C(F)(F)F)CSCCNC(=O)Nc2cccc(c2)C(F)(F)F RDR03443 CC1C(=O)N/C(=N\N=C(C)C)/S1 RF01457 CC(=O)OC1CCC2(C3CCC\4(C(C3CC=C2C1)CC/C4=N\NC(=O)N)C)C NRB03846 CC(=O)O[C@]1(CCC2C1(CCC3C2CCC4=CC(=O)C(=C)CC34C)C)C NRB03849 COC(=O)C(C(F)(F)F)(NC(=O)c1cccc(c1)Cl)O RJC01591 CC(C)(C)c1ccc(c(c1)[N+](=O)[O-])NC(=O)C(Cl)(Cl)Cl RF01617 CC(C)(C)c1ccc(c(c1)Cl)NC(=O)C2CC2 RF01618 COC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1)O RJC01589 Cc1cccc(c1NC(=O)NCCSCc2c(cccc2Cl)Cl)C RDR03427 Cc1c(c(nc(n1)C(C)(C)C)O)Cl RF01713 CC(C)(C)c1ccc(c(c1)N)NC(=O)c2ccco2 RF01715 CC(C)(C)c1ccc(c(c1)NC(=O)c2ccco2)NC(=O)CN3CCOCC3 RF01726 Cc1cccc(c1)C(CC2(CCCCC2)CN(C)C)OC(=O)c3ccc(cc3)[N+](=O)[O-].Cl NRB02291 CC(=C(c1ccc(cc1)N(C)C)/C(=N/O)/C)C NRB02308 C/C=C(\c1ccccc1)/C(=N/OC(=O)c2ccc(cc2)[N+](=O)[O-])/C NRB02309 c1cc(ccc1/C=N/NC(=S)NCC2CCCO2)Cl RDR00927 c1cc2c(cc1C(F)(F)F)nn[nH]2 RH00264 c1ccnc(c1)/C=N/OC(=O)Nc2ccc(cc2)C(F)(F)F RF01636 Cc1ccc(cc1)S(=O)(=O)N2CC3CCCC2C3 NRB02395 c1cc(cc(c1)F)NC(=O)/C=C/C(=O)O RDR01086 c1ccc(cc1)CNS(=O)(=O)c2ccc-3c(c2)Cc4c3ccc(c4)S(=O)(=O)NCc5ccccc5 RJC00500 CC(C)(C)c1ccc(c(c1)NC(=O)c2cccs2)NC(=O)CN3CCOCC3 RF01727 Cc1ccc(cc1)/N=C\2/N(C(=O)C3(S2)CC3)c4ccc(cc4)C RDR03390 Cc1cc(nc(n1)SCC(=O)c2ccc(cc2)Cl)O RDR00962 Cc1ccc(cc1)S/C=C/C(=O)c2ccc(cc2)Cl NRB03906 Cc1ccc(c2c1CCC3C2CCC4(C3CCC4=O)C)OC NRB03872 c1cc(ccc1C(=O)/C=C/Sc2ccc(cc2)Cl)I NRB03909 CN(C)/C=C/c1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] RH00292 c1cc(c(cc1C(F)(F)F)C(=O)O)F RH00293 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1)OCc2ccccc2 RJC01580 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1)OCc2ccc(cc2)F RJC01581 C[C@@]1(CCC2C1(CCC3C2CC[C@@H]4C3(CC(=C)CC4)C)C)O NRB03881 c1ccc(cc1)CCNC(=S)N2CCOCC2 RDR01143 c1cc(cc(c1)F)NC(=S)N2CCOCC2 RDR01145 CCOC(=O)CSc1nc2c3ccccc3c4ccccc4c2nn1 NRB02591 Cc1cccc(c1n2c(nnn2)SCC=C)C RDR01149 c1ccc2c(c1)cc([nH]2)c3ccccc3Cl RDR01153 c1ccc(cc1)C2C(=O)c3cccc4c3c(ccc4)C2=O NRB05242 c1cc(ccc1COc2ccc(cc2)/C(=N/OC(=O)C(Cl)(Cl)Cl)/N)Cl RF01859 CS/C(=N\C#N)/NCc1ccco1 RF01966 CSc1cccc(c1)NC(=O)CCC(=O)O RDR01116 CCn1c(n[nH]c1=S)C(c2ccccc2)O RJC00520 c1cc(oc1)C(=O)Nc2cc(c(cc2F)Br)F RDR03538 CC(=O)N[C@@H](Cc1ccc(cc1)OC(=O)C)C(=O)O RJC01674 CCOC(=O)c1cc(no1)c2c(cccc2Cl)Cl RF02000 Cc1cc(=O)c2nncn2[nH]1 NRB05215 c1c2c(cc3c1C(=O)CCO3)OCCC2=O NRB05219 CSc1cccc(c1)NC(=O)/C=C/C(=O)O RDR01117 COc1ccc(c(c1)NC(=O)/C=C/C(=O)O)OC RDR01127 c1ccc(cc1)Cc2c(c3ccccc3n(c2=O)c4ccccc4)O NRB05249 CC(=O)Nc1cccc(c1)c2cc(no2)c3c(cccc3Cl)Cl RF01870 CC(C)CC(c1ccccc1)C(=O)c2ccccc2 NRB02493 CCC(C)c1cc(nc2n1c3ccccc3n2)N NRB02556 C1C2CC3CC1CC(C2)OC3=O NRB02502 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)OC2C3CC4CC(C3)CC2C4 NRB02503 c1cc(ccc1C(=O)CSC(=O)N2CCOCC2)Cl RF01922 c1ccc(cc1)C(C(CO)N2C(=O)c3ccccc3C2=O)O NRB03979 CCCCN1CCC(CC1)(C#N)O RJC00496 CC(=O)CCCCn1c(=O)c2c(ncn2C)n(c1=O)C RJC01667 COc1ccc(cc1C(=O)NCCc2ccc(cc2)S(=O)(=O)NC(=O)NC3CCCCC3)Cl RJC01668 COc1cc2c(cc1OC)nc([nH]2)C=C NRB05222 COc1ccc2cccc3c2c1C=CC3=O NRB05226 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2cc(c(cc2OC)Cl)OC RDR01132 c1cc(c(c(c1)Cl)Cl)NC(=O)CCC(=O)O RDR01139 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Oc2ccc(cc2OC)C3N(CCS3)C(=O)NC)OC(=O)C)OC(=O)C)OC(=O)C NRB03998 Cc1cccc(c1C)Nc2c(cncn2)C#N NRB05231 Cc1cccc(c1n2c(=S)[nH]nn2)C RDR01146 Cc1cccc(c1n2c(nnn2)SC)C RDR01147 c1ccc2c(c1)C(=O)C(C(=O)N2)(Cl)Cl NRB05243 c1ccc2c(c1)cc([nH]2)c3ccc(cc3)Cl RDR01154 c1cc(ccc1COc2ccc(cc2)/C(=N/OC(=O)C3CC3)/N)Cl RF01867 COC(=O)c1c(noc1C(=O)NN)c2c(cccc2Cl)Cl RF02043 COc1cc(cc(c1)OC)NC(=S)NNC(=O)CSc2nc3cccnc3s2 RH00360 CC1=NC=CC2C1C=C(C(=O)N2)C#N RH00361 CCc1c(c2ccccc2n(c1=O)c3ccccc3)O NRB05269 CCc1ccccc1NC(=S)NNS(=O)(=O)c2ccc(cc2)C RDR01207 CC(Cc1cccc(c1)O)(C(=O)O)N RJC01671 CC(C)(C)C(=O)Nc1cccc(c1)c2cc(no2)c3c(cccc3Cl)Cl RF01981 CC(Cc1ccc(cc1)O)(C(=O)OC)N.Cl RJC01672 CCCCCCCCCCCCNC(=O)C(=O)c1ccccc1NC(=O)C(=O)Nc2ccccc2C(=O)C(=O)NCCCCCCCCCCCC NRB02477 c1cc(ccc1C(=O)CSC(=S)N2CCOCC2)Cl RF01946 CC1([C@@H](NC(S1)[C@H]([C@@H]([C@@H](CO)O)O)O)C(=O)O)C NRB03989 CC1([C@@H](NC(S1)c2ccc(cc2)Cl)C(=O)O)C NRB03990 COc1ccc(cc1)c2c(c(=S)[nH]c(n2)SC)C#N NRB02566 CC(=O)O[C@H]1[C@@H](Oc2ccccc2C1=O)c3ccccc3 RJC01641 Cc1ccc(cc1)C(=O)C2=NNCC2c3c4ccccc4cc5c3cccc5 RJC01644 c1ccc(cc1)C(=O)CC(c2ccsc2)SC(=S)N RDR03555 c1ccc(cc1)C2C=C(NC(=S)N2)c3ccccc3 RDR03562 c1cc(ccc1/C(=N/O)/N)OCc2ccc(cc2Cl)Cl RF01893 CC(C)c1ccc(cc1)S(=O)(=O)NNC(=O)CSc2nc3cccnc3s2 RH00366 c1ccc(cc1)c2cc(nc3n2c4ccccc4n3)N NRB02554 CC(=O)NC(COC(=O)C)C(c1ccc(cc1)[N+](=O)[O-])OC(=O)C NRB03971 C(C1C2[C@@H]([C@@H]([C@H](O1)OC3[C@@H]([C@@H]([C@@H](OC3CO)OC4[C@@H]([C@@H]([C@@H](OC4CO)OC5[C@@H]([C@@H]([C@H](OC5CO)OC6[C@@H]([C@@H]([C@@H](OC6CO)OC7[C@@H]([C@@H]([C@@H](OC7CO)OC8[C@@H]([C@@H]([C@@H](OC8CO)OC9[C@@H]([C@@H]([C@@H](O2)OC9CO)O)O)O)O)O)O)O)O)O)O)O)O)O)O)O)O)O RJC01701 c1ccc2cc(ccc2c1)c3c(c4ccccc4[nH]3)/C=C/[N+](=O)[O-] RDR01166 c1ccc(cc1)NNC(=S)Nc2cccc(c2)F RDR01179 Cc1ccc(cc1)S(=O)(=O)Oc2c3ccccc3[nH]c(=O)c2Cc4ccccc4 NRB05250 c1cc(c(c(c1)F)c2[nH]nc(n2)c3ccncc3)N RH00343 CC(=O)N1C2C(=O)OCC1(SC2(C)C)[C@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C NRB03993 CC(=O)N1[C@@H](SC([C@@H]1C(=O)O)(C)C)c2cccc(c2)[N+](=O)[O-] NRB03994 c1ccc2c(c1)[nH]c(n2)c3cccc(n3)c4[nH]c5ccccc5n4 NRB03961 CN(c1ccccc1)c2[nH]c(=O)c(c(n2)c3ccc(cc3)OC)C#N NRB02573 c1ccc(c(c1)C(=O)N\2C(=O)CS/C2=N\c3ccc(cc3)Cl)Cl RF02002 c1cc(c(c(c1)Cl)C(=O)NC(=S)Nc2ccc(cc2)Cl)F RF02005 CCCCCCCCOc1ccc(cc1)c2nnc(s2)COc3ccc(cc3)OCCCCCCCC RJC00516 c1ccc(cc1)NC(=O)c2cc(cc3c2-c4ccc(cc4C3=O)[N+](=O)[O-])[N+](=O)[O-] RJC01711 c1ccc(cc1)c2c(c(=S)[nH]nc2c3ccccc3)C#N NRB05209 c1ccc2cnc(cc2c1)/N=C/c3cc(cc(c3O)Cl)Cl NRB03963 c1ccc(c(c1)/C=N/c2ccc(cc2Cl)Br)Cl RDR01206 c1ccc(cc1)c2c(c3ccccc3oc2=O)O NRB05261 Cc1ccc(cc1)/C=C/2\CCCC(C2=O)CN(C)C.Cl NRB03968 c1cc(ccc1C[C@@H](C(=O)O)N)[N+](=O)[O-] RJC01694 COc1ccc2c(c1)nnc(n2)NN NRB04013 c1ccc2cnc(cc2c1)C(=N)c3ccc(cc3)Cl NRB04019 c1ccc(cc1)COC[C@@H](C(=O)O)N RJC01683 CC(C)CC(c1ccccc1)C(c2ccccc2)O NRB02489 c1cc(c(nc1)Sc2nc3cccnc3s2)N RH00380 c1cc2c(nc1)sc(n2)SCC(=O)NN RH00353 c1ccc2c(c1)nc(s2)Cc3nc4ccccc4s3 RJC00512 CCOc1c2cc(c(cc2ncc1C(=O)OCC)Cl)F RH00367 CC(=CC(=O)NNC(=O)CSc1nc2cccnc2s1)C RH00370 c1ccc(cc1)/C(=N\Oc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])/CNC(c3ccccc3)(c4ccccc4)c5ccccc5 NRB02472 COC(=O)C(c1ccc(cc1[N+](=O)[O-])Cl)C(=O)OC RH00373 c1ccc2c(c1)ccc3c2cc(cc3)C(=O)C4=NNCC4c5c6ccccc6cc7c5cccc7 RJC01649 c1ccc2c(c1)cc3ccccc3c2C4CNN=C4C(=O)c5cc6ccccc6c7c5cccc7 RJC01650 c1ccc(c(c1)/C=N/c2cccnc2)O RDR01096 c1ccc2c(c1)n3c(=O)c(cnc3s2)C(=O)O RDR03470 CO[C@@H]1[C@H]([C@H]([C@@H]([C@H](O1)CO)O)O)O NRB05166 c1cc(cc(c1)C(F)(F)F)CSCCNC(=O)Nc2ccc(cc2)OC(F)(F)F RDR03430 CC(=O)C(CCC#N)(CCC#N)C(=O)OC NRB02544 CCOC(=O)c1c(c(n[nH]c1=O)c2ccccc2)c3ccccc3 NRB05214 c1ccc2c(c1)ccc(n2)N=Cc3cc(cc(c3O)Cl)Cl NRB03965 Cc1cc(c(cc1C)NC(=O)/C=C/C(=O)O)C RDR01126 C=CCn1c2ccccc2c3c1ccc(c3)c4ccc5c(c4)c6ccccc6n5CC=C NRB03958 Cc1ccc(cc1)CS(=O)(=O)CC(COc2ccc(cc2)F)O RDR03435 Cc1cc(n(c(=O)c1C#N)NC(=S)NC2CC3CC2C=C3)C RH00318 Cc1cc(n(c(=O)c1C#N)NC(=S)NCc2cccs2)C RH00319 C[C@@]1(CCC2C1(CCC3C2CCC4=CC(=O)CCC34C)C)O NRB03896 Cc1ccc(cc1)S(=O)(=O)N(CCC=C)C(C)C NRB02440 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2nc3cccnc3s2 RH00350 Cc1cc(c(cc1C)NC(=O)CCC(=O)O)C RDR01128 C([C@@H]1[C@H]([C@@H]([C@H]([C@H](O1)OC[C@@H]2[C@H]([C@@H](C(O2)(CO)O)O)O)O)O)O)O NRB05188 Cc1ccc(cc1)CS(=O)(=O)CC(COCc2ccc(cc2)OC)O RDR03472 Cc1ccc(cc1)C(=O)/C=C/C=C/C=C/N(C)C NRB05220 Cc1cc(ccc1Br)NC(=S)N2CCOCC2 RDR01141 Cc1cc(ccc1NC(=S)N2CCOCC2)Br RDR01142 Cc1ccc(cc1)S(=O)(=O)O[C@H]2[C@H]3[C@@H](CO[C@H](O3)c4ccccc4)O[C@@H]([C@@H]2OS(=O)(=O)c5ccc(cc5)C)OC NRB05189 CO[C@H]1[C@H]([C@@H]([C@@H](CO1)O)O)O NRB05195 CC(C(=O)Nc1ccc(cc1)OC(F)(F)F)Oc2ccc(cc2)OC(F)(F)F RDR03488 Cc1ccc(cc1)S(=O)(=O)OC[C@@H]2CC3CCC2[C@@H](C3)OS(=O)(=O)c4ccc(cc4)C NRB02411 c1ccc(cc1)c2ccc(cc2)c3csc(n3)NC(=O)c4cc(ccc4O)Cl RDR01109 c1ccc(cc1)COc2ccc(cc2)C#N RF01818 c1cc(ccc1OCC(=O)NN)OC(F)(F)F RDR03498 CN(C)/C=C(/C(=O)OC)\NC(=O)c1ccccc1 RJC00511 c1cc2cc(ccc2cc1CC#N)CC#N NRB05225 c1ccc(cc1)CNC(=O)c2cc(cc3c2-c4ccc(cc4C3=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] RJC01714 CN(C)/C=C/C=c/1\c2cccc3c2c(c1=O)ccc3 NRB05227 Cc1ccc(cc1C)NC(=S)NNC(=O)CSc2nc3cccnc3s2 RH00358 c1cc2c3c(c1)c(cc(=O)n3CCC2)O NRB02372 COc1ccc2c(c1)[nH]c(=O)c(c2O)c3ccccc3 NRB02373 c1ccc2c(c1)c(=O)c3ccccc3[nH]2 NRB02376 COc1ccc(cc1)COCC(CS(=O)(=O)Cc2ccccc2)O RDR03471 CC(C)(CO)NCC(COc1ccc(cc1)F)O RDR03479 CCCCN(C)C(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC00507 c1cc(cc(c1)NC(=O)CCC(=O)O)C(F)(F)F RDR01118 COc1ccc(cc1)CNC(=O)CSc2nc3cccnc3s2 RH00355 COc1ccc(cc1)C(=C2SCCS2)C#N RDR03512 c1c(cc(cc1C(F)(F)F)N2C(=O)CC3(C2=O)CCCC3)C(F)(F)F RDR03517 c1cc(ccc1C(=C2SCCS2)C#N)[N+](=O)[O-] RDR03513 c1ccc(cc1)SC(C(=O)Nc2cc(c(cc2F)Br)F)(F)F RDR03539 c1ccc2c(c1)nc(nn2)N/N=C/c3cc(cc(c3O)Cl)Cl NRB03964 c1cc(c(cc1N2C(=O)CC3(C2=O)CCCC3)Cl)Cl RDR03518 CC(C)(C)c1ccc(c(c1)Cl)NC(=O)C(Cl)Cl RF01611 CC(C)(C)c1ccc(c(c1)Br)NC(=O)C(Cl)Cl RF01612 CC(C)(C)c1ccc(c(c1)Br)NC(=O)C(Cl)(Cl)Cl RF01616 c1ccc(cc1)CSC([C@@H]([C@H]([C@H]([C@@H](CO)O)O)O)O)SCc2ccccc2 NRB05197 CC(C)C[C@@H](C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 NRB05198 CC(=O)N[C@@H](CC(=O)N)C(=O)OC NRB05216 Cc1ccc(cc1C)/N=C/c2ccccc2Cl RDR01130 c1cc(ccc1n2c(n[nH]c2=S)COc3ccc(cc3)OC(F)(F)F)Cl RDR03520 COc1ccc(c(c1)NC(=O)CCC(=O)O)OC RDR01129 COC(=O)C1=C(C2(CC(=C(C(C1)(C2)C(=O)O)O)C(=O)OC)C(=O)O)O NRB02512 C/C(=N\OC(=O)c1ccccc1)/c2ccc(cc2)[N+](=O)[O-] NRB02515 c1ccc(cc1)n2c(n[nH]c2=S)COc3ccc(cc3)OC(F)(F)F RDR03521 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)C(C)C RDR01157 Cc1ccc(cc1)S(=O)(=O)O[C@H]2CC3CCCC2C3 NRB02521 CO[C@@H]1[C@@H]([C@H]([C@@H](CO1)O)O)O NRB05191 CSc1nc2cccnc2s1 RH00330 c1ccc(cc1)CCNC(=S)N/N=C/c2ccccc2Cl RDR01112 CN(C)/C=C/C=C/C=C/C(=O)c1ccc(cc1)Br NRB05221 c1cc(ccc1c2c(c(=O)[nH]c(n2)Nc3ccc(cc3)Cl)C#N)Cl NRB02570 c1ccc(cc1)CSc2[nH]c(=O)c(c(n2)c3ccccc3)C#N NRB02577 c1ccc(cc1)N/C=C/2\CCCCC2=O NRB05230 c1ccc(cc1)c2c(c(nnc2c3ccccc3)N4CCOCC4)c5ccccc5 NRB05208 COc1ccc2c3c1cccc3C(=O)CC2 NRB05236 CC(C)(C)c1ccc(cc1)OC(=O)c2ccc(s2)[N+](=O)[O-] RF01744 CCOC(=N)c1ccc(s1)[N+](=O)[O-].Cl RF01771 c1cc(ccc1NC(=O)/C=C/C(=O)O)S(=O)(=O)Nc2nccs2 RDR01250 c1ccc2cc(ccc2c1)c3cc4ccccc4[nH]3 RDR01160 c1cc(c(cc1n2c(=O)c3ccc(cc3nc2S)Cl)Cl)Cl RDR01258 COc1cc(ccc1OS(=O)(=O)C)/C=N/NC(=S)Nc2ccc(cc2)F RDR01262 Cc1cc(ccc1Br)NC(=S)N2CCCCC2 RDR01218 c1cc(c(cc1NC(=S)N2CCCCC2)Cl)Br RDR01219 Cc1ccc(cc1C)NC(=S)N2CCCCC2 RDR01222 CCCOc1ccccc1/C=N/NC(=S)Nc2cccc(c2)F RDR01224 CCCOc1ccccc1/C=N/NC(=S)Nc2ccc(cc2)F RDR01225 CCCOc1ccccc1/C=N/NC(=S)NC(C)(C)C RDR01227 C/C(=N\O)/c1cc2ccccc2oc1=O NRB04000 c1cc(c(cc1NC(=O)/C=C/C(=O)O)Cl)Br RDR01193 CC(=O)Nc1ccc(cc1)c2ccccc2 RJC01733 CCc1ccccc1NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)Cl RDR01208 COc1cccc(c1)/N=C/c2cc(c(c(c2)OC)OC)OC RDR01209 CC(=O)OC[C@H]([C@@H]([C@@H]([C@H](C1N[C@H](C(S1)(C)C)C(=O)O)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB03992 c1cc-2c(cc1[N+](=O)[O-])C(=C(C#N)C#N)c3c2c(cc(c3)[N+](=O)[O-])C(=O)NC4CCCCC4 RJC01716 c1cc(c(cc1C(F)(F)F)NC(=S)N2CCOCC2)Cl RDR01191 CCOc1ccccc1/C=N/NS(=O)(=O)c2ccc(cc2)C RDR01192 CCCCNC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC01724 Cc1ccc(c(c1)C)C2C(=S)NN=N2 RDR01200 Cc1cc(c(c(c1)C)Nc2nc(cs2)c3ccc(cc3)[N+](=O)[O-])C.Br RDR01305 CCCCNc1nc(cs1)c2ccc(cc2)c3ccccc3.Br RDR01308 Cn1c2ccccc2c3c1ccc(c3)Cl RJC01741 c1ccc(c(c1)N)NC(=S)Nc2c(cccc2Cl)Cl RDR01215 CCCCN(C)CC(Cn1c2ccccc2c3c1cccc3)O RJC01743 CN(C)CC(Cn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br)O RJC01745 c1ccc2c(c1)c3ccccc3n2CC(CN4CCN(CC4)CC(Cn5c6ccccc6c7c5cccc7)O)O RJC01728 c1ccc(cc1)Cn2c3ccc(cc3c4c2c(cc(c4)Br)Br)Br RJC01731 c1cc2c(cc1Cl)c3cc(ccc3n2CC(CN4CCN(CC4)CC(Cn5c6ccc(cc6c7c5ccc(c7)Cl)Cl)O)O)Cl RJC01727 COC(=O)C1=NNC(=NN1)C(=O)OC NRB04029 CS/C(=N\C#N)/NCc1cccnc1 RF01964 COC(=O)c1c(noc1NC(=O)O/N=C(/c2c(cccc2Cl)Cl)\N)c3c(cccc3Cl)Cl RF02248 c1ccc2c(c1)C(=O)C(C2=O)c3ccc(cc3)Cl RJC01750 c1ccc2c(c1)C(=C(C2=O)c3ccc(cc3)[N+](=O)[O-])O RJC01754 CCOC(=O)c1c(c2c(nc(nc2s1)SC)c3ccc(cc3)OC)N NRB02584 c1ccc2c(c1)C(=C(C2=O)c3cccc(c3)[N+](=O)[O-])O RJC01753 c1cc(ccc1COc2ccc(cc2)/C(=N/OC(=O)C(Cl)Cl)/N)Cl RF01858 c1cc(c(cc1Cl)Cl)Oc2cnc(nc2)O RF01931 CC\1=NN(C(=O)/C1=C\c2ccccc2)C(=O)C(C)Oc3ccc(cc3Cl)Cl RJC00521 Cc1cc(nc2c1/C(=N\O)/CC(C2)(C)C)c3ccccc3 RJC00527 C1CCC(CC1)/N=C\2/N(C(=O)C3(S2)CC3)C4CCCCC4 RDR03601 CCCCCCCCCCN(CCCCCCCCCC)S(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)N(CCCCCCCCCC)CCCCCCCCCC)C2=C(C#N)C#N RJC01719 c1ccc2c(c1)cccc2C3C(=O)c4ccccc4C3=O RJC01756 c1ccc(cc1)Nc2ccc3ccccc3c2/N=N\c4ccccc4O NRB04026 c1ccc(cc1)C(=O)Nc2ccncc2 NRB04027 C=CCOc1cc(=O)[nH]c2c1cccc2 NRB05270 c1c(c(cc(c1F)Br)F)NC(=O)C(Cl)(Cl)Cl RDR03581 CC1=NN(C(=O)C1)c2ccccc2 NRB05254 CCOC(=O)C(C#N)N=C(C#N)C#N.c1ccncc1 NRB05264 COc1cc(ccc1OC(=O)c2ccc(c(c2)Cl)Cl)/C=N/NC(=S)Nc3cc(ccc3Cl)Cl RDR01239 Cc1cccc(c1C)C(=O)Nc2cc(c(cc2F)Br)F RDR03574 COc1cc(ccc1OC(=O)c2ccc(c(c2)Cl)Cl)/C=N/NC(=S)Nc3ccc(cc3)F RDR01240 CCCCCCCCCCCCCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC01707 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)N(CCO)CCO RJC01708 CCOC(=O)/N=C(/c1ccc(cc1)Cl)\c2cc3ccccc3cn2 NRB04047 CS/C(=N\C#N)/NCc1ccccn1 RF01965 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2c(cccc2Cl)Cl RDR01217 CCCOc1ccccc1/C=N/NC(=S)Nc2ccc(c(c2)C)C RDR01230 CCCOc1ccccc1/C=N/NC(=S)Nc2cc(ccc2Cl)Cl RDR01231 Cc1cc(=O)oc2c1C(=O)CC(C2)(C)C RJC00528 COc1cccc(c1)C(=O)Nc2cc(c(cc2F)Br)F RDR03570 c1cc(ccc1C(=O)Nc2cc(c(cc2F)Br)F)Cl RDR03572 c1cc(ccc1C(F)(F)F)/N=C\2/N(C(=O)C3(S2)CC3)c4ccc(cc4)C(F)(F)F RDR03605 c1cc2c(cc1Br)c3cc(ccc3n2CC(CN4CCN(CC4)CC(Cn5c6ccc(cc6c7c5ccc(c7)Br)Br)O)O)Br RJC01726 c1cc(cc(c1)/N=C\2/N(C(=O)C3(S2)CC3)c4cccc(c4)C(F)(F)F)C(F)(F)F RDR03606 Cc1cc(nc(n1)c2ccccn2)S RDR03752 CC(C(=O)O)NC(=O)c1ccc(cc1)Cl RJC00567 COc1ccc(cc1)NC(=S)NC(=O)c2c(cccc2F)F RF02016 c1cc(cc(c1)NC(=S)NC(=O)c2c(cccc2F)F)C(F)(F)F RF02017 Cc1ccc(cc1)S(=O)(=O)Oc2c3ccccc3n(c(=O)c2Cc4ccccc4)C NRB05245 CC(C)(C)NC(=O)c1cccc-2c1C(=O)c3c2cccc3 RJC01722 CCCNC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC01723 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)NCCO RJC01710 c1cc(cc(c1)Cl)/N=C\2/N(C(=O)C3(S2)CC3)c4cccc(c4)Cl RDR03607 c1ccc(c(c1)C(=O)NC(=S)Nc2ccc(cc2)Cl)Cl RF01991 Cc1cs/c(=N\c2ccc(cc2)OC)/n1C(=O)c3ccccc3Cl RF02010 CC(=O)CS/C(=N\c1ccc(cc1)Cl)/NC(=O)c2c(cccc2Cl)F RF02011 c1cc(c(c(c1)F)C(=O)NC(=S)Nc2ccc(cc2)Cl)F RF02015 Cn1c(nc2ccccc2c1=O)/C=C/C=C/N3CCCC3 NRB04062 c1ccc(cc1)SC(C(=O)NNC(=O)c2ccsc2)(F)F RDR03624 COc1cc(c(cc1Cl)OC)n2c(=O)c3ccccc3nc2SC RDR01277 CCOC(=O)c1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)Cl RDR01267 Cc1cc(ccc1n2c(=O)c3ccccc3nc2S)Br RDR01286 c1cc(ccc1c2csc(n2)/C=C/C=C/N3CCOCC3)Br NRB04056 c1ccc\2c(c1)CN(/C2=N/c3cccc(c3)[N+](=O)[O-])c4cccc(c4)[N+](=O)[O-] RJC00552 c1ccc(cc1)CCn2c(=O)c3ccccc3nc2S RDR01271 COc1ccccc1Nc2nc(cs2)c3ccc(cc3)[N+](=O)[O-].Br RDR01306 CNC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC00505 CCNC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC00506 c1ccc2cc(ccc2c1)c3csc(n3)NC(=O)c4cc(ccc4O)Br RDR01111 c1ccc(cc1)COc2ccc(cc2)/C(=N/OC(=O)C(Cl)Cl)/N RF01855 c1ccc2c(c1)c(=O)n3ccccc3n2 NRB04067 c1ccc(cc1)c2cc(ncc2c3ccccc3)/C=C/C=C/N4CCCC4 NRB04068 CCOC(=O)c1ccc(c(c1)/N=C/c2ccccc2O)Cl RDR01268 COc1cc(c(cc1Cl)OC)n2c(=O)c3ccccc3nc2SCC=C RDR01281 CSc1nc2ccccc2c(=O)n1CCc3ccccc3 RDR01275 c1cc(ccc1NC(=O)CCC(=O)O)S(=O)(=O)Nc2nccs2 RDR01288 Cc1cc(nc(n1)NC(=S)c2ccc(cc2)NC(=O)/C=C/C(=O)O)C RDR01289 CCOC(=O)c1c(c(=O)oc2c1c(nn2c3ccccc3)O)C RJC00532 c1ccc2c(c1)c3cc(ccc3n2CN4CCOCC4)Cl RJC01734 c1cc2c(cc1Cl)c3cc(ccc3n2CN4CCCCC4)Cl RJC01735 c1cc2c(cc1Br)c3cc(cc(c3n2CC(CN4CCNCC4)O)Br)Br.Cl.Cl RJC01736 c1cc2c(cc1Br)c3cc(ccc3n2CC(CN4CCNCC4)O)Br.Cl.Cl RJC01737 c1ccc(cc1)C(=O)/C=C/2\C(=O)Nc3c([nH]c(=S)[nH]c3=O)N2 NRB02588 c1ccc(cc1)COc2ccc(cc2)/C(=N/OC(=O)C(Cl)(Cl)Cl)/N RF01856 c1c(ccc(c1)Br)/C=C\2/C(=O)/C(=C/c3ccc(cc3)Br)/CCC2 NRB03969 CC(=O)NC(CO)C(c1ccc(cc1)[N+](=O)[O-])O NRB03972 c1ccc2c(c1)C(=O)N(C2=O)C(CO)C(c3ccc(cc3)[N+](=O)[O-])O NRB03975 c1ccc2c(c1)cc(c3c2cccc3)C4CNN=C4C(=O)c5cc6ccccc6c7c5cccc7 RJC01662 CCOCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC01747 c1ccc(cc1)/N=C\2/N(C(=O)C3(S2)CC3)c4ccccc4 RDR03613 c1ccc2c(c1)C(=O)C(C2=O)c3ccc(cc3)F RJC01749 Cc1cc(nc2c1c(nn2C)O)C RJC00535 C1C2CC3CC1CC(C2)(C3)C(=N)N.Cl RF02105 c1cc(c(c(c1)Cl)/C=N/OC(=O)Nc2csnc2c3c(cccc3Cl)Cl)Cl RF02130 c1ccc2c(c1)ccn3c2nnn3 NRB05288 C/C(=C\c1ccc(cc1)SC)/[N+](=O)[O-] P00093 CCCCCCCCN1CCC(CC1)CCCC2CCN(CC2)CCCCCCCC NRB02533 CSc1c(c(c(nn1)c2ccccc2)c3ccccc3)c4ccccc4 NRB05203 c1cc(cnc1)n2c(n[nH]c2=S)c3ccc(cc3)Cl RDR03493 c1ccnc(c1)NNC(=O)Nc2csnc2c3c(cccc3Cl)Cl RF02213 Cc1c(nc2ccccc2n1)O RF02078 CC(=O)Nc1ccc(cc1)c2ccc(cc2)NC(=O)C RJC01730 c1cc(c(c(c1)Cl)c2nsc(=O)o2)Cl RF02103 Cc1cc(nc(n1)C23CC4CC(C2)CC(C4)C3)O RF02106 COC(=O)c1c(nsc1C(=O)OC)c2c(cccc2Cl)Cl RF02114 c1ccc(c(c1)CSc2nc3cc(ccc3c(=O)n2c4ccc(c(c4)Cl)Cl)Cl)Cl RDR01317 Cc1cc(nc(n1)SCc2ccc(cc2)Cl)O RDR01323 Cc1c(cccc1Cl)Nc2nnc(s2)C RDR01325 c1ccc(cc1)c2[nH]c3cc4c(cc3n2)nc([nH]4)c5ccccc5 RJC00557 c1ccc(cc1)c2c(c(nnc2c3ccccc3)N4CCOCC4)C#N NRB05212 COc1cccc(c1OC)CNC(=O)CSc2nc3cccnc3s2 RH00364 c1cc2c(nc1)sc(n2)SCC(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RH00368 Cc1cc(ccc1S(=O)(=O)NNC(=O)CSc2nc3cccnc3s2)[N+](=O)[O-] RH00369 c1ccc(cc1)/C=C/C=C/c2nnn(n2)c3ccc(cc3)Cl NRB04091 c1ccc2c(c1)C=C(N3C2NN4C(N3)c5ccccc5C=C4C(=O)c6cccc(c6)C(F)(F)F)c7cccc(c7)C(F)(F)F NRB04099 CC1(CC2=C(C(Nc3ccccc3N2)c4ccco4)C(=O)C1)C RJC00548 Cc1ccnc(c1)/N=C/2\c3ccccc3CN2c4cc(ccn4)C RJC00550 CC(C)n1c(nnc1SCc2ccccc2)COc3ccc(cc3)OC(F)(F)F RDR03528 Cc1nnc(s1)NC(C)C RDR01353 c1ccc\2c(c1)CN(/C2=N/c3ccc(cc3)Cl)c4ccc(cc4)Cl RJC00551 CC(C)(C)NS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)NC(C)(C)C RJC01780 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3ccccc3Br RJC01784 Cc1c(cccc1[N+](=O)[O-])NC(=O)C2CCCCC2 RJC01789 CC1C(=O)N/C(=N/N=C\C23CC4CC(C2)CC(C4)C3)/S1 RF02150 c1ccc(cc1)C2=CC(SC(=S)N2)c3ccsc3 RDR03556 c1cc(ccc1OCc2n[nH]c(=S)o2)OC(F)(F)F RDR03524 CC(=O)OCc1ccc(c(c1OC(=O)C)OC(=O)C)COC(=O)C NRB02542 c1ccc(cc1)NS(=O)(=O)c2ccc-3c(c2)C(=O)c4c3ccc(c4)S(=O)(=O)Nc5ccccc5 RJC01779 c1ccc2cc(ccc2c1)c3csc(n3)/N=C/c4cc(cc(c4O)Cl)Cl RDR01299 Cc1c(cccc1[N+](=O)[O-])/N=C/N(c2cccc(c2C)[N+](=O)[O-])C(=O)c3ccccc3 RJC01786 CCOC(=O)c1c(c2c(nc(nc2s1)SC)c3ccc(cc3)Cl)N NRB02583 CSc1nc2c3ccccc3c4ccccc4c2nn1 NRB02589 c1ccc2c(c1)cc[n+](c2C(=O)c3ccc(cc3)Cl)[N-]C#N NRB04077 c1cnccc1C2N[C@@H](CS2)C(=O)O NRB03982 c1ccc(c(c1)/C=N/NC(=S)Nc2ccc(cc2)F)Cl RDR01113 c1cc2c(nc1)sc(n2)SCC(=O)c3ccc(cc3)Br RH00348 c1cc2c(nc1)sc(n2)SCC(=O)c3ccc(cc3)OC(F)(F)F RH00349 c1cc(c(c(c1)Cl)c2c(csn2)NC(=O)O/N=C(/c3c(cccc3Cl)Cl)\N)Cl RF02215 CCCCCCCCCCCC(=N)OC.Cl NRB05273 c1cc(cnc1)CNc2[nH]nc(n2)N RF02193 c1ccc(cc1)c2[nH]c(=O)cc(n2)O NRB05285 Cc1cc(c(c2c1sc(c2C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)OC)C)Cl PD00004 c1c(cnc(n1)N)Br RJC00628 c1ccc(cc1)CCNC(=S)Nc2ccc(cc2)NC(=O)c3ccccc3O RDR01431 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=S)Nc3ccc(c(c3)Cl)Cl)O RDR01433 CC1=CC[C@@H](CC1=O)C(C)(C)OC(=O)C RJC00604 CCOC(=O)c1cc2ccc3ccccc3c2s1 PD00012 CCN(CC)CCOC(=O)c1ccc(cc1)N[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)CO)O)O)O.Cl RJC00575 CCOc1c2ccccc2c3c(n1)nc(n3Nc4ccc(cc4)Br)c5ccc(cc5)OC NRB04090 Cn1c2c(c3c(c(=O)n2c4ccccc4)[n+](on3)[O-])c(=O)n(c1=O)C RJC01814 CCOC(=O)c1cnc(nc1N)S/C=C/C(=O)c2ccccc2 NRB04149 c1cc(c(cc1NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F)C#N RDR03708 c1cc(ccc1C2=NCCO2)NS(=O)(=O)c3ccc(cc3)Cl RDR03715 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=S)Nc3cccc(c3Cl)Cl)O RDR01434 COc1ccc(cc1)/C(=C/c2c(cccc2Cl)Cl)/C#N RDR01462 CC(=O)c1ccc(cc1)N2C(=O)c3ccccc3C2=O PD00209 c1cc2c(cc1Cl)C=C(CO2)C(=O)O RDR03723 COC(=O)CCC1CC2(CCC1=O)OCCO2 RJC01805 COC(=O)c1cccc(c1)CSC(=S)N2CCCC2 RDR03757 Cc1ccc(c(c1)Br)NC(=O)CCS(=O)(=O)Cc2ccccc2 RDR03759 CCOC(=O)NN(C1=CC(Oc2c1cccc2)c3ccccc3)C(=O)OCC NRB02669 c1ccc2c(c1)c(c[nH]2)/C(=C/c3ccc(cc3)F)/C#N PD00112 CC(C)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)N3C(=O)CCC3=O RDR03718 COc1ccc(cc1)CC2(CCC3(CC2)OCCO3)O RJC01800 c1ccc(cc1)C2C(NC(=N2)N)C(=O)c3ccccc3 NRB02691 COCCOC(=O)c1c(nccn1)C(=O)Nc2cc(cc(c2)OC)OC PD00083 Cn1c2ccccc2c(c(c1=O)[N+](=O)[O-])C(C(=O)OC)C(=O)OC RJC01812 c1ccnc(c1)/C(=C/c2ccc(cc2)C(F)(F)F)/C#N PD00103 CN(C)NC(=O)Nc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC RF02253 COC(=O)c1c(noc1NC(=O)NCc2ccccn2)c3c(cccc3Cl)Cl RF02258 c1cc2c(cc1Cl)C=C(CO2)C(=O)Oc3ccc(cc3Cl)Cl RDR03737 COC(=O)C1CN(CCC1=O)Cc2ccccc2 RJC01808 CCc1c(c2ccccc2n(c1=O)C)OS(=O)(=O)c3ccc(cc3)Br RJC01810 c1cc(ccc1NC(=O)C2=Cc3cc(ccc3OC2)Cl)Cl RDR03726 c1ccc2c(c1)ccc3c2sc(c3)C(=O)Nc4cccnc4 PD00020 CC(C)(C)c1ccc(cc1)N2C(=O)CC(C2=O)C/C=C/c3ccccc3 PD00068 c1cc(cc(c1)S(=O)(=O)N)NC(=O)Nc2cccc(c2)S(=O)(=O)N RJC00584 CC(=O)N1C(C(C(=N1)c2ccccc2OCc3ccccc3)OC(=O)C)c4ccc(cc4)OC NRB02695 COC(=O)c1c(noc1NC(=O)N/N=C/c2c(cccc2Cl)Cl)c3c(cccc3Cl)Cl RF02262 c1ccc2c(c1)c(=S)[nH]c(=S)[nH]2 PD00041 COc1ccc(cc1)C(C(=O)c2ccc(cc2)OC)O RJC00580 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3[nH]c(nn3)SC RF02295 COC(=O)c1cc(=O)nc(s1)N RF02299 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(o2)c3cccc(c3)[N+](=O)[O-] RDR01389 CC(=O)c1cc2ccccc2c3c1cccc3 RJC00601 c1ccc(cc1)C(=O)COC(=O)c2ccccc2Nc3ccccc3F RDR01412 c1ccc(cc1)C(=O)COC(=O)c2ccccc2Nc3cccc(c3)F RDR01413 c1ccn2cc(nc2c1)c3ccc(cc3)[N+](=O)[O-] RDR01384 COc1ccc(cc1)Oc2ccc(cn2)C(F)(F)F NRB02708 Cc1c(c(no1)c2c(cccc2Cl)F)C3=NCCO3 RDR03687 CN(C)c1ccc(cc1)c2nc3c(s2)C(=O)CCC3 RJC01794 c1ccc(cc1)CNCCNCc2ccccc2.Cl.Cl RJC00581 Cc1ccc(cc1)C2N[C@H](C(S2)(C)C)C(=O)O RJC00589 Cc1ccc(cc1C)NC(=O)c2ccccc2O RDR01397 Cc1ccc(cc1C)/N=C/c2ccc(o2)c3ccc(cc3)[N+](=O)[O-] RDR01374 Cc1cccc(c1n2c(nnn2)SCc3ccccc3Cl)C RDR01378 CO/N=C/1\CC(Oc2c1cccc2)c3ccccc3 NRB02662 c1c(cnc(c1Cl)N2C(=O)CSCC2=O)C(F)(F)F PD00059 CNC(=O)NNC(=O)c1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC RF02176 c1ccc(cc1)C2C/C(=N\OC(=O)Nc3cccc(c3)Cl)/c4ccccc4O2 NRB02663 c1cc(ccc1Oc2ccc(cn2)C(F)(F)F)Oc3ccc(cn3)C(F)(F)F NRB02709 Cc1cccc(c1NC(=O)C(C(F)(F)F)C(F)(F)F)C RDR03655 Cc1cccc(c1n2c(nnn2)SCc3ccc(cc3)Cl)C RDR01380 CCc1nnc(s1)NC(=O)c2ccccc2O RDR01382 COc1ccccc1C2(CCN(CC2)Cc3ccccc3)O RJC01804 c1ccc(cc1)NC(=O)c2cc3ccc4ccccc4c3s2 PD00015 c1cnccc1CN2C(=O)CSCC2=O PD00057 c1ccc(c(c1)C(=O)O)Nc2ccccc2F RDR01405 CCOC(=O)/C(=C/c1ccccc1)/C(=O)c2ccccc2OCc3ccccc3 NRB02625 COc1ccc(cc1)N2C(=O)c3c(nccn3)C2=O PD00073 CSc1nn2c(=O)c(nnc2s1)Cc3ccccc3 NRB04141 CC(Cc1c[nH]c2c1cccc2)(C(=O)OC)N RJC01802 COC(=O)c1c(noc1C(=O)NNC(=S)Nc2ccccc2)c3c(cccc3Cl)Cl RF02185 c1cc2c(cc1Cl)c(=S)[nH]c(=S)[nH]2 PD00042 c1cc(ccc1SC2CC(=O)N(C2=O)Cc3ccncc3)Cl PD00051 c1cc(cnc1)N2C(=O)CSCC2=O PD00055 CCSc1nnc2n1nc3c4ccccc4c5ccccc5c3n2 NRB04129 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)/C=N/NC(=S)NCc3ccco3 RDR01387 Cc1cc(c(cc1Cl)C)S(=O)(=O)N(/C=N/c2cccc(c2C)[N+](=O)[O-])c3cccc(c3C)[N+](=O)[O-] RJC01792 CSc1[nH]c(nn1)C23CC4CC(C2)CC(C4)C3 RF02165 c1ccc(cc1)COc2ccccc2C(=O)[C@@H]3[C@@H](N3C4CCCCC4)c5ccc(cc5)Cl NRB02656 CCOC(=O)CSc1nnc(c(=O)n1c2ccccc2)c3ccccc3 NRB04144 c1ccc2c(c1)ccc3c2sc(c3)C(=O)Oc4cccc(c4)C(F)(F)F PD00028 c1ccc(c(c1)/C=N/c2ccc(cc2)NC(=O)c3ccccc3O)Cl RDR01416 c1ccc2c(c1)C=C(N3C2NN4C(N3)c5ccccc5C=C4C#N)C#N NRB04100 CC(C)(C)NC(=S)N/N=C/c1ccc(o1)c2ccc(cc2)[N+](=O)[O-] RDR01371 CC(C)NC(=S)N/N=C/c1ccc(o1)c2ccc(cc2)[N+](=O)[O-] RDR01372 c1ccc(cc1)CSc2nnc3n2nc4c5ccccc5c6ccccc6c4n3 NRB04130 COC(=O)C1=CN2c3ccccc3SC2(C(=C1C(=O)OC)C(=O)OC)C(=O)OC PD00009 c1ccc(cc1)c2nc(c(=O)[nH]n2)Cc3ccc(cc3)Cl NRB04136 Cn1c(=O)c(c(nc1SC)c2ccc(cc2)Cl)C#N NRB04138 Cc1ccc(cc1)NC(=O)NNC(=O)c2cc3ccc4ccccc4c3s2 PD00025 c1cc-2c(cc1S(=O)(=O)N(CCO)CCO)Cc3c2ccc(c3)S(=O)(=O)N(CCO)CCO RJC01776 COc1ccc(cc1)/C=N/c2ccc(cc2)NC(=O)c3ccccc3O RDR01418 c1ccc(c(c1)C(=O)Nc2ccc(cc2)/N=C/c3ccco3)O RDR01422 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(o2)c3ccc(cc3)[N+](=O)[O-] RDR01373 c1cc(cc(c1)F)NC(=S)N/N=C/c2ccc(o2)c3ccc(cc3)[N+](=O)[O-] RDR01375 c1ccc2c(c1)/C(=C/C(=O)Oc3cc(cc(c3)Cl)Cl)/OC2=O RDR03694 c1ccc2c(c1)ccc3c2sc(c3)C(=O)N/N=C/c4ccc(cc4)C(F)(F)F PD00022 c1ccc2c(c1)-c3ccccc3C2=NNc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-] RJC01775 CCOC(=O)NC(=S)NC12CC3CC(C1)CC(C3)C2 RJC00588 c1cc(cnc1)Nc2nc(cs2)c3ccc(cc3)Cl RDR03652 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2ccc3c(c2)OCCO3 RDR01295 CCCCN(C)CC(Cn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br)O RJC01742 CC(=O)C1=C(c2cc(c(cc2C1=O)Cl)Cl)O RJC01758 CC(C)(C)/C=C(\C#N)/C(C)(C)C RJC01759 CC(C)(C)CC(C#N)(C(C)(C)C)O RJC01761 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCC(CC2)c3ccccc3OC RJC01785 C1C2CC3CC1CC(C2)(C3)C(=O)NNC(=S)N RF02154 C1C2CC3CC1CC(C2)(C3)c4[nH]c(nn4)S RF02159 CN(C)NC(=O)c1csnc1c2c(cccc2Cl)Cl RF02195 c1ccc2c(c1)ccc(n2)C(=O)c3cccc(c3)C(F)(F)F NRB04080 c1ccc2c(c1)nnc3n2c(nn3)SCC(=O)O NRB04082 CCCCN(C)CC(Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl)O RJC01744 CCCCN(C)CC(Cn1c2ccc(cc2c3c1ccc(c3)Br)Br)O RJC01746 CC(C(=O)O)NC(=O)c1ccc(cc1)[N+](=O)[O-] RJC00565 c1ccc(cc1)n2c(cc(=O)[nH]c2=O)N RJC00571 c1cc(oc1)CNC(=S)N/N=C/c2cc(c(c(c2)Br)O)Br RDR01354 CCOC(=O)Cn1c(noc1=O)c2c(cccc2Cl)Cl RF02238 c1cc(ccc1CSc2nc3cc(ccc3c(=O)n2c4ccc(c(c4)Cl)Cl)Cl)Cl RDR01318 CC(=O)N(c1cc2ccccc2cn1)N(C(=O)C)C(=O)C NRB04101 c1ccc2c(c1)ccc3c2sc(c3)C(=O)NNC(=O)c4ccc(cc4Cl)Cl PD00023 c1cc(ccc1c2cnc(s2)/C=C/C=C/N3CCOCC3)Br NRB04057 COc1cc(ccc1O)/C=N/NC(=S)NCc2ccco2 RDR01355 c1cc(c(c(c1)Cl)Cl)n2ccnc2S RDR01357 CC(=O)c1ccc(s1)[N+](=O)[O-] RJC00615 CSc1nnc(o1)c2cccs2 RDR03671 CC(=O)ON=C1c2cc(ccc2-c3c1cc(cc3)[N+](=O)[O-])[N+](=O)[O-] RJC01781 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl RJC01782 Cc1cc(nc(n1)SCc2ccccc2Cl)O RDR01322 COC(=O)c1cc(=O)n2c(c1C(=O)c3cccs3)SCC2 PD00063 c1cnc(c(n1)C(=O)Nc2cc(cc(c2)Cl)Cl)C(=O)O PD00070 COCCCNC(=S)Nc1c(cccc1Cl)Cl RDR01335 Cc1cc(nc(c1C(=O)C)NC(C)(C)C)NC(C)(C)C RJC00594 c1ccc(cc1)CNc2nc3c4ccccc4c5ccccc5c3nn2 NRB04125 c1ccc2c(c1)ccc(=O)n2Nc3ccc(cc3)Br NRB04059 Cc1ccc(cc1C)Nc2nnc(s2)C RDR01326 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3ccccc3[N+](=O)[O-] RJC01783 CC(=O)Nc1ccc(c(c1)C(F)(F)F)Br RDR03711 c1ccc2c(c1)C3(C(=O)N2CC4(CCC=CC4)C#N)OCCO3 RJC01793 CCOC(=O)c1cnc(nc1N)S/C=C/C(=O)c2ccc(cc2)Cl NRB04151 c1ccc(cc1)C(=O)/C=C/Sc2ccc(cn2)C(F)(F)F NRB04152 Cc1c(c(no1)c2ccccc2Cl)C3=NCCO3 RDR03686 Cc1c(cccc1[N+](=O)[O-])/N=C/N(c2cccc(c2C)[N+](=O)[O-])C(=O)C3CCCCC3 RJC01787 Cc1cccc(c1n2c(nnn2)SCc3ccc(cc3)Br)C RDR01377 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)/C=N/NC(=S)Nc3ccc(cc3)F RDR01385 c1cc(cc(c1)c2[nH]c3ccc(cc3n2)C(=O)O)c4[nH]c5ccc(cc5n4)C(=O)O.Cl RJC00559 COC(CNC(=S)Nc1cccc(c1Cl)Cl)OC RDR01347 c1cc(sc1)CNc2[nH]nc(n2)N RF02194 Cc1ccc(cc1)C(=O)NCCO RDR03640 c1ccc(cc1)COc2ccccc2C([C@H]3[C@@H](N3C4CCCCC4)c5ccc(cc5)Cl)O NRB02651 Cn1c2c(cc3cc(ccc3n2)F)c(=O)n(c1=O)C RJC01815 COC(=O)c1cc(=O)n2c(c1C(=O)c3ccc(cc3)Cl)SCC2 PD00061 c1cnc2c(n1)C(=O)N(C2=O)c3cc(cc(c3)Cl)Cl PD00071 c1ccc2c(c1)/C(=C/C(=O)Oc3cccc(c3)C(F)(F)F)/OC2=O RDR03693 c1cc(c(c(c1)Cl)c2c(csn2)C(=O)O/N=C(/c3c(cccc3Cl)Cl)\N)Cl RF02201 CCCC1C2C(C(=O)N(C2=O)c3ccccc3)ON1c4ccc(c(c4)Cl)Cl PD00034 CN(C)NC(=O)Nc1csnc1c2c(cccc2Cl)Cl RF02210 c1cc(c(c(c1)Cl)c2c(csn2)NC(=O)NN3CCCCC3)Cl RF02211 COC(=O)c1c(noc1C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-])c3c(cccc3Cl)Cl RF02175 c1c(cc(cc1C(F)(F)F)NC(=O)/C=N/O)C(F)(F)F P00217 c1ccc(cc1)Nc2nc3ccccc3c(=O)o2 P00256 c1ccc(cc1)COc2ccccc2C(=O)/C(=C\c3ccccc3)/n4ccnc4 NRB02626 c1ccc2c(c1)c3ccccc3c4c2nc(nn4)Nc5ccc(cc5)Cl NRB04123 COc1ccc(cc1)Nc2nc3c4ccccc4c5ccccc5c3nn2 NRB04124 c1ccc2c(c1)c3ccccc3c4c2nc(nn4)N5CCCCC5 NRB04126 c1cc(ccc1c2ccc(o2)/C=N/NC(=S)NCC3CCCO3)[N+](=O)[O-] RDR01363 Cn1c2ccccc2c(c(c1=O)Cc3ccccc3)OC(=O)c4ccccc4 NRB05272 c1cc(ccc1n2nc(nn2)/C=C/C=C/N3CCOCC3)Cl NRB04083 c1ccc(cc1)/C=C\2/C(=O)N(OC2=O)c3ccccc3 RJC00538 c1ccc(cc1)C(=O)COC(=O)c2cc3ccccc3cc2OC(=O)c4ccc(cc4)Cl RDR01490 c1ccc2cc(c(cc2c1)C(=O)OCC(=O)c3ccc(cc3)Cl)OC(=O)c4ccc(cc4)Cl RDR01491 c1cc(oc1C(=O)N)[N+](=O)[O-] RF02316 c1cc(ccc1N2C(=O)CCC2=O)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl RDR03720 c1cc(c(c(c1)Cl)CSC(=O)Nc2ccc(cc2)Cl)Cl RF02465 c1ccc2c(c1)ccc3c2sc(c3)C(=O)NCc4ccc(cc4)C(F)(F)F PD00019 c1ccc(cc1)C2Cn3c(nnn3)-c4ccccc4O2 NRB02673 c1ccc(cc1)C2CNC(=O)c3ccccc3O2 NRB02674 Cc1c(c(no1)c2ccccc2)C(=O)OCC(=O)c3ccccc3 RDR01483 COc1ccccc1/C=N/NC(=S)NCc2ccco2 RDR01452 c1cc(c(cc1NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F)Br RDR03703 CN(C)N/C(=N\O)/c1c(cccc1Cl)Cl RF02310 COc1ccc(cc1)C2C(C(=NN2)c3ccccc3OCc4ccccc4)O NRB02693 c1ccc2c(c1)c(cc(=O)o2)Sc3ccc(cc3)Cl NRB02735 Cn1cccc1/C(=C/c2cccc3c2cccc3)/C#N PD00118 CCC1(C(=O)c2cc3ccccc3cc2C1=O)CC NRB04174 c1cc(c(c(c1)Cl)NNC(=O)NS(=O)(=O)c2ccc(cc2)Cl)Cl RF02424 c1cc(ccc1S(=O)(=O)NC(=O)NNc2cc(cc(c2)Cl)Cl)Cl RF02425 c1ccc(c(c1)Nc2c(c(ns2)O)C#N)Cl RF02367 Cc1ccc(cc1Cl)NC(=S)C(C#N)C(=O)N RF02392 c1ccc(cc1)c2cc(=O)c3ccc(cc3o2)OCC#N NRB02680 c1ccc(cc1)c2cc(=O)c3c(o2)cc(cc3Cl)Cl NRB02681 CCOC(=O)c1ccc(cc1)c2cc(=O)c3ccccc3o2 NRB02682 c1ccc(c(c1)C(F)(F)F)NNC(=O)NS(=O)(=O)c2ccc(cc2)Cl RF02426 Cc1ccc2c(c1)nc([nH]2)S/C=C\C(=O)c3ccccc3 NRB04158 Cn1ccnc1S/C=C/C(=O)c2ccc(cc2)Cl NRB04164 Cn1cccc1/C(=C\c2ccc3c(c2)OCO3)/C#N PD00117 c1ccc(cc1)C(=O)CSc2c3ccccc3nc(n2)SCC(=O)c4ccccc4 PD00210 c1ccc2c(c1)c(=O)n3c(n2)SCC3 PD00216 Cc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3ccc(cc3)OC PD00091 c1ccc(cc1)N/N=C/c2c(c3ccccc3oc2=O)Cl NRB02736 CC(=O)/C(=N\Nc1ccccc1)/C(=O)OCc2ccccc2 NRB02739 Cc1cc(=O)[nH]c(n1)N/N=C/c2ccccc2O NRB04183 c1ccc(cc1)C(=O)/C=C/Sc2c(c(cc(n2)c3cccs3)C(F)(F)F)C#N NRB04155 COC(=O)C1=C(C(=C(C1=O)C(=O)OC)c2ccccc2)c3ccccc3 PD00096 CCCCCCCCCCCCCCc1c(nc(s1)N)c2ccccc2 RJC00645 C[C@]12CCCC(C1CC[C@@]3([C@@H]2CCO3)C)(C)C RJC00646 c1ccc2c(c1)c(nc(n2)SCC(=O)c3ccc(cc3)Cl)SCC(=O)c4ccc(cc4)Cl PD00214 CC(=O)Nc1ccc(c(c1)C(F)(F)F)C#N RDR03709 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C3=NCCO3 RDR03714 Cn1c(=O)c2ccccc2nc1SC PD00218 COc1cc(cc(c1OC)OC)C(=O)OCC(=O)c2ccccc2 RDR01454 c1ccc(cc1)C(=O)/C=C(/C(=O)Nc2ccccc2)\Nc3ccccc3 RJC01833 c1ccc(c(c1)C(=O)OCC(=O)c2ccc(cc2)Cl)NCc3ccco3 RDR01428 CCNC(=S)Nc1ccc(cc1)NC(=O)c2ccccc2O RDR01429 c1ccnc(c1)/C(=C/c2cccs2)/C#N PD00144 COc1ccc(cc1)Cc2c(=S)[nH]nc(n2)c3ccccc3 NRB04137 Cc1c(=O)n2c(nn1)sc(n2)SC NRB04139 CCSc1[nH]c(=O)c(c(n1)C)C NRB04181 CC(=O)OCc1ccccc1Sc2ccc(cc2C(=O)NC)[N+](=O)[O-] RJC01858 c1ccc(cc1)NC(=S)SCc2c(cccc2Cl)Cl RF02457 c1cc(ccc1Nc2c(c(ns2)O)C#N)Cl RF02366 CC(C)c1ccc(cc1)Nc2c(c(ns2)O)C#N RF02384 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3nc(=O)cc(s3)C(=O)OC RF02302 Cc1ccc(cc1)N2C(=O)C=C(C2=O)Sc3ccc(cc3)Cl PD00230 c1cc(ncc1Cl)NC(=O)CSCC(=O)O PD00231 Cc1ccc2c(c1)cc3c(n2)c4c(n(c(=O)n(c4=O)C)C)n(c3=O)c5ccccc5 RJC01846 COc1cccc2c1OCC(=C2)C#N RDR03729 CNC(=O)c1ccccc1Sc2ccc(cc2C(=O)NC)OC RJC01850 Cn1cccc1/C(=C\c2ccc(cc2)C#N)/C#N PD00119 Cn1cccc1/C(=C/c2cc(c(c(c2)OC)OC)OC)/C#N PD00120 CCOC(=O)c1ccccc1Sc2ccc(cc2C(=O)OCC)[N+](=O)[O-] RJC01842 CCOC(=O)c1cnc(nc1N)S/C=C/C(=O)c2ccc(cc2)C NRB04150 CC(=O)c1cc(c(c(c1O)n2nc3ccccc3n2)O)n4nc5ccccc5n4 NRB02696 c1ccc(c(c1)C(F)(F)F)Nc2c(c(ns2)O)C#N RF02433 COC(=O)c1c(noc1NC(=O)NN2CCOCC2)c3c(cccc3Cl)Cl RF02255 COC(=O)c1c(noc1NC(=O)NCc2cccs2)c3c(cccc3Cl)Cl RF02259 CN(C)C1C(C(SC(=C1c2ccccc2)c3ccccc3)c4ccccc4)[N+](=O)[O-] NRB02732 COC(=O)c1c(noc1NC(=O)NN2CCCCC2)c3c(cccc3Cl)Cl RF02254 CC1(OC(=O)C(=CNc2ccccc2)C(=O)O1)C NRB02805 c1ccc2c(c1)c(=O)[nH]/c(=N\c3ccc(cc3)OC(F)(F)F)/o2 PD00139 CN(C)C(=O)Nc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC RF02260 CCCCNC(=O)Nc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC RF02261 c1ccc2c(c1)c(c[nH]2)/C(=C/c3ccc(cc3Cl)Cl)/C#N PD00115 COCc1cc(n(n1)c2ccccc2)O RF02406 CCc1c(c([nH]c1C)C(=O)OCc2ccccc2)C NRB04225 c1ccc(c(c1)C(=O)OCC(=O)c2ccc(cc2)Cl)NC(=O)c3ccc(cc3)Cl RDR01449 COc1cccc(c1OC)/C=N/NC(=S)NCc2ccco2 RDR01453 COc1ccc(cc1)N2C(=O)CC(C2=O)c3ccccc3 PD00136 CC(C)NC(=O)c1ccccc1Sc2ccc(cc2C(=O)NC(C)C)[N+](=O)[O-] RJC01841 CCOC(=O)CSc1[nH]nc(c(=O)n1)Cc2ccc(cc2)Cl NRB04132 Cc1c(=O)n(c(=S)[nH]n1)/N=C/c2ccc(cc2)Cl NRB04134 CC(CCCC(=O)C)C1CCC2C1(CCC3C2CC=C4C3(CCC(C4)O)C)C NRB04201 c1cc(ccc1c2csc(n2)N)Cl RJC00636 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2F)Cl)Cl NRB04234 Cc1nc(nc(n1)N(C)C)N RF02693 CSc1nc(nc(n1)N)c2cc(cc(c2)Cl)Cl RF02700 COc1ccc(cc1)NC(=O)C2=Cc3cccc(c3OC2)OC RDR03738 Cc1ccc(cc1)Sc2cc(nc(n2)c3ccccn3)C RDR03750 c1cc(ccc1C2=NCCO2)NC(=O)c3ccc(cc3)C(F)(F)F RDR03784 c1cc(ccc1C(c2cc3c(cc2O)OCO3)N4CCOCC4)C(F)(F)F RDR03785 COc1ccc(cc1OC)/N=N/c2ccc(c(c2)OC)OC RJC01837 CNC(=O)c1ccccc1Sc2ccc(cc2C(=O)NC)[N+](=O)[O-] RJC01840 Cc1ccc(cc1)S(=O)(=O)Oc2c3ccccc3n(c(=O)c2c4ccccc4)C NRB02802 Cc1ccc(cc1)S(=O)(=O)Oc2cc(=O)n(c3c2cccc3)C NRB02803 Cc1ccc(cc1)S(=O)(=O)Nc2cccc3c2c(ccc3)Br RJC01848 Cc1cccc(c1C(=O)/C=C(/C(=O)O)\O)C RJC01822 CC(=O)OCc1ccccc1Sc2ccc(cc2C(=O)NC)Cl RJC01854 c1ccc(c(c1)/C=N/c2ccc(cc2)NC(=O)c3ccccc3O)O RDR01417 c1ccc(cc1)C(=O)/C=C/2\C(=O)OCCN2 RJC01832 CCOC(=O)Cc1c([nH]c(c1CC(=O)OCC)C(=O)OCC)C NRB02792 c1ccnc(c1)/C(=N/Nc2ccc(cc2)OC(F)(F)F)/C#N PD00172 c1ccc(cc1)C(=O)/C=C/Sc2nc3ccccc3o2 NRB04159 c1ccc(cc1)NS(=O)(=O)c2ccc-3c(c2)Cc4c3ccc(c4)S(=O)(=O)Nc5ccccc5 RJC01778 c1cc(c(c(c1)Cl)Cl)n2ccnc2SCc3ccc(cc3)Cl RDR01360 c1cc(oc1)CNC(=S)N/N=C/c2ccc(o2)c3ccc(cc3)[N+](=O)[O-] RDR01362 COC(=O)/C(=C/C(=O)c1ccc(cc1)Cl)/O RJC01825 Cc1ccc(c(c1)C)C(=O)/C=C(/C(=O)Nc2ccccn2)\O RJC01827 Cc1ccc(c(c1)C(=O)NC)Sc2ccccc2COC(=O)C RJC01862 CC(=O)OCc1ccccc1Sc2ccc(cc2C(=O)O)OC RJC01864 c1cc(ccc1S(=O)(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl RF02418 Cc1cc(ccc1Cl)c2csc(n2)N RJC00671 c1cc(ccc1C(=O)Cc2c(=O)[nH]cnn2)Cl NRB04146 CSc1nc2c(cc(s2)c3ccccc3)nn1 NRB04148 COC(=O)c1c(noc1C(=O)N/N=C/c2ccccn2)c3c(cccc3Cl)Cl RF02174 CNc1nc(ns1)C23CC4CC(C2)CC(C4)C3 RF02202 CN1CCN(CC1)/C=C/C=C/c2nnn(n2)c3ccc(cc3)Cl NRB04084 CCN(CC)/C=C/C=C/c1nnn(n1)c2ccc(cc2)Cl NRB04085 c1cc(ccc1n2nc(nn2)/C=C/C=C/C#N)Cl NRB04086 c1ccnc(c1)/C(=C/c2ccc(cc2)O)/C#N PD00157 Cc1c(c(c(nc1C)S/C=C/C(=O)c2ccccc2)C#N)C NRB04154 c1ccc(cc1)C(=O)/C=C/Sc2[nH]c3cc(c(cc3n2)Cl)F NRB04157 c1cc2c(cc1F)sc(n2)N RJC00659 Cc1ccc(cc1)/C(=C/c2c(cccc2Cl)Cl)/C#N RDR01463 c1ccc(c(c1)C(=O)Nc2ccc(cc2)/N=C/c3cccs3)O RDR01421 CN(C)c1ccc(cc1)/C=N/c2ccc(cc2)NC(=O)c3ccccc3O RDR01425 c1ccc(cc1)C(=O)COC(=O)c2ccccc2NCc3ccco3 RDR01427 CCCCCCC1C2C(C(=O)N(C2=O)c3ccccc3)ON1c4ccc(c(c4)Cl)Cl PD00035 c1ccc(cc1)Cc2c(=O)n(c3nc4ccccc4c(=O)n3n2)N NRB04109 c1ccc2c(c1)ccc3c2sc(c3)C(=O)Oc4ccc(cc4Cl)Cl PD00027 CSc1nc2ccccc2c(=O)n1c3ccc(cc3)F RDR01343 CC12CCC3c4ccc(cc4CCC3C1CCC2O)Oc5ccc(cc5)[N+](=O)[O-] NRB04210 c1ccc(cc1)C2CC(=O)N(C2=O)c3ccc(cc3)F PD00180 c1ccc(cc1)C2C(=Cc3c4ccccc4ccc3O2)[N+](=O)[O-] PD00143 c1ccc(c(c1)C(=O)Nc2ccc(cc2)/N=C/c3cccnc3)O RDR01419 c1ccc(c(c1)C(=O)OCC(=O)c2ccc(cc2)Br)Sc3ccc(cc3C(=O)OCC(=O)c4ccc(cc4)Br)[N+](=O)[O-] RJC01843 Cc1cccc(c1n2c(=O)c3ccccc3nc2SCc4ccccc4)C RDR01345 CC(=O)OC[C@@H]1[C@@H]2[C@H]([C@@H](O1)n3cnc4c3ncnc4N)OC(O2)(C)C RJC00602 c1cc(c(c(c1)F)C(=O)Nc2ccc(c(c2)C(F)(F)F)Br)F RDR03704 c1ccc(c(c1)C(=O)Nc2ccccn2)O RDR01388 c1ccc(c(c1)C(=O)Nc2ccc(cc2)[N+](=O)[O-])O RDR01408 c1ccc(cc1)C(=O)COC(=O)c2ccccc2Nc3ccc(cc3)F RDR01414 Cc1cc(ccc1[N+](=O)[O-])C(=O)OCC(=O)c2ccc(cc2)Cl RDR01479 c1cc(ccc1N2C(=O)CCC2=O)S(=O)(=O)Oc3ccc(cc3)F RDR03782 c1cc(cc(c1)OS(=O)(=O)c2ccc(cc2)N3C(=O)CCC3=O)C(F)(F)F RDR03783 c1ccc(cc1)C(=O)COC(=O)c2ccccc2Cl RDR01455 Cc1ccc(cc1)C(=O)OCC(=O)c2ccccc2 RDR01456 c1ccc(cc1)Nc2c(c(ns2)O)C#N RF02350 c1ccc(cc1)CCN2CCC(CC2)O NRB04193 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)CO PD00122 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)/C=N/NC(=S)Nc3cccc(c3)F RDR01386 c1ccc(cc1)SC(C(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl)(F)F RDR03804 c1ccc(c(c1)C(=O)N)Sc2ccc(cc2C(=O)N)[N+](=O)[O-] RJC01839 CC(C)(C#Cc1ccccn1)O RF02309 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)COC(=O)c4ccc(cc4)C(F)(F)F PD00125 c1ccnc(c1)/C(=C/c2ccc(cc2)C#N)/C#N PD00106 Cc1c(c(c(c(c1[N+](=O)[O-])C(C)(C)C)[N+](=O)[O-])C)C(=O)CSc2ccccn2 RDR01435 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=O)c3ccccc3O)[N+](=O)[O-] RDR01439 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2csnc2c3c(cccc3Cl)Cl)Cl RF02206 c1cc(c(c(c1)Cl)c2c(csn2)NC(=O)NN3CCOCC3)Cl RF02212 CC1(CC(CC(N1)(C)C)Nc2ccc(cc2)Nc3ccccc3)C RJC01813 C(C(=O)O)Sc1nn2c(=O)c(nnc2s1)N NRB04115 c1ccc2c(c1)c(=O)[nH]c(=S)[nH]2 PD00036 CCCCn1c2ccccc2c(c(c1=O)C(=O)C)O NRB02822 CCO/C=N/c1c2cnc(nc2sc1C(=O)OCC)SC NRB04184 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=O)c3ccc(cc3)Cl)O RDR01440 c1ccc2c(c1)cccc2/C=C(\C#N)/c3ccccn3 PD00215 CCOc1ccc(cc1OCC)C(=O)C RJC01847 c1cc(cnc1)CN2C(=O)CC(C2=O)Sc3ccc(cc3)Cl PD00047 c1ccnc(c1)NC(=O)CSCC(=O)O PD00052 c1ccnc(c1)/C(=C/c2ccc3c(c2)OCO3)/C#N PD00105 c1cc(ccc1c2ccc(o2)/C=N/NC(=S)Nc3ccc(c(c3)Cl)Cl)[N+](=O)[O-] RDR01364 c1ccc2c(c1)c(c[nH]2)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N PD00185 Cc1ccc(cc1F)N/C(=C(/C#N)\c2ccccn2)/SC PD00191 c1ccnc(c1)/C=C(\C#N)/c2ccccn2 PD00145 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=S)Nc3ccc(cc3)Cl)O RDR01430 CCOC(=O)Cc1cc([nH]c1C(=O)OCC)C NRB04218 CC(C)c1nc(nc(n1)SC)N RF02690 COc1ccc(cc1)C(=O)OCC(=O)c2ccccc2 RDR01485 CCOC(=O)C(c1ccccc1)C(=O)Cc2ccccc2 NRB02815 Cc1c(c(nc(n1)c2ccncc2)NCCNc3ccc(cn3)C(F)(F)F)Cl RDR03879 c1ccc(cc1)Oc2ccc(cc2)OC(=O)N3CCC(CC3)OC(=O)n4ccnc4 RJC01915 Cc1ccc(cc1)S(=O)(=O)OC[C@@H]2COc3cc4c(cc3O2)OCO4 RJC01941 CCCCCCNC(=O)OCCCCCCNC(=O)OC1CCN(CC1)Cc2ccccc2 RJC01942 CSc1nc(nc(n1)N)c2cccs2 RF02724 c1cc(c(nc1)NCCNCC(COc2ccc(cc2)F)O)C(F)(F)F RDR03853 CC1(c2ccccc2-n3c1cc(c(c3=O)c4ccccc4)O)C NRB02860 Cn1c2c(c3c(c1=O)[n+](on3)[O-])c(=O)n(c(=O)n2c4ccccc4)c5ccccc5 RJC01886 c1ccc2c(c1)c(=O)n(c(n2)SCc3ccc(cc3)[N+](=O)[O-])Cc4ccc(cc4)[N+](=O)[O-] PD00228 c1ccc2cc(ccc2c1)c3cn4ccccc4n3.Br RDR01635 c1ccc(cc1)Oc2ccc(cc2)OC(=O)N3CCC(CC3)O RJC01900 CCCCCCNC(=O)OCCCCCCNC(=O)OC1CCNCC1.CC(=O)O RJC01905 CC(=O)Oc1ccc(cc1OC)/C=C/2\C(=O)OC(=N2)c3ccccc3 PD00281 c1ccc(cc1)/C=C/2\C(=O)c3ccccc3S2=O RJC00741 CC(C)(C)c1ccc(cc1)N2C(=O)CSC2=N RF02588 c1cc(ncc1Cl)N2C(=O)CSCC2=O PD00232 CC(C)(C)c1nc(nc(n1)OC)N RF02684 Cc1nc(nc(n1)SC)N RF02687 c1ccc(cc1)C2CC(c3ccccc3O2)O RJC00736 Cc1cc(cc(c1NC(=O)/C=C/C(=O)O)C)C(C)(C)C RDR03911 c1ccc2cc(ccc2c1)OC(=O)Oc3ccc4ccccc4c3 RJC00748 Cc1c(c(nc(n1)c2ccncc2)NCCNc3c(cccn3)C(F)(F)F)Cl RDR03870 c1ccc(c(c1)C(=O)Nc2ccc(cc2)/N=C/c3cc(cc(c3O)Cl)Cl)O RDR01519 COc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2)Cl NRB04235 CC(=O)N(C(=O)C)N(C)c1nc(ns1)c2ccccc2 RDR03956 c1ccc(c(c1)C(=O)Nc2cccc(c2)NC(=O)/C=C/C(=O)O)O RDR01526 Cc1cc(=O)oc2c1cc(c(c2)OS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl RDR01556 c1ccc(cc1)n2c3c(cn2)c(ncn3)N RJC00689 CCNC(=S)Nc1cccc(c1)NC(=O)c2ccccc2O RDR01511 c1cc(c(c(c1)F)NC(=O)NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)F RDR04020 C=CCCN1c2ccccc2C(=NCC1=O)c3ccccc3 RJC01932 c1cc(ccc1N2C(=O)c3c(nccn3)C2=O)F PD00255 c1cc(nc(c1)NCCNc2nc(ns2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F RDR03944 Cc1cc(c(cc1Cl)C)S/C(=C/C(=O)OC)/C(=O)OC PD00304 COc1cc(cc(c1OC)OC)N2C(=O)CC3(CCCC3)CC2=O PD00309 c1cc(ccc1NC(=O)CC2(CCCC2)CC(=O)O)OC(F)(F)F PD00310 CN(C)C(=O)O/N=C(/c1ccc(cc1)C2SCCS2)\N RF02568 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2csc3c2cccc3 PD00147 Cn1c2c(c3c(c1=O)cc4ccc(cc4n3)Cl)c(=O)n(c(=O)n2C)C RJC01887 c1cc(ccc1NC(=O)CC2(CCCC2)CC(=O)O)F PD00314 c1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3)F NRB04257 Cc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(c(c3)Cl)Cl NRB04259 CCCCn1c(cc(nc1=S)N)O RDR01547 c1ccc(cc1)NC(=O)O/N=C(/c2ccc(cc2)C3SCCS3)\N RF02570 c1cc(ccc1C2SCCS2)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N RF02571 CC(C(=O)N1CCN(CC1)c2ccccc2OC)Nc3ccccn3 RJC01899 CC(C)N(C1C(=O)N(c2ccc(cc2C(=N1)c3ccccc3)Cl)C)C(C)C RJC01902 C/C(=C\c1ccc(cc1)N(C)C)/[N+](=O)[O-] PD00318 Cc1ccc(cc1)OCCC(=O)O RJC00750 c1cc(ccc1OCCC(=O)O)Cl RJC00752 CCc1c(c(c([nH]1)C(=O)OCC)CCC(=O)OCC)C(=O)OCc2ccccc2 NRB04227 c1ccc2c(c1)c(cs2)C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N PD00152 CCC1(CCCCN(C1=O)C)c2cccc(c2)OC RJC01911 CCOC(=O)/C(=C\1/N(C(CS1)(C)O)c2c(cccc2F)F)/C#N RF02496 c1cc(ccc1C2SCCS2)/C(=N/O)/N RF02543 CC1CCCC(N1C(=S)NCc2ccco2)C RDR01545 CN(C)/C=C/1\Cc2ccccc2C1=O PD00297 CN(C)/C=C/1\CCCc2ccccc2C1=O PD00299 c1cc(ccc1C(=O)/C=C/OC(=O)c2ccc(cc2)Cl)Cl NRB04240 c1cc(cnc1)NC(=O)CCC(=O)O RDR01549 c1cc(cnc1)NC(=O)/C=C/C(=O)O RDR01550 Cc1cc(cc(c1N2C(=O)CC(C2=O)Sc3cc(c(cc3C)Cl)C)C)C(C)(C)C RDR03914 Cc1cc(cc(c1NN=C(C(=O)C)C(=O)C)C)C(C)(C)C RDR03915 c1ccc(cc1)C(=O)c2ccccc2C(=O)OCC(=O)c3ccc(cc3)Cl RDR01503 c1ccc(c(c1)C(=O)Nc2cccc(c2)N)O RDR01504 CCCc1c(nc2n(c1=O)c(cs2)c3ccccc3)C RDR01528 COc1cccc(c1C(=O)OCC(=O)c2ccccc2)OC RDR01533 CCCCCCCCC/C(=N\O)/c1ccccn1 RJC00758 Cc1cccc(c1)C(=O)Oc2ccc(cc2)/C=C(\C#N)/c3ccccn3 PD00158 COc1ccc(cc1)C(=O)/C=C/OC(=O)c2ccc(cc2)Cl NRB04242 c1cc(ccc1C2=CC(=O)C(C(=O)O2)C(=O)c3ccc(cc3)Br)Br RJC00768 c1ccc(cc1)NC(=S)NC(=N)N2CCOCC2 RJC00770 c1cc(ccc1C(=O)/C=C/OC(=O)c2ccc(c(c2)Cl)Cl)Cl NRB04241 COc1ccc(cc1)C(=O)NNC(=O)/C=C/C(=O)O RJC00782 c1ccc(cc1)c2nc(sn2)Oc3cc(cc(c3)Cl)Cl RDR03909 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nc(sn2)Oc3cc(cc(c3)Cl)Cl RDR03910 Cc1ccc(cc1)n2c(nnn2)c3cnc(nc3c4ccc(cc4)Cl)c5ccccc5 NRB04246 c1ccc(cc1)n2c(nnn2)c3cnc(nc3c4cccc(c4)Cl)N NRB04248 CS(=O)(=O)Oc1c(=O)c2ccccc2oc1c3ccccc3 RJC00731 CC(=O)c1ccc(cc1)N/N=C\2/c3ccccc3C=C(C2=O)C(=O)Nc4ccccc4 NRB02907 c1cc(ccc1NC=C2C(=O)CCCC2=O)Cl NRB02830 c1ccc(cc1)NC=C2C(=O)CCCC2=O NRB02832 CCCCc1c(c2cccc3c2n(c1=O)c4c3cccc4)O NRB02883 CCc1c(c([nH]c1C)C(=O)OC(C)(C)C)C NRB04223 c1ccnc(c1)/C(=C/c2ccc(cc2)OC(=O)c3cccs3)/C#N PD00161 Cc1c(c2nnnn2c(n1)c3ccccn3)Cl RDR03800 CCCc1c(nc2n(c1=O)c(cs2)c3ccc(cc3)Cl)C RDR01529 c1cc(c(c(c1)Cl)CSC(=S)Nc2ccc(cc2)Cl)Cl RF02458 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)SCc3c(cccc3Cl)Cl RF02467 Cn1cnnc1S/C=C/C(=O)c2ccc(cc2)Cl NRB04163 Cc1ccc(cc1)S(=O)(=O)N(c2ccc3c(c2Cl)C(=O)c4ccccc4C3=O)S(=O)(=O)c5ccc(cc5)C NRB04165 c1cc(ccc1C(=O)c2ccc(cc2)Br)[N+](=O)[O-] NRB04195 CC(=O)CCc1c[nH]c2c1cccc2 NRB02761 c1ccc2c(c1)ccc(c2OC(=O)c3ccc(cc3)Cl)C(=O)OCC(=O)c4ccc(cc4)Cl RDR01492 c1ccc2c(c1)c(cs2)C(=O)/C(=C/c3ccc(cc3Cl)Cl)/C#N PD00153 CC1=NNC(=O)C1Oc2ccc(cc2Cl)Cl RDR03765 Cc1ccc(cc1Cl)N/N=C(\C#N)/c2ccccn2 PD00178 c1cc(ccc1CS(=O)(=O)C2CCCCC2O)Cl RDR03788 CCN(CC)c1nc2ccccc2c(=O)s1 RDR03793 c1ccc2c(c1)CCc3c(ccs3)C2O NRB04197 c1ccc2c(c1)C(=O)C(C(=O)N2)(N3CCOCC3)N4CCOCC4 NRB02835 c1ccc2c(c1)c(cs2)C(=O)/C(=C/c3cccc(c3)F)/C#N PD00155 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2Cl)Cl)F NRB04237 COc1ccc(cc1)Oc2ccc(cc2)S(=O)(=O)c3ccc(cc3)c4ccc(cc4)S(=O)(=O)c5ccc(cc5)Oc6ccc(cc6)OC RJC01871 c1cc(c(cc1N2C(=O)CSC2=N)Cl)F RF02586 CN(C)C(=O)Oc1c(cn(c(=O)c1c2ccccc2)Cc3ccccc3)c4ccccc4 NRB02801 c1ccc(c(c1)C(=O)OCC(=O)c2ccc(cc2)Cl)Cl RDR01474 c1cc(c(c(c1)Cl)C(=O)OCC(=O)c2ccc(cc2)Cl)Cl RDR01475 Cn1c2c(c(cc(=O)n2c3ccccc3)Nc4ccc(cc4)Cl)c(=O)n(c1=O)C RJC01817 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)F)c4ccc(cc4)F PD00289 CC12CCC3C(C1CC[C@H]2O)CCC4=CC(=O)CCC34C NRB04205 c1ccnc(c1)/C(=C/c2ccc(cc2)OC(=O)c3cc(cc(c3)Cl)Cl)/C#N PD00159 c1ccnc(c1)/C(=C/c2ccc(cc2)OC(=O)c3ccc(cc3)C(F)(F)F)/C#N PD00160 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2Cl)Cl)Cl NRB04238 c1cc(cc(c1)F)C(=O)O/C=C/C(=O)c2ccc(cc2)Cl NRB04239 CCCCCCCCCCCCSC1CC(=O)N(C1=O)c2ccc(cc2)Cl PD00247 CCCCCCCCCCCCSC1CC(=O)N(C1=O)c2ccc(cc2)OC PD00251 c1cc(ccc1C2N(C(=O)CS2)CCN3C(SCC3=O)c4ccc(cc4)Cl)Cl PD00261 c1ccc(c(c1)CO)Sc2ccc(cc2C(=O)O)Cl RJC01852 CC(=O)OCc1ccccc1Sc2ccc(cc2C(=O)O)Cl RJC01853 c1ccc(c(c1)CO)Sc2ccc(cc2C(=O)O)[N+](=O)[O-] RJC01856 c1ccc(cc1)/N=C/c2c(c3cccc4c3n(c2=O)CCC4)O NRB02811 c1ccc2c(c1)c(=O)n3c(n2)S(=O)(=O)CC3 PD00225 c1cc(ccc1C(=O)COC(=O)c2ccc3cc(ccc3c2)OC(=O)c4ccc(cc4)Cl)Cl RDR01493 c1cc(ccc1/C=N/NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)C(F)(F)F RDR03919 COc1ccc(cc1)/C=N/c2cccc(c2)NC(=O)c3ccccc3O RDR01507 C1CNCC1N.Cl.Cl RJC00676 Cc1ccc(cc1)/C=C(\C#N)/c2cccs2 PD00269 c1cc(sc1)/C(=C/c2ccc3c(c2)OCO3)/C#N PD00270 c1ccc(cc1)C2CC(=O)N(C2=O)Cc3cccs3 PD00184 Cc1ccc(cc1)c2cc(n(c(=O)c2C#N)C(=O)C)c3ccc(cc3)C PD00088 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)COC(=O)Nc4cccc(c4)Cl PD00130 CC(C)(C)c1ccc(cc1)N2C(=O)CC(C2=O)c3ccccc3 PD00133 CS/C(=C(/C#N)\c1ccccn1)/Nc2cccnc2 PD00177 Cn1c2c(c(c(c1=O)[N+](=O)[O-])N)c(=O)n(c(=O)n2c3ccccc3)c4ccccc4 RJC01869 Cc1c(c(nc(n1)c2cccnc2)N(C)C)Cl RDR03819 C[C@@]1(CCC2C1(CCC3C2CC[C@@H]4C3(C/C(=C\c5ccccc5)/C(=O)C4)C)C)O NRB04209 CC1(CCc2ccc(cc2O1)OCC(=O)Nc3ccccc3Br)C RJC00698 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)COC(=O)Nc4ccc(cc4)OC(F)(F)F PD00132 COc1cc(cc(c1OC)OC)C(=O)OCC(=O)c2ccc(cc2)Cl RDR01476 Cc1cc(ccc1[N+](=O)[O-])C(=O)OCC(=O)c2ccccc2 RDR01478 c1ccc(cc1)C(=O)COC(=O)c2ccccc2NC(=O)c3ccc(cc3)Cl RDR01448 CC(=O)Oc1cc(c(cc1OC)OC(=O)C)c2cc(c(cc2OC(=O)C)OC)OC(=O)C RJC01889 CN(S(=O)(=O)c1ccc(cc1)F)S(=O)(=O)c2ccc(cc2)Cl RJC01872 c1ccc(cc1)C(=O)COC(=O)c2ccc(cc2NC(=O)c3ccc(cc3)Cl)Cl RDR01450 c12c([nH]c(n1)S)nc(nc2O)N RJC00691 CC(=O)OC[C@@H]([C@@H]([C@H]([C@@H]1N2[C@@H](CS1)C(=O)OC2[C@H]([C@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00872 CCOc1ccc(c(c1N2CCOCC2)[N+](=O)[O-])OCC NRB02924 C1CCC(CC1)NC(=S)N2CCCCC2 RDR01662 c1cc(ccc1NC(=N)NC(=N)NN)F.Cl RDR01650 CCN(CCC#N)c1ccc(cc1)NN=C2c3ccccc3C=CC2=O NRB02983 c1ccc(cc1)c2c(c3cccc(c3[nH]c2=O)F)O NRB02818 c1ccc2c(c1)c(c(c(=O)o2)/C=N/c3ccc(cc3)Cl)O NRB02821 c1cc(c(cc1Cl)Cl)N2C(=O)CSC2=N RF02583 c1ccc2c(c1)C=CC(=O)C2=NNc3ccccc3Cl NRB02966 c1ccc2c(c1)C=CC(=O)C2=NNc3ccc(cc3)I NRB02970 CC\1=NN(C(=O)/C1=N/Nc2ccc(cc2)N3CCCCC3)c4ccccc4 NRB02917 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccccc4 RJC00733 CCN(CC)c1ccc(cc1)/C=C/c2ccc(cc2C#N)[N+](=O)[O-] NRB02930 c1ccc2c(c1)nc(n2CCC(=O)O)CCC(=O)O NRB04296 CCc1ccc(cc1)C(=O)/C=C/Sc2ccc(cc2)Cl NRB04298 c1cc(cc(c1)Br)C(=O)/C=C/Sc2ccc(cc2)Cl NRB04299 c1c(cc(cc1Cl)Cl)N2C(=O)CC3(CCCC3)CC2=O PD00313 c1ccc(cc1)CN2C/C(=C\c3ccc(cc3)F)/C(=O)/C(=C/c4ccc(cc4)F)/C2 PD00328 c1ccc(cc1)c2cc(nc(n2)SCc3ccccc3Cl)O RDR01582 c1ccc(cc1)OCCC(=O)O RJC00749 CCCCCCNC(=O)OCCCCCCNC(=O)OC1CCN(CC1)C(=O)Oc2ccc(cc2)Oc3ccccc3 RJC01917 c1cscc1/C=C/2\C(=O)C3CCN2CC3 PD00298 c1ccc(cc1)C2CC(=O)c3ccccc3S2(=O)=O RJC00740 C=CCOc1ccc(cc1)/C=C(\C#N)/c2ccccn2 PD00306 c1ccc(cc1)NNC(=S)N PD00320 Cc1cc(ccc1NNC(=S)N)Cl PD00321 COc1ccc(cc1OC)CC(=O)NNC(=O)CSCC(=O)O PD00361 c1ccc(cc1)CCC=C(c2ccc(cc2)Cl)c3ccc(cc3)Cl RJC00773 c1cc(ccc1C(=O)NN/C=C/C(=O)O)[N+](=O)[O-] RJC00774 Cc1cc(=O)oc2c1cc(c(c2)OC(=O)N(C)C)Cl RDR01558 COc1cc(cc(c1OC)OC)NC(=S)Nc2ccc3c(c2)OCCO3 PD00366 C/C(=N\N=C(\c1ccccc1)/C)/c2ccccc2 RJC00784 COc1ccc(cc1)N/N=C\2/c3ccccc3C=C(C2=O)O NRB02956 Cc1cc(ccc1NC(=S)NC(C)(CO)CO)Cl RDR01567 c1ccc2c(c1)CC(OC2=O)[N+](=O)[O-] PD00301 CCC/C(=N\O)/c1ccccn1 RJC00757 c1ccnc(c1)/C(=N/O)/C2CCCCC2 RJC00762 COc1ccc(cc1)/C=C\2/c3ccc(cc3C(=O)O2)[N+](=O)[O-] NRB02933 CC(CO)(CO)NC(=S)Nc1ccc(cc1)F RDR01565 c1ccc(cc1)C23[C@H](C4C5C2C6[C@H](C3C4C6C5)O)O RJC00822 CN(C)c1ccc(c2c1cccc2)/C=C(/C#N)\c3ccc(cc3)[N+](=O)[O-] NRB02939 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nc(sn2)N3CCOCC3 RDR03893 COC1(C2([C@@H]3[C@@H](C=C[C@@H]([C@@H]3C1(C(=C2Cl)Cl)Cl)O)O)Cl)OC RJC00826 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])N3CCOCC3 NRB02946 c1ccc(cc1)Cn2c3cc(ccc3oc2=S)Cl RDR03898 c1ccc2c(c1)C=CC(=O)C2=NNc3ccc(cc3)F NRB02964 CC(=O)Oc1ccc(cc1)c2coc3cc(cc(c3c2=O)OC(=O)C)OC(=O)C RJC00833 C=C(C(CCCCOc1ccc(cc1)Cl)O)C(=O)[O-].[Na+] RJC01919 c1ccc(c(c1)C(C(=O)Nc2ccc(cc2)Cl)O)Cl RJC01928 c1ccc(c(c1)S(=O)(=O)NC(=O)c2ccc(cc2)C(F)(F)F)Cl RDR04016 C1CCCCCC(CCCCC1)CCC(=O)O RJC01939 c1ccc2c(c1)nc3n2c(=O)c4cccc5c4c3ccc5 PHG00154 CCNc1nc(nc(n1)SC)NC(C)C RJC00747 CSc1nc(nc(n1)N)C23CC4CC(C2)CC(C4)C3 RF02813 Cc1c(c(no1)c2ccccc2)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N RF02855 Cc1ccc(cc1)/C(=C/c2ccc(cc2)NC(=O)C)/C#N PHG00062 COc1ccc(cc1)/C=C(\C#N)/c2ccc(cc2)OC PHG00067 Cc1ccc(cc1)/C(=C/c2ccc(cc2)OC)/C#N PHG00068 c1ccc2c(c1)c(=O)c(cn2C3CCCCC3)C(=O)N RJC01922 COc1ccc(cc1)C=C2CCC(=O)CC2 RJC01927 CC(=O)C(=NNc1ccc(cc1)C#N)C(=O)C NRB02958 CC(=O)C(=NNc1ccc(cc1)Cl)C(=O)C NRB02959 CSc1nc(nc(n1)N)c2ccncc2 RF02732 COc1ccc(cc1OC)CCN2C(=O)c3cccc4c3c(ccc4Br)C2=O PHG00218 CCOC(=O)OCCN1C(=O)c2cccc3c2c(ccc3Br)C1=O PHG00220 Cc1cc(=O)oc2c1ccc(c2O)O RJC00743 c1cc2c(cc1Cl)C(=O)C(C(=O)N2)(Cl)Cl NRB02884 CSc1nc(nc(n1)N2CCCCC2)N RF02737 c1ccc(c(c1)C(=O)O)NC(=O)Nc2ccc(cc2)C(F)(F)F PD00364 c1ccc2c(c1)c(=O)oc(n2)Nc3ccc(cc3)C(F)(F)F PD00365 CC(=O)Nc1ccc(cc1)/C=C(\C#N)/c2ccc(cc2)OC PHG00061 COc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(c(c3)Cl)Cl NRB04329 COc1ccccc1C(=O)OCC(=O)c2ccc(cc2)Cl RDR01628 CC(C)(C)c1nc2cc(c(cc2c(=O)o1)OC)OC RDR03907 CC\1=NN(C(=O)/C1=N/Nc2ccc(cc2)C#N)c3ccccc3 NRB02904 CCCCN1C(=O)C(=C(/C(=N\Nc2ccc(cc2)C#N)/C1=O)C)C#N NRB02906 CSc1nc(nc(n1)N2CCSCC2)N RF02734 CCCCNC(=O)NS(=O)(=O)c1ccccc1C(F)(F)F RF02735 c1ccc(cc1)CN2C/C(=C\c3sccc3)/C(=O)/C(=C/c4sccc4)/C2 PD00329 Cc1ccc(cc1)N2C(=O)CCC2=O PD00333 Cc1ccc(cc1)NC(=O)c2ccccc2[N+](=O)[O-] PD00338 c1ccc(c(c1)C(=O)Nc2ccc(cc2F)F)[N+](=O)[O-] PD00339 CC(C)(C)c1nc(nc(n1)O)N RF02758 CC(=O)SC1CC(=O)N(C1=O)c2ccc(c(c2F)F)F PD00353 CC(C)(C)c1nc(nc(n1)NNS(=O)(=O)c2ccccc2C(F)(F)F)N RF02939 COC(=O)C(=C1C2CC3CC(C2)CC1C3)C(=O)OC RJC00823 CC1(OC(=O)C(=C2C3C4CC5C2C6C3CC4C56)C(=O)O1)C RJC00825 c1ccc(cc1)n2c(nnn2)c3cnn(c3c4cccc(c4)Cl)c5ccc(cc5Cl)Cl NRB04322 c1ccc2c(c1)C(=O)N(C2=O)CN(CCc3ccc(cc3)Cl)CN4C(=O)c5ccccc5C4=O PD00336 Cc1c(c(nc(n1)c2ccccn2)NCCNc3cccc(n3)C(F)(F)F)Cl RDR03871 CC(C)(C)c1nc(nc(=O)n1C)N RF02851 Cc1ccc(cc1)/C(=C/c2ccc3c(c2)OCO3)/C#N PHG00070 C1C2C3CC4C2C5C1C3C(=O)C45 RJC00812 c1ccc(cc1)C23C4C5CC6C4C(O2)C7C6C5C37 RJC00813 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C)NC(=O)C RJC01969 Cc1c(c(no1)c2cccc(c2Cl)Cl)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N RF02859 C1C2C3CC(=O)C2C4C1C3C=C4Br RJC00817 Cc1cc(=O)oc2c1cc(c(c2)OS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)Cl RDR01557 Cc1ccc(cc1)n2c(nnn2)c3cnn(c3c4ccc(cc4)Cl)c5ccc(cc5)Cl NRB04317 Cc1nc(cs1)c2cccnc2 RDR03966 CCCCC1(CCN(CC1)Cc2ccccc2)O RJC01938 CN(C)/N=C(\c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/Sc2ccc(cc2)Br RDR03952 CN(C)/N=C(\c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/Sc2ccc(c(c2)OC)OC RDR03953 Cc1ccc(cc1)C(=O)/C=C(\O)/C(=C/C(=O)c2ccc(cc2)C)/O RJC00789 Cc1c(c(c(=O)n(c1c2ccccc2)c3ccccn3)c4ccccc4)O RJC00803 COC(=O)[C@@H]1[C@@H]([C@@H]([C@H](C(O1)O)O)O)O RJC00828 Cn1c(=O)c(c(c(n1)c2ccccc2)O)/N=N/c3ccccc3 RJC00807 c1ccc2c(c1)c(=O)c(cn2C3CCCCC3)C(=O)O RJC01923 Cc1ccc(cc1)/C(=C/c2ccccc2OC)/C#N RDR01629 Cc1c(c(c(cn1)CO)/C=N/O)O RJC00832 Cc1ccc(c(c1)C)NC(=N)NC(=N)N RDR01690 c1cc(ccc1/C(=C/c2cc(cc(c2O)Cl)Cl)/C#N)[N+](=O)[O-] PHG00018 Cc1ccc(cc1)/C(=C/c2ccco2)/C#N PHG00037 CN1C(=NC(NC1=O)/N=C/N(C)C)C2CC2 RF02844 c1ccc\2c(c1)C=CC(=O)/C2=N\Nc3ccc(cc3)N4CCCCC4 NRB02918 CCN(CC)c1ccc(cc1)N/N=C\2/c3ccccc3C=CC2=O NRB02920 c1cc(c(c(c1)Cl)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])Cl PHG00053 c1cc(cc(c1)[N+](=O)[O-])/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00055 COc1ccc(c(c1N2CCOCC2)[N+](=O)[O-])OC NRB02923 COc1c(cc(cc1Br)[N+](=O)[O-])Br RDR01643 COc1ccc(cc1)/C(=C/c2ccccc2OC)/C#N RDR01630 c1ccc(cc1)NC(=O)C2=Cc3ccccc3/C(=N/Nc4ccc(cc4)Cl)/C2=O NRB02909 CC\1=NN(C(=O)/C1=N/Nc2ccc(cc2)OC)c3ccccc3 NRB02911 CCCCN1C(=O)C(=C(/C(=N\Nc2ccc(cc2)OC)/C1=O)C)C#N NRB02912 c1cc(ccc1S(=O)(=O)N2CCc3c(c4cc(ccc4[nH]3)F)C2)Cl RJC01948 c1cc(ccc1F)S(=O)(=O)N2CCc3c(c4cc(ccc4[nH]3)F)C2 RJC01950 CC(C)(C)C(=O)OCC(=S)N RF02972 c1ccc2c(c1)c(nc(n2)SCC(=O)c3ccc(cc3)Br)SCC(=O)c4ccc(cc4)Br PD00206 c1cc(cc(c1)Br)C(=O)/C=C/Sc2c(cccc2Cl)Cl NRB04301 COc1ccc(cc1)N/N=C\2/c3ccccc3C=CC2=O NRB02913 Cc1ccc(cc1C)NC(=S)NCCCN2CCOCC2 RDR01621 c1cc(ccc1C(=O)/C=C/Sc2ccc(cn2)C(F)(F)F)F NRB04304 CN(C)C(=O)Oc1cc(nc(n1)SC)c2ccccc2 RDR01583 CCCCNC(=O)NS(=O)(=O)c1ccccc1Cl RF02699 CN1C(=O)c2cccc3c2c(cc(c3)[N+](=O)[O-])C1=O NRB04269 CC1(CS/C(=N/c2ccc(cc2)F)/N1)CO RDR01572 CCc1c(c2c(n(c1=O)C)n(c(=O)n(c2=O)C)C)O RJC01881 CN(C)c1nc2ccccc2c(=O)s1 RDR03794 CC(=O)C(CCC(=O)OC)(CCC(=O)OC)C(=O)C NRB02750 c1ccc(cc1)CNc2nc(ns2)c3ccccc3 RDR03958 c1cc2c(cc1[N+](=O)[O-])[nH]c(=O)[nH]2 RJC00810 C=CCNC(=S)NC(=N)N1CCOCC1 RJC00793 c1cc(cnc1)c2csc(n2)c3ccc(cc3)Cl RDR03963 c1ccc(cc1)n2c(nnn2)c3cnn(c3c4cccc(c4)Cl)c5ccc(c(c5)Cl)Cl NRB04321 CC1(CS/C(=N\c2ccc(c(c2)Cl)Cl)/N1)CO RDR01573 CC1(CS/C(=N\c2ccc(cc2)OC)/N1)CO RDR01574 CC(C)c1ccc(cc1)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00050 C/C(=N\OC(=O)c1ccc(cc1)C(C)(C)C)/c2csc3c2cccc3 PD00148 CCOC(=O)C1=C(N(C(=NC1c2ccccc2)SC)C(=O)C)C NRB02855 CC(=O)Nc1nc(cs1)c2cccnc2 RDR03962 c1ccc(cc1)c2nc(cs2)c3cccnc3 RDR03965 Cn\1c(cs/c1=N\C(=S)NCCc2ccccc2)c3ccc(cc3)Cl RDR01632 c1ccc(cc1)c2nc(sn2)N3CCOCC3 RDR03889 Cc1c(c(nc(n1)c2ccccn2)SCc3ccccc3)Cl RDR03984 CCC1(COC2(c3ccccc3NC2=O)OC1)CC PD00375 COc1ccc(cc1OC)CCNC(=O)N PHG00007 Cc1c(c(nc(n1)c2cccnc2)NCc3ccccc3)Cl RDR03950 CSc1nc(nc(n1)N)c2cccnc2 RF02731 Cc1ccc(cc1)S(=O)(=O)N2CCc3c(c4cc(ccc4[nH]3)F)C2 RJC01951 c1ccc2c(c1)C=CC(=O)C2=NNc3ccccc3O NRB02978 c1ccc2c(c1)C=CC(=O)C2=NNc3cccc(c3)O NRB02979 C(CCC(=O)O)CC(C(=O)O)N RJC00670 c1cc(cnc1)/C=C(\C#N)/c2cccs2 PD00271 c1cc(sc1)/C(=C/c2ccc(cc2)C(F)(F)F)/C#N PD00272 COc1ccc(c(c1OC)OC)/C=C(\C#N)/c2cccs2 PD00273 CNS(=O)(=O)Cc1ccc(cc1)[N+](=O)[O-] RJC01929 Cc1ccc(cc1)S(=O)(=O)OCCCCN2C(=O)CC3(CCCC3)CC2=O RJC01930 c1cc(oc1)C(=O)OCC(=O)c2ccc(cc2)Cl RDR01611 c1cc(c(c(c1)O)O)C(=O)OCC(=O)c2ccc(cc2)Cl RDR01609 CSc1nc(=O)[nH]n1c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] RJC01924 COC(=O)c1ccccc1S(=O)(=O)N2CCc3c(c4cc(ccc4[nH]3)F)C2 RJC01947 CC\1=NN(C(=O)/C1=N/Nc2ccc(cc2)N3CCOCC3)c4ccccc4 NRB02915 c1ccc2c(c1)C=CC(=O)C2=NNc3cccc(c3)[N+](=O)[O-] NRB02972 Cc1cccc(c1)NN=C2c3ccccc3C=CC2=O NRB02975 CC1=C(C(C(=C(N1)C)C#N)c2ccccc2[N+](=O)[O-])C#N RJC00797 CCSc1nc(nc(n1)N)C(C)C RF02722 CC(C)(C)C(=O)CSc1c2ccccc2nc(n1)SCC(=O)C(C)(C)C PD00207 COc1cccc(c1C(=O)OCC(=O)c2ccc(cc2)Cl)OC RDR01534 c1ccc(cc1)C(=O)COC(=O)c2cccc(c2)I RDR01537 CSc1nc(nc(n1)N)c2ccccn2 RF02651 CC(=O)SC1CC(=O)N(C1=O)c2ccc(cc2)C(C)(C)C PD00351 c1ccc(cc1)c2ccc(cc2)C(=O)/C=C(\c3ccccc3)/C(=O)c4ccccc4 PD00363 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N RF02856 COc1ccccc1NN=C2c3ccccc3C=CC2=O NRB02976 COc1nc(nc(n1)N)C2CC2 RF02686 CSc1nc(nc(n1)N)C2CC2 RF02696 c1ccc(cc1)c2cc(nc(n2)S)O RDR01576 CSc1nc(cc(n1)O)c2ccccc2 RDR01577 c1ccc(cc1)C(=NNC(=O)/C=C/C(=O)O)c2ccccc2 RJC00783 CN(C)c1cc(c(cc1OC)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])OC NRB02943 CN(C)c1ccc(cc1[N+](=O)[O-])/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] NRB02944 Cc1c(c(no1)c2ccccc2)C(=O)OCC(=O)c3ccc(cc3)Cl RDR01484 CC(C1CC1)Nc2ccccc2.Cl RJC01874 COc1ccc(cc1)C(=O)OCC(=O)c2ccc(cc2)Cl RDR01486 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)I PD00368 Cc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3)Cl NRB04258 c1ccc(cc1)c2cc(nnc2N3CCCC3)c4ccccc4 RDR03998 CN(C)c1nc(nc(n1)SC)N RF02697 CCSc1nc(nc(n1)N)C RF02707 c1cc\2c(cc1[N+](=O)[O-])C(=O)O/C2=C\c3cc4c5c(c3)CCCN5CCC4 NRB02935 c1ccc(cc1)CN(Cc2ccccc2)c3ccc(cc3)/C=C(\C#N)/c4ccc(cc4)[N+](=O)[O-] NRB02947 Cc1ccc(cc1)S(=O)(=O)CC(CN2CCCC2=O)O RDR04031 Cc1cc(c(c(c1)C)NC(=N)NC(=N)NN)C.Cl RDR01647 CN(C)c1nc(ns1)c2ccccc2 RDR03891 c1ccc(cc1)C2=NCC(=O)Nc3c2cccc3 RJC01933 c1ccc2c(c1)C=CC(=O)C2=NNc3cccc(c3)Cl NRB02965 COc1ccc(cc1)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] NRB02941 CC(C)(C)CC(C)(C)NC(=O)c1c(cccc1OC)OC RF00046 CC(=O)Nc1cc2cc(ccc2oc1=O)Br PHG00461 Cc1ccc(cc1)C(=O)CSc2nc(c(s2)C(=O)c3ccc(cc3)C)N NRB04401 CC(C)(C)CC(C)(C)NC(=O)c1ccccc1Cl RF00018 c1cc(c(c(c1)Cl)Cl)NC(=O)c2c(cccc2F)F RF00022 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H](C(O1)OC(C)(C)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00888 CO/N=C(/c1ccco1)\C(=O)Oc2c(c(c(c(c2Cl)Cl)Cl)Cl)Cl NRB03005 C[C@H]1[C@@H]([C@H]([C@H]([C@H](O1)OC[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)Oc3c(=O)c4c(cc(cc4OC(=O)C)OC(=O)C)oc3c5ccc(c(c5)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00889 CCOC(=O)C(C(F)(F)F)(NC(=O)C)OC RJC01972 c1ccc(cc1)C2=N/C(=C\c3cccc(c3)F)/C(=O)O2 NRB02990 CCOc1ccccc1/C=C(\C#N)/c2cccc(c2)Cl PHG00581 c1cc(ccc1C(C(CO)NC=C(C#N)C#N)O)[N+](=O)[O-] NRB04395 CC(=O)N1[C@@H](CS[C@@H]1[C@@H]([C@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)O)C(=O)N(C)C RJC00870 CCc1ccc(cc1)/C(=C/c2ccccc2Cl)/C#N PHG00905 c1cc(c(cc1NC(=O)/C=C/C(=O)O)O)C(=O)O RDR01892 COc1ccc(cc1)CCN2C(=O)CNC2=S RF03175 c1cc(cc(c1)Cl)CN2C(=O)CNC2=S RF03181 CC(=O)OC[C@H]([C@H]([C@@H](/C=N/N=C(N)N)OC(=O)C)OC(=O)C)OC(=O)C.Cl RJC00884 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] PD00341 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)NCCO)[N+](=O)[O-] PHG00966 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)CC4CCCO4)[N+](=O)[O-] PHG00991 COc1cc(cc(c1OC)OC)/C=c\2/c(=O)n3c4ccccc4nc3s2 RJC00852 CCOC(CNC(=O)[C@H](Cc1ccccc1)NC(=O)C)OCC RJC00856 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)Br RJC00859 c1cc(c(cc1NC(=O)CCC(=O)O)O)C(=O)O RDR01893 CCSC([C@@H]([C@H]([C@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)SCC NRB04507 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)[N+](=O)[O-] RJC00861 c1cc(ccc1NC(=O)NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)Cl RDR04007 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)Cc4ccco4)[N+](=O)[O-] PHG00961 CC(C)(C)CC(C)(C)NC(=O)c1ccc(cc1)[N+](=O)[O-] RF00001 c1ccc(cc1)/C=C/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00048 c1cc(ccc1/C(=C/c2ccc(c(c2)Cl)Cl)/C#N)[N+](=O)[O-] PHG00054 COc1ccc(cc1)/C(=C/c2ccc3c(c2)OCO3)/C#N PHG00069 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OCc2ccccc2)OC(=O)C)OC(=O)C)OC(=O)C RJC00900 c1ccc(cc1)CCNS(=O)(=O)c2cccc3c2nsn3 RJC00905 c1cc(ccc1C#N)S(=O)(=O)N2CCc3c(c4cc(ccc4[nH]3)F)C2 RJC01952 c1ccc2c(c1)C=CC(=O)C2=NNc3ccccc3F NRB02962 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1C)C)NC(=O)C RJC01975 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)NCCO)[N+](=O)[O-] PHG01006 c1ccc(cc1)C2CC(=O)N(C(=O)C2)c3ccc(cc3F)I PD00374 CCOC(=O)C(C(F)(F)F)(NC(=O)CC#N)O RJC01981 CC(=O)Oc1ccc(cc1OC)/C=C(\C(=O)OC)/NC(=O)c2ccccc2 NRB03000 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)Cc4cccnc4)Br PHG01018 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1C(F)(F)F)Cl)NC(=O)C RJC01986 c1ccnc(c1)CCN2C(=O)c3cccc4c3c(ccc4SCCO)C2=O PHG01042 C1COCCN1CCCNC(=S)N2CCOCC2 RDR01618 CSC(=CC(=O)c1cccc2c1cccc2)SC NRB04345 c1ccc(cc1)N/C(=C\C(=O)c2ccc(cc2)F)/SCc3c(cccc3Cl)Cl NRB04346 CC(C)(CCC(C)(C)N1C(=O)c2cccc3c2c(ccc3)C1=O)N4C(=O)c5cccc6c5c(ccc6)C4=O PHG00954 c1cc([nH]c1)C(=O)NNC(=O)C(F)(F)F RF03090 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)CCCN4CCOCC4)[N+](=O)[O-] PHG00531 CC1CN=C(S1)N(c2cccc(c2)C(F)(F)F)C(=O)Nc3ccccc3 RJC02017 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)CC4CCCO4)Br PHG01019 c1ccc(cc1)CCN2C(=O)CNC2=S RF03152 c1cnccc1CCN2C(=O)CNC2=S RF03155 c1c(nc[nH]1)CCN2C(=O)CNC2=S RF03162 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCCN4CCOCC4 PHG00872 CCc1ccc(cc1)/C(=C/c2cccc3c2cccc3)/C#N PHG00901 c1cc(ccc1NC(=O)NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)OC(F)(F)F RDR04008 C1C2C3C4C1C5C2C6C3C4C5(O6)CC(=O)O RJC00820 c1cc(c(c(c1)Cl)Cl)NC(=O)c2cccs2 RF00024 Cc1cc(nc(c1C#N)OC(=O)c2cccs2)C RF00032 c1cc(oc1/C=N/NC(=O)[C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O)[N+](=O)[O-] NRB04437 c1cc(ccc1[N+](=O)[O-])OCCCOc2ccc(cc2)[N+](=O)[O-] RDR01899 CC(=O)NC(=O)NC(C(=O)OC)(C(F)(F)F)O RJC01970 Cc1csc([n+]1C)NC2CCCCC2.[I-] RDR01702 C[n+]1c(csc1NC2CCCCC2)c3ccccc3.[I-] RDR01703 Cc1ccc(cc1)S(=O)(=O)/C(=C(/Nc2ccccc2)\SC)/C#N NRB04334 COc1ccc(cc1)n2c(nnn2)c3cnn(c3c4ccc(cc4)Cl)c5ccc(cc5)Cl NRB04318 CC(=O)OC[C@H]1[C@H]([C@@H]([C@H]([C@H](O1)OC2[C@H](O[C@H]([C@@H]([C@H]2OC(=O)C)OC(=O)C)OC)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00886 CCOC(=O)C(C(F)(F)F)(NC(C)C)NC(=O)c1ccccc1 RJC01995 COc1ccc(cc1)/C(=C/c2ccc(c(c2)OC)OC)/C#N PHG00071 c1cc(c(cc1NC(=S)N2CCCCCC2)Cl)Cl RDR01587 Cc1csc(=S)n1CC(=O)O NRB04503 CCOC(=O)C(C(F)(F)F)(NC1CCCCC1)NC(=O)C RJC01977 CCOC(=O)C(C(F)(F)F)(NC(=O)C)OC(C)C RJC01978 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2F)I)CC(=O)O PD00373 CC(C)(C)CC(C)(C)NC(=O)C(C)(C)C RF00019 c1cc(c(c(c1)Cl)Cl)NC(=O)C(Cl)Cl RF00021 CCOC(=O)C(C(F)(F)F)(NC(=O)c1cccc(c1)C(F)(F)F)O RJC01984 c1cc(ccc1/C(=C/c2ccc3c(c2)OCO3)/C#N)[N+](=O)[O-] PHG00045 COc1ccc(cc1OC)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00046 Cc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccc(cc3F)Cl NRB04330 CCc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3Cl)Cl NRB04332 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCCN4CCN(CC4)CCCN5C(=O)c6cccc7c6c(ccc7)C5=O PHG00933 c1cc(c(c(c1)Cl)C(=O)O/N=C(\c2ccc(o2)[N+](=O)[O-])/N)F RF02891 CC1(C2CCC1(C(C2)NC(=O)c3ccc(cc3)C(C)(C)C)C)C RJC01956 COc1cccc(c1)C(=O)OCC(=O)c2ccc(cc2)Cl RDR01612 Cc1nc(nc(n1)N/N=C/c2ccccc2O)N.Cl RF02942 c1ccc2c(c1)C=CC(=O)C2=NNc3ccccc3C#N NRB02973 c1ccc2c(c1)C=CC(=O)C2=NNc3cccc(c3)C#N NRB02974 CC1CCCC(N1C(=S)NCCCN2CCOCC2)C RDR01617 c1cc2c(ccc(c2c(c1)C(=O)O)C(=O)O)N PHG00507 c1ccc(cc1)COc2cccc(c2)/C=C(\C#N)/c3ccc(cc3)[N+](=O)[O-] PHG00052 c1ccc(cc1)n2c(nnn2)c3cnn(c3c4cccc(c4)Cl)c5ccc(cc5)Cl NRB04320 c1ccc(cc1)n2c(nnn2)c3cnn(c3c4cccc(c4)Cl)c5ccc(cc5)F NRB04323 C1CCC(CC1)NC(=S)N2CCOCC2 RDR01664 c1cc(oc1)CNC(=S)NC2CCCCC2 RDR01665 C1CCC(CC1)NC(=S)NCCO RDR01669 c1cc(ccc1/N=N/c2ccc(cc2)[N+](=O)[O-])N3C(=O)CSC3=S NRB04354 C[C@@]1\2CCC(C1)C(/C2=N\OC(=O)c3ccc(cc3)C(C)(C)C)(C)C RJC01965 CCCNC(=S)NC(=N)N1CCOCC1 RJC00857 c1cc(ccc1C(=O)/C=C/OC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl NRB04308 c1ccc(cc1)C(=O)C(=C2SCCCS2)C#N NRB04384 CCOC(=O)C(C(F)(F)F)(NC(C)C)NC(=O)C RJC01971 c1cc(ccc1/C=N/NC(=S)NCCCN2CCOCC2)Cl RDR01624 c1ccc(cc1)n2c(nnn2)c3cnn(c3c4ccc(cc4)Cl)c5ccc(c(c5)Cl)Cl NRB04319 C1C2CC3CC1CC(C2)(C3)NC(=O)NC(=O)CC#N RJC00844 CN(Cc1cccc(c1)Cl)/C(=N/C(=N\[N+](=O)[O-])/N)/SC NRB04391 CC(C)c1nc(nc(=O)n1C)/N=C/N(C)C RF02876 CC1(OC(=O)C(C(=O)O1)[C@@H]2C3C4CC5C2C6C3CC4C56)C RJC00824 COCCCNC(=O)c1ccc(cc1)[N+](=O)[O-] RF00006 CC(C)(C)CC(C)(C)NC(=O)c1cccs1 RF00010 CC(=O)c1ccc(c(c1)CSc2nnnn2c3ccc(c(c3)OC)OC)OC RDR01623 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)OC RJC00858 c1cc(ccc1c2cc3cc(ccc3oc2=O)Cl)[N+](=O)[O-] PHG00120 c1ccc(c(c1)C(=O)Nc2cccc(c2Cl)Cl)Cl RF00034 c1ccc(c(c1)C(=O)Nc2ccc(c(c2)N)Cl)O RDR01631 COc1cc(cc(c1OC)OC)C(=O)Nc2cccc(c2Cl)Cl RF00023 CCOC(=O)/C(=C/c1ccc(c(c1)OC)OC)/NC(=O)c2ccccc2 NRB02996 CC(=O)Nc1cc2cc(cc(c2oc1=O)Cl)Cl PHG00471 C/C(=C\c1cc(ccc1OC)Br)/[N+](=O)[O-] PD00323 CC1(C2CCC1(C(C2)NC(=O)c3c(cccc3Cl)Cl)C)C RJC01954 Cc1cccc2c1c(=O)cc(o2)c3ccc(cc3)Cl RJC00808 COc1ccc(cc1)C(=O)/C=C/OC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB04309 COc1ccc(cc1)C(=O)/C=C/Oc2ccc(cc2)Cl NRB04311 c1cc(ccc1S(=O)(=O)CC(CN2CCCC2=O)O)Cl RDR04026 c1ccc(cc1)C(C(=O)O)Nc2ccccc2C(=O)O PHG00205 CCOc1ccc(cc1)N2C(=O)c3cccc4c3c(cc(c4)[N+](=O)[O-])C2=O PHG00251 Cc1ccc(cc1)NC(c2ccccc2)C(=O)O PHG00304 CC(=O)ON1C(=O)c2cccc3c2c(ccc3)C1=O PHG00126 c1cc(ccc1C(=S)N)C(F)(F)F RF03219 Cc1c(c(nc(c1[N+](=O)[O-])C)O)C#N RF00054 Cc1cc(nc(c1C#N)Sc2ccccn2)C RF00063 c1ccc(cc1)C2OCC3C(O2)C(C(C(O3)OC4C(C(C5C(O4)COC(O5)c6ccccc6)O)O)O)O NRB02994 CC(=O)Nc1ccc(cc1)Cc2ccc(cc2)NC(=O)C PHG00073 Cc1ccc(cc1)/C(=C/c2cccc(c2)[N+](=O)[O-])/C#N PHG00856 c1cc(ccc1CN2C(=O)CNC2=S)[N+](=O)[O-] RF03169 COC(=O)c1ccc(nc1)C(=O)O RF03028 Cc1ccc(cc1)c2csc(n2)CO RF03062 COc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2F)Cl NRB04306 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2F)Cl)Br NRB04307 c1cc(c(cc1CCN2C(=O)CNC2=S)O)O RF03082 c1cn(cn1)CCCN2C(=O)CNC2=S RF03083 c1ccc(cc1)/C=C/C=C/N=N/C(=N)N RJC00841 c1cc(ccc1C(=O)/C=C/OC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)F NRB04310 c1ccc(cc1)c2ncc(c(n2)c3cccc(c3)F)c4nnnn4c5ccccc5 NRB04314 CCc1ccc(cc1)/C(=C/c2ccc(cc2)OC)/C#N PHG00902 Cc1cccc(c1/N=C/2\NC(CS2)(C)CO)C RDR01575 CC(=O)N1[C@H](CSC1[C@@H]([C@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)O)C(=O)N(C)C RJC00871 CCCN1CCCC(C1)NC(=S)Nc2ccc(cc2C)Br RDR01684 CCOC(=O)C(C(F)(F)F)(NC(=O)C)OCc1ccccc1 RJC01973 CCOC(=O)C(C(F)(F)F)(NC(=O)C)OCc1ccc(cc1)F RJC01974 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1OC)NC(=O)C RJC01976 COCCCNC(=O)c1ccc(cc1)/N=C/c2ccccc2O RF00012 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCNCCN4C(=O)c5cccc6c5c(ccc6)C4=O PHG00899 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CC4CCC(CC4)CN5C(=O)c6cccc7c6c(ccc7)C5=O PHG00900 c1ccc(cc1)S(=O)(=O)CC(=O)c2ccc(cc2)Cl RJC00860 CNC(=S)NC1CCCCC1 RDR01698 c1cc(oc1)C2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)O2 PHG00928 CC(C(=O)Nc1ccc(cc1)OC)ONC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RDR04084 CSc1nc(nc(n1)N2CCOCC2)N RF02736 CC1(C2CCC1(C(C2)NC(=O)c3ccc(cc3Cl)Cl)C)C RJC01955 CC1(C2CCC1(C(C2)NC(=O)c3ccco3)C)C RJC01958 COc1cccc(c1OC)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00079 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1)OCC RJC01993 COC(=O)c1ccc(nc1)C(=O)OC RF02989 CC1(C2C(=O)N3C(C(=O)N2C4(S1)C(=O)c5ccccc5C4=O)C(SC36C(=O)c7ccccc7C6=O)(C)C)C RJC00878 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC)OC(=O)C)OC(=O)C)OC(=O)C RJC00887 CC1(CS/C(=N\C2CCCCC2)/N1)C RDR01674 COc1ccccc1NC(=N)SCc2ccccc2.Cl RDR01677 Cc1cccc(c1NC(=N)NC(=N)N)C RDR01689 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)F)/C(=O)O2 NRB02989 CC(=O)OC[C@H]([C@H]([C@@H]([C@H](C(=O)c1ccccc1)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00839 C1CN2C(=N1)SC3=NCCN3C2=S NRB04292 COc1ccc(cc1)C(=O)/C=C/Sc2ccc(cc2)Cl NRB04297 c1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3)Cl NRB04255 c1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3Cl)Cl NRB04256 c1ccc(c(c1)CN2C(=O)CNC2=S)Cl RF03171 COc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccc(cc3F)Cl NRB04331 c1ccc(cc1)CN2C(=O)c3cccc4c3c(ccc4)C2=O PHG00876 COCCCNC(=O)c1cccs1 RF00008 CC(C)(C)CC(C)(C)NC(=O)c1c(cccc1F)F RF00011 CC(=O)OC[C@@H]([C@@H]([C@H]([C@@H](C(OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00831 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)N2CCOCC2)OC(=O)C)OC(=O)C)OC(=O)C NRB04436 c1ccc(cc1)CN2C(=O)CNC2=S RF03069 C([C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NN=C(N)N)O)O)O)O.N(=O)(=O)O RJC00879 c1ccnc(c1)CN2C(=O)CNC2=S RF03149 CC(=O)Nc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PHG00602 Cc1cc(ccc1Br)NC(=S)N2CCCCCC2 RDR01584 COc1cccc(c1OC)C2Nc3ccccc3C(=O)N2 RDR01590 c1cc(ccc1C(CS(=O)(=O)c2ccc(cc2)Br)(c3ccc(cc3)F)O)F RDR03989 Cc1cc(cc(c1[N+](=O)[O-])C)C(C)(C)C RDR03880 c1cc(ccc1/C=N/NC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)Cl RDR03920 CC(C)(C)CC(C)(C)NC(=O)c1cc(c(c(c1)OC)OC)OC RF00016 CC(C)(C)CC(C)(C)NC(=O)C(Cl)Cl RF00017 CCC1CCC(N(C1)C(=S)Nc2ccc(cc2C)Br)C RDR01685 CCC1CCC(N(C1)C(=S)Nc2ccc(c(c2)Cl)Cl)C RDR01686 CC(C)c1ccc(cc1)/N=C\2/NC(CS2)(C)C RDR01694 CC1CN=C(S1)Nc2ccc(cc2F)F RJC02016 Cn1c(nc2ccccc2c1=O)/C=C/c3ccccc3Cl NRB03068 c1cc(ccc1C(=O)/C(=C/2\NCCO2)/C#N)Cl NRB04337 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)CC4CCCO4)[N+](=O)[O-] PHG00960 c1cc2cccc3c2c(c1)C(=O)N(C3=O)Cc4ccco4 PHG00950 c1cc(ccc1N/N=C/Cc2nnnn2c3ccc(cc3)I)[N+](=O)[O-] NRB03175 c1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] NRB03177 c1c(c(cc(c1Cl)Cl)Cl)NC(=O)C(Cl)(Cl)Cl RF00049 CCOC(=O)CSc1c(c(cc(n1)C)C)C#N RF00050 c1cc(ccc1[N+](=O)[O-])OCCCCCCOc2ccc(cc2)[N+](=O)[O-] RDR01935 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2F RDR01938 c1cc(ccc1[N+](=O)[O-])OCCCCOc2ccc(cc2)[N+](=O)[O-] RDR01901 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Oc2ccc3ccccc3c2)OC(=O)C)OC(=O)C)OC(=O)C RJC00892 c1cc(c(c(c1)Cl)Cl)NC(=O)c2ccc(cc2)[N+](=O)[O-] RF00025 c1cc(c(c(c1)Cl)Cl)NC(=O)C(Cl)(Cl)Cl RF00026 CSC1=N/C(=C\c2ccc(s2)[N+](=O)[O-])/C(=O)N1CCOc3ccc(cc3)Cl RF03362 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(C)(C)CC(C)(C)C RF00040 Cc1cc(nc2c1c(n[nH]2)N)C RF00042 Cc1ccc(cc1)S(=O)(=O)/N=C\2/NC(C(O2)c3ccc(cc3)[N+](=O)[O-])CO NRB04410 c1ccc(cc1)CCNC(=S)N/N=C/c2cccs2 RDR01793 c1ccc2c(c1)c(=O)c(co2)/C=N/NC(=O)N RF00060 c1ccc2c(c1)c(=O)c(co2)/C=N/NC(=S)N RF00061 Cc1c(c(nc(c1[N+](=O)[O-])C)N2CCCCC2)C#N RF00093 CC1C(O/C(=N\S(=O)(=O)c2ccc(cc2)Cl)/N1C)c3ccccc3 NRB04414 CSC1=N/C(=C\c2ccc(cc2Cl)Cl)/C(=O)N1Cc3ccccc3 RF03197 c1ccc2c(c1)nc(o2)S/C=C/C(=O)c3ccc(cc3)Cl NRB04446 CCN(/C=C/c1nnnn1c2ccc(cc2)Cl)c3ccccc3 NRB03134 CCNc1nc(cs1)c2ccccc2.Br RDR01764 CCSc1ccc2c3c1cccc3C(=O)N(C2=O)Cc4ccccc4 PHG01049 CC1CN=C(S1)N(c2cccc(c2)F)C(=O)NC RJC02023 CN(C)c1ccc(cc1)/C=N/c2ccc3c(c2)OCO3 RB00007 CCOc1ccc(cc1/C=N/c2ccc3c(c2)OCO3)Br RB00008 Cn1c2c(con2)c(=O)n(c1=O)C RJC02067 CCOc1ccc(cc1)NC(=S)Nc2ccc(c(c2)Cl)Cl RB00014 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)/C=C/C(=O)O)Cl RB00018 c1ccc(cc1)Sc2ccc3c4c2cccc4C(=O)N(C3=O)NCCO PHG01048 c1cc2c(cc1N3C(=O)C=CC3=O)OCO2 RB00021 c1ccc(cc1)OCCN2C(=O)CNC2=S RF03258 Cc1cccc(c1)N(C2=NCC(S2)C)C(=O)Nc3ccccc3 RJC02028 Cc1ccccc1N(C2=NCC(S2)C)C(=O)Nc3ccccc3 RJC02030 c1ccc(c(c1)CO)S(=O)c2ccc(cc2C(=O)O)Cl RJC02055 CSC1=N/C(=C\c2ccccc2Cl)/C(=O)N1Cc3ccc(cc3)Cl RF03321 CSC1=N/C(=C\c2ccc(cc2)Cl)/C(=O)N1Cc3ccc(cc3)Cl RF03323 C1[C@H](NC(S1)C(=O)O)C(=O)O NRB04469 c1ccc(cc1)C(=O)c2ccccc2N/C=C/c3nnnn3c4ccc(cc4)Cl RJC02070 CSC1=N/C(=C/c2cccnc2)/C(=O)N1Cc3ccc(cc3)Cl RF03333 Cc1csc([n+]1C)Nc2cccc3c2cccc3.[I-] RDR01837 c1ccc(c(c1)OCCN2C(=O)CNC2=S)Cl RF03354 CC(=O)N1[C@@H](SC([C@H]1C(=O)O)(C)C)[C@H]([C@@H]([C@@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB04427 COc1nc(nc(n1)SC)N RF03315 CC(C)c1c2cc3c4c(c2oc(=O)c1Br)CCCN4CCC3 RJC00929 CCCc1ccc(nc1)c2ccc(cc2)C#N RJC00934 CC[n+]1c(csc1Nc2c(cc(cc2C)C)C)C.[I-] RDR01894 CC[n+]1ccsc1Nc2c(cccc2C)C.[I-] RDR01897 Cc1ccc(cc1)S(=O)(=O)NN[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC02172 c1cc(ccc1/C(=N/O)/N)C(F)(F)F RF03217 Cc1cc(nc(c1C(=O)O)O)C RF00089 Cc1c(c(nc(c1[N+](=O)[O-])C)N2CCOCC2)C#N RF00090 Cc1ccc(cc1)[C@@H]2N([C@H](C(S2)(C)C)C(=O)O)C(=O)C NRB04428 C[C@H]1[C@@H]([C@H]([C@H]([C@@H](O1)O[C@@H]2[C@H]([C@@H]([C@H](O[C@H]2Oc3cc(c4c(c3)O[C@@H](CC4=O)c5ccc(cc5)O)O)CO)O)O)O)O)O NRB04426 c1ccnc(c1)S/C=C/C(=O)c2ccc(cc2)Cl NRB04443 c1ccc(cc1)n2c(nnn2)/C=C/N3CCCC3 NRB03137 CC(C)(C)c1ccc(cc1)OC(=O)c2ccc(cc2Cl)Cl RDR01856 CSc1nc(nc(n1)N)c2ccc(cc2)C(F)(F)F RF03259 c1cc(ccc1OCCN2C(=O)CNC2=S)Cl RF03277 Cc1cc(ccc1Br)NC(=S)N/N=C/c2coc3ccccc3c2=O RF00107 c1cc(ccc1c2nc3c(c(n2)O)CSCC3)C(F)(F)F RF03920 Cc1cccnc1NC(=S)Nc2ccccc2Cl RB00089 CSC1=N/C(=C\c2ccccc2O)/C(=O)N1Cc3ccc(cc3)Cl RF03322 CCOC(=O)/C(=C/1\NC(C(O1)c2ccccc2)CO)/C#N NRB04408 CC(=O)OC[C@@H]([C@H]([C@H]([C@@H]([C@H]1N[C@@H](C(S1)(C)C)C(=O)OC)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB04433 c1ccc(cc1)[C@@H]2N[C@@H](CS2)C(=O)O NRB04457 c1cc(ccc1n2c(nnn2)/C=C/N3CCCCCC3)Br NRB03129 CSC1=N/C(=C\c2ccc(cc2)Cl)/C(=O)N1CCOc3ccc(cc3)Cl RF03341 C/C(=N\N=C(N)N)/c1ccccc1 NRB04483 c1ccc(cc1)Nc2nc(nc(=N)n2c3ccccc3)N NRB04479 COc1ccc(cc1)N/C(=N/C(=N)N)/N NRB04481 c1ccc(cc1)CN2C(=O)c3cccc4c3c(ccc4Sc5ccccc5)C2=O PHG01050 Cc1ccc(cc1)n2c(nnn2)/C=C/N3CCOCC3 NRB03140 Cn1c2c(c3c(c1=O)cc4ccc(cc4n3)[N+](=O)[O-])c(=O)n(c(=O)n2C)C RJC02059 COC(=O)c1cc(cc2c1NS(=O)S2)Cl RF03420 CN(C)/C=C/c1nnnn1c2ccc(cc2)Br NRB03121 Cc1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccn3 RB00003 c1cc2c(cc1/N=C/c3cc(ccc3O)Br)OCO2 RB00005 COc1ccc(cc1)OCCN2C(=O)CNC2=S RF03363 CN(C)/C=C\1/C(=O)N(C(=N1)SC)CCOc2ccc(cc2)Cl RF03366 Cc1ccc(cc1C)N/C(=N/C(=N\[N+](=O)[O-])/N)/SC NRB04392 Cn1c2c(c3c(c1=O)cc4cc(ccc4n3)[N+](=O)[O-])c(=O)n(c(=O)n2c5ccccc5)c6ccccc6 RJC02093 c1cc(cnc1)C/N=C/c2ccc(cc2Cl)Cl RF03428 COc1nc(nc(n1)OC)N RF03347 Cc1ccc2cc3c(c4c(n(c3=O)C)n(c(=O)n(c4=O)C)C)nc2c1 RJC02066 c1cc(ccc1[C@@H]2N[C@@H](CS2)C(=O)O)[N+](=O)[O-] NRB04465 CSC1=N/C(=C\c2ccccc2O)/C(=O)N1Cc3ccco3 RF03546 c1cc2c(cc1NC(=O)/C=C/C(=O)O)OCO2 RB00020 COc1ccc(cc1OC)C2CC(=O)Nc3ccccc3S2 RJC02089 CCOC(=O)CNC(=S)NN(C)C RF03388 CN(C)N1C(=O)/C(=C/c2cccc(c2)Cl)/N=C1SC RF03406 CC(=O)OCC(=O)c1ccc(cc1)C(F)(F)F RF03413 c1cc(ccc1C(=O)COC(=O)C(C(C(=O)OCC(=O)c2ccc(cc2)C(F)(F)F)O)O)C(F)(F)F RF03436 CC1([C@@H](NC(S1)c2cc(c(c(c2)OC)OC)OC)C(=O)O)C NRB04489 CC(C)(C)c1ccc(cc1)OC(=O)c2ccc(c(c2)Cl)Cl RDR01855 c1cc(oc1)CN2C(=O)CNC2=S RF03540 C/C(=N\N=C(NC(=O)C)NC(=O)C)/c1ccc(cc1)Br NRB04564 Cc1c(c(nc(c1[N+](=O)[O-])C)Sc2ccc(cc2)Cl)C#N RF00092 CN(C)N1C(=O)/C(=C/c2ccc(cc2)Cl)/N=C1SC RF03404 CN(C)N1C(=O)/C(=C/c2ccccc2Cl)/N=C1SC RF03405 CCc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccccc3C(=O)O RJC02075 c1ccc2c(c1)c(=O)c(co2)/C=N/NC(=O)CC#N RF00097 COc1ccc(cc1)NC(=S)N/N=C/c2coc3ccccc3c2=O RF00106 CSC1=N/C(=C\c2ccc(cc2)[N+](=O)[O-])/C(=O)N1CCOc3cccc(c3)Cl RF03417 C1C2CC3(CC1CC(C2)(C3)CO)CO RJC00940 C1C2CC3(CC1CC(C2)(C3)Br)CC(=O)O RJC00941 Cc1cc(nc(c1C#N)S)C RF00112 CC(C)(C)C(=O)OCC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F RF03422 c1cc(c(c(c1)Cl)C2N[C@@H](CS2)C(=O)O)Cl NRB04461 Cc1cc(nc2c1c(c(s2)C(=O)c3ccc(cc3)Cl)N)C RF00119 c1ccc(cc1)S(=O)(=O)CC(CN2CCCC2=O)O RDR04088 c1cc(cc(c1)F)NC(=N)NC(=N)NN.Cl RDR01649 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccc(cc1Cl)Cl)O RJC01987 CC(C(=O)NC(Cc1ccccc1)C(=O)O)NC(=O)OC(C)(C)C RJC01992 CC[n+]1c(csc1Nc2c(cccc2C)C)C.[I-] RDR01783 Cc1cc(ccc1[N+](=O)[O-])C(=O)N/N=C/c2coc3ccccc3c2=O RF00101 c1ccc2c(c1)c(=O)c(co2)/C=N/NC(=O)CCc3ccc(cc3)O RF00102 Cc1cc(cc(c1)OC(=O)c2ccc(cc2Cl)Cl)C RDR01794 Cc1cc(cc(c1)OC(=O)c2ccc(c(c2)Cl)Cl)C RDR01795 c1ccc2c(c1)c(=O)c(co2)/C=N/NC(=S)NCc3ccco3 RF00105 c1cc2cccc3c2c(c1)C(=O)N(C3=O)NCCO PHG00956 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)Cc4cccnc4)[N+](=O)[O-] PHG00963 C/N=C(/NC1CCCCC1)\SCc2ccccc2.Cl RDR01700 c1ccc(cc1)C2C(=O)Nc3ccccc3S2 PHG00186 c1cc(ccc1c2cc3cc(ccc3oc2=O)Br)[N+](=O)[O-] PHG00099 CN1C(=O)c2cccc3c2c(cc(c3Br)N)C1=O PHG00169 c1cnccc1CN2C(=O)CNC2=S RF03150 c1ccc(cc1)N/C=C\2/C(=O)c3ccccc3OC2=O NRB03062 CCc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(c(c3)Cl)Cl NRB04455 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C)NC(=O)Nc2ccccc2 RJC01998 c1ccc(c(c1)C2N[C@@H](CS2)C(=O)O)O NRB04462 c1cc(ccc1C2N[C@@H](CS2)C(=O)O)Cl NRB04463 COc1ccc(cc1)/N=C\2/N(C(=O)CS2)CCc3ccc(c(c3)OC)OC RDR01745 COc1ccc(cc1)CN2C(=O)CNC2=S RF03174 c1cc(ccc1CCN2C(=O)CNC2=S)Cl RF03153 COC(=O)c1ccc(nc1)C(=O)Nc2ccc(cc2)C(F)(F)F RF03164 c1ccc(cc1)C2=NN([C@@H](S2)[C@@H]([C@@H]([C@H]([C@H](CO)O)O)O)O)c3ccccc3 RJC00851 c1ccnc(c1)CCN2C(=O)c3cccc4c3c(ccc4)C2=O PHG00951 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1OC)NC(=O)Nc2ccccc2 RJC01999 CC1([C@@H](NCS1)C(=O)O)C NRB04496 CC1([C@@H](NC(S1)c2ccc(cc2)SC)C(=O)O)C NRB04492 CSC1=N/C(=C/c2cccnc2)/C(=O)N1Cc3ccccc3 RF03198 COc1ccc(cc1)NC(=S)NCCc2ccc(c(c2)OC)OC RDR01741 Cc1cccc(c1NC(=S)NCCc2ccc(c(c2)OC)OC)C RDR01742 CSC1=N/C(=C/c2cccnc2)/C(=O)N1CCOc3ccccc3Cl RF03372 Cc1ccc(cc1)n2c(nnn2)c3c[nH]c4c3cccc4 RJC02078 CC1(C=Cc2c(cc(c3c2OC(CC3=O)c4ccccc4)OC)O1)C RJC02082 CC[n+]1c(csc1Nc2ccc(cc2C)C)C.[I-] RDR01896 CCOC(=O)c1ccc(cc1)NC(=N)SCc2ccccc2.Cl RDR01676 Cc1cc(c(c(c1)C)NC(=N)Nc2nc(cc(n2)O)C)C RDR01656 c1ccc(cc1)CCNC(=S)Nc2cccnc2 RDR01659 c1cc(cnc1)NC(=S)NCc2ccc(c(c2)Cl)Cl RDR01660 COc1ccc(cc1Br)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00078 c1ccc(c(c1)C(=O)NCCOC(=O)c2ccccc2Cl)Cl RF00115 c1ccc2c(c1)CCN(C2CNC(=O)C3CCCCC3)C(=O)CN4CCOCC4 RJC00907 Cc1cc(c(c(c1)C)/N=C/c2ccc(c(c2)OC)OC(=O)c3ccc(cc3)Cl)C RDR01888 c1ccc2c(c1)cccc2NC(=O)c3ccc(c(c3)Cl)Cl RDR01816 c1ccc2c(c1)cccc2Nc3nc(cs3)c4ccc(cc4)Cl RDR01834 Cc1csc(n1)Nc2cccc3c2cccc3 RDR01836 Cc1cc(nc2c1c(c(s2)C(=O)c3ccccc3Cl)N)C RF00124 Cc1cc(nc2c1c(nn2C)N)C RF00080 Cc1cc(nc(c1C#N)Sc2ccccc2N)C RF00058 CC(=O)OC[C@@H]1[C@]2(CO[C@H]([C@@H]([C@H]2OC(=O)C)OC(=O)C)OC3[C@@H](CO1)OC([C@@H]([C@H]3OC(=O)C)OC(=O)C)Oc4ccccc4)OC(=O)C RJC00891 c1ccc(cc1)Cc2c(c3ccccc3[nH]c2=O)O NRB03058 C1CSC(N1)[C@@H]([C@@H]([C@H]([C@H](CO)O)O)O)O RJC00847 c1cc2c(c(c1)S(=O)(=O)N(CCC#N)C3CCCCC3)nsn2 RJC00908 CN(CCC#N)S(=O)(=O)c1cccc2c1nsn2 RJC00909 COc1ccc(cc1)C(=O)N/N=C/c2coc3ccccc3c2=O RF00103 CCN(CC)/C=C/c1nnnn1c2ccc(cc2)Cl NRB04450 COc1ccc(cc1OC)CCNC(=S)Nc2ccc(c(c2)Cl)Cl RDR01743 c1cc(c(c(c1)Cl)C(=O)NCCOC(=O)c2c(cccc2Cl)F)F RF00117 Cc1ccc(cc1)n2c(nnn2)/C=C/N(C)c3ccccc3 NRB03124 Cc1ccc(c(c1)C)Nc2[n+](c(cs2)C)C.[I-] RDR01797 CN(C)N1C(=O)c2cccc3c2c(ccc3Br)C1=O PHG01022 Cc1ccc(c(c1)[N+](=O)[O-])OC(=O)c2ccc(c(c2)Cl)Cl RDR01798 Cc1cc(c(c(c1)Cl)OC(=O)c2ccc(cc2Cl)Cl)Cl RDR01802 c1ccc2c(c1)cccc2NC(=O)c3ccccc3O RDR01818 c1cc(cc(c1)[N+](=O)[O-])/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PHG00604 COc1cc(cc(c1OC)OC)C(=O)Nc2cc3cc(cc(c3oc2=O)Br)Br PHG00783 c1ccc(cc1)CNC(=O)c2ccccc2Cl RF00002 CC(C)(C)CC(C)(C)NC(=O)c1cccc(c1)/N=C/c2ccccc2O RF00004 Cc1cccc(c1/N=C\2/N(C(=O)CS2)CCc3ccc(c(c3)OC)OC)C RDR01746 COc1cc(c(cc1Cl)OC)n2c(=O)c3ccccc3nc2SCC(=O)c4ccccc4 RDR01735 CCSc1ccc2c3c1cccc3C(=O)N(C2=O)NCCO PHG01047 C(=O)(N)NNC(=O)NNC(=O)N PHG00977 c1cc2c(ccc3c2c(c1)C(=O)N(C3=O)CCCN4CCOCC4)[N+](=O)[O-] PHG00967 c1cc(ccc1CSc2nccn2c3cc(ccc3Cl)Cl)Cl RDR01792 COc1ccc(cc1OC)CCNC(=S)Nc2ccc(cc2Cl)Cl RDR01744 CN/N=C/c1ccc(o1)c2ccc(cc2)[N+](=O)[O-] RDR01751 CC(C)N(CCC#N)S(=O)(=O)c1cccc2c1nsn2 RJC00906 Cc1ccc2c(c1)c3c([nH]2)C(=O)CCC3 RJC00911 Cc1cc(nc(c1C#N)SC)C RF00083 Cc1ccc(c(c1)N/C=C/c2nnnn2c3ccccc3)C(=O)c4ccccc4 RJC02069 c1ccnc(c1)CCN2C(=O)c3cccc4c3c(ccc4[N+](=O)[O-])C2=O PHG00962 CCOC(=O)c1ccc(cc1)NC(=N)SCc2ccc(cc2)Cl.Cl RDR01679 c1ccc(cc1)Cc2c(c3cccc4c3n(c2=O)c5c4cccc5)O NRB03018 Cc1cccc(c1)N(C2=NCC(S2)C)C(=O)NC RJC02027 Cc1cc(nc(c1C#N)SCc2c(c(c(c(c2C)C)C)C)C)C RF00081 CC(=O)OC[C@@H]([C@@H]([C@H]([C@@H](C(=O)Nc1ccc(cc1)Br)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00899 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NC(=O)N)OC(=O)C)OC(=O)C)OC(=O)C RJC00901 CN1/C(=N/O)/CC(=O)N(C1=O)C RJC02060 Cc1c2c(no1)n(c(=O)n(c2=O)C)C RJC02061 COc1ccccc1c2nnc(n2c3ccccc3)SCC(=O)O NRB04598 Cc1c(c(=O)n(n1C)c2ccccc2)NN=C3C(=O)OC(OC3=O)(C)C RJC02136 Cc1cc(nc(c1C#N)SCCC#N)C RJC02138 Cc1cc(nc2c1c(c(s2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)N)C RF00162 c1cc(ccc1C#N)OC(=O)c2ccc(c(c2)Cl)Cl RDR02076 c1cc(ccc1C#N)OC(=O)c2ccc(cc2Cl)Cl RDR02077 Cc1c(c(=O)n(n1C)c2ccccc2)N/N=C\3/C(=NN(C3=O)c4ccccc4)C RJC02141 CSc1c(c(cc(n1)c2cccs2)C(F)(F)F)C#N RF00201 COc1cc(cc(c1OC)OC)C(=O)Oc2ccc(cc2Cl)Cl RDR01940 COc1cccc(c1C(=O)NCCc2ccccc2)OC RDR01958 CS/C(=N\C(=N/[N+](=O)[O-])\N)/NCc1ccccc1Cl NRB04393 CS/C(=N\C(=N/[N+](=O)[O-])\N)/Nc1ccc(cc1)Cl NRB04394 C1COCCN1CC(=O)C23CC4CC(C2)CC(C4)C3 RJC00975 Cc1cc(nc(c1C#N)SS(=O)(=O)c2c(c(cc(n2)C)C)C#N)C RF00156 c1c(cc(cc1C(F)(F)F)/N=N/N2CCOCC2)C(F)(F)F RF00188 Cc1ccc(cc1)C(=O)/C=C/2\C(=O)NCCN2 RJC00932 C1C2CC3CC1CC(C2)NC3=O RJC00933 c1cc(c(c(c1)Cl)Cl)/N=N/N2CCOCC2 RF00189 c1cnn2c1[C@@H](n3c(ccn3)C2O)O RF03885 c1cc(sc1)c2cc(c(c(n2)O)C#N)C(F)(F)F RF00195 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NC(=S)N[C@@H]2[C@H]([C@@H]([C@H]([C@@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB04543 C/C(=N\NC(=O)N)/c1ccccc1 NRB04544 c1ccc(cc1)C(=S)NNc2ccccc2 NRB04545 c1cc(ccc1n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl NRB03182 COc1cc(cc(c1OC)OC)C(Sc2ccccc2)Sc3ccccc3 NRB03046 c1ccc2c(c1)c(=O)c(co2)/C=N/NC(=O)c3cccnc3 RF00099 c1ccnc(c1)S/C=C/C(=O)c2cccc(c2)Br NRB04444 c1ccc(cc1)c2cc(=O)n3c(csc3n2)c4ccccc4 RDR01713 C1C2CC3CC1CC(C2)(C3)CC(=O)N RJC00935 c1ccc2c(c1)CC(=C3c4ccccc4CC3=O)C2 NRB03165 C1C2CC3(CC1CC(C2)(C3)CC(=O)O)CC(=O)O RJC00937 c1ccc(cc1)C(=O)CC(=O)C(=O)Nc2ccccc2 RJC00939 c1cc(c(cc1Cl)Cl)NC(=O)c2cnccc2C(F)(F)F RF03973 c1cc(ccc1n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])I NRB03184 Cc1cc(ccc1Br)NC(=O)C(Cl)(Cl)Cl RDR02030 CC(C)c1ccc(cc1)N2Cc3cc(ccc3[N+](=C2)C)C(C)C.[I-] RB00045 CSC(=N)Nc1ccccc1.I NRB04582 c1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccccc4 RJC02112 CSC1=N/C(=C\c2ccc(s2)[N+](=O)[O-])/C(=O)N1Cc3ccco3 RF03548 COc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccccc3C(=O)O RJC02076 c1ccc(c(c1)C(=O)O)N/C=C/c2nnnn2c3ccc(cc3)F RJC02077 c1ccc(cc1)c2cn(c(n2)N)Nc3ccccc3 NRB04593 c1ccc(cc1)/C(=C/C=C(C#N)C#N)/Sc2nnnn2c3ccccc3 RJC02080 c1ccc(cc1)C2=NN(C(C2)c3ccc4c(c3)OCO4)c5ccccc5 RJC02120 Cc1ccc(cc1)C2=NN(C(C2)c3ccccc3)c4ccccc4 RJC02124 CC(=O)NC(C(F)(F)F)(C(F)(F)F)N(c1nc2ccccc2s1)c3nc4ccccc4s3 RJC02085 COc1cc(cc(c1OC)OC)C(=O)Oc2ccc(cc2)C#N RDR02079 Cn1c2c(c3c(c1=O)cc4cc(ccc4n3)F)c(=O)n(c(=O)n2c5ccccc5)c6ccccc6 RJC02094 c1ccnc(c1)SC2CC(=O)N(C2=O)c3ccc(cc3Br)Cl RB00001 COc1ccccc1C2CC(=NN2c3ccccc3)c4ccccc4 RJC02114 COc1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccccc4 RJC02115 c1ccc(cc1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccccc4 RJC02117 c1ccc2c(c1)c(c(nn2)O)O RF03470 c1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccn3 RB00002 COc1ccc(cc1OC)C2CC(=NN2c3ccccc3)c4ccccc4 RJC02121 c1cc(ccc1C(=O)NN)C(F)(F)F RF03473 c1ccc(cc1)C(=O)c2cc(ccc2N3C(=O)C=CC3=O)Cl RB00019 c1cc(c(c(c1)Cl)Cl)N/C(=N/C(=N)N)/N NRB04516 CSC(=C(C#N)C#N)NC(c1ccccc1)C(=O)O NRB04525 c1cc(=O)oc2c1cc(c(c2)O)O[C@H]3[C@@H]([C@H]([C@@H]([C@H](O3)CO)O)O)O RJC00925 COc1ccc(cc1Br)/C=C\2/C(=O)NC(=O)N2 RB00049 c1cc(cc(c1)NC(=S)NCCO)C(F)(F)F RB00077 Cc1cc(=O)oc2c1cc3c4c2CCCN4CCC3 RJC00927 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Oc2c(cc(cc2Br)Br)Br)OC(=O)C)OC(=O)C)OC(=O)C NRB04531 c1cc2c(cc1[N+](=O)[O-])sc(n2)N NRB04532 c1cc(ccc1NC(=S)NCCO)Cl RB00016 c1cc(ccc1NC2=NCCS2)Cl RB00017 COc1ccc(c(c1)NC(=S)NCCO)OC RB00274 c1ccc(cc1)C(=O)NC(=S)NCCc2ccccn2 RB00276 c1ccc(cc1)C(=O)c2cc(ccc2N3C(=O)CC(C3=O)Sc4ccccc4N)Cl RB00022 CCOC(=O)Nc1nc2c(s1)c3c(s2)CCCC3 RJC00923 Cc1ccc(cc1)C23CC4CC(C2)CC(C4)C3 RJC00943 CSC1=N/C(=C\c2ccc(cc2)Cl)/C(=O)N1Cc3ccco3 RF03547 CCc1ccc(cc1)C(=O)/C=C/S/C(=N/C#N)/SC NRB03187 Cc1cccnc1NC(=S)Nc2cccc(c2)C(F)(F)F RB00090 Cc1cc(nc2c1c(c(s2)C(=O)c3ccc(cc3)[N+](=O)[O-])N)C RF00122 COc1cccc(c1)NC(=S)NC(=O)c2ccccc2 RB00290 Cc1cc(c2c(c1)c(=O)c3cc(c(nc3o2)N)C#N)C RJC01064 COc1cc(cc(c1OC)OC)C(=O)NCc2ccco2 RDR01939 Cc1cc(cc(c1)OC(=O)c2cc(c(c(c2)OC)OC)OC)C RDR01942 c1ccc(cc1)NC(=O)Sc2ccc(cc2F)F RF03745 CC(=O)OC[C@@H]([C@@H]([C@H]([C@@H](C(=O)O)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB04524 CC(=O)O.c1cc(c(cc1Cl)Cl)/C=N/N=C(N)N NRB04536 c1cnccc1c2nc(nc(n2)N)N RDR01973 c1ccc(cc1)C2=NN(C(C2)c3c(cccc3Cl)Cl)c4ccccc4 RJC02119 c1ccc2c(c1)C(=O)N(C2=O)CCC34CC5CC(C3)CC(C5)C4 RJC00952 c1ccc2c(c1)C(=O)N(C2=O)CC34CC5CC(C3)CC(C5)(C4)Br RJC00954 c1cc(c(cc1)O)/C=N/c2ccc(cc2)OCCCOc3ccc(cc3)/N=C/c4c(cccc4)O RDR01977 C(COC(=O)C(Cl)(Cl)Cl)NC(=O)C(Cl)(Cl)Cl RF00114 Cc1cc(nc(c1C#N)SCC(=O)c2ccc(cc2)[N+](=O)[O-])C RF00121 CC1CCCC(N1C(=O)c2cc(c(c(c2)OC)OC)OC)C RDR01957 COc1cc(cc(c1OC)OC)C(=O)NCCc2ccccc2 RDR01959 c1ccc(cc1)n2ccc(n2)/C=N/c3ccc(cc3)Cl RF03905 Cn1c2ccccc2c(c(c1=O)c3ccccc3)OS(=O)(=O)c4ccc(cc4)Br RJC02090 CCOc1ccc(cc1OC)C2CC(=NN2c3ccccc3)c4ccccc4 RJC02122 CN(C)c1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccccc4 RJC02127 CC1([C@@H](NC(S1)c2ccccc2)C(=O)O)C NRB04491 c1cc(cnc1)c2nc(nc(n2)N)N RDR01974 c1coc(c1)/C=N/c2ccc(cc2)OCCCOc3ccc(cc3)/N=C/c4occc4 RDR01975 CC1([C@@H](NC(S1)C(=O)O)C(=O)O)C NRB04495 CC1(C(NC(S1)(C)C)C(=O)O)C NRB04497 Cc1cccc(c1/N=C(/N(C)C)\SC)C.I RDR01987 c1ccc(cc1)/C=N/N=C(N)N NRB04482 Cc1ccc(c(c1)C)N/C(=N/C)/SC.I RDR01997 c1cc(ccc1N)OCCCCCCOc2ccc(cc2Cl)Cl RDR02004 COc1ccc(cc1OC)/C(=C\c2ccc(cc2)Cl)/C(=O)O RDR01933 COc1cc(cc(c1OC)OC)C(=O)Nc2cccc(c2)F RDR01937 Cc1cc(nc2c1c(c(s2)C(=O)c3ccc(cc3)F)N)C RF00125 Cc1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccccc4 RJC02128 CC1(CC(=O)C(=NNc2ccccc2C(F)(F)F)C(=O)C1)C RJC02134 c1cc(ccc1N/N=C/Cc2nnnn2c3ccc(cc3)Cl)[N+](=O)[O-] NRB03173 CC(=O)OC[C@@H]([C@H]([C@H]([C@@H]([C@H]1N[C@H](C(S1)(C)C)C(=O)OC)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB04501 Cc1c(c(=O)n(n1C)c2ccccc2)NN=C3C(=O)CC(CC3=O)(C)C RJC02142 Cc1c(c([nH]n1)N)c2ccccc2 RJC02145 Cc1cc(c(c(c1)C)NC(=O)c2c(cccc2OC)OC)C RDR01953 c1ccc(cc1)n2c(nnn2)/C=C/N3CCCCCC3 NRB03130 c1cc(ccc1n2c(nnn2)/C=C/N3CCCCC3)Br NRB03133 Cc1cc(nc(c1C#N)OC)C RF00141 Cc1cc(nc2c1c(c(s2)C(=O)Nc3ccc(c(c3)Cl)Cl)N)C RF00126 Cc1cc(nc2c1c(c(s2)C(=O)Nc3cccc(c3)SC)N)C RF00127 Cc1c(c(nc(c1[N+](=O)[O-])C)NC)C#N RF00128 Cc1c(c(nc(c1[N+](=O)[O-])C)N(C)C)C#N RF00129 CCOc1ccc(cc1OC)C2CC(=O)Nc3ccccc3S2 RJC02097 c1cc(ccc1N/N=C/Cc2nnnn2c3ccc(cc3)Br)[N+](=O)[O-] NRB03174 CC(=O)OC[C@@H]([C@@H]([C@H]([C@@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB04555 CCOC(=O)c1c(n[nH]c1NNC(=S)Nc2ccccc2Cl)C NRB04563 Cc1cc(nc2c1c(c(s2)C(=O)c3ccc(cc3)Cl)n4cccc4)C RF00139 c1cncc(c1C(F)(F)F)C(=O)O RF03948 C1C2CC3CC1CC(C2)(C3)C(=O)NO RJC00955 CSC1=N/C(=C\c2ccccc2Cl)/C(=O)N1CCOc3cccc(c3)Cl RF03415 c1ccc(cc1)c2cc(nc(n2)SCC(=O)c3ccc(cc3)[N+](=O)[O-])O RDR01708 c1ccc(cc1)c2cc(=O)n3c(csc3n2)c4ccc(cc4)[N+](=O)[O-] RDR01712 CC(C)c1ccc(cc1)NC(=S)Sc2ccc(cc2F)F RF03751 Cc1cc(nc(c1C#N)OC(C)C)C RF00142 CCOCCOc1c(c(cc(n1)C)C)C#N RF00143 CCCN/C(=C/1\C(=O)C(=O)N(C1=O)c2ccccc2)/c3ccccc3 RJC02102 c1ccc(cc1)C2=NN(C(C2)c3cccc(c3)Cl)c4ccccc4 RJC02116 Cc1nc(c(c(n1)SC)C#N)N RF03694 c1ccc(cc1)N/N=C/c2ccc(o2)c3ccc(cc3)[N+](=O)[O-] RDR01752 c1ccc(cc1)Nc2ccccc2C(=O)OCC(=O)c3ccc(cc3)Cl RDR01756 Cc1cc(nc(c1C#N)Sc2cc(nc(n2)N)C)C RDR02040 Cc1cc(nc(n1)N)NCc2cccnc2 RDR02058 Cc1cc(nc(n1)N)NCCc2ccc(c(c2)OC)OC RDR02059 CC(=O)OC[C@H]([C@H]([C@@H](C(=O)[O-])OC(=O)C)OC(=O)C)OC(=O)C.[K+] NRB04523 C1CCc2c(c\3c(nn2)CCC/C3=N/O)C1 RJC02164 CCOC(=O)C(C)Oc1ccc(cc1)NC(=O)C(Cl)Cl RDR02013 CCOC(=O)C(C)Oc1ccc(cc1)NC(=O)C(Cl)(Cl)Cl RDR02014 CC1([C@@H](N[C@H](S1)CNC(=O)Cc2ccccc2)C(=O)O)C NRB04527 c1cc(c(cc1Br)Cl)NC(=O)C(Cl)(Cl)Cl RDR02031 Cc1cc(ccc1NC(=S)NCCc2ccc(c(c2)OC)OC)Cl RDR01767 C1C2CC3CC1CC(C2)(C3)CC(=O)NN RJC00936 c1ccc(c(c1)CC2=NCCN2)Cl RB00038 CCC(=O)OCCC(=O)N1C=Cc2ccccc2C1C#N RB00063 CC(C)(/C(=N\O)/c1ccccc1)NO RJC02154 Cc1cc(c(cc1C)N/C(=N/C)/SC)C.I RDR01980 c1cnnc2c1-c3c(non3)CC2 RJC02158 Cc1cnnc2c1-c3c(non3)CC2 RJC02159 COc1ccc(c(c1)c2cc(nc(c2)c3cccc(c3)[N+](=O)[O-])c4ccccc4)OC RB00119 c1cc(ccc1C[C@@H](C(=O)O)N)[N+](=O)[O-] RJC02057 Cc1cc(nc2c1c(c(s2)C(=O)C)N)C RF00145 c1ccc2c(c1)c(=O)c(co2)/C=N/NC(=O)c3ccco3 RF00098 Cn1cc(c(n1)/C=N/O)Cl RF03966 c1cc(ccc1C23CC4CC(C2)CC(C4)(C3)Br)[N+](=O)[O-] RJC00956 COC(=O)CNC(=O)NC12CC3CC(C1)CC(C3)C2 RJC00966 c1ccc2c(c1)nc(o2)S/C=C/C(=O)c3ccc(cc3)F NRB04635 C([C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NNC(=S)N)O)O)O)O NRB04541 Cc1cc(nc(n1)N)OC(C)C RDR02028 Cc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] NRB03178 Cc1cc(ccc1NC(=O)C(Cl)(Cl)Cl)Br RDR02029 c1ccc(cc1)C(C#N)O[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)CO[C@H]3[C@@H]([C@H]([C@@H]([C@H](O3)CO)O)O)O)O)O)O NRB04549 c1cc(oc1C(=O)NN)[N+](=O)[O-] NRB04554 CCOC(=O)C(C(C(=O)c1ccc(c(c1)OC)OCc2ccccc2)C(=O)OCC)C(=O)c3ccc(c(c3)OC)OCc4ccccc4 NRB03040 c1ccc2c(c1)c(=O)n(c(n2)SCC(=O)c3ccc(cc3)Cl)c4ccc(c(c4)Cl)Cl RDR01733 c1ccc(cc1)Sc2ccc3c4c2cccc4C(=O)N(C3=O)CCc5ccccn5 PHG01040 CCCSc1ccc2c3c1cccc3C(=O)N(C2=O)CCc4ccccn4 PHG01044 COc1ccc(c(c1)OC)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccccc4 RJC02131 CC(C(=O)C12CC3CC(C1)CC(C3)C2)N(C)C.Cl RJC00964 C([C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NN=C(N)N)O)O)O)O.Cl NRB04542 Cc1ccc(cc1)S(=O)(=O)NNC(=S)NC(C)(C)C NRB04573 CN(C)CCOC(=O)C12CC3CC(C1)CC(C3)C2 RJC00973 c1cc(ccc1OC(=O)c2ccc(cc2Cl)Cl)F RDR02007 COc1cc(cc(c1OC)OC)C2CC(=NN2c3ccccc3)c4ccccc4 RJC02123 CCSC([C@H]([C@@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)SCC NRB04508 c1cc(ccc1C#N)OC(=O)c2ccc(cc2)Cl RDR02075 CC1CN=C(S1)N(c2ccc(c(c2)Cl)F)C(=O)Nc3ccccc3 RJC02024 c1ccc(c(c1)C#N)N/C=C/c2nnnn2c3ccc(cc3)F RJC02071 Cc1ccc2c(c1)c3c(n2CCC#N)C(=O)CCC3 RJC00914 c1ccc2c(c1)C=CN(C2C#N)C(=O)C3=CCCCC3 RJC00917 c1cnccc1CNC(=S)N RB00196 Cc1ccnc(n1)S/C=C/C(=O)c2ccccc2 NRB04641 c1cnccc1/C=C(/C#N)\C(=O)N RB00243 Cc1c(cc(nc1c2ccccc2)c3ccc(cc3)Cl)c4ccccc4 NRB03282 Cn1cc(c(n1)/C=C(\C#N)/S(=O)(=O)c2ccccc2)Cl RF04086 COc1ccc(cc1)C(CC(=O)c2ccccc2)SC(=O)c3ccccc3 RB00258 c1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)SC(=O)c3ccccc3 RB00261 c1cc(ccc1C#N)OS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl RDR02081 c1cc(ccc1n2c(nnn2)/C=C/N3CCCCC3)F NRB03215 CC([C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC)OC(C)(C)C.C1CCC(CC1)N RJC02223 Cc1cc(c(cc1C)NC(=N)SC)C.I RDR02103 Cc1cc(c(cc1C)N/C(=N/C)/NN)C.I RDR02105 Cc1cc(nc(c1C#N)SC(c2ccccc2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C RF00239 c1cc(ccc1S(=O)(=O)O[C@H]2CN3CCC2CC3)Br.Cl RJC01010 CCc1ccc(cc1)NC(=N)NC(=N)N.Cl RDR02130 c1cc(sc1)c2cc(c3c(c(sc3n2)C(=O)c4ccc(cc4)[N+](=O)[O-])N)C(F)(F)F RF00204 Cc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3)[N+](=O)[O-] NRB03169 CCc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3)[N+](=O)[O-] NRB03170 CCc1ccc(cc1)C(=O)/C=C/Sc2ccccn2 NRB04629 COc1ccc(cc1)C(=O)/C=C/Sc2ccccn2 NRB04630 c1ccnc(c1)S/C=C/C(=O)c2ccc(cc2)F NRB04631 Cc1cc(ccc1NC(=N)NC(=N)N)Cl.Cl RDR02089 C=CCSc1[nH]c2ccccc2n1 RDR02091 Cc1cc(nc(c1C#N)SC(c2ccccc2)C(=O)Nc3ccc(cc3)C(C)C)C RF00240 Cc1cc(c(cc1C)/N=C(\NN)/N(C)C)C.I RDR02110 CC(C)(C)S(=O)(=O)/C(=C/c1c(cn(n1)C)Cl)/C#N RF04095 Cn1cc(c(n1)/C=C(\C#N)/C(=O)c2ccc(cc2)Cl)Cl RF04096 Cn1cc(c(n1)C=C(C#N)C#N)Cl RF04100 Cc1cc(nc(c1C#N)SC(c2ccccc2)C(=O)Nc3cc(c(cc3OC)Cl)OC)C RF00243 Cc1cc(nc(c1C#N)SC(c2ccccc2)C(=O)Nc3ccc4c(c3)OCO4)C RF00245 Cc1cc(nc(c1C#N)SC(c2ccccc2)C(=O)NC(C)(C)C)C RF00248 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)N2CCC[C@H]2C(=O)O RJC02221 CC(C)(C)OC[C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)N RJC02222 Cc1cc(nc(c1C#N)SC(c2ccccc2)C(=O)Nc3c(cccc3F)F)C RF00238 c1ccc(cc1)c2ccc(cc2)n3c(nnn3)/C=C/N4CCCCCC4 NRB03221 C#CCSc1[nH]c2ccccc2n1 RDR02092 C#CCSc1nnc(o1)c2ccco2 RDR02099 c1cncc(c1C(F)(F)F)c2nnc(o2)C3CCCCC3 RF04091 Cn1cc(c(n1)/C=C(\C#N)/S(=O)(=O)c2ccccn2)Cl RF04093 c1ccc(cc1)n2c(nnn2)/C=C/Nc3ccccc3C(=O)O NRB03235 Cc1ccccc1SC(CC(=O)c2ccccc2)c3ccc(cc3)OC RB00257 c1ccc(cc1)C(=O)NC(=S)NCc2cccnc2 RB00197 c1cncc(c1C(F)(F)F)c2nc(no2)c3cc(cc(c3)Cl)Cl RF04110 COc1ccc(cc1OC)CCNC(=O)C(c2ccccc2)Sc3ccccn3 RF00266 c1ccc(cc1)C(C(=O)Nc2c(cccc2F)F)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N RF00275 Cc1cc(no1)NC(=O)Nc2cnccc2C(F)(F)F RF04125 c1cc(cnc1)CNC(=O)Nc2cnccc2C(F)(F)F RF04126 CCOC(=O)C1=C(NC(=O)NC1c2ccccc2)C RF00278 CCOC(=O)C1=C(NC(=O)NC1c2ccc(c(c2)Cl)Cl)C RF00279 CCOC(=O)C1=C(NC(=O)NC1c2cc(c(c(c2)OC)OC)OC)C RF00281 Cc1cc(nc(c1C#N)SC(c2ccccc2)C(=O)Nc3cc(ccc3Cl)C(F)(F)F)C RF00247 COc1ccc(cc1)N/C=C\c2nnnn2c3ccccc3 NRB03226 c1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)O NRB03230 c1cc(ccc1n2c(nnn2)/C=C/N3CCOCC3)F NRB03218 CCc1cccc(c1N2C(=NC(=NC2(C)C)N)N)CC.Cl RB00303 c1ccc(cc1)n2c(nnn2)/C=C\Nc3ccccc3Cl NRB03227 c1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)Cl NRB03228 c1cc(sc1)c2nc(cs2)CNC(=O)Nc3ccc(cc3Cl)Cl SCR01339 c1cc(sc1)c2nc(cs2)CNC(=O)Nc3ccc(cc3)C(F)(F)F SCR01338 CC(=O)N1[C@@H](CS[C@H]1[C@@H]([C@H]([C@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)C(=O)OC NRB04625 Cc1ccc(cc1Cl)/N=C/c2cccs2 RB00129 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2ccc(cc2)Cl NRB04626 Cc1cc(c(c(c1)C)n2c(nnn2)SC)C RDR02133 c1cc(ccc1NC(=O)C(Cl)Cl)Br RDR02141 Cc1ccc(cc1)n2c(nnn2)C/C=N\NC(=S)N NRB03237 c1cc2c(cc1Cl)[nH]c(=O)[nH]c2=O RB00270 Cc1ccc2c(c1)c(=O)[nH]c(=O)[nH]2 RB00271 CC(C)c1ccc2c(c1)c(=O)c3cc(c(nc3o2)N)C#N RJC01059 COc1ccc(c(c1)NC2=NCCS2)OC RB00275 c1ccc(cc1)C(C(=O)Nc2cc(c(cc2Cl)Cl)Cl)Sc3ccc(cc3)Cl RF00282 Cc1cccc(c1NC(=O)C(c2ccccc2)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N)Cl RF00284 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC[C@@H]2[C@H]([C@@H]([C@H]([C@@H](O2)OC(C#N)c3ccccc3)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C NRB04615 Cc1cc(=O)[nH]c(n1)N/N=C\c2cccc3c2cccc3 NRB04621 CCOc1ccc(cc1)/N=C/c2cccs2 RB00127 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2)[N+](=O)[O-])C RF00289 c1cc(ccc1n2c(nnn2)C/C=N\NC(=S)N)F NRB03240 c1cc(ccc1n2c(nnn2)C/C=N\NC(=S)N)Cl NRB03241 c1cc(ccc1n2c(nnn2)C/C=N\NC(=S)N)Br NRB03242 c1cc(ccc1n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])F NRB03181 c1ccc(cc1)C(=O)NC(=S)N2CCOCC2 RB00139 c1ccc(cc1)C(=O)NC(=S)N2CCCC2 RB00141 c1ccc(cc1)CCN2C(=O)C=CC2=O RB00158 Cc1cc(c(c(c1)C)NC(=O)C(C)(C)C)C RDR02145 Cc1cccc(c1n2c(nnn2)SCC#C)C RDR02152 Cc1ccc(c(c1)C)n2c(nnn2)SCC#C RDR02153 Cc1c(cc(nc1c2ccc(cc2)F)c3ccccc3)c4ccccc4 NRB03278 Cc1c(cc(nc1c2ccc(cc2)Cl)c3ccccc3)c4ccccc4 NRB03280 CCOC(=O)NC(=S)NCCO RB00163 C1C2CC(C1C=C2)NC(=S)NCCO RB00164 CCOC(=O)CSC(=S)Nc1ccc(cc1)OC RDR02158 CC1=C(N2C([C@H](C2=O)NC(=O)[C@H](c3ccccc3)N)SC1)C(=O)[O-].[Na+] RJC02206 COC(=O)/C=C/1\C(=O)C=C(O1)c2ccccc2 RJC00987 CCOC(=O)C1=C(NC(=O)NC1c2ccccc2Cl)C RF00285 CCc1ccc(cc1)n2c(nnn2)C/C=N/NC(=S)N NRB03238 c1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)C(=O)O NRB03231 c1ccc(cc1)n2c(nnn2)/C=C\Nc3cccc4c3cccc4 NRB03232 c1ccc(cc1)n2c(nnn2)C/C=N\NC(=S)N NRB03236 CCOC(=O)NC(=S)NN RB00159 Cc1ccc(cc1)N/C=C\c2nnnn2c3ccccc3 NRB03224 COc1ccccc1N/C=C\c2nnnn2c3ccccc3 NRB03225 CCOC(=O)CSC(=S)Nc1c(cc(cc1C)C)C RDR02159 CCOC(=O)CSC(=S)Nc1ccc(cc1)Cl RDR02160 CCOC(=O)CSC(=S)Nc1ccccc1Cl RDR02161 c1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc4ccccc4c3 NRB03233 c1ccc(cc1)n2c(nnn2)/C=C/Nc3cccc(c3)Cl NRB03234 CCc1cccc(c1NC(=O)C(c2ccccc2)Sc3ccccn3)CC RF00257 Cc1cccc(c1)c2nc(nc(n2)N)N RDR02083 c1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)Br NRB03229 c1cc(sc1)/C=N/c2ccc(cc2)O RB00133 c1ccc(cc1)C(=O)OC[C@@H]2[C@H]([C@@H](/C(=N/OC(=O)c3ccccc3)/CO2)OC(=O)c4ccccc4)OC(=O)c5ccccc5 RJC02209 C/C(=N\N=C(N)N)/c1cccs1 RJC02212 CCOC(=O)/C=C(\C)/NN=C(c1ccccc1)c2ccccc2 RJC00982 c1ccc(cc1)c2ccc(cc2)n3c(nnn3)C/C=N/NC(=S)N NRB03244 c1ccc(cc1)C2=CC(=O)C3(C2=C(C=C(O3)c4ccccc4)c5ccc(cc5)Br)c6ccccc6 NRB03245 Cc1cc(nc(c1C#N)SCC#C)C RF00202 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)N(C)C)C RF00287 CC1(N=C(N=C(N1c2c(cccc2Cl)Cl)N)N)C.Cl RB00301 CN1c2ccccc2/C(=N/O)/C1=O RJC02195 Cc1cc(ccc1NC(=N)NC(=N)N)Br RDR02132 Cc1cc(c(c(c1)C)n2c(nnn2)SCC=C)C RDR02135 CSc1c(c(nc(n1)c2cccnc2)N)C#N RF04037 c1c(c(n[nH]1)/C=N/O)Br RF03952 c1cc(ccc1NC(=O)c2cnccc2C(F)(F)F)Cl RF03968 Cn1cc(c(n1)c2nc(on2)c3ccccc3C(F)(F)F)Cl RF04178 c1cc(cc(c1)Cl)c2nnc(o2)c3cnccc3C(F)(F)F RF04087 COc1cc(c(cc1NC(=O)C(c2ccccc2)Sc3ccc(cc3)Cl)Cl)OC RF00254 c1ccc(cc1)C(C(=O)Nc2cc(ccc2Cl)C(F)(F)F)Sc3ccccn3 RF00255 CC(C)(C)C(=O)Nc1ccc(cc1)Br RDR02140 c1ccc(cc1)C(C(=O)Nc2cc(c(cc2Cl)Cl)Cl)Sc3ccccc3N RF00283 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)NCCC(=O)O RJC02202 c1ccc(cc1)n2c(c3c(n2)CCSC3)O RF03842 CCOC(=O)c1ccc(cc1)c2ccc(o2)/C=N/NC(=S)Nc3ccc(cc3)OC RDR01930 c1ccc(c(c1)NC(=S)N/N=C/c2cc[nH]n2)F RF03912 COc1ccc(cc1OC)CCNC(=O)C(c2ccccc2)Sc3ccc(cc3)Cl RF00264 Cc1cccc(c1NC(=O)C(C)(C)C)C RDR02148 Cc1c(c(nc(n1)S)O)CC=C RDR02150 Cc1ccc(cc1)c2cc(cc(n2)c3ccccc3)c4ccccc4 NRB03269 COc1cc(c(cn1)C(=O)N)C(F)(F)F RF04202 CCc1cccc(c1NC(=O)C(c2ccccc2)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N)CC RF00276 c1ccc(cc1)C(C(=O)Nc2cc(c(cc2Cl)Cl)Cl)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N RF00277 c1ccc(cc1)C(C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Sc3ccccc3N RF00288 Cc1ccc(cc1)S(=O)(=O)NC(=N)NCCC[C@@H](C(=O)O)NC(=O)OC(C)(C)c2cc(cc(c2)OC)OC RJC02203 Cc1cccc(c1Nc2nnc(s2)S)C RB00138 COc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3)[N+](=O)[O-] NRB03171 CCc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] NRB03179 CCOC(=O)CSC(=S)NC(C)c1ccccc1 RDR02156 CCOC(=O)CSC(=S)Nc1ccccc1OC RDR02157 Cc1cc(c(c(=O)o1)C(=O)C)O RJC00983 C#CCSc1c(c(cc(n1)c2cccs2)C(F)(F)F)C#N RF00200 C[C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)N RJC02199 CCOC(=O)C1=C(NC(=O)NC1c2cccs2)C RF00280 c1cc(sc1)c2cc(c3c(c(sc3n2)C(=O)c4ccc(cc4)Cl)N)C(F)(F)F RF00203 CC(=O)c1c(c2c(cc(nc2s1)c3cccs3)C(F)(F)F)N RF00208 c1cc(ccc1NC(=N)NC(=N)N)Br.Cl RDR02131 CCc1ccc(cc1)n2c(nnn2)/C=C/N(C)C NRB03208 COc1ccc(cc1)n2c(nnn2)/C=C/N3CCCC3 NRB03209 CC(C)(C)OCC(C(=O)ON1C(=O)CCC1=O)NC(=O)OCc2ccccc2 RJC02196 Cc1ccc(cc1)NC(=S)NNC(=O)c2ccco2 RJC02198 Cc1nc(c(c(n1)SC)C#N)n2cccc2 RF03721 CC(=O)OC[C@H]([C@H]([C@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C NRB04556 c1ccc(c(c1)C(=O)O)Nc2cccc(c2)C(F)(F)F RJC02179 Cc1cc2c(cccc2nn1)N RJC02157 c1ccc(cc1)c2ccc(cc2)n3c(nnn3)/C=C/N4CCCCC4 NRB03217 c1cc(ccc1Cc2ccncc2)[N+](=O)[O-] RJC02189 COC(=O)c1ccccc1/N=N/Nc2ccc(cc2)Br RB00235 c1ccc2c(c1)c(=O)n(nn2)c3ccc(cc3)Br RB00242 c1cc(c(cc1[N+](=O)[O-])Cl)Oc2ccc(cc2Cl)Cl RF04046 Cc1cc(c(cc1C)N2C(=O)C(=C(C2=O)C)C)C RB00298 CCSC([C@H]([C@H]([C@@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)SCC NRB04509 c1cc(ccc1c2nc(nc(n2)N)N)Cl RDR02035 Cc1cc(nc(n1)N)Sc2ccccn2 RDR02039 c1cc(ccc1N/C(=N/C(=N)N)/N)Cl NRB04514 Cc1cc-2c(nn1)CCc3c2non3 RJC02160 c1cc(ccc1n2c(nnn2)/C=C/N3CCCCCC3)F NRB03220 C=CCN(CC=C)C(=S)NC(=O)c1ccccc1 RB00193 COC(=O)/C=C/1\C(=O)C=C(O1)c2ccc(cc2)Cl RJC00993 COc1ccc(cc1)C2=CC(=O)/C(=C\C(=O)OC)/O2 RJC00994 c1ccc(cc1)C(=O)NC(=S)N2CCCCC2 RB00210 CSc1c(c(nc(n1)c2ccccn2)N)C#N RF04036 CSc1c(c(nc(n1)c2ccncc2)N)C#N RF04038 c1ccnc(c1)S/C=C/C(=O)c2ccc(cc2)Br NRB04632 c1ccc(cc1)C(C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N RF00291 CC1(N=C(N=C(N1c2ccccc2C(F)(F)F)N)N)C.Cl RB00302 c1cc(ccc1NC(=O)/C=C/C(=O)O)Oc2ccc(cc2)Cl RB00149 c1ccc(cc1)c2cc-3c(nn2)CCc4c3non4 RJC02161 CN(C)/C(=N/c1ccc(cc1)Cl)/SC.I RDR01989 CN(C)/C(=N/c1ccc(cc1)F)/SC.I RDR01993 C/N=C(/Nc1ccccc1OC)\SC.I RDR01994 CC(C)c1ccc(cc1)N2Cc3cc(ccc3N=C2)C(C)C RB00030 Cc1cc(cnn1)c2ccccc2 RJC02162 CS/C(=N\C#N)/S/C=C/C(=O)c1ccc(cc1)Br NRB03189 COc1cc2ccc(=O)oc2cc1OC NRB03190 c1cc(ccc1C(=O)CC(C(=O)O)Sc2ccc(cn2)C(F)(F)F)Br NRB04689 c1ccc(c(c1)Nc2nnc(s2)S)Cl RB00135 CCOc1ccccc1Nc2nnc(s2)S RB00136 c1ccnc(c1)SCC(=O)Nc2cccc(c2Cl)Cl RF00175 c1cc(c(c(c1)Cl)Cl)NC(=O)CSc2ccc(cc2)Cl RF00177 c1c(ccc(c1)NC(=O)/C=C/C(=O)O)Cc2ccc(cc2)NC(=O)/C=C/C(=O)O RB00152 c1ccc2c(c1)C(=O)N(C2=O)CC34CC5CC(C3)CC(C5)C4 RJC00953 c1cc(c(cc1NC(=O)C(Cl)(Cl)Cl)Cl)Br RDR02032 c1ccc(cc1)c2ccc(cc2)n3c(nnn3)C/C=N/Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-] NRB03185 Cc1ccc(cc1)C(=O)/C=C/S/C(=N/C#N)/SC NRB03186 Cc1cc\2c(nn1)CCC/C2=N/O RJC02152 CC(C)(C(=O)c1ccccc1)NO.Cl RJC02155 Cc1cc(nc(n1)SC(=O)OC(C)(C)C)C RJC02187 Cc1ccc(c(c1)C)Nc2nnc(s2)S RB00137 Cc1cc(nc2c1c(c(s2)C(=O)Nc3cc(ccc3Cl)C(F)(F)F)N)C RF00163 CC(=O)N1[C@@H](CSC1[C@H]([C@@H]([C@@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)C(=O)OC RJC02188 c1ccc(cc1)C(=O)NC(=S)NNC(=O)c2ccco2 RJC02191 c1cncc(c1C(F)(F)F)NC(=O)NC2CCCCC2 RF03996 c1cncc(c1C(F)(F)F)NC(=O)Nc2cc(cc(c2)Cl)Cl RF03998 c1cc(c(cc1F)F)CNC(=O)Nc2cnccc2C(F)(F)F RF03999 Cc1c(c(on1)/C=C/c2c(cn(n2)C)Cl)[N+](=O)[O-] RF04102 c1cncc(c1C(F)(F)F)C(=O)NN RF04050 COc1ccc(c(c1)OC)C2=NN(C(C2)c3ccccc3)c4ccccc4 RJC02125 c1ccc(cc1)C2=NN(C(C2)c3cccc(c3)O)c4ccccc4 RJC02129 c1ccc(cc1)/C=N/NC(=S)Nc2ccccc2 NRB04585 Cc1cccc(c1C)NC(=O)C(c2ccccc2)Sc3c(c(cc(n3)C)C)C#N RF00244 c1ccc(cc1)C(=O)NC(=S)NCc2ccncc2 RB00195 c1cc(ccc1n2c(nnn2)/C=C/N3CCCC3)F NRB03210 c1ccc(cc1)c2ccc-3c(n2)CCc4c3cccc4 NRB03206 c1ccc(cc1)C(C(=O)Nc2ccc(cc2)F)Sc3ccc(cc3)Cl RF00250 CCc1cccc(c1NC(=O)C(c2ccccc2)Sc3ccc(cc3)Cl)CC RF00253 CSc1c(c(nc(n1)c2ccc(cc2)Cl)N)C#N RF04041 CC1=C(C(=O)N(C1=O)c2ccc(cc2)Cl)C RB00216 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=S)N(C2=O)c3ccccc3)c4ccccc4 RJC02266 Cc1c(cc(nc1c2ccccc2)c3ccc(cc3)OC)c4ccccc4 NRB03277 Cc1c(cc(nc1c2ccccc2)c3ccc(cc3)Br)c4ccccc4 NRB03285 c1ccnc(c1)/C=C(\C#N)/C(=O)N RB00244 CC(C)c1ccc(cc1)C(CC(=O)c2ccc(cc2)OC)Sc3ccccc3 RB00266 c1ccc(cc1)/C(=C/C(=C/2\C(=O)N=C(S2)N3CCOCC3)/c4ccc(cc4)Cl)/CC(=O)c5ccc(cc5)Cl NRB03291 Cc1c(cc(nc1c2ccccc2)c3ccccc3)c4ccccc4 NRB03294 c1ccc(c(c1)N/C=C\C2=NN=NC2c3ccc(cc3)Br)Cl NRB03295 c1cc(ccc1c2nc(cs2)NC(=O)Nc3ccc(cc3)Cl)C(F)(F)F RF04287 c1cc(cnc1)NC(=O)Nc2csc(n2)c3ccc(cc3)C(F)(F)F RF04289 Cc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccc(c(c3)Cl)F NRB03297 CCc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccc(c(c3)Cl)F NRB03298 c1cc(ccc1/N=N/N2CCOCC2)[N+](=O)[O-] RF00306 CCOC(=O)c1cc(cnc1)Br RDP00009 c1c(cc(cc1C(F)(F)F)n2c(c(nn2)C#N)N)C(F)(F)F RF00382 c1cc(oc1)CNC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02198 COc1ccc(c(c1)C(=O)Nc2c(cccc2F)F)Br RF00414 c1cc(ccc1C#N)OC(=O)c2ccc(cc2)[N+](=O)[O-] RDR02078 c1ccc(cc1)CCNc2ccc(cc2C(=O)O)[N+](=O)[O-] RDR02087 c1cc(c(cc1SCSc2ccc(c(c2)Cl)Cl)Cl)Cl RJC01110 c1cc(ccc1c2[nH]nnn2)Cl RJC01112 Cc1ccc2cc(ccc2n1)Cl RJC01119 Cn1cc(c(n1)c2nc(cs2)c3ccc(cc3)Cl)Cl RF04201 c1cnc(nc1)SCc2nc(on2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RF04229 c1ccc(cc1)C(C(=O)Nc2cc(ccc2Cl)C(F)(F)F)Sc3ccc(cc3)Cl RF00251 c1ccc(cc1)C(C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Sc3ccc(cc3)Cl RF00252 c1cc(c(cc1c2nc(no2)c3cnccc3C(F)(F)F)Cl)Cl RF04160 c1cc(c(cc1Cl)Cl)c2nc(no2)c3cnccc3C(F)(F)F RF04165 c1cncc(c1C(F)(F)F)c2nc(on2)c3cc(cc(c3)Cl)Cl RF04166 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)N[C@@H](Cc2ccccc2)C(=O)O RJC02220 C1(C(=O)NC(=O)NC1=O)[N+](=O)[O-] RDP00108 COC(=O)c1cc(cnc1)Br RF04619 Cc1cc2c(cc1C)nsn2 RDP00075 c1cc(sc1)c2nc(no2)COC(=O)Nc3ccc(cc3)Cl RF04234 c1ccc(cc1)c2cc(nc(c2)c3ccc(cc3)Br)c4ccc(cc4)Br NRB03273 Cc1ccc(cc1)c2c(c(cc(n2)c3ccccc3)c4ccccc4)C NRB03274 CC(C)(C)C(=O)OC/C(=N/OC(=O)c1cccs1)/N RF04216 c1ccc(cc1)n2c(c(cn2)c3nnnn3c4ccccc4)C(F)(F)F NRB04659 Cc1ccnc(n1)S/C=C/C(=O)c2ccc(cc2)Cl NRB04644 Cc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2)C(F)(F)F NRB04645 c1cncc(c1C(F)(F)F)/C(=N/O)/N RF04149 c1ccc(cc1)N/N=C(\C#N)/C(=S)N RJC01056 Cc1cccc(c1NC(=O)C(C)Oc2ccc(cc2Cl)Cl)C RDR02207 c1cc2c(cc1COC(=O)OCc3ccc4c(c3)OCO4)OCO2 RF00389 CC(C)(C)OC(=O)CC[C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)N RJC02214 COc1cc(cc(c1)OC)COC(=O)N[C@@H](Cc2c[nH]c3c2cccc3)C(=O)O.C1CCC(CC1)NC2CCCCC2 RJC02225 CC(C)[C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)NC2CCCCC2 RJC02227 C1CS(=O)(=O)CC1S(=O)(=O)N2CCOCC2 RJC02232 c1ccc(cc1)Cn2c(c(nn2)C(=O)O)C(=O)O RJC01070 Cc1cc(c(c(c1)C)NC(=O)c2ccc(cc2[N+](=O)[O-])Cl)C RDR02189 Cc1ccc(c(c1)C)NC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02190 Cc1ccnc(n1)S/C=C/C(=O)c2ccc(cc2)OC NRB04643 Cc1cccc(c1C)NC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02192 c1cc(c(cc1Cl)[N+](=O)[O-])C(=O)Oc2ccc(cc2Cl)Cl RDR02195 c1cc(ccc1C#N)OC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02196 Cc1ccc(c(c1)[N+](=O)[O-])OS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl RDR02241 c1cc(c(c(c1)Cl)SCSc2c(cccc2Cl)Cl)Cl RJC01080 Cn1c(nnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)C(F)(F)F NRB04680 CC(C)C[C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)N RJC02217 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)N[C@@H](CCCCNC(=O)OCc2ccccc2)C(=O)O RJC02218 c1cc(ccc1c2nc(no2)c3cnccc3C(F)(F)F)F RF04169 Cn1cc(c(n1)/C(=N/OC(=O)c2ccccc2C(F)(F)F)/N)Cl RF04176 Cc1ccc(cc1)C(=O)C/C(=C\C(=C\2/C(=O)N=C(S2)N3CCOCC3)\c4ccc(cc4)C)/c5ccccc5 NRB03255 CN(C[C@H]([C@@H]([C@H]([C@H](CO)O)O)O)O)C=C(C#N)C#N RJC02205 C1C2C(S2)CS1(=O)=O RJC02228 c1ccc(cc1)CNS(=O)(=O)C2CCS(=O)(=O)C2 RJC02235 CC(C)(C)OC(=O)C[C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)N RJC02210 c1ccc(cc1)c2c(n3ccccc3n2)Sc4ccc(cc4)[N+](=O)[O-] RJC02248 CCOC(=O)c1ccc(cc1)OCc2ccc(cc2)[N+](=O)[O-] RDR02201 Cc1c(c(nc(n1)SCC=C)O)CC=C RDR02203 Cc1ncc(c(n1)C(F)(F)F)c2nnnn2c3ccccc3 NRB04667 c1ccc(cc1)/C=C/2\C(=O)Nc3ccccc3S2 RB00331 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)Nc3ccccc3S2 RB00332 COC(=O)c1ccccc1NC(=S)Sc2ccc(cc2)Cl RF00625 CCOC(=O)C1=C(NC(=O)NC1c2ccc(o2)c3ccc(cc3)[N+](=O)[O-])C RF00627 CCOC(=O)C1=C(NC(=O)NC1c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C RF00628 Cc1ccc(cc1)N/C=C\c2nnnn2c3ccc(cc3)F NRB03310 Cc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)C)c4ccccc4 NRB03271 Cc1ccc(cc1)n2c(nc3c2ccc(c3)[N+](=O)[O-])C NRB04700 CCC(C)[C@@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)N RJC02216 c1cc(ccc1c2nc(no2)c3cnccc3C(F)(F)F)Cl RF04159 c1ccc(c(c1)c2nc(no2)c3cnccc3C(F)(F)F)F RF04168 CC(C(=O)Oc1ccc(cc1Cl)Cl)Oc2ccc(cc2Cl)Cl RDR02212 CCOC(=O)CSC(=S)Nc1ccc(cc1C)C RDR02163 Cc1cccc(c1NC(=O)c2ccc(cc2[N+](=O)[O-])Cl)C RDR02191 Cc1ccc(c(c1)C)NC(=S)NC(C)(C)C#C RDR02217 CCOC(=O)c1ccc(cc1)OC(=O)c2ccc(c(c2)Cl)Cl RDR02229 c1ccc2c(c1)cc-3oc(ccc23)c4ccc(cc4)Cl NRB04670 c1ccc2c(c1)NC(=O)/C(=C\c3ccc(cc3)Cl)/S2 RB00334 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)C(F)(F)F)F NRB04647 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)C(F)(F)F)Cl NRB04648 c1ccc(cc1)c2ncc(c(n2)C(F)(F)F)c3nnnn3c4ccccc4 NRB04678 Cc1ccc(c(c1)NC(=O)CSc2nnc(n2C)C(F)(F)F)OC NRB04679 Cc1ccc(cc1)C(=O)/C=C/OC(=O)c2ccc(cc2)Cl NRB04649 c1ccc(cc1)n2c(nnn2)c3cn[nH]c3C(F)(F)F NRB04658 Cc1ccc(cc1C#N)NC(=O)CSc2ccc(cn2)C(F)(F)F NRB04684 C1CCN(CC1)S(=O)(=O)C2CCS(=O)(=O)C2 RJC02233 Cc1c(c(c(nc1C)S)C#N)C RF00378 C1C(C(CS1(=O)=O)SC(=N)N)O.Cl RJC02236 Cc1ccc(cc1)C(=O)N(c2ccccc2)C(C)C3CC3 RJC02254 Cc1ccc(c(c1)[N+](=O)[O-])OC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02197 Cc1ccc(c(c1)C)NC(=O)C(C)(C)C RDR02200 c1cc(ccc1[N+](=O)[O-])OS(=O)(=O)c2ccc(cc2Cl)Cl RDR02234 Cc1ccc(c(c1)[N+](=O)[O-])OS(=O)(=O)c2ccc(cc2Cl)Cl RDR02240 CCOC(=O)c1ccc(cc1)OC(=O)c2ccc(cc2Cl)Cl RDR02230 Cc1cc(c(c(c1)C)NC(=O)C(C)Oc2ccc(cc2Cl)Cl)C RDR02205 Cc1cc(ccc1NC(=O)C(C)Oc2ccc(cc2Cl)Cl)Cl RDR02208 Cc1cccc(c1Nc2nnc(s2)C(F)(F)F)C RDR02249 CCOC(=O)c1ccc(c(c1)Cl)OC(=O)c2ccc(c(c2)Cl)Cl RDR02237 CCOC(=O)c1ccc(c(c1)Cl)OC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02238 CC(C(=O)Nc1ccc(cc1)Br)Oc2ccc(cc2Cl)Cl RDR02147 c1ccc(cc1)C(C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Sc3ccccn3 RF00256 COc1ccc(cc1OC)CCNC(=O)C(c2ccccc2)Sc3ccccc3N RF00261 CC(C)(C)CC(C)(C)NC(=O)C(c1ccccc1)Sc2ccccc2N RF00263 CC(C)S/C(=N\C#N)/S/C=C/C(=O)c1ccc(cc1)Cl NRB03264 COc1ccc(cc1)c2cc(nc(c2)c3ccccc3)c4ccccc4 NRB03266 COC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F RF04568 c1ccc2c(c1)NC(=O)/C(=C/c3ccc4c(c3)OCO4)/S2 RB00335 Cc1cc(nc(n1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C RF00392 Cc1ccc(cc1)C(=O)C/C(=C\C(=C\2/C(=O)NC(=S)S2)\c3ccc(cc3)C)/c4ccccc4 NRB03249 c1ccc(cc1)c2nc(no2)c3cnccc3C(F)(F)F RF04154 c1ccc(cc1)CC(=O)c2ccc(cc2)Br RJC01073 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2O)OC)C RF00290 COc1cc(cc(c1OC)OC)/C=C/[N+](=O)[O-] RB00156 c1ccc(cc1)n2c(nnn2)c3cnc(nc3c4ccc(cc4)Cl)c5cccnc5 NRB04665 COc1ccc(cc1)NC(=O)c2cc(ccc2Br)OC RF00418 C1[C@H]([C@@H]([C@@H](C=C1C(=O)O)O)O)O RJC01089 Cc1ccc(cc1)c2cc(nc(c2C)c3ccccc3)c4ccccc4 NRB03275 Cc1ccc(cc1)c2cc(c(c(n2)c3ccccc3)C)c4ccccc4 NRB03276 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)N[C@@H](CCSC)C(=O)O.C1CCC(CC1)N RJC02219 COc1ccc(c(c1)/C=C\2/C(=O)Nc3ccccc3S2)OC RB00336 c1cc(ccc1C#N)c2ccc(cc2)C#N RJC01092 Cc1c(cc(nc1c2ccc(cc2)Br)c3ccccc3)c4ccccc4 NRB03283 Cc1c(cc(nc1c2ccccc2)c3ccccc3)c4ccc(cc4)Br NRB03284 c1cc(ccc1n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Br NRB03183 C1C(C1C(=O)NN)C(=O)NN RJC02180 COc1ccc(cc1)n2c(nnn2)/C=C/N3CCCCC3 NRB03214 c1cc(ccc1n2c(nnn2)/C=C/N3CCCCC3)Cl NRB03216 c1ccc(c(c1)CNC(=O)c2cnccc2C(F)(F)F)Cl RF04003 CC(C(=O)Nc1ccc(cc1)OC)Oc2ccc(cc2Cl)Cl RDR02210 CC(C(=O)Nc1ccc(cc1Cl)Cl)Oc2ccc(cc2Cl)Cl RDR02211 c1ccc(c(c1)SCSc2ccccc2Cl)Cl RJC01076 c1cc(cc(c1)Cl)S(=O)(=O)CS(=O)(=O)c2cccc(c2)Cl RJC01077 c1ccc(c(c1)S(=O)(=O)CS(=O)(=O)c2ccccc2Cl)Cl RJC01078 CCN(CC)c1ccc(cc1)C2C(=C(NC(=O)N2)C)C(=O)OCC RJC02265 Cc1c(cc(nc1c2ccccc2)c3ccc(cc3)F)c4ccccc4 NRB03279 CC(C)NCC(COc1ccccc1CC=C)O.Cl RJC02271 Cc1ccc(cc1)c2nc(c(c(n2)SC)C#N)N RF04040 CSc1c(c(nc(n1)c2ccc(cc2)C(F)(F)F)N)C#N RF04042 c1ccc(cc1)C2=NNC(=S)SC2 NRB04606 Cc1cc(c(c(c1)C)N2C(=NC(=NC2(C)C)N)N)C.Cl RB00304 CC12C3C4CC5C3C1C(=O)C5C4C2=O RJC02257 c1ccc(cc1)c2nnc(o2)c3ccc(cc3)Br RJC01085 CC(C)NC(=O)Nc1csc(n1)c2ccc(cc2)C(F)(F)F RF04291 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)[N+](=O)[O-])C RJC02261 c1ccc(cc1)CCn2c3ccc(cc3c(cc2=O)O)[N+](=O)[O-] RDR02253 c1ccc(c(c1)c2[nH]nnn2)Br RJC01091 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])/N=N/N2CCOCC2 RF00307 CCOC(=O)C1=C(NC(=O)NC1c2coc3ccccc3c2=O)C RF00321 c1ccc2c(c1)NC(=O)/C(=C\c3cccs3)/S2 RB00337 c1ccc(cc1)n2cnc3c2ccc(c3)[N+](=O)[O-] NRB04702 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)Cl)C RJC02262 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)OC)C RJC02263 CCCCc1c(c2ccccc2o1)C(=O)c3cc(c(c(c3)I)OCCN(CC)CC)I.Cl RJC02270 CC(C)(C)C(=O)Nc1cccc(c1Cl)Cl RDP00115 Cc1ccc(cc1)c2cc(nc(c2)c3ccccc3)c4ccccc4 NRB03265 c1ccc(cc1)c2cc(cc(n2)c3ccccc3)c4ccc(cc4)Cl NRB03267 COc1ccc(c(c1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br RF00412 CCO/C(=C/1\C(=O)NC(=S)S1)/C RB00180 c1ccnc(c1)SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F RF00179 c1ccc(c(c1)N)SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F RF00180 c1cc(ccc1SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F)Cl RF00181 c1cc(c(cc1C(F)(F)F)/N=N/N2CCOCC2)Cl RF00187 c1cc(ccc1CNC(=O)c2cnccc2C(F)(F)F)Cl RF04004 Cc1c2c(n[nH]c2nc(c1[N+](=O)[O-])C)N RF00431 Cc1ccc(cc1)C(=O)/C=C/Sc2nccc(n2)C NRB04642 COC(=O)COC(=O)c1ccccc1[N+](=O)[O-] RJC02317 c1ccc(cc1)CNCC(c2ccc(cc2)[N+](=O)[O-])O RJC02318 Cn1cc(c(n1)/C=C(\C#N)/C(=O)c2ccco2)Cl RF04097 Cn1cc(c(n1)/C=C(\C#N)/C(=O)N)Cl RF04099 Cc1c(c(on1)/C=C/c2ccn[nH]2)[N+](=O)[O-] RF04106 CC(C)(C)C(=O)OC/C(=N/OC(=O)c1ccc(cc1)Cl)/N RF04197 Cc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)Br NRB03328 c1cc2c(cc1F)nsn2 RDP00058 COc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)Br NRB03329 c1cc(c(cc1c2nn(c(=O)o2)c3ccc(cn3)C(F)(F)F)Cl)Cl RF04851 COC(=O)c1ccc2c(c1)nccn2 RDP00059 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NS(=O)(=O)c3ccc(cc3)C)C(=O)OC RDP00060 COc1ccc2c(c1)nsn2 RDP00061 c1ccc(cc1)N2CCN(C2Cc3nnnn3c4ccc(cc4)Cl)c5ccccc5 NRB03338 c1ccc(cc1)/C(=C/C(=C/2\C(=O)N=C(S2)N3CCOCC3)/c4ccccc4)/CC(=O)c5ccccc5 NRB03288 c1ccc(cc1)NC(=O)Nc2csc(n2)c3ccc(cc3)C(F)(F)F RF04286 Cc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)OC NRB03318 CCCCCCCCCCCCSC(=S)Nc1cc(ccc1Cl)Cl RF00588 c1cc(ccc1N/C=C/c2nnnn2c3ccc(cc3)Br)Cl NRB03327 COc1ccc(cc1)N/C=C\c2nnnn2c3ccc(cc3)OC NRB03319 CCOC(=O)Cn1c2c(nc1NCCc3ccccc3)n(c(=O)n(c2=O)C)C RJC01278 c1ccc2c(c1)c(=O)c3cc(ccc3s2)C(F)(F)F RJC01285 COc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccccc3OC NRB03314 COc1ccccc1N/C=C/c2nnnn2c3ccc(cc3)Br NRB03317 COc1ccc(cc1)N/C=C\c2nnnn2c3ccc(cc3)F NRB03320 CC(C)(C(=O)O)ONC(=O)Nc1ccccc1Cl RF04677 CCOC(=O)c1ccc(cc1)NC(=O)CCC(=O)O RDP00030 c1ccc(cc1)/C(=C/C(=O)c2ccccc2)/CC(=O)c3ccccc3 NRB03351 Cn1/c(=N\C(=N\C#N)\SC)/nc(n1C)SC RDP00087 CCOC(=O)[C@H](CCSC)N.Cl RDP00088 COc1ccccc1C(=O)c2ccccc2 RDP00089 c1cc2c(cc1C(F)(F)F)nsn2 RDP00073 CC(C)C1(C(=O)N=C2N1C(=O)c3c2cccc3)C RJC02309 COC(=O)c1ccc2c(c1)nn[nH]2 RDP00072 Cc1cc(c(c(c1)C)NC(=S)NC(=O)c2cc(ccc2Br)OC)C RDR02331 c1ccc(cc1)COc2cccc(c2C#N)Cl RJC01108 CC(C)(C)C(=O)CS(=O)(=O)c1ccc(cc1)Cl RJC01109 Cc1cc(nc2c1c(c(s2)C#N)N)C RF00546 COc1ccc(cc1)NC(=O)Cc2ccc(cc2)[N+](=O)[O-] RF00480 c1ccc2c(c1)N/C(=C(/C#N)\C(=O)c3ccco3)/S2 RJC02246 c1ccc(cc1)N(c2ccc(cc2)F)C(=O)C34CC5CC(C3)CC(C5)C4 RJC02247 Cc1cc(ccc1NC(=O)C(C)Oc2ccc(cc2)I)Br RDR02317 Cc1cc(ccc1NC(=O)C(C)Oc2ccc(cc2)C(C)(C)C)Br RDR02318 CCOC(=O)C1=C(NC(=CC1=C(C#N)C#N)C)C RJC02313 CCOC(=O)/C(=N/Nc1ccccc1Cl)/C(=O)C RJC02321 Cc1ccc(cc1)c2cc(c3c(n2)-c4ccccc4CCC3)c5ccccc5 NRB03350 CC(=O)O/N=C/c1c(cn(n1)C(=O)NC)Br RF04852 COC(=O)c1ccc(cc1)CN.Cl RJC02323 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNc3ccccc3 RF00562 c1ccc2c(c1)c(=O)c(c3n2c4ccccc4[nH]3)C#N RJC02304 COc1ccc(c(c1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl)Br RF00582 CCOC(=O)Cc1csc(n1)N/N=C/c2ccc(cc2)Cl RF00583 CCCCCCCCCCCCSC(=S)Nc1ccc(c(c1)C)Br RF00587 c1cc(ccc1N/C=C\c2nnnn2c3ccc(cc3)F)Br NRB03330 Cc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)OC)c4ccccc4 NRB03344 COCCOc1ccc(cc1C(=O)O)/N=C/c2ccccc2O RDR02340 C1CCC(CC1)Nc2c(c(=O)c2=O)NC3CCCCC3 RDP00145 CC(C)C(=O)NNc1c(cc(cn1)C(F)(F)F)Cl RF04805 CCOC(=O)NNc1c(cc(cn1)C(F)(F)F)Cl RF04806 c1cc(c(c(c1)F)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)F RF04808 Cc1cc(c(c(c1)C)NC(=O)C(C)Oc2ccc(cc2)C(C)(C)C)C RDR02319 c1ccc(cc1)/C(=C/2\CCCc3ccccc3C2=O)/CC(=O)c4ccccc4 NRB03370 COc1cccc(c1C(=O)NNc2ccc(cn2)C(F)(F)F)OC RF04812 CC(=O)n1cc(c(n1)/C=N/OC(=O)NC)Br RF04823 COc1ccccc1n2c(=O)c3ccccc3nc2SCC#C RDR02338 COc1ccc(cc1)n2c(=O)c3ccccc3nc2SCC=C RDR02339 CC1(C2CCC1(C(C2)N)C)C.Cl RDP00128 c1ccc2c(c1)c(=O)n(c(n2)S)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RDR02334 COc1ccc(cc1)/C(=C/C(=O)c2ccccc2)/CC(=O)c3ccccc3 NRB03362 c1ccc(cc1)/C(=C/2\Cc3ccccc3C2=O)/CC(=O)c4ccccc4 NRB03366 c1cc2c(cc1C(=O)NN)nsn2 RDP00096 c1ccc2cnc(cc2c1)C(C#N)c3ccc4c(c3[N+](=O)[O-])C(=O)c5ccccc5C4=O RJC02308 c1cc(c(nc1)OCC(F)(F)F)C(=O)N RF04864 c1cc(c(nc1)OCC(F)(F)F)C(=O)Nc2ccc(cc2)Cl RF04879 CC(=O)Nc1cc(cc(c1)C(=O)O)C(=O)O RJC02327 CC1=CC(NC(=S)N1)(C)C NRB04774 Cn1c2ccccc2c(cc1=O)OC(=O)N(C)C NRB04777 c1cc(ccc1c2ccc(o2)/C=N/O)S(=O)(=O)N RDR02359 C1CNc2c(c(=O)c2=O)NC1 RDP00155 CN1C2CCCCC2(C(=O)CC1c3ccccc3)O RJC01143 COc1cccc(c1C(=O)NNC(=S)N)OC RF00516 COc1ccc(c(c1)c2[nH]c(nn2)SCC(=O)c3ccc(cc3)Cl)Br RF00519 CC1(O[C@H]([C@H](O1)C(=O)c2ccccc2)c3cccc(c3)[N+](=O)[O-])C RJC01161 CC(C)(C)C(=O)Nc1ccc(cc1)S(=O)(=O)N RDR02322 CC(c1ccccc1)NC(=O)Cc2ccc(cc2)[N+](=O)[O-] RF00523 CC(C)(C)C(=O)n1cc(c(n1)/C=N/OC(=O)NC)Br RF04828 c1ccc(cc1)/C(=C/C(=O)c2ccc(cc2)Br)/CC(=O)c3ccc(cc3)Br NRB03355 Cc1ccc(cc1)C(=O)/C=C(\CC(=O)c2ccc(cc2)Cl)/c3ccccc3 NRB03360 COc1ccc(cc1)C(=O)/C=C(\CC(=O)c2ccc(cc2)Cl)/c3ccccc3 NRB03361 c1ccc(cc1)CNc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] NRB04731 CC(C(=O)Nc1ccc(cc1)S(=O)(=O)N)Oc2ccc(cc2)C(C)(C)C RDR02354 CC(C(=O)Nc1ccc(cc1)S(=O)(=O)N)Oc2ccc(cc2)I RDR02355 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNc3cc(ccc3Cl)Cl RF00552 Cc1c(c(no1)c2c(cccc2Cl)Cl)CO RF00619 Cc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)[N+](=O)[O-])c4ccccc4 NRB03346 c1ccc(cc1)c2cc(nc(c2)c3ccc(cc3)F)c4ccccc4 NRB03348 CCOc1c(c(=O)c1=O)Nc2ccc(cc2)C(=O)OCC RDP00149 CN1CCN(c2c1c(=O)c2=O)C RDP00150 CCCCCCCCCCCCSC(=S)Nc1cccc(c1C)Cl RF00591 CCCCCCCCCCCCSC(=S)Nc1cccc(c1)SC RF00593 CCCCCCCCCCCCSC(=S)NCC1CCCO1 RF00596 c1cc(ccc1SC(=S)NC2CCCCC2)Cl RF00605 c1ccc(cc1)CNc2c(c(=O)c2=O)NCc3ccccc3 RDP00132 CCCNc1c(c(=O)c1=O)NCCC RDP00134 c1ccc(cc1)[C@H]2[C@@H](C2(Cl)Cl)c3ccccc3 RJC01159 CC1(O[C@H]([C@H](O1)C(=O)c2ccc(cc2)OC)c3ccc(cc3)[N+](=O)[O-])C RJC01163 CCOC(=O)/C(=N/Nc1cccc(c1)C)/C(=O)C RJC02320 c1ccc(cc1)S(=O)(=O)C(CCC(=O)O)(CCC(=O)O)C#N RJC02324 CN(c1ccc(c(c1)Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)Oc3ccc(cc3)Cl RF04760 CN(c1ccc(c(c1)Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04773 CCCCCCCCCCCCCCCc1c\2c(on1)CCC/C2=N/O RJC01199 CCc1cccc(c1NC(=O)CSc2ccc(cc2)Cl)CC RF00336 Cc1ccccc1N/C=C\c2nnnn2c3ccc(cc3)OC NRB03304 CC(C)C(CCCN(C)CCc1ccc(c(c1)OC)OC)(C#N)c2ccc(c(c2)OC)OC.Cl RJC01232 CCOC(=O)Cc1csc(n1)NN=C(C)C.Cl RF00711 c1ccc(cc1)C(=O)NCc2nnc3n2cc(cc3Cl)C(F)(F)F RF04853 c1c(cncc1Br)C(=O)N RDP00037 C=CCS/C(=N\C#N)/S/C=C/C(=O)c1ccc(cc1)Br NRB03262 c1cc(ccc1c2nc(cs2)NC(=O)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F RF04288 c1ccc2c(c1)NC(=O)CS2 RB00326 c1cc(c(cc1C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl)Cl RF04802 CC(C)C(=O)NNc1ccc(cn1)C(F)(F)F RF04825 CCCc1c(nc(nc1O)SCc2ccc(cc2)Cl)C RDR02301 c1cc(cc(c1)C(F)(F)F)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl RF04833 CC(C(=O)Nc1ccc(cc1)Br)Oc2ccc(cc2)C(C)(C)C RDR02315 Cc1cc(nc(n1)c2ccncc2)O RDR02269 c1cc(ncc1C(F)(F)F)S RF04700 CC(=O)CSc1[nH]c(nn1)c2ccc(cc2)Cl RF00513 c1cc(ccc1n2c(nnn2)/C=C/Nc3ccc(c(c3)Cl)F)Br NRB03302 c1ccc(cc1)c2ccc(cc2)c3nnc(o3)c4ccc(cc4)c5ccccc5 RJC01083 c1ccc(cc1)n2c(nnn2)/C=C/Nc3ccc(c(c3)Cl)F NRB03296 c1ccc2c(c1)C(=O)c3ccc(c(c3C2=O)[N+](=O)[O-])C(=O)O RJC02296 COc1ccc(cc1)c2ccc(cc2C#N)OC RJC01103 c1ccc2c(c1)c(c3ccccc3n2)N NRB04719 CCNc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] NRB04730 CC(=O)CSc1[nH]c(nn1)c2ccccc2 RF00493 COc1cc(cc(c1OC)OC)C2CC(=NN2c3ccccc3)c4ccc(cc4)Cl RDR02307 CCOC(=O)/C(=C/c1ccccc1[N+](=O)[O-])/C#N RJC02283 CC(=O)C(C(=O)c1ccccc1[N+](=O)[O-])C(=O)OC RJC02284 COc1ccc(c(c1)C(=O)NNC(=S)N)Br RF00502 CSc1[nH]c(nn1)c2ccc(cc2)Cl RF00506 CCOc1ccc(cc1)C(=O)CC(C(=O)O)SCc2ccc(cc2)Cl NRB04683 C1=CC2C3C(C1O2)C(=O)N(C3=O)O RDP00003 c1ccc(cc1)CN2CCC(CC2)(C#N)O RJC01072 c1ccc(cc1)CNc2c3c([nH]cn3)ncn2 RJC01074 CC(C(=O)Nc1ccccc1OC)Oc2ccc(cc2Cl)Cl RDR02209 c1ccc(cc1)N2C(CC(=N2)c3ccccc3Cl)c4cc(cc(c4O)Cl)Cl RDR02304 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)Cl)c4ccc5c(c4)OCO5 RDR02305 c1cc(ccc1CC(=O)Nc2ccc3c(c2)OCO3)[N+](=O)[O-] RF00486 COc1ccccc1N/C=C\c2nnnn2c3ccc(cc3)Cl NRB03316 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)[N+](=O)[O-])c4ccco4 RDR02308 c1ccc(cc1)c2nc([nH]n2)SCC(=O)c3ccc(cc3)Cl RF00494 c1cc(ccc1C(=O)NNC(=S)N)Cl RF00497 COc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)Cl NRB03324 CN(C)CCCNC(=O)c1c(c(cc(c1OC)Cl)Cl)OC RF00635 c1ccc(cc1)c2c(n3ccccc3n2)S/N=C(/c4ccccc4)\C(F)(F)F RJC02250 Cc1ccc(cc1)Oc2c(c(c(c(c2F)F)Oc3ccc(cc3)C)F)F RJC02253 c1ccc(cc1)c2c(n3ccccc3n2)Sc4ccc(cc4)Cl RJC02249 C1CCC(CC1)N2C(=O)CCC2=O RDP00015 Cc1ccccc1N/C=C\c2nnnn2c3ccc(cc3)Cl NRB03306 Cc1ccccc1N/C=C\c2nnnn2c3ccc(cc3)Br NRB03307 CCOC(=O)C(c1ccccc1)N.Cl RDP00069 Cc1ccc2c(c1C)nsn2 RDP00105 c1ccc2c(c1)[nH]c(n2)C(C#N)C(=O)c3ccc(cc3Cl)Cl RJC02310 Cc1csc(n1)c2c3ccc(cc3c(=O)n(c2N)Cc4ccccc4)[N+](=O)[O-] RJC02312 CCCNC(=O)O/N=C(/c1c(onc1c2c(cccc2Cl)Cl)C)\N RF00806 c1cc(c(c(c1)Cl)NC(=O)c2ccc(cc2)F)Cl RJC02275 c1ccc(cc1)/C(=C/c2ccccc2[N+](=O)[O-])/C#N RJC02281 CC(=O)Nc1cccc(c1)C(F)(F)F RDP00039 CCOC(=O)c1ccc(cc1)N2C(=O)C=C(C2=O)C RDP00041 CCOC(=O)[C@H](Cc1c[nH]c2c1cccc2)N.Cl RDP00077 CC(C)c1ccc(cc1)/C=C\2/C(=O)Nc3ccccc3S2 RB00333 c1cc(c(cc1Cl)Cl)NC(=O)NC(=O)c2cnccc2C(F)(F)F RF04503 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])NC(=O)C RDP00018 CC(=O)N1CCc2c1c(cc(c2)Br)[N+](=O)[O-] RJC02274 c1cc(ccc1N/C=C\c2nnnn2c3ccc(cc3)F)Cl NRB03325 CCOC(=O)c1ccc(cc1)N2C(=O)CCC2=O RDP00033 c1cc(ccc1[N+](=O)[O-])Oc2ccc(cc2Cl)Cl RDP00053 c1c2c(cc(c1F)Cl)nsn2 RDP00065 c1ccc(cc1)c2nc3n(n2)c(cs3)c4ccc(cc4O)O RF00498 c1cc(ccc1CC(=O)NC2CCCCCCC2)[N+](=O)[O-] RF00524 c1cc(ccc1SCC(=O)O)Cl RF00560 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN3CCCCC3 RF00556 Cc1ccc(cc1)N/C=C\c2nnnn2c3ccc(cc3)OC NRB03309 c1ccc(cc1)N2CCN(C2Cc3nnnn3c4ccc(cc4)F)c5ccccc5 NRB03337 Cn1cc(c(n1)/C=N/Nc2ccc(cc2Cl)Cl)Br RF04137 CCCCCC#CC(=O)N=c1[nH]c2cc(c(cc2[nH]1)C)C RJC01132 COc1ccc(cc1OC)CCNC(=O)Cc2ccc(cc2)[N+](=O)[O-] RF00490 C=CCSc1[nH]c(nn1)c2ccccc2 RF00501 CC1=C(C(=O)OC1(C)CN(C)C)Cl RJC01147 c1cc(ccc1c2[nH]c(nn2)S)Cl RF00505 c1cc(ccc1N/C=C\c2nnnn2c3ccc(cc3)Cl)Br NRB03331 CC(=O)Nc1ccc(cc1NC(=O)C)C(=O)OC RDP00054 CCc1cccc(c1Nc2ncnc(n2)N)CC RDR02604 c1ccc2c(c1)ccc(c2I)OC(=O)c3ccc(c(c3)Cl)Cl RDR02606 c1cc(c(cc1Cl)Cl)n2c(=O)cc(c(n2)C(=O)O)O NRB04807 c1ccc(cc1)CS/C(=N\C#N)/S/C=C/C(=O)c2cccc(c2)Br NRB03486 Cc1c(oc(cc1=O)C(=O)O)C NRB04763 c1cc(c(cc1c2nn(c(=O)o2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl RF04803 Cc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)Cl)c4ccccc4 NRB03347 COc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)Cl)c4ccccc4 NRB03345 c1ccc(cc1)c2cc(nc-3c2CCCc4c3cccc4)c5ccccc5 NRB03349 CCC(=O)Oc1ccc(cc1)NC(=S)NCCCO RDR00003 Cc1c2ccc(cc2oc(=O)c1Cc3ccccc3)OS(=O)(=O)C RDR02427 Cc1ccc(cc1)C(=O)/C(=C(\CC(=O)c2ccccc2)/c3ccccc3)/C NRB03364 Cc1c(c(nc(c1[N+](=O)[O-])C)Sc2ccccc2)C#N RF00658 CCC(=O)Oc1ccc(cc1)NC(=S)Nc2c(cc(cc2C)C)C RDR00020 CC(=O)OCCCNc1[nH]c2c(n1)n(c(=O)n(c2=O)C)C RJC01281 Cc1c(c(nc(n1)S)O)Cc2cccc(c2)C(F)(F)F RDR02443 Cc1ccc(cc1)C(=O)C/C(=C\2/CCc3ccccc3C2=O)/c4ccccc4 NRB03369 Cc1ccc(cc1)Sc2cc(c(c(n2)Sc3ccc(cc3)C)C#N)C RF00667 CCCCc1c(c2ccc(cc2n(c1=O)CC)C)O NRB04784 Cc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)Cl NRB03323 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Nc2c(cc(cn2)C(F)(F)F)Cl RF04693 c1ccc(c(c1)/C=C(/C#N)\S(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl RF04733 c1ccc(cc1)Cc2c(c3cccc4c3n(c2=O)c5c4CCCC5)O NRB04795 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCCCO)CC(=O)NCCCO RJC01282 Cc1nnc(s1)Nc2ccc(cc2)Cl RDR02363 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F RDR02377 CCOC(=O)C(C)Oc1ccc(cc1Cl)NS(=O)(=O)c2cc(ccc2OC)OC RDR02467 COc1ccc(c(c1)NC(=O)C(Cl)Cl)OC RDR02473 c1cc(ccc1N)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F RDR02378 Cc1ccc2cccc(c2n1)Cl RJC01118 c1cc(ccc1CC(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] RF00479 c1ccc2c(c1)c3c([nH]2)CCCC3 RJC02362 c1cc(c(c(c1)n2ccnc2)C#N)n3ccnc3 RF00675 Cc1cc(c2c(c1)occ(c2=O)/C=C/3\C(=O)N(C(=S)S3)c4cccc(c4)Cl)C RF00683 CCCc1c(nc(nc1O)SCC#C)C RDR02380 CCOC(=O)C(C)Oc1ccc(c(c1)NC(=O)c2ccc(cc2[N+](=O)[O-])Cl)C RDR02382 CCOC(=O)[C@H](CCCNC(=N)N)NC(=O)c1ccccc1.Cl RDP00259 Cc1ccc(c(c1)C)NC(=S)Nc2ccccc2N RDR00005 c1ccc(c(c1)N)NC(=S)Nc2cccc(c2)C(F)(F)F RDR00008 c1ccc(cc1)c2[nH]c(nn2)S RF00489 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN(C)C RF00561 CN(C(=O)c1ccccc1)C(=O)N(C)C(=O)c2ccccc2 RF00696 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N(C)C(=O)N(C)C(=O)c3c(onc3c4c(cccc4Cl)F)C RF00698 Cc1cc(nc(c1C#N)OC)OC RF00652 COc1ccc(cc1)C(=O)C/C(=C\C(=O)c2ccccc2)/c3ccccc3 NRB03359 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=S)N RF00748 Cc1ccc(cc1)S(=O)(=O)O[C@@H]2CO[C@H]3[C@@H]2OCC3OS(=O)(=O)c4ccc(cc4)C NRB04852 Cc1c(c(nc(c1[N+](=O)[O-])C)Sc2cc(ccc2OC)OC)C#N RF00659 Cc1c(c(nc(c1[N+](=O)[O-])C)S(=O)(=O)c2ccccc2)C#N RF00662 c1cc(ccc1N/C=C\c2nnnn2c3ccc(cc3)Br)O NRB03427 Cc1ccc(c(c1)C)N2C(=O)/C(=C\c3coc4cc(cc(c4c3=O)C)C)/SC2=S RF00685 Cc1ccc(cc1)C(=O)C/C(=C\2/CCCc3ccccc3C2=O)/c4ccccc4 NRB03371 COc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)O NRB03435 CC(C)N(C(C)c1[nH]c(=O)c2ccccc2n1)C(=O)Nc3ccc(c(c3)Cl)Cl NRB03446 CC(C)Oc1c(c(=O)c1=O)N2CCOCC2 RDP00180 CCOc1c(c(=O)c1=O)N2CCOCC2 RDP00151 CCOC(=O)c1ccc2c(c1)Nc3c(c(=O)c3=O)N2 RDP00153 C1COCCN1c2c(c(=O)c2=O)N3CCOCC3 RDP00154 COc1ccc(c(c1)[N+](=O)[O-])N2CCCCC2 NRB03378 c1ccc(cc1)Nc2c(c(=O)c2=O)Nc3ccccc3 RDP00133 CCOc1c(c(=O)c1=O)NN(C)C RDP00135 COc1cc(ccc1N2CCCCC2)[N+](=O)[O-] NRB03388 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])OC NRB03389 c1ccc(cc1)C(=O)C/C(=C\C(=C/2\Cc3ccccc3C2=O)\c4ccccc4)/c5ccc(cc5)Br NRB03428 Cc1cc(ccc1N2CCCC2)[N+](=O)[O-] NRB03400 CC1(CC(=CC(=O)C1)/C=C/c2ccc(cc2)Br)C RJC01200 c1ccc(cc1)C(=O)/C=C/S/C=C/C(=O)c2ccccc2 NRB03475 COc1ccc(cc1)C(=O)/C=C/S/C=C/C(=O)c2ccc(cc2)OC NRB03477 c1cc(ccc1C(=O)CC(=O)C(=O)Nc2ccc(cn2)Br)Cl RJC01219 Cc1c(c(nc(c1[N+](=O)[O-])C)Sc2ccc(cc2)Br)C#N RF00660 CC1[C@@H]2[C@@]3(OC(C(O3)[C@@](O2)(O1)C)C)C RJC01176 Cc1[nH]n(c2c(c(=O)c2=O)n(n1)C)C RDP00169 c1cc2c(cc1F)Nc3c(c(=O)c3=O)N2 RDP00187 CC1C(C1(C(=O)c2ccccc2)C(=O)c3ccccc3)(C)C RJC01186 CCOc1c(c(=O)c1=O)N2CCN(CC2)c3c(=O)c(=O)c3OCC RDP00192 CCOc1c(c(=O)c1=O)N2CCCC2 RDP00194 c1c(cc(c2c1nsn2)Cl)C(F)(F)F RDP00195 CC(C)(C)C(=O)CC(c1ccc(cc1)Cl)Nc2ccccc2 RJC01195 CC(C)(C)C(=O)CC(c1ccccc1)Nc2ccccc2 RJC01196 Cc1ccc(cc1)Sc2cc(c(cc2OC)[N+](=O)[O-])C NRB03391 COc1c(cc(c(c1NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)Cl)Cl RF00680 Cc1ccc(cc1)Sc2c(c(c(c(n2)C)[N+](=O)[O-])C)C#N RF00661 CCOC(=O)c1c(c(nc(c1[N+](=O)[O-])C)O)C#N RF00743 Cc1c(c(no1)c2c(cccc2Cl)F)C#N RF00744 COc1cc(ccc1N=NN2CCOCC2)Cl NRB03413 c1cc(c(cc1C(F)(F)F)Nc2ncnc(n2)N)Cl RDR02608 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN3CCCCC3 RF00930 Cc1ccc(cc1)C(=O)/C=C/S/C(=N/C#N)/SCc2ccccc2 NRB03522 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C(=N/OC(=O)N(C)C)/N RF00807 CCOc1c(c(=O)c1=O)NCc2ccccc2 RDP00148 CCc1[nH]n(c2c(c(=O)c2=O)n(n1)C)C RDP00184 C1CCN(CC1)c2c(c(=O)c2=O)N3CCOCC3 RDP00199 CCOc1c(c(=O)c1=O)N2CC(OC(C2)C)C RDP00201 CCNc1c(c(=O)c1=O)NCC RDP00204 CCOc1c(c(=O)c1=O)Nc2ccccc2O RDP00185 c1ccc(c(c1)C(=O)N)Br RDP00161 CC(C)(C(=O)N)Oc1ccc(cc1)Cl RDP00163 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nc(on3)CSc4ccccn4 RF00810 c1ccc(cc1)c2cc(c(c-3c2C(=O)c4c3cccc4)C(=O)c5ccccc5)c6ccc(cc6)Cl NRB03433 c1c(ccc(c1)F)C(=O)/C=C/S/C=C/C(=O)c2ccc(cc2)F NRB03478 COC(=O)c1cc(nc(c1)OCC(F)(F)F)OCC(F)(F)F RF04928 Cc1ccc2c(c1)Nc3c(c(=O)c3=O)N2 RDP00178 c1ccc2c(c1)CCC(O2)C(=O)O RJC01246 CN(C)/C=C/c1nnnn1c2ccc3ccccc3c2 NRB03492 CCOC(=O)c1ccc2c(c1)nc(c(n2)C)C RDP00190 Cc1c(nc2cc(ccc2n1)C(=O)OC)C RDP00206 C1COCCN1c2c(c(=O)c2=O)N RDP00207 CCOc1c(c(=O)c1=O)N2CCSCC2 RDP00215 CCCc1c(nc2ccccc2n1)C RDP00216 Cc1cc2c(cc1C)nc(c(n2)C)C RDP00196 CCc1ccc(cc1)n2c(nnn2)/C(=C/N(C)C)/C(=O)C NRB03493 Cc1cc(cc(c1Cl)C)OCc2ccccc2 RDP00218 COC(=O)CNC(=O)c1ccccc1 RDP00222 c1cc(ccc1SC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl RF00602 Cc1c(c(no1)c2c(cccc2Cl)F)C(=S)N RF00747 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=N)N.Cl RF00749 Cc1c(c(no1)c2c(cccc2Cl)Cl)C#N RF00723 Cc1cccc2c1NC(=O)C(C2=O)c3ccccc3 RJC01270 c1ccc2c(c1)c(c(c(=O)[nH]2)[N+](=O)[O-])O RJC01271 CNC(=O)O/N=C/c1c(cn(n1)C)Br RF04801 CCCCCCCCCCCCSC(=S)Nc1ccc(cc1)F RF00592 CCCCCCCCCCCCSC(=S)Nc1cc(ccc1C)Cl RF00594 CCCCCCCCCCCCSC(=S)Nc1ccc(c(c1)Cl)Cl RF00595 Cc1c(c(no1)c2c(cccc2Cl)F)/C(=N/OC(=O)c3ccco3)/N RF00798 c1cc(ccc1N/C=C\c2nnnn2c3ccc(cc3)F)OC(F)(F)F NRB03481 CC(C)(C)c1ccc(cc1)/C(=N/O)/N RF00724 Cc1ccc(cc1)Cc2c(nc(nc2O)S)C RDR02413 c1cc(ccc1CNC(=O)C(Cl)Cl)C(=O)NN RJC02326 CC(C)(C)c1ccc(cc1)C(=O)N(C)C(=O)N(C)C(=O)c2ccc(cc2)C(C)(C)C RF00764 Cc1cc(nc(c1C(=O)O)O)O RF00769 CC1C(=O)N(C(=O)O1)c2cc(cc(c2)Cl)Cl RF04913 c1ccc(cc1)[I+]c2c(c3ccccc3[nH]c2=O)[O-] NRB04776 c1cc(ccc1C(c2ccc(cc2)Cl)C(=O)O)Cl RJC02290 C1CCN(C1)c2c(c(=O)c2=O)N3CCOCC3 RDP00208 c1ccc(cc1)CNc2c(c(=O)c2=O)N RDP00209 CCOC(=O)CNC(=O)c1ccccc1 RDP00211 Cn1c2c(c(=O)n(c1=O)C)[nH]c(n2)NCCc3ccccc3 RJC01277 Cc1ccc(cc1)/C(=C/C(=C\2/Cc3ccccc3C2=O)/c4ccccc4)/CC(=O)c5ccccc5 NRB03431 c1ccc(cc1)NC(=Nc2ccccc2)Nc3ccccc3 RJC02332 Cc1ccc(cc1)N/C=C\c2nnnn2c3ccc(cc3)Cl NRB03311 Cc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccccc3OC NRB03313 c1ccc(c(c1)NC(=O)c2ccc(cc2)F)I RJC02288 CS/C(=N\C#N)/S/C=C/C(=O)c1cccc(c1)Br NRB03485 Cc1c(c(=O)[nH]c(c1/N=N/c2ccc(cc2)[N+](=O)[O-])O)C#N NRB04791 Cc1c(nc2cc(ccc2n1)C(F)(F)F)C RDP00217 C=CCS/C(=N\C#N)/S/C=C/C(=O)c1cccc(c1)Br NRB03487 c1ccc2c(c1)cc-3oc4ccccc4cc23 NRB03490 CCc1c(c(c(=O)n(c1c2ccccc2)c3nccs3)Cc4ccccc4)O NRB04797 c1cc2c(cc1[N+](=O)[O-])nsn2 RDP00064 Cc1ccc(cc1)C(=O)C/C(=C\C(=O)c2ccc(cc2)C)/c3ccccc3 NRB03352 c1ccc(cc1)/C(=C/C(=O)c2ccc(cc2)F)/CC(=O)c3ccc(cc3)F NRB03353 Cc1ccc(cc1)C(=O)/C=C(\CC(=O)c2ccccc2)/c3ccccc3 NRB03356 c1ccc(cc1)C(=O)OC[C@@H]2[C@H]([C@@H]([C@H]([C@@H](O2)OC(=O)c3ccccc3)OC(=O)c4ccccc4)OC(=O)c5ccccc5)OC(=O)c6ccccc6 RJC02349 c1cc(ncc1C(=O)O)OCC(F)(F)F RF04860 C1CSCCN1c2c(c(=O)c2=O)N RDP00219 Cc1c(c(nc(n1)S)O)Cc2ccccc2 RDR02412 CCOC(=O)C(C)Oc1ccc(cc1)S(=O)(=O)N RDR02367 COC(=O)C1C(C(S(=O)(=O)CS1(=O)=O)C(=O)OC)c2ccccc2 RJC02335 CC(C)(C)c1ccc(cc1)c2nc(on2)CS(=O)(=O)c3ccc(cc3)Cl RF00788 COc1ccc(cc1)N/C=C\c2nnnn2c3ccc(cc3)Cl NRB03321 Cc1cc(nc(=S)[nH]1)C.Cl RJC02291 c1cc(ccc1C(=O)/C=C/C(=O)c2ccc(cc2)F)F RJC01100 c1cc(ncc1C(=O)N)OCC(F)(F)F RF04949 C=CCS/C(=N\C#N)/S/C=C/C(=O)c1ccccc1F NRB03484 c1ccc(cc1)C2CS(=O)(=O)CS(=O)(=O)C2 RJC02334 CC(C)(C)c1ccc(cc1)c2nc(on2)CSc3ccccn3 RF00790 Cc1c(c(no1)c2c(cccc2Cl)F)/C(=N/OC(=O)c3ccc(cc3)C(C)(C)C)/N RF00797 c1cc(oc1)CNc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] RJC02336 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)NCCCC(=O)O RJC02340 c1cc(ccc1CN2CCOCC2)C(=O)O.Cl RJC02333 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])NCCCC(=O)O RJC02337 c1ccc2c(c1)c(=O)c(c3n2cccc3)C#N RJC02293 c1cc2c(ccc(c2nc1)NCCO)[N+](=O)[O-] RJC01127 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN3CCCCCC3 RF00557 COc1ccccc1N/C=C\c2nnnn2c3ccc(cc3)F NRB03315 CNC(=O)n1cc(c(n1)/C(=N\OCc2ccccc2)/N)Br RF05207 CC1(C(=O)N(C(=O)NO1)CCc2cccs2)C RF05243 CNC(=O)NC1CCS(=O)(=O)C1 RJC02398 c1ccc(cc1)N/C(=N\O)/c2cccc(c2)C(F)(F)F RF05117 c1c(cnc(c1[N+](=O)[O-])O)C(F)(F)F RF04994 C#CCOC(=O)Nc1ccc(nc1)OCC(F)(F)F RF05274 Cc1ccc(cc1)S(=O)(=O)O[C@H]2[C@H]3[C@@H](COC(O3)c4ccccc4)O[C@@H]([C@@H]2OC(=O)c5ccccc5)OC NRB04857 Cc1cc2c(c(nnc2O)N)c(n1)O RF00735 Cc1cc2c(cc1Cl)nsn2 RDP00248 c1cc(cc(c1)N/C(=N/O)/c2cccnc2)C(F)(F)F RF05152 CO/N=C(\c1c(c[nH]n1)Br)/N RF05200 CSc1c(c(cc(n1)Nc2cccc(c2)[N+](=O)[O-])C(F)(F)F)C#N RF05466 CC(=O)OC[C@H]([C@@H]([C@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C RJC01374 CCSC([C@@H]([C@H]([C@@H]([C@@H](CO)O)O)O)O)SCC NRB04841 CS/C(=N\C#N)/S/C=C/C(=O)c1ccccc1F NRB03374 c1ccc(cc1)N/C=C\C(=N\c2ccccc2)\c3ccc(cc3)Cl NRB03375 CC(=O)c1c(c2ccccc2n(c1=O)c3ccccc3)O NRB04787 Cn1c2ccccc2c(c(c1=O)C#N)O NRB04790 CNC(=O)n1cc(c(n1)/C(=N/OC(=O)NC)/N)Br RF05199 CC1(O[C@@H]2[C@H]([C@H](O[C@@H]2O1)C(COS(=O)(=O)C)OS(=O)(=O)C)OS(=O)(=O)C)C NRB04850 Cc1ccc(cc1)S(=O)(=O)O[C@H]2COC3[C@@H]2OC[C@H]3OS(=O)(=O)c4ccc(cc4)C NRB04851 Cc1ccc(cc1)/C=C/2\CCCc3ccccc3C2=O RJC01407 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)F RDR02491 CC1(O[C@@H]2[C@H]([C@H](O[C@@H]2O1)C(CC#N)OS(=O)(=O)C)OCc3ccccc3)C NRB04848 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F RDR02489 c1ccc(cc1)/C=C/C=N/N=C(N)N RJC02352 c1ccc2c(c1)c3c(c(=O)o2)C(c4c(c5ccccc5oc4=O)O3)c6ccc(cc6)[N+](=O)[O-] NRB04868 CS(=O)(=O)Nc1ccc2c(c1)c(=O)c3ccccc3o2 NRB04875 CCCCc1c(nc(nc1O)S)C RDR02438 CCc1cccc(c1NS(=O)(=O)c2ccc(cc2)NC(=O)C)CC RDR02480 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)O)CC=C RDR02493 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl RDR02498 Cc1nc2ccc(cc2s1)NC(=O)c3ccccc3 RJC02420 CC(=O)Oc1ccc(cc1)C2NC(CS2)C(=O)O RJC02350 CCCCc1c(nc(nc1O)N2CCCC2)C RDR02501 COCCCNS(=O)(=O)c1ccc(cc1)NC(=O)c2ccc(cc2)Cl RDR02517 CC1=NNC(=O)C1Cc2ccccc2 RDR02395 CCc1cccc(c1NC(=S)Nc2ccc(cc2)C)CC RDR00013 CC1(c2ccccc2NC1=S)C RJC02408 COc1ccc(cc1)/C=C/c2nc3ccccc3s2 RJC02413 Cc1nc2cc(c(cc2n1C)[N+](=O)[O-])[N+](=O)[O-] RJC02414 c1cc(ccc1NC(=O)c2ccc(c(c2)Cl)Cl)S(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F RDR02485 CCN\1c2ccccc2S/C1=C/C(=S)Nc3ccccc3 RJC02416 c1ccc(cc1)CCNC(=S)N/N=C/c2c3ccccc3[nH]c2c4ccc(cc4)Cl RDR02526 Cc1cccc(c1NC(=O)CCN2CCOCC2)C RDR02555 c1c(ccc(c1)Cl)C(=O)/C=C/S/C=C/C(=O)c2ccc(cc2)Cl NRB03513 Cc1cc(c(cc1)C(=O)/C=C/S/C=C/C(=O)c2c(cc(cc2)C)C)C NRB03514 Cc1cccc(c1NS(=O)(=O)c2ccc(cc2)NOC(=O)C)C RDR02596 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl RDR02496 c1cc(cc(c1)NC(=S)Nc2ccc(cc2)NC(=S)Nc3cccc(c3)C(F)(F)F)C(F)(F)F RDR00040 c1ccc(cc1)c2csc(n2)N/N=C/c3c(cn[nH]3)Br.Br RF05308 CC1C(=O)N2C(=O)/C(=C\c3ccc(cc3)OC)/N=C2S1 NRB04872 COC(=O)Cc1ccc2c(c1)c(=O)c3ccccc3o2 NRB04873 CN(C)c1ccc(cc1)/C=C/c2nc3c4ccccc4ccc3s2 RJC02419 CCO/N=C(\c1c(c[nH]n1)Br)/N RF05201 Cc1cc(ccc1NC(=S)NC(=O)c2ccc(cc2)[N+](=O)[O-])Br RDR00054 CN(C)/C=C/C=C\1/C(=O)OC(=N1)c2ccccc2 NRB04886 c1ccc(cc1)c2ccc-3c4ccccc4cc3o2 NRB03510 CCc1c(c-2c3ccccc3cc2oc1C)C NRB03511 Cc1cccc(c1NC(=O)CCN2CCCC2)C RDR02557 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2c(cccc2Cl)Cl RDR02591 Cc1cc(ccc1Br)NS(=O)(=O)c2ccc(cc2)NC(=O)C RDR02478 Cc1cc2c(c(c1)C#N)CCCCCCCCCC2 NRB04879 Cc1ccc(cc1)c2nc(cc(n2)O)C RDR02584 CN1CCC(=C(c2ccccc2)c3ccccc3)C1.Cl RJC01308 CN\1c2ccccc2C=C/C1=C\C=C3c4ccccc4-c5c3cccc5 NRB04885 CC(C)NC(=S)N/N=C/c1cc[nH]n1 RF05316 CC(C(=O)O)Oc1ccc2ccccc2c1I RDR02568 CC(C(=O)Oc1ccc2ccccc2c1I)Oc3ccc(cc3)I RDR02574 c1cc(ccc1N)Oc2c(c(c(c(c2F)F)Oc3ccc(cc3)N)F)F RJC02400 Cc1csc([n+]1C)Nc2ccccc2OC.[I-] RDR00207 CCOC(=O)CNC(=O)c1cccs1 RJC02458 CCOC(=O)CNC(=O)c1ccc(cc1)OC RJC02461 Cn1cnnc1SCc2ccccc2[N+](=O)[O-] RJC02462 c1ccc(c(c1)C(F)(F)F)NC(=S)Nc2ccccc2N RDR00065 c1cc(c(c(c1)F)NC(=O)CN2CCCCC2)F RDR02565 CC(=O)OC[C@H]([C@@H]([C@@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC02378 c1ccc2c(c1)c3c(c(=O)o2)C(c4c(c5ccccc5oc4=O)O3)c6cccc(c6)[N+](=O)[O-] NRB04869 c1ccc(cc1)NC(=S)N/N=C/c2c(cn[nH]2)Br RF05281 Cc1cccc(c1NC(=O)CCN2CC(OC(C2)C)C)C RDR02558 CC(=O)Nc1ccc(cc1)Oc2c(c(c(c(c2F)F)Oc3ccc(cc3)NC(=O)C)F)F RJC02401 c1ccc(c(c1)Nc2ncnc(n2)N)F RDR02602 COc1ccc(cc1)Oc2cc(c(cc2Oc3ccc(cc3)OC)C(=O)O[Na])C(=O)O[Na] RJC02466 CC(=O)OC[C@H]([C@H]([C@@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C RJC01373 CS(=O)(=O)c1ccc2ccn(c2c1)O RJC02382 Cc1ccc(c(c1)NC(=O)C)C RJC01302 c1ccc(cc1)COC(CNC2CCCCC2)CNC3CCCCC3.Cl.Cl NRB03525 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl RDR02497 CC(C)(C)c1ccc(cc1)OS(=O)(=O)c2ccc(cc2Cl)Cl RDR02499 c1cc(cc2c1cc[nH]2)C(=O)O RJC02385 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)C(C)(C)C RDR02511 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)OC RDR02512 c1cc(ccc1NC(=S)N/N=C/c2c(cn[nH]2)Br)Cl RF05282 C/C(=N\Nc1ccccc1)/c2cc(cc(c2O)Cl)Cl RDR02549 c1cc(c(c(c1)F)NC(=O)CN2CCOCC2)F RDR02563 c1cc(ccc1c2csc(n2)N/N=C\c3c(c[nH]n3)Br)Cl.Br RF05311 COc1ccc(cc1OC)C(Cc2ccccc2)N.Cl NRB03527 c1ccc(cc1)CCSCC(=O)O RJC01304 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccccc2Cl RDR02593 CN(C)/C=C(/c1nnnn1c2ccc(cc2)OC)\C(=O)c3ccccc3 NRB03501 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2I)I RDR02598 CCOC(=O)c1cc(nc(c1C#N)SCC=C)C RF00843 CCOC(=O)c1cc(nc(c1C#N)S(=O)(=O)C)C RF00844 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3cc(ccc3Cl)Cl RF00928 Cc1ccc(cc1)COC(CN2CCCCCC2)CN3CCCCCC3.Cl.Cl NRB03524 CCOC(=O)c1cc(ccc1OS(=O)(=O)c2ccc(cc2)NC(=O)C)Cl RDR02594 CC1([C@@H](SCN1)C(=O)[O-])C.[K+] RJC02371 c1ccc(cc1)/C=C/c2nc3ccccc3o2 RJC02417 CC1(c2ccccc2N3C1=CC4(C(c5ccccc5N4CC3)(C)C)C)C RJC02421 CC1(c2ccc3ccccc3c2N=C1/C=C/c4ccc(cc4)N(C)C)C RJC02422 Cc1ccc2c(c1C)Nc3c(c(=O)c3=O)N2 RDP00179 Cc1c(nc2cc(ccc2n1)Cl)C RDP00197 Cc1cc(ccc1NC(=O)C)I RDP00225 Cc1cccc(c1)c2nc(cc(n2)O)C RDR02587 Cc1ccc(c(c1)[N+](=O)[O-])OS(=O)(=O)c2ccc(cc2)NC(=O)C RDR02588 COCCCNS(=O)(=O)c1ccc(cc1)NS(=O)(=O)c2cc(ccc2OC)OC RDR02617 c1c[nH]nc1/C=N\NC(=S)NC2CCCCC2 RF05317 c1ccc(cc1)CSC23CC4CC(C2)CC(C4)C3 RJC01240 CC(C)NCC(COc1cccc2c1cccc2)O.Cl RJC01228 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N RF00732 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN(C)C RF00926 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3ccccc3 RF00927 CC(C)(C)NC(=O)N/N=C/c1c(cn[nH]1)Br RF05287 Cc1ccccc1CO/N=C\c2c(c[nH]n2)Br RF05346 CCOC(=O)c1nc(on1)Oc2ccc(cc2Cl)Cl RF05313 c1cc(ccc1NC(=S)N/N=C\c2cc[nH]n2)Cl RF05320 c1ccc2c(c1)ccc3c2Cc4c5ccccc5ccc4OCO3 RJC01319 c1ccc2cc3c(cc2c1)cc([nH]3)S(=O)(=O)[O-].[Na+] RJC01295 c1ccc(cc1)C2=NOC(=O)C2 RF00778 c1ccc(cc1)C\2=NOC(=O)/C2=N/O RF00779 CC(C)(C)c1ccc(cc1)c2nc(on2)CSc3ccc(cc3)Cl RF00785 c1c(cc(nc1OCC(F)(F)F)OCC(F)(F)F)C(=O)NNC2=NCCCN2 RF04937 c1cc(c(nc1)OCC(F)(F)F)C(=O)NCc2ccc(cc2Cl)Cl RF04940 c1ccc(cc1)C2C(=O)N=C(S2)N/N=C\c3c(c[nH]n3)Br RF05306 CCCCCCCCC(=O)N(CC(C)/C(=N/c1ccccc1)/Nc2ccccc2)c3ccccc3.Cl RJC01316 CCCCCCCCCCCCC(=O)N(CC(C)/C(=N/c1ccccc1)/Nc2ccccc2)c3ccccc3.Cl RJC01317 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(cs3)c4cc5cc(ccc5o4)Cl RF00848 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nc(on3)CS(=O)(=O)c4ccc(cc4)Cl RF00812 Cc1c(c(nc(c1Cl)C)O)C#N RF00816 c1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)OC(F)(F)F NRB03516 Cc1ccc(cc1)C(=O)/C=C/S/C=C/C(=O)c2ccc(cc2)C NRB03476 Cc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)OC(F)(F)F NRB03480 Cc1c(nc2cc(ccc2n1)[N+](=O)[O-])C RDP00198 c1cc(cc(c1)C(F)(F)F)C(c2cccc(c2)C(F)(F)F)O RJC01288 CCC1NC(CS1)C(=O)O RJC02372 CN(C)/C=C(/c1nnnn1c2ccccc2)\C(=O)c3ccc(cc3)Cl NRB03507 c1ccc(c(c1)/C=N/NC(=S)NN)[N+](=O)[O-] RJC02366 Cc1ccc(cc1)c2csc(n2)c3c(onc3c4c(cccc4Cl)F)C RF00845 C=CCNC(=O)Nc1ncc(s1)[N+](=O)[O-] RJC01294 CC(=O)OC[C@H]([C@H]([C@H](C(=O)N)OC(=O)C)OC(=O)C)OC(=O)C RJC02369 CN(C)/C=C(/c1nnnn1c2ccccc2)\C(=O)c3cccc(c3)Cl NRB03506 COc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)OC(F)(F)F NRB03519 CCOC(=O)CNC(=O)c1cccc(c1)Cl RJC02427 CCCNc1c(c(=O)c1=O)N RDP00243 Cc1cc2c(cc1Cl)[nH]nn2 RDP00249 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2Cl)C(F)(F)F RDR02379 CCCC(=O)/C(=C\N(C)C)/c1nnnn1c2ccccc2 NRB03498 CCOC(=O)C1=C(NC(=O)N(C1c2ccccc2)C(=O)C)C NRB04808 c1cc(ccc1NC(=S)Nc2ccc(cc2)F)F RDR00029 Cc1cc(c(c(c1)C)Nc2nnns2)C RDR00033 c1ccc(cc1)C(=O)OC(CN2CCCCC2)CN3CCCCC3.Cl.Cl NRB03523 Cc1ccc(cc1)S(=O)(=O)O[C@@H]2[C@@H]3[C@@H](C(C(=O)O3)OS(=O)(=O)c4ccc(cc4)C)O[C@H]2OC NRB04843 Cc1cc(nn1c2ccccc2)NC(=O)N(C)C RF00836 Cc1cc(nn1c2ccccc2)NC(=O)OC RF00839 CCCCCCCc1c(c2ccccc2[nH]c1=O)O RJC01260 Cc1c(c(no1)c2c(cccc2Cl)F)/C(=N/OC(=O)c3c(onc3c4c(cccc4Cl)Cl)C)/N RF00799 c1ccc(cc1)c2c(n3ccccc3n2)Sc4ccc(cc4)I RJC02347 c1ccc(cc1)Cc2c(c3c(c4ccccc4[nH]c3=O)oc2=O)O NRB04813 CCC(=O)Nc1cc(c(nc1)OC)C(F)(F)F RF05094 c1ccc2c(c1)nc(s2)SCSc3nc4ccccc4s3 RJC02405 CC(C)c1ccc(cc1)Nc2nnns2 RDR00038 Cc1cc(c(c(c1)C)/N=C\2/N(C(=O)CS2)Cc3ccco3)C RDR00193 COc1ccccc1c2nn(c(=O)o2)c3c(cccn3)C(F)(F)F RF04882 COc1ccccc1c2nn(c(=O)o2)c3cc(ccn3)C(F)(F)F RF04908 Cc1cc(nn1c2ccccc2)NC(=O)OCC#C RF00837 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(on3)c4c(onc4c5c(cccc5Cl)Cl)C RF00802 COC(=O)c1ccc(nc1)OCC(F)(F)F RF04859 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)NCCCC(=O)O RJC02341 c1ccc(cc1)c2c(n3ccccc3n2)Sc4ccccc4 RJC02346 c1ccc(cc1)[C@@H](C#N)O[C@@H]2[C@H]([C@@H]([C@H](C(O2)CO[C@H]3[C@@H]([C@H]([C@@H]([C@H](O3)CO)O)O)O)O)O)O RJC02360 Cc1cc(nc(n1)N2CCOCC2)O RDR02447 c1cc(ccc1NNC(=O)c2cc(nc(c2)OCC(F)(F)F)OCC(F)(F)F)F RF04974 Cc1cc2cc(ccc2[nH]1)[N+](=O)[O-] RJC02389 CC(=O)OC[C@@H]([C@H]([C@@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C RJC01375 COc1ccc(cc1)Oc2cc(c(cc2Oc3ccc(cc3)OC)C#N)C#N RJC02438 c1cc(ccc1c2nc(on2)c3ccno3)C(F)(F)F RF05389 CNc1c(c(cc(n1)c2cccs2)C(F)(F)F)C#N RF01020 CC(C)(C)c1ccc(cc1)c2nc(on2)c3ccno3 RF05390 c1cc(oc1c2nc(on2)c3ccno3)[N+](=O)[O-] RF05391 CC(=O)CC(c1ccc(cc1)[N+](=O)[O-])c2c(c3ccccc3oc2=O)OC(=O)C NRB04865 CC(=O)CC(c1cccc(c1)[N+](=O)[O-])c2c(c3ccccc3oc2=O)OC(=O)C NRB04866 CCCOc1ccccc1NC(=O)/C=C/C(=O)N RJC02756 C1CC(=O)N(C1=O)OC(=O)CNC(=O)CCCCC(=O)NCC(=O)ON2C(=O)CCC2=O RJC01340 c1ccc(c(c1)O)OCCCCCOc2ccccc2O NRB03608 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3c(cccc3C)C RDR02654 c1c(cc(cc1C(F)(F)F)NC(=O)CN2CCOCC2)C(F)(F)F RDR02659 COc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3F)F NRB03517 CSc1nc(cc(n1)N)N RDR02422 c1ccc(cc1)C23C(NC(=O)N2)(NC(=O)N3)c4ccccc4 RJC02748 COc1cc(cc(c1OC)OC)/C=N/OC(=O)c2ccc(cc2Cl)Cl RDR02692 COCCCNC(=S)Nc1cccc2c1cccc2 RDR00237 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNC(=S)NC(C)(C)C RF00935 CC(C)S(=O)(=O)CC(=O)NCC(=O)OC RJC02484 CC(C)NC(=S)Nc1cccc2c1cccc2 RDR00246 c1ccc(cc1)C\2=NOC(=O)/C2=N/Nc3ccc(c(c3)Cl)Br RF00975 c1ccc(cc1)C\2=NOC(=O)/C2=N/Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F RF00977 Cc1cc(c(c(c1)Cl)OS(=O)(=O)c2ccc(cc2)NC(=O)C)Cl RDR02589 c1cc(c(cc1N)C(=O)O)SCC(=O)O RJC02357 CC(=O)n1cc(c2c1cccc2)OC(=O)C RJC02358 COCCCNS(=O)(=O)c1ccc(cc1)NC(=O)c2ccc(cc2Cl)Cl RDR02518 CC(C)(C)NCC(COc1ccc(cc1)OC)O.Cl RDR02613 C[C@@]12CCC3C4CC[C@](C4(CCC3C1(C/C(=C\c5ccccc5)/C(=O)C2)C)C)(C)O NRB03682 c1cc(ccc1/C=C/2\C(=O)N3CCCSC3=N2)[N+](=O)[O-] NRB03559 Cc1ccccc1CO/N=C\c2c(cn(n2)C(=O)NC)Br RF05351 CCOC(=O)CNC(=O)c1ccccc1Cl RJC02442 c1ccc2c(c1)n(c(=S)s2)CCn3c4ccccc4sc3=S RJC02406 CC12CC[C@H](C[C@@H]1CCC3C2CCC4(C3CCC4=O)C)O NRB03688 c1ccc(cc1)CCNC(=S)Nc2cc(c(cc2Cl)Cl)Cl RDR00093 c1ccc(c(c1)CCC(c2ccc3c(c2)OCCO3)N)Cl.Cl NRB03538 CC(C)c1ccc(cc1)NC(=S)NCCc2ccccc2 RDR00101 Cc1cc(c(c(c1)C)NC(=S)NCCNCc2ccccc2)C RDR00114 CCc1ccccc1NC(=S)Nc2c(cccc2CC)CC RDR00115 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Sc2ccccc2)OC(=O)C)OC(=O)C)OC(=O)C RJC01345 Cc1cc(cc(c1)OS(=O)(=O)c2ccc(cc2)NC(=O)C)C RDR02590 Cc1ccc(cc1[N+](=O)[O-])OS(=O)(=O)c2ccc(cc2)NC(=O)C RDR02592 CCc1ccc(cc1)NC(=S)NCCc2ccc(c(c2)OC)OC RDR00106 c1ccc2c(c1)ccc(c2I)OC(=O)c3ccc(cc3)Cl RDR02605 Cc1ccc(cc1)S(=O)(=O)Oc2ccc3ccccc3c2I RDR02607 CC(=O)OC[C@@H]1[C@@H]([C@@H](C(=C(O1)C#N)OC(=O)C)OC(=O)C)OC(=O)C RJC01348 COc1ccc(cc1OC)CCn2cnc3c2ccc(c3)C(F)(F)F RDR02619 Cc1cc(ccc1NC(=O)CN2CCOCC2)Br RDR02638 c1ccc(cc1)C\2=NOC(=O)/C2=C\c3ccc(s3)[N+](=O)[O-] RF00974 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N3CCOCC3)CC(CN4CCN(CC4)C)O.Cl.Cl NRB03552 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCc3ccco3)CC(CN(Cc4ccccc4)Cc5ccccc5)O NRB03553 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)S(=O)(=O)c2ccccc2)OC(=O)C)OC(=O)C)OC(=O)C RJC01346 c1ccc(cc1)SCCn2c(=O)c3ccccc3[nH]c2=O RJC02445 Cc1cc2c(c(nnc2O)N)c(n1)Sc3ccc(cc3)Cl RF00981 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)NCCCOC RDR02615 COC(=O)CNC(=O)CSc1ccccn1 RJC02430 COC(=O)CNC(=O)CSc1ccccc1 RJC02431 c1ccc(c(c1)C(=O)NCC(=O)O)Cl RJC02443 c1ccc2c(c1)c(=O)c3cc(ccc3o2)C(=O)O NRB03554 CC(Cn1c2c(nc1N(Cc3ccccc3)Cc4ccccc4)n(c(=O)n(c2=O)C)C)O NRB03547 Cc1cc(ccc1NC(=S)NCCCNC2CCCCC2)Cl RDR00107 CN(C)/C=N/c1c(non1)c2ccccc2 RF00987 CN(C)/C=N/c1c(non1)c2ccc(cc2)Cl RF00991 c1cc(ccc1C(=O)NNC(=O)c2ccno2)Cl RF05357 c1cn[nH]c1/C=N/N=C/2\NC(=O)CS2 RF05360 c1ccc(cc1)C(=O)OC[C@@H]2[C@H]([C@@H](C(=CO2)OC(=O)c3ccccc3)OC(=O)c4ccccc4)OC(=O)c5ccccc5 RJC01351 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H](CO1)OC(=O)C)OC(=O)C)OC(=O)C RJC01352 Cc1cccc(c1NC(=S)NCCO)C S01188 c1cc(c(cc1C(F)(F)F)NC(=O)CCN2CCOCC2)Cl RDR02643 Cc1cc(ccc1Br)NC(=O)CCN2CCOCC2 RDR02645 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CCCCn3cnc4c3c(=O)n(c(=O)n4C)C NRB03565 CC1=C(C(NC(=O)N1)c2ccc(cc2)Cl)C(=O)C RJC02752 c1ccc(c(c1)NC(=S)SCCSC(=S)Nc2ccccc2Cl)Cl RDR02628 c1ccc(cc1)C(Cc2cccnc2)(c3ccc(cc3)Cl)O RF01093 c1cc(cc(c1)Cl)C(=O)NNC(=O)c2ccno2 RF05356 c1ccc(cc1)CCNC(=S)Nc2cccc(c2Cl)Cl RDR00091 CC(=O)O[C@@H]1CO[C@@H]([C@H]([C@@H]1OC(=O)C)OC(=O)C)c2nc3ccccc3s2 RJC01362 c1ccc(cc1)CCNC(=S)Nc2c(cccc2Cl)Cl RDR00099 c1cc(ccc1c2csc(n2)NC(=O)CN3CCCCC3)Cl RDR02621 Cc1cccc(c1NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccccc3)C RDR02653 c1ccnc(c1)SCC(=O)NCC(=O)O RJC02464 COc1ccc(cc1)C(=O)NCC(=O)N RJC02465 CC(C)(C)c1cc2c(cc(cc2[N+](=O)[O-])C(C)(C)C)c(c1)[N+](=O)[O-] RJC02468 c1ccc(cc1)C(=O)OC[C@@H]2[C@H]([C@H]([C@@H](O2)C#N)OC(=O)c3ccccc3)OC(=O)c4ccccc4 RJC01365 CCc1cccc(c1NC(=S)Nc2cccc(c2Cl)Cl)CC RDR00118 c1cc(ccc1c2csc(n2)NC(=O)CCN3CCCC3)Cl RDR02635 c1cc2c(cc1S(=O)(=O)N3CCCCCC3)OCCO2 RJC02762 c1cc(ccc1C(=O)Nc2ccc(cc2I)I)Cl RDR02599 c1ccc(cc1)C(=O)O[C@@H]2CO[C@H]([C@@H]([C@@H]2OC(=O)c3ccccc3)OC(=O)c4ccccc4)C#N RJC01367 Cn1ccc(n1)/C=N/N=C\2/NC(=O)CS2 RF05421 C=C1COC(=O)N1Cc2ccccc2Cl RF05444 c1cc(c(c(c1)Cl)Cl)NC(=S)NCCC(=O)O RDR00159 c1cc(c(c(c1)Cl)Cl)NC(=S)NCc2ccco2 RDR00178 c1cc(ccc1c2csc(n2)NC(=O)c3ccc(cc3)Cl)Cl RDR02636 CCOC(=O)c1cc2cc(ccc2oc1=O)Cl RDR02664 c1ccc(cc1)c2c(c(oc2c3ccccc3)N)C#N RJC02473 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@H](O1)OC)OC(=O)C)OC(=O)C)OC(=O)C RJC01370 COc1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2I)I)OC RDR02688 c1c(c([nH]n1)/C=N/NC(=S)NC2CCCCC2)Br RF05280 CC(C)(C)NC(=S)N/N=C\c1c(c[nH]n1)Cl RF05321 Cc1c(cccc1Cl)NC(=S)NCc2ccco2 RDR00182 c1cc2c(=O)c3cc(ccc3oc2c(c1)Cl)C(=O)O NRB03555 CCOC(=O)CN1C(=O)C(N(C1=O)CC(=O)c2ccccc2)(c3ccccc3)c4ccccc4 NRB03557 c1cc(cc(c1)[N+](=O)[O-])/C=C/2\C(=O)N3CCCSC3=N2 NRB03558 c1ccc(cc1)N2C(C3C(O2)C(=O)N(C3=O)c4ccccc4)c5ccc(cc5)F RJC02758 CC(=O)OC[C@@H]([C@@H]([C@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C RJC01372 COc1cc(c(cc1CC#N)OC)CC#N RJC02469 c1cc(c(nc1)OCC(F)(F)F)C(=O)NCc2ccc(cc2)Cl RF04938 CN(C)/C=C(/c1nnnn1c2ccc(cc2)Cl)\C(=O)c3ccccc3 NRB03503 CN(C)/C=C(/c1nnnn1c2ccc(cc2)Br)\C(=O)c3ccccc3 NRB03504 c1cc(cc(c1)Cl)c2nnc(o2)c3ccno3 RF05365 Cc1ccc(cc1)C(=O)OC[C@@H]2[C@H](C[C@@H](O2)C#N)OC(=O)c3ccc(cc3)C RJC01366 c1c(cc(cc1C(F)(F)F)NC(=O)CN2CCCC2)C(F)(F)F RDR02661 c1cc(c(cc1NC(=S)NCCC(=O)O)Cl)Cl RDR00160 c1ccnc(c1)SCc2cccc(n2)CSc3ccccn3 RJC02449 Cc1ccc(cc1)OCC(=O)Nc2ccc(cc2)NC(=O)C NRB03561 c1cc(ccc1c2cc3cc(ccc3o2)Cl)[N+](=O)[O-] RDR02648 Cc1cccc(c1NS(=O)(=O)c2ccc(cc2)N)C RDR02650 CCOC(=O)c1c(c[nH]n1)c2ccc(cc2Cl)Cl RF04996 Cc1cc(ccc1NC(=S)Nc2cccc(c2)C(F)(F)F)Br RDR00035 c1cc(oc1)CNC(=S)Nc2ccc(cc2)Cl RDR00170 CCCNC(=S)Nc1ccc(cc1)Cl RDR00171 Cc1nnc(s1)SCC(=O)Nc2ccc(cc2)Br RJC02485 Cc1nnc(s1)SCC(=O)Nc2ccc(cc2)C(=O)C RJC02486 CCOC(=O)c1cc2cc(ccc2oc1=O)Br RDR02665 COc1c(cccc1Cl)c2cn3ccccc3n2 RDR02680 c1cc(oc1)CN\2C(=O)CS/C2=N\c3ccc(cc3)Cl RDR00172 COCCCNC(=S)N/N=C/c1ccco1 RDR00174 COc1ccccc1/N=C\2/N(C(=O)CS2)Cc3ccco3 RDR00175 CCOC(=O)c1ccc(cc1)Nc2[n+](c(cs2)C)C.[I-] RDR00198 Cc1cccc(c1Nc2[n+](c(cs2)C)C)C.[I-] RDR00205 c1ccc(cc1)COC(=O)NCC#N RJC02477 Cc1csc([n+]1C)Nc2ccc(cc2)Cl.[I-] RDR00206 CC(C)(C)c1ccc(cc1)C(=O)CCN(C)C.Cl NRB03603 CC(=O)CC(c1ccccc1)c2c(c3ccccc3oc2=O)OC(=O)C NRB04864 CCN(Cc1ccccc1)c2nc3c(n2CCO)c(=O)n(c(=O)n3C)C NRB03546 Cc1cc(c(cc1C)NC(=S)NCCCOC)C RDR00210 COCCCNC(=S)Nc1cccc(c1)C(F)(F)F RDR00231 COc1cc(cc(c1OC)OC)/C=N/OC(=O)c2ccc(cc2)Cl RDR02689 CCSc1ccc(cc1)C(=O)NCC(=O)O RJC02455 c1cc(sc1)C(=O)NCC(=O)O RJC02457 Cc1ccc(c(c1)C)NC(=S)NCc2ccco2 RDR00186 CCOC(=O)C1=C(N=C2N(C1c3ccccc3)C(=O)CS2)C RJC02753 c1cc(ccc1NC(=S)CCC(=S)Nc2ccc(cc2)Cl)Cl RDR02629 CCCS/C(=N\CC)/Nc1c(cccc1C)C.I RDR00239 CCCCc1ccc(cc1)C(=O)CCN(C)C.Cl NRB03604 c1ccc(cc1)c2csc(n2)NC(=O)c3ccc(cc3)Cl RDR02637 CC(C)SCC(=O)NCC(=O)N RJC02487 CC1(O[C@@H]2[C@H]([C@H](O[C@@H]2O1)C(COC(=O)c3ccccc3)O)OC(=O)c4ccccc4)C NRB04853 Cc1cc(nn1c2ccccc2)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F RF00840 c1cc(c(nc1)OCC(F)(F)F)C(=O)NCc2ccc(c(c2)Cl)Cl RF04939 CN(C)C(=O)c1ccc(nc1)OCC(F)(F)F RF04950 CO[C@H]1[C@@H]([C@H]([C@H](O1)COC(=O)c2ccccc2)OC(=O)c3ccccc3)OC(=O)c4ccccc4 RJC01371 CN(C)C(=O)Oc1c2ccccc2on1 RF01308 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3ccc(c(c3)Cl)Cl RF01311 Cc1ccc(c(c1)C)N/N=C\2/C(=NNC2=O)C RJC02943 CC\1=NN(C(=O)/C1=N\Nc2ccccc2)c3ccccc3 RJC02944 CC(C)SCC(=O)Nc1ccc(cc1)Br RJC02488 CN(C)c1c(c(cc(n1)c2cccs2)C(F)(F)F)C#N RF01021 c1cc(sc1)c2cc(c(c(n2)Sc3ccc(cc3)Cl)C#N)C(F)(F)F RF01028 CCOC(=O)c1cc(nc(c1C#N)SC)C RF00841 CCOC(=O)c1cc(nc(c1C#N)SCC#C)C RF00842 c1ccc(c(c1)N/C(=N\O)/c2c(cccc2F)F)Cl RF05120 COCCCNC(=S)N/N=C/c1ccc(c(c1)Cl)Cl RDR00374 c1ccc2c(c1)c(ccc2/N=N\c3ccc(cc3)S(=O)(=O)N)N RDR00470 c1c(cc(cc1C(F)(F)F)/N=C/2\NCCN/C(=N/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)/SS2)C(F)(F)F RDR00498 c1ccc2c(c1)nc3c(n2)Sc4ccccc4N3 RJC01449 c1c(c(c(cn1)Cl)N)Cl RF01230 Cc1cc(nc(n1)c2cccs2)OC(=O)N(C)C RF01060 Cc1ccc(cc1)NC(=S)NCCCOC RDR00305 CC(C)(CO)NC(=S)Nc1ccc(cc1)F RDR00451 CC(C)c1ccc(cc1)NC(=S)N/N=C/c2ccccc2Cl RDR00349 COc1ccc(cc1)NC(=S)N/N=C/c2ccc(cc2)Cl RDR00354 CCOC(=O)c1cc(nc2c1cccc2)C3CC3 NRB03622 CCCCc1c(nc(nc1O)N)C RDR02663 Cc1ccn2cc(nc2c1)c3cccc(c3OC)Cl RDR02679 c1ccc2c(c1)c(=O)c(c-3[nH]c4ccccc4nc23)Cl RJC01466 c1ccc(c(c1)Sc2c(c(c(s2)Sc3ccccc3Br)[N+](=O)[O-])[N+](=O)[O-])Br RJC01467 CCOC(=O)C(C(F)(F)F)(NC(=O)c1cccc(c1)C)O RJC02676 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)Cl RJC02678 CC(=O)c1ccc(cc1)NC(=O)CSc2nncn2C RJC02504 CC12CCC3(C=C1CCC4C2C(=O)CC5(C4CCC56OCCO6)C)OCCO3 NRB03657 CC12CCC3C(C1CCC2O)CCC4=CC(=O)CCC34 NRB03703 CC1CC2C3CC[C@H]4CC(CCC4(C3[C@@H](CC2([C@]1(C(=O)C)O)C)O)C)O NRB03680 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H](CO1)OC(=O)C)OC(=O)C)OC(=O)C RJC01353 c1cc2c(c(c1)[N+](=O)[O-])C(=O)CC2=O RJC01388 C[C@]12CCC3C(C1CCC2=O)CCC45C3(C4)CCC(=O)C5 NRB03681 C[C@@]1(CCC2C1(CCC3C2CCC4=CC(=O)CCC34)C)O NRB03676 c1cc(ccc1NC(=S)NCCCNC2CCCCC2)Cl RDR00335 c1cc(c(cc1Cl)NC(=S)NCCCNC2CCCCC2)Cl RDR00339 C/C(=N\CCc1ccccc1)/C2CCOC2=O NRB03567 c1ccc(cc1)C(=O)NCC(=O)N RJC02447 CCOC(=O)CNC(=O)c1ccc(cc1)SCC RJC02444 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C(\C)/C(C)(C)C RF01182 c1ccc2c(c1)c(=O)c(co2)C(=O)O RF01275 CC(=O)OC12CCC(=O)C=C1CCC3C2CCC4(C3CCC4=O)C NRB03667 CC(=O)OCC(=O)[C@]1(CCC2C1(CCC3C2CC[C@@]4(C3(CCCC4)C)C)C)O NRB03672 Cc1ccc(cc1)C(=O)NC(C(=O)OC)(C(F)(F)F)O RJC02664 CCOc1ccccc1C(=O)NC(C(=O)OC)(C(F)(F)F)O RJC02665 CCOC(=O)CSc1ccc2nnc(n2n1)c3ccccc3 RH00154 c1ccc(cc1)c2nnc3n2nc(cc3)SCCO RH00156 c1ccc(cc1)c2nnc3n2nc(cc3)Oc4cccc(c4)C(F)(F)F RH00163 CNC(=O)Oc1c2cc(ccc2on1)Cl RF01327 CC12CCC3C(C1CCC2OC(=O)c4ccccc4)CC5[C@@]6(C3(CCC(C6)O)CO5)Br NRB03663 CCc1c(c2ccccc2[nH]c1=O)O RJC01476 COC(=O)C1(N=C(OC(=N1)N2CCOCC2)c3ccccc3)C(F)(F)F RJC02650 c1ccc(cc1)c2nnc3n2nc(cc3)Sc4cccc(c4)C(F)(F)F RH00148 COc1ccc2nnc(n2n1)c3ccccc3 RH00152 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3ccccn3 RF01320 CC1CC(CC(C1)(C)C)NC(=S)NCCO S01233 CC1(CS/C(=N\c2ccc(cc2)F)/N1)C RDR00452 CC1(CS/C(=N\c2ccccc2F)/N1)C RDR00459 Cc1cccc(c1/N=C\2/NC(CS2)(C)C)C RDR00461 CCOC(=O)C(C(F)(F)F)(Nc1cc(on1)C)NC(=O)c2cccc(c2)C RJC02672 CCOC(=O)c1ccc2c(c1)sc(n2)NC(=O)c3ccc(c(c3)Cl)F RH00142 Cc1c(c(no1)c2c(cccc2Cl)Cl)COC(=O)c3ccc(cc3)[N+](=O)[O-] RF01303 c1cc2c(cc1Cl)onc2O RF01288 Cc1c(c(no1)c2c(cccc2Cl)Cl)COC(=O)c3ccc(cc3)Cl RF01298 c1ccc(cc1)c2nnc3n2nc(cc3)Sc4ccc(cc4)Cl RH00146 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3ccc(cc3Cl)Cl RF01312 Cc1cc(cc(c1)Sc2ccc3nnc(n3n2)c4ccccc4)C RH00151 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3ccccc3 RF01317 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3c(cncc3Cl)Cl RF01218 CCC(=O)OC1CCC2C1(CCC3C2CCC4=CC(=O)CCC34C)C NRB03689 CCOC(=O)c1ccc(cc1)NCN2C(=O)c3ccccc3C2=O S01184 CCOC(=O)C1(N=C(OC(=N1)N2CCCCC2)c3cccc(c3)C)C(F)(F)F RJC02671 c1ccc(cc1)C23CCCC(C2)(CC3)I RJC01486 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNc3c(cncc3Cl)Cl RF01241 CCOC(=O)C1=NN(C(=NN1c2ccc(cc2)[N+](=O)[O-])C(=O)OCC)c3ccc(cc3)[N+](=O)[O-] RJC02939 CC\1=NNC(=O)/C1=N\Nc2ccccc2Cl RJC02940 Cc1ccccc1N/N=C\2/C(=NNC2=O)C RJC02941 CC(C)CCCC(C)C1CCC2C1(CCC3C2CC(C4=CC(CCC34C)O)O)C NRB03714 c1cc(sc1)C(=O)OCC(=O)c2ccc(cc2)Cl RDR02812 COc1ccc(cc1)NC(=O)/C=C/C(=O)O S01322 Cc1ccc(cc1)NC(=O)/C=C\C(=O)O S01331 COC(=O)C(C(F)(F)F)(NC(=O)COc1ccccc1)O RJC02666 COc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)NCc2cccnc2 RJC02667 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3ccc(cc3)N(C)C RF01316 CC(=O)OC1CCC2C1(CCC3C2CCC4C3(CC(=O)CC4)C)C NRB03692 CC(=O)OC1CCC2C1(CCC3C2CC[C@@H]4C3([C@H]([C@H]5C[C@H]5C4)O)C)C NRB03694 CCC(=O)OC1CCC2(C(C1)CCC3C2C(=O)CC4(C3CC=C4C(=O)C)C)C NRB03698 CC1=C(CC2C(C1)C(=O)N(C2=O)c3ccc(cc3)N4CCOCC4)C RJC02930 CC12CCC3C(C1CCC2O)CC4[C@@]5(C3(CCC(C5)O)CO4)Br NRB03696 CC12CCC(=O)C=C1CCC3C2CCC4(C3CC[C@]4(C#C)O)C NRB03706 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3cccnc3 RF01324 CC(C)(C)NC(=O)Oc1c2ccc(cc2on1)Cl RF01326 COCCCNC(=S)Nc1ccc2cn[nH]c2c1 RDR00248 CC12CCC3c4ccc(cc4CCC3C1CCC2=O)Oc5ccc(cc5)N(C)C NRB03655 COCCCNC(=S)N/N=C/c1ccc(c(c1)Br)OC RDR00282 COc1c(nccn1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)Br RJC02929 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3ccccc3[N+](=O)[O-] RF01319 CC(=O)O[C@@H]1CC2(C(CCC3C2CCC4(C3CCC4OC(=O)C)C)CC1=O)C NRB03691 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3ccc(cc3)F RF01314 c1ccc(cc1)CCN\2C(=O)CS/C2=N/c3c(cccc3Cl)Cl RDR00102 CCc1cccc(c1Nc2nc3c(s2)ccc(c3Cl)Cl)CC RDR00121 c1cc(cc(c1)Cl)C(=O)NCC(=O)N RJC02452 CCOC(=O)CC1=NC(=O)CS1 RJC01338 c1cc(sc1)C(=O)NCC(=O)N RJC02459 COCCCNC(=S)Nc1cccc(c1)SC RDR00269 Cc1cc(c(c(c1)C)NC(=S)NCCCOC)C RDR00303 Cc1c(cccc1Cl)NC(=S)N/N=C/c2ccccc2Cl RDR00322 c1ccc(c(c1)/C=N/NC(=S)Nc2cc(ccc2Cl)Cl)Cl RDR00325 c1ccc(cc1)C2C3C(N4CN2C(C(C4c5ccccc5)C3=O)c6ccccc6)c7ccccc7 RJC02951 c1ccc(c(c1)CSc2ccccn2)[N+](=O)[O-] RJC02460 COc1ccc(cc1)C(=O)NCC(=O)O RJC02463 c1ccc(cc1)c2nnc(o2)[C@H]3[C@@H]([C@H]([C@H]([C@H](O3)COC(=O)c4ccccc4)OC(=O)c5ccccc5)OC(=O)c6ccccc6)OC(=O)c7ccccc7 RJC01357 CC(=O)Oc1cccc(c1)NC(=O)CC2C(=O)Nc3ccccc3S2 RJC02932 CC\1=NN(C(=O)/C1=N\Nc2ccc(cc2)F)c3ccccc3 RJC02937 CCOC(=O)c1c(c(sc1NC(=O)C(F)(F)F)C(=O)OCC)C RJC01406 CCOC(=O)C1=C(NC2=C(C1c3ccccc3)C(=O)CC(C2)(C)C)C RJC01409 Cc1ccc(c(c1)C)N/N=C\2/C(=NN(C2=O)c3ccccc3)C RJC02933 CC(=O)c1ccc(cc1)NC(=O)COc2ccc(cc2)OC RJC02509 CC(C(=O)O)Nc1c(=O)[nH]c(=O)[nH]n1 RJC02540 CCCOC(=O)C(C)Nc1c(=O)[nH]c(=O)[nH]n1 RJC02542 c1ccc(cc1)CCNC(=O)C(Cc2ccccc2)N3C(=O)c4ccccc4C3=O RJC02543 CC(=O)OC1CCC2(C3CCC4(C(C3CC=C2C1)CCC4C(=O)OC5CC6CCC5C6)C)C NRB03707 COCCCNC(=S)Nc1ccc(cc1)OC RDR00215 CC[N+]1=C(SCC1)Nc2c(cccc2C)C.[I-] RDR00216 CCc1cccc(c1NC(=S)Nc2ccc(cc2)C(C)C)CC RDR00123 c1ccc(cc1)C(=O)O[C@@H]2CO[C@H]([C@H]([C@@H]2OC(=O)c3ccccc3)OC(=O)c4ccccc4)OC(=O)c5ccccc5 RJC01363 CCCSc1ccc2c(c1)nc([nH]2)NC(=O)C RJC02474 Cc1cc(nc(n1)c2ccccn2)O RF01053 CCc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3c(cccc3Cl)Cl RF01150 CN(C)c1ccc(cc1)/C=N/c2ccc(c(c2)O)C(=O)O RDR00293 Cc1cc(ccc1/N=C/c2cc(cc(c2O)Cl)Cl)Br RDR00330 CC1=C(C(NC(=S)N1)c2ccccc2)C(=O)OC RJC01410 Cc1cccc(c1NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl)C RDR02651 Cc1cccc(c1NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl)C RDR02652 c1cc(ccc1NC(=S)N/N=C/c2cc(cc(c2O)Cl)Cl)F RDR00289 CC12CCC3C(C1CCC2O)CCC4=CC(=O)/C(=C(\C(F)(F)F)/[O-])/CC34C.[K+] NRB03669 CC(C)NC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl RDR00290 CC12CCC3C(C1CCC2OC(=O)c4ccccc4)CCC5=CC(=O)CCC35CO NRB03670 CC(=O)Nc1ccc(cc1)NC(=S)NCCCOC RDR00297 C[C@@]12CCC3C4CCC(=O)C4(CCC3C1(CCC(=O)C2)CO)C NRB03674 CN(C)c1ccc(cc1)/C=N/NC(=S)Nc2cc(ccc2Cl)Cl RDR00326 c1cc(c(cc1Cl)n2ccnc2S)Cl RDR00372 c1ccc(cc1)Nc2nnc(s2)S S01205 c1cc(c(cc1Cl)NC(=S)NCCC(=O)O)Cl RDR00139 Cc1cccc(c1)N(c2ccccc2)c3ccc(cc3)c4ccc(cc4)N(c5ccccc5)c6cccc(c6)C RJC02479 CC1(c2ccccc2N(C13C=Cc4cc(cc(c4O3)[N+](=O)[O-])Br)C)C RJC02480 Cc1cc(c(c(c1)C)N/C(=N/CCCOC)/SC)C.I RDR00358 Cc1c(c(no1)c2c(cccc2Cl)Cl)COC(=O)c3ccc(cc3[N+](=O)[O-])Cl RF01301 CN(C)C(=O)Oc1c2cc(ccc2on1)Cl RF01305 CCCC(Nc1ccccn1)n2c3ccccc3nn2 RJC01431 CC(=O)NC12CC3CC(C1)CC(C3)(C2)O[N+](=O)[O-] NRB03630 CCOC(=O)c1cc(nc2c1cccc2)c3cccs3 NRB03635 c1ccc(cc1)c2ccc(cc2)c3cc(c4ccccc4n3)C(=O)O NRB03636 COc1cc(c(cc1OC)Br)CNc2ccccc2 NRB03611 CC(=O)c1cc(cs1)[N+](=O)[O-] NRB03624 CSC(=N)Nc1cc(ccc1Cl)Cl.I RDR00145 CN(C)C(=O)Oc1c2ccc(cc2on1)Cl RF01306 CCOC(=O)/C(=N\Nc1ccccc1)/c2csc(n2)N RJC02555 c1ccc2c(c1)cccc2OC(=O)/C=C/c3cccs3 RDR02805 CCOC(=O)c1cc(nc2c1cccc2)C34CC5CC(C3)CC(C5)C4 NRB03626 CC(C)c1ccc(cc1)NC(=S)N/N=C/c2ccc(c(c2)OC)OC RDR00348 C(C(CC(C(C(F)(F)F)(F)F)(F)F)C(=O)O)C(=O)O RJC01439 CCOC(=O)Cc1csc(n1)NC(=O)c2cccc(c2)Cl RJC02494 c1ccc2c(c1)c(=O)n(c(=O)[nH]2)CCSc3ccc(cc3)Cl RJC02498 CC(C)(C)c1cc2c(c(=N)[nH][nH]c2=O)c(=O)[nH]1 RF01043 Cc1cc(nc(n1)c2cccs2)O RF01046 Cc1c(c(nc(n1)c2ccccn2)O)Cl RF01049 COCCC(=O)NC12CC3CC(C1)CC(C3)C2 NRB03632 CCOc1ccc(cc1)NCN2C(=O)c3ccccc3C2=O S01262 COc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccccc3 S01253 CCOc1ccc(cc1)NC(=S)NCCO S01256 C/C(=N/OC(=O)Nc1ccccc1Cl)/C2CC2 RJC02841 CCOc1ccc(cc1)NC(=O)/C=C/C(=O)O S01328 c1ccc(cc1)C2=N/C(=C\c3cccc(c3)[N+](=O)[O-])/C(=O)O2 S01274 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)[N+](=O)[O-])/C(=O)O2 S01282 CC1CN=C(S1)N(c2ccc(cc2)Cl)C(=O)Nc3cccc(c3)Cl RJC02655 CSc1c(c(cc(n1)Nc2cccc(c2)C(F)(F)F)C(F)(F)F)C#N RF05463 Cc1cc(c(c(=O)o1)c2cc[nH]n2)O RF01179 c1ccc2c(c1)Nc3c(nc4ccc(cc4n3)Cl)S2 RJC01451 CC1CN=C(S1)N(C(C)c2ccccc2)C(=O)Nc3ccc(cc3)Cl RJC02662 c1ccc(c(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)C(C(F)(F)F)C(F)(F)F)Cl RJC02690 Cc1ccc(cc1)N2C(=O)C=CC2=O S01335 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)NCc2cccnc2 RJC02668 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)NCc2ccccn2 RJC02669 CCc1[nH]c(=O)c2cnn(c2n1)c3ccccc3 RJC02767 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)Cl)NC(=O)c2cccc(c2)C RJC02698 CC12CS(=O)(=O)CC1SC(=N)N2 RJC02854 Cc1ccc(c2c1nc(c(c2)C)Sc3ccc(cc3)Cl)F RH00137 c1ccc2c(c1)c(c(c(c2CN3CCCCC3)O)O)CN4CCCCC4 RJC02768 CC(=O)Oc1ccccc1/C(=C/C=C(c2ccccc2)c3ccccc3)/N4CCOCC4 RF01254 c1ccc2c(c1)c(=O)c(co2)C#N RF01263 Cc1c(c(ccn1)O)OCC(=O)O RF01266 c1ccc(cc1)Nc2nn(c(=S)n2c3ccccc3)CCC(=O)O RJC02851 CC(C)(C)NS(=O)(=O)C1CCS(=O)(=O)C1 RJC02852 CC1=C(Sc2ccccc2N1)C(=O)NN RH00160 CCOc1ccc(cc1)/N=C\2/NCCS2 S01260 C/C=C/CC(=O)NCC(=O)O RJC02501 c1ccc(cc1)CC2C(=O)NC(=N)S2 RJC02857 c1ccc(cc1)c2nnc3n2nc(cc3)Oc4ccc(cc4)F RH00164 Cc1c(ccc(c1OC(=O)c2cccs2)C(=O)C)OCc3ccccc3 RH00165 c1cc(ccc1c2ccc(cc2)S(=O)(=O)NC3CCS(=O)(=O)C3)S(=O)(=O)c4ccc(cc4)Cl RJC02858 Cc1cccc(c1NC(=O)/C=C/c2cccs2)C RDR02734 CC\1=NNC(=O)/C1=N\Nc2ccc(cc2)Br RJC02942 Cc1cc(c(c(c1)C)NC(=O)/C=C/c2cccs2)C RDR02735 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nccn2C RJC02512 Cc1ccc(cc1)S(=O)(=O)OCC23CCC(=O)C=C2CCC4C3CCC5(C4CCC5=O)C NRB03664 Cc1csc([n+]1CCCOC)Nc2ccc(cc2)OC.[I-] RDR00395 Cc1cc(c(c(c1)C)Nc2[n+](c(cs2)C)CCCOC)C.[I-] RDR00396 C/C=C/CC(=O)NCC(=O)NN RJC02502 COc1ccccc1C(=O)Nc2cccc(c2)Oc3c(c(c(c(c3F)F)F)F)F RJC02745 CC1CC(CC(C1)(C)C)/N=C\2/NCCS2 S01234 Cc1cc(no1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)N(C)C RJC02652 Cn1cnnc1SC/C=C/c2ccccc2 RJC02515 CC(=C)C(=O)Oc1c2ccccc2cc3c1cccc3 RJC02811 CC1=NOC2(C1C3C(C2)C3(C)C)O RJC02546 c1ccc2c(c1)nc3ccc(cc3n2)C(=O)O RJC02548 CCOC(=O)c1cc2cc(cc(c2oc1=O)Cl)Cl RDR00341 CC(C)c1ccc(cc1)NC(=S)N/N=C/c2cccs2 RDR00347 CC1CN=C(S1)N(CCc2ccccc2)C(=O)Nc3cccc(c3)Cl RJC02660 CNS(=O)(=O)C1CCS(=O)(=O)C1 RJC02779 Cc1c(=S)[nH]c(=S)[nH]n1 RJC02781 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccc(cc1)OC)O RJC02654 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)c2cccc(c2)C RJC02673 c1cc(ccc1OS(=O)(=O)CCN2C(=O)C3(CCCCCC3)NC2=O)Cl RJC02772 c1ccc(cc1)C(=O)Oc2ccc3c4ccccc4c(=O)oc3c2 RJC02774 CCOC(=O)Cc1csc(n1)NC(=O)CSc2nncn2C RJC02514 c1cc(sc1)/C=C/C(=O)Nc2cc(ccc2Cl)C(F)(F)F RDR02740 COc1cccc(c1C(=O)Nc2ccc(c(c2)Cl)Br)OC RDR02728 Cn1cnc(c1C(=O)O)n2oo2 RJC02780 CCOC(=O)CNC(=O)CSc1nnc(s1)SCC(=O)NCC(=O)OCC RJC02519 c1ccc(c(c1)NC(=O)/C=C/c2cccs2)F RDR02736 c1cc(sc1)/C=C/C(=O)Nc2ccc(cc2)F RDR02737 c1cc(sc1)/C=C/C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F RDR02738 c1cc(ccc1CCC(=O)c2c(cc(cc2O)O)O)O RJC02792 CC(C(=O)OC)Nc1c(=O)[nH]c(=S)[nH]n1 RJC02784 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C)NC(=O)c2cccc(c2)C RJC02674 Cn1cnnc1SCC(=O)Nc2ccc(cc2)Br RJC02505 Cc1c(ccc(c1OC(=O)c2ccc(c(c2)Cl)Cl)C(=O)C)OCc3ccccc3 RH00166 c1ccc(cc1)CC2C(=O)NC(=O)N2 RJC02813 CCOC(=O)Cc1csc(n1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)OCC RJC02564 Cc1ccc(cc1)Cn2c(c(cn2)Br)/C=N/NC(=S)NC(C)(C)C RF05503 CCc1cc2c(=O)c(c(oc2c(c1O)CN(C)C)C(F)(F)F)c3nc4ccccc4s3 RJC02783 Cc1ccc(c(c1)[N+](=O)[O-])OC(=O)/C=C/c2cccs2 RDR02750 Cn\1c2ccccc2s/c1=N/N=C3CCCCC3 RJC02961 c1cc(sc1)/C=C/C(=O)Oc2c(cc(cc2Br)Br)Br RDR02744 CCOC(=O)c1ccc(c(c1)Cl)OC(=O)/C=C/c2cccs2 RDR02754 c1cc(sc1)/C=C/C(=O)Oc2ccc(cc2)I RDR02758 CCOC(=O)c1c(n(nn1)c2cc(cc(c2)Cl)Cl)O SEW00003 c1cc(ccc1NC(=S)NCCO)I S01487 CCc1ccc(cc1)NC(=O)c2c(cccc2OC)OC RDR02729 CCCCc1c(nc(nc1O)SCC#C)O RDR02764 Cc1ccnc(c1)N(C2=NCC(S2)C)C(=O)Nc3cccc(c3)Cl RJC02657 c1ccc(cc1)C2c3c(c4ccccc4[nH]3)CC(N2)C(=O)O RJC02535 CCOC(=O)c1ccc(cc1)NC(=O)CSc2cccc(n2)C(=O)O RJC02524 CCOC(=O)c1ccc(cc1)OC(=O)/C=C/c2cccs2 RDR02755 c1cc(c(c(c1)Cl)OC(=O)/C=C/c2cccs2)Cl RDR02756 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCc1ccccn1 RJC02595 c1cc(c(c(c1)F)CNCC(COc2ccc(c(c2)Cl)Cl)O)N RDR03027 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)NC(=O)c3ccccc3 RJC02782 c1cc(sc1)C(=O)OCC(=O)c2ccc(cc2)[N+](=O)[O-] RDR02813 c1cc(ccc1c2csc(n2)c3c(cn[nH]3)Br)Cl RF05499 CC(C)(C)NC(=S)N/N=C/c1c(cnn1Cc2ccc(cc2)Cl)Br RF05501 c1ccc(cc1)CCn2c3ccc(cc3[nH]c2=S)C(F)(F)F RDR02789 c1cc(ccc1n2c(nnn2)SCC(=O)Nc3nc(cs3)CC(=O)O)O RJC02526 c1ccc2c(c1)C(c3ccccc3O2)C(=O)O RH00001 CCCCCCCCCCCC(=O)Nc1cc(ccc1OC)OC RG00117 c1ccc2c(c1)NC(=O)C(S2)CC(=O)Nc3ccc(cc3)C(F)(F)F RJC02534 CCCCCCNC(=O)C1c2ccccc2Oc3c1cccc3 RH00029 CC(=O)c1ccc(o1)/C=C/C(=O)Nc2ccccc2 RJC02785 CCCc1c(nc(nc1OC(=O)N(C)C)c2ccc(cc2)C)C RDR02768 c1cc(sc1)c2c(c(=O)[nH]c(n2)SCC(=O)c3ccc(cc3)OC(F)(F)F)C#N RH00009 c1ccc(cc1)CCNC(=O)/C=C/c2cccs2 RDR02739 c1ccc2c(c1)C(c3ccccc3O2)C(=O)NN RH00018 c1ccc2c(c1)nc(o2)SCC(=O)Nc3ccc(cc3)Br RJC02506 c1cc(c(cc1[N+](=O)[O-])C(=O)O)N2CCOCC2 RDR02718 c1ccc(cc1)C(=O)Nc2nc(cs2)CC(=O)O RJC02531 c1cc(ccc1C2=NCCO2)OCCO RJC02532 Cn1c(=O)c(c(n2c1nnc2)c3cccs3)C#N RH00022 C(CCO)CC1C(=O)NC(=O)N1 RJC02804 c1cc(sc1)/C=C/C(=O)Oc2ccc(cc2)[N+](=O)[O-] RDR02752 CC(C)(C)C(=O)Nc1ccc(cc1)c2cc3cc(ccc3o2)Cl RDR02753 CCOC(=O)CNC(=O)CSc1nnnn1c2ccc(cc2)O RJC02523 COc1ccc(cc1)NC(=O)Nc2ccc(cc2)Cc3ccc(cc3)NC(=O)Nc4ccc(cc4)OC RJC02837 C1CS(=O)(=O)CC1S(=O)(=O)Nc2c(c(c(c(c2F)F)F)F)F RJC02547 c1ccc2c(c1)c3ccc(cc3oc2=O)OC(=O)c4ccccc4Cl RJC02819 Cc1cc(ccc1Cl)C(=O)CSc2[nH]c(=O)c(c(n2)c3cccs3)C#N RH00007 Cc1cnnc2c1c3c(cc2)non3 RJC02826 c1ccc(cc1)c2cc3c(ccc4c3non4)nn2 RJC02827 C[C@@]1(CCC2C1(CCC3C2CC[C@@H]4C3(CCC5(C4)OCCO5)C)C)O NRB03695 CC(=O)OC1CCC2C1(CCC3C2CCC4C3(C(=O)CCC4)C)C NRB03697 CCCCOC(=O)C(C)Nc1c(=O)[nH]c(=S)[nH]n1 RJC02539 c1ccc(cc1)CCn2c3ccc(cc3nc2SCc4ccccc4)C(F)(F)F RDR02791 CC(=O)O.CC\1(CCCC/C1=N/O)NO RJC02822 CCCc1c(nc(nc1O)c2cccc(c2)C)C RDR02798 Cc1c(c(=O)[nH]c(=O)[nH]1)[N+](=O)[O-] RH00044 Cc1c(c2c(n1O)ccc3c2non3)C(=O)C RJC02828 c1cc(sc1)/C=C/C(=O)Nc2ccc(c(c2)Cl)Cl RDR02821 c1cc(c(c(c1)Cl)Cl)NC(=O)/C=C/c2cccs2 RDR02823 C1C2CC(C(=O)C1CC(C2=O)(Br)Br)(Br)Br RJC02957 c1cc(ccc1C/C(=N/O)/N)[N+](=O)[O-] S01213 COc1ccc(cc1OC)/C=C\2/C(=O)OC(=N2)c3ccccc3 S01235 c1cc(sc1)c2cc(c3cc(ccc3n2)Br)C(=O)O NRB03634 c1ccc(c(c1)OC(=O)/C=C/c2cccs2)Cl RDR02757 c1cc(sc1)c2c(c(=O)[nH]c(n2)SCC(=O)c3ccc(cc3)Br)C#N RH00006 CCCCc1c(nc(nc1O)SC)O RDR02763 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCc1ccccc1 RJC02571 CCOC(=O)Cc1csc(n1)NC(=O)C/C=C/C RJC02500 c1ccc(cc1)/C=C/C=C/2\C(=O)OC(=N2)c3ccccc3 S01257 COC(=O)C1c2ccccc2Oc3c1cccc3 RH00011 COc1ccc(cc1OC)CCNc2ccccc2[N+](=O)[O-] RDR02781 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)OC RJC02681 c1cc(nc(c1)SCC(=O)Nc2nc(cs2)CC(=O)O)C(=O)O RJC02525 c1ccc(cc1)CCC(=O)c2ccc3c(c2)OCCCCCO3 NRB03609 CC1=C(C(NC(=O)N1)c2ccc(cc2)OC)C(=O)OC RJC01411 CCOC(=O)C(C)Nc1c(=O)[nH]c(=S)[nH]n1 RJC02538 Cc1c(c(=O)[nH]nc1c2cccs2)C RH00049 Cc1ccc(cc1)CNc2nc(c(c(=O)n2C)C#N)c3cccs3 RH00032 c1ccc2c(c1)C(c3ccccc3O2)c4nnc(o4)c5cccc(c5)F RH00034 c1ccc2c(c1)C(c3ccccc3O2)C(=O)NNC(=O)c4cccc(c4)C(F)(F)F RH00035 c1cc(ccc1C#N)OCCO RJC02530 COc1cc(cc(c1OC)OC)/C=C\2/C(=O)OC(=N2)c3ccccc3 S01273 c1ccc2c(c1)C(c3ccccc3O2)C(=O)NNC(=O)c4cccc(c4)[N+](=O)[O-] RH00037 c1ccc2c(c1)C(c3ccccc3O2)c4nnc(o4)c5cccc(c5)[N+](=O)[O-] RH00038 Cc1c(c2c(n1OC)ccc3c2non3)C(=O)C RJC02829 c1ccc2c(c1)CCC/C(=C\c3ccc(cc3)C#N)/C2=O RJC01412 COc1ccc(cc1)NC(=S)N/N=C/c2ccc(c(c2)OC)O RDR00353 CN(CCC#N)c1ccc(cc1)/C=N/NC(=S)Nc2ccc(cc2)OC RDR00355 CCOc1ccc(cc1)C2C(=C(NC(=S)N2)C)C(=O)OC RJC01416 COc1ccc(cc1OC)CCn2c3ccc(cc3[nH]c2=S)C(F)(F)F RDR02790 CCOC(=O)c1c(n(c2c1c3c(cc2)non3)O)C RJC02820 COc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)OC RJC02687 CC(C)C(C(=O)Nc1ccc(cc1)Cl)N2C(=O)c3ccccc3C2=O RJC02550 c1ccc(cc1)C2=N/C(=C/c3ccccc3[N+](=O)[O-])/C(=O)O2 S01320 CC1CC(=O)NN=C1c2cccs2 RH00054 Cc1cc(c(c(c1)C)OC(=O)/C=C/c2cccs2)C RDR02806 c1cc2c(c3c1nncc3)non2 RJC02824 c1cc(sc1)/C=C/C(=O)Oc2ccc(cc2Cl)[N+](=O)[O-] RDR02807 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2[nH]c(=O)c(c(n2)c3cccs3)C#N RH00010 Cc1cccc(c1)C(=O)NC(C(=O)OC)(C(F)(F)F)O RJC02675 CCOC(=O)CSc1[nH]nc(c(=O)n1)NCC(=O)OC RJC02844 Cc1ccc(c(c1)[N+](=O)[O-])NC(=O)CC2C(=O)Nc3ccccc3S2 RJC02842 COc1ccc(cc1)NC(=O)/C=C/c2cccs2 RDR02820 c1cc(sc1)/C=C/C(=O)Nc2cc(ccc2Cl)Cl RDR02822 CCOC(=O)/C(=N\Nc1ccc(cc1)C(=O)C)/c2csc(n2)N RJC02552 CCOC(=O)/C(=N\Nc1cccc(c1)C(F)(F)F)/c2csc(n2)N RJC02554 COc1ccc(cc1)S(=O)(=O)NCCNC(=O)N2CCOCC2 RDR03014 Cc1cc2c(ccc3c2non3)nn1 RJC02825 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccc2 RJC02695 c1c(cc(cc1C(F)(F)F)N2C(=O)CCCC2=O)C(F)(F)F S10670 CC(=O)Nc1cccc(c1)Oc2c(c(c(c(c2F)F)F)F)F RJC02746 CCOC(=O)c1c(n(c2c1c3c(cc2)non3)OC)C RJC02830 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(nn2)OC RJC02567 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NNc1ccccc1 RJC02570 CCOC(=O)CCn1c(=S)n(c(n1)Nc2ccccc2)c3ccccc3 RJC02853 Cc1cc2c(c(n1)Sc3ccc(cc3)Cl)C(=O)NC2=O RF01129 CN(C)C(=O)Oc1c(c(cc(n1)c2cccs2)C(F)(F)F)C#N RF01131 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)C(=O)O RJC02563 c1ccc(cc1)/C(=N/NC(=O)c2ccccc2)/C(=O)O RJC02962 c1ccc(cc1)C2=NNC(=O)CC2 RH00053 Cc1ccc(cc1)S(=O)(=O)OS(=O)(=O)c2ccc(cc2)C SB01946 CCOC(=O)c1c(n(nn1)c2ccc(cc2)Cl)O SEW00002 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cc(on1)C RJC02565 CCCCCCCCOc1ccc(cc1)C(=O)c2ccc(cc2)F RJC02859 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2nc3ccccc3s2 RJC02683 Cn1ccnc1SCC(=O)Nc2ccc(cc2)Br RJC02510 C[C@@H]1CC2(C3CCC4(C(C3CCC2=CC1=O)CC[C@]4(C)O)C)C NRB03662 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=S)Nc2ccc(cc2)OC RDR00356 c1ccc2c(c1)Nc3c(nc4ccc(cc4n3)Cl)O2 RJC01447 c1ccc2c(c1)c(c(c(=O)[nH]2)Br)O RJC01448 CCC1(CC(=O)N(C(=O)C1)c2ccc(c(c2)Cl)F)C S10924 CC1CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)I S10928 CC1=NN(C2(C1C3C(C2)C3(C)C)O)C(=O)N RJC02740 COc1ccc(cc1Br)/C=C\2/C(=O)OC(=N2)c3ccccc3 S01303 Cc1ccnc(c1)N(C2=NCC(S2)C)C(=O)Nc3ccc(cc3)Cl RJC02658 c1cc(cc(c1)Cl)Cn2c(c(cn2)Br)C#N RF05469 c1cc(ccc1Cn2c(c(cn2)Br)C#N)Cl RF05470 CCCCCCCCCCCCCCCCC\1CCCC/C1=N/O RJC02848 c1c(c(c(o1)C(F)(F)F)C(=O)O)C(=O)O RJC02731 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3cccs3 RJC03015 c1ccc(c(c1)/C=C/[N+](=O)[O-])Cl S01393 COc1ccc(cc1)/C=C/[N+](=O)[O-] S01396 c1cc(ccc1C(=O)NC(=S)Nc2ccc(cc2)I)[N+](=O)[O-] S10935 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cc(ccn1)C RJC02592 c1cc2c(cc1Br)c(ncn2)O RH00197 c1ccc(cc1)Cc2cc(n[nH]c2=O)c3cccs3 RH00057 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCCc1cc2ccccc2[nH]1 RJC02597 c1ccc(cc1)COc2ccc(cc2Cl)Cc3cc(n[nH]c3=O)c4cccs4 RH00223 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(c2)C(F)(F)F RJC02682 c1ccc(cc1)Nc2nn(c(=S)n2c3ccccc3)CCC#N RJC02849 Cc1cc(ccc1Cl)C(=O)CSc2[nH]c(=O)c3cnn(c3n2)c4ccc(cc4)F RH00144 Cn1c(=O)c(c(nc1NCc2ccc(cc2)OC)c3cccs3)C#N RH00031 c1cc(c(cc1Cl)Cl)/C=C/[N+](=O)[O-] S01394 CCC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cc(ccn1)C RJC02591 c1cc(c(nc1)Oc2ccc(cc2Cl)Cl)C(=O)N RH00205 Cc1ccc(cc1)CNc2ccc3nnc(n3n2)c4ccccc4 RH00217 c1cc(c(cc1F)[N+](=O)[O-])/C=C/N2CCCC2 RH00214 COc1ccc(c(c1/C=C/[N+](=O)[O-])[N+](=O)[O-])OC RH00219 c1ccc(c(c1)CN2CCN(CC2)c3cccc4c3cc[nH]4)Cl RJC03025 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccccc3Br RJC03039 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3c(cccc3Cl)Cl RJC03040 c1cc(sc1)/C=C/C(=O)Oc2ccc(cc2)Cl RDR02743 CC(C)(C)c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccccc3 RJC03037 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)Cc4ccc(cc4Cl)Cl RJC03028 c1ccc(c(c1)CN2CCN(CC2)c3cccc4c3cc[nH]4)F.Cl.Cl RJC03032 c1cc(ccc1CSc2nnc(o2)CCCc3nnc(o3)SCc4ccc(cc4)Br)Br RJC02887 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3ccc(cc3)Cl RJC03046 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)Cc4ccc(c(c4)Cl)Cl.Cl.Cl RJC03048 c1ccc(cc1)C(=O)Nc2cccc(c2)Oc3c(c(c(c(c3F)F)F)F)F RJC02744 CCCCCCCCCCCC[NH+]1CCN(CC1)c2cccc3c2cc[nH]3.[Cl-] RJC03024 CCOC(=O)c1cnn2c1nc(c3c2cccc3)Nc4cc(ccc4OC)C RH00083 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(=O)CSc2nnnn2c3ccccc3 RJC02865 c1cc(c(cc1CSC(=N)N)Cl)Cl.Cl S01442 Cc1cc2c(cc1C)[nH]c(=S)[nH]2 S01443 COc1ccc(cc1OC)CCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJC03065 c1cc(c(c(c1)Cl)/C=C/[N+](=O)[O-])Cl S01398 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3Cl)Cl)/C(=O)O2 S01409 CC(=O)SC1CC(=O)N(C1=O)c2cc(cc(c2)Cl)Cl S10661 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3ccco3 RJC03018 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3ccccc3Br RJC03019 COc1ccccc1C2CCN(CC2)C(=O)c3cccs3 RJC03020 COc1ccc(cc1OC)CCNC(=O)C2CCCCC2 RJC03056 Cc1cc(c(cc1Cl)C)S(=O)(=O)NC2CCN(CC2)Cc3ccccc3 RJC03051 CC(C1CC1)N(c2ccccc2)C(=O)c3ccccc3Cl RJC02747 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(c(c2Cl)Cl)Cl RJC03061 Cc1cc(c(cc1Cl)C)S(=O)(=O)NCCc2ccc(c(c2)OC)OC RJC03062 Cn1c2c(c3c(c1=O)nc(o3)c4ccc(cc4)Cl)c(=O)n(c(=O)n2C)C RJC03109 CCOC(=O)C(C#N)c1c2ccccc2n(c(=O)c1[N+](=O)[O-])C RJC03110 c1cnccc1C2N(C(=O)CS2)CC3CC3 S10864 CC1CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)C(C)(C)C S10866 c1cc(ccc1COc2c3ccc(cc3ncn2)Cl)F RH00221 CC(=O)C(=NNc1ccc(cc1)C(F)(F)F)C(=O)C RH00218 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)c3ccccc3OC RJC03021 CCOC(=O)c1ccc(cc1)NC(=O)CCCN2CCN(CC2)Cc3ccccc3.Cl.Cl RJC03050 c1ccc2c(c1)C3C=CC2C=C3 RJC02978 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)Cl RJC03057 COc1ccc(cc1OC)CCNS(=O)(=O)c2cccc(c2Cl)Cl RJC03059 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)NCCc2ccc(c(c2)OC)OC RJC03064 C1CCC(CC1)C2C(CCC(=O)N2)[N+](=O)[O-] S10650 COc1ccc(cc1OC)CCNC(=O)c2ccco2 RJC03066 c1cc(oc1)/C=N/C2CCCCCCCCCCC2 S01516 c1cc(sc1)c2cc(c(=O)[nH]n2)CC3CCCCC3 RH00204 CCOC(=O)c1ccc(cc1)N2C(=O)C3CCC(CC3C2=O)C S10867 Cn1c2c(c3c(c1=O)nc(o3)c4ccc(c(c4)Cl)Cl)c(=O)n(c(=O)n2C)C RJC03111 CCOC(=O)C1(c2c(cc(cc2OC)OC)NC1=O)O RH00209 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3ccc(cc3)C#N RJC03052 CCOC(=O)c1cnn2c1nc(c3c2cccc3)N4CC(CC(C4)C)C RH00080 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccco3 RJC03043 COC(=O)c1ccccc1Sc2c(nc3n2cccc3)c4ccccc4 RJC02873 c1ccc(cc1)c2c(n3ccccc3n2)Sc4ccccc4[N+](=O)[O-] RJC02874 C1C2CC3(CC1CC(C2)(C3)C(C(C(F)(F)F)F)(F)F)C(=O)O RJC02875 Cc1ccc(cc1)/C=C/[N+](=O)[O-] S01418 c1cc(ccc1N2C(=O)CCCC2=O)F S10659 c1c(cc(cc1C(F)(F)F)NC(=O)CCCC(=O)O)C(F)(F)F S10666 Cc1cccc(c1N2C(=O)CC(C2=O)SC(=O)C)C S10674 CCOC(=O)c1cnn2c1nc(c3c2cccc3)Oc4cc(cc(c4)C(F)(F)F)C(F)(F)F RH00073 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Oc4ccc(cc4)NC(=O)c5ccc(cc5)C RJC02882 Cc1ccc(cc1)n2c(n[nH]c2=S)N RJC02866 COc1ccc(cc1)OC(=O)Nc2ccc(cc2)Cc3ccc(cc3)NC(=O)Oc4ccc(cc4)OC RJC02868 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3cccs3 RJC03044 c1c(cc(c2c1c(ncn2)O)Br)Br RH00195 Cc1ccc(cc1)S(=O)(=O)CC(COc2ccc(cc2)Br)O RDR03073 c1ccc(cc1)S(=O)(=O)CC(COc2ccc(cc2)Br)O RDR03074 Cc1cccc(c1)Oc2c(c(c(c(c2F)F)Oc3cccc(c3)C)F)F RJC02869 C1C=CC2CC(CC1C2=O)C(=O)O RJC02878 C/C(=N\O)/c1ccc(cc1)OC(=O)c2ccc(o2)Br RJC02880 C1=C(C(=O)C=C(C1=O)Br)CCCCCCC2=CC(=O)C(=CC2=O)Br RJC02977 CC(C)(C)c1cc(c(c(c1)C(C)(C)C)N=S=Nc2c(cc(cc2C(C)(C)C)C(C)(C)C)C(C)(C)C)C(C)(C)C RJC02883 C(Cc1nnc(o1)S)Cc2nnc(o2)S RJC02884 Cc1ccc(cc1C)n2c(=O)c3c(cccc3F)nc2SCC(OC)OC RH00182 CC(C1CC1)N(Cc2ccccc2)C(=O)CCC(=O)O RJC02881 c1ccc(cc1)CSc2nnc(o2)CCCCc3nnc(o3)SCc4ccccc4 RJC02888 C(CCCCc1nnc(o1)S)CCCc2nnc(o2)S RJC02885 COc1cc(c(cc1Br)OC)CCOCCOCCc2cc(c(cc2OC)Br)OC RJC02968 COc1ccc(c(c1)S(=O)(=O)CC(COc2ccccc2Cl)O)OC RDR03059 c1cc(ccc1OCC(CS(=O)(=O)c2ccc(cc2)Cl)O)Cl RDR03060 c1cc(c(cc1N2C(=O)C=CC2=O)Cl)Cl S01347 c1c(cc(cc1Cl)Cl)NC(=O)CCCC(=O)O S10678 c1cc(ccc1NC(=O)CCCC(=O)O)F S10657 c1cc(cc(c1)/C=N/N=C/c2cc(ccc2)[N+](=O)[O-])[N+](=O)[O-] S01491 c1ccc(cc1)CC(c2ccccc2)NCN3C(=O)c4ccccc4C3=O S01499 c1cc(ccc1NC(=O)/C=C/C(=O)O)Cl S01355 c1cc(c(cc1F)F)NC(=O)CCCC(=O)O S10664 CCOC(=O)c1cnn2c1nc(c3c2cccc3)Sc4ccc(cc4)C RH00071 CC(=O)SC1CC(=O)N(C1=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F S10662 Cc1ccc(cc1)S(=O)(=O)NCCc2ccc(c(c2)OC)OC RJC03058 COc1ccc(c(c1)CCOCCOCCc2cc(ccc2OC)OC)OC RJC02983 CC1=CC(=O)C(=CC1=O)CCCC2=CC(=O)C=CC2=O RJC02987 CCOc1ccc(cc1)NC(=S)NC(Cc2ccccc2)c3ccccc3 S01518 CNC(=O)Oc1ccccc1OCC(=O)NCc2ccccc2Cl RDR03042 Cc1c(cccc1Cl)N2C(=O)C=CC2=O S01339 COc1cccc(c1)NC(=O)/C=C\C(=O)O S01338 Cc1ccc(cc1)CNc2ccccn2 S01597 CCOC(=O)c1c(nc(n1c2ccc(cc2)C(C)C)SC)N SEW00052 CCOC(=O)c1c(n(nn1)c2ccc(cc2)C(C)C)O SEW00007 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(=O)CSc2nncn2c3ccccc3 RJC02864 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl RJC03053 COc1ccc(cc1OC)CCNC(=O)c2ccccc2Br RJC03055 Cc1ccc(cc1C)Oc2ccc3nnc(n3n2)c4ccccc4 RH00169 CCOC(=O)Cc1csc(n1)NC(=O)CSc2nnc(s2)SCC(=O)Nc3nc(cs3)CC(=O)OCC RJC02518 Cn1c(=O)c(c(nc1SC)c2cccs2)C#N RH00014 COc1ccc(cc1OC)CCNC(=O)c2cccc(c2)[N+](=O)[O-] RJC03067 c1ccc(cc1)n2c(c(c(n2)CC#N)C#N)N S01481 CCCCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCC(c1ccccc1)O RJC02584 Cc1cccc(c1NC(=O)CCCC(=O)O)C S10677 c1c(cc(cc1Cl)Cl)N2C(=O)CCCC2=O S10679 Cc1cccc(c1N2C(=O)CSCC2=O)C S10689 COC(=O)C/C(=N\Nc1cc(cc(c1)Cl)Cl)/C(=O)OC SEW00044 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC2CCN(CC2)Cc3ccccc3 RJC03047 c1ccc2cc(ccc2c1)CN3CCN(CC3)c4cccc5c4cc[nH]5 RJC03049 Cc1ccc(cc1C)n2c(=O)c3c(cccc3F)[nH]c2=S RH00172 Cc1cc(c(cc1OC)Cc2cc(c(cc2OC)C)OC)OC RJC02967 c1cc(ccc1S(=O)(=O)C2=CC34CCCCC3(C2)C=C(C4)S(=O)(=O)c5ccc(cc5)Cl)Cl RJC02976 CCOC(=O)c1ccc(cc1)NC(=O)CSCc2ccco2 RJC02527 COc1ccc(cc1)C2C3C(C(=O)N(C3=O)c4ccccc4)ON2c5ccccc5 RJC02833 c1ccc(c(c1)C2NC(CS2)C(=O)O)O RJC02835 c1cc(ccc1Cc2ccc(cc2)NC(=O)Oc3ccc(cc3)Br)NC(=O)Oc4ccc(cc4)Br RJC02838 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)c2cccc(c2)C(F)(F)F RJC02691 CCOC(=O)C(C(F)(F)F)(NC(=O)c1cccnc1)O RJC02692 CN(C)/C=N\c1ccc2nnc(n2n1)c3ccccc3 RH00183 CCOc1ccccc1C(=O)NC(C(=O)OCC)(C(F)(F)F)O RJC02693 CCOc1ccccc1C2=NC(N=C(O2)N(C)C)(C(F)(F)F)C(F)(F)F RJC02696 Cc1ccc(cc1)S(=O)(=O)OCCc2cc(ccc2OC)OC RJC02969 COc1ccc(c(c1)C(=O)CCCC(=O)c2cc(ccc2OC)OC)OC RJC02970 Cc1cc(oc1C)C=C2C(=O)CC(CC2=O)(C)C RH00188 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(c(c1)F)F RJC02580 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1nnc(s1)c2ccccc2 RJC02581 c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccc(cc3Cl)Cl RJC03002 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)Cl)Cl RJC02685 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccn2 RJC02686 c1ccc(cc1)c2nnc3n2nc(cc3)N/C=N/O RH00184 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)F)NS(=O)(=O)c2ccc(cc2)C RJC02704 CC1=CC(=O)C(=CC1=O)CCOCCC2=CC(=O)C(=CC2=O)C RJC02988 Cc1ccc(cc1Cl)N2C(=O)C=CC2=O S01336 COc1ccc(c(c1)OCCOCCOc2cc(ccc2OC)OC)OC RJC02984 Cc1ccc(cc1N2C(=O)C=CC2=O)Cl S01340 c1cc(c(c(c1)Cl)Cl)NC(=O)/C=C/C(=O)O S01346 c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccccc3Cl RJC03001 CCOC(=O)c1c(n(nn1)c2cc(cc(c2)Cl)Cl)Sc3ccccn3 SEW00013 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCc1cccnc1 RJC02599 Cn1c(=O)c(c(nc1NCc2ccccc2)c3cccs3)C#N RH00028 c1ccc(cc1)C2=N/C(=C\c3ccc4c(c3)OCO4)/C(=O)O2 S01296 c1ccc2c(c1)C(c3ccccc3O2)c4nnc(o4)c5cccc(c5)C(F)(F)F RH00040 Cc1cccc(c1)NC(=O)Nc2ccc(cc2)Cc3ccc(cc3)NC(=O)Nc4cccc(c4)C RJC02836 c1ccc2c(c1)cccc2Oc3ccc(cc3)S(=O)(=O)c4ccc(cc4)Oc5cccc6c5cccc6 RJC02718 CC(C1CC1)N(c2ccccc2)C(=O)c3ccccc3 RJC02719 c1cc(c(cc1OCC(CNCc2cc(cc(c2)Cl)Cl)O)Cl)Cl RDR03026 CC(=O)Oc1ccc(c2c1cc3c(ccc(c3c2)OC(=O)C)OC(=O)C)OC(=O)C RJC02997 CCN(CC)S(=O)C12CC3CC(C1)CC(C3)C2 RJC02736 c1ccc(cc1)N2C(=O)CC(C2=O)SCc3ccc(cc3)Cl S10651 Cc1ccc(cc1C)n2c(=O)c3c(cccc3F)nc2SC RH00178 c1ccc(cc1)c2nnc3n2nc(cc3)N RH00173 Cc1cc2c3c(c1)c(c(c(=O)n3CCC2)c4ccccc4)OCc5ccc(cc5)F RH00175 c1ccc2c(c1)C(c3ccccc3O2)C(=O)NNC(=O)c4cccc(c4)F RH00016 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C RJC02680 CCCCCCCCCCCCC\1CCCC/C1=N/O RJC02846 CC(=O)/C=C/1\C(c2ccccc2N1C)(C)C RJC02847 c1cc(ccc1S(=O)(=O)CC(COc2ccc(c(c2)Cl)Cl)O)Cl RDR03006 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)NC(=O)c3ccccc3 RJC03011 c1ccc(c(c1)CNC(=O)COc2ccccc2O)Cl RDR03031 CCOC(=O)c1cnn2c1nc(c3c2cccc3)Sc4cccc(c4)OC RH00070 COc1ccc(cc1)N2C(=O)CC(C2=O)SCc3ccc(cc3)Cl S10653 Cc1ccc(cc1)C(=O)Nc2cccc(c2)Oc3c(c(c(c(c3F)F)F)F)F RJC02741 CCOC(=O)C(C(F)(F)F)(Nc1cccc(n1)C)NC(=O)c2cccc(c2)C RJC02699 c1cc2c3c(c1)c(c(c(=O)n3CCC2)C4CCCCC4)O RH00168 Cc1cc2c3c(c1)c(c(c(=O)n3CCC2)c4ccccc4)O RH00170 c1cc(c(cc1Cl)Cl)N2C(=O)C=CC2=O S01348 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)NC(=O)c4ccc(cc4)C RJC02715 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)NC(=O)c4ccccc4Cl)Cl RJC02716 c1ccc(cc1)CN2CCC(CC2)NC(=O)C3CCC3 RJC03036 CCOC1=NC(N=C(O1)N2CCOCC2)(C(F)(F)F)C(F)(F)F RJC02573 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cc(ccc1C)F RJC02574 c1ccc2c(c1)cccc2NC(=O)/C=C/C(=O)O S01361 Cc1cccc(c1NC(=O)/C=C/C(=O)O)C S01371 Cc1cccc(c1N2C(=O)C=CC2=O)C S01372 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C)NS(=O)(=O)c2ccc(cc2)C RJC02705 CCOC(=O)C(c1ccc(cc1)F)(C(F)(F)F)NC(=O)OCC RJC02706 COc1ccccc1NC(=O)/C=C\C(=O)O S01337 COc1ccccc1N2C(=O)C=CC2=O S01342 CCOC(=O)C(C(F)(F)F)(Nc1cc(ccn1)C)NC(=O)c2cccc(c2)C RJC02701 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc(cc3)Cl RJC03038 c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3cccc(c3)[N+](=O)[O-] RJC03007 c1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl RJC03008 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3ccc(cc3Cl)Cl RJC03012 COc1ccccc1C2CCN(CC2)Cc3ccccc3 RJC03003 COc1c(cc(cc1)/C=N/N=C/c2cc(c(cc2)OC)OC)OC S01460 COc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccn2 RJC02689 c1ccc2c(c1)c3ccc(cc3oc2=O)OC(=O)c4ccco4 RJC02775 CCOC(=O)Cc1csc(n1)NC(=O)CSc2cccc(n2)C(=O)O RJC02521 COC(=O)C(c1c(cccn1)[N+](=O)[O-])C(=O)OC RH00042 COc1ccccc1C2CCN(CC2)CCCOc3ccc(cc3)Cl.Cl RJC03034 c1ccc(cc1)SC(=C(Sc2ccccc2)Sc3ccccc3)C(F)(F)F RJC02723 COC1C2C3CCC(C2C(O1)OC)C(C3)O RJC02994 COC(=O)C1(N=C(OC(=N1)N2CCCCC2)c3ccccc3)C(F)(F)F RJC02710 CC(C1CC1)N(c2ccccc2)C(=O)c3ccc(cc3)F RJC02712 c1cc(cc(c1)[N+](=O)[O-])CN2CCN(CC2)c3cccc4c3cc[nH]4 RJC03030 CC(=O)Oc1ccc(c2c1C(=O)c3c(ccc(c3C2=O)OC(=O)C)OC(=O)C)OC(=O)C RJC02998 Cc1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccccc3 RJC03000 Cn1c(=O)cc(c2c1n(c(=O)n(c2=O)C)C)N3CCCCC3 RJC03103 c1ccc(cc1)Oc2ccc(cc2)N3C(=O)C=CC3=O S01644 CCc1ccc2cc3c(c4c(n(c3=O)C)n(c(=O)n(c4=O)C)C)nc2c1 RJC03104 c1ccc(cc1)c2c(c3ccc(c(c3[nH]c2=O)Cl)Cl)O RJC03105 CCc1nc2c(o1)c3c(n(c2=O)C)n(c(=O)n(c3=O)C)C RJC03113 c1ccc(c(c1)N2CCC(CC2)CCCC3CCN(CC3)c4ccccc4[N+](=O)[O-])[N+](=O)[O-] S01698 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)C3CCCCC3 RJC03013 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3ccc(cc3)Cl RJC03016 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3cccc(c3)[N+](=O)[O-] RJC03017 CC(C)Oc1cccc(c1)NC(=O)c2ccccc2C(F)(F)F SEW00135 COc1ccc(cc1OC)CNc2ccccc2C(=O)O S01683 c1ccnc(c1)NC(=S)Nc2ccc(cc2)Cl S01684 c1ccnc(c1)NC(=S)Nc2ccc(cc2)I S01685 CC(C)Oc1cccc(c1)NC(=O)c2ccc(o2)[N+](=O)[O-] SEW00138 CSc1c(c(sn1)SC)C#N SEW00142 CSc1c(c(sn1)SC)C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW00147 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1)OC)/C#N S10880 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1)Cl)/C#N S10887 CCCOC(C(F)(F)F)(C(F)(F)F)NC(=O)CC RJC02579 COC(=O)N1C2CC(C1(C(F)(F)F)C(F)(F)F)C=C2 RJC02587 c1ccc(cc1)NC(=S)NCCO S01421 COc1ccc(c(c1OC)OC)Cc2cc(n[nH]c2=O)c3cccs3 RH00200 c1cc(c(nc1)Oc2ccc(cc2Cl)Cl)C#N RH00202 c1cc(sc1)c2cc(c(=O)[nH]n2)Cc3ccc(c(c3)Cl)Cl RH00199 CCOC(=O)c1c(nc(n1Cc2ccco2)SC)N SEW00112 Cc1ccccc1C(=O)Nc2cccc(c2)OC(C)C SEW00134 CCC1(CC(=O)N(C(=O)C1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C S10922 CCC(C)(CC(=O)Nc1ccc(cc1)Cl)CC(=O)O S10923 c1cc(ccc1NC(=O)COCC(=O)O)I S10929 c1cc(ccc1N2C(=O)COCC2=O)I S10930 CC(C)Oc1cccc(c1)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC SEW00137 CSc1c(c(sn1)SC)C(=O)N SEW00143 CC(C)(C)c1ccc(cc1)NC(=S)NC(=O)c2ccc(cc2)[N+](=O)[O-] S10937 Cc1nc2c(o1)c3c(n(c2=O)C)n(c(=O)n(c3=O)c4ccccc4)c5ccccc5 RJC03122 CCc1nc2c(o1)c3c(n(c(=O)n(c3=O)C)C)n(c2=O)c4ccccc4 RJC03124 CSc1c(c(sn1)SC)C(=O)NC(=O)Nc2ccc(cc2F)F SEW00146 Cn1ccnc1SCC(=O)Nc2ccccc2C#N RJC03128 CC(C)(C)OC(=O)/C(=C/C1CCCCC1)/C#N S10892 Cn1ccnc1SCC(=O)Nc2ccc(c(c2)Cl)F RJC03129 c1cc(ccc1N2C(=O)C=CC2=O)Cl S01357 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cn1)C)NC(=O)c2cccc(c2)C RJC02700 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)CCCOc4ccc(cc4)Cl RJC03029 c1ccc(cc1)CN2CCN(CC2)CCCOc3ccc(cc3)Cl.Cl.Cl RJC03033 c1ccc(cc1)C(=O)CC(CC(=O)c2ccccc2)c3cccc4c3cccc4 S01547 c1ccc(cc1)CN2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])SC4CCCCC4)/SC2=S RJC03167 c1ccc(cc1)CN2C(=O)/C(=C\c3cc(ccc3[N+](=O)[O-])Sc4ccccc4)/SC2=S RJC03170 COc1cc(c(cc1Br)Br)OC RJC03240 COC(=O)c1c(n(nn1)c2ccc(c(c2)Cl)F)C(=O)OC SEW00064 COC(=O)c1cc(n(n1)c2cc(cc(c2)Cl)Cl)O SEW00045 COc1ccc(cc1)c2c(n(nn2)c3ccc(cc3Cl)Cl)N SEW00040 c1cc(c(cc1F)F)N2C(=O)COCC2=O S10762 COC(=O)c1c(n(nn1)c2cc(cc(c2)Cl)Cl)C(=O)OC SEW00041 COC(=O)C/C(=N\Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C(=O)OC SEW00033 COC(=O)C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C(=O)OC SEW00034 Cc1cc(ccc1N2C(=O)C=CC2=O)I S01528 COc1ccc(cc1)c2c(n(nn2)c3cc(cc(c3)Cl)Cl)N SEW00039 CC1(CC(=O)N(C(=O)C1)c2cc(cc(c2)Cl)Cl)C S10801 CC(C)(CC(=O)Nc1ccc(cc1)Cl)CC(=O)O S10804 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl RJC03071 c1ccc(cc1)CN2CCN(CC2)C(=O)c3c(cccc3Cl)Cl RJC03073 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cccc(c3)[N+](=O)[O-] RJC03075 c1cc(ccc1C(=O)N2CCN(CC2)C(=O)C3CCCCC3)Cl RJC03089 CC1(CC(=O)N(C(=O)C1)c2ccc(cc2)Cl)C S10806 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)Cc3ccccc3 RJC03072 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc(cc3)C#N RJC03076 c1ccc(cc1)CN2CCN(CC2)C(=O)c3ccccc3Br.Cl RJC03079 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl RJC03077 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCN(CC2)Cc3ccccc3 RJC03078 CC(C)(CC(=O)Nc1cc(cc(c1)Cl)Cl)CC(=O)O S10800 CC(C)(CC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)CC(=O)O S10802 c1c(csc1C=C(C#N)C#N)Br S10772 c1c(csc1/C=C/[N+](=O)[O-])Br S10775 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3cccc(c3Cl)Cl.Cl RJC03081 C/C(=C\c1cc(cs1)Br)/[N+](=O)[O-] S10776 CC1(CC(=O)N(C(=O)C1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C S10803 COc1ccc(cc1OC)CCNC(=O)Cc2ccccc2F RJC03068 c1ccc(cc1)CN2CCN(CC2)C(=O)C3CCCCC3.Cl RJC03069 CC(=O)Nc1ccc(cc1)C2=N/C(=C/c3cc(cs3)Br)/C(=O)O2 S10780 CC(=O)Nc1ccc(cc1)NC(=O)C RH00100 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)c5c4CCCC5)O RH00102 c1ccc2c(c1)c(=O)[nH]c3n2ncc3C(=O)O RH00109 c1ccc(cc1)CN2C(=O)C3C(N(OC3C2=O)c4ccccc4)c5ccc(cc5)F RJC02912 c1cc(ccc1OCC(CS(=O)(=O)c2ccc(cc2)Cl)O)Br RDR03077 COc1ccc(cc1)C(CC(=O)c2ccccc2)CC(=O)c3ccccc3 S01543 CCN(CC)c1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccccc3 S01564 Cc1cc(c(cc1Cl)C)S(=O)(=O)N2CCN(CC2)Cc3ccccc3.Cl RJC03080 c1ccc(cc1)CN2CCN(CC2)C(=O)c3ccco3.Cl RJC03084 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3 RJC03086 c1ccc(cc1)CC(=O)N2CCN(CC2)Cc3ccccc3.Cl RJC03082 c1ccc(cc1)CN2CCN(CC2)C(=O)c3ccc(cc3Cl)Cl.Cl RJC03083 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3cccc(c3)C(F)(F)F RJC03085 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3)C(F)(F)F RJC03087 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3 RJC03088 c1c(cc(cc1C(F)(F)F)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3)C(F)(F)F RJC03091 CC1CC(=O)N(C1=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F S10731 CCOC(=O)c1c(n(nn1)c2cc(cc(c2)Cl)Cl)SCc3c(cccc3Cl)F SEW00011 CCOC(=O)c1c(n(nn1)c2cc(cc(c2)Cl)Cl)Sc3ccc(cc3)C SEW00012 CCOC(=O)c1c(nc(n1c2ccc(cc2)C(C)C)SC)NC(=O)C(C)C SEW00074 CC(C)c1ccc(cc1)N/C(=N/C#N)/SC SEW00050 CC(C)(C)c1cc(c(s1)C(=O)OC)CSc2ccc(cc2)Cl SEW00506 Cc1cc(c(cc1Cl)C)SCc2cc(sc2C(=O)OC)C(C)(C)C SEW00510 CC(C)(C)c1cc(c(s1)C(=O)OC)CSc2ccccn2 SEW00511 c1cc(cc(c1)[N+](=O)[O-])NC2[C@@H]([C@H]([C@@H]([C@H](O2)CO)O)O)O RJC03292 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4cc(ccc4Cl)Cl RJC03165 CCOC(=O)c1c(nc(n1c2ccccc2OC)SC)N SEW00080 CC1=C(C(NC(=O)N1C)c2ccc(cc2)OC)C(=O)O RJC02900 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3 RJC03090 c1cc(c(cc1Cl)Cl)C(=O)N2CCN(CC2)C(=O)C3CCCCC3 RJC03092 COc1cc(cc(c1OC)OC)C(CC(=O)c2ccccc2)CC(=O)c3ccccc3 S01546 c1cc(ccc1Oc2c(cc(cn2)Cl)Cl)Oc3c(cc(cn3)Cl)Cl RJC02909 CCOC1=NC(N=C(O1)N=C(SC)SC)(C(F)(F)F)C(F)(F)F RJC02601 CCOC(=O)c1ccc(cc1)NC(=O)CSCC(=O)O S10825 CCOC(=O)c1ccc(cc1)N2C(=O)CSCC2=O S10826 CCOC(=O)c1ccc(cc1)N2C(=O)CS(=O)(=O)CC2=O S10827 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cccc(c1)C(=O)C RJC02603 COC(=O)c1c(n(nn1)c2ccc(c(c2)Cl)F)O SEW00062 CC(C)(CC(=O)Nc1ccc(cc1)F)CC(=O)O S10807 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1OC)OC RJC02604 CCOC(=O)c1c(nc(n1c2ccccc2OC)SC)NC(=O)c3ccc(cc3)C(C)(C)C SEW00086 COc1ccc(c(c1)S(=O)(=O)CC(COc2ccc(cc2)Br)O)OC RDR03076 CCOC(=O)c1c(nc(n1c2ccccc2OC)SC)NC(=O)Nc3ccccc3 SEW00091 CN(C)S(=O)(=O)N(C)C RH00085 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCCc1ccc(c(c1)OC)OC RJC02600 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cccc(c1C)Cl RJC02605 CCOC(C(F)(F)F)(C(F)(F)F)NC(=O)Nc1ccc(cc1)Br RJC02606 CCOC(C(F)(F)F)(C(F)(F)F)NC(=O)Nc1ccc(cc1)F RJC02609 c1cc(ccc1S(=O)(=O)CC(COc2ccc(cc2Cl)Cl)O)Cl RDR03056 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)C#N RJC02616 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)N1CCCCC1 RJC02618 C1CC1NC(=S)SCCN.Cl RDR03078 C=CCNC(=S)SCCN.Cl RDR03079 CC1CC(CC(C1)(C)C)NC(=O)/C=C/C(=O)O S01511 COc1ccc(cc1)c2cn3ccccc3n2 RJC02877 CC1=C(C(N(C(=O)N1C)C)c2ccc3ccccc3c2)C(=O)OCc4ccccc4 RJC02898 CC1=C(C(NC(=O)N1C)c2ccc3ccccc3c2)C(=O)OCc4ccccc4 RJC02899 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/NCc3ccccc3)/C(=O)N2c4ccccc4 RJC03100 C/C(=C\C(=O)c1ccccc1)/NCC#N RH00095 CCC(=O)Nc1cc(ccc1C)F RH00098 CCC(=O)Nc1ccc(c(c1)Cl)F RH00099 CCOC(C(F)(F)F)(C(F)(F)F)NC(=O)Nc1ccccc1C(F)(F)F RJC02610 c1cc(ccc1n2c(c(cn2)C#N)N)F RH00101 c1cc(ccc1n2c(c(cn2)C(=O)N)N)F RH00103 CCC(=O)Nc1ccc(cc1OC)OC RH00104 CCOC(=O)C(C(=O)OCC)C(C(F)(F)F)(C(F)(F)F)NC(=O)Nc1ccc(cc1)C(F)(F)F RJC02614 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)C(C)C RJC02615 Cc1ccc(cc1C)n2c(=O)c3c(cccc3F)nc2SCC(C)C RH00179 C1CCC23CC(=O)CC2(C1)CC(=O)C3 RJC02979 C1=CC(=O)C(=CC1=O)CCCCCCC2=CC(=O)C=CC2=O RJC02981 C1=C(C(=O)C=C(C1=O)Br)CCCCCC2=CC(=O)C(=CC2=O)Br RJC02986 C12C(C(OC1C(=O)O)C(=O)O)C(C2(F)F)(F)F RJC02913 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCc1ccco1 RJC02625 CCOC(=O)NC(c1ccccc1)(C(F)(F)F)C(F)(F)F RJC02626 c1ccc(cc1)CSc2nnc(o2)CCCCCCCCc3nnc(o3)SCc4ccccc4 RJC02890 CCC(C)(CC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)CC(=O)O S10918 CCC1(CC(=O)N(C(=O)C1)c2cc(cc(c2)Cl)Cl)C S10921 CNC(=S)NNC(=S)NC1CCCCC1 RJC03148 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3ccc(cc3)F RJC03142 CCN(c1ccc(cc1)/C=N/N=C/c2ccc(cc2)N(CC)CC)CC S01571 CCc1nc2c(o1)c3c(n(c2=O)C)n(c(=O)n(c3=O)c4ccccc4)c5ccccc5 RJC03114 CC1CCC2C(C1)C(=O)N(C2=O)c3cc(cc(c3)Cl)Cl S10874 CC1CCC2C(C1)C(=O)N(C2=O)c3cccc(c3)C#C S10879 C1CCC(CC1)C(=O)N2CCN(CC2)C(=O)C3CCCCC3 RJC03093 c1cc(ccc1S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3)Cl RJC03095 C1=CC(=O)C(=CC1=O)CCC2=CC(=O)C=CC2=O RJC02982 CCOC(=O)C(c1ccc(cc1)NC(=O)c2ccc(c(c2)Cl)Cl)(C(F)(F)F)O RJC02711 CC1=[N+](c2cc(ccc2C1(C)C)C(F)(F)F)C.[I-] RJC02721 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)Cl)F RJC02639 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(c2)C(F)(F)F RJC02641 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cc(on2)C RJC02633 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)NCc2ccco2 RJC02644 CC1CN=C(S1)N(c2ccccc2)C(=O)Nc3ccc(cc3)Cl RJC02629 CC1=C(C(NC(=O)N1C)c2ccc(cc2)OC)C(=O)Nc3ccccc3 RJC02893 CC1=C(C(NC(=O)N1C)c2ccc3ccccc3c2)C(=O)OC(C)(C)C RJC02894 CC1=C(C(NC(=O)N1C)c2ccccc2)C(=O)OC(C)(C)C RJC02896 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)F RJC02631 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)NCCc2ccccc2 RJC02632 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cn2)C RJC02634 CCCCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NN1CCN(CC1)C RJC02583 c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccc4ccccc4c3 RJC03005 COC(=O)C/C(=N\Nc1ccccc1C(F)(F)F)/C(=O)OC SEW00032 c1cc(ccc1C(=O)CCC(=O)O)Cl RH00125 CCOC(=O)c1ccc2c(c1)sc(n2)N/C=N/O RH00127 CCOC(=O)c1ccc2c(c1)sc(n2)n3cccc3 RH00133 C1(C(C1C(=O)O)C(=O)O)C(=O)O RJC02914 C1C(C1(C(=O)O)C(=O)O)C(=O)O RJC02917 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C(=O)C RJC02647 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1OC)OC)NC(=O)c2ccccc2Cl RJC02649 Cc1ccnc(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2C RJC02648 c1cc(ccc1c2nnc3n2nc(cc3)N4CCCCC4)C(F)(F)F RH00112 c1cc(ccc1n2c3c(cn2)c(=O)[nH]c(n3)SCCO)F RH00114 COc1ccc2nnc(n2n1)c3ccc(cc3)C(F)(F)F RH00115 c1cc(ccc1c2nnc3n2nc(cc3)NC4CC4)C(F)(F)F RH00113 CCOC(=O)c1cnn(c1N)c2ccc(cc2)F RH00119 CCOC(=O)Cc1nnc(o1)c2ccccc2 RH00067 CCCCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ncccn1 RJC02577 CCc1c(c2ccccc2n(c1=O)C)O RJC03106 C1C2C=CC1C(C2C(=O)N)C(=O)O S10847 Cn1c2c(c(cc(=O)n2c3ccccc3)Nc4ccc(cc4)OC)c(=O)n(c1=O)C RJC03107 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)Nc3ccc(cc3)C(C)(C)C S10902 CCOC(=O)c1ccc2c(c1)sc(n2)N/C=C(\C#N)/C(=O)OCC RH00131 CCOC(=O)c1ccc2c(c1)sc(n2)NC=C(C(=O)OCC)C(=O)OCC RH00132 c1cc2c(cc1NC(=O)CSCC(=O)O)OCO2 S10833 c1cc2c(cc1N3C(=O)CSCC3=O)OCO2 S10834 CCOC(=O)c1ccc2c(c1)sc(n2)N/C=N/OC(=O)c3cccs3 RH00135 CC1CCC2C(C1)C(=O)N(C2=O)c3ccc(c(c3)Cl)F S10870 CC1CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)F S10875 Cc1ccc(cc1C)n2c(=O)c3c(cccc3F)nc2SCC=C RH00180 c1ccc2c(c1)cccc2N3C(=O)C=CC3=O S01362 COc1ccc(cc1OC)CCN2C(=O)C=CC2=O S01356 C(C(=O)N)(C(F)(F)F)C(F)(F)F RJC02724 c1cc(cc(c1)Cl)CSC(=N)N.Cl S01620 CC(=O)c1ccc(cc1)NCN2C(=O)c3ccccc3C2=O S01629 CCOC(=O)c1c(c2cccc3c2n(c1=O)CCC3)O RJC03099 Cn1c2c(c(cc(=O)n2c3ccccc3)Nc4ccc(cc4)F)c(=O)n(c1=O)C RJC03101 c1ccc(c(c1)N2C(=O)C=CC2=O)N3C(=O)C=CC3=O S01882 Cc1ccccc1C(=O)NNC(=S)NC S04407 CC(C)c1cccc(c1N2C(=O)C=CC2=O)C(C)C S04412 CNC(=S)NNC(=O)c1ccccc1Cl S04413 CC\1=NN(C(=O)/C1=C\c2ccc(o2)c3cccc(c3)[N+](=O)[O-])c4ccccc4 RJC03287 C#Cc1cccc(c1)NC(=S)NC(=O)c2ccc(cc2)[N+](=O)[O-] S10936 COc1ccc(cc1)/C=C(\C(=O)O)/NC(=O)c2ccccc2 S01722 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc(cc3)[N+](=O)[O-] RJC03041 Cc1ccc(c(c1)C)NC(=S)NCCO S01471 Cc1ccc(o1)C=C(C#N)C#N S11249 CC(=O)NC(Cc1ccccc1)C(=O)OC RJC03267 CC(C)/C(=N/NC(=O)c1ccc(cc1)Cl)/C(=O)O RJC03270 Cn1c(=O)c2cc3c(cc2c1=O)c(=O)n(c3=O)C RJC03275 Cc1cc(c(c(c1)C(C)(C)C)OC(=O)C(C)C)C(C)(C)C RJC03276 c1ccc(cc1)C(=O)CCCC(=O)c2ccccc2 RJC03277 CSc1nc(c(n1Cc2ccco2)C#N)N SEW00105 Cc1ccccc1NC(=S)Nc2ccccn2 S01678 CCOC(=O)c1c(noc1N)c2c(cccc2Cl)Cl SEW00100 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3cc(ccc3O)Cl)C2=O S11165 Cn1/c(=N/N=c/2\oc3c(n2C)cccc3)/oc4c1cccc4 RJC03254 CC1(CC1NC(=O)OCc2ccccc2)NC(=O)OCc3ccccc3 RJC03259 CC(C)(C)n1c(=S)[nH]nn1 RJC03265 Cc1cc(c(cc1CSC(=N)N)C)CSC(=N)N.Cl.Cl S01870 CC1=CC(=O)C(=CC1=O)Br RJC03273 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)O)C RJC02921 COc1c(nccn1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)F RJC02924 CCOC(=O)C1CCCCN1C(=O)c2c(nsc2SC)SC SEW00246 CCCCOC(=O)c1nnc(o1)c2ccc(cc2)Cl SEW00259 CCOC(=O)c1c(nc(n1Cc2cccs2)SC)NC(=O)C SEW00101 CCOC(=O)c1c(nc(n1Cc2cccs2)SC)NC(=O)c3ccc(o3)[N+](=O)[O-] SEW00102 CCc1ccc(cc1)NC(=S)NC(=O)c2c(onc2c3ccccc3Cl)C S10900 CCCCCCCCC/C=C/CC1CC(=O)N(C1=O)c2ccc(cc2)C(C)(C)C S10909 Cc1ccc(cc1C)Nc2n[nH]c(=S)s2 S01846 COc1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3N S01865 c1ccc(cc1)/C=N/c2ccccc2 S02104 Cc1ccc(cc1N2C(=O)CCCC2=O)Cl S11533 CC(C(=O)O)SCSC(C)C(=O)O S11659 C/C(=C\c1ccc2c(c1)OCO2)/[N+](=O)[O-] S11082 CCCCOC(=O)c1nnc(o1)c2ccc(cc2)[N+](=O)[O-] SEW00260 Cc1ccc(cc1)NC(=S)N(C)C S01811 c1ccc(cc1)C2=N/C(=C\c3ccsc3)/C(=O)O2 S11119 c1ccc(cc1)CN2C(SCC2=O)c3ccccc3O S11127 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1)C#N)/C#N S10894 CC1(SCCS1)c2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl RJC03134 c1ccc(cc1)/C=C/C(=O)O/N=C/c2ccc3c(c2)OCO3 RJC03137 COc1cc(cc(c1OC(=O)Cc2ccccc2)[N+](=O)[O-])C3SCCS3 RJC03138 CNC(=O)NNC(=N)c1ccccn1 SEW00366 c1c(cc(c2c1sc(n2)N3CCCCC3)Cl)Cl SEW00292 c1c(cc(c2c1sc(n2)N3CCCC3)Cl)Cl SEW00293 Cc1cc(c(cc1Cl)C)SCc2ncon2 SEW00296 c1ccc2c(c1)c(cs2)CC(=O)O S11080 CCOC(=O)/C(=C/c1ccc(o1)C)/C#N S11250 CN(C)C(=S)Nc1cccc2c1cccc2 S01848 c1cc(ccc1N2CCOCC2)N3C(=O)C=CC3=O S04434 Cc1cccc-2c1CCc3c2ccc(c3)C(C)C RJC03279 CC(C)(C)c1ccc(cc1)NC(=O)c2c(nsc2SC)SC SEW00241 COc1ccc(cc1)NC(=S)Nc2ccccn2 S01853 CC(=O)CC(=O)Nc1cc(ccc1Cl)Cl RJC03256 Cc1c(snn1)c2nc(no2)CSc3ccc(cc3)Cl SEW00462 CC(C)c1cccc(c1NC(=O)/C=C/C(=O)O)C(C)C S04409 CC1(CC2=C(C(=O)C1)Sc3ccccc3N2)C S11372 c1ccc(cc1)C2C(C2C(=O)NN)C(=O)NN RJC03262 Cc1ccc(cc1)C2C3C(NC(C(C3=O)C(N2)c4ccc(cc4)C)c5ccc(cc5)C)c6ccc(cc6)C RJC03264 Cc1cc(cc(c1)NC(=S)N(C)C)C S04420 c1ccc2c(c1)C(=O)C(C2=O)C(C[N+](=O)[O-])c3cccc(c3)Br S11433 C/C(=C\c1c[nH]c2c1cccc2)/[N+](=O)[O-] S11461 c1ccc2c(c1)C3CC(=NN3C2=O)c4ccc(s4)Cl S11466 Cc1ccc(cc1)S(=O)(=O)NN=C(C)C RJC03280 C1=C(C(=O)C=C(C1=O)Br)Br RJC03281 COc1c(nccn1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cc(cc(c3)Cl)Cl RJC02926 c1ccc2c(c1)C(=O)C(C2=O)C(C[N+](=O)[O-])c3c(cccc3Cl)F S11423 c1ccc2c(c1)C(=O)N(C2=O)N3C(=O)c4ccccc4C3=O S01910 c1ccc2c(c1)c(=O)[nH][nH]c2=O S01911 C1CCC(CC1)Nc2nnc(s2)S S01925 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1)F)/C#N S11472 CN(C)C(=S)NC1CCCCC1 S01812 Cc1c(c(=O)n(n1C)c2ccccc2)/N=C/c3ccc(o3)c4cccc(c4)[N+](=O)[O-] RJC03290 Cc1c(c(=O)n(n1C)c2ccccc2)/N=C/c3ccc(o3)c4ccc(cc4)[N+](=O)[O-] RJC03291 c1ccc2c(c1)Oc3ccccc3S2 RJC03297 CSc1ccc(cc1)C2C(=Cc3ccccc3O2)[N+](=O)[O-] S11422 CCOc1ccc(cc1)C2N([C@H](CS2)C(=O)O)C(=O)C RJC03302 COc1ccc(c(c1)/C=C/[N+](=O)[O-])OC S11460 C[C@H](c1ccccc1)NC(=O)C(=O)NC(C)c2ccccc2 RJC03244 c1ccc(cc1)/C=C/c2n[nH]nn2 RJF01475 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC23CC4CC(C2)CC(C4)C3 RJF01478 c1cc(ccc1N)S(=O)(=O)NC23CC4CC(C2)CC(C4)C3 RJF01481 c1ccc2c(c1)c(cs2)CSc3ccc(cc3)[N+](=O)[O-] S11328 c1cc2c(cc1Cl)nc(s2)N3CCCC3 SEW00231 C/C(=C\c1ccc(cc1)F)/[N+](=O)[O-] S11474 COc1ccc(cc1OC)CCNC(=S)NCCc2ccc(c(c2)OC)OC S01942 c1cc(oc1)CNc2c3c([nH]cn3)ncn2 RJC03303 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4c(cccc4Cl)Cl RJF00049 CC(C)(C)S(=O)(=O)/C(=C/c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C#N SEW00698 CNC(=S)N/N=C/c1cc(cc(c1)C(F)(F)F)C(F)(F)F SEW00702 CSc1c(c(sn1)SC)c2n[nH]nn2 SEW00322 CN(C)/C=N/NC(=O)Cn1nc(nn1)c2ccc(cc2)C(F)(F)F SEW00315 Cc1cccc(c1C)NC(=S)N(C)C S04418 Cc1c(snn1)c2nc(no2)CSc3ccccn3 SEW00463 c1ccc2c(c1)c(cs2)CSc3ccccc3[N+](=O)[O-] S11327 c1ccc(c(c1)S(=O)(=O)NNC(=N)c2ccccn2)Cl SEW00352 CC1CCN(CC1)c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] S01827 c1cc(c(cc1Cl)[N+](=O)[O-])N2CCCCC2 S01833 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)NNC(=N)c2ccccn2 SEW00353 CCCc1cc(=O)[nH]c(n1)SCc2nc(on2)c3c(nns3)C SEW00427 CN(C)C(=O)Oc1cccc(c1)NC(=O)c2cc(cc(c2)Cl)Cl SEW00302 CSc1nnc(s1)Nc2ccc(cc2Cl)Cl S11174 C1CC(CC=C1)C2C(CCC(=O)N2)[N+](=O)[O-] S11290 c1ccc2c(c1)C=C(C(O2)c3c(cccc3Cl)Cl)[N+](=O)[O-] S11301 Cc1cc(nc(n1)N2CCOCC2)OCCOC RJF01467 CC(C)c1ccc(cc1)NC(=S)NN(C)C S04445 Cc1cc(no1)NC(=O)NC(=O)c2c(nsc2SC)SC SEW00164 c1ccc(cc1)COc2cc(ccc2)/C=N/N=C/c3cc(ccc3)OCc4ccccc4 S01813 c1ccc(c(c1)C(F)(F)F)N/C(=N/C#N)/N2CCCC2 SEW00324 Cc1c(cccc1Cl)NC(=S)Nc2c(cccc2C(C)C)C(C)C S04442 c1ccnc(c1)C(=N)NNS(=O)(=O)c2ccc(cc2)Cl SEW00350 c1ccnc(c1)N2C(SCC2=O)c3ccc(cc3Cl)Cl S11430 CSc1c(c(sn1)SC)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW00239 CNc1nnc(s1)SCc2csc3c2cccc3 S10950 Cc1cc(nc(n1)NC(=O)C(C)(C)C)Nc2ccc(c(c2)Cl)F RJF01455 CC(C)c1cccc(c1NC(=S)Nc2cccc(c2)Cl)C(C)C S04429 c1cc(ccc1NC(=O)/C=C/C(=O)O)N2CCOCC2 S04433 CCOC(=O)c1ccc(cc1)NC(=O)NC(=O)c2c(nsc2SC)SC SEW00151 CSc1c(c(sn1)SC)C(=O)NC(=O)Nc2ccc(cc2)Cl SEW00153 CCOC(=O)C1=C(NC(=S)NC1c2c(cccc2Cl)F)C S11032 C/C(=N\N=C\1/NC(=O)C(S1)CC(=O)O)/c2csc3c2cccc3 S11067 C/C(=N\NC(=S)N)/c1ccncc1 S11073 CCOC(=O)C1=C(NC(=S)NC1c2cccc(c2)Br)C S11044 CC(C)Nc1nc2cc(ccc2s1)Cl SEW00232 C/C(=N\NC(=S)N)/c1ccccn1 S11074 CCOc1ccc(cc1)C(=O)/C=C/C(=O)Nc2ccc(cc2)F RJC03153 c1cscc1/C=C/[N+](=O)[O-] S10991 C/C(=N\NC(=O)N)/c1csc2c1cccc2 S11079 CCOC(=O)/C(=C/c1ccsc1)/C#N S10997 c1ccc(c(c1)N2C(=O)/C(=C\c3cc(ccc3SC4CCCCC4)[N+](=O)[O-])/SC2=S)Cl RJC03168 CCOC(=O)C1=C(NC(=O)NC1c2c(cccc2Cl)F)C S11030 Cc1cc(c(cc1Cl)Cl)SC2CC(=O)N(C2=O)c3ccc(cc3)F S11005 CCOC(=O)C1=C(NC(=S)NC1c2cccs2)C S11034 CCCCNC(=S)NCCCC S11041 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3cc(ccc3Cl)Cl RJC03172 COc1cc(cc(c1OS(=O)(=O)c2cc(ccc2Cl)Cl)[N+](=O)[O-])C3SCCS3 RJC03173 Cc1[n+](c2ccccc2s1)C.[I-] S11049 COc1ccc(c(c1)OC)/C=C/[N+](=O)[O-] S01886 COc1ccc(cc1/C=C/[N+](=O)[O-])Br S01894 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)S(=O)(=O)Nc2nccs2 RJC02623 C1CCCC(CCC1)NC(=S)SCCN.Cl RDR03081 c1cc(ccc1n2c3c(cn2)c(=O)[nH]c(=S)[nH]3)F RH00107 c1cc(ccc1SC2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl)Cl RJC03163 Cc1ccc(c(c1)C)N/N=C/Cc2nnnn2c3ccccc3 RJC03198 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(c(c3)Cl)Cl S02027 c1ccc2c(c1)NC(=O)C(S2)CC(=O)O S11679 CC(C)c1cccc(c1NC(=S)Nc2cccc(c2)SC)C(C)C S04431 Cc1ccc(cc1C)Cc2n[nH]nn2 RJF01470 CSc1nnc(o1)CCCCCCCCc2nnc(o2)SC RJC02889 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)N RJC02892 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NC(C)c1ccccc1 RJC02622 c1ccc(cc1)CNc2cc(=O)n(c(=O)n2c3ccccc3)c4ccccc4 RJC03116 CCCCNC(=O)NNC(=N)c1ccccn1 SEW00367 c1ccnc(c1)C(=N)NNC(=O)Nc2ccc(cc2)Cl SEW00369 CNC(=S)NNC(=N)c1ccccn1 SEW00371 CCC1(C(C(N=N1)(C)CC)O)C RJC02927 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3ccc(cc3)Br RJC03143 CCc1cccc(c1N2C(=O)CC(C2=O)Sc3ccccc3N)CC S02114 Cc1ccc(cc1NC(=S)NNC(=O)Cn2nc(nn2)c3cccc(c3)[N+](=O)[O-])Cl RJF01457 c1ccc(c(c1)C(F)(F)F)NC(=S)NNC(=N)c2ccccn2 SEW00373 c1ccc(cc1)/C=C/c2nc(no2)COc3ccc(cc3Cl)Cl SEW00377 CC(C)c1ccc(cc1)NC(=O)NC(=O)c2ncon2 SEW00391 CCOC(=O)COc1cccc(c1)NC(=O)c2ccccc2Cl SEW00225 Cc1ccc(cc1)n2c(nnn2)c3cnc(nc3c4ccc(cc4F)F)N RJC03200 c1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3 RJC03096 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ncccn2 RJC02636 Cc1ccc(cc1F)NC(=C2C(=O)c3ccccc3C2=O)C#N S10957 c1cscc1C=C(C#N)C#N S10996 CSc1c(c(sn1)SC)C(=O)NC(=O)N2CCOCC2 SEW00150 c1cc(cc(c1)Cl)CNC(=O)/C=C/C(=O)O S11150 CN(C)/C=C(\c1nnnn1c2ccccc2)/C(=O)c3ccc(c(c3)Cl)Cl RJC03191 CC1=CC(=O)C(=CC1=O)CCCCCC2=CC(=O)C(=CC2=O)C RJC03238 COc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])OC RJC03241 c1ccc2c(c1)c(cs2)CNC(=O)Nc3cc(cc(c3)Cl)Cl S11115 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)Cl RJC02638 c1cc(ccc1n2c3c(cn2)c(ncn3)O)F RH00118 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)c5c4CCCC5)OC(=O)c6cccs6 RH00120 c1ccc(c(c1)N2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Cl)/SC2=S)Cl RJC03171 CN(C)C(=S)Nc1ccccc1 S01810 c1cc(ccc1SCc2ncon2)Cl SEW00295 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2)Br)C S11043 c1ccc(cc1)CN2C(=O)c3ccccc3C2=O S01822 Cc1cc(c(cc1Cl)C)S(=O)(=O)Cc2cc(sc2C(=O)OC)C(C)(C)C SEW00516 Cc1ccc(cc1)S(=O)(=O)Cc2cc(sc2C(=O)OC)C(C)(C)C SEW00517 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)c5c4CCCC5)OC(=O)c6cccc(c6)C(F)(F)F RH00122 CCOC(=O)c1ccc2c(c1)sc(n2)/N=C/N(C)C RH00126 CCCOc1ccccc1N2C(=O)C3C(N(OC3C2=O)c4ccccc4)c5ccc(cc5)N(C)C RJC02923 CC1=CC(=O)C(=CC1=O)CCCCCCC2=CC(=O)C(=CC2=O)C RJC03239 c1cc(ccc1c2nnn(n2)CC(=O)NN)C(F)(F)F SEW00314 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=S)Nc3ccc(cc3F)F RJF01479 Cn1c2ccccc2c(c(c1=O)SC(=S)N(C)C)O RJC03397 CN(C)/C=C/1\C(=O)OC(=N1)c2ccccc2 RJC03399 CC(C)(C)c1cc(c(s1)C(=O)OC)CS(=O)(=O)c2ccccn2 SEW00518 CSc1c(c(sn1)SC)C(=O)NC(=O)Nc2c(cc(cc2F)F)F SEW00181 COc1ccc(c(c1)NC(=O)CSCC(=O)O)OC S10831 CC(C)(C)c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3ccc(cc3)Cl RJC03094 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1)N(C)C)/C#N S10893 COc1cc(cc(c1OC)OC)/C=N/c2ccccc2C(=O)O S01728 c1cc(cc(c1)Cl)NC(=O)CSCCSCC(=O)Nc2cccc(c2)Cl RJC03132 CSc1c(c(sn1)SC)C(=O)NC(=O)N2CCSCC2 SEW00152 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4ccco4 RJF00048 CSc1c(c(sn1)SC)C(=O)NC(=O)Nc2cccnc2 SEW00162 CSc1c(c(sn1)SC)C(=O)NC(=O)NNc2c(cc(cc2Cl)Cl)Cl SEW00168 Cc1ccc(o1)/C=C(\C#N)/C(=O)OC S11251 Cc1ccc(o1)/C=C/2\C(=O)OC(=N2)c3ccccc3 S11252 Cn1ccnc1SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F RJC03127 Cc1cc(cnc1NC(=S)Nc2ccc(cc2F)F)Br RJC03131 c1ccc(cc1)Oc2ccc(cc2)NCN3C(=O)c4ccccc4C3=O S01647 Cc1cc(c(cc1Cl)Cl)SCc2ncon2 SEW00294 CC(C)(C)NS(=O)(=O)NC(C)(C)C RJC03260 CSc1nnc(s1)NCc2cccc(c2)Cl S11177 CCCc1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccc4ccccc4c3 S11232 CC1CN(CC(O1)C)c2nc3c(s2)cc(cc3Cl)Cl SEW00297 CN(C)C(=O)Oc1cccc(c1)NC(=O)c2ccccc2C(F)(F)F SEW00300 CCOC(=O)Sc1ccc2ccccc2c1 S11233 c1ccc2cc(ccc2c1)SCCC(=O)O S11238 Cc1ccc(cc1N2C(=O)CCC(C2=O)(C)C)Cl S11530 c1cc(ccc1N2CC(=O)N(CC2=O)/N=C/c3ccc(o3)[N+](=O)[O-])I S14327 c1ccc(cc1)Oc2cccc(c2)C3C(=Cc4cc(ccc4O3)Cl)[N+](=O)[O-] S14129 CC1(N(N=C(S1)Nc2ccccc2)C(=O)C(C)(C)C)C S14133 C1CCCCCC2(CCCCC1)NNC(=S)NN2 RJC03321 CC(CC(=O)Nc1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl SEW00551 c1ccc2c(c1)C(=O)C(C2=O)C(C[N+](=O)[O-])c3c(cccc3Cl)Cl S11269 c1ccc2c(c1)C=C(C(O2)c3c(cccc3Cl)F)[N+](=O)[O-] S11304 COc1ccc(s1)/C=C/2\C(=O)OC(=N2)c3ccccc3 S11313 C1CCC(CC1)NC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)NC4CCCCC4 S01859 CC(C)(CC(=O)Nc1ccc(cc1Cl)Cl)CC(=O)O S11485 CC1(CC(=O)N(C(=O)C1)c2cc(ccc2Cl)Cl)C S11488 c1cc(c(cc1Br)Cl)NC(=O)/C=C/C(=O)O S01904 c1cc(c(cc1F)F)NC(=O)CCC(=O)O S11581 c1cc(ccc1C(N2CCOCC2)N3CCOCC3)Cl S11565 C/C(=N\N=C(NC(=O)C)NC(=O)C)/c1cccs1 RJC03314 CCOC(=O)/C(=C/c1ccc(cc1)[N+](=O)[O-])/C#N S11894 CC1(CC(=O)N(C(=O)C1)c2ccc(c(c2)Cl)Cl)C S11490 c1c(ccc(c1)Cl)/C=N/N=C/c2ccc(cc2)Cl S01980 c1cc(ccc1C(N2CCSCC2)N3CCSCC3)[N+](=O)[O-] S11555 Cc1c(cccc1Cl)N2C(=O)CC(C2=O)Sc3ccccc3N S02033 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)Cl)/C(=O)N2CCc4ccc(cc4)Cl S11516 CN(C)C(=S)Nc1ccc(cc1)Cl S01843 Cc1ccc(cc1C)NC(=S)N(C)C S01844 Cc1ccc(cc1Nc2nc3nc(cc(n3n2)NCC4CC4)C)Cl RJF01458 c1ccc(cc1)NC(=O)NNC(=O)Cn2nc(nn2)c3cccc(c3)[N+](=O)[O-] RJF01462 CC(C)(C)c1cc(c(s1)C(=O)OC)CS(=O)(=O)c2ccc(cc2)Cl SEW00508 C1(C(=O)NC(=O)N1)NC(=O)N RJC03317 CCO/C=C\1/C(=O)N(C(=S)S1)Cc2ccccc2 S02013 COc1c(c(ccc1)/C=N/N=C/c2c(c(ccc2)OC)OC)OC S02020 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)C(C)(C)C RJC03330 Cc1c(c(on1)c2ccco2)NC(=O)NN(C)C SEW00468 Cc1ccc(cc1N2C(=O)CC(CC2=O)(C)C)Cl S11528 CC(CC(=O)Oc1ccc(cc1)C(F)(F)F)S(=O)(=O)c2ccc(cc2)Cl SEW00565 CC1CC(=O)c2cc(ccc2S1)Cl SEW00543 c1cc(ccc1c2nnc(o2)/C(=N/O)/N)[N+](=O)[O-] SEW00270 c1c(cc(c2c1sc(n2)N3CCOCC3)Cl)Cl SEW00291 c1ccc(cc1)S(=O)(=O)NNC(=N)c2ccccn2 SEW00351 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)Cl)/C(=O)N2c4ccc(cc4)F S11514 c1ccc(cc1)C(=S)SCC(=O)O S01990 CCN1c2ccccc2C(=O)C(C1=O)(Cl)Cl RJC03343 CC(C)(C)c1ccc(s1)c2nc(no2)CSc3ccc(cc3)Cl SEW00631 Cc1ccc(cc1Cl)N2C(=O)CC(C2=O)Sc3ccccc3N S02030 CCO/C=C\1/C(=O)N(C(=S)S1)CCc2ccc(c(c2)OC)OC S02011 CC1C/C(=N\Nc2ccc(cc2)Br)/c3cc(ccc3S1)Cl SEW00547 CC(C)(CC(=O)Nc1cccc(c1Cl)Cl)CC(=O)O S11483 COc1cccc(c1)Nc2ccc(nn2)c3ccccc3 RJC03337 CC1c2c(nns2)-c3cc(ccc3S1(=O)=O)Cl SEW00595 CSc1c(c(sn1)SC)C(=O)N2CCSCC2 SEW00245 c1ccnc(c1)C(=N)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW00354 Cc1cccc(c1N2C(=O)/C(=N\O)/C(=N2)C(=O)OC)Cl SEW00365 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc3c(cc(=O)oc3c2)C(F)(F)F RJF00060 c1cc(cc(c1)C(F)(F)F)c2nc(on2)c3ccsc3 SEW01954 c1cc(ccc1N2CC(=O)N(CC2=O)/N=C/c3ccc(o3)[N+](=O)[O-])OC(F)(F)F S14326 c1c(cc(cc1Cl)Cl)NC(=O)c2csnn2 SEW00637 c1c(cc(cc1C(F)(F)F)NC(=O)NC(=O)c2csnn2)C(F)(F)F SEW00639 Cc1cc(n(n1)c2ccccc2)NC(=O)c3c(c4cccc5c4n(c3=O)CCC5)O RJC03348 c1ccc2c(c1)cccc2N3C(=O)CC(C3=O)Sc4ccccc4N S02041 CC(C)N(C(C)C)C(=O)NC(=O)c1csnn1 SEW00645 CC1C/C(=N\Nc2ccc(cc2)Br)/c3cc(ccc3S1(=O)=O)Cl SEW00578 CC1C/C(=N\Nc2cc(cc(c2)Cl)Cl)/c3cc(ccc3S1(=O)=O)Cl SEW00580 c1ccc(cc1)COc2cc(nnc2c3ccccc3)OCc4ccccc4 RJC03362 CC(C)Oc1cccc(c1)NC(=O)c2csnn2 SEW00635 c1cnccc1C(N2CCOCC2)N3CCOCC3 S11569 CC(CC(=O)O/N=C(/c1ccc(cc1)C(F)(F)F)\N)S(=O)(=O)c2ccc(cc2)Cl SEW00555 CC(CC(=O)O/N=C/c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl SEW00559 CC(CC(=O)O/N=C/c1ccc(cc1)C#N)S(=O)(=O)c2ccc(cc2)Cl SEW00560 Cc1cc(nc(n1)SCc2c(cccc2Cl)F)OC(=O)N(C)C RJF00084 COCCOc1ccc(cc1)NC(=O)c2ccc(cc2[N+](=O)[O-])Cl RJF00068 CC(CC(=O)O/N=C/c1c(cccc1Cl)Cl)S(=O)(=O)c2ccc(cc2)Cl SEW00562 Cc1ccc(cc1NC(=O)CCC(=O)O)Cl S11551 Cc1ccc(cc1N2C(=O)CCC2=O)Cl S11552 c1cc(ccc1C(N2CCOCC2)N3CCOCC3)[N+](=O)[O-] S11553 CC1C(=O)N(C(S1)c2cccnc2)CCc3ccc(cc3)OC S11654 CC1C(=O)N(C(S1)c2cccnc2)Cc3ccc(cc3)OC S11661 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3csc4c3cccc4 S11577 c1ccc(cc1)C(C2C(=O)Nc3ccccc3S2)C(=O)O S11681 c1cc(ccc1CSCc2ccc(cc2)Cl)c3csnn3 SEW00677 CC1C(=O)N(C(S1)c2cccnc2)c3ccc(cc3)Cl S11644 Cc1ccc(cc1NC(=O)C2C3CC(C2C(=O)O)C=C3)Cl S11536 Cc1ccc(cc1NC(=O)CSCC(=O)O)Cl S11538 Cc1ccc(cc1N2C(=O)CSCC2=O)Cl S11539 c1c(nns1)C(=O)NC(=O)N2CCCC2 SEW00646 Cc1cccc(c1)Nc2ccc(nn2)c3ccccc3 RJC03344 Cc1c(=O)nc2n(c1O)ccs2 RJC03350 c1ccc(cc1)CNc2cc(=O)c(n[nH]2)c3ccccc3 RJC03387 Cc1ccc(cc1NC(=O)/C=C\C(=O)O)Cl S11541 Cc1ccc(cc1N2C(=O)c3cccnc3C2=O)Cl S11543 CC(CC(=O)Oc1ccc(cc1)C#N)S(=O)(=O)c2ccc(cc2)Cl SEW00566 c1c(nns1)C(=O)NC(=O)N2CCOCC2 SEW00643 c1ccc(cc1)/C=C/SCC(=O)O S11590 Cc1c(nc2n(c1=O)c3ccccc3s2)O RJC03354 c1ccc(cc1)c2cc(c(c(=O)n2c3ccccc3)Sc4ccccc4)O RJC03395 c1ccc(c(c1)NC(=O)/C=C/C(=O)O)Cl S02046 Cc1c(c2ccccc2n(c1=O)C)O RJC03345 c1cc(ccc1NC(=O)c2csnn2)Cl SEW00634 c1ccc(cc1)c2c(c3cc(c(cc3[nH]c2=O)Cl)Cl)O RJC03369 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2cc(ccc2O)Cl S02045 CC1(c2ccccc2-n3c1cc(c(c3=O)Cc4ccccc4)O)C RJC03349 CCc1c(nc2n(c1=O)c3ccc(cc3s2)OC)O RJC03352 c1cc(c(cc1NC(=O)NC(=O)c2csnn2)Cl)F SEW00642 CCCCc1c(nc2n(c1=O)c3ccccc3s2)O RJC03358 Cn1c2ccccc2c(c(c1=O)Sc3ccccc3)O RJC03359 CCOC(=O)c1csnn1 SEW00615 c1cc(ccc1/C(=N/OC(=O)c2csnn2)/N)C(F)(F)F SEW00657 c1c(cc(cc1C(F)(F)F)NC(=O)c2csnn2)C(F)(F)F SEW00636 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1)[N+](=O)[O-])/C#N S11895 CN1C(CC(=N1)c2ccc3ccccc3c2)c4ccc(cc4)F S14222 CNNC(=S)Nc1cccc(c1)SC S04458 Cc1c(cccc1Cl)NC(=S)NNC S04460 c1ccc(cc1)c2ccc3nnnn3n2 RJC03376 c1ccc(cc1)CN2c3ccccc3C(=O)C(C2=O)(Cl)Cl RJC03377 c1ccc(cc1)c2cn3ccsc3n2 RJC03415 COc1ccccc1C(C[N+](=O)[O-])Sc2ccccc2N S11749 c1cc(c(cc1)Cl)/C=N/N=C/c2c(cccc2)Cl S02120 c1ccc(c(c1)NC(=O)NC(=O)c2csnn2)Cl SEW00641 CCc1cccc(c1NC(=S)NC(=O)c2ccccc2)CC S02115 CCc1cccc(c1NC(=S)N)CC S02116 c1c(nns1)C(=O)NC(=O)N2CCCCC2 SEW00644 c1c(cc(cc1Cl)Cl)N2C(=O)CCC2=O S11592 Cc1ccc(cc1)SC(=O)c2csnn2 SEW00681 c1ccc(cc1)c2c(cc3nnnn3n2)O RJC03380 c1cc(ccc1c2nc(on2)c3csnn3)C(F)(F)F SEW00661 Cc1ccc(cc1)c2csnn2 SEW00674 CCc1cccc(c1NC(=S)NN)CC S02118 CN(C)C(=S)NCCc1ccc(c(c1)OC)OC S02182 CN(C)CN1C(=O)c2ccccc2C1=O S02061 CCOC(=O)N/N=C/1\CCS(=O)(=O)c2c1cc(cc2)Cl SEW00602 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCOCCO RJC03159 Cc1c(nc(nn1)c2ccccn2)O SEW00402 C1CC2CC1CC2NC(=S)NN3C4CSC3CS4 SEW00410 c1cc(c(cc1Cl)Cl)OC(=O)c2csnn2 SEW00684 CC(C)(C)c1cccc(c1O)C2(C(=O)c3ccccc3C2=O)O S11843 CC1CC(CC(C1)(C)C)NC(=S)N(C)C S02069 Cc1cc(no1)NC(=O)NC(=O)c2csnn2 SEW00647 c1cnc(nc1)NC(=O)NC(=O)c2csnn2 SEW00648 c1ccc2c(c1)nc(s2)NC(=O)NC(=O)c3csnn3 SEW00649 c1ccc(cc1)/C=C/SCCC(=O)O S11610 c1cc(ccc1S(=O)(=O)/C(=C/c2ccc(cc2F)F)/C#N)Cl SEW00721 c1ccc2c(c1)C(=O)N(C2=O)CC#N S02063 CCOc1ccc(cc1)/C=C/[N+](=O)[O-] S02064 c1cc(ccc1c2ncc3c(n2)-c4cc(ccc4SC3)Cl)C(F)(F)F SEW01850 c1ccc2cc(ccc2c1)CC(=O)N/N=C/c3ccccc3[N+](=O)[O-] RJC03301 Cc1cc(=O)n2c3ccccc3[nH]c2n1 RJC03304 Cc1c(c(n(n1)c2ccccc2)O)Cc3c(cccc3Cl)Cl RJF00040 c1ccc(cc1)C(=O)NC(=S)Nc2ccccn2 S02172 CC1(CC2=C(CC3(CN2)C(=O)CC(CC3=O)(C)C)C(=O)C1)C S02154 CC1C(=O)N(C(S1)c2ccc(cc2)C(F)(F)F)c3ccc(cc3)C(F)(F)F S11730 COC(=O)/C(=C/c1ccc(cc1)C(F)(F)F)/C#N S11736 Cc1cc(ccc1C(F)(F)F)/C=C\2/C(=O)OC=N2 S11739 c1ccc2c(c1)c(=O)oc(n2)c3ccc(cc3)Cl S02126 c1ccc2c(c1)c(=O)oc(n2)c3cccc(c3)Cl S02127 CC1C(=O)N(C(S1)c2cccnc2)c3ccc(cc3F)F S11645 CC(C(c1ccc(cc1)F)Sc2ccccc2N)[N+](=O)[O-] S11817 Cc1ccc(cc1C)NC(=S)NCCO S01747 CC(=O)c1csc2c1cccc2 S10994 COc1ccc(cc1OC)CCNC(=S)NN S02162 c1ccc(cc1)c2nc(on2)c3csnn3 SEW00659 c1cc(ccc1c2nc(on2)c3csnn3)Cl SEW00660 CC(C)(CC(=O)Nc1cccc(c1)Cl)CC(=O)O S11481 CC(C)(C)S(=O)(=O)/C(=C/c1ccc(cc1F)F)/C#N SEW00718 c1cc2c(cc1Cl)C(=O)CCS2 SEW00590 CNC(=O)NNC(=O)c1csc(n1)c2ccc(cc2Cl)C(F)(F)F SEW01935 COc1ccc(cc1)NC2CC(=O)N(C2=O)c3ccc(cc3)OC S14274 c1ccc(cc1)Cn2c3ccccc3c(c(c2=O)Cl)O RJC03381 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc4c(cc(=O)oc4c3)C(F)(F)F RJF00012 C1CCC(CC1)n2c(nnn2)S S02145 c1ccc(cc1)Cn2c(nnn2)S S02146 CCOC(=O)/C(=C/c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C#N SEW00708 c1cc(ccc1CSc2ccc(cc2)Cl)c3csnn3 SEW00710 Cc1ccc(c(c1)C)NC(=S)Nc2ccccn2 S01808 Cc1ccc(cc1C)NC(=S)Nc2ccccn2 S01809 Cc1ccccc1C(=O)/C(=C/N(C)C)/c2nnnn2c3ccc(cc3)Cl RJC03195 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2F)F)/C#N SEW00719 c1ccnc(c1)S(=O)(=O)/C(=C/c2ccc(cc2F)F)/C#N SEW00720 c1[nH]c2c(n1)c(ncn2)NCCO RJC03312 CC(=O)NC(Cc1c[nH]c2c1cccc2)C(=O)O RJC03313 CC(C)(C)c1ccc(cc1)NC2=CC(=O)N(C2=O)c3ccc(cc3)C(C)(C)C S14277 COc1ccc(cc1OC)CCNC(=S)NC(=O)c2ccc(cc2Cl)Cl S02166 CC1CC(CC(C1)(C)C)NC(=S)NC(=O)c2ccc(c(c2)Cl)Cl S02167 c1c(cc(cc1Cl)Cl)OC(=O)c2csnn2 SEW00683 c1cc(ccc1CS(=O)(=O)c2ccc(cc2)Cl)c3csnn3 SEW00711 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)NCCc3ccc(c(c3)OC)OC S02183 CC(C)N1CN(C(=S)SC1)C(C)C S01973 Cc1ccc(cc1)C(=O)/C(=C/N(C)C)/c2nnnn2c3ccc(cc3)Cl RJC03196 CN(C)C(=O)Oc1cccc(c1)NC(=O)c2c(cccc2F)F SEW00303 CC1(C2CCC1(C(C2)(C#N)Nc3ccccc3)C)C RJC03507 c1ccc2c(c1)cc(o2)CSC(=N)N.Cl S11866 Cc1ccc(cc1[N+](=O)[O-])NC(=O)c2ccccc2F S11493 COc1ccc(c(c1)[N+](=O)[O-])NC(=O)c2cc(cc(c2)Cl)Cl S11494 CC(C)(CC(=O)Nc1ccc(c(c1)Cl)Cl)CC(=O)O S11489 Cc1c(c2cc(cc(c2[nH]c1=O)Cl)Cl)O RJC03390 Cc1c(c(c(=O)n(c1c2ccccc2)c3ccccc3)Sc4ccccc4)O RJC03393 COc1ccc(cc1)/N=C/2\c3ccccc3NC2=O S11704 c1ccc2c(c1)c(cs2)CNC(=O)/C=C\C(=O)O S11716 CCOC(=O)N/N=C/c1cc(cc(c1)C(F)(F)F)C(F)(F)F SEW00701 c1cc(ccc1CCNC(=N)N[N+](=O)[O-])Cl S11825 CC1C/C(=N\Nc2cc(cc(c2)Cl)Cl)/c3cc(ccc3S1)Cl SEW00545 Cc1ccc(cc1[N+](=O)[O-])NC(=O)c2ccc(cc2)C(F)(F)F S11480 COc1c(cc(cc1)Br)/C=N/N=C/c2c(ccc(c2)Br)OC S01901 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2cc(ccc2OC)Br S01902 CCCCCCCCCCCCCCCCCCC(C(C)(C)C)(C(C)(C)C)O RJC03179 c1cc(oc1)CN2C(=O)CSC2=S S01954 C1CCC(CC1)N2CN(C(=S)SC2)C3CCCCC3 S01956 CC1C/C(=N\Nc2ccc(cc2)I)/c3cc(ccc3S1(=O)=O)Cl SEW00581 CCOC(=O)N/N=C/1\CC(S(=O)(=O)c2c1cc(cc2)Cl)C SEW00584 CC1(CC(=O)N(C(=O)C1)c2cccc(c2)Cl)C S11482 c1ccc(cc1)/C=N/NC(=N)N/N=C/c2ccccc2 RJC03328 CC(C)(C)c1cc(c(s1)C(=O)OC)CSc2ccccc2 SEW00509 CCOC(=O)C1=C(NC(=O)NC1)C S11879 Cc1cccc(c1O)C2(C(=O)c3ccccc3C2=O)O S11882 c1cc2c(cc(=O)oc2cc1O)C(F)(F)F RJF00002 c1ccc(cc1)c2cc(c(c(=O)n2c3ccccc3)S(=O)(=O)c4ccccc4)O RJC03394 c1ccc(cc1)c2ccc(nn2)Nc3ccccc3 RJC03335 c1ccc(cc1)c2ccc(nn2)Nc3ccc(cc3)Cl RJC03336 CCN(CC)C(=O)Oc1ccc2c(cc(=O)oc2c1)C(F)(F)F RJF00013 Cc1ccc(cc1C)/N=C\2/NCCS2 S01748 c1ccc(c(c1)N)SC(CC(=O)c2ccc(cc2)Cl)c3ccsc3 S11134 Cc1ccc(cc1)C(=O)CC(c2ccsc2)Sc3ccccc3N S11135 c1cc(ccc1Cn2nc(nn2)c3ccc(cc3)Cl)F RJF01553 COC(=O)c1c(ccs1)c2ccc(o2)c3ccn(n3)C(=O)c4ccc(cc4)Cl SEW01908 CCn1cc(c(=O)c2c1ccc(c2)C(F)(F)F)C(=O)OC SEW00796 c1cc(ccc1c2csnn2)NS(=O)(=O)c3ccc(cc3)Cl SEW00797 c1ccc(c(c1)Cn2nc(nn2)c3ccc(cc3)Cl)F RJF01559 CCCC1=NNC(=O)C1CC=C RJF01560 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)Cl)OCC(=O)NN RJF01564 CC(C)(C)NC(=S)N(C)C S04512 c1ccc(c(c1)CN2CC(CC2=O)C(=O)O)Cl SEW00806 c1ccc2c(c1)cccc2/C=N\N=C(N)N RJC03325 c1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3N S02003 c1csc2c1-c3c(cnc(n3)C45CC6CC(C4)CC(C6)C5)CS2 SEW01898 CCOC(=O)Cn1c(=O)cc(c2c1CCCC2=O)C(F)(F)F SEW01903 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)O RJF01538 c1cc(ccc1c2csnn2)NC(=O)c3ccc(cc3)Cl SEW00789 c1cc(ccc1c2csnn2)NS(=O)(=O)c3ccc(cc3F)F SEW00798 CS(=O)(=O)c1c(c(sn1)S(=O)(=O)C)C(=O)N SEW00805 CCc1cccc(c1NC(=C2C(=O)c3ccccc3C2=O)C#N)C S12033 c1cc(ccc1c2csnn2)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW00800 c1cc(c(cc1CN2CC(CC2=O)C(=O)O)Cl)F SEW00808 c1cc(cc(c1)Cl)CNC(=O)C2C3C=CC(C2C(=O)O)O3 S12003 CC(CC(=O)Nc1ccccc1)S(=O)(=O)c2ccc(cc2)Cl SEW00550 CC(CC(=O)Nc1cccc(c1)C#C)S(=O)(=O)c2ccc(cc2)Cl SEW00552 c1cc(sc1)C(=O)Nc2ccc(cc2)c3csnn3 SEW00795 c1ccc(c(c1)C(=O)Nc2ccc(cc2)c3csnn3)C(F)(F)F SEW00788 c1cc(c(c(c1)Cl)C(=O)Nc2ccc(cc2)c3csnn3)F SEW00790 c1cc(ccc1c2csnn2)NC(=O)c3cc(cc(c3)Cl)Cl SEW00791 CCc1cccc(c1N2C(=O)C=CC2=O)C S12019 CCc1cccc(c1N2C(=O)CC(CC2=O)(C)C)C S12040 CCc1cccc(c1N2C(=O)c3cccnc3C2=O)C S12044 c1cc(ccc1C(F)(F)F)N2C(=O)CSC2=O S12056 CN(C)/C=C\1/C(=O)N(C(=O)S1)c2ccccc2 S12055 CCCc1ccc(cc1)N2C(=O)C3CCC(CC3C2=O)C S12234 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)F)c4cc(cc(c4)C(F)(F)F)C(F)(F)F RJF00112 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)F)c4ccc(c(c4)Cl)F RJF00113 c1c(cc(cc1Cl)Cl)NC(=N)NC(=N)N.Cl RJF00091 c1ccc(cc1)c2c(nc3n(c2=O)c4ccccc4s3)O RJC03360 CC1(CC(=O)N(C(=O)C1)c2ccc(cc2Cl)Cl)C S11486 CCc1cccc(c1N2C(=O)CCCC2=O)C S12028 CCc1cccc(c1N2C(=O)CC(C2=O)C)C S12042 c1ccc(cc1)N2C(=O)CSC2=O S12054 c1cc2c(cc1[N+](=O)[O-])c(=O)oc(n2)c3ccc(cc3Cl)Cl S02435 c1ccc2c(c1)C(=O)NC(N2)C3CCCCC3 S12243 Cc1c(c(nc(n1)c2ccccn2)O)Cc3c(cccc3Cl)Cl RJF00096 COCCOc1ccccc1NC(=S)SCCSC(=S)Nc2ccccc2OCCOC RJF00101 COCCOc1ccccc1NC(=O)c2ccc(cc2[N+](=O)[O-])Cl RJF00070 c1ccc(cc1)N/N=C/c2ccc(cc2)Cl S02311 c1ccc(cc1)CN2CN(C(=S)SC2)Cc3ccccc3 S01960 c1cc2c(cc1Cl)C(=O)CCS2(=O)=O SEW00597 CCOC(=O)/C=C/1\CSCC(N1)C(=O)OCC SEW00604 CCCc1c(c(nc(n1)c2ccccn2)O)C(C)C=C RJF01666 c1ccc(c(c1)c2nc3c(cc(cc3Br)Br)c(=O)o2)F S02268 COc1cccc(c1OC)/C=C\2/C(=O)N(C(=S)S2)CCc3ccc(c(c3)OC)OC S02317 Cc1c(cc(c(c1)/N=C/c2ccc(cc2)Cl)/N=C/c3ccc(cc3)Cl)C S02304 Cc1ccc(cc1)N2C(c3ccccc3C2=O)C(=O)c4cc(c(cc4O)C)C S11889 CCn1c(=O)c2ccccc2[nH]c1=S S02205 Cc1c(c(on1)C)c2nc(no2)CSc3ccc(cc3)Cl SEW00762 c1ccc(cc1)/C=C/S(=O)(=O)CC(=O)O S11599 COc1ccc2c(c1)sc3n2c(=O)c(c(n3)O)c4ccccc4 RJC03357 Cc1c(c(on1)C)c2nc(no2)CSc3ccccn3 SEW00764 CCNC(=S)NNc1ccccc1 S02279 c1ccc2c(c1)c(=O)oc(n2)c3ccc(cc3)F S02265 Cc1cc(c(c(c1)C2(C(=O)c3ccccc3C2=O)O)O)C S11886 Cc1ccc(cc1)N2C(c3ccccc3C2=O)C(=O)c4cc(ccc4O)OC S11893 COC(=O)/C(=C/c1ccc(cc1)[N+](=O)[O-])/C#N S11896 c1cc(ccc1c2cnco2)NC(=O)c3ccc(cc3)Cl SEW00754 CC(=O)c1ccc(o1)c2ccsc2C(=O)OC SEW01856 CC1=NN(C(=O)C1CC(=C)C)S(=O)(=O)c2ccccc2Cl RJF01583 COc1cccc(c1OC)/C=C/[N+](=O)[O-] S14295 CCOC(=O)CNc1cc(cc(c1)Cl)Cl S14311 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)OCC(=O)C RJF01594 Cc1c(snn1)C(=O)Nc2ccc(cc2)c3cnco3 SEW00760 Cc1ccc(cc1)SCc2nc(on2)c3c(noc3C)C SEW00765 c1cc(c(cc1NC(=N)NC(=N)N)Cl)F.Cl RJF00044 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4ccccc4Cl RJF00046 Cc1c(=O)n(c2ccccc2n1)C SEW00767 c1cc(ccc1c2cnco2)NC(=O)c3cc(sc3)[N+](=O)[O-] SEW00758 c1ccc(cc1)NC2=CC(=O)N(C2=O)c3ccccc3 S14273 c1cc(ccc1NC2CC(=O)N(C2=O)c3ccc(cc3)Cl)Cl S14275 COc1ccc(cc1OC)CCN2C(=O)/C(=C/c3ccccc3Cl)/SC2=S S02314 Cc1ccc(cc1)c2cnco2 SEW00783 COc1ccc(cc1OC)CCN2C(=O)/C(=C\c3cccc4c3cccc4)/SC2=S S02316 C/C(=C\c1ccc(cc1)[N+](=O)[O-])/[N+](=O)[O-] S11898 CCOC(=O)c1ccc(cc1)NC(=S)NC(=O)c2ccccc2 S02240 c1ccc(c(c1)C(=O)O/N=C(/CCS(=O)(=O)c2ccc(cc2)Cl)\N)Cl SEW00737 Cc1c(c[nH]n1)c2nc(sn2)Nc3ccccc3 SEW01865 COc1ccc(cc1OC)CC(=O)NCc2cccc(c2)Cl S11966 CCOc1cc(=O)oc2c1cccc2 S11989 CC(C)c1ncc2c(n1)-c3cc(ccc3SC2)Cl SEW01851 CC(C)(C)c1ccc(cc1)OC(=O)c2csnn2 SEW00750 c1ccc(cc1)C(=O)Nc2ccc(cc2)c3cnco3 SEW00753 c1cc(c(cc1/N=C\2/N(C(=O)CS2)c3ccc(c(c3)Cl)F)Cl)F RJF00163 c1ccc(cc1)SC2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl S14290 c1ccc(cc1)SC2CC(=O)N(C2=O)c3ccc(cc3)F S14291 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)O RJF01573 c1cc(ccc1c2csnn2)[N+](=O)[O-] SEW00752 c1cc(ccc1c2cnco2)NC(=O)c3ccc(cc3F)F SEW00755 C/C(=N\Nc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])/c2ccc(o2)c3ccsc3C(=O)OC SEW01860 C/C(=N\NC(=O)N)/c1ccc(o1)c2ccsc2C(=O)OC SEW01864 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)Cl)OCC(=O)O RJF01580 Cc1c(cn(n1)S(=O)(=O)c2ccc(cc2)Cl)c3nc(sn3)Nc4ccccc4 SEW01872 Cc1c(cn(n1)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3nc(sn3)Nc4ccccc4 SEW01873 Cc1ccc(cc1)N2C(c3ccccc3C2=O)C(=O)c4ccc(cc4O)C S11885 Cc1ccc(c(c1C)O)C2(C(=O)c3ccccc3C2=O)O S11890 c1cc(cnc1)CNC(=S)Nc2ccc(c(c2)Cl)F RJF00165 c1cc(c(cc1CNC(=O)Nc2cc(sc2)[N+](=O)[O-])Cl)F SEW00834 c1ccc(cc1)N2C(=O)/C(=C/c3ccc(cc3)F)/SC2=O S12078 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)O RJF00016 CNNC(=S)Nc1ccc(cc1)Cl S04459 CNNC(=S)Nc1cccc(c1)C(F)(F)F S04461 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)Cl)O RJF00021 Cc1c2cc(c(cc2oc(=O)c1Cc3c(cccc3Cl)Cl)O)Cl RJF00028 c1cc(ccc1C(=O)O/N=C(/CCS(=O)(=O)c2ccc(cc2)Cl)\N)Cl SEW00736 CCCc1cc(=O)oc2c1ccc(c2)O RJF01525 CCc1ccc(c(c1)C2(C(=O)c3ccccc3C2=O)O)O S11847 Cc1ccc(cc1)N2C(c3ccccc3C2=O)C(=O)c4cc(ccc4O)C S11876 c1cc(ccc1C(=O)O/N=C(/CCS(=O)(=O)c2ccc(cc2)Cl)\N)[N+](=O)[O-] SEW00738 CN(C)NC(=S)Nc1cccc(c1)C(F)(F)F S04448 CN(C)NC(=S)Nc1cccc(c1Cl)Cl S04473 CC1(N(N=C(S1)Nc2ccccc2)C(=O)c3ccc(cc3)C(C)(C)C)C S14137 CCOc1cccc2c1OC(C(=C2)[N+](=O)[O-])c3ccc(cc3)F S14161 Cc1ccc(cc1)NC(=S)NN(C)C S04475 c1ccc(cc1)C2=N/C(=C\c3ccccc3Cl)/C(=O)O2 S02121 c1ccc2c(c1)c(=O)oc(n2)c3ccc(c(c3)Cl)Cl S02128 c1cc(ccc1/C(=N/OC(=O)c2csnn2)/N)Cl SEW00655 Cc1c(c(no1)c2ccccc2Cl)c3nc4ccccc4c(=O)o3 S02187 CC(C)(C)c1ccc(s1)c2nc(no2)CSc3ccccn3 SEW00628 COC(=O)c1c(ccs1)c2ccc(o2)C=C(C(=O)OC)C(=O)OC SEW01883 CN(C)NC(=S)Nc1cccc(c1)SC S04446 Cc1cc(cc(c1)/N=C/c2cc(ccc2O)Br)C S04508 Cc1cc(cc(c1)/N=C/c2cc(cc(c2O)Cl)Cl)C S04509 CN(C)NC(=S)Nc1ccc(cc1)OC S04455 C/C(=N\Cc1ccccc1)/c2ccc(c(c2O)O)O S04456 c1cc(cc(c1)F)/C=C/[N+](=O)[O-] S14126 c1ccc2c(c1)ccc3c2C=C(C(O3)c4ccc(cc4)F)[N+](=O)[O-] S14136 CC(=O)N1c2ccccc2C(=O)C1=O S04457 COC(=O)c1c(ccs1)c2ccc(o2)c3cc[nH]n3 SEW01906 COC(=O)c1c(ccs1)c2ccc(o2)c3ccn(n3)C(=O)c4cccs4 SEW01907 COC(=O)c1c(ccs1)c2ccc(o2)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl SEW01910 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=S)NC RJF01499 CCCc1cc(nc(n1)SCc2c(cccc2Cl)F)O RJF01504 c1cc(ccc1/C=C/[N+](=O)[O-])[N+](=O)[O-] S11897 COc1ccc(cc1OC)CCNC(=S)NC(=O)c2ccccc2 S02101 CCc1cccc(c1NC(=O)/C=C/C(=O)O)CC S02111 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=N/NC(=O)N SEW00703 Cc1c(c2ccccc2o1)CCOC(=O)c3ccc(cc3)C(F)(F)F S11671 c1ccc(cc1)N2C(CC(=N2)c3ccc4ccccc4c3)c5ccc(cc5)F S14216 CCOC(=O)C1C(CC(=CC1=O)c2ccc3ccccc3c2)c4ccc(cc4)F S14217 Cc1cc(nc(n1)SCc2c(cccc2Cl)Cl)Nc3ccc(cc3F)F RJF01487 CCCC1=NNC(=O)C1Cc2c(cccc2Cl)Cl RJF01524 CN(C)/C=C/1\CSc2c(ccs2)C1=O SEW01897 c1cc(ccc1NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)S(=O)(=O)NC34CC5CC(C3)CC(C5)C4 RJF01495 Cc1cc(nc(n1)SCc2c(cccc2Cl)Cl)Nc3ccc(cc3)F RJF01496 COc1cccc2c1OC(C(=C2)[N+](=O)[O-])c3ccc(cc3)F S14147 c1cc(cc(c1)C(F)(F)F)/C=C/[N+](=O)[O-] S14149 CCCc1cc(nc(n1)SCc2c(cccc2Cl)Cl)O RJF01505 c1cc(ccc1C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Oc4ccc(cc4)NC(=O)c5ccc(cc5)Cl)Cl RJC03408 CCCc1c(c(nc(n1)SC)O)Cc2c(cccc2Cl)Cl RJF01526 CCOC(=O)c1c(nc(s1)c2ccc(cc2Cl)C(F)(F)F)C SEW01920 CN(C)NC(=S)Nc1cccc(c1)Cl S04447 CCCC1=NNC(=O)C1Cc2c(cccc2Cl)F RJF01532 Cc1ccc(cc1C)NC(=S)NN(C)C S04449 Cc1cc(c(c(c1)C)NC(=S)NCCO)C S02482 Cc1cc(c(c(c1)C)NC2=NCCS2)C S02483 Cc1cc(c(c(c1)C)Nc2nnc(s2)S)C S02486 CCCCC(C(=O)N/N=C/c1ccc(cc1)OC)C(=O)N/N=C/c2ccc(cc2)OC S04763 c1ccc(c(c1)/C=N/c2ccc(cn2)Cl)O S04829 CCCc1c(nc(nc1O)SCc2c(cccc2Cl)F)C RJF00080 Cc1c(cn(n1)C(=O)c2ccccc2)c3nc(sn3)Nc4ccccc4 SEW01869 Cc1c(cn(n1)C(=O)C)c2nc(sn2)Nc3ccccc3 SEW01870 CCCc1cc(nc(n1)SCC(=O)c2ccc(cc2)Cl)O RJF01519 c1cc(ccc1NC2CC(=O)N(C2=O)c3ccc(cc3)F)F S14268 c1c2c(cc(=O)oc2cc(c1Cl)O)C(F)(F)F RJF00020 CC1CC(CC(C1)(C)C)NC(=S)NC(=O)c2ccc(cc2Cl)Cl S02171 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc4c(cc(=O)oc4c3)C(F)(F)F RJF00057 c1ccc(cc1)N2C(CC(=N2)c3ccc4ccccc4c3)c5ccc(cc5)C(F)(F)F S14215 CCOC(=O)C1C(CC(=CC1=O)c2ccc3ccccc3c2)c4ccc(cc4)C(F)(F)F S14218 CC(C)(C)C(=O)CSc1nc2ccccc2c(=O)n1c3ccccc3 S14241 CC(=O)Cc1nc(sn1)Nc2ccccc2 SEW01855 C/C(=N/NC(=S)Nc1ccc(cc1Cl)Cl)/c2ccc(o2)c3ccsc3C(=O)OC SEW01863 Cc1cc(nc(n1)SCc2c(cccc2Cl)Cl)Nc3ccc(c(c3)Cl)F RJF01486 c1cc(ccc1C(=O)Nc2ccc(cc2)S(=O)(=O)NC34CC5CC(C3)CC(C5)C4)Cl RJF01488 c1ccc(cc1)CN2CCC3(CC2)NC(=O)c4ccccc4O3 S14246 CC1(OC(=O)C(=Cc2ccc(cc2OC)OC)C(=O)O1)C S14253 c1ccc(cc1)NNC(=S)Nc2ccccc2C(F)(F)F S04528 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3cccc(c3)F S04536 c1ccc2c(c1)C(=O)N(C2=O)CNc3ccc(cc3)N4CCOCC4 S04546 c1cc(ccc1/N=C/c2cc(ccc2O)Br)S(=O)(=O)Nc3nccs3 S04548 CCCc1cc(=O)oc2c1ccc(c2)OC(=O)/C=C/c3cccs3 RJF01536 CC(C)(CC(=O)O)Sc1ccc(cc1)Cl SEW00725 c1ccc(c(c1)C(=O)O/N=C(/CCS(=O)(=O)c2ccc(cc2)Cl)\N)C(F)(F)F SEW00735 Cc1cccc(c1)NC(=S)NCCc2ccccn2 S02196 c1ccc2c(c1)c(cs2)CSCc3c(cccc3Cl)Cl S11559 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=C/[N+](=O)[O-] SEW00707 Cc1ccc2c(c1)c(=O)n(c(n2)SCC(=O)C(C)(C)C)c3ccccc3 S14242 CN(CCC#N)c1ccc(cc1)/C=N/c2ccc(cc2)Cl S04516 CCc1ccc(cc1)/N=C/c2ccc(cc2)N(C)CCC#N S04517 CN(CCC#N)c1ccc(cc1)/C=N/c2ccc(cc2)OC S04520 Cc1ccc(cc1)n2c(=O)c3ccccc3nc2SCC(=O)C(C)(C)C S14243 CCCC1=NN(C(=O)C1Cc2c(cccc2Cl)F)C(=O)C(C)(C)C RJF01555 CC1(OC(=O)C(=Cc2cccc(c2OC)OC)C(=O)O1)C S14255 COc1ccc2c(c1)cc(c(=O)o2)C(=O)O S14261 CC1(OC(=O)C(=Cc2cc(c(cc2OC)OC)OC)C(=O)O1)C S14262 CC1=NNC(=O)C1Cc2ccc(cc2)F RJF01570 CC(C)(C)NC(=S)Nc1cc(ccc1Cl)Cl S04526 c1cc(ccc1CSc2ccc(cn2)C(F)(F)F)c3ncns3 SEW01930 c1cc(cc(c1)F)N2C(=O)C=CC2=O S04534 Cc1ccc(cc1)C(C[N+](=O)[O-])Sc2ccc(cc2)N S14250 c1cc(ccc1C2N(C(=O)CS2)c3ccc(cc3)C(F)(F)F)C(F)(F)F S11729 CCOC(=O)/C(=C/c1ccc(cc1)C(F)(F)F)/C#N S11732 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1)C(F)(F)F)/C#N S11735 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)C(F)(F)F)/C(=O)O2 S11738 Cc1ccc(cc1NC(=O)CCCC(=O)O)Cl S11531 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccccc3F S04582 CCOC(=O)COc1ccc2c(c(c(=O)oc2c1)Cc3c(cccc3Cl)Cl)C RJF01556 c1cc(ccc1OC/C(=N\OC(=O)c2ccsc2)/N)Cl SEW01952 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/OC(=O)c3cccs3 SEW01926 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)NN RJF01571 CCOc1ccc(cc1)/N=C/c2ccc(cc2)N(C)CCC#N S04518 c1cc(cc(c1)NC(=O)/C=C/C(=O)O)C(=O)O S02636 Cc1cc(ccc1NC(=S)Nc2ccc3ccccc3c2)Br S04893 CNNC(=S)Nc1ccc(cc1)OC S04469 CCc1ccc(cc1)NC(=S)NN(C)C S04474 CCOc1ccc(cc1)NC(=S)NCc2cccnc2 S04493 CC1(OC(=O)C(=Cc2ccc(c(c2OC)OC)OC)C(=O)O1)C S14263 CCCC1=NN(C(=O)C1Cc2c(cccc2Cl)F)C(=O)/C=C/c3cccs3 RJF01557 COc1ccc(cc1OC)CCN2C(=O)CSC2=S S01951 CCOc1ccc(cc1)N2CN(C(=S)SC2)c3ccc(cc3)OCC S01957 COc1cc2cc(c(=O)oc2cc1OC)C(=O)O S14270 CCN1CCC2(CC1)NC(=O)c3ccccc3O2 S14271 CCCCC(C(=O)N/N=C/c1ccc(cc1)C(C)C)C(=O)N/N=C/c2ccc(cc2)C(C)C S04760 CCCCC(C(=O)N/N=C/c1ccc(cc1)C)C(=O)N/N=C/c2ccc(cc2)C S04762 Cc1cc(no1)/N=C/c2cc(cc(c2O)Cl)Cl S04777 CCCc1cc(=O)oc2c1ccc(c2)OS(=O)(=O)c3cc(c(cc3Cl)Cl)C RJF01541 CCCc1cc(=O)oc2c1ccc(c2)OC(=O)c3ccccc3Cl RJF01545 c1ccc(cc1)C2=Nc3ccccc3SC(C2)c4c(cccc4Cl)Cl S02357 c1ccc(cc1)C(=O)CC(c2cccc(c2)[N+](=O)[O-])Sc3ccccc3N S02359 c1cc(ccc1c2c(nco2)C#N)C(F)(F)F SEW01983 CCn1cc(c(=O)c2c1ccc(c2)C(F)(F)F)C(=O)N/N=C/c3ccccc3Cl SEW00812 CCn1cc(c(=O)c2c1ccc(c2)C(F)(F)F)C(=O)NNC(=S)Nc3ccc(cc3)Cl SEW00813 CCn1cc(c(=O)c2c1ccc(c2)C(F)(F)F)C(=O)NNC(=S)Nc3ccccc3C(F)(F)F SEW00814 CCCc1cc(=O)oc2c1ccc(c2)OC(=O)c3ccc(cc3)Cl RJF01533 CCCc1c(c(nc(n1)SC)O)C RJF01534 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)OCC RJF01566 CCOC(=O)COc1ccc2c(c(c(=O)oc2c1)Cc3c(cccc3Cl)F)C RJF01569 c1c(cc(cc1Cl)Cl)NC(=S)NCCO RJF00150 c1c(cc(cc1Cl)Cl)/N=C\2/N(C(=O)CS2)c3cc(cc(c3)Cl)Cl RJF00162 CCn1cc(c(=O)c2c1ccc(c2)C(F)(F)F)C(=O)NNC(=O)C SEW00830 c1cc(ccc1c2nnc(s2)N)[N+](=O)[O-] S02659 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(o2)c3ccsc3C(=O)OC)C(=O)OC SEW02070 c1ccc(cc1)c2cc(oc2c3ccccc3)c4ccc(cc4)Br S14399 c1cc(c(cc1F)F)NC(=S)NNC(=O)Cn2nc(nn2)N3CCOCC3 RJF00236 Cc1c(c(c(c(c1[N+](=O)[O-])C(C)(C)C)[N+](=O)[O-])C)C(=O)Cn2nc(nn2)N3CCOCC3 RJF00239 c1c(cc(cc1Cl)Cl)NC(=S)NNC(=O)Cn2nc(nn2)N3CCOCC3 RJF00242 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OCC(=O)NN RJF01572 c1cc(ccc1CN2CC(CC2=O)C(=O)O)C(F)(F)F SEW00809 COc1cc(=O)oc2c1cccc2 S11995 c1cc(cc(c1)Cl)CNC(=O)Nc2cc(sc2)[N+](=O)[O-] SEW00833 c1ccc(cc1)C(=O)CC(c2ccc(cc2)[N+](=O)[O-])Sc3ccccc3N S02364 c1ccc(cc1)C2=Nc3ccccc3SC(C2)c4ccc(cc4)[N+](=O)[O-] S02367 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2ccccc2Cl)N S12159 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2ccco2)N S12165 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2c(cccc2Cl)F)N S12166 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N\c3ccc(c(c3)Cl)F RJF00171 c1cc(c(cc1F)F)NC(=S)NCCCN2CCOCC2 RJF00174 Cc1c(c(on1)/C=C/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] SEW00815 Cc1c(c(on1)/C=C/c2cc(cc(c2)Cl)Cl)[N+](=O)[O-] SEW00816 CCc1cccc(c1NC(=O)/C=C/C(=O)O)C S12018 CCc1cccc(c1NC(=O)CCCC(=O)O)C S12024 COc1ccc(cc1)NC2=CC(=O)N(C2=O)c3ccc(cc3)OC S14279 CCOC(=O)CNc1cc(cc(c1)C(F)(F)F)C(F)(F)F S14312 Cc1ccc(cc1)C(C[N+](=O)[O-])c2c(n(c(=O)n(c2=O)C)C)N S12161 CCn1cc(c(=O)c2c1ccc(c2)C(F)(F)F)C(=O)NNC(=O)C(Cl)(Cl)Cl SEW00831 c1cc(cnc1)CNC(=O)Nc2cc(sc2)[N+](=O)[O-] SEW00832 c1cc(sc1)CNC(=O)Nc2cc(sc2)[N+](=O)[O-] SEW00835 C1COCCN1c2nnn(n2)CC(=O)NN RJF00235 c1cc(c(cc1/C=C/[N+](=O)[O-])Cl)Cl S12121 Cc1cc(c(cc1C)Nc2nnc(s2)S)C S02404 c1cc(c(cc1Cl)Br)NC(=O)/C=C\C(=O)O S02407 c1cc(c(cc1Cl)Br)N2C(=O)C=CC2=O S02409 CCOC(=O)/C(=C(\C)/N)/N=N/c1ccccc1 S12134 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2ccc(cc2Cl)Cl)N S12157 COCCOc1ccc(cc1)NC(=S)N2CCOCC2 RJF00072 Cc1cc(nc(n1)SCc2c(cccc2Cl)Cl)O RJF00106 Cc1c(c(nc(n1)SC)O)Cc2c(cccc2Cl)F RJF00108 c1cc(c(cc1Nc2ncnc(n2)N)Cl)F RJF00103 COc1cc(cc(c1OC)OC)C=C(C#N)C#N S02457 CCOC(=O)N/N=C(\C)/c1ccccc1O SEW00840 c1cc(c(c(c1)Cl)CSc2nc(cc(n2)O)C(F)(F)F)F RJF00201 Cc1c(c(on1)C)c2nc(no2)CS(=O)(=O)c3ccc(cc3)Cl SEW00846 Cc1nnc(s1)Nc2cccc(c2)F RJF00210 Cc1c(c(nc(n1)N2CCSCC2)O)CC=C RJF00226 CN(C)C(=S)Oc1ccc2c(cc(=O)oc2c1)C(F)(F)F RJF00228 c1cc(ccc1CNC(=O)c2ccc(cc2)Cl)c3csnn3 SEW00850 c1cc(c(c(c1)Cl)Cn2nc(nn2)N3CCCCC3)F RJF00327 c1ccc(c(c1)/N=C/c2cc(ccc2O)Br)SCCC#N S04839 Cc1c(c(nc(n1)S)O)Cc2c(cccc2Cl)F RJF00107 CCOC(=O)c1ccc(cc1)N2C(=O)C=CC2=O S02262 COc1ccc(cc1OC)CCN2C(=O)/C(=C/c3c(c(c(c(c3F)F)F)F)F)/SC2=S S02324 Cc1ccc(cc1Cl)N2C(=O)CC(C2=O)Sc3ccccc3C(=O)O S02334 c1cc(ccc1c2csnn2)NC(=O)C(Cl)(Cl)Cl SEW00786 Cc1c(c(on1)C)c2nc(no2)CSc3ccccc3 SEW00843 c1cc(cc(c1)Cl)c2cnco2 SEW00955 CN(C)C(=S)NCc1ccc(cc1)F S14533 c1cc(ccc1CNC(=S)NCc2ccc(cc2)F)F S14534 Cc1cccc(c1N(C2=NCCC(=O)S2)C(=O)c3ccoc3)C RJF01733 CCc1cccc(c1N(C2=NCCC(=O)S2)C(=O)C)C RJF01739 CCc1cccc(c1N(C2=NCCC(=O)S2)C(=O)c3ccco3)C RJF01740 c1cc(ccc1OCc2nc(on2)c3ccsc3)Cl SEW01964 c1ccc2c(c1)C(=O)NC(N2)c3c(cccc3Cl)F S12245 CC(=O)C1CNc2ccccc2C1(c3ccccc3)O S12255 CCOC(=O)CNc1ccc(cc1)C(F)(F)F S14332 CCOC(=O)c1c(nc2ccc(cc2c1c3ccccc3)Cl)C S12260 COc1cc2c(cc1OC)N3C(=O)c4ccccc4C3(OC2=O)O S14349 CC(C)(C)C(=O)Nc1ccc(cc1)c2csnn2 SEW00787 c1cc(ccc1NC(=O)NC(=O)c2csc(n2)c3ccc(cc3Cl)C(F)(F)F)F SEW01978 Cc1c(c(nc(n1)SCc2c(cccc2Cl)Cl)O)Cc3c(cccc3Cl)Cl RJF00255 Cc1c(c(on1)C)c2nc(no2)CS(=O)(=O)c3ccccc3 SEW00845 c1cc(ccc1CNC(=O)c2cc(cc(c2)Cl)Cl)c3csnn3 SEW00852 CC(C)(C)NC(=O)NCc1ccc(cc1)c2csnn2 SEW00854 CCCCC(C(=O)N/N=C/c1cc(c(cc1)OCC)OC)C(=O)N/N=C/c2cc(c(cc2)OCC)OC S04752 c1cc(ccc1CNC(=S)Nc2ccc(c(c2)Cl)Cl)c3csnn3 SEW00858 C=CCNC(=S)NCc1ccc(cc1)c2csnn2 SEW00860 CCCCC(C(=O)N/N=C/c1sccc1)C(=O)N/N=C/c2sccc2 S04753 CNC(=O)NCc1ccc(cc1)c2csnn2 SEW00853 c1ccc(cc1)NC(=O)NCc2ccc(cc2)c3csnn3 SEW00855 c1ccc(cc1)C(=O)Cn2nc(nn2)N3CCOCC3 RJF00232 c1cc(ccc1CNC(=O)Nc2ccc(cc2)Cl)c3csnn3 SEW00856 c1ccc(c(c1)C(F)(F)F)NC(=S)NCc2ccc(cc2)c3csnn3 SEW00857 c1cc(cc(c1)Cl)CNC(=O)N S12185 c1cc(cc(c1)NC(=S)NNC(=O)Cn2nc(nn2)N3CCOCC3)C(F)(F)F RJF00246 Cc1cc(cc(c1)N2C(=O)C=CC2=O)C S14371 c1c(cc(cc1Cl)Cl)NC(=S)Nc2cc(cc(c2)Cl)Cl RJF00280 c1cscc1c2nc(no2)COc3c(cc(cc3Cl)F)Cl SEW01987 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccccc2CCC(=O)O S12188 c1c(cc(c(c1Cl)N/N=C/c2cc(sc2Cl)Cl)Cl)Cl SEW02002 c1cc(c(c(c1)F)c2nc3ccc(cc3c(=O)o2)SC#N)F S12196 c1ccc(cc1)C(=O)Oc2cccc3c2CCC3=O S12199 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)Cc3cccnc3 S12235 CCCCC(C(=O)N/N=C/c1ncccc1)C(=O)N/N=C/c2ncccc2 S04754 CCCCC(C(=O)N/N=C/c1c(cccc1)Cl)C(=O)N/N=C/c2c(cccc2)Cl S04757 c1cc(sc1)C(=O)NCc2ccc(cc2)c3csnn3 SEW00861 c1cc(c(cc1NC(=S)N)Cl)Cl S12174 Cc1cc(cc(c1)N2C(=O)CC(C2=O)Sc3ccccc3N)C S14372 c1cc(c(c(c1)Cl)Cn2nc(nn2)N3CCOCC3)Cl RJF00247 Cc1c(nc(nc1OC(=O)N(C)C)SCc2c(cccc2Cl)F)C RJF00274 CC(=O)Nc1nc(nc(n1)NC(=O)C)c2ccccc2C(F)(F)F RJF01642 c1cc(oc1/C=N/N2CC(=O)N(CC2=O)c3cc(cc(c3)Cl)Cl)[N+](=O)[O-] S14383 c1ccc(cc1)c2cc(oc2c3ccccc3)c4ccc(cc4)Cl S14393 COc1ccc(cc1)N2C(=O)CC(C2=O)N3CCCCC3 S12371 Cc1c(c(nc(n1)SCc2c(cccc2Cl)F)O)Cc3c(cccc3Cl)Cl RJF00258 Cc1c(c(nc(n1)S)O)CC2CC2 RJF00264 CN1C2(CC(O1)COC(=O)c3ccc(cc3)C(F)(F)F)C4CC5CC(C4)CC2C5 S14397 CCCc1cc(nc(n1)NC#N)O RJF01620 CCCC(/N=C/c1c(ccc(c1)Cl)O)/N=C/c2c(ccc(c2)Cl)O S14362 Cc1c(nc(nc1OC(=O)N(C)C)SCc2c(cccc2Cl)Cl)C RJF00267 Cc1ccccc1c2nc(nc(n2)N)N RJF01626 Cc1c(c(nc(n1)S)O)Cc2ccc(cc2)F RJF01657 Cc1ccc2c(c1)C(=O)OC3(N2C(=O)c4c3cccc4)O S14346 COc1ccc(cc1)N2C(=O)CC(C2=O)N3CCOCC3 S12374 CCOC(=O)c1ccc(cc1)N2C(=O)CC(C2=O)N3CCSCC3 S12375 CC(C)Cc1ccc(cc1)C(=O)CC2c3ccccc3C(=O)O2 S14466 COc1cc(cc(c1)N/N=N/c2ccccc2C(=O)OC)C(F)(F)F S04920 c1ccc(cc1)c2nc(no2)COc3ccc(cc3Cl)Cl SEW02035 COc1ccccc1c2nc(no2)COc3ccc(cc3Cl)Cl SEW02036 COc1cccc(c1)c2nc(no2)COc3ccc(cc3Cl)Cl SEW02037 CN(C)C(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F S04786 c1ccc(c(c1)NC(=O)/C=C/C(=O)O)Br S04787 c1cc(cc(c1)Cl)C(=O)NNC(=S)N S04479 c1cc(ccc1NC(=O)CCC(=O)O)OC(F)(F)F S14176 c1cc(ccc1N2C(=O)CCC2=O)OC(F)(F)F S14177 C1C2CC3CC1CC(C2)C3(CC#N)C#N S14185 CSc1cccc(c1)NC(=S)NCc2cccnc2 S04495 c1ccc(cc1)C(=O)NC(CC(=O)O)C(=O)O S02474 Cc1cc(c(c(c1)C)NC(=S)NN)C S02484 CC(C)C(=O)Nc1nc(nc(n1)NC(=O)C(C)C)c2ccccc2C(F)(F)F RJF01640 c1cc(c(cc1OCC(F)(F)F)c2csnn2)OCC(F)(F)F SEW00874 CC(C)Cc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3ccc(cc3)C(F)(F)F S14468 CC1=CC2CC1C3C2C(=O)N(C3=O)c4ccc(cc4)OC(F)(F)F S14356 CC1=CC2CC1C3C2C(=O)N(C3=O)c4ccc(cc4)C(F)(F)F S14357 CCOc1ccccc1/N=C\2/NCCS2 S02531 Cc1c(c(c(c(c1C)C)CSC(=[NH2+])N)C)C S02526 Cc1cc(cc(c1)NC(=O)/C=C\C(=O)O)C S14370 Cc1ccc(cc1F)NC(=S)NC(=O)c2cc(c(c(c2)OC)OC)OC S02563 Cc1c(c(on1)C)C(=O)NCc2ccc(cc2)c3csnn3 SEW00864 c1cc(ccc1CNS(=O)(=O)c2ccc(cc2F)F)c3csnn3 SEW00866 c1cc(ccc1NC(=O)C2CC2)S(=O)(=O)NC34CC5CC(C3)CC(C5)C4 RJF01507 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(c(c2)Cl)F)/C#N SEW00870 Cc1cc(nc(n1)SCc2c(cccc2Cl)Cl)OC(=O)c3ccc(cc3)C(C)(C)C RJF00283 CCCCCc1c(nc(nc1O)S)C RJF01647 CC(=O)c1ccccc1N2C(=O)C3C4CC(C3C2=O)C=C4 S12276 c1ccnc(c1)C2N(C(=O)CS2)c3ccc(cc3)C(F)(F)F S12286 COc1ccc(cc1OC)CCNC(=S)NC(=O)c2cc(c(c(c2)OC)OC)OC S02561 c1ccc(c(c1)C(=O)N)NC(=O)C2C3CC(C2C(=O)O)C=C3 S12293 c1ccc(c(c1)C(=O)Nc2ccccc2C(=O)N)C(=O)O S12294 CN1C(=O)/C(=C\N(C)C)/C(=N1)c2ccccc2O S12303 COc1cc(cc(c1OC)OC)C(=O)NC(=S)Nc2ccc3c(c2)OCO3 S02565 c1ccc2c(c1)cc(o2)CSCc3c(cccc3Cl)Cl S11952 COc1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccc5ccccc5c4 S14210 c1cc2c(cc(=O)oc2cc1N)C(F)(F)F RJF00052 Cc1cc(nc(n1)SCc2c(cccc2Cl)Cl)OC(=O)c3ccco3 RJF00286 c1cc(ccc1C(=O)Cn2nc(nn2)N3CCCC3)Cl RJF00291 c1cc(c(cc1/C=N/O)Cl)F SEW00875 CC(=O)Nc1ccc(cc1)C2=N/C(=C\c3cc(c(c(c3)OC)OC)OC)/C(=O)O2 S02586 Cc1c(c(nc(n1)S)O)Cc2ccc(c(c2)Cl)Cl RJF01660 Cc1cc(c(c(c1)C)NC(=S)N(C)C)C S02487 c1ccc(cc1)/C=C/c2nc3ccccc3c(=O)o2 S02488 CNC(=O)O/N=C/c1ccc(c(c1)Cl)F SEW00877 c1cc(c(cc1/C=N/OC(=O)C2CC2)Cl)F SEW00880 c1cc(c(c(c1)Cl)Cn2nc(nn2)N3CCCC3)Cl RJF00305 C1CCN(C1)c2nnn(n2)CC(=O)NN RJF00309 c1ccnc(c1)/C=N/NC(=O)Cn2nc(nn2)N3CCCCC3 RJF00311 c1ccc2c(c1)c(=O)oc(n2)c3ccc(cc3)[N+](=O)[O-] S02574 CCCc1cc(nc(n1)c2cccc(c2)C)O RJF01521 CCCc1c(c(nc(n1)S)O)C RJF01522 Cc1c(c(nc(n1)SC(C)C=C)O)Cc2ccc(cc2)F RJF01663 CC(C)(C)C(=O)Nc1nc(nc(n1)NC(=O)C(C)(C)C)c2ccccc2Cl RJF01664 CCOC(=O)CNc1ccc(cc1)I S14315 CCOC(=O)CNc1ccc(cc1)F S14316 c1cc(ccc1C(=O)O/N=C/c2ccc(c(c2)Cl)F)Cl SEW00881 c1cc(cc(c1)NC(=S)NCCCC(=O)O)C(F)(F)F RJF01715 c1cc(cnc1)/C=N/NC(=O)Cn2nc(nn2)N3CCCCC3 RJF00325 c1cc(c(cc1Cl)Cl)/C=N/NC(=O)Cn2nc(nn2)N3CCCCC3 RJF00326 COc1ccccc1C(CC(=O)c2ccccc2)Sc3ccccc3N S02340 Cc1ccc(cc1)C(=O)CC(c2ccc(cc2)[N+](=O)[O-])Sc3ccccc3N S02341 Cc1ccc(cc1)C2=Nc3ccccc3SC(C2)c4ccc(cc4)OC S02345 COc1ccc(cc1OC)C2CC(=Nc3ccccc3S2)c4ccccc4 S02347 CC\1=NN(C(=O)/C1=N/O)c2cccc(c2)Cl S12126 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OS(=O)(=O)c4cc(c(cc4Cl)Cl)C RJF01546 CCCc1cc(=O)oc2c1ccc(c2)OC(=O)c3ccc(cc3)C(C)(C)C RJF01547 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)Cl)c4cc(cc(c4)C(F)(F)F)C(F)(F)F RJF00116 CCCc1cc(nc(n1)NC(=N)Nc2cc(ccc2Cl)C(F)(F)F)O RJF01614 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)OCC(=O)c3ccc(cc3)Cl RJF01576 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)OCC(=O)C(C)(C)C RJF01577 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)NNC(=O)c3ccc(cc3)Cl RJF01579 CCCc1cc(nc(n1)NC(=N)Nc2ccc(cc2F)F)O RJF01615 Cc1ccc(c(c1)NC(=O)/C=C/C(=O)O)C S04584 Cc1ccc(c(c1)C)N2C(=O)CC(C2=O)Sc3ccccc3N S04591 CCCc1c(c(nc(n1)SCc2ccc(cc2)F)O)CC=C RJF01584 CCCC1=NN(C(=O)C1CC=C)S(=O)(=O)c2ccc(cc2)Cl RJF01592 COc1ccc(cc1)C(=O)CC2c3ccccc3C(=O)O2 S04713 CCCC1=NN(C(=O)C1Cc2c(cccc2Cl)F)C(=O)c3ccc(cc3)Cl RJF01551 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/OCc3cc(cc4c3OCOC4)F SEW01942 CN(C)C(=S)Nc1cccc(c1)F S04561 c1ccc(cc1)C2=Nc3ccccc3SC(C2)c4ccc(cc4)Cl S02346 c1ccc(cc1)C(=O)CC(c2c(cccc2Cl)Cl)Sc3ccccc3N S02355 COc1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccccc4 S02356 CCCCC(C(=O)N/N=C/c1c(c(cc(c1)Cl)Cl)O)C(=O)N/N=C/c2c(c(cc(c2)Cl)Cl)O S04750 c1c(cc(cc1Cl)Cl)/N=C/2\NCCS2 RJF00152 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N\c3cc(cc(c3)Cl)Cl RJF00153 Cc1ccc(c(c1)N2C(=O)C=CC2=O)C S04585 c1cc(c(cc1F)F)NC(=S)Nc2ccc(cc2F)F RJF00157 COc1ccc(cc1OC)C(CC(=O)c2ccccc2)Sc3ccccc3N S02337 CC(C)(C)CC(C)(C)NC(=O)/C=C/C(=O)O S04637 CCCCCCNC(=O)/C=C/C(=O)O S04679 Cc1ccc(c(c1)NC(=S)N(C)C)C S04716 Cc1ccc(cc1)C(=O)CC(c2ccc(cc2)OC)Sc3ccccc3N S02338 c1cc(cc(c1)F)NC(=S)NC2CCCCCCCCCCC2 S04565 c1ccc2c(c1)C(OC2=O)CC(=O)c3ccc(cc3)[N+](=O)[O-] S04568 CC1(OC(=O)C(=Cc2c(cc(cc2OC)OC)OC)C(=O)O1)C S14264 COC(=O)c1c(ccs1)c2ccc(o2)/C=C(\C#N)/S(=O)(=O)C SEW01884 COC(=O)c1c(ccs1)c2ccc(o2)C=C(C#N)C#N SEW01885 c1cc(ccc1Cn2nc(nn2)N3CCCCC3)Cl RJF00333 c1cc(ccc1/C=N/NC(=O)Cn2nc(nn2)N3CCCC3)Cl RJF00338 CCOC(=O)/C(=C/c1ccc(s1)[N+](=O)[O-])/C#N S05244 Cc1c(c(nc(n1)SCc2c(cccc2Cl)Cl)O)Cc3c(cccc3Cl)F RJF00340 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)N)Oc3ccc(cc3Cl)Cl RJF01710 Cc1c(c(on1)/C=C/c2ccc(cc2F)F)[N+](=O)[O-] SEW00817 c1cc(ccc1/C(=N\N)/Cn2nc(nn2)N3CCCCC3)Cl RJF00330 CC(C)(C)C(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl RJF01716 c1cc(ccc1NC(=S)NCCCC(=O)O)Cl RJF01722 c1cc(sc1)c2ccc(s2)C=C(C#N)C#N SEW02156 Cc1ccc(o1)/C=N/NC(=S)N S12436 c1ccnc(c1)C2N(C(=O)CS2(=O)=O)c3ccc(cc3)C(F)(F)F S12288 CC(C)Cc1ccc(cc1)C(=O)/C=C/c2cccc(c2)[N+](=O)[O-] S14492 Cc1ccc(cc1)N2C(=O)C(C(C2=O)N3CCOCC3)c4ccccc4 S12414 c1cc(ccc1CN2C(SCC2=O)c3ccncc3)F S14510 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccc(cc3)c4csnn4 SEW00838 CCOC(=O)N/N=C(\C)/c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F SEW00841 Cc1c(c(on1)C)c2nc(no2)CSCc3ccc(cc3)Cl SEW00842 c1ccc(c(c1)/C=N/Nc2ccc(cn2)[N+](=O)[O-])OC(F)(F)F SEW02147 c1cc(ccc1c2csnn2)NC(=O)C3C4CC(C3C(=O)O)C=C4 SEW00987 c1cc(ccc1c2csnn2)NC(=O)CSCC(=O)O SEW00988 Cc1ccc(cc1C)N2C(=O)CC(C2=O)N3CCCCC3 S12384 CCOc1c(c(c(c(n1)N)C#N)c2cccc(c2OC)OC)C#N S02756 CC(C)Cc1ccc(cc1)C(=O)CC(c2cccc(c2)[N+](=O)[O-])Sc3ccccc3N S14500 c1cc(ccc1NCn2c3ccc(cc3nn2)Cl)I S14501 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2cccc3 S02762 c1cc(ccc1CNC(=O)/C=C/C(=O)O)F S14504 CSc1nnc(o1)c2cccc(c2)[N+](=O)[O-] SEW00822 Cc1ccc(cc1)S(=O)(=O)c2c(scn2)NC SEW00824 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(c(c3)Cl)Cl)O RJF01678 CCCNC(=O)NNC(=O)Cn1nc(nn1)N2CCOCC2 RJF01817 c1cc(c(cc1Cl)NC(=O)c2cc(cc(c2)Cl)Cl)OC(=O)c3cc(cc(c3)Cl)Cl S14559 Cc1c(c(no1)c2ccccc2Cl)c3nc4ccc(cc4c(=O)o3)I S12522 CC(=O)c1ccccc1NC(C#N)c2ccccc2 S12546 Cc1c(c(nc(n1)SCc2c(cccc2Cl)F)O)Cc3c(cccc3Cl)F RJF00334 c1cc(cc(c1)Cl)n2c(nnc2SCC3CC3)C4CC4 RJF01762 c1cc(cc(c1)NC(=S)NNC(=O)Cn2nc(nn2)N3CCCC3)C(F)(F)F RJF00337 c1cc(cc(c1)N)c2cnco2 SEW00990 c1cc2c(cc1NC(=S)NN)OCO2 S02420 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2ccccc2OC)N S12164 C/C(=C\c1cccc(c1)OC)/[N+](=O)[O-] S12170 Cc1cccc(c1/C=N/NC(=S)Nc2ccc(cc2Cl)Cl)Cl SEW01050 Cc1cc(c(n1c2ccc(cc2)C(F)(F)F)C)C(=O)C(F)(F)F SEW01052 c1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2)c3csnn3)\N SEW01054 c1cc(ccc1c2csnn2)/C(=N/OC(=O)c3ccc(cc3)Cl)/N SEW01055 COc1ccc(cc1NC(=O)COCC(=O)O)Cl S12645 CC1=CC(=O)N(C1=O)c2cc(ccc2OC)Cl S12646 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc4c(c3)OCCO4 S05266 Cc1cc(c(c(c1)C)NC(=O)/C=C/C(=O)O)C S02802 Cc1cc(c(c(c1)C)NC(=O)CC2C(=O)NC(=N)S2)C S02812 c1cc(c(cc1C(F)(F)F)N2C(=O)C=CC2=O)Cl S04911 c1ccc(c(c1)NC(=S)Nc2cc(c(cc2Cl)Cl)Cl)Br S04914 c1cc(c(cc1F)F)N2C(=O)c3ccncc3C2=O S12321 c1cc(c(cc1Cl)Cl)N2C(=O)c3ccncc3C2=O S12323 CCOC(=O)c1ccc(cc1)N2C(=O)c3ccncc3C2=O S12324 c1ccc2c(c1)nnn2CNc3ccc(cc3)C(F)(F)F S14444 CC(C)(C)C(=O)Nc1nc(nc(n1)NC(=O)C(C)(C)C)c2ccccc2C(F)(F)F RJF01670 c1cc(cnc1)CN\2C(=O)CS/C2=N\c3ccc(cc3F)F RJF00169 CCOc1ccccc1NC(=S)NCCO S02445 c1ccc(cc1)C(=O)Oc2ccccc2CCC(=O)O S12190 Cc1cc(c(cc1C)NC(=S)N(C)C)C S02405 c1cc(c(cc1N2C(=O)C=CC2=O)Cl)Br S02408 c1cc2c(cc1NC(=S)NCCO)OCO2 S02422 c1cc2c(cc1N3C(=O)C=CC3=O)OCCO2 S05229 COC(=O)c1ccccc1/N=N/Nc2cccc(c2)C(F)(F)F S02737 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccccc3SCCC#N S04843 Cc1ccc(cc1N2C(=O)C=CC2=O)N3C(=O)C=CC3=O S04909 c1ccc2c(c1)c(=O)[nH]c(n2)c3ccccc3C(=O)O S12296 CC1=C(C2(c3ccccc3NC2=O)C(=C(O1)N)C#N)C(=O)C S14426 c1cc(sc1)SC2CC(=O)N(C2=O)c3ccc(cc3)F S14439 c1ccc2c(c1)nnn2CNc3ccccc3OC(F)(F)F S14441 c1ccc(cc1)C(=O)NC(=S)Nc2cccc(c2)C(F)(F)F S02633 CCCc1c(c(nc(n1)c2ccccn2)O)Cc3c(cccc3Cl)F RJF01808 CCCc1c(c(nc(n1)c2ccccn2)O)CC3CC3 RJF01809 CCOC(=O)C1=C(OC(=C(C12c3ccccc3NC2=O)C#N)N)C S14427 COc1ccc(cc1)C(=O)CC(c2ccccc2)C(=O)c3ccccc3 S14416 CCOC(=O)c1c(nc2ccccc2c1c3ccccc3)C S12267 CC(=O)c1ccccc1NC(=O)CSCC(=O)O S12270 CC1(CC2=C(C(=O)C1)C3(C(=C(O2)N)C#N)C(=O)c4ccccc4C3=O)C S14423 CC1=C(C2(c3ccccc3NC2=O)C(=C(O1)N)C#N)C(=O)OC(C)(C)C S14425 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S05042 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)/C=N/NC(=O)Cn3nc(nn3)N4CCOCC4 RJF00298 CCOC(=O)Cn1nc(nn1)N2CCCC2 RJF00301 c1cc(c(cc1C(=O)Cn2nc(nn2)N3CCCCC3)Cl)Cl RJF00303 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(c(c3)Cl)Cl)OS(=O)(=O)c4ccc(cc4)Cl RJF01689 C=CCCN1C(=O)c2ccccc2C1=O S05273 c1cc(sc1)/C=C(/c2ccsc2)\C(=O)N3CCOCC3 SEW02128 c1ccc(cc1)/C(=C/C(=O)c2ccc(cc2)F)/C(=O)c3ccccc3 S14401 c1cnccc1/C=N/NC(=O)Cn2nc(nn2)N3CCCCC3 RJF00314 CCCc1c(c(nc(n1)c2ccccn2)O)CC=C RJF01673 Cc1c(nc(nc1OC(=O)c2ccc(cc2)C(C)(C)C)SCc3c(cccc3Cl)F)C RJF00281 C1CCN(CC1)c2n[nH]nn2 RJF00289 c1cc(ccc1C(=O)Cn2nc(nn2)N3CCCCC3)Cl RJF00292 c1ccc(c(c1)/C=N/NC(=O)Cn2nc(nn2)N3CCOCC3)Cl RJF00295 CC(C)(C)c1cc(nc(n1)NC(=N)Nc2ccc(cc2F)F)O RJF01796 c1cc(ccc1C#N)c2csnn2 SEW00982 Cc1cc(c(n1c2ccccc2)C)C(=O)C(F)(F)F SEW00977 c1cc(ccc1c2csnn2)NC(=O)/C=C/C(=O)O SEW00984 c1ccc(cc1)C(=O)Cn2nc(nn2)N3CCCCC3 RJF00306 CCOC(=O)Cn1nc(nn1)N2CCCCC2 RJF00308 Cc1ccccc1c2nc(nc(n2)NC(=O)C)NC(=O)C RJF01675 c1cc(c(c(c1)Cl)c2nc(nc(n2)N)N)Cl RJF01676 CCOC(=O)/C(=C\c1c(c(c(c(c1)/C=C(\C(=O)OCC)/C#N)N(C)C)C#N)N(C)C)/C#N SEW02049 C/C(=N\Nc1cc(ccc1Cl)Cl)/Cc2nc(sn2)Nc3ccccc3 SEW02064 c1cc(sc1)CNC(=S)Nc2cc(cc(c2)Cl)Cl RJF00373 CC(C)c1ccc(cc1)N2C(=O)C=CC2=O S02846 CC(C)c1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3N S02848 CCO/C=C\1/C(=O)N(C(=S)S1)c2ccc(cc2)C(C)C S02849 CC(C)c1ccc(cc1)NC(=S)NC(=O)c2ccccc2 S02850 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(o3)c4ccsc4C(=O)OC)C(=O)OC SEW02071 Cc1c(c(c(c(n1)C)C(=O)O)c2ccsc2)C(=O)O SEW02072 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(c(c3)Cl)Cl)OS(=O)(=O)C RJF01683 c1ccc(cc1)N2C(=O)CC(C2=O)N3CCOCC3 S12347 CN(C)c1c(cc(c(c1C#N)N(C)C)C=C(C#N)C#N)C=C(C#N)C#N SEW02047 CN(c1c(c(c(cc1/C=C(\S(=O)(=O)C)/C#N)/C=C(\S(=O)(=O)C)/C#N)N(C)C)C#N)C SEW02048 c1ccc(cc1)c2cc(oc2c3ccccc3)c4ccc(cc4)F S14408 Cc1c(c(c(c(n1)C)C(=O)OC)c2ccsc2)C(=O)OC SEW02068 c1cc(cc(c1)Cl)c2c(nco2)C#N SEW02044 c1ccc(cc1)S(=O)(=O)/C(=C/c2cc(sc2Cl)Cl)/C#N SEW02050 COC(=O)c1c(ccs1)c2ccc(o2)/C=N/c3ccc(cc3)Cl SEW02055 c1cc(cnc1)/N=C/c2cc(sc2Cl)Cl SEW02061 COC(=O)c1c(ccs1)c2ccc(o2)C3C4=C(CCCC4=O)NC5=C3C(=O)CCC5 SEW02069 c1cc(ccc1c2csnn2)NNC(=O)c3ccc(cc3)Cl SEW00948 c1cc(ccc1N2C(=O)c3ccncc3C2=O)Cl S12343 Cc1ccc(cc1N2C(=O)c3ccncc3C2=O)Cl S12344 c1ccc2c(c1)cccc2C3CC(=Nc4ccccc4S3)c5ccc(cc5)Cl S05101 c1cc(ccc1C(=O)NNC(=S)N)[N+](=O)[O-] S02652 c1ccc(cc1)C(=O)NC(=S)Nc2cccc(c2)[N+](=O)[O-] S02660 c1ccc(c(c1)N2C(=O)C=CC2=O)Br S04788 COc1ccc(cc1)c2nc(no2)COc3ccc(cc3Cl)Cl SEW02038 c1cc(cc(c1)C(F)(F)F)c2c(nco2)C#N SEW02042 COc1ccc(cc1)CNc2ccccn2 S04793 c1ccc(c(c1)/C=N/c2ccccc2SCCC#N)O S04837 CC1c2ccsc2CCN1C(=S)Nc3ccccc3Cl SEW00940 CC(=O)Nc1ccc(cc1)C2=N/C(=C/c3cccc(c3OC)OC)/C(=O)O2 S02573 c1cc(cc(c1)[N+](=O)[O-])c2nc3cc(ccc3c(=O)o2)Cl S02582 c1ccc(cc1)c2nnnn2c3cc(cc(c3)C(F)(F)F)C(F)(F)F S05046 c1cc(cc(c1)F)n2c(nnn2)c3ccc(c(c3)Cl)Cl S05055 COc1cc(c(c(c1)OC)/C=C\2/C(=O)OC(=N2)c3ccccc3)OC S02598 c1cc(c(cc1Cl)NC(=S)N)Cl S02620 c1cc(ccc1C(F)(F)F)Nc2n[nH]c(=S)s2 S05057 Cc1ccc(cc1)N2C(=O)CC(C2=O)Sc3cccs3 S14450 Cc1ccccc1C(=O)NNc2ccc(cc2)c3csnn3 SEW00947 c1c(cc(c(c1/C=N/c2c(cc(cn2)Cl)Cl)O)Cl)Cl S04827 c1ccc2c(c1)C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/CO2 S14382 c1ccc(cc1)/C(=C/C(=O)c2ccc(cc2)Cl)/C(=O)c3ccccc3 S14391 CCCc1cc(nc(n1)NC(=N)Nc2cc(cc(c2)Cl)Cl)O RJF01616 c1ccnc(c1)S(=O)(=O)/C(=C/c2ccc(c(c2)Cl)F)/C#N SEW00871 CC(=O)Nc1ccc(cc1)C2=N/C(=C\c3cccc4c3cccc4)/C(=O)O2 S02587 c1cc(ccc1CSC(=N)N)c2csnn2.Br SEW00912 c1csc2c1sc(c2)C(=O)N SEW02086 c1cc(ccc1CNC(=O)C2CC2)c3csnn3 SEW00915 c1cc(sc1)/C=C(/c2ccsc2)\C(=O)N SEW02112 c1cc(ccc1C2c3ccsc3CCN2)Cl SEW00928 Cc1ccc(cc1Cl)NC(=S)N2CCc3c(ccs3)C2C SEW00938 CCOC(=O)N/N=C(\C)/c1ccc(cc1)O SEW00897 Cc1ccc(cc1Cl)Nc2nnc(o2)c3cccc(c3)[N+](=O)[O-] SEW00923 COc1ccc(cc1)c2cc(c(o2)c3ccccc3)c4ccccc4 S14418 c1ccc(cc1)/C(=C/C(=O)c2ccc(cc2)C(F)(F)F)/C(=O)c3ccccc3 S14419 CC(C)(C)S(=O)(=O)/C(=C/c1ccc(c(c1)Cl)F)/C#N SEW00872 Cc1c-2c(=O)n(nc2c3ccccc3o1)C S12307 c1cc(ccc1CNS(=O)(=O)c2ccc(c(c2)Cl)F)c3csnn3 SEW00867 c1cc(ccc1C2=NCCc3c2ccs3)Cl SEW00927 c1cc(ccc1N2C(=O)CC(C2=O)N3CCOCC3)Cl S12351 CC(C)Cc1ccc(cc1)/C(=N/NC(=S)N)/C S14458 COc1ccc(cc1N2C(=O)COCC2=O)Cl S12647 COc1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2)c3csnn3)\N SEW01056 Cc1c(c(on1)C)C(=O)O/N=C(/c2ccc(cc2)c3csnn3)\N SEW01059 CCCc1c(c(nc(n1)SC(C)C=C)O)CC=C RJF01686 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)NC(=O)C3CC3)Oc4ccc(cc4Cl)Cl RJF01746 c1cc(ccc1CNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3csnn3 SEW00868 CC(C)Cc1ccc(cc1)/C(=N/N=C/2\NC(=O)C(S2)CC(=O)O)/C S14459 COc1ccc(cc1)N2C(=O)CC(C2=O)N3CCSCC3 S12370 Cc1ccc(n1c2ccc(cc2)[N+](=O)[O-])C SEW00942 c1ccc(c(c1)C(=O)NNc2ccc(cc2)c3csnn3)C(F)(F)F SEW00946 CCC(=O)Nc1nc(nc(n1)NC(=O)CC)c2ccccc2C RJF01671 Cc1ccc(cc1C)N2C(=O)c3ccncc3C2=O S12345 CCCCCC1C(=NNC1=O)COC RJF01672 CCCc1c(c(nc(n1)SC)O)CC=C RJF01679 CCCc1c(c(nc(n1)SCC#C)O)CC=C RJF01680 Cc1cccc(c1NC(=S)NCCCC(=O)O)C RJF01723 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl)Oc4ccc(cc4Cl)Cl RJF01724 c1cc(cc(c1)F)Cn2nc(nn2)N3CCCCC3 RJF00331 CN(C)C(=S)Nc1ccc2c(c1)OCCO2 S05267 COc1ccc(cc1OC)CCNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S05284 c1cc(cc(c1)Cl)/C=C/2\CSc3c(ccs3)C2=O SEW02094 COc1ccc(cc1)C(CC(=O)c2ccccc2)Sc3ccccc3N S02354 Cc1ccc(c(c1)C)C(=O)CC(c2c(cccc2Cl)Cl)Sc3ccccc3N S02360 COc1cccc(c1)/C=C/[N+](=O)[O-] S12156 c1cc(sc1C=C(C#N)C#N)[N+](=O)[O-] S05237 c1cc(cc(c1)[N+](=O)[O-])c2nnnn2c3cccc(c3)F S05047 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc4c(c3)OCCO4 S05239 c1cc(ccc1C(=O)CSc2nnnn2c3ccc(cc3)F)Cl S05120 c1cc2c(cc1NC(=S)NN)OCCO2 S05265 c1ccc2c(c1)nnn2CNc3ccc(cc3)OC(F)(F)F S14447 CC(C)Cc1ccc(cc1)C(=O)/C=C(/c2ccccc2)\C(=O)c3ccccc3 S14451 Cc1c(c(c(c(n1)C)C(=O)OC)c2cc(sc2)S(=O)(=O)/N=C/N(C)C)C(=O)OC SEW02143 c1cc(ccc1NCn2c3ccc(cc3nn2)Cl)OC(F)(F)F S14452 c1ccc(cc1)C2=Nc3ccccc3SC(C2)c4cccc(c4)[N+](=O)[O-] S02362 c1ccc(cc1)Oc2ccccc2C(=O)N/N=C/c3cc(cc(c3O)Cl)Cl S04718 Cc1c(c(=O)n([nH]1)C(=O)C2CC2)Cc3ccc(cc3)F RJF01605 c1cc(sc1)/C=C(/c2ccsc2)\C(=O)Sc3ccc(cn3)C(F)(F)F SEW02131 Cc1c(c(c(c(n1)C)C(=O)OC)c2cc(sc2)S(=O)(=O)N3CCOCC3)C(=O)OC SEW02132 c1cc(sc1)/C=C(/c2ccsc2)\C(=O)Nc3ccc(cc3)Cl SEW02109 c1cc(c(cc1Cl)Cl)OCC2=C(c3cc(ccc3SC2)Cl)Cl SEW02124 Cc1c(c(c(c(n1)C)C(=O)OC)c2cc(sc2)S(=O)(=O)N3CCSCC3)C(=O)OC SEW02133 Cc1c(c(c(c(n1)C)C(=O)OC)c2cc(sc2)S(=O)(=O)N3CCCC3)C(=O)OC SEW02134 Cc1c(c(c(c(n1)C)C(=O)OC)c2cc(sc2)S(=O)(=O)Nc3ccc(cc3)OC)C(=O)OC SEW02140 CC(C)(C)c1ccccc1N2C(=O)C=CC2=O S14474 CC(CC(=O)Nc1ccccc1C(C)(C)C)CC(=O)O S14481 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)Cl)c4ccc(c(c4)Cl)F RJF00119 c1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)Sc3ccccc3N S02339 COc1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccc(cc4)OC S02343 Cc1ccc(cc1)C2=Nc3ccccc3SC(C2)c4cccc(c4)[N+](=O)[O-] S02344 c1ccc(cc1)Oc2ccccc2C(=O)N/N=C/c3cc(ccc3O)Br S04720 CSc1cccc(c1)N2C(=O)C=CC2=O S02724 CC(C)Cc1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)Sc3ccccc3N S14488 CCC(=O)Nc1nc(nc(n1)NC(=O)CC)c2ccccc2Oc3ccc(cc3Cl)Cl RJF01712 COc1ccc(c(c1)/C=N/NC(=O)Cn2nc(nn2)N3CCCCC3)OC RJF00322 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2)OC)C(=O)OC SEW02190 c1cc(sc1)c2ccc(s2)/C=N/Nc3c(cc(cc3Cl)Cl)Cl SEW02174 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(\Cn2nc(nn2)N3CCCC3)/c4ccc(cc4)Cl RJF00359 Cc1c(c(nc(n1)SCC2CC2)O)Cc3ccc(c(c3)Cl)Cl RJF01780 c1ccc(c(c1)C(=O)NNC(=O)Cn2nc(nn2)N3CCOCC3)Cl RJF00370 CCCc1c(c(nc(n1)SCC2CC2)O)CC=C RJF01793 c1cc2c(cc1Cl)C(=C(CS2)CN3CCSCC3)Cl SEW02178 c1cc(ccc1CNC2=NCCS2)F S14515 CC(=C)Cc1c(nc(nc1O)SCC2CC2)COC RJF01792 CC(C)(CO)NC(=S)NC1CC1 RJF00379 c1cc(sc1)CN\2C(=O)CS/C2=N\c3cc(cc(c3)Cl)Cl RJF00380 COCc1cc(nc(n1)SCC2CC2)O RJF01763 c1ccc(cc1)/N=N/c2nnc(s2)Nc3cccc(c3)C(F)(F)F S05000 c1cc(c(cc1Cl)Cl)C(=O)NNC(=O)Cn2nc(nn2)N3CCOCC3 RJF00364 Cc1cc(c(cc1C)NC(=S)NC(=O)c2ccccc2)C S02842 c1cc2c(cc1[N+](=O)[O-])C(=O)N(C2=O)CO S05531 Cc1nc(cc(n1)O)c2ccccc2 RJF00516 COCc1cc(=O)oc2c1ccc(c2)O RJF00525 CN(C)C(=O)Oc1ccc2c(cc(=O)oc2c1)COC RJF00526 c1cc(ccc1c2nnc(o2)SCC(=O)c3ccc(cc3)F)C(F)(F)F S12692 c1ccc(cc1)C(C#N)Nc2cc(cc(c2)Cl)Cl S12557 c1ccnc(c1)C2N(C(=O)CS2)Cc3ccc(cc3)F S14511 c1cc(c(cc1Cl)Cl)C(=O)NNC(=O)Cn2nc(nn2)N3CCCC3 RJF00342 Cc1ccc(c(c1)C)/N=C\2/N(C(=O)CS2)CCc3ccc(c(c3)OC)OC S12461 c1ccc(cc1)CS/C(=N/N=C2CCCCC2)/NC(=O)Nc3ccccc3 S12467 c1cc(cc(c1)NC(=O)/C=C/C(=O)O)C(F)(F)F S02721 c1(nnc(s1)NC(=N)NC(=N)N)C(F)(F)F.Cl RJF00600 CC(C)c1ccc(cc1)N2CN(C(=S)SC2)c3ccc(cc3)C(C)C S02844 CC(C)c1ccc(cc1)NC(=O)/C=C/C(=O)O S02845 c1cc(ccc1c2csnn2)/N=C/c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW00994 c1cc(ccc1c2csnn2)N3C(=O)C4C5CC(C4C3=O)C=C5 SEW00999 COc1cc(cc(c1)OC)/C=C\2/C(=O)OC(=N2)c3ccccc3 S12695 Cc1cn(c2c1cccc2)CCC#N SEW02253 c1cc(ccc1/C=N/c2ccc(cc2)c3csnn3)[N+](=O)[O-] SEW00993 CC1CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)c4csnn4 SEW01001 c1cc(ccc1c2csnn2)N3C(=O)C=CC3=O SEW00998 c1cc(c(cc1/C=N/NC(=S)N)Cl)F SEW01003 c1ccc(c(c1)C(F)(F)F)NC(=S)NNc2ccc(cc2)c3csnn3 SEW00950 c1ccc(cc1)/C(=C/C(=O)c2ccco2)/C(=O)c3ccccc3 S14517 c1ccc(cc1)/C(=C\C(=O)c2cccs2)/C(=O)c3ccccc3 S14518 c1cc(ccc1CNC(=S)NN)F S14523 CNC(=S)N1CCc2c(ccs2)C1c3ccc(cc3)Cl SEW01029 Cc1ccc(cc1NCN2C(=O)CNC2=S)Cl S12483 Cc1c(nc(c(n1)C#N)C#N)C SEW01007 c1cc(ccc1CN)c2csnn2.Cl CC16413 c1ccc(c(c1)C2C(CCC(=O)N2)[N+](=O)[O-])Cl S05368 c1cc(ccc1C2c3ccsc3CCN2C(=O)c4ccc(cc4)Cl)Cl SEW01018 COc1ccc(cc1)C(=O)N2CCc3c(ccs3)C2c4ccc(cc4)Cl SEW01019 CCNC(=O)/C(=C/c1ccc(cc1)C)/C#N S05391 c1cc(sc1)c2ccc(s2)/C=N/c3ccc(cc3)Cl SEW02186 c1cc(c(cc1NC(=S)NCCCC(=O)O)Cl)F RJF01765 c1ccc(cc1)C(=O)NC(=S)Nc2c(cc(cc2Cl)Cl)Cl S02725 CC(=O)c1ccc(cc1)NCN2C(=O)/C(=C\N(C)C)/NC2=S S12492 CC(=O)NNC(=O)c1cc2c(s1)ccs2 SEW02169 Cc1ccc(c(c1)NC(=O)c2cc(cc(c2)Cl)Cl)OC(=O)c3cc(cc(c3)Cl)Cl S14555 c1csc2c1sc(c2)C(=O)NNC(=O)C(F)(F)F SEW02170 CC(C)C(=O)NNC(=O)c1cc2c(s1)ccs2 SEW02171 Cc1ccccc1/C=N/N=C\2/NC(=O)CCS2 S14539 c1cc(ccc1c2nc3cc(ccc3o2)Cl)F S14578 Cc1c(c(nc(n1)SCC(=O)C(C)(C)C)O)Cc2c(cccc2Cl)F RJF00444 Cc1cc(nc(c1)/N=C/c2ccccc2O)C S04828 Cc1c(c(c(c(n1)C)C(=O)OC)c2cc(sc2)S(=O)(=O)Nc3ccc(c(c3)Cl)F)C(=O)OC SEW02141 c1cc(ccc1c2csnn2)N/N=C/c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW00962 c1cc(cc(c1)[N+](=O)[O-])c2cnco2 SEW00985 Cc1ccc(c(c1)NC(=O)c2ccc(cc2)C(F)(F)F)OC(=O)c3ccc(cc3)C(F)(F)F S14556 Cc1ccc(cc1)NCN2C(=O)c3ccc(cc3C2=O)[N+](=O)[O-] S05587 c1cc2c(cc1Cl)C(=CCS2(=O)=O)SCCC(=O)O SEW02182 CC(C)(C)c1ccc(cc1)C(=O)Nc2cc(ccc2OC(=O)c3ccc(cc3)C(C)(C)C)Cl S14560 c1ccc(cc1)C(=O)NC(=S)Nc2ccccc2NC(=S)NC(=O)c3ccccc3 S03104 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N/c3c(cc(cc3Br)F)Br RJF00414 Cc1cc(nc(n1)N)Nc2cc(cc(c2)Cl)Cl RJF00402 CC(C)(C)c1ccc(cc1)/N=C/2\N(C(=O)CS2)CCc3ccc(c(c3)OC)OC RJF00411 c1c(cc(cc1Cl)Cl)NC(=O)C2CC2 RJF00415 c1ccc(cc1)c2csc(n2)NC(=O)C3CC3 RJF00426 CCCc1c(nc(nc1O)SCC(=O)C(C)(C)C)C RJF00437 c1cc(sc1)CN\2C(=O)CS/C2=N\c3c(cc(cc3Br)F)Br RJF00413 CCSc1nc(cc(n1)O)c2ccccc2 RJF00514 CC1CN(CC(O1)C)c2ccc(cc2)NC(=S)NCc3cccs3 RJF00391 c1ccc(cc1)N2C(=O)CC(C2=O)N3CCN(CC3)C4CC(=O)N(C4=O)c5ccccc5 S12579 c1cc(cc(c1)Cl)n2c(nnn2)SCC(=O)c3ccc(cc3)F S12596 c1cc(ccc1/C=N/NC(=S)N)F S12746 Cc1cc(nc(n1)N)Nc2ccc(c(c2)Cl)F.Cl RJF00401 c1cc(sc1)c2ccc(s2)/C=N/c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW02185 CCOC(=O)c1ccc(c(c1)NC(=S)NCCO)Cl S05419 Cc1ccc(c(c1)OC(=O)c2ccccc2)NC(=O)c3ccccc3 S14569 Cc1ccc2c(c1)oc(n2)c3ccc(cc3)C(F)(F)F S14573 Cc1c(c(nc(n1)N)O)Cc2c(cccc2Cl)Cl RJF00433 COc1cccc(c1)N2C(=O)C=CC2=O S02937 Cc1cc(c(n1c2ccc(cc2)Cl)C)C(=O)O SEW01045 COc1cccc(c1)N2C(=O)CC(C2=O)Sc3ccccc3N S02938 Cc1cc(nc(n1)NC(=O)C2CC2)O RJF00436 COc1ccc(c(c1)C=C(C#N)C#N)OC S02895 CCCc1c(nc(nc1OC(=O)N(C)C)SCC(=O)C(C)(C)C)C RJF00438 c1cc(sc1)CN\2C(=O)CS/C2=N\C3CC3 RJF00389 CC1CN(CC(O1)C)c2ccc(cc2)/N=C\3/N(C(=O)CS3)CCc4ccc(c(c4)OC)OC RJF00398 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(c(c3)Cl)Cl S02903 COc1ccc(cc1NC(=O)/C=C/C(=O)O)Cl S12608 COc1ccc(cc1N2C(=O)C=CC2=O)Cl S12609 Cc1cc(nc(n1)SCC(=O)C(C)(C)C)O RJF00456 Cc1cc(nc(n1)N)Nc2ccc(cc2F)F.Cl RJF00403 CC[n+]1c(csc1Nc2ccc(cc2)N3CC(OC(C3)C)C)C.[I-] RJF00405 c1cc(ccc1C2c3ccsc3CCN2C(=O)C4CC4)Cl SEW01036 Cc1cccc(c1/C=N/NC(=S)N)Cl SEW01049 COc1ccc(cc1N2C(=O)c3ccncc3C2=O)Cl S12624 CC1(CC(=O)N(C(=O)C1)c2cc(ccc2OC)Cl)C S12629 Cc1cc(c(n1c2cc(cc(c2)Cl)Cl)C)C(=O)C(F)(F)F SEW01051 CC(C)c1ccc(cc1)NCN2C(=O)c3ccccc3C2=O S02912 c1ccc(cc1)C(=O)CC(c2ccc3c(c2)OCO3)Sc4ccccc4N S02950 C=CCNC(=S)N1CCc2c(ccs2)C1c3ccc(cc3)Cl SEW01030 c1cc(ccc1C2c3ccsc3CCN2S(=O)(=O)c4ccc(cc4)Cl)Cl SEW01032 CC1CC(CC(C1)(C)C)NC(=S)NC2(CCCCC2)C#C S02935 c1ccc(c(c1)C(F)(F)F)NC(=S)N2CCc3c(ccs3)C2c4ccc(cc4)Cl SEW01031 Cc1c(c(c(c(n1)C)C(=O)OC)c2ccc(cc2)OC)C(=O)OC SEW02191 Cc1c(c(nc(n1)SCC(=O)C(C)(C)C)OC(=O)N(C)C)Cc2c(cccc2Cl)Cl RJF00462 CC(C)(C)C(=O)Cn1nc(nn1)N2CCCC2 RJF00465 COc1ccc(cc1N2C(=O)CSCC2=O)Cl S12613 COc1ccc(cc1N2C(=O)CC(C2=O)Sc3ccccc3N)Cl S12614 COc1ccc(cc1N2C(=O)C=C(C2=O)c3ccccc3)Cl S12623 c1cc(ccc1c2csnn2)/C(=N/O)/N SEW01053 c1cc(ccc1c2csnn2)/C(=N/OC(=O)c3ccc(cc3)[N+](=O)[O-])/N SEW01057 Cc1cn(c2c1cccc2)CCC(=O)O SEW02254 Cc1c2ccccc2n3c1C(=O)CC3 SEW02255 CC(C(=O)N/N=C/c1cc(c(c(c1)OC)OC)OC)n2nc(nn2)N3CCOCC3 RJF01886 Cc1cc(c(n1c2cc(cc(c2)Cl)Cl)C)C(=O)O SEW01062 Cc1c(cccc1Cl)NC(=S)NC(=O)c2ccccc2 S02668 CC(C)(CC(=O)Nc1cc(ccc1OC)Cl)CC(=O)O S12628 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3cccc(c3)C(F)(F)F S02991 Cc1c(c(nc(n1)SCC(=O)C(C)(C)C)O)Cc2c(cccc2Cl)Cl RJF00447 Cc1c(c(nc(n1)c2ccc(c(c2)Cl)F)OC(=O)N(C)C)CC=C RJF00477 CCCCCCCc1c(nc(nc1O)S)COC RJF01888 CC(C)(C)C(=O)Cn1nc(nn1)N2CCOCC2 RJF00475 COc1ccc(cc1NC(=S)N)Cl S12633 c1ccc(c(c1)/C=N/OC(=O)c2c(cccc2Cl)F)OC(F)(F)F SEW02209 CC/N=C(/Nc1ccc(cc1)C(C)(C)C)\SCC2CC2.Br RJF00485 c1cc(ccc1c2csnn2)NNC(=O)c3cc(cc(c3)Cl)Cl SEW00949 c1cc(ccc1C(F)(F)F)NCn2c3ccc(cc3nn2)Cl S14454 c1cc(ccc1NCn2c3ccc(cc3nn2)Cl)F S14455 CN(C)C(=S)Nc1cccc(c1)C(F)(F)F S02992 CC(C)NC(=O)NNC(=O)C(C)n1nc(nn1)N2CCOCC2 RJF01838 c1c(cc(cc1C(F)(F)F)NC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(F)(F)F S05471 Cc1c(c(nc(n1)SC)O)CC2CC2 RJF00481 Cc1ccc(c(c1)OC(=O)c2ccc(cc2)C(F)(F)F)NC(=O)c3ccc(cc3)C(F)(F)F S14570 COCc1cc(nc(n1)S)O RJF00490 COc1cc(cc(c1)OC)N2C(=O)C=CC2=O S12653 Cc1c(c(nc(n1)c2cccnc2)O)CC3CC3 RJF00488 COCc1cc(nc(n1)SC)O RJF00491 Cc1ccc2c(c1)nc(o2)c3cccs3 S14577 Cc1ccc(n1c2ccc(cc2)c3csnn3)C SEW00931 CC1c2ccsc2CCN1C(=S)NC SEW00936 CCOC(=O)C1=C(OC(=C(C12c3ccccc3NC2=O)C#N)N)c4ccccc4 S14430 c1ccc(cc1)N2C(=O)CC(C2=O)Sc3cccs3 S14437 c1cc(c(c(c1)Cl)Cn2nc(nn2)N3CCCCC3)Cl RJF00316 CCOc1ccc(cc1)N2C(=O)c3ccccc3C2=O S05509 c1ccc2c(c1)C(=O)N(C2=O)Cc3cccnc3 S05517 CCOc1ccc(cc1)NCN2C(=O)c3ccc(cc3C2=O)[N+](=O)[O-] S05532 c1cc(ccc1NCN2C(=O)c3ccc(cc3C2=O)[N+](=O)[O-])Cl S05541 c1cc(sc1)c2ccc(s2)/C=N/O SEW02193 Cc1ccc2c(c1)nc(o2)c3ccc(cc3)C(C)(C)C S14575 CC(C(=O)NNC(=O)c1ccc(cc1)Cl)n2nc(nn2)N3CCOCC3 RJF01846 CC(C(=O)NNC(=O)c1ccccc1Cl)n2nc(nn2)N3CCOCC3 RJF01849 CC(C(=O)NNS(=O)(=O)c1cccc(c1)C(F)(F)F)n2nc(nn2)N3CCOCC3 RJF01850 CCN(CC)C(=O)Oc1c(c(nc(n1)c2ccccn2)COC)CC3CC3 RJF01823 CC(C)NC(=O)NNC(=O)Cn1nc(nn1)N2CCCC2 RJF01824 CC(C(=O)NNS(=O)(=O)c1ccc(cc1)Cl)n2nc(nn2)N3CCOCC3 RJF01851 CC(C(=O)NN)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01855 c1cc(c(cc1NC(=O)/C=C/C(=O)O)Cl)F S12356 c1cc(c(cc1N2C(=O)C=CC2=O)Cl)F S12357 c1cc(c(cc1N2C(=O)CC(C2=O)N3CCCCC3)Cl)F S12372 c1cnccc1/C=N/NC(=O)Cn2nc(nn2)N3CCCC3 RJF00313 CCCc1c(c(nc(n1)c2ccccn2)OC(=O)N(CC)CC)Cc3c(cccc3Cl)F RJF01813 CNC(=O)NNC(=O)Cn1nc(nn1)N2CCCCC2 RJF01814 Cc1ccc(cc1C)N2C(=O)CC(C2=O)N3CCOCC3 S12388 c1cc(cc(c1)Cl)/C=C/[N+](=O)[O-] S05525 Cc1cc(c(c(c1)C)NC(=S)N)C S03098 c1cc(sc1)CNC(=O)NC(=O)c2ccc(cc2)c3csnn3 SEW01152 c1cc(ccc1/C(=N/OC(=O)c2ccc(cc2Cl)Cl)/Cn3nc(nn3)N4CCCCC4)Cl RJF00385 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N\c3cc(cc(c3)C(F)(F)F)C(F)(F)F S05288 CC(=O)c1cc2c([nH]1)ccs2 SEW02099 C/C(=N\C(=S)c1ccc(cc1)Cl)/N(C)C SEW02102 Cc1nc(sn1)c2ccc(cc2)Cl SEW02104 c1cc(c(cc1F)F)NC(=S)NNC(=O)Cn2nc(nn2)N3CCCCC3 RJF00347 CCOC(=O)/C(=C/c1ccc(s1)c2cccs2)/C#N SEW02158 CCCc1cc(=O)n2c(csc2n1)c3ccc(cc3)Cl RJF01919 Cc1ccc(cc1C)N2C(=O)C=C(C2=O)c3ccccc3 S12401 CCSc1nc2ccc(cc2c(=O)n1c3ccc4c(c3)OCCO4)C S05371 CC1=CC(=O)N(C1=O)c2ccc(cc2)F S12423 c1ccc(cc1)CS/C(=N/N=C/c2cccs2)/N S12431 CCNC(=O)/C(=C/c1cccs1)/C#N S05396 Cc1ccc2c(c1)nnn2CNc3ccc(cc3)OC(F)(F)F S14460 CC(C)Cc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3ccc(cc3)Cl S14471 Cc1ccc(c(c1)C)N2C(=O)C=CC2=O S12378 c1ccnc(c1)/C=N/NC(=O)Cn2nc(nn2)N3CCCC3 RJF00315 c1cc(c(cc1F)F)NC(=S)NNC(=O)Cn2nc(nn2)N3CCCC3 RJF00349 c1cc(ccc1/C(=N/OC(=O)c2ccc(cc2Cl)Cl)/Cn3nc(nn3)N4CCOCC4)Cl RJF00358 COc1ccc(cc1)/C=N/N=C(\N)/SCc2ccc(cc2)F S12409 COc1ccc(cc1)/C=N/N=C(\NC(=O)Nc2ccccc2)/SCc3ccc(cc3)F S12410 C1CC1NC(=S)NCCO RJF00363 c1cc(sc1)c2ccc(s2)/C=N/Nc3ccc(cn3)[N+](=O)[O-] SEW02176 CN(C)/N=C(\Cn1nc(nn1)N2CCCC2)/c3ccc(cc3)Cl RJF00318 CC(C)Cc1ccc(cc1)C(=O)CC(c2ccc(cc2)C(F)(F)F)Sc3ccccc3N S14489 C=CC/N=C\1/NC(=O)C(S1)CC(=O)Nc2ccc(cc2)Cl S05934 CCCCCCCc1c(n[nH]c1O)COC RJF01892 CC(C(=O)NNC(=O)NC(C)(C)C)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01894 c1cc(cnc1)/C=C/2\C(=O)N(C(=S)S2)Cc3ccncc3 S03142 c1cc(c(cc1NC(=S)NNC(=O)Cn2nc(nn2)N3CCCC3)Cl)F RJF00351 c1cc(ccc1CNC(=O)N)F S14532 CCCc1c(c(nc(n1)c2ccccn2)OC(=O)N(C)C)Cc3c(cccc3Cl)F RJF01811 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N\C3CC3 RJF00384 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)OC S02819 CCCC1c2ccsc2CCN1C(=S)Nc3ccccc3C(=O)OC SEW01146 CCCC1c2ccsc2CCN1C(=S)NC SEW01147 CC(C(=O)NNC(=O)c1cc(ccc1OC)OC)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01905 Cc1ccc(cc1)CN2C(=O)C=CC2=O S14672 Cc1ccc(cc1)CN2C(SCC2=O)c3cccnc3 S14674 c1cnccc1CN2CN(C(=S)SC2)Cc3ccncc3 S14683 c1cc(cnc1)CN2CN(C(=S)SC2)Cc3cccnc3 S14685 COc1cccc(c1)Nc2nnc(s2)S S03055 c1ccc(cc1)CCN2C(=O)CSC2=S S03086 CCOC(=O)C1CSC(C(=O)N1)CC(=O)Nc2ccccc2 S14689 c1ccc2c(c1)CCC/C(=C\c3ccc(cc3)Cl)/C2=O S14708 c1ccc(cc1)C(=O)NC(=S)Nc2c(cccc2Cl)Cl S03092 CNC(=O)NNC(=O)Cn1nc(nn1)N2CCCC2 RJF01812 c1cc(cc(c1)Cl)n2c(nnn2)SCC(=O)c3ccc(cc3)Cl S12597 c1ccc(cc1)/C=C/2\C(=O)N(C(=N2)c3ccccc3)c4ccccc4 S12548 c1ccc(cc1)C(C#N)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S12549 Cc1ccc(cc1N2C(=O)C3CCC(CC3C2=O)C)F S12865 Cc1ccc(cc1NC(=O)C2C3CC(C2C(=O)O)C=C3)F S12866 c1ccc(cc1)c2csc(n2)NC(=N)NC(=N)N.Cl RJF00586 c1cc(c(cc1Cl)NC(=N)NC(=N)N)Cl.Cl RJF00588 c1cc(c(c(c1)Cl)/N=C\2/NCCS2)Cl S03102 c1ccc(cc1)C(=S)NCc2cccnc2 S03154 c1cc(cc(c1)Cl)NC(=S)NNC(=O)C2CC2 RJF00638 c1cc(c(cc1NC(=N)NC(=N)N)Cl)Cl.Cl RJF00648 c1ccc(cc1)c2ccc(cc2)C(=O)CSc3nnnn3c4cccc(c4)Cl S12598 c1cc(sc1)C(=O)N2CCc3c(ccs3)C2c4ccc(cc4)Cl SEW01022 COCc1cc(nc(n1)c2ccccc2)O RJF00617 c1cc(c(cc1Nc2ncnc(n2)N)Cl)Cl RJF00656 COc1cc(ccc1OC(=O)c2cc(c(c(c2)OC)OC)OC)C=C(C#N)C#N S03148 c1ccc(cc1)C(=S)NCCc2ccccn2 S03155 CC(C)(C)C(=O)Oc1ccc(cc1)c2csnn2 SEW01160 c1cc(ccc1c2csnn2)OS(=O)(=O)c3ccc(c(c3)Cl)F SEW01163 c1ccc(c(c1)S(=O)(=O)Oc2ccc(cc2)c3csnn3)Cl SEW01165 CN(C)C(=O)Nc1ccccc1 S03159 CCCCNC(=O)Oc1ccc(cc1)c2csnn2 SEW01169 c1cc(ccc1/C=N/Nc2ccc(cc2)c3cnco3)Cl SEW01176 c1cc2c(cc1[N+](=O)[O-])NC3(N2)CCCCC3 S03183 CC(C)NC(=O)N1CCc2c(ccs2)C1c3ccc(cc3)Cl SEW01027 c1ccc(c(c1)c2nc3ccc(cc3c(=O)o2)I)Cl S12479 c1cc(ccc1C2=NCCc3c2ccs3)OC(F)(F)F SEW02189 CN1C2(CC(O1)COS(=O)(=O)c3ccc(cc3)[N+](=O)[O-])C4CC5CC(C4)CC2C5 S14549 c1cc(sc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N S14752 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)NNC(=S)NC(=O)c3ccc(cc3)Cl RJF01964 c1cc(ccc1/C=N/c2ccc(cc2)c3cnco3)[N+](=O)[O-] SEW01181 c1ccc2c(c1)cc(o2)C3N(C(=O)CS3)c4ccc(cc4)F S12820 COc1cc(cc(c1OC)OC)Nc2ncnc(n2)N RJF00567 COc1ccccc1Nc2ncnc(n2)N RJF00568 c1ccc(c(c1)NC(=N)NC(=N)N)Cl.Cl RJF00570 Cc1ccc(cc1NC(=O)/C=C\C(=O)O)F S12851 Cc1ccc(cc1N2C(=O)C=CC2=O)F S12852 CN1C2(CC(O1)COS(=O)(=O)c3ccc(cc3)Cl)C4CC5CC(C4)CC2C5 S14548 Cc1ccc(c(c1)NC(=O)c2ccc(cc2)C(C)(C)C)OC(=O)c3ccc(cc3)C(C)(C)C S14557 c1cc(ccc1C(=O)Nc2cc(ccc2OC(=O)c3ccc(cc3)C(F)(F)F)Cl)C(F)(F)F S14558 c1cc(ccc1c2csnn2)OC(=O)Nc3ccc(cc3)Cl SEW01171 Cc1c(c(c(o1)/N=C/c2ccc(cc2)F)c3ccc(cc3)F)C#N S12792 c1cc(cc(c1)[N+](=O)[O-])c2nnco2 SEW01182 CSc1ccccc1Nc2ncnc(n2)N RJF00562 COCc1cc(nc(n1)NC(=N)Nc2c(cccc2F)F)O RJF00563 c1cc(ccc1c2cnco2)NC(=O)/C=C\C(=O)O SEW01186 Cc1ccc(cc1)S(=O)(=O)NCCc2cccs2 S12721 CCOC(=O)C1=C(NC(=O)NC1c2cc(cc(c2)OC)OC)C S12701 COc1ccc(cc1OC)c2cc(=S)sc(c2C#N)N SEW01110 c1cc(ccc1c2csnn2)OC(=O)c3ccc(cc3)Cl SEW01112 COc1ccc(cc1N2C(=O)c3cccnc3C2=O)Cl S12618 CC(=O)c1ccc(s1)c2cccs2 SEW02215 c1ccc(c(c1)/C=N/OCc2cc(cc(c2)Br)Br)OC(F)(F)F SEW02219 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(cc3)Br S03023 C#Cc1cccc(c1)NC(=N)NC(=N)N.Cl RJF00559 c1cc(sc1)CCNC(=O)c2ccc(cc2)C(F)(F)F SEW01174 c1cc(ccc1/C=N/c2ccc(cc2)c3cnco3)Cl SEW01178 CC1(CC(=CC(=O)C1)NCCCCCCCCNC2=CC(=O)CC(C2)(C)C)C S03035 Cc1cc(c(n1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)C(=O)C(F)(F)F SEW01072 Cc1ccnc(c1)N2C(=O)CCC2=O S14593 c1cc(cnc1)N2C(=O)CCC2=O S14602 c1ccnc(c1)c2n[nH]c(=S)s2 S12761 c1ccc(c(c1)/C=C\2/C(=O)N(C(=S)S2)c3ccc(cc3)Cl)[N+](=O)[O-] S12757 c1cc(ccc1c2csnn2)OC(=O)C3CC3 SEW01161 COc1ccc(cc1NCN2C(=O)c3ccccc3C2=O)Cl S12674 c1cc(ccc1c2nnc(o2)S)C(F)(F)F S12682 CN1C(C2CCCc3ccccc3C2=N1)c4ccc(cc4)F S14629 CC(C(=O)NNC(=O)C1CC1)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01857 CN(C)/C=C/C(=O)c1ccc(s1)c2cccs2 SEW02221 C/C(=C\c1cc(cc(c1)OC)OC)/[N+](=O)[O-] S12685 CCOC(=O)/C(=C/c1cc(cc(c1)OC)OC)/C#N S12689 CC1=N/C(=C\c2cc(cc(c2)OC)OC)/C(=O)O1 S12696 CS(=O)(=O)NNC(=O)Cn1nc(nn1)c2ccccc2C(F)(F)F RJF01866 CC(C(=O)NNS(=O)(=O)c1cccc(c1)Cl)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01870 COc1ccc(cc1)C(=O)Oc2ccc(cc2)c3csnn3 SEW01113 COc1ccc(cc1N2C(SCC2=O)c3cccnc3)Cl S12663 CC(C(=O)NNC(=O)C)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01858 Cc1ccc(cc1)S(=O)(=O)N(CCc2cccs2)CC(=O)O S12728 CN(C)C(=O)Oc1cc(nc(n1)c2ccncc2)COC RJF00498 Cc1c(c(on1)C)C(=O)Oc2ccc(cc2)c3csnn3 SEW01116 COc1cc(cc(c1)OC)C(C[N+](=O)[O-])Sc2ccccc2N S12686 CC(C)(C)C(=O)NNC(=O)Cn1nc(nn1)c2ccccc2C(F)(F)F RJF01864 CC(C(=O)NNS(=O)(=O)c1cccc(c1)C(F)(F)F)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01865 Cc1ccc(cc1)/N=N\c2c(nn(c2O)c3ccccc3)C(=O)OC SEW02279 COC(=O)c1c(c(n(n1)c2ccccc2)O)/N=N\c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW02280 Cc1cc(c(cc1C)/N=c/2\oc(cs2)C(C)(C)C)C RJF00536 CC(C)(C)C(=O)O/N=C(/c1ccc(cc1)c2csnn2)\N SEW01092 Cc1ccccc1C(=O)Oc2ccc(cc2)c3csnn3 SEW01114 Cn1cc(c(=O)c2c1cccc2)c3ccccc3C(=O)N S12845 c1cc(cc(c1)[N+](=O)[O-])NC(=O)/C=C/C(=O)O S12846 c1cc(cc(c1)[N+](=O)[O-])N2C(=O)C=CC2=O S12847 Cc1ccc(cc1NC(=S)N)F S12850 COc1cc(cc(c1)OC)N2C(=O)CSCC2=O S12661 CC(C)(C)OC(=O)/C(=C/c1cc(cc(c1)OC)OC)/C#N S12690 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(cc3)F S03038 c1ccc(cc1)NC(=O)N2CCc3c(ccs3)C2c4ccc(cc4)C(F)(F)F SEW01212 c1ccc(cc1)c2nc(no2)c3ccc(cc3)c4csnn4 SEW01076 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc(cc4)[N+](=O)[O-] SEW01080 c1ccnc(c1)N2C(=O)COCC2=O S14596 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CCCC(=O)O S14611 c1cc(ccc1c2csnn2)c3csnn3 SEW01099 COc1ccc(cc1NC(=O)CSCC(=O)O)Cl S12612 c1cc(ccc1C2c3ccsc3CCN2S(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)Cl SEW01034 c1ccc(c(c1)/C=N\OC(=O)c2ccsc2)OC(F)(F)F SEW02210 c1cc(ccc1c2csnn2)C(=S)N SEW01067 c1ccc(c(c1)c2nnn(n2)CC(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F)C(F)(F)F RJF01863 Cc1ccc(cc1Cl)NC(=O)n2c(ccn2)c3ccc(s3)c4cccs4 SEW02232 Cc1ccnc(c1)NC(=O)CCC(=O)O S14589 c1ccnc(c1)N2C(=O)CCC2=O S14591 c1ccnc(c1)NC(=O)COCC(=O)O S14594 CC(=O)O/N=C(/c1ccc(cc1)c2csnn2)\N SEW01091 c1ccc(c(c1)c2nnn(n2)CC(=O)NNS(=O)(=O)c3cccc(c3)Cl)C(F)(F)F RJF01869 CCCNC(=O)NNC(=O)C(C)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01877 CC(C(=O)N/N=C/C(C)(C)C)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01883 COc1cc(cc(c1OC)OC)C(=O)O/N=C/c2ccccc2OC(F)(F)F SEW02211 c1cc(ccc1C2C3=C(c4cc(ccc4OC3)F)OC(=C2C#N)N)Cl SEW02216 c1cc(ccc1NC(=O)/C=C/C(=O)O)Br S03020 COc1cc(cc(c1)OC)NC(=O)C2C3CC(C2C(=O)O)C=C3 S12657 Cc1c(c(nc(n1)SCC(=O)C(C)(C)C)O)CC=C RJF00446 c1ccc(c(c1)c2nnn(n2)CC(=O)NNS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F RJF01868 c1ccc(cc1)NN2C(=O)c3cccc4c3c(ccc4)C2=O S05575 CNN1C(=O)c2cccc3c2c(ccc3)C1=O S05578 CN(C)N1C(=O)c2ccccc2C1=O S05580 COc1ccc(cc1)CN2C(SCC2=O)c3ccccn3 S14637 Cc1c(cc(c(=O)o1)NC(=O)c2ccccc2)C(=O)C S14651 C/C(=N\Cc1ccccc1OC)/c2ccccc2O S14654 c1cc(ccc1Nc2ncnc(n2)N)Br RJF00545 CC(C(=O)NNC(=S)Nc1ccccc1Cl)n2nc(nn2)N3CCOCC3 RJF01837 CC(C(=O)NN)n1nc(nn1)N2CCOCC2 RJF01826 COc1ccc(cc1)C(=O)n2c(ccn2)c3ccc(s3)c4cccs4 SEW02261 c1cc(sc1)c2ccc(s2)C(=O)c3ccc(cc3F)F SEW02249 c1cc(c(cc1Cl)Cl)OCc2nc(on2)c3ccoc3 SEW02251 c1cc(cc(c1)C(F)(F)F)c2nc(no2)COc3ccc(cc3Cl)Cl SEW02252 c1cc(ccc1CN2CN(C(=S)SC2)Cc3ccc(cc3)F)F S14677 CCOC(=O)C1(C(CC(=CC1=O)c2ccc(cc2)OC)c3ccc4ccccc4c3)CCC#N S14636 CN1/C(=N/c2ccc(cc2)OC)/SCC(=N1)c3ccccc3 S14773 COc1cc(cc(c1)OC)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)Cl S12705 COc1cc(cc(c1)OC)/C=N/N=C\2/NC(=O)CS2 S12737 c1ccc2c(c1)CCC/C(=C\c3ccc(cc3)F)/C2=O S14624 CC(C(=O)NNC(=S)NC)n1nc(nn1)N2CCOCC2 RJF01836 c1ccc2c(c1)C(=O)N(C2=O)c3ccc(cc3)Cl S05513 c1ccc2c(c1)C(=O)N(C2=O)Cc3ccncc3 S05514 Cc1cc(ccc1F)NC(=S)NCCO S05496 Cc1ccc(c(c1)C)/N=C\2/NCCS2 S03044 Cc1c(nc(nc1O)S)COC RJF00506 CN(C)C(=S)Nc1ccc(cc1F)F RJF00539 c1cc(c(c(c1)F)NC(=N)NC(=N)N)F.Cl RJF00542 c1cc(oc1)C(CC(=O)c2ccc(cc2)F)CC(=O)c3ccc(cc3)F S05892 c1ccc2c(c1)CCC/C(=C\c3c(cccc3Cl)F)/C2=O S14625 COc1ccc(cc1)CN2C(SCC2=O)c3cccnc3 S14631 CC(C(=O)NNS(=O)(=O)c1ccc(cc1)Cl)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01871 CC(C(=O)NNC(=O)NC)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01872 CCCC1c2ccsc2CCN1C(=S)Nc3ccc(cc3Cl)Cl SEW01145 Cc1cc(ccc1F)n2c(nnn2)S S05501 c1ccc(cc1)Oc2ccc(cc2)NCN3C(=O)c4ccc(cc4C3=O)[N+](=O)[O-] S05535 c1ccc2c(c1)C(C(=O)N2)(C3C(=O)NC(=O)NC3=O)C4C(=O)NC(=O)NC4=O S02822 Cc1c(c(c(c(c1C)NC(=O)/C=C/C(=O)O)C)C)NC(=O)/C=C/C(=O)O S02829 c1ccc(c(c1)c2nnn(n2)CC(=O)N/N=C/c3c(cccc3Cl)Cl)C(F)(F)F RJF01906 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(cc3)F)O RJF01910 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(cc3)F)OC(=O)N(C)C RJF01911 Cc1ccc(o1)/C=C/2\CCCc3ccccc3C2=O S14622 Cc1cccc(c1NC(=N)NC(=N)N)Cl.Cl RJF00547 c1cc(cc(c1)Nc2ncnc(n2)N)C(F)(F)F RJF00552 c1cc(c(c(c1)F)Nc2ncnc(n2)N)F RJF00553 CN(C)C(=S)Nc1ccc(cc1)S(=O)(=O)N2CCCCC2 S03040 c1ccc2c(c1)CCC/C(=C\C3CCCCC3)/C2=O S14623 CC(C)(C)c1ccc(cc1)OC(=O)NC(=O)c2ccc(cc2)c3csnn3 SEW01156 CSc1cccc(c1)NC(C#N)c2ccccc2 S12787 CC(=O)Nc1ccc(cc1)C2=N/C(=C/c3cccs3)/C(=O)O2 S05424 c1cc(ccc1Cc2ccc(cc2)N3C(=O)C=CC3=O)N4C(=O)C=CC4=O S12770 CCCC1c2ccsc2CCN1C(=O)Nc3c(occ3c4c(cccc4Cl)Cl)C SEW01143 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)Cl)OCC(=O)OCC(=O)c4ccc(cc4)Cl RJF01928 c1ccc(cc1)C(C#N)Nc2ccc(cc2)C(F)(F)F S12781 COc1cccc(c1)NC(=N)NC(=N)N.Cl RJF00557 Cc1cccc(c1Nc2ncnc(n2)N)Cl RJF00558 CCCC1c2ccsc2CCN1C(=O)c3ccc(cc3)Cl SEW01124 c1cc(ccc1c2csnn2)C(=O)N SEW01125 COc1ccc(cc1)N2C(=O)CC(C2=O)c3ccc(cc3)[N+](=O)[O-] S12475 c1cc(c(cc1Cl)Cl)c2nc3ccc(cc3c(=O)o2)I S12478 Cc1ccc(cc1)n2c(=O)n(c(=O)s2)Cc3ccc(cc3)F S14530 COc1ccccc1CCNC(=O)N S14531 c1cc(c(cc1NC(=S)NNC(=O)Cn2nc(nn2)N3CCCCC3)Cl)F RJF00348 c1ccc(cc1)c2ccc(cc2)C(=O)CSc3nnc(s3)c4ccccn4 S12775 c1cc(ccc1c2csc(n2)NC(=N)NC(=N)N)Cl.Cl RJF00587 CCCC1c2ccsc2CCN1C(=O)Nc3ccc(cc3)Cl SEW01141 c1ccnc(c1)c2c(nnc(n2)c3ccccn3)c4ccccn4 S12786 c1ccc(cc1)CCN2CN(C(=S)SC2)CCc3ccccc3 S03085 CO/C=C\1/C(=O)N(C(=S)S1)CCc2ccccc2 S03088 c1ccc(c(c1)Nc2ncnc(n2)N)Cl RJF00607 c1ccc2c(c1)CCC/C(=C\c3cccs3)/C2=O S14713 COc1ccc(cc1)CNC2(C(=O)c3ccccc3C2=O)NC(=O)c4ccc(cc4)C(F)(F)F S14715 c1ccc(cc1)NC(=O)NCCO S03160 CN(C)C(=O)Sc1nnc(n1c2ccc(cc2)Cl)C3CC3 RJF00630 c1ccc2c(c1)CC/C(=C\C3CCCCC3)/C2=O S12902 CN1C(C2CCCc3ccccc3C2=N1)c4ccc(cc4)N(C)C S14720 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)Cc3ccc(cc3)NC(=S)NC(=O)c4ccccc4 S03177 c1cc(sc1c2ccno2)/C(=N/O)/N SEW02268 CC(C(=O)NNC(=O)c1ccc(cc1Cl)Cl)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01903 Cc1ccc(cc1)CNC(=O)/C=C/C(=O)O S14671 c1cc(ccc1c2csnn2)OS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW01162 c1ccc2c(c1)CCC/C(=C\c3ccc(cc3Cl)Cl)/C2=O S14710 COc1ccc(cc1OC)CCNC(=S)c2ccccc2 S03157 Cc1ccc(cc1NC(C#N)c2ccccc2)F S12872 CC(C)c1ccc(cc1)C2C(=Cc3ccccc3O2)[N+](=O)[O-] S14741 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)Cl)OCC(=O)OCC(=O)C(C)(C)C RJF01933 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)C(F)(F)F)C(=O)O S12890 c1cc(cc(c1)Cl)n2c(=S)[nH]nn2 S03205 CC(C)c1ccc(cc1)C(C[N+](=O)[O-])Sc2ccccc2N S14726 c1ccc2c(c1)CC/C(=C\c3ccncc3)/C2=O S12909 c1c(cc(cc1C(F)(F)F)NC(=S)N2CCCCCC2)C(F)(F)F S05649 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(cc3)F)OC(=O)c4ccco4 RJF01941 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(cc3)F)OC(=O)c4cc(ccc4OC)OC RJF01942 c1cc(sc1)C(=O)Oc2ccc(cc2)c3csnn3 SEW01118 CCCCCCCc1c(n[nH]c1O)C RJF01893 CC(C(=O)NNC(=O)c1ccc(cc1)Cl)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01896 c1cc(c(c(c1)Cl)NC(=O)NC(=O)c2ccc(cc2)c3csnn3)Cl SEW01132 Cc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)Cl)OCC(=O)OCC(=O)c4ccccc4 RJF01934 CCOC(=O)N/N=C(\C)/COc1ccc(cc1)c2csnn2 SEW01200 c1cc(ccc1C2c3ccsc3CCN2C(=O)c4ccc(cc4)Cl)C(F)(F)F SEW01204 c1cc(ccc1c2cnco2)N3C(=O)C4C5CC(C4C3=O)C=C5 SEW01192 C/C(=N\Nc1cc(cc(c1)Cl)Cl)/COc2ccc(cc2)c3csnn3 SEW01196 c1ccc(c(c1)NC(=S)NNC(=O)c2ccncc2)Cl S03292 CC(C)(C)C(=O)Cn1nc(nn1)c2ccncc2 RJF01944 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(cc3)F)OS(=O)(=O)c4cccc(c4)C(F)(F)F RJF01946 C/C(=N\CCc1ccc(c(c1)OC)OC)/c2ccc3ccccc3c2 S05776 c1cc(oc1)CNC(=S)Nc2ccc(cc2)Oc3ccc(cc3)Cl S05784 Cc1ccc(cc1Cl)/N=C\2/NCCS2 S03124 c1ccnc(c1)/C=C/2\C(=O)N(C(=S)S2)Cc3ccncc3 S03143 Cc1ccc(cc1)NC(=N)NC(=N)N.Cl RJF00649 Cc1ccc(cc1Cl)NC(=N)NC(=N)N.Cl RJF00655 c1cc(sc1c2ccno2)S(=O)(=O)N3CCOCC3 SEW02275 Cc1ccc(cc1NC(=O)CSCC(=O)O)F S12870 CCN(CC)S(=O)(=O)c1ccc(s1)c2ccc(s2)S(=O)(=O)N(CC)CC SEW02299 c1ccc2c(c1)CCC/C(=C\c3ccc(cc3)[N+](=O)[O-])/C2=O S14709 CCOC(=O)NC(=S)Nc1ccc(cc1)Oc2ccc(cc2)Cl S05793 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(cc3)F)OC(=O)COC RJF01945 CN1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)C(F)(F)F S12903 c1ccc2c(c1)CC/C(=C\c3ccc(cc3)F)/C2=O S12910 c1cc(ccc1c2csnn2)OC/C(=N/O)/N SEW01203 CC(C)(C)c1ccc(cc1)C(=O)N2CCc3c(ccs3)C2c4ccc(cc4)C(F)(F)F SEW01206 c1cc(ccc1C2=NCCc3c2ccs3)C(F)(F)F SEW01177 c1cc(cnc1)/C=N/c2ccc(cc2)c3cnco3 SEW01179 Cc1ccc(cc1NCN2C(=O)c3ccccc3C2=O)F S12876 CCOC(=O)NC(=S)Nc1cc(cc(n1)C)C S05810 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2c5ccccc5 S12923 Cc1ccc(cc1)CNC2(C(=O)c3ccccc3C2=O)NC(=O)c4ccc(cc4)C(F)(F)F S14716 c1cc(sc1)c2ccc(s2)c3ccnc(n3)N SEW02312 c1cc(ccc1CNC(=N)NC(=N)N)C#N.Cl RJF00661 c1cc(ccc1NC(=N)NC(=N)N)Oc2ccc(cc2)Cl.Cl RJF00668 c1ccc2c(c1)CC/C(=C\c3ccc(cc3)C(F)(F)F)/C2=O S12899 Cc1ccc(cc1)NC(=N)Nc2nc(cc(n2)O)COC RJF00673 Cc1cccc(c1)Nc2nnc(s2)S S03258 c1cc(c(cc1NC(=S)NN)Cl)Br S03260 CC(C)c1ccc(cc1)/C=C/[N+](=O)[O-] S14725 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4ccccc4Cl RJF01953 CC(C)c1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccccc3 S14727 c1cc(ccc1c2ccc(s2)C(=O)N)Cl SEW01166 c1ccc(cc1)C(C#N)Nc2ccc(cc2Cl)Cl S12780 c1ccc(cc1)C(C#N)Nc2ccc(cc2)I S12784 c1ccc(cc1)c2c(nnc(n2)c3ccccn3)c4ccccc4 S12785 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)C(F)(F)F)C(=O)C1)C S14754 Cc1cc(nc(n1)NC(=N)Nc2ccc(cc2Cl)Cl)O RJF00680 c1cc(c(cc1C(F)(F)F)NC(=S)Nc2ccc(cc2F)F)N3CCCCC3 RJF00686 c1cc(c(cc1C(F)(F)F)NC(=S)Nc2ccc(cc2F)F)N3CCCC3 RJF00689 CCC(C)(C)NC(=S)N(C)C S05723 Cc1c(c(c(c(c1C)N2C(=O)C=CC2=O)N3C(=O)C=CC3=O)C)C S05718 c1cc2c(cc1/N=C/c3ccc(s3)[N+](=O)[O-])OCCO2 S05765 Cc1c(cnc(n1)C2CC2)c3nc(sn3)Nc4ccccc4 SEW02334 c1cc(ccc1NC(=O)/C=C/C(=O)O)F S03036 Cc1ccc(cc1N2C(=O)CC(C2=O)Sc3ccccc3N)F S12858 c1cc(ccc1NC(=N)NC(=N)N)F.Cl RJF00572 CC(C)(C)c1cs/c(=N\c2ccc(cc2F)F)/o1 RJF00573 c1cc(c(c(c1)Cl)Cl)NC(=N)NC(=N)N.Cl RJF00579 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=S)Nc4ccc(cc4F)F)C(F)(F)F RJF00687 CCCNC(=O)NNC(=O)Cn1nc(nn1)c2cccc(c2)C(F)(F)F RJF02124 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)Cc3ccc(cc3)F RJF02127 CN1C(C2CCCc3ccccc3C2=N1)c4cccs4 S14719 c1cc(ccc1C2C(CCC(=O)N2)[N+](=O)[O-])Cl S06284 c1cc(ccc1OS(=O)(=O)c2ccc(s2)c3ccno3)Cl SEW02318 Cc1ccc(o1)/C=C/2\CCc3ccccc3C2=O S12912 COCc1cc(nc(n1)NC(=N)Nc2ccc(c(c2)Cl)Cl)O RJF00672 Cc1ccc(cc1N2C(=O)c3cccnc3C2=O)F S12863 c1ccc(c(c1)/N=C/c2ccc(s2)[N+](=O)[O-])Br S05768 c1cc(cnc1)CNC(=S)Nc2ccc(cc2)Oc3ccc(cc3)Cl S05783 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccccc3)C(=O)C1)C S14753 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=S)Nc4cc(cc(c4)Cl)Cl)C(F)(F)F RJF00692 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4ccc(cc4Cl)Cl RJF01956 Cc1cc(cc(c1)NC(=S)NC2CCCCC2)C S05696 Cc1cc(ccc1NC(=S)N/N=C/c2cccs2)F S06326 c1cc(ccc1C2CCCCC2)NC(=N)NC(=N)N.Cl RJF00719 c1cc(c(cc1C(F)(F)F)NC(=S)NC2CCCCC2)Cl S05698 Cc1c(c(c(c(c1C)C)NC(=O)/C=C/C(=O)O)NC(=O)/C=C/C(=O)O)C S05717 CC(C)(C)C1=NN(/C(=N\c2ccc(cc2)OC)/SC1)C S14782 CC(C)(C)C(=O)Oc1cc2c(cc1Cl)c(cc(=O)o2)COC RJF02001 Cc1c2ccccc2n3c1/C(=N/Nc4ccc(cc4Cl)Cl)/CC3 SEW02314 Cc1c2ccccc2n3c1/C(=N/Nc4cccc(c4)C(F)(F)F)/CC3 SEW02315 CC(C)(C)C1=NN(/C(=N\c2ccc(cc2)F)/SC1)C S14780 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4cc(ccc4OC)OC RJF01965 Cc1c2ccccc2n3c1/C(=N/Nc4ccccc4)/CC3 SEW02310 Cc1c2ccccc2n3c1/C(=N/Nc4ccc(cc4)C(F)(F)F)/CC3 SEW02311 c1cc(cnc1)C=C(C#N)C#N S14755 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cccs3)C(=O)C1)C S14757 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C/c2ccccc2Cl SEW02351 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C/c2ccc(cc2Cl)Cl SEW02355 c1cc(cc(c1)OS(=O)(=O)c2ccc(s2)c3ccc(s3)S(=O)(=O)Oc4cccc(c4)C(F)(F)F)C(F)(F)F SEW02305 CN1/C(=N/c2ccccc2Cl)/SCC(=N1)c3ccccc3 S14771 CC(C)Cc1ccc(cc1)C2=CC(C(C(=O)N2)C(=O)N)c3ccc(cc3)C#N S14774 CC(C)(C)c1ccc(cc1)c2nc(nn2c3ccccc3)OS(=O)(=O)c4ccc(cc4)Cl S14745 c1cc(ccc1C2C(=C(OC3=C2C(=O)CCC3)N)C#N)Cl S14750 Cc1ccc2c(cc(nc2c1)c3ccc(cc3)NC(=O)C)C(=O)O S05805 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4ccc(cc4)Cl RJF01966 c1cc(sc1)c2ccc(s2)c3ccnc(n3)S SEW02319 CC(=O)c1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3N S05855 CCCc1cc(=O)oc2c1ccc(c2)OC(C)C(=O)NNC(=S)Nc3ccc(c(c3)Cl)Cl RJF01986 CCCc1cc(=O)oc2c1ccc(c2)OC(C)C(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F RJF01991 CSc1ccccc1NC(=N)NC(=N)N.Cl RJF00550 COc1ccc(cc1)CNC(=O)/C=C/C(=O)O S14618 COc1ccc(cc1)CN2C(=O)C=CC2=O S14619 c1ccc2c(c1)CCC/C(=C\c3ccc(cc3)C(F)(F)F)/C2=O S14621 COc1ccc(cc1)c2csnn2 SEW01104 c1cc(cc(c1)Cl)S(=O)(=O)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl RJF02036 CCCc1cc(=O)oc2c1ccc(c2)OC(C)C(=O)NN RJF01970 c1cc(sc1)c2ccc(s2)c3ccnc(n3)SCC(=O)c4ccc(cc4)Br SEW02323 Cc1c2ccccc2n3c1/C(=N/O)/CC3 SEW02327 C1CN(CCN1C(=S)NCCCN2CCOCC2)C(=S)NCCCN3CCOCC3 S06099 CC(C(=O)N/N=C/c1c(cccc1Cl)Cl)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01884 c1cc(c(cc1F)Cl)NC(=O)CS(=O)(=O)Nc2ccc(cc2Cl)F SEW02241 COc1ccc(cc1)C(=O)c2ccc(s2)c3cccs3 SEW02248 Cc1c(c(n(n1)C)O)/N=N/c2ccc(c(c2)Cl)Cl SEW02342 c1c(cc(cc1Cl)Cl)c2nnn(n2)CC(=O)NN RJF02005 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)[N+](=O)[O-] SEW02367 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)NN RJF02110 c1ccc(c(c1)NC(=S)NNC(=O)Cn2nc(nn2)c3cccc(c3)C(F)(F)F)Cl RJF02111 Cc1cc(c(cc1CSC(=N)Nc2ccccc2Cl)C)CSC(=N)Nc3ccccc3Cl S05998 c1cc(ccc1C2C=C(C(=O)N2c3ccc(cc3)OC(F)(F)F)Nc4ccc(cc4)OC(F)(F)F)C(F)(F)F S14812 CN(c1c(cc(cn1)Cl)C(F)(F)F)/N=C/c2ccc(cc2)Cl SEW02352 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)NNS(=O)(=O)c3cccc(c3)Cl RJF01988 COc1ccccc1CNC(=O)/C=C/C(=O)O S14657 Cc1ccc(cc1)CN2CN(C(=S)SC2)Cc3ccc(cc3)C S14675 COc1ccc(cc1)CN2CN(C(=S)SC2)Cc3ccc(cc3)OC S14676 c1cc(ccc1NC(=O)CS(=O)(=O)Nc2ccc(cc2)Cl)Cl SEW02239 CC(C)(C)C1=NN(/C(=N\c2ccccc2)/SC1)C S14789 Cc1cccc(c1C)Nc2ncnc(n2)N RJF00650 c1c(cc(cc1Cl)Cl)c2nnn(n2)CC(=O)NNC(=O)C3CC3 RJF02010 Cc1c(cnc(n1)c2ccc(cc2)C(=O)N)c3nc(sn3)Nc4ccccc4 SEW02341 Cc1c2ccccc2n3c1C(=O)/C(=C/c4ccccc4)/C3 SEW02347 c1ccc(c(c1)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)N3CCCCCC3 S05660 CN(c1c(cc(cn1)Cl)C(F)(F)F)/N=C/c2ccc(cc2Cl)Cl SEW02354 Cc1cc(c(c(c1)C)Nc2ncnc(n2)N)C RJF00608 CN(C)C(=S)NCCCN1CCOCC1 S05872 c1ccc(cc1)COc2ccc(cc2)C=C(C#N)C#N S14803 Cc1cccc(c1C)NC(=N)NC(=N)N.Cl RJF00551 COc1cc(cc(c1OC)OC)NC(=N)NC(=N)N.Cl RJF00554 COCc1cc(nc(n1)SCC#C)O RJF00493 CC(C)(C)C(=O)CSc1nc(cc(n1)O)COC RJF00499 CN(C)C(=O)Oc1cc(nc(n1)SC)COC RJF00502 CCCCCCCC1C(=NN(C1=O)S(=O)(=O)c2ccc(cc2)Cl)C RJF01897 Cc1c2ccccc2n3c1C(=O)/C(=C/c4ccc(cc4Cl)Cl)/C3 SEW02344 Cc1c2ccccc2n3c1C(=O)/C(=C/c4ccc(cc4)C(F)(F)F)/C3 SEW02345 c1ccc(cc1)COc2ccc(cc2)/C=C/[N+](=O)[O-] S14801 c1ccc(cc1)CCNC(=S)c2ccccc2 S03158 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)N/N=C\c3c(cccc3Cl)Cl RJF02014 Cc1c(cccc1Cl)NC(=S)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl RJF02018 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C/c2ccccc2 SEW02349 c1ccc2c(c1)C(=O)C(C2=O)(NCc3ccc(cc3)F)NC(=O)c4ccc(cc4)C(F)(F)F S14717 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C/c2ccc(cc2)Cl SEW02353 c1cc(c(c(c1)Cl)/C=N\NC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl)Cl RJF02025 CN(c1c(cc(cn1)Cl)C(F)(F)F)/N=C/c2ccc(cc2O)O SEW02356 COc1ccc(cc1)CN2C(SCC2=O)c3ccncc3 S14634 c1ccc(c(c1)/C=N/NC(=O)Cn2nc(nn2)c3ccccc3C(F)(F)F)Cl RJF01881 COc1ccc(cc1)NC(=S)N2CCCC(=N2)c3ccccc3 S14798 Cc1ccc(cc1)NC(=S)N2CCCCCC2 S05653 CN(c1c(cc(cn1)Cl)C(F)(F)F)/N=C/c2ccccc2Cl SEW02350 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NNC(=S)Nc3ccc(cc3)C(F)(F)F RJF02022 CC(C)(C)NNC(=S)Nc1cccc(c1)F S06244 Cc1c2c(nn(c2oc(=O)c1Br)c3ccccc3)C(=O)OC SEW02287 COC(=O)c1c(c(n(n1)c2ccccc2)O)/N=N/c3cccc(c3Cl)Cl SEW02289 c1cc(c(c(c1)Cl)/C=N/N=C/2\NC(=O)CS2)F S12740 Cc1ccc(o1)/C=N/N=C/2\NC(=O)CS2 S12741 c1cc(ccc1NC(=N)NC(=N)N)F S05614 c1ccc2c(c1)c(c[nH]2)C=C(C#N)C#N S03064 c1cc(ccc1NC(=N)NC(=N)N)I.Cl RJF00651 Cc1ccc(cc1N2C(=O)COCC2=O)F S12860 c1cc(ccc1C2c3ccsc3CCN2C(=S)Nc4ccc(cc4Cl)Cl)C(F)(F)F SEW01214 c1cc(sc1c2ccno2)S(=O)(=O)N3CCCCC3 SEW02273 c1cc(sc1c2ccno2)S(=O)(=O)N3CCCC3 SEW02274 c1cc(sc1c2ccno2)S(=O)(=O)N3CCSCC3 SEW02276 c1cc(ccc1NC(=N)NC(=N)N)Cl.Cl RJF00576 c1cc(cc(c1)Cl)NC(=N)NC(=N)N.Cl RJF00580 CCCC1c2ccsc2CCN1C(=O)c3cc(cc(c3)OC)OC SEW01127 COc1ccccc1NC(=O)NC(=O)c2ccc(cc2)c3csnn3 SEW01131 c1cc(ccc1c2csnn2)C(=O)NC(=O)N3CCCCC3 SEW01137 CC(C)Cn1c(=O)c2ccccc2[nH]c1=S S06470 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)S(=O)(=O)Nc3cccc(c3)C(F)(F)F SEW02428 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)SC SEW02445 c1ccc(cc1)N/N=C/2\CCCc3c2c(co3)C(=O)O SEW02431 CN(c1c(cc(cn1)Cl)C(F)(F)F)/N=C/2\CCCc3c2c(co3)C(=O)O SEW02432 C=C1CC(=O)N(C1=O)c2ccc(cc2)OC(F)(F)F S14731 c1ccc(cc1)C(=O)N/C(=C\c2cccs2)/C(=O)Nc3ccc(cc3)F S14729 CNC(=S)Nc1ccc(cc1)Oc2ccccc2 S06147 CCn1c2ccccc2c3c1ccc(c3)N4C(=O)C=CC4=O S06150 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(ccc3F)F RJF02145 CCOC(=O)c1c(c(on1)N)C#N SEW02469 c1cc(c(c(c1)Cl)C(=O)NCc2ccc(s2)c3cccs3)Cl SEW02477 CCOC(=O)c1ccc(cc1)NC(=S)N(Cc2ccccc2)C(C)C S06114 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)c4cccc(c4)C(F)(F)F)C(F)(F)F SEW02446 CC(C)S(=O)(=O)c1c(n(nn1)c2cc(cc(c2)Cl)Cl)N SEW01273 c1cc(cc(c1)NC(=O)NCc2c(ccs2)COc3ccc(cc3)Cl)C(F)(F)F SEW02478 CC(C)Cc1ccc(cc1)C(=O)/C=C/N(C)C S14936 CC(=O)COc1ccc(cc1)c2csnn2 SEW01194 c1c(cc(cc1C(F)(F)F)NC(=S)NC2CCCCC2)C(F)(F)F S05695 c1ccc(cc1)n2c(nc(n2)O)c3cccs3 S14739 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)S(=O)(=O)Oc3ccc(cc3)F SEW02422 Cc1c(c(c(c(c1CSC(=N)N)C)CSC(=N)N)C)CSC(=N)N S06041 CC(C(=O)O)SC1CC(=O)N(C1=O)c2ccccc2 S12992 COc1cc(cc(c1OC)OC)C(=O)Nc2cc(ccc2Cl)C(F)(F)F S03315 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F RJF02123 CCOC(=O)/C(=C/c1ccccc1C)/C#N S12946 Cc1ccccc1C2NC(CS2)C(=O)O S12948 c1cc(cc(c1)NC(=O)C(Cl)(Cl)Cl)c2nnco2 SEW01227 Cc1c2ccc(cc2oc(=O)c1Cc3ccc(cc3)F)OS(=O)(=O)c4cccc(c4)Cl RJF01947 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)COC RJF01955 CN1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)F S12915 c1cc(sc1)c2ccc(s2)CNC(=O)c3ccc(cc3)Cl SEW02459 c1ccc2c(c1)cccc2/C=N/NC(=S)Nc3cccc(c3)Cl S03265 c1cc(cc(c1)Cl)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(ccc3F)F RJF02116 Cc1ccccc1/C=C(\C#N)/C(=O)OC(C)(C)C S12949 CC(C)NC(=O)NNC(=O)Cn1nc(nn1)c2cccc(c2)C(F)(F)F RJF02126 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)Cc3ccc(c(c3)Cl)F RJF02129 c1ccc2c(c1)c3c([nH]2)C(N(CC3)S(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(F)(F)F SEW02454 COc1ccc(cc1)/C=C/2\CCc3ccccc3C2=O S12919 c1ccc(c(c1)C(F)(F)F)NC(=S)N2CCc3c(ccs3)C2c4ccc(cc4)C(F)(F)F SEW01213 COc1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N S14749 COCc1cc(nc(n1)NC(=N)Nc2ccc(cc2Cl)Cl)O RJF00674 CN(c1c(cc(cn1)Cl)C(F)(F)F)NC(=O)c2ccccc2 SEW02382 c1cc(ccc1c2csnn2)C(=O)Nc3nccs3 SEW01327 c1cc(oc1)CNC(=O)c2ccc(cc2)c3csnn3 SEW01329 c1cc(cc(c1)NC(=O)c2cccs2)c3ncon3 SEW01258 c1cc(ccc1NS(=O)(=O)c2ccc(s2)c3ccc(s3)S(=O)(=O)Nc4ccc(cc4)[N+](=O)[O-])[N+](=O)[O-] SEW02451 c1ccc(c(c1)C(=O)O)SC2CC(=O)N(C2=O)c3ccc(cc3)Cl S06031 Cc1cc(nc(n1)NC(=N)Nc2ccc(c(c2)Cl)Cl)O RJF00676 c1cc(ccc1Nc2ncnc(n2)N)Oc3ccc(cc3)Cl RJF00678 c1ccc(c(c1)C(F)(F)F)NC(=N)NC(=N)N.Cl RJF00679 COCc1cc(nc(n1)NC(=N)Nc2ccc(cc2)Oc3ccc(cc3)Cl)O RJF00681 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)c3ccccc3 SEW02442 CCN(CC)C(=S)Oc1ccc(cc1Cl)Cl S06010 CC(=O)N1C(SC(=N1)N(C(=O)C)/N=C/c2ccc(cc2)Cl)c3ccc(cc3)Cl S14839 COc1ccc(cc1)/C=N/NC(=S)N/N=C/c2ccc(cc2)OC S14840 Cc1ccc(cc1)Sc2ccccc2NC(=O)C(Cl)(Cl)Cl S06380 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)NNC(=S)Nc3ccccc3OC RJF01960 CC(=O)Oc1cc2c(cc1Cl)c(cc(=O)o2)COC RJF02002 CC(=O)N1C(SC(=N1)N(C(=O)C)/N=C/c2ccc(cc2)C(F)(F)F)c3ccc(cc3)C(F)(F)F S14837 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3C=Cc4ccccc4C3C#N S06275 CN(c1c(cc(cn1)Cl)C(F)(F)F)NC(=O)CC#N SEW02378 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2ccccc2 SEW02379 Cc1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3C(=O)O S06030 CC(=O)Nc1cccc(c1)c2nnco2 SEW01226 c1cc(ccc1C(=O)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl)Cl RJF02045 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)c4ccc(cc4)Cl)C(F)(F)F SEW02394 c1ccc(cc1)c2c(nccn2)c3ccccc3 S12966 Cc1ccc(cc1Nc2ncnc(n2)N)I RJF00723 Cc1cc(c(cc1Cl)C)S(=O)(=O)c2nc3ccc(cc3s2)Cl SEW01277 COc1ccc(cc1)C(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F SEW02448 C=CC/N=C/1\NC(=O)C(S1)CC(=O)Nc2ccccc2 S05940 CC1(CC2=C(C3CCCCC3O2)C(=O)C1)C S12962 CN(c1c(cc(cn1)Cl)C(F)(F)F)NC(=O)c2ccccc2Cl SEW02383 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C(=O)Nc3ccc(cc3OC)OC SEW02391 c1c(ccc(c1)F)/C=N/NC(=S)N/N=C/c2ccc(cc2)F S14829 c1ccc(cc1)N2C(=O)CSC2=S S06033 c1c(nc(nc1O)C2CC2)C(F)(F)F RJF00722 Cc1ccc(cc1)Sc2ccccc2NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C S06335 COc1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3C(=O)O S06032 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)OC(F)(F)F SEW02370 c1cc(cc(c1)F)Nc2ncnc(n2)N RJF00709 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NNC(=O)c3ccc(cc3)Cl RJF02050 c1ccc2c(c1)cccc2/C=N/NC(=S)Nc3c(cccc3Cl)Cl S03264 Cc1c(c(n(n1)C)O)/N=N/c2cccc3c2cccc3 SEW02373 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2ccccc2Cl SEW02380 c1cc(c(cc1F)Br)Nc2ncnc(n2)N RJF00715 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccccc2C(F)(F)F RJF02056 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C(=O)Oc3ccc(cc3)Br SEW02398 CN1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)OCC=C S14823 CC(C)NC(=O)NNC(=O)Cn1nc(nn1)c2cc(cc(c2)Cl)Cl RJF02066 c1cc(c(cc1C(F)(F)F)NC(=S)Nc2cc(cc(c2)Cl)Cl)N3CCCCC3 RJF00697 COC(=O)c1cccc(c1)NC(=N)NC(=N)N.Cl RJF00705 c1cc(cc(c1)Cl)S(=O)(=O)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl RJF02033 CS(=O)(=O)NNC(=O)Cn1nc(nn1)c2cccc(c2Cl)Cl RJF02037 c1cc(cc(c1)NC(=O)c2ccc(cc2)Cl)c3ncon3 SEW01233 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)Cc3c(cccc3Cl)Cl RJF02040 c1cc(cc(c1)F)NC(=N)NC(=N)N.Cl RJF00703 COc1ccc(cc1OC)CCn2c(=O)c3cc4c(cc3c2=O)c(=O)n(c4=O)CCc5ccc(c(c5)OC)OC S03288 c1cc(c(cc1C(F)(F)F)NC(=S)Nc2ccc(c(c2)Cl)F)N3CCCC3 RJF00693 c1ccc(c(c1)c2nnc(o2)N)[N+](=O)[O-] S14873 c1cc2c(cc1F)-c3c(cnc(n3)C4CC4)CO2 SEW02372 CC1(CC2=C(C(C3=C(N2)CC(CC3=O)(C)C)c4ccccc4Cl)C(=O)C1)C S06314 CCOC(=O)c1ccc(cc1)/N=C/c2ccc(cc2)Cl S03434 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC(=O)c2ccc(cc2)Cl SEW02381 c1cc(c(cc1NC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl)Cl)Br RJF02027 Cc1cccc(c1S(=O)(=O)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl)Cl RJF02038 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C(=O)Nc3ccc(cc3)Cl SEW02389 CC(C)c1ccc(cc1)/C=N/NC(=S)N/N=C\c2ccc(cc2)C(C)C S14841 c1cc(c(cc1Cl)Cl)C(=O)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl RJF02046 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C(F)(F)F RJF02048 COCc1cc(=O)oc2c1cc(c(c2)O)Cl RJF01996 CC(=O)Oc1ccc2c(cc(=O)oc2c1)COC RJF01999 Cc1cc(ccc1Br)NC(=S)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl RJF02019 CN(c1c(cc(cn1)Cl)C(F)(F)F)NC(=O)c2ccc(cc2)Cl SEW02384 CC(=O)c1ccc(cc1)N2C(=O)C=CC2=O S03357 COc1cc(cc(c1OC)OC)/C(=N/O)/N S03367 CC1c2nc3ccccc3n2CN(CO1)c4ccc(cc4)OC S14875 COCc1cc(nc(n1)N)O RJF00700 Cc1cccc(c1)c2nc(cc(n2)O)COC RJF00701 c1ccc2c(c1)C(=Cc3ccc(cc3)C(F)(F)F)c4ccccc4C2=O S14919 c1ccc2c(c1)C(=Cc3ccc(cc3)Cl)c4ccccc4C2=O S14921 CC(=O)N1C(SC(=N1)N(C(=O)C)/N=C/c2ccc(cc2)F)c3ccc(cc3)F S14838 Cc1c(cnc(n1)c2ccncc2)c3nc(sn3)Nc4ccccc4 SEW02340 c1cc(ccc1C2C=C(C(=O)N2c3ccc(cc3)OC(F)(F)F)Nc4ccc(cc4)OC(F)(F)F)Cl S14813 C=CCOc1ccc(cc1)C(C[N+](=O)[O-])Sc2ccccc2N S14818 c1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3C(=O)O S06029 CC1c2nc3ccccc3n2CN(CO1)c4ccc(cc4)OC(F)(F)F S14865 CC(c1[nH]c2ccc(cc2n1)Cl)O S14867 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NNC(=O)c3ccc(cc3Cl)Cl RJF02064 c1cc(c(cc1C(F)(F)F)NC(=S)Nc2cc(cc(c2)Cl)Cl)N3CCCC3 RJF00696 c1ccc(cc1)/C=C/C(=O)NC(=S)NNC(=O)Cn2nc(nn2)N3CCCCC3 RJF02073 C=CCOc1ccc(cc1)/C=C/2\CCCc3ccccc3C2=O S14824 c1ccc2c(c1)ccc3c2C=C(C(O3)c4c(cccc4Cl)Cl)[N+](=O)[O-] S14915 c1ccc(cc1)C2c3cc(ccc3NC(=N)N2C(=N)N)Cl.Cl RJF00706 COc1cc(cc(c1OC)OC)C(=O)Nc2cccc(c2)C(F)(F)F S03313 Cc1c2ccccc2n3c1/C(=N/OC)/CC3 SEW02369 CN(c1c(cc(cn1)C(F)(F)F)Cl)/N=C/c2ccc(cc2O)O SEW02357 c1cc(c(c(c1)Cl)CSc2nnc(n2c3ccc(cc3)Cl)C4CC4)F RJF00634 Cc1ccc(cc1NC(=N)NC(=N)N)I.Cl RJF00716 c1cc(ccc1C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ccc(cc3)C(F)(F)F)Cl RJF02095 CC1c2nc3ccccc3n2CN(CO1)c4ccc(cc4)F S14874 CCCNC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(on2)C RJF02096 c1cc(cc(c1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3nnco3 SEW01331 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)Cl)c3nnco3 SEW01333 CCOC(=O)c1ccc(cc1)NC(=S)N2CCN(CC2)C(=S)Nc3ccc(cc3)C(=O)OCC S06101 CCCNC(=O)NNC(=O)Cn1nc(nn1)c2cc(cc(c2)Cl)Cl RJF02065 CC(=O)OCc1ccc(o1)C=C(C#N)C#N S12935 C=CCOc1ccc(cc1)/C=C/2\CCc3ccccc3C2=O S14820 C=CCOc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccccc3 S14821 c1ccc(c(c1)NC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl)F RJF02009 c1cc(ccc1C(F)(F)F)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F RJF02093 c1cc(cc(c1)Cl)CNC(=O)c2ccc(cc2)c3csnn3 SEW01335 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2F)F)c3ncon3 SEW01250 Cc1ccccc1/C=C\2/C(=O)OC(=N2)c3ccccc3 S12944 CC(C)(C)n1c(ccn1)c2ccc(s2)c3cccs3 SEW02416 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)S(=O)(=O)Oc3ccc(cc3)C#N SEW02425 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)C(C)C SEW02368 c1c(cc(cc1Cl)Cl)c2nnn(n2)CC(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF02034 COc1ccc(cc1OC)S(=O)(=O)Nc2cccc(c2)c3ncon3 SEW01247 CC(=O)c1ccc(cc1)NC(=O)/C=C\C(=O)O S03356 c1c(c2c(o1)CCCC2=O)C(=O)O SEW02412 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C(=O)Oc3ccc(cc3)C(C)(C)C SEW02400 c1cc(ccc1C(=O)Oc2ccc(cc2Cl)Cl)Cl S06071 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C(=O)N SEW02406 COc1ccccc1c2nc(no2)c3cccc(c3)C(F)(F)F SEW02409 c1ccc2c(c1)c(cs2)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N S14923 C/C(=N\NC(=S)N)/c1cc2ccccc2o1 S13029 c1ccc2c(c1)ccc3c2C=C(C(O3)c4ccc(cc4)Cl)[N+](=O)[O-] S14918 Cc1c(cccc1Cl)NC(=S)Nc2ccc(cc2)S(=O)(=O)Nc3cc(ccc3F)F RJF02107 c1ccc2c(c1)cccc2C3C(=Cc4c5ccccc5ccc4O3)[N+](=O)[O-] S14917 c1cc(c(cc1Br)Cl)NC(=S)N2CCCCCC2 S05651 c1cc(sc1c2ccc(s2)S(=O)(=O)N3CCOCC3)S(=O)(=O)N4CCOCC4 SEW02290 c1cc(sc1c2ccc(s2)S(=O)(=O)N3CCCC3)S(=O)(=O)N4CCCC4 SEW02298 CC1c2cnc(nc2-c3cc(ccc3S1)Cl)N SEW01285 c1ccc(cc1)N/N=C/C(=O)Nc2ccccc2C(=O)O S14896 c1ccc2c(c1)ccc3c2C=C(C(O3)c4c(cccc4Cl)F)[N+](=O)[O-] S14916 c1ccc(cc1)N2C(=O)CC(C2=O)SCCC(=O)O S12993 c1cc(ccc1N)S(=O)(=O)Nc2cc(ccc2F)F RJF02101 COc1ccc(cc1)N2Cn3c4ccccc4nc3CSC2 S14911 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/C(=S)N S14966 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)NNC(=S)Nc3ccc(cc3)C(F)(F)F RJF02114 CCCNC(=O)NNC(=O)Cn1nc(nn1)c2cccc(c2Cl)Cl RJF02068 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2)C(F)(F)F RJF02074 COc1ccc(c(c1)C(=O)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl)OC RJF02080 CN(C)/C=C\1/C(=NN(C1=O)c2ccccc2)C(=O)OC SEW02277 c1cc(ccc1C(=O)CSc2nnc(n2c3ccc(cc3)Cl)C4CC4)Cl RJF00639 c1cc(cc(c1)Cl)n2c(nnc2S)C3CC3 RJF00640 COc1cc(cc(c1)OC)/C=C/2\CCc3ccccc3C2=O S12911 CN(C)/C=C/C(=S)c1cccs1 S14950 c1cc(ccc1c2nnc(o2)N)N S14957 CC(=O)Nc1ccc(cc1)/C=C/[N+](=O)[O-] S14963 CC(C)(C)NC(=O)NNc1nc2ccc(cc2s1)Cl SEW01352 CC(CS(=O)(=O)c1ccc(cc1)Cl)C(=O)O SEW01356 CCOC(=O)c1cc(nn1c2nc3ccc(cc3s2)Cl)C SEW01284 COc1ccc(cc1)CNC(=S)NN S14992 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)Cl)/C(=O)S2 S15000 CC(=O)Nc1ccc(cc1)C2=N/C(=C/c3cccc(c3)OC)/C(=O)O2 S15001 CCCCCCCCCCCCSC1CC(=O)N(C1=O)c2ccccc2 S13002 c1cc(cc(c1)[N+](=O)[O-])/C=C/[N+](=O)[O-] S13012 c1cc(ccc1N2C(=O)C=CC2=O)OC(F)(F)F S13069 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C#N SEW02410 Cc1ccc2c(c1)oc(=S)[nH]2 S06035 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)N RJF02082 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2)S(=O)(=O)Nc3ccc(cc3)C(F)(F)F RJF02083 c1ccc2c(c1)cc(o2)C(=O)CSc3nnnn3c4cccc(c4)Cl S13051 c1cc(c(cc1F)F)NC(=S)NCCC(=O)O RJF00746 c1cc(ccc1NC(=O)/C=C/C(=O)O)OC(F)(F)F S13068 c1cc(sc1)c2cc([nH]n2)NC(=N)NC(=N)N.Cl RJF00729 c1cc(ccc1N)S(=O)(=O)Nc2cc(cc(c2)Cl)Cl RJF00748 c1cc(c(cc1NC(=S)NCCC(=O)O)Cl)F RJF00751 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2F)F RJF00752 c1cc(cc(c1)NC(=S)NCCC(=O)O)C(F)(F)F RJF00755 Cc1ccc(cc1F)NC(=S)NCCC(=O)O RJF00758 c1ccc(c(c1)C(F)(F)F)NC(=S)NCCC(=O)O RJF00757 c1cc(cc(c1)F)NC(=S)NCCC(=O)O RJF00759 c1cc(ccc1NC(=S)NCCC(=O)O)Cl RJF00760 c1cc(c(c(c1)Cl)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(cc(c3)Cl)Cl)F RJF00763 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(cc(c3)Cl)Cl RJF00767 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)Cc3c(cccc3Cl)F RJF02132 c1c(c\2c(o1)CCC/C2=N\N3CCCCC3)C(=O)O SEW02433 c1c(cc(c(c1Cl)N/N=C/2\CCCc3c2c(co3)C(=O)O)Cl)Cl SEW02434 C=C1c2ccccc2C(=O)N1c3cc(cc(c3)Cl)Cl S14886 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)NNC(=O)c3ccc(cc3Cl)Cl RJF02138 c1cc(ccc1C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(ccc3F)F)Cl RJF02142 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3ccc(cc3)F)C2=O S06959 c1ccc2c(c1)C(=O)C(=C(C#N)NCc3cccnc3)C2=O S06963 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F SEW01290 c1cc(ccc1C/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/N)c3csnn3 SEW01293 COc1c(c(ccc1)/C=N/N=C/c2c(c(ccc2)OC)O)O S03456 c1cc(sc1)c2ccc(s2)CNC(=O)CSCC(=O)O SEW02583 CC(C)(C)C1=NN(C(=O)C1)c2nc3ccc(cc3s2)Cl SEW01297 c1cc(sc1)C(=O)O/N=C(/Cc2ccc(cc2)c3csnn3)\N SEW01302 c1ccc(cc1)NC(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F SEW02481 c1cc(ccc1C/C(=N/OC(=O)c2csnn2)/N)c3csnn3 SEW01303 CC(C)(C)C(=O)O/N=C(/Cc1ccc(cc1)c2csnn2)\N SEW01307 CN(C)S(=O)(=O)Oc1ccc(cc1)C#N SEW02485 CCOC(=O)c1csc(n1)Cc2ccc(cc2)c3csnn3 SEW01319 c1cc(ccc1c2csnn2)C(=O)Nc3ccc(cc3)Cl SEW01321 Cc1cc(cc(c1I)C)C(C)(C)C SEW02501 c1ccc(c(c1)NC(=O)/C=C\C(=O)O)OC(F)(F)F S13070 c1cc(ccc1C(F)(F)F)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(ccc3F)F RJF02119 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)NNS(=O)(=O)c3ccc(cc3)C(F)(F)F RJF02120 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)Cn2nc(nn2)c3cccc(c3)C(F)(F)F RJF02139 COc1cc(cc(c1)OC)C=C2C(=O)c3ccccc3C2=O S12975 Cc1ccccc1/C=C/2\CCc3ccccc3C2=O S12988 c1cc(sc1)c2ccc(s2)CNC(=O)NC(=O)c3ccc(cc3)Cl SEW02495 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSCC(=O)O)C(F)(F)F SEW02504 CC1=CC(=O)N(C1=O)c2ccc(cc2)OC(F)(F)F S13087 CC1(CCC(=O)N(C1=O)c2ccc(cc2)OC(F)(F)F)C S13089 c1ccc2c(c1)cccc2/C=C(/C#N)\C(=S)N S14969 c1cc(c(cc1Cl)NC(=O)/C=N/O)Cl S13096 c1cc(c2c(c1Cl)C(=O)C(=O)N2)Cl S13100 CNC(=S)Nc1ccc(cc1)Oc2ccc(cc2)/N=C/c3ccncc3 S06195 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NN RJF02011 c1cc(ccc1NC(=S)N)OC(F)(F)F S13090 CN(C)C(=S)NCCC1=CCCCC1 S14986 COc1ccc(cc1)CNC(=S)NCCO S14990 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cccc(c3)C(F)(F)F RJF00771 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ccc(cc3F)F RJF00772 COc1cccc(c1)/C=C/2\C(=O)OC(=N2)c3ccccc3 S14998 CC(=O)Nc1nc(cc(n1)O)COC RJF00786 Cc1c(nc(nc1O)SCc2c(cccc2Cl)F)COC RJF00799 c1cc(cc(c1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)c3nnco3 SEW01330 CCCCNC(=O)Nc1cccc(c1)c2nnco2 SEW01338 CC1CC(=O)N(C1=O)c2ccccc2OC(F)(F)F S13097 c1ccc(c(c1)N2C(=O)c3cccnc3C2=O)OC(F)(F)F S13099 CC1/C(=C\N(C)C)/C(=O)c2cc(ccc2S1)Cl SEW01280 c1ccc2c(c1)c3c([nH]2)C(N(CC3)S(=O)(=O)c4ccc(c(c4)Cl)Cl)C(F)(F)F SEW02456 COc1ccc(cc1)CNc2n[nH]c(=S)s2 S14993 CC(=C)Cc1c(nc(nc1O)SC)COC RJF00994 c1ccc2c(c1)c(cs2)CN3C(=O)COCC3=O S13293 c1cc2c(cc1F)-c3c4cc(ccc4ncc3CO2)Cl SEW02556 c1cc(oc1)c2c(c(sc2C(=O)O)C(=O)O)c3ccco3 SEW02557 Cc1c(c(nc(n1)SC)O)CC(=C)C RJF00921 CCCCc1c(nc(nc1O)S)COC RJF00999 COc1ccccc1CNC(=S)NN S14973 COc1ccccc1CNC(=S)NCCO S14974 Cc1ccc(cc1)CNC(=S)NCCO S14981 c1cc(cc(c1)/N=C/c2c(cccc2Cl)F)c3ncon3 SEW01346 c1ccc(cc1)C2=CC(=O)N(C2=O)c3ccc(cc3)OC(F)(F)F S13120 c1cc(sc1)c2nc(no2)c3ccc(s3)c4ccno4 SEW02559 c1cc(ccc1/C=C/[N+](=O)[O-])Cl S03529 CC(=O)O/N=C(/Cc1ccc(cc1)c2csnn2)\N SEW01309 Cc1ccc(cc1)CSc2nc3ccc(cc3s2)[N+](=O)[O-] S03533 c1cc(ccc1Cc2nc(cs2)c3ccc(cc3)Cl)c4csnn4 SEW01315 c1cc(ccc1Cc2nc(cs2)c3ccc(cc3)[N+](=O)[O-])c4csnn4 SEW01316 c1ccc2c(c1)C(=O)N(C2=O)CNc3ccc(cc3)OC(F)(F)F S13074 CC1CC(=O)N(C1=O)c2ccc(cc2)OC(F)(F)F S13086 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3cccc(c3)C(F)(F)F RJF02158 c1ccc(cc1)NC(=O)Nc2cccc(c2)c3nnco3 SEW01339 Cc1cc(ccc1Br)n2c(=O)c3ccccc3[nH]c2=S S06543 c1cc2c(cc1NC(=N)NC(=N)N)OCCO2.Cl RJF00843 c1cc2c(cc1Nc3ncnc(n3)N)OCO2 RJF00844 COc1ccccc1NC(=O)c2ccc(cc2)c3csnn3 SEW01323 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cccs3)C(F)(F)F RJF00780 c1cc(cc(c1)/N=C/c2ccc(cc2)C#N)c3ncon3 SEW01347 Cc1cc(nc(n1)c2ccc(cc2)C(=O)N)O RJF00785 CCCCc1c(nc(nc1O)C2CC2)C RJF00797 c1cc(c(cc1Cl)NC(=N)NC(=N)N)O.Cl RJF00798 Cc1c(nc(nc1O)c2ccccn2)COC RJF00833 CCOC(=O)CN1C(=O)CC(CC1=O)c2cc(c(c(c2)OC)OC)OC S13209 c1cc(c(cc1Cl)C#N)N2C(=O)C=CC2=O S03563 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl RJF02166 CCO/C=C\1/C(=O)NC(=S)S1 S03457 c1ccc(cc1)C(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF00862 c1ccn(c1)c2ncnc(n2)Nc3cccc(c3)Cl RJF00871 c1ccc(cc1)/C=N/C(/N=C/c2ccccc2)c3ccccc3 S03463 Cc1c(c(nc(n1)SCC#C)O)Cc2c(cccc2Cl)F RJF00873 c1cc(c(c(c1)Cl)/C=N/c2ccc(cc2C#N)Cl)Cl S03547 c1ccc2c(c1)c3c([nH]2)C(NCC3)C(F)(F)F SEW02393 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3cccc(c3)C(F)(F)F RJF02163 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F RJF02165 COC(=O)C1=CC2C3C(C1C4C2C(=O)N(C4=O)c5cc(cc(c5)Cl)Cl)C(=O)N(C3=O)c6cc(cc(c6)Cl)Cl S13133 COc1ccccc1Nc2ncnc(n2)n3cccc3 RJF00878 Cc1cccc(c1)c2nc(c(c(n2)O)CCC(C)C)C RJF00881 CC(C)CNC(=O)/C=C\C(=O)O S06478 c1cc(ccc1C(=O)N2C(=O)c3ccc(cc3C2=O)[N+](=O)[O-])Cl S06506 CCOC(=O)c1c(ocn1)c2ccc(cc2Cl)Cl SEW01386 CC(C)c1ccc(c(c1)Br)NC(=N)NC(=N)N.Cl RJF00714 CCOC(=O)C1=C(n2c(=CC1c3ccc(cc3)OC)s/c(=C\c4ccc(cc4)OC)/c2=O)N S06587 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)N/N=C/c3c(cccc3Cl)Cl RJF02169 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)N/N=C/c3c(cccc3Cl)F RJF02170 COc1cccc(c1OC)/C=C/2\C(=O)OC(=N2)c3cccs3 S06426 COc1cc(cc(c1OC)OC)C2CC(=O)N(C(=O)C2)c3ccc(cc3)OC(F)(F)F S13182 c1cc(sc1C2NC(CS2)C(=O)O)[N+](=O)[O-] S06066 COc1c(c(cc(c1)/N=C/c2ccc(cc2)/C=N/c3cc(c(c(c3)OC)OC)OC)OC)OC S06067 c1ccc2c(c1)c(cs2)/C(=C/c3ccc(cc3)F)/C#N S14924 Cc1c(nc(nc1O)SCC#C)COC RJF00864 COc1cccc(c1)NC(=N)NC(=N)N RJF00867 c1ccc2c(c1)cccc2NC(=O)CC3C(=O)NC(=N)S3 S15021 c1ccc(c(c1)Nc2ncnc(n2)n3cccc3)Cl RJF00870 Cc1c(c(nc(n1)S)O)CCC(C)C RJF00872 c1cc(sc1)c2ccc(s2)CNC(=O)/C=C\C(=O)O SEW02510 c1cc(sc1)c2ccc(s2)CNC(=O)C3C4CC(C3C(=O)O)C=C4 SEW02511 c1ccc(c(c1)NC(=O)NCc2c(ccs2)CSc3ccc(cc3)Cl)F SEW02522 c1cc(cc(c1)NC(=O)NCc2c(ccs2)CSc3ccc(cc3)Cl)C(F)(F)F SEW02524 CC(C)(C)C(=O)Cn1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF00854 c1ccc(cc1)c2nc(no2)c3cccc(c3)C(F)(F)F SEW02407 c1cc(cc(c1)C(F)(F)F)c2nc(on2)c3cccc(c3)Cl SEW02408 C=C1c2ccccc2C(=O)N1c3ccc(cc3)C(F)(F)F S14860 C=C1c2ccccc2C(=O)N1c3ccc(cc3)F S14861 CC(C)C(C(=O)O)NS(=O)(=O)c1ccccc1 S03581 Cc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccc(cc3)Cl S06418 c1ccc(cc1)/C=C/C(=O)NCC(=O)O S06424 CSc1nnc(s1)/N=C/c2ccccc2O S15031 c1cc(cc(c1)C(F)(F)F)c2nnc(o2)c3ccc(cc3Cl)Cl RJF02157 c1cc(ccc1NC(=O)/N=C\2/C(=S)N(C(=O)N2c3ccc(cc3)OC(F)(F)F)c4ccc(c(c4)Cl)Cl)OC(F)(F)F S15048 Cc1ccccc1/C=N/NC(=S)N S12951 Cc1c(cccc1)/C=N/N=C/c2c(cccc2)C S12955 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)S(=O)(=O)Nc3cc(c(c(c3)OC)OC)OC SEW02429 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)C(C)C S03329 c1cc(sc1)c2ccc(s2)CNC(=O)c3ccc(s3)[N+](=O)[O-] SEW02484 c1ccc(cc1)c2c(nco2)C(=O)NN SEW01409 CC(=C)Cc1c(nc(nc1O)S)COC RJF00991 CCOC(=O)c1ccc(cc1)/N=C/c2ccc(c(c2)Cl)Cl S03435 CC1(CC2=C(C(C3=C(N2)CC(CC3=O)(C)C)c4cccs4)C(=O)C1)C S06316 Cc1ccc(cc1NC(=S)N/N=C/c2cccc3c2cccc3)Cl S06323 c1ccnc(c1)NS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F SEW01289 c1cc(cc(c1)C(F)(F)F)c2n[nH]nn2 RJF02108 c1cc(ccc1S(=O)(=O)c2nc3ccc(cc3s2)Cl)Cl SEW01276 CN(C)C(=S)NCc1ccccc1OC S14975 COc1ccccc1Cn2c(=S)[nH]nn2 S14978 Cc1ccc(cc1)CNC(=S)N(C)C S14987 c1cc2c(cc1Cl)sc(n2)SCC(=O)N SEW01281 COc1cc(cc(c1OC)OC)N2C(=O)C=CC2=O S03341 Cc1cc(cc(c1C#N)C)C(C)(C)C SEW02502 COc1ccc(c(c1OC)OC)C=C(C#N)C#N S03345 Cc1nc(no1)c2cc(c(c(c2)OC)OC)OC S03370 c1ccc(cc1)n2c(nnn2)SCC(=O)c3ccc(cc3)[N+](=O)[O-] S03372 CCOC(=O)CN(/C=N/C#N)c1ccc(cc1)OC SEW01262 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)NNC(=S)Nc3ccc(c(c3)Cl)Cl RJF02113 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)c3ccc(cc3)Cl RJF02134 CNC(=O)c1c(ocn1)c2ccc(cc2)Cl SEW01413 c1cc(ccc1/C=N/Nc2ccc(cc2Cl)C#N)Cl SEW01417 Cc1cc(no1)NC(=O)/C=C/C(=O)O S03621 C#CCSc1nnc(s1)N S06815 CC(C)(C)c1ccc(cc1)C(=C(C#N)C#N)O S06859 CC(C)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2Cl)C#N SEW01391 c1ccc(c(c1)NC(=N)NC(=N)N)Oc2ccc(cc2Cl)Cl.Cl RJF00728 Cc1ccc(cc1C)N2C(=O)C3CCCCC3C2=O S13354 c1cc2c(cc1Cl)c(cs2)CNC(=O)/C=C/C(=O)O S13355 COc1ccc(cc1)C2c3ccsc3CCN2C(=O)c4cccs4 SEW01499 Cc1ccccc1NC(=S)N2CCCCC2C S00053 Cc1c(c(nc(n1)NC(=O)C)O)CCC(C)C RJF00894 Cc1c(c(nc(n1)SCC#C)OC(=O)N(C)C)Cc2c(cccc2Cl)F RJF00883 CC(C)(C)c1nc(no1)c2ccc(s2)c3ccno3 SEW02552 CCN(CC)CCCNC(=O)/C=C/C(=O)O S07065 c1ccc2c(c1)CCC/C(=C\c3ccc4c(c3)OCO4)/C2=O S15205 Cc1c(c2ccccc2o1)CC(=O)Nc3ccc(cc3)C(C)(C)C S15116 C=CCOc1ccc(cc1)/C=C\2/C(=O)C3CCN2CC3 S15121 Cc1ccc(cc1)/C=C\2/C(=O)C3CCN2CC3 S15124 c1cc(sc1)c2ccc(s2)C(=O)N3CCOCC3 SEW02571 Cc1ccc(c(c1)C)NC(=S)Nc2ccccc2C S00054 c1ccn(c1)c2ncnc(n2)Nc3ccc(cc3)F RJF00877 c1cc(ccc1C2CC(=O)N(C2=O)c3ccc(cc3)OC(F)(F)F)NC(=O)C(F)(F)F S15091 COc1ccc(cc1)/N=C/C2=C(c3cc(ccc3OC2)Cl)Cl SEW02592 c1cc(ccc1NC(=N)NC(=N)N)Cl RJF00885 c1cc(cc(c1)OC(=O)c2ccc(s2)c3cccs3)C(F)(F)F SEW02580 c1cc(c(cc1N2C(=N)C(=S)N(C2=O)c3ccc(c(c3)Cl)Cl)Cl)Cl S15051 Cc1c(c(on1)C)C(=O)O/N=C(/Cc2ccc(cc2)c3csnn3)\N SEW01301 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/Cc2ccc(cc2)c3csnn3)\N SEW01295 c1cc(ccc1C/C(=N/OC(=O)c2ccc(o2)[N+](=O)[O-])/N)c3csnn3 SEW01304 c1cc(ccc1C/C(=N/OC(=O)C2CC2)/N)c3csnn3 SEW01308 CS/C(=N\C#N)/NCc1ccc(s1)c2cccs2 SEW02573 CCN(CC)C(=O)c1ccc(s1)c2cccs2 SEW02574 Cc1cc(no1)NC(=N)NC(=N)N.Cl RJF00946 c1cc(ccc1OCCC(=O)Nc2nccs2)F SEW01430 c1cc(ccc1OCCC(=O)N2CCSCC2)F SEW01431 c1ccc(cc1)C(=O)NC(=S)Nc2cccnc2 S15062 Cc1cc(no1)NC(=O)CCC(=O)O S03622 Cn1cnnc1SCc2ccc(cc2)c3csnn3 SEW01438 c1ccc(cc1)C(=O)NC(=O)NCc2ccc(s2)c3cccs3 SEW02493 c1cc(cc(c1)C(F)(F)F)C(=O)NC(=O)NCc2ccc(s2)c3cccs3 SEW02494 c1ccc(c(c1)N2C(=O)C=CC2=O)OC(F)(F)F S13071 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(cc3)OC(F)(F)F S13075 c1cc(ccc1NC(=O)CCOc2ccc(cc2)F)Cl SEW01424 c1cc(ccc1OCCC(=O)Nc2cc(cc(c2)Cl)Cl)F SEW01425 c1cc(ccc1C2CCCCC2)/N=C/3\NC(=O)C(S3)CC(=O)Nc4ccc(cc4)F S15016 c1cc(ccc1N/N=C/2\CCOc3c2cc(cc3)F)[N+](=O)[O-] SEW01447 CCOC(=O)c1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccc(cc3)C S03689 CC(C)(C)c1ccc(cc1)C(=O)NCc2csc3c2cc(cc3)Cl S13450 c1ccc(c(c1)C2OC(=O)c3ccccc3S2)Cl S06705 c1cc2c(cc1Cl)c-3c(cn2)COc4c3cc(cc4)Cl SEW02593 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)C RJF00931 Cc1c(c(nc(n1)SCC(=O)C(C)(C)C)O)CC(=C)C RJF00939 c1cc(ccc1C(=O)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl RJF01009 Cc1ccc(cc1)CNC2=NCCS2 S14983 Cc1ccc(cc1)CNc2n[nH]c(=S)s2 S14984 Cc1ccc(cc1)Cn2c(=S)[nH]nn2 S14985 c1cc(ccc1N2C(=O)CSCC2=O)OC(F)(F)F S13119 COc1ccc(c(c1)OC)C(C[N+](=O)[O-])Sc2ccccc2N S13384 c1ccc(cc1)C2N(C(=O)CS2)c3ccc(cc3)Cl S06691 C=CCC1CC(=O)N(C1=O)c2ccc(cc2)Cl S15214 C=CCC1CC(=O)N(C1=O)c2ccc(cc2)C(F)(F)F S15217 c1cc(cnc1)C2N(C(=O)CS2)c3cc(cc(c3)Cl)Cl S06723 COc1ccc(c(c1)N2C(=O)C=CC2=O)OC S07163 c1cc(cnc1)c2c(c(=O)[nH]c(=S)[nH]2)C#N S15219 c1ccc2c(c1)C/C(=C\c3ccc(cc3)F)/C2=O S15222 COc1ccc(c(c1)O)/C=N/c2nnc(s2)SC S15033 c1ccc(cc1)c2cc(nc(c2C#N)O)c3ccccc3 S06676 c1ccc(cc1)c2c(nco2)C(=O)O CC10201 Cc1cc(c(cc1CSc2nc3ccc(cc3s2)[N+](=O)[O-])C)CSc4nc5ccc(cc5s4)[N+](=O)[O-] S03534 CC(C)c1ccc(cc1)NC(=O)c2ccc(cc2)c3csnn3 SEW01322 c1cc(cc(c1)N/N=C(\C#N)/C(=O)c2ccsc2)C(F)(F)F SEW02696 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)OC(=O)N(C)C)CC(=C)C RJF00958 CCCCCCCC1CC/C(=C/c2cccc(c2)[N+](=O)[O-])/C1=O S15226 c1ccc(c(c1)C(=O)O)NC(=O)C(F)(F)F S03711 COc1cccc(c1)c2c(c(=O)[nH]c3c2-c4ccc(cc4CC3)OC)C#N S15103 CC1=NN(C(=O)C1=C2SCCS2)c3ccccc3 S15106 CCOc1cccc(c1O)/C=N/c2nnc(s2)SC S15032 c1c(cc(c(c1Cl)NNC(=O)c2cnc3n(c2=O)CCS3)Cl)Cl SEW01394 c1c(cc(cc1C(F)(F)F)NNC(=O)c2cnc3n(c2=O)CCS3)C(F)(F)F SEW01395 CC(C)(C)c1ccc(cc1)N2C(=O)C=CC2=O S06736 CCOC(=O)CNC(=O)c1ccc(cc1)C(F)(F)F S15002 C1CCN(CC1)c2nnn(n2)CC(=O)NNC(=S)NC(=O)C3CC3 RJF02189 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nnn(n2)CC(=O)NNC(=S)NC(=O)C3CC3 RJF02191 c1cc(sc1)c2ccc(s2)C(=O)Sc3ccc(cc3)Cl SEW02614 c1cc(cc(c1)/N=C/C2=C(c3cc(ccc3SC2)Cl)Cl)C(F)(F)F SEW02616 Cc1ccc(c(c1)C(=O)O)NC(=O)C(F)(F)F S03703 COc1ccc2c(c1)CC/C(=C\c3cc(cc(c3)OC)OC)/C2=O S13245 c1cc(ccc1C2CCCCC2)/N=C/3\NC(=O)C(S3)CC(=O)Nc4ccc(cc4)OC(F)(F)F S15017 c1ccc(c(c1)n2c(=S)[nH]nn2)F S15024 c1ccc(c(c1)CSc2nnc(n2c3ccc(c(c3)Cl)Cl)Cn4nc(nn4)c5cc(cc(c5)C(F)(F)F)C(F)(F)F)Cl RJF02201 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=S)NC(=O)C3CC3 RJF02203 c1ccc(c(c1)/C=N/NC(=S)Nc2cccc(c2)F)O RJF01010 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(c(c2)Cl)Br S03724 CCCCCCCCCCCCSC(=S)c1c(nn(c1O)c2ccccc2)C S15109 c1cc(sc1)/C=C/C(=O)NC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl RJF02174 c1cc(cnc1)N2C(SCC2=O)c3ccc(cc3)Cl S06686 c1ccc(cc1)C2N(C(=O)CS2)c3cccnc3 S06689 Cc1cc(cc(c1)NC(=O)CC2C(=O)N/C(=N\c3ccc(cc3)C4CCCCC4)/S2)C S15018 c1c(cc(cc1Cl)Cl)c2nnn(n2)CC(=O)NNC(=S)NC(=O)C3CC3 RJF02193 CCOC(=O)c1ccc(cc1)N2C(SCC2=O)c3ccccc3 S06692 c1cc(sc1)/C=C/C(=O)NC(=S)NNC(=O)Cn2nc(nn2)N3CCOCC3 RJF02187 c1c(cc(cc1Cl)Cl)N2C(=O)C=CC2=O S06729 C1CC1C(=O)NC(=S)NNC(=O)Cn2nc(nn2)N3CCOCC3 RJF02190 CC(C)(C)c1ccc(cc1)N2C(SCC2=O)c3cccnc3 S06731 c1ccc(cc1)c2c(nco2)C(=O)Nc3ccccc3 SEW01375 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NNC(=S)NC(=O)C3CC3 RJF02195 CC(=O)N/C(=C\c1cc(c(c(c1)OC)OC)OC)/C(=O)O SEW02605 CN1C(C2CCc3cc(ccc3C2=N1)OC)c4ccc(cc4)F S13256 c1cc(sc1)/C=C/C(=O)NC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF02175 c1cc(sc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2)S(=O)(=O)Nc3cc(ccc3F)F RJF02184 c1cc(ccc1C2N3C(OCC3(CO2)CO)c4ccc(cc4)[N+](=O)[O-])[N+](=O)[O-] S13228 c1ccc2c(c1)c(cs2)CNC(=O)c3ccccc3C(=O)O S13296 CC(C)c1nc(no1)c2ccc(s2)c3ccno3 SEW02561 CN(C)/C=N/C(=O)c1ccc(s1)c2cccs2 SEW02564 COc1cc(cc(c1OC)OC)N2C(=O)CC(C2=O)Sc3ccccc3N S03501 c1ccc(cc1)CCNC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)NCCc4ccccc4 S03507 c1cc(cc(c1)C(F)(F)F)c2nnc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF02159 c1ccc2c(c1)c(cs2)CNC(=O)CSCC(=O)O S13271 COc1ccc2c(c1)CC/C(=C\c3ccc(cc3)C(F)(F)F)/C2=O S13244 c1cc(cc(c1)C(F)(F)F)/C=N/Cc2ccc(s2)c3cccs3 SEW02515 c1ccc(c(c1)NC(=O)NCc2c(ccs2)COc3ccc(cc3)Cl)F SEW02516 CC(=O)c1c(c(c(s1)C(=O)O)c2ccco2)c3ccco3 SEW02517 CN(C)/C=C/1\C(=O)N(C(S1(=O)=O)c2cccnc2)c3ccc(cc3F)F S13387 Cc1cccc(c1NC(=S)Nc2cccc(n2)C)C S00081 C#CCSc1nnnn1c2cccc(c2)Cl S07148 c1c(scc1/C=N/N=C/c2csc(c2)[N+](=O)[O-])[N+](=O)[O-] S13251 c1cc(oc1)c2c(sc(c2c3ccco3)C(=O)N)C#N SEW02533 c1c(c(=O)n2c(n1)SCC2)C(=O)O SEW01382 c1cc(c(cc1C#N)Cl)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW01389 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(c(c3)Cl)Br S06546 c1cc(sc1)c2ccc(s2)C/N=C/c3ccc(cc3)Cl SEW02514 c1ccn(c1)c2ncnc(n2)Nc3cccc(c3)C(F)(F)F RJF00876 COc1ccccc1NC(=S)NCC2CCC(CC2)CNC(=S)Nc3ccccc3OC S00037 COc1ccccc1NC(=S)NCCc2ccc(c(c2)OC)OC S00039 COc1ccccc1NC2=NC(CS2)(CO)CO S13274 CCOC(=O)c1cnc2n(c1=O)CCS2 SEW01371 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3ccc(cc3)C(C)(C)C S06875 COC(=O)c1ccc(cc1)c2csnn2 SEW01372 CCOC(=O)c1c(ocn1)c2ccc(cc2)Cl SEW01373 COc1ccc(cc1)NC(=O)/C=C/c2ccccc2 S06516 CC(=O)N1C(=O)c2ccc(cc2C1=O)[N+](=O)[O-] S06535 CC1(OC(=O)C(=C2SCCCS2)C(=O)O1)C S13192 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2cccc(c2)Cl S13208 CCOC(=O)c1c(ocn1)c2ccc(cc2)C(F)(F)F SEW01379 CC(C)(C#C)NC(=C1C(=O)c2ccccc2C1=O)C#N S06961 COc1ccc2c(c1)CC/C(=C\c3ccc(cc3)F)/C2=O S13242 COc1ccc(cc1OC)/C=C/[N+](=O)[O-] S06777 c1ccc2c(c1)C(=C(C#N)C#N)C(=O)N2 S06782 c1cc(c(cc1C(F)(F)F)Cl)S(=O)(=O)N SEW01355 Cc1ccc(o1)/C=C/2\CCc3cc(ccc3C2=O)OC S13246 CN1C(C2CCc3cc(ccc3C2=N1)OC)c4ccc(cc4)C(F)(F)F S13253 CC1=N/C(=C/c2cc(c(c(c2)OC)OC)OC)/C(=O)O1 SEW02604 CS/C(=N\C#N)/NCc1c(ccs1)COc2ccc(cc2)Cl SEW02525 c1cc(ccc1C(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl RJF00861 Cc1cccc(c1)NC2=NC(CS2)(CO)CO S13273 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)C(=O)c4c(onc4c5ccccc5)C S06917 COc1ccc2c(c1)c-3c(cn2)COc4c3cc(cc4)Cl SEW02594 COc1ccccc1NC(=S)Nc2ccccn2 S00034 CCCCCCCC1CC/C(=C/c2ccc(cc2)C#N)/C1=O S15228 CC(C)(C)c1ccc(cc1)c2nc3ccccc3c(=O)o2 S06721 CC(C)(C)c1ccc(cc1)NC(=S)N(C)C S06746 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NNC(=S)NC(=O)/C=C/c3cccs3 RJF02177 COc1ccc(c(c1)c2nc3ccccc3c(=O)o2)Br S06924 c1cc(ccc1/C=C/2\CC/C(=C/c3ccc(cc3)C(F)(F)F)/C2=O)C(F)(F)F S15058 COc1c(c(c2c(n1)/C(=C/c3ccc(cc3)F)/CCC2)c4ccc(cc4)F)C#N S15059 c1c(ccc(c1)C(F)(F)F)/C=C\2/C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/CCCC2 S15063 c1cc(cc(c1)C(F)(F)F)c2nc(on2)c3ccc(s3)c4cccs4 SEW02619 CCOC(=O)c1c(ocn1)c2cccc(c2)C(F)(F)F SEW01507 Cc1c(c(on1)/C=C/c2c(ccs2)C3OCCO3)[N+](=O)[O-] SEW02704 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)CN4CCCCC4 S15069 COc1cccc(c1)/C=C(\C#N)/C(=O)OC S15105 Cc1ccc(cc1)N2C(=O)C(=C3SCCS3)C(=N2)C S15110 c1cc(ccc1c2csc(n2)NC(=S)NC(=O)C3CC3)Cl RJF02207 c1cnc(nc1)NS(=O)(=O)c2ccc(cc2Cl)C(F)(F)F SEW01291 c1cc(ccc1C/C(=N/OC(=O)c2cc(cc(c2)Cl)Cl)/N)c3csnn3 SEW01294 c1cc2c(cc1[N+](=O)[O-])c(nnc2O)O S06365 Cc1c(c2ccccc2o1)CC(=O)Nc3ccc(cc3)C(F)(F)F S15115 Cc1c(c(nc(n1)SCC(=O)C(C)(C)C)O)CCC(C)C RJF00907 COCc1c(c(nc(n1)S)O)Cc2c(cccc2Cl)F RJF00908 COc1ccc-2c(c1)CCc3c2nc(c(c3c4ccc(cc4)C(F)(F)F)C#N)OC S15075 COc1c(c(c2c(n1)-c3ccccc3CC2)c4ccc(cc4)C(F)(F)F)C#N S15076 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)CN4CCCC4 S15071 CCc1cccc(c1NC(=S)Nc2ccccc2OC)CC S00052 Cc1c(c(nc(n1)S)O)CC(=C)C RJF00916 CCOC(=O)c1ccc(cc1)N2C(=O)C3CC=C(CC3C2=O)C S03568 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C(=O)ONC(c3ccc(cc3)OS(=O)(=O)N(C)C)N SEW02506 COc1ccc(cc1)/N=C/C2=C(c3cc(ccc3OC2)F)Cl SEW02508 Cc1c(c(nc(n1)SCCC(C)C)O)CCC(C)C RJF00909 Cc1c(c(nc(n1)SCc2c(cccc2Cl)Cl)O)CCC(C)C RJF00898 COc1ccc(cc1)NC(=S)Nc2cccc(c2)C(F)(F)F S00024 c1ccc(cc1)NC(=O)c2c(ocn2)c3ccc(cc3)Cl SEW01411 CCOc1ccc(cc1OC)C2Nc3ccccc3C(=O)N2 S03611 c1ccc2c(c1)c(nn(c2=O)CN3CCOCC3)c4ccc(cc4)Cl S15085 c1cc(ccc1C(F)(F)F)NC2=NCCCS2 S15086 COc1ccccc1NC(=S)NC(c2ccccc2)c3ccccc3 S00036 c1ccc2c(c1)c(cc(=O)o2)Nc3ccc(cc3)OC(F)(F)F S13370 CCCCCCCCCCCCN1CN(C(=S)SC1)CCCCCCCCCCCC S07010 Cc1cccc(c1C)C(=O)Oc2ccccc2/C=N/N=C\3/N(C(=O)CS3)c4cccc(c4)Cl RJF00988 c1cc(cnc1)C2N(C(=O)CS2)c3ccc(cc3Cl)Cl S07044 CCCCc1c(nc(nc1O)SC)COC RJF01001 CCSc1nc(c(c(n1)O)Br)N RJF01005 CC1(C/C(=N\Nc2ccc(cc2)C(F)(F)F)/c3cc(c(c(c3O1)O)O)C(C)(C)C)C SEW02680 CC(C(c1ccc2c(c1)OCO2)c3c(n(c(=O)n(c3=O)C)C)N)[N+](=O)[O-] S13314 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2c(cccc2F)OC)N S13322 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nnn(n2)CC(=O)NNC(=O)C3CC3 RJF01023 C/C(=N\Cc1ccc2c(c1)OCO2)/c3ccccc3O S03777 COc1ccc2c(c1)CC/C(=C\c3ccc(cc3)OCC=C)/C2=O S15136 COc1ccc(cc1)/C=C/2\CCc3cc(ccc3C2=O)OC S15138 c1ccc2c(c1)CCC/C(=C\c3ccccc3Cl)/C2=O S15143 c1ccc2c(c1)CC/C(=C\c3ccccc3Cl)/C2=O S15144 CCCCCCCC1CC/C(=C\c2ccc(cc2)SC)/C1=O S15152 COc1ccc2c(c1)CC/C(=C\c3ccc(cc3Cl)Cl)/C2=O S15156 c1ccc2c(c1)C/C(=C/c3ccc(cc3)Cl)/C2=O S15158 COc1ccc(cc1)/C=C/2\Cc3ccccc3C2=O S15166 CSc1ccc(cc1)NC(=O)/C=C/C(=O)O S03868 CSc1ccccc1N2C(=O)C=CC2=O S03871 Cc1c(c2ccccc2o1)CC(=O)Nc3ccc(cc3)OC(F)(F)F S15114 Cc1nc(no1)c2ccc(s2)c3ccno3 SEW02554 c1cc(sc1)CSC(=O)NC(=O)c2ccc(s2)c3cccs3 SEW02563 c1cc(sc1)c2ccc(s2)C(=O)Nc3ccc(cc3)Cl SEW02570 c1cc(c(cc1NC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl)Cl RJF00942 c1c(cc(cc1Cl)Cl)OC(=O)c2cnc3n(c2=O)CCS3 SEW01454 COc1ccc(cc1)OC(=O)c2cnc3n(c2=O)CCS3 SEW01455 COc1ccc(cc1)C2c3ccsc3CCN2C(=O)c4ccc(cc4)C(F)(F)F SEW01497 c1cc(ccc1c2cn3c(n2)SCC3)[N+](=O)[O-] SEW01458 c1c(cc(cc1Cl)Cl)NC(=O)c2cnc3n(c2=O)CCS3 SEW01459 CC(C)(C)C(=O)N1CCc2c(ccs2)C1c3ccc(cc3)OC SEW01512 Cc1cccc(c1NC(=S)NCC2CCC(CC2)CNC(=S)Nc3c(cccc3C)C)C S00166 Cc1ccccc1NC(=S)NCCc2ccccn2 S00168 c1cc(ccc1/C(=N/OC(=O)CCOc2ccc(cc2)F)/N)Cl SEW01464 c1cc(ccc1C2SCCS2)/C(=N/OC(=O)CCOc3ccc(cc3)F)/N SEW01465 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)Br S06995 CCCCCCCCCCCC/N=C(\C)/c1ccccc1O S07008 Cc1c(c(nc(n1)N)O)CCC(C)C RJF00893 Cc1cc(ccc1Nc2ncnc(n2)n3cccc3)Br RJF00895 c1ccc(cc1)/C/2=N/CCNC(=O)c3c2cccc3 S15066 CCOc1ccc(cc1)/C=C/2\CCc3ccccc3C2=O S13715 c1ccnc(c1)S(=O)(=O)/C(=C/c2ccc(cc2Cl)C(F)(F)F)/C#N SEW01602 Cc1c(c(c(c(c1C)C)CSC(CC(=O)c2ccccc2)c3ccc(c(c3)OC)OC)C)C S04004 c1ccc(cc1)CC(=O)NC2(C(=O)c3ccccc3C2=O)O S13722 CSc1ccc(cc1)C(=O)C(CC(=O)c2ccc(cc2)Cl)c3cccs3 S13498 Cn1c(cc(c1c2ccc(cc2)SC)c3cccs3)c4ccc(cc4)Cl S13499 c1cnccc1c2c(c(=O)[nH]c(=S)[nH]2)C#N S15230 Cn1c(nnc1S(=O)(=O)Cc2ccc(cc2)c3csnn3)C(F)(F)F SEW01439 c1cc2c(cc1F)C(=O)CCO2 SEW01443 c1cc(c(cc1C(F)(F)F)N/N=C\2/CCOc3c2cc(cc3)F)Cl SEW01446 CN\1C=CC=C/C1=C\2/C(=O)OC(=N2)c3ccccc3 S13560 c1c(c(sc1Br)S(=O)(=O)N2CCCC2)Br SEW02659 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)O SEW02660 CC(C)(C)NS(=O)(=O)c1c(cc(s1)Br)Br SEW02661 c1cc(cc(c1)Cl)CNS(=O)(=O)c2c(cc(s2)Br)Br SEW02663 c1cc(c(cc1NC(=O)/C=C/C(=O)O)F)F S03834 c1cc(c(cc1N2C(=O)C=CC2=O)F)F S03835 c1ccc2c(c1)c(=O)n(c(n2)SCc3ccc(cc3)/C=C/c4c(cccc4Cl)F)Cc5ccco5 RJF01157 c1c(c(sc1S(=O)(=O)N)Cl)Br SEW02664 COC(=O)c1c(c(c(s1)C(F)(F)F)c2ccccc2)N SEW02673 CSC(=N)NC(=S)Nc1cccc(c1)Cl RJF01047 Cc1ccc(cc1NC(=S)NC(=N)SC)Cl RJF01049 c1ccc(c(c1)c2[nH]nnn2)C(F)(F)F RJF01052 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2CCOC(=O)Nc5ccc(cc5)Cl S15186 C#CCn1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF00989 COC(=O)c1ccccc1SC(=O)c2cnc3n(c2=O)CCS3 SEW01402 c1ccc(cc1)c2nc(no2)c3ccc(s3)c4ccno4 SEW02545 c1cc(cc(c1)Cl)c2nc(no2)c3ccc(s3)c4ccno4 SEW02546 Cc1cc(ccc1NCN2C(=O)c3ccccc3C2=O)Br S03867 CSc1ccccc1NC(=O)/C=C/C(=O)O S03869 c1cc(c(cc1CNC(=O)/C=C/C(=O)O)Cl)Cl S03872 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(c(c3)F)F S03836 COc1ccc2c(c1)CC/C(=C/c3ccc(cc3)SC)/C2=O S15161 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2cccc(c2)[N+](=O)[O-] S03849 COc1cc(c(cc1Cl)OC)NC(=S)NCCO S03877 Cc1cc(ccc1N2C(=O)C=CC2=O)Br S03866 c1cc(c(cc1Cl)Cl)NC(=O)/C=N/O S15172 c1ccc2c(c1)CC/C(=C\c3cccnc3)/C2=O S15174 CN(C)/C=N/C(=S)c1c(ccs1)COc2ccc(cc2)Cl SEW02624 Cc1cccc(c1C)NC(=O)/C=C/C(=O)O S03914 CC(=O)N/C(=C\c1ccc(cc1)Cl)/C(=O)O SEW02607 c1cc(sc1)c2ccc(s2)c3nc(no3)c4ccc(cc4)C(F)(F)F SEW02613 c1cc(c(cc1F)F)NC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF00943 c1cc(ccc1C2NC(CO2)(CO)CO)[N+](=O)[O-] S13227 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)O)CCC(C)C RJF00896 CC(=O)N1CCc2c(ccs2)C1c3ccc(cc3)OC SEW01511 Cc1ccccc1NC(=S)NCC2CCC(CC2)CNC(=S)Nc3ccccc3C S00165 Cc1csc2c1[nH]c(=O)n(c2=O)CCN3CCSCC3 S13667 Cc1ccccc1NC(=S)Nc2ccc(cc2)SC S00102 CC1(C/C(=N\Nc2c(cccc2Cl)Cl)/c3cc(c(c(c3O1)O)O)C(C)(C)C)C SEW02684 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl S06994 c1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S S00203 COc1ccc(c(c1)C(=O)O)Nc2cc(ccc2Cl)C(F)(F)F S07197 c1ccc(cc1)NC(=N)NC(=N)N.Cl RJF01059 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)Br SEW02649 C/C(=N\Cc1ccc(cc1)C#N)/c2ccccc2O S03739 CC(C)c1ccc2c(c1)CCC3C2(CCCC3(C)CNC(=O)/C=C/C(=O)O)C S03989 Cc1c(oc(n1)C)/C(=N/Nc2c(cc(cc2Cl)Cl)Cl)/C SEW01551 CC(C)(C)c1ccc(s1)C(=O)c2cccs2 SEW01553 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3ccc(c(c3)Cl)Cl)C(F)(F)F RJF01085 CSc1ccc(cc1)/C=C/2\CCc3ccccc3C2=O S13679 c1ccc2c(c1)CC/C(=C\c3ccc(cc3Cl)Cl)/C2=O S13683 CC(=O)Nc1ccccc1OCC(CS(=O)(=O)c2ccc(cn2)C(F)(F)F)O SEW02685 CSc1ccc(cc1)/C=C/2\CCCc3ccccc3C2=O S15195 Cc1ccc(cc1)CSc2ccccc2[N+](=O)[O-] S07229 c1cc(cc(c1)C(F)(F)F)CSc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] S07230 Cc1ccc(cc1Nc2nc3nc(cc(n3n2)O)COC)Cl RJF01082 c1ccc2c(c1)CCC3C2=NN(C3c4ccccc4Cl)CCO S15146 CCSc1nc(c(c(n1)O)CC(=C)C)C RJF00965 CC(=C)Cc1c(nc(nc1O)SCC(=O)C(C)(C)C)COC RJF01088 CN(C)/C=C/1\C(=O)N(C(=O)S1)c2ccc(cc2)OC(F)(F)F S13583 c1cc(ccc1NC(=S)Nc2ccc(cc2)OC(F)(F)F)OC(F)(F)F S13585 c1cc(ccc1NC(=S)NCCO)OC(F)(F)F S13587 c1cc(ccc1NC(=S)NN)OC(F)(F)F S13597 c1ccc(c(c1)N2CCOCC2)OC(=O)Nc3ccc(cc3)OC(F)(F)F S13604 c1cc(ccc1NC2=NCCCS2)OC(F)(F)F S13622 c1cc(sc1)C(=O)c2cccs2 SEW02655 COc1ccc2c(c1)CC/C(=C\c3ccc(cc3)Cl)/C2=O S15137 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nnn(n2)CC(=O)NN RJF00926 Cc1ccc(cc1)NC(=S)Nc2cccc(c2)C(F)(F)F S00236 Cc1ccc(cc1)NC(=S)Nc2ccc(cc2)C S00245 Cc1ccc(cc1)C(=O)CC(c2ccc(c(c2)OC)OC)Sc3ccccc3N S03728 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F RJF01090 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3ccccc3F)C(F)(F)F RJF01096 COc1ccccc1N\2C(=O)CS/C2=N\N=C\c3ccccc3O RJF00967 Cc1ccc(cc1Cl)c2nc(nc(n2)N)N RJF01100 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2CCOC(=O)c5ccc(cc5)C(F)(F)F S15179 c1cc(c(c(c1N2C(=O)CSCC2=O)F)F)F S13470 COc1cc(ccc1O)/C=N/NC(=S)Nc2cccc(c2)F RJF01011 CC(C(c1cccs1)c2c(n(c(=O)n(c2=O)C)C)N)[N+](=O)[O-] S13313 c1ccc2c(c1)cccc2N3C(=N)C(=S)N(C3=O)c4ccc(c(c4)Cl)Cl S15050 COc1ccc(cc1)C2c3ccsc3CCN2S(=O)(=O)c4ccc(cc4)Cl SEW01488 c1ccc(cc1)C/N=C/c2cccs2 SEW02695 C/C(=N\Cc1cccnc1)/c2ccccc2O S03765 c1cc(ccc1c2c(nco2)C#N)Cl SEW01420 CC(C)(C)c1ccc(cc1)C(=O)NCc2ccc(cc2)Cl S07105 COc1cc(cc(c1OC)OC)NC(=O)CCOc2ccc(cc2)F SEW01426 c1ccc2c(c1)c(cs2)CNC(=O)COCC(=O)O S13292 c1cc(sc1)/C=C/C(=O)NC(=S)NNC(=O)Cn2nc(nn2)N3CCCC3 RJF02185 c1cc(cnc1)NC(=O)NC(=O)c2ccc(s2)c3cccs3 SEW02537 c1ccc(c(c1)/C=N/N=C\2/N(C(=O)CS2)c3cccc(c3)F)OC(=O)c4ccc(cc4)Cl RJF01016 COc1cc(c(cc1Cl)OC)NC(=S)N S03774 CCOC(=O)c1ccc(cc1)NC(=S)Nc2ccccc2F S03772 CC(C)(C)S(=O)(=O)/C(=C/c1c(ccs1)C2OCCO2)/C#N SEW01621 CCOC(=O)c1cccc(c1)CSC(=N)N.Cl S07313 c1ccc(cc1)NC(=O)OCCSc2nc3ccccc3s2 S07346 c1ccc(cc1)CN(Cc2cccs2)C(=O)c3cccs3 SEW02709 c1cc(cnc1)/N=C\2/NC(=O)C(S2)CC(=O)Nc3ccc(cc3)OC(F)(F)F S13393 c1ccc2c(c1)c(cc(=O)o2)Nc3ccc(cc3)F S13400 C/C(=N\Cc1ccc(c(c1)Cl)Cl)/c2ccccc2O S03802 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccccc3 S06886 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)C(=O)c4c(onc4c5c(cccc5Cl)Cl)C S06916 CCc1ccccc1NCN2C(=O)c3ccccc3C2=O S03684 Cc1c(c(nc(n1)SCC(=O)C(C)(C)C)OC(=O)N(C)C)CC(=C)C RJF00957 c1cc(ccc1C(F)(F)F)NC(=O)c2cnc3n(c2=O)CCS3 SEW01460 c1cc(c(cc1NC(=O)c2cnc3n(c2=O)CCS3)Cl)F SEW01461 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)CCOc2ccc(cc2)F)/N SEW01466 COc1cc(c(cc1Cl)OC)NC(=S)NC(=O)c2ccccc2 S03773 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2ccc(c(c2F)C#N)N(C)C)N S13321 Cc1ccc(cc1C)NC(=O)C2CCCCC2C(=O)O S13353 CCOC(=O)c1ccc(cc1)NC(=S)NCCCN2CCOCC2 S03783 c1cc(ccc1CNC(=S)Nc2ccc(cc2)Cl)C#N S03789 c1cc(c(c(c1)Cl)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)F RJF00918 c1cc(c(c(c1)Cl)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl RJF00919 c1cc(ccc1CNC(=S)Nc2cc(ccc2Cl)Cl)C#N S03804 CCc1ccc(cc1)NC(=O)/C=C/C(=O)O S03807 c1cc(ccc1NC2=NC(CS2)(CO)CO)F S13260 c1cc(ccc1/N=C/C2=C(c3cc(ccc3SC2)Cl)Cl)Cl SEW02609 COc1ccc(cc1)/N=C/C2=C(c3cc(ccc3SC2)Cl)Cl SEW02610 c1cc(c(c(c1NC(=S)N)F)F)F S13513 Cn1c(cc(c1c2ccc(cc2)F)c3ccc(cc3)OC)c4ccc5ccccc5c4 S13512 COc1ccc(cc1)C2=NCCc3c2ccs3 SEW01483 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)C(C)(C)C)C S13474 CCOc1ccc(cc1)n2c(nnn2)SCC(=O)C(C)(C)C S13475 Cc1cccc(c1NC(=S)NCc2ccc(cc2)C#N)Cl S03793 CCOC(=O)c1ccc(cc1)NC(=S)NCc2ccc(cc2)C#N S03794 c1c(ccc(c1)C(F)(F)F)/C=C\2/C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/CCC2 S15054 c1c(ccc(c1)F)/C=C\2/C(=O)/C(=C/c3ccc(cc3)F)/CCC2 S15056 c1cc(cc(c1)C(F)(F)F)c2nc(no2)c3ccc(s3)c4ccno4 SEW02547 Cc1ccc(cc1)N2C(=O)C(=C3SCCCS3)C(=N2)C S15111 c1cc(cnc1)C2N(C(=O)CS2(=O)=O)Cc3ccc(cc3)F S15113 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc3c(cc(=O)oc3c2)COC RJF01136 COc1c(c(c2c(n1)-c3ccccc3C2)c4c(cccc4Cl)F)C#N S13714 c1ccc(c(c1)/C=N/c2ccc(cc2)OC(F)(F)F)O S13563 Cc1cccc(c1C)NC(=N)NC(=N)N RJF01025 c1cc2c(cc1NC(=N)NC(=N)N)OCO2 RJF01027 c1cc(ccc1OCCC(=O)O)F SEW01421 c1c(c(=O)n2c(n1)SCC2)c3nc(on3)CCCC(=O)O SEW01456 Cc1ccc(cc1)S(=O)(=O)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01029 COc1ccc(cc1OC)S(=O)(=O)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01030 c1cc(ccc1NC(=S)NN)Cl S00196 c1ccc(c(c1)/C=N/NC(=O)CCn2nc(nn2)c3cccc(c3Cl)Cl)Cl RJF02211 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CCC(=O)N/N=C/c3ccc(cc3)Cl RJF02213 CC(C(c1ccccc1OC)c2c(n(c(=O)n(c2=O)C)C)N)[N+](=O)[O-] S13319 CC(C)(C)c1ccc(cc1)C(=O)N2CCOCC2 S06987 c1ccc(c(c1)NC(=O)CC2C(=O)N/C(=N\c3ccc(cc3)C4CCCCC4)/S2)Oc5ccc(cc5Cl)Cl S06989 c1cc(c(c(c1NC(=O)/C=C\C(=O)O)F)F)F S13456 c1cc(c(cc1C(F)(F)F)Cl)/C=N/Nc2nc3ccc(cc3s2)Cl SEW01608 Cc1ccc(cc1Cl)NC(=S)NNC(C)(C)C S07295 c1ccc(c(c1)c2nc(nc(n2)N)N)C(F)(F)F RJF01071 COC(=O)c1ccc(c(c1)N2C(=O)C=CC2=O)C(=O)OC S13652 Cc1cccc(c1)NC(=S)Nc2ccc(cc2NC(=S)Nc3cccc(c3)C)C S00086 Cc1ccc2c(c1)c(=O)n(c(n2)SCC(=O)C(C)(C)C)c3ccc(c(c3)C)Br S13489 Cc1ccc(cc1)c2cc(c(n2C)c3ccc(cc3)C(F)(F)F)c4cccs4 S13497 CCOc1ccc(cc1)n2c(nnn2)SCC#C S07176 Cc1cccc(n1)NC(=S)Nc2ccc(cc2)OC S00011 COc1cc(cc(c1OC)OC)NS(=O)(=O)c2ccc(cc2Cl)C#N SEW01390 c1cc(cnc1)NS(=O)(=O)c2ccc(cc2Cl)C#N SEW01392 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)OC(F)(F)F S13611 C#CCOC(=O)c1cccc(c1)CSC(=N)N.Cl S07331 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)OC(F)(F)F S13613 Cc1ccccc1NC(=S)NCCc2ccc(cc2)OC S00340 Cc1cccc(c1)NC(=S)Nc2ccccn2 S00360 CC(C)(C)c1ccc(cc1)C(=O)NCc2ccco2 S07189 c1ccc(c(c1)/C=N/N=C\2/N(C(=O)CS2)c3cccc(c3)F)OC(=O)/C=C/c4cccs4 RJF01017 c1ccn(c1)c2ncnc(n2)Nc3cc(ccc3Cl)C(F)(F)F RJF01019 c1c(c(sc1S(=O)(=O)N)Br)Cl SEW02666 CC(C)(C)NNC(=S)Nc1cccc(c1)C(F)(F)F S07296 CN1C(C2CCCc3ccccc3C2=N1)c4ccc5c(c4)OCO5 S15209 c1cc(cc(c1)[N+](=O)[O-])/C=C/2\CSc3ccc(cc3C2=O)Cl S15268 Cc1cccc2c1c(=O)n(c(=S)[nH]2)c3ccc(cc3)OC(F)(F)F S13612 CSc1cccc(c1)NC(=S)Nc2ccc(cc2)F S04076 c1ccc(cc1)OC(=O)NC(=O)c2cccc(=O)o2 SEW01612 Cc1cc(nn(c1=O)CCO)O S15398 c1ccc2c(c1)nc(s2)SCCOC(=O)Nc3ccc(cc3)Cl S07358 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2CCOC(=O)C5CC5 S15181 CCc1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccccc3N S03810 COc1ccc(cc1)C2c3ccsc3CCN2 SEW01484 c1ccc2c(c1)CC/C(=C\c3cccs3)/C2=O S15290 Cc1ccc(cc1F)N2C(=O)CC(C2=O)CC=C S15210 c1ccc2c(c1)CCC3C2=Nc4ccccc4SC3c5cccs5 S15490 c1ccc2c(c1)c(nn(c2=O)CCO)O S15400 CC(C)NC(=S)Nc1ccc(c(c1)Cl)F RJF01226 CC(C)CNC(=S)Nc1ccc(c(c1)Cl)F RJF01227 c1cc(ccc1/C=C/2\COc3ccc(cc3C2=O)F)Cl SEW01541 c1ccc(c(c1)N2CCCCC2)OC(=O)Nc3ccc(cc3)OC(F)(F)F S13603 COc1ccc(c(c1)C(=O)O)Nc2cccc(c2)Cl S07382 Cc1cc(ccc1Br)n2c(=S)[nH]nn2 S07171 COc1ccc(cc1)C2c3ccsc3CCN2S(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SEW01489 c1c(c(=O)n2c(n1)SCC2)c3nc(on3)CSCC(=O)O SEW01475 CC(C)(CO)NC(=O)c1cc(ccc1Br)OC S07026 Cc1ccc(cc1)/C=C/2\CCc3ccccc3C2=O S15491 c1cc(cnc1)C(=O)Oc2ccc(cc2)c3csnn3 SEW01528 c1cc(ccc1n2c(=S)[nH]nn2)OC(F)(F)F S13590 CC1CN(CC(O1)C)c2ccccc2OC(=O)Nc3ccc(cc3)OC(F)(F)F S13602 CC(C)c1ccc(cc1)N2C(=O)C(SC2=O)c3ccccc3 S07146 Cc1cc(c(c(c1)C)n2c(=S)[nH]nn2)C S07169 c1cc(c(c(c1)Cl)/C=C/c2ccc(cc2)CSC(=N)Nc3cc(cc(c3)Cl)Cl)F.Br RJF01154 Cc1ccc(nc1)n2cc3ccccc3c2C#N S13535 CN(C)/C=N\C(=S)c1c(ccs1)CSc2ccc(cc2)Cl SEW02626 c1cc(ccc1SCc2ccsc2c3ncns3)Cl SEW02632 c1cc(ccc1Nc2n[nH]c(=S)s2)OC(F)(F)F S13598 CCOC(=O)c1ccc(cc1)NC(=S)NNC(C)(C)C S07297 COc1cc(cc(c1OC)OC)/C=C(\C#N)/C(=O)c2ccsc2 SEW02720 CC1=CC(=O)N(C1=O)c2ccc(c(c2)F)F S03927 c1cc(cc(c1)C(F)(F)F)c2nc(on2)c3cc(sc3)[N+](=O)[O-] SEW02739 c1cc(ccc1c2cc(=O)c3ccc(cc3o2)OCC(CS(=O)(=O)c4ccc(cc4)Cl)O)Cl SEW02752 CC(C)(C)c1ccc(cc1)C(=O)N(C)C S07386 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3ccc(c(c3)Cl)Br)C(F)(F)F RJF01099 Cc1c(c(nc(n1)c2ccc(cc2)Cl)O)CC(=C)C RJF01122 Cc1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S S00227 c1cc(c(cc1/N=C/c2cc(ccc2O)Br)F)F S03839 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(c(c2)F)F S03841 COC(=O)c1ccccc1NC(=O)/C=C\C(=O)O S03894 c1cc(c(cc1C(F)(F)F)Cl)N/C=C(\C#N)/C(=O)c2ccsc2 SEW02729 COC(=O)c1ccccc1N2C(=O)C=CC2=O S03895 CC(C)(C)c1ccc(cc1)NC(=O)c2cc(c(cc2C(=O)O)Cl)Cl S15499 c1c(cc(cc1C(F)(F)F)N/N=C\2/CCCNC2=O)C(F)(F)F SEW02698 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)SC)C(=O)C1)C S15250 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cccc4c3cccc4)C(=O)C1)C S15251 COC(=O)c1ccc(c(c1)NC(=O)/C=C/C(=O)O)C(=O)OC S13649 c1ccc(cc1)C2C3=C(c4ccccc4CC3)NC(=S)N2 S15324 COc1ccc(cc1)C2c3ccsc3CCN2C(=O)c4ccccc4Cl SEW01496 COc1ccccc1NC(=S)Nc2ccccc2OC S00068 Cc1ccc(c(c1)C)NC(=S)Nc2ccc(cc2C)C S00139 CC(C)(C)c1ccc(cc1)N/C=C(\C#N)/C(=O)c2ccsc2 SEW02730 Cc1ccc(cc1F)NC(=S)Nc2ccc(cc2)Cl S00403 CC(C)(C)c1ccc(cc1)N2C(=O)c3cc(c(cc3C2=O)Cl)Cl S15501 CN(C)C(=O)Oc1cc(nc(n1)c2cc(cc(c2)Cl)Cl)COC RJF01257 c1ccc2c(c1)C/C(=C\c3cccc(c3)[N+](=O)[O-])/C2=O S15220 C=CCOc1ccc(cc1)C2C(=C(OC3=C2C(=O)CCC3)N)C#N S15236 CCOC(=O)Nc1cc(ccc1C(=O)OC)C(=O)OC S13647 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nc(on2)c3cc(sc3)[N+](=O)[O-] SEW02748 COC(=O)c1ccccc1N2C(=O)CC(C2=O)Sc3ccccc3N S03900 CN(C)C(=S)Nc1ccccc1C(=O)OC S03902 CC(C)(C)c1ccc(cc1)/C=C/2\CCCc3ccccc3C2=O S15201 CC(C)(C)c1ccc(cc1)C2C3CCCc4ccccc4C3=NN2C S15202 C#CCOC(=O)Nc1ccc(cc1)Cl S07271 CC(C)(C)NNC(=S)Nc1ccc(cc1)F S07292 Cc1cc(ccc1NC(=O)/C=N/O)Cl S13719 c1ccc2c(c1)C(=O)C(C2=O)(NC(=O)c3ccc(cc3)C(F)(F)F)O S13721 c1cc(ccc1CNC(=S)Nc2ccc(cc2)F)C#N S04075 c1ccc(c(c1)c2nnn(n2)Cc3c(cccc3Cl)F)C(F)(F)F RJF01133 COCc1cc(=O)oc2c1ccc(c2)NC(=O)C3CC3 RJF01143 Cc1ccc(cc1Cl)c2nnn(n2)CC(=O)NN RJF01146 c1cc(ccc1C2=NN(/C(=N\c3ccc(cc3)OC(F)(F)F)/SC2)CCO)[N+](=O)[O-] S15316 c1cc(c(cc1Cl)Cl)C2C(=C(OC3=C2C(=O)CCC3)N)C#N S15243 c1ccc2c(c1)c(=O)n(c(n2)SCc3ccc(cc3)/C=C/c4c(cccc4Cl)F)c5ccc(cc5)F RJF01155 Cc1cc(nc(n1)SCc2ccc(cc2)/C=C/c3c(cccc3Cl)F)O RJF01156 CC(C)(C)NNC(=S)Nc1cccc(c1)OC S07293 c1cscc1C(=O)CC#N SEW02693 Cc1ccc(cc1/N=C\2/N(N=C(CS2)c3ccccc3)C)Cl S15302 C=CCC1CC(=O)N(C1=O)c2cccc(c2)C#C S15218 Cc1ccc(cc1)C2=NN(/C(=N\c3ccc(cc3)OC(F)(F)F)/SC2)CCO S15317 c1ccc(cc1)NC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)Nc4ccccc4 S00429 c1ccc2c(c1)cc([nH]2)c3ccc(cc3)F SEW02763 C1CCCCCC(CCCCC1)NC(=S)NN S00457 Cc1ccc(cc1Cl)c2nc(cc(n2)OC(=O)N(C)C)C(F)(F)F RJF01123 CCOC(=O)C1=c2n(c(=O)/c(=C\c3ccc(cc3)SC)/s2)C(=C(C1c4ccc(cc4)SC)C(=O)OCC)N S15341 COC(=O)c1ccc(c(c1)N2C(=O)CC(C2=O)Sc3ccccc3N)C(=O)OC S13653 COC(=O)c1ccc(c(c1)NC(=O)COCC(=O)O)C(=O)OC S13658 Cc1csc2c1[nH]c(=O)n(c2=O)CCO S13660 CN(C)C(=O)Oc1cc(nc(n1)c2ccc(cc2)Cl)COC RJF01089 Cc1c(c(c(c(c1C)C)CNC(=S)NN)C)C S04016 Cc1ccc(cc1Cl)c2nc(c(c(n2)OC(=O)N(C)C)CC(=C)C)COC RJF01120 CN(C)C(=S)Nc1cc(c(cc1OC)Cl)OC S03882 Cc1c(cccc1Cl)NC(=S)NC2CCCCCCCCCCC2 S00398 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)C(F)(F)F)C#N)N)C S13702 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)C#N)N)C S13705 c1ccc2c(c1)C/C(=C\c3ccc(cc3)C(F)(F)F)/C2=O S13708 c1ccc2c(c1)C/C(=C\c3ccc(cc3Cl)Cl)/C2=O S13710 c1csc2c1[nH]c(=O)n(c2=O)CCO S13661 C/C(=C\c1ccc(cc1)Cl)/[N+](=O)[O-] S04023 CCOC(=O)c1c(nc(s1)c2c(ccs2)COc3ccccc3)C SEW01707 c1ccc(cc1)NC(=O)c2cccc(=O)o2 SEW01560 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)Nc3cccc(c3)SC S04018 CC(C)(C)NNC(=S)Nc1cccc(c1)Cl S07291 COc1ccccc1c2c3c(nc(c2C#N)OC)-c4ccccc4CC3 S13689 COc1ccc(cc1)C2c3ccsc3CCN2C(=S)Nc4ccc(cc4Cl)Cl SEW01485 COc1ccc(cc1)C2c3ccsc3CCN2C(=S)NCC=C SEW01487 Cn1c(nnc1SCc2ccc(cc2)c3csnn3)C(F)(F)F SEW01435 c1ccnc(c1)SCc2ccc(cc2)c3csnn3 SEW01436 CCOC(=O)Cn1nc(nn1)c2ccc(c(c2)Cl)C RJF01132 Cc1cc(cc2c1NC(=O)C2=O)Cl S13720 CC(C)(C)NC(=S)Nc1ccccc1Cl RJF01216 Cc1ccc(cc1Cl)c2nnn(n2)CC(=O)C(C)(C)C RJF01128 c1ccc2c(c1)cc(o2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl SEW01581 CC(C)(C)S(=O)(=O)/C(=C/c1cc2ccccc2o1)/C#N SEW01583 c1cc(ccc1S(=O)(=O)/C(=C/c2cc(sc2)[N+](=O)[O-])/C#N)Cl SEW01584 c1c2c(cc(c1Cl)Cl)c(=O)n(nc2O)CCO S15497 CCOC(=O)c1csc(n1)c2ccc(cc2Cl)C(F)(F)F SEW01587 c1cc(ccc1S(=O)(=O)/C(=C/c2ccc(cc2Cl)C(F)(F)F)/C#N)Cl SEW01603 COc1c(c(c2c(n1)-c3ccccc3CC2)c4ccc(cc4Cl)Cl)C#N S13690 c1cc(ccc1N/N=C(\C#N)/C(=O)c2ccsc2)Cl SEW02694 c1cc(ccc1N/N=C(\C#N)/C(=O)c2ccsc2)OC(F)(F)F SEW02697 C/C(=C\c1ccccc1Cl)/[N+](=O)[O-] S03994 C/C(=C\c1cccs1)/[N+](=O)[O-] S03995 Cn1c(nnc1SCc2ccc(cc2)c3nnco3)C(F)(F)F SEW01517 COc1ccc(cc1)NC(=S)Nc2ccc(cc2)SC S00099 CC(C)(C)S(=O)(=O)/C(=C/c1cc(sc1)[N+](=O)[O-])/C#N SEW01586 CC(C)(C)c1ccc(cc1)NC(=O)N(C)C S07254 c1cc(c(cc1Cl)Cl)n2c(=S)[nH]nn2 S07473 COC(=O)c1c(ccs1)Br SEW02691 Cc1ccc(cc1)NC(=S)NNC(C)(C)C S07294 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)OCC=C)C(=O)C1)C S15245 c1ccc2c(c1)cc(o2)/C=C(\C#N)/S(=O)(=O)c3ccccn3 SEW01582 Cc1c(c(nc(n1)N)O)CC(=C)C RJF00938 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)O)CC(=C)C RJF00940 c1c(c(=O)n2c(n1)SCC2)/C(=N\O)/N SEW01449 CCCCCCCCCCCCN1C(SCC1=O)c2cccnc2 S07497 Cc1cc(oc(=O)c1)C(=O)OC SEW01567 c1ccc2c(c1)cc([nH]2)c3ccc(c(c3)Cl)F SEW02771 c1ccc2c(c1)cc([nH]2)c3ccc(c(c3)F)F SEW02776 Cc1c(c(c(c(c1C)C)CNC(=O)/C=C/C(=O)O)C)C S04011 Cc1cc(oc(=O)c1)C(=O)Nc2ccccc2 SEW01570 CC(C)(C)c1ccc(cc1)C(=O)Nc2cc(cc(c2)Cl)Cl S07534 c1cc(ccc1OS(=O)(=O)c2c(cc(s2)Br)Br)Cl SEW02669 Cc1c(oc(n1)C)c2ccn(n2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW01572 c1ccnc(c1)S(=O)(=O)/C(=C/c2cc(sc2)[N+](=O)[O-])/C#N SEW01585 c1ccc(cc1)C(=O)c2ccccc2N3C(=O)C=CC3=O S03980 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)C S15252 COCc1cc(=O)oc2c1ccc(c2)NS(=O)(=O)C RJF01161 c1ccc(c(c1)/C=N/N=C\2/N(C(=O)CS2)c3cccc(c3)F)O RJF01012 Cc1ccc2c(c1)c(=O)n(c(n2)SCC(=O)C(C)(C)C)c3ccc(cc3)OC S13487 c1cc(c(cc1NC(=S)N)Cl)Br S03725 CCc1ccc(cc1)N2C(=O)C=CC2=O S03808 CC(CCc1ccccc1)C/C=N/Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] SEW02780 c1c(c(cc(c1Cl)Cl)Cl)NC(=S)NCCCO S04187 c1cc(c(cc1Cl)NC(=S)NCCCO)Cl S04188 CSc1cccc(c1)NC(=O)N S04034 c1cc(ccc1NC(=S)NC2CCCCCCCCCCC2)F S00460 c1ccc2c(c1)CC/C(=C\c3ccccn3)/C2=O S15169 Cc1ccc(cc1Cl)Nc2ncnc(n2)n3cccc3 RJF01041 COc1ccccc1/C=C\2/C(=O)C3CCN2CC3 S13878 CN1/C(=N/c2ccc(cc2)Cl)/SCC(=N1)c3ccccc3 S15263 Cc1ccc(cc1)C(=O)NC(=S)NC(=O)NC S15264 CC(=O)N1C(=O)c2ccccc2C1=O S13730 c1cc(cc(c1)Cl)NC(=N)SCc2ccc(cc2)/C=C/c3c(cccc3Cl)F.Br RJF01158 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCO S15270 c1cc(c(c(c1)Cl)/C=C/2\COc3ccc(cc3C2=O)F)F SEW01542 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)C3CC3 S15253 CN1/C(=N/c2ccc(cc2)OC(F)(F)F)/SCC(=N1)c3ccccc3 S15256 c1cc(ccc1C(=O)NCc2csc3c2cc(cc3)Cl)C(F)(F)F S13447 c1cc(ccc1C(=O)NCc2csc3c2cc(cc3)Cl)F S13448 COc1ccc(cc1)C(CC(=O)c2ccc3ccccc3c2)C(=O)c4ccc(cc4)F S13507 C#CCSc1nnnn1c2ccc(c(c2)Cl)Cl S07178 Cc1c(c(n(n1)S(=O)(=O)c2ccccc2)O)CC(=C)C RJF01195 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3cc(ccc3C)Cl S13640 COC(=O)c1ccc(c(c1)N2C(=O)CSCC2=O)C(=O)OC S13646 c1c(c(sc1Br)S(=O)(=O)N2CCSCC2)Br SEW02662 CC1=NN(C(=O)C1CC(=C)C)C(=O)c2c(cccc2Cl)Cl RJF01200 C/C(=C\c1ccc(s1)Br)/[N+](=O)[O-] S04022 CSc1c(ccs1)/C=N/O SEW02717 c1cc(ccc1/C=C(\C#N)/C(=O)c2ccsc2)C(F)(F)F SEW02719 CC(=O)Nc1ccccc1OCC(CS(=O)(=O)Cc2ccc(cc2)Cl)O SEW02674 c1ccc(cc1)c2c[nH]nc2C(F)(F)F SEW02809 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)N3CCCC3 SEW02813 Cc1cc(no1)NC(=O)c2cc(c(s2)C(F)(F)F)c3ccccc3 SEW02814 CC(C)(C)NC(=S)NCC1CC1 RJF01241 CC(C)(C)c1csc(n1)c2c(ccs2)CS(=O)(=O)c3ccc(cc3)Cl SEW01724 c1ccc(cc1)/C=C/2\CCCc3ccccc3C2=O S15203 c1cc(ccc1NC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)Nc4ccc(cc4)Cl)Cl S00387 Cc1c(oc(n1)C)/C(=N\OC(=O)c2ccccc2)/C SEW01654 Cc1ccc(cc1C)NC(=C2C(=O)c3ccccc3C2=O)C#N S15446 CCOC(=O)c1ccc(cc1)/N=C/c2cc(cc(c2O)I)I S00540 Cc1cc(ccc1/N=C/c2ccc(c(c2)OC)OCc3ccccc3)Br S00602 c1cc(ccc1NC(=S)NCC2CC2)Cl RJF01268 c1ccc2c(c1)C(=O)C(C2=O)(NC(=O)c3ccc(cc3)C(F)(F)F)N4CCCCC4 S13742 Cc1csc([n+]1C(C)C)Nc2ccc(c(c2)Cl)F.[I-] RJF01246 Cc1cccc(c1NC(=S)NCCC(=O)O)C RJF01261 c1ccnc(c1)c2nc(cc(n2)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F RJF01192 c1cc(c(cc1Cl)Cl)/N=C\2/NCCS2 S04109 COc1ccc(cc1OC)Cc2nnc(o2)N S15380 c1cc(=O)n(nc1O)CCO S15381 c1ccc2c(c1)C3N4C2OCC4(CO3)CO S13755 Cc1ccc(cc1)C(=O)C2C(NC(C2c3cccs3)c4ccc(cc4)Cl)c5ccc(cc5)C(F)(F)F S13778 c1cc(c(c(c1)Cl)Cl)NC2=NCCS2 S04126 c1cc(ccc1N2C(=O)CSC2=O)OC(F)(F)F S13582 c1cc(ccc1NC2=NCCS2)OC(F)(F)F S13588 CCOC(=O)c1c(ocn1)c2ccco2 SEW01565 c1ccc(c(c1)/C=N/N=C\2/N(C(=O)CS2)CC3CC3)Cl RJF01279 CC(C(=O)O)NC(=O)c1ccccc1 S07576 COc1cc(ccc1OC(=O)/C=C/c2cccs2)/C=N/c3cc(cc(c3)Cl)Cl RJF01283 c1ccc(cc1)/C(=N\NC(=O)c2ccc(cc2)Cl)/C(=O)O S13855 c1cc(ccc1/C=C\2/C(=O)C3CCN2CC3)F S13876 c1c(c(sc1Br)S(=O)(=O)N2CCOCC2)Br SEW02658 CC1(CC(=CC(=O)C1)NC(=O)Nc2ccc(cc2)Cl)C S07362 c1cc(c(cc1F)N2C(=O)C=CC2=O)F S03893 c1ccc2c(c1)CCC(=C2Cl)/C=N/O SEW01827 COc1ccc2c(c1)CCC(=C2Cl)/C=N/O SEW01829 c1cc(c(c(c1)Cl)SCc2ccc(cc2)c3ncns3)Cl SEW01830 c1cc(cc(c1)Br)N2C(=O)C=CC2=O S04151 c1cc(c(c(c1)Cl)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl)Cl RJF01374 Cn1nc(nn1)c2cc(cc(c2)Cl)Cl RJF01380 COc1ccc2c(c1)CCC3C2=Nc4ccccc4SC3c5ccc(cc5)C(F)(F)F S15506 c1cc(c(c(c1)Cl)Cl)Nc2nnc(s2)S S04127 c1cc(c(c(c1)Cl)/C=C\2/C(=O)C3CCN2CC3)F S13916 CC(=O)c1ccc(cc1)N/N=C\2/CCCNC2=O SEW02726 C1COCCN1CCCNC(=S)NN S03974 c1cc(sc1)C(=O)n2cc3c(n2)-c4cc(ccc4SC3)Cl SEW01834 COc1ccc(cc1OC)NC(=O)/C=C/C(=O)O S04110 COc1ccc(cc1OC)N2C(=O)C=CC2=O S04111 COc1ccc(cc1/C=C/2\C(=O)C3CCN2CC3)Br S13879 C#Cc1cccc(c1)NC(=O)c2cc3ccccc3oc2=O S13900 c1cc(cc(c1)Nc2ncnc(n2)N)C#N RJF01386 c1cc(cc(c1)[N+](=O)[O-])Nc2ncnc(n2)N RJF01387 C[n+]1c(ccc2c1cccc2)/C=C/c3ccc(cc3Cl)N(C)C.[I-] S04121 c1cc(c(c(c1)Cl)Cl)NC(=S)NCCO S04125 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)c5ccccn5)C(=O)N(C4=O)c6ccc(cc6)OC(F)(F)F)C2=O S13910 c1cc(c(cc1I)F)N2C(=O)C=CC2=O S07757 COc1ccc(c(c1)C(=O)Nc2ccc(cc2F)I)Br S07759 COC(=O)CS/C(=C(\C=N\O)/c1ccccc1)/C(F)(F)F SEW02910 c1cc(ccc1c2nc(on2)c3cnc4n(c3=O)CCS4)Cl SEW01537 c1cc(ccc1c2nc(on2)c3cnc4n(c3=O)CCS4)C(F)(F)F SEW01538 c1c(c(=O)n2c(n1)SCC2)C(=O)N SEW01539 c1ccc(cc1)n2c(=S)sc(n2)Nc3cc(ccc3Cl)Cl S03934 COCc1cc(=O)oc2c1ccc(c2)N RJF01106 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nc4cc(ccc4c(=O)o3)Cl S04139 Cc1c(nc(o1)C(=O)N)c2ccccc2 SEW01668 Cc1cccc(c1)N2C(=O)C3C(NC(=C4C(=O)c5ccccc5C4=O)C3C2=O)c6ccccn6 S13911 c1ccc2c(c1)C(=O)C(=C3C4C(C(N3)c5ccccn5)C(=O)N(C4=O)c6ccc(cc6)Cl)C2=O S13912 COc1ccccc1/C=C(\C#N)/C(=O)N S13825 COc1ccc(cc1OC)CC/N=C/c2ccccc2O S04153 COc1ccc(cc1OC)CC/N=C/c2cc(ccc2O)Br S04157 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)F)CC4CC4 RJF01264 CC(C)c1ccc(cc1)/C=C/2\CCc3cc(ccc3C2=O)OC S15505 Cc1ccc(cc1Cl)c2nc(c(c(n2)O)C)C RJF01127 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C(=N/O)/N SEW02865 CC(C)(C)c1ccc(cc1)C(=O)N/N=C(\c2ccccc2)/C(=O)O S13849 COC(=O)/C(=C\c1cccc2c1cccc2)/C#N S07731 c1ccc(cc1)c2cc(sc2C(F)(F)F)c3nc(no3)c4ccccc4 SEW02898 COc1ccc(cc1)/C=C\2/C(=O)C3CCN2CC3 S13925 c1cc(ccc1/C=C/2\C(=O)C3CCN2CC3)[N+](=O)[O-] S13926 c1ccc(cc1)c2c(c(ns2)N3CCOCC3)C#N SEW02750 CS(=O)(=O)/C(=C/c1ccsc1/C=C(\C#N)/S(=O)(=O)C)/C#N SEW01699 Cc1ccc(cc1)NC(=S)NCC2CCC(CC2)CNC(=S)Nc3ccc(cc3)C S00243 C1CCC2(CC1)NC(=O)CS2 S15369 CN1C(C2CCc3ccccc3C2=N1)c4cccs4 S15291 c1ccc(cc1)c2cc(sc2C(F)(F)F)c3nc(no3)c4cccc(c4)C(F)(F)F SEW02871 c1cc(ccc1C/N=C/c2cc(ccc2O)Br)C#N S04210 c1ccc(cc1)C(=O)CC(c2ccc(cc2)F)Sc3ccccc3C(=O)O S15464 c1ccc(cc1)C2=C3C(c4c2cc(cc4)F)Sc5ccccc5C3=O S15470 CCOc1ccc(cc1/C=C(\C)/[N+](=O)[O-])Br S04213 COc1ccc(cc1)C(=O)N/N=C(\c2ccccc2)/C(=O)O S13859 CC(C)c1ccc2c(c1)ccc[n+]2C.[I-] S13865 c1cc(ccc1/C=C/2\C(=O)C3CCN2CC3)C(F)(F)F S13871 CSc1ccc(cc1)/C=C/2\C(=O)C3CCN2CC3 S13872 Cc1ccc(cc1NC(=S)N(CCO)N)Cl S15295 C1CCC2(C1)NC(=O)CS2 S15370 COc1ccc(cc1)c2cc(nc(c2C#N)O)c3ccccc3 S07544 c1ccc2c(c1)C(=O)C(C2=O)(NCc3ccc(cc3)Cl)NC(=O)c4ccc(cc4)C(F)(F)F S13741 CCOc1ccc(cc1C=C(C#N)C#N)Br S04214 CCOC(=O)/C(=C/c1cccc(c1)Cl)/C#N S04228 Cc1c(oc(n1)C)/C(=N\OC(=O)c2ccsc2)/C SEW01657 c1csc(c1Br)C#N SEW02722 Cc1ccc(cc1)/C=N/N=C\2/N(C(=O)CS2)CC3CC3 RJF01280 COc1cc(ccc1OC(=O)/C=C/c2cccs2)/C=N/c3ccc(cc3)Cl RJF01281 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)Oc3cccc(c3)C(F)(F)F SEW02787 COc1ccc(cc1)OC(=O)c2cc(c(s2)C(F)(F)F)c3ccccc3 SEW02788 Cc1c(nc(nc1O)SCc2ccc(cc2)/C=C/c3c(cccc3Cl)F)C RJF01125 CCOc1ccc2c(c1)sc(n2)NC(=S)Nc3ccccc3OC S00420 Cc1ccc(cc1)C(=O)NC2(C(=O)c3ccccc3C2=O)NCc4ccc(cc4)Cl S13752 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)Oc3ccccc3 SEW02786 c1cc(c(cc1F)N/N=C\2/CCCNC2=O)F SEW02725 COc1ccc(cc1)NC(=S)N(CCO)N S15311 c1cc(c(cc1Cl)N/N=C\2/CCCNC2=O)Cl SEW02741 COC(=O)c1ccc(c(c1)NC(=O)CSCC(=O)O)C(=O)OC S13645 c1cc(cc(c1)C(F)(F)F)CSc2ccc(cc2)[N+](=O)[O-] S07233 CSc1ccc(cc1)/C=C/2\Cc3ccccc3C2=O S13691 CCOC(=O)C1=C(OC(=C(C1c2cc(cc(c2)OC)OC)C#N)N)C S13701 c1cc(c(cc1Cl)Cl)c2nc(on2)c3cc(sc3)[N+](=O)[O-] SEW02758 Cc1ccc(cc1)N/N=C(\C#N)/C(=O)c2ccsc2 SEW02700 COc1ccccc1/C=C/2\CCc3ccccc3C2=O S13685 COc1c(c(c2c(n1)-c3ccccc3C2)c4ccc(cc4)SC)C#N S13700 c1ccc2c(c1)C/C(=C\c3c(cccc3Cl)F)/C2=O S13711 COc1c(c(c2c(n1)-c3ccccc3C2)c4ccc(cc4)C(F)(F)F)C#N S13712 c1cc(ccc1c2c(c(ns2)N3CCOCC3)C#N)C(F)(F)F SEW02762 Cc1ccc(cc1)C(=O)NC2(C(=O)c3ccccc3C2=O)NCCc4ccc(cc4)Cl S13753 Cc1ccc(cc1)/C=C/2\CCc3cc(ccc3C2=O)OC S15329 CN1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)C#N S13845 c1cc2c(c(c1)N3C(=O)C=CC3=O)CCCC2 S07429 Cc1ccc(cc1)C(=O)CC(c2cccc(c2)[N+](=O)[O-])SCc3c(c(c(c(c3C)C)C)C)C S04003 c1ccc2c(c1)c(=O)n(c(n2)SCc3ccc(cc3)/C=C/c4c(cccc4Cl)F)c5ccc(c(c5)Cl)F RJF01164 Cc1c(c(no1)c2ccccc2)c3nc4ccccc4c(=O)o3 S04145 c1csc(c1C2OCCO2)C=C(C#N)C#N SEW01665 CC1=NNC(=O)C1CC(=C)C RJF01190 c1cc(c(c(c1)Cl)/C=N/Cc2ccc(cc2)Cl)F S13785 c1cc(sc1)C2NC(=O)CS2 S08134 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3Cl)Br S04201 c1cc2c(c(c1)NC(=O)/C=C\C(=O)O)CCCC2 S07428 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)Nc3cccc(c3)C(F)(F)F SEW02768 CC(c1ccc(cc1)/C=N/N=C/c2ccc(cc2)C(C)C)C S04058 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)/C=C/4\N=C(OC4=O)c5ccccc5)/C(=O)O2 S04064 Cc1ccc(n1c2ccc(cc2)/C=C(/C#N)\S(=O)(=O)C(C)(C)C)C SEW01693 CC(C)(C)c1csc(n1)c2c(ccs2)CSc3ccc(cc3)Cl SEW01703 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3ccc4c(c3)OCCO4)C2=O S07562 c1cc(sc1)C/N=C/c2cc(ccc2O)Cl S07677 c1ccc(cc1)C/N=C/c2cc(cc(c2O)Br)Br S04204 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC2c3ccccc3C(=O)O2 SEW01840 CCCCNC(=S)Nc1ccc(cc1F)F RJF01201 Cc1cccc(c1)c2nc(cc(n2)OC(C)C)COC RJF01204 CS(=O)(=O)/C(=C/c1c(ccs1)C2OCCO2)/C#N SEW01667 COC(=O)c1cc2c(s1)-c3cc(ccc3SC2)Cl SEW01676 Cc1ccc(n1c2ccc(cc2)Br)C SEW01677 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CC3CC3 S15254 CCCN1Cc2c(n(c(=O)n(c2=O)C)C)NC1 S15255 c1c(ccc(c1)/C=C/[N+](=O)[O-])/C=C/[N+](=O)[O-] S15343 CN(C)C(=S)NCc1cccs1 S07639 Cc1cc(ccc1N2C(SCC2=O)c3cccnc3)Br S07665 CCOC(=O)C1=c2n(c(=O)/c(=C\c3ccccc3)/s2)C(=C(C1c4ccccc4)C(=O)OCC)N S15344 Cc1c(nc(o1)C(=O)NC(=O)Nc2cccc(c2)C(F)(F)F)c3ccccc3 SEW01673 c1cc(sc1C=C(C#N)C#N)Br S04027 Cc1ccc(cc1)N2C(=O)/C(=C/N(C)C)/C(=N2)C S13836 c1ccc2c(c1)cccc2CC(=O)NC(CC(=O)O)C(=O)O S07583 c1cc(cnc1)CN2C(SCC2=O)c3cccnc3 S07598 CC1(CC(=CC(=O)C1)OC(=O)c2ccc(cc2)Cl)C S07438 CC1(CC(=CC(=O)C1)OC(=O)c2ccc(cc2)C(C)(C)C)C S07441 Cc1ccc(cc1)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl RJF01373 Cc1cc(c(cc1Cl)C)SCC(COc2ccc3c(=O)cc(oc3c2)c4ccc(cc4)Cl)O SEW02765 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)Oc3ccc(cc3Cl)Cl SEW02777 CSc1c(ccs1)/C=C(/C#N)\S(=O)(=O)C SEW02778 c1cc(ccc1CNC(=S)N(CCO)N)Cl S15356 c1ccc(cc1)SC(=O)c2cccc(=O)o2 SEW01559 c1cc(cnc1)NC(=O)CCSc2cccs2 SEW01788 CC(C)CCSc1nnc(s1)N S08083 C/C(=N\O)/c1cc(c(s1)C(F)(F)F)c2ccccc2 SEW02965 c1cc2c(cc1Cl)C(=O)CCO2 SEW01816 c1ccc2c(c1)nc(s2)/C=N/Nc3cccc(c3)C(F)(F)F SEW02967 CC(c1ccc2cc(ccc2c1)OC)C(=O)Nc3ccc(cc3)OC(F)(F)F S14046 Cc1c(c(nc(n1)c2ccccn2)NCc3ccccc3)Cl SEW02971 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)Nc3ccccn3 SEW02817 c1ccc(cc1)C2=N/C(=C/c3cccc(c3)Cl)/C(=O)O2 S04106 c1cc(ccc1SCc2nc(on2)c3ccsc3)Cl SEW01731 Cc1cc(ccc1OCc2ccc(cc2)C(=O)O)Cl S08029 c1cc(cc(c1)Cl)/C=N/NC(=S)N S08064 CCCCCSc1nnc(s1)N S08081 c1ccc(cc1)SC(=O)c2cc3c(s2)-c4cc(ccc4SC3)Cl SEW01784 c1ccc(cc1)SCC(COc2ccc(cc2)c3csnn3)O SEW02829 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(c(c3)Cl)Br S07986 COc1ccc(cc1)SCC(CNCc2ccc(cc2)Cl)O.Cl SEW02945 c1cc(c(cc1Cl)Cl)OCc2nc(on2)c3ccsc3 SEW01740 c1ccc(cc1)C2=N/C(=C\c3ccccc3Br)/C(=O)O2 S04107 Cc1ccc(cc1)Nc2nnc(s2)S S00596 c1ccc(cc1)C(=O)N2c3ccccc3C=CC2C#N S15361 C1CCC2(CC1)NC(=O)CS2(=O)=O S15372 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)C(C)(C)C S07944 c1ccc2c(c1)C(=O)C(=O)N2CNc3ccc(cc3F)F S07982 Cc1ccc(cc1)C2C3CCc4cc(ccc4C3=Nc5ccccc5S2)OC S15509 c1cc(ccc1C(F)(F)F)N2C(=O)c3cc(c(cc3C2=O)Cl)Cl S15512 CCCCCCCCCCCCN1C(S(=O)(=O)CC1=O)c2cccnc2 S15433 CC(C)c1ccc(cc1)/C=C/2\CCc3ccccc3C2=O S15437 CC(C)c1ccc(cc1)C2C3CCc4ccccc4C3=NN2C S15441 Cc1cc(nn(c1=O)c2ccccc2)O S15443 CCOC(=O)C/C(=N/Nc1ccc(cc1)[N+](=O)[O-])/C S15534 CCCSC(=S)c1c(nn(c1O)c2ccc(cc2)C)C S15550 CC(C)(C)c1ccc(cc1)NC(=C2C(=O)c3ccccc3C2=O)C#N S15445 c1ccc(cc1)NC(=C2C(=O)c3ccccc3C2=O)C#N S15449 c1c(c(cc(c1Cl)Cl)Cl)n2c(nnn2)S S04132 CC(C)(C)/N=C(/NCC1CC1)\NN.I RJF01262 CC(C)c1ccc(cc1)C2C3CCc4cc(ccc4C3=NN2C)OC S15507 C#Cc1cccc(c1)N2C(=O)c3cc(c(cc3C2=O)Cl)Cl S15508 CC(C)c1ccc(cc1)NC(=S)NN S15429 CC(CS(=O)(=O)c1ccc(cc1)Cl)(CS(=O)(=O)c2ccccc2Cl)O SEW03129 CC(c1ccc2cc(ccc2c1)OC)C(=O)N/N=C/c3ccccc3O S14049 CNNC(=S)NCCC1=CCCCC1 S14052 c1ccc2c(c1)CCCC2(CC#N)C#N S14058 c1ccc(c(c1)CC(=O)NNC(=S)Nc2ccc(cc2)OC(F)(F)F)Cl S14085 CN(C)C(=S)Nc1ccc(c(c1)Cl)Br S04208 CN(C)C(=S)Nc1ccc(cc1Cl)Br S04209 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)Cl)CC4CC4 RJF01263 Cc1cc(nc(n1)c2cccc(c2)Cl)O RJF01212 CC(C)(C)NC(=S)Nc1ccc(cc1F)F RJF01213 CC1CN(CC(O1)C)c2ccccc2O S08887 c1cc(c(c(c1)Cl)NC(=O)N2CCOC23CCCCC3)Cl S08893 c1cc(c(c(c1)Cl)C(CC(=O)N)CC(=O)N)Cl S08922 Cc1ccc(cc1)/N=C/c2cc(cc(c2O)I)I S00686 c1cc(cnc1)C2N(C(=O)CS2)c3ccc(cc3F)F S07727 COC(=O)/C(=C/c1ccc(cc1)Cl)/C#N S07747 c1cc(c(cc1I)Cl)N2C(=O)C=CC2=O S07748 c1cc2c(cc1Br)C3(C(=O)N2CN4CCOCC4)OCCO3 S13961 COc1ccc(c(c1)C(=O)Nc2ccc(cc2Cl)I)Br S07752 c1cc2c(cc1Cl)nc(o2)S S04169 CCN(CC)C(=S)Oc1c(c(nc(n1)c2ccc(cc2)Cl)C)CC(=C)C RJF01214 Cc1c(oc(n1)C)/C(=N\OC(=O)c2ccc(cc2)C(F)(F)F)/C SEW01647 c1cc(sc1)CN2CN(C(=S)SC2)Cc3cccs3 S07629 Cc1cccc(c1)/N=C/c2cc(cc(c2O)I)I S00677 c1cc(sc1)CN2C(=O)CSC2=S S07634 c1ccc2c(c1)cccc2CC(=O)NCc3cccs3 S07668 c1cc(n(c1)c2cc(cc(c2)Cl)Cl)C=C(C#N)C#N SEW02999 c1ccc(cc1)c2c(snn2)c3ccccc3 SEW03000 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)O/N=C(/c3ccccc3)\N SEW02897 COc1cc(ccc1OC(=O)/C=C/c2cccs2)/C=N/c3ccc(cc3F)F RJF01282 c1ccc(cc1)/C=N/C2CCCCCCCCCCC2 S00795 c1cc(cnc1)C/N=C/c2cc(ccc2O)Br S04156 c1ccc2c(c1)cccc2CC(=O)NN S07413 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/C(=O)c2ccsc2 SEW02721 Cc1cc(ccc1Br)/N=C/c2ccc(cc2)[N+](=O)[O-] S00607 CCOC(=O)N/N=C(\Cc1ccccc1)/c2ccccc2 SEW02990 c1c(cc(cc1C(F)(F)F)NC(=N)NC(=N)N)C(F)(F)F RJF01321 c1ccc2c(c1)cccc2CC(=O)Nc3ccc(cc3F)F S07793 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(cc3F)F S07815 CCOC(=O)/C=C/1\CCCCCN1 SEW02808 CC(C)(C)NC(=O)c1cc(c(s1)C(F)(F)F)c2ccccc2 SEW02812 CC1=CCC2C(C1)C(=O)N(C2=O)c3cc(cc(c3)Cl)Cl S07819 CN(C)/N=C/c1ccc(o1)[N+](=O)[O-] S13933 COC(=O)/C(=C/c1ccccc1Cl)/C#N S07705 c1ccc(c(c1)N)SC(C[N+](=O)[O-])c2ccc(cc2)C(C[N+](=O)[O-])Sc3ccccc3N S15348 c1ccc2c(c1)CC/C(=C\c3ccc(cc3)C#N)/C2=O S13844 c1cc(cc(c1)C(F)(F)F)/C(=N/O)/N SEW02866 CC(=O)n1c(cc(n1)c2nccs2)SC SEW02867 Cc1csc([n+]1C(C)(C)C)Nc2cc(ccc2Cl)C(F)(F)F.[I-] RJF01309 C1CC1CNC(=S)NCCNC(=S)NCC2CC2 RJF01313 Cc1cccc(c1/N=C(/NC(=O)c2ccc(cc2)OC)\SC)C S09001 Cc1cc(c(c(c1)Br)NC(=S)NC(=O)c2ccccc2)Br S09051 Cc1ccc(cc1)c2nc(on2)c3cc(c(s3)C(F)(F)F)c4ccccc4 SEW02905 c1ccc(cc1)OC(=O)c2c(nccn2)N SEW02906 c1ccc(cc1)c2cc(sc2C(F)(F)F)c3nnc(o3)c4ccc(cc4Cl)Cl SEW02908 Cc1c(c(=O)oc2c1c(n[nH]2)C)Cc3c(cccc3Cl)F RJF01341 c1cc(ccc1C(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl)Cl RJF01342 CC(=O)c1cc(c(s1)C(F)(F)F)c2ccccc2 SEW02864 CCOC(=O)C1CSC(C(=O)N1)CC(=O)Nc2ccc(cc2)OC(F)(F)F S13992 Cc1ccc(c(c1)C(=O)Nc2ccc(cc2)Br)N S08548 CC(C)(C)c1csc(n1)c2c(ccs2)COc3ccc(cc3)Cl SEW01709 CCOC(=O)c1c(nc(s1)c2c(ccs2)COc3ccc(cc3)Cl)C SEW01710 Cc1cc(ccc1N2C(=O)CC(C2=O)Sc3ccccc3N)Br S08074 CCCCCCCSc1nnc(s1)N S08085 COC(=O)c1c(c2c(s1)-c3cc(ccc3SC2)Cl)N SEW01714 Cc1c(nc(o1)C(=O)NNC(=O)Nc2cccc(c2)C(F)(F)F)c3ccccc3 SEW01716 c1cc(c(cc1C2NC(=O)CS2)Cl)Cl S08129 Cc1c(nc(o1)C(=O)NNC(=O)NC)c2ccccc2 SEW01718 c1ccc(cc1)C2=C3C(c4c2cc(cc4)Cl)Sc5ccccc5C3=O S15461 c1ccc2c(c1)c(=O)oc(n2)c3ccccc3NS(=O)(=O)c4ccc(cc4)F S15482 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl S07820 c1ccc(cc1)/C=C/2\C(=O)N(C(=S)S2)c3cccc(c3)Br S07829 C1CCC(=CC1)CCNC(=O)/C=C\C(=O)O S14005 Cc1cc(ccc1Br)NC(=S)NN S04185 c1cc(ccc1/N=C/c2cc(cc(c2O)[N+](=O)[O-])[N+](=O)[O-])F S00816 COC(=O)/C(=C/c1ccc(cc1Cl)Cl)/C#N S07990 c1cc(c(cc1Br)Cl)NC(=S)NCCCO S04194 COC(=O)c1ccc(o1)CO/N=C(/c2ccc(cc2)C(F)(F)F)\N SEW01761 CC(=O)N(c1c2c(sc1C(=O)OC)-c3cc(ccc3SC2)Cl)C(=O)C SEW01768 COc1ccsc1/C=C/2\CSc3ccc(cc3C2=O)Cl SEW02943 c1ccc2c(c1)c(=O)n(c(n2)SCc3ccc(cc3)/C=C/c4c(cccc4Cl)F)c5ccc(cc5F)F RJF01163 CCC(CC)(C#C)Nc1ccsc1C(=O)O SEW02792 c1cnccc1NC(=S)N SEW02754 C/C(=C\c1ccc(cc1)/C=C(/[N+](=O)[O-])\C)/[N+](=O)[O-] S15347 c1cc(ccc1Nc2nnc(s2)S)Cl S00897 CN1C/C(=C\c2ccccc2)/C(=O)/C(=C/c3ccccc3)/C1.Cl S07872 c1cc2c(cc1Cl)-c3c(cc(s3)C(=O)O)CS2 SEW01776 c1cc2c(cc1Cl)-c3c(cc(s3)C(=O)N)CS2 SEW01779 CCOC(=O)c1csc(n1)c2c(ccs2)COc3ccccc3 SEW01706 c1ccnc(c1)S(=O)(=O)Cc2nc(on2)c3ccsc3 SEW01743 c1ccc(cc1)/C=C/2\C(=O)C3CCN2CC3 S15515 CC1=CC2(C3C(C1C4C2C(=O)N(C4=O)c5ccc(cc5)OC(F)(F)F)C(=O)N(C3=O)c6ccc(cc6)OC(F)(F)F)C S13994 c1cc(ccc1NC(=O)NCCC2=CCCCC2)OC(F)(F)F S14003 CC1=CC(=O)N(C1=O)c2cc(cc(c2)Cl)Cl S14008 C1CCC(=CC1)CCNC(=S)NN S14011 c1ccc2c(c1)CC/C(=C\c3ccc(cc3)[N+](=O)[O-])/C2=O S15522 C1CCC(=CC1)CCNC(=S)N(CCO)N S15354 CC(C)(C)c1ccc(cc1)n2c(nnn2)c3ccccc3 S07486 COC(=O)/C(=C/c1ccc(cc1)SC)/C#N S15338 COc1cc(cc(c1OC)OC)/C=N/c2ccc(cc2)Oc3ccc(cc3)Cl S00400 CC1(CC(=O)c2ccc(cc2O1)O)C S13733 CCCCCC1C/C(=C\c2ccc(cc2)C(F)(F)F)/C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/C1 S15557 CC1=C[C@]2(C3C(=O)N(C(=O)C3[C@@H]1C4C2C(=O)N(C4=O)c5cc(cc(c5)Cl)Cl)c6cc(cc(c6)Cl)Cl)C S13993 CC(C)(C)c1ccc(cc1)C(=N)SC(c2ccccc2)C(=O)C(F)(F)F SEW02955 c1ccc2c(c1)nc(s2)/C=N/Nc3ccccc3Cl SEW02964 CCOC(=O)/C(=C/c1ccccc1Br)/C#N S04230 c1ccc2c(c1)CCC3C2=Nc4ccccc4SC3c5ccc(cc5)C(F)(F)F S15495 COc1ccccc1/C=C/2\C(=O)OC(=N2)c3ccccc3 S04237 Cc1ccc(cc1Cl)NC(=S)NC2CCCCCCCCCCC2 S00401 CSc1c(ccs1)/C=C(/C#N)\C(=O)c2cccs2 SEW02782 CN(C)c1ccc(cc1)/C=C(\C#N)/C(=O)N S13826 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC3=CC(=O)CC(C3)(C)C S07440 c1cc(ccc1/N=C/c2ccc(s2)Cl)Cl SEW03832 COC(=O)/C(=C/c1ccc(cc1)F)/C#N S08234 CC(C)c1ccc(cc1)n2c(=O)n(sc2=O)c3ccc(cc3)SC(F)(F)F S13830 CCCCc1c(nc(nc1O)c2ccc(cc2)Cl)C RJF01211 C=C(C(CC(=O)O)C(=O)O)C(=O)O SB00530 c1ccc(c(c1)/N=C/c2cc(cc(c2O)I)I)Cl S00679 c1cc(ccc1/N=C/c2cc(cc(c2O)Br)Br)Oc3ccc(cc3)Cl S00828 CCc1cc(nc(n1)SCc2c(cccc2Cl)F)O RJF01413 c1cc(ccc1/C=C\2/C(=O)C3CCN2CC3)Cl S13920 c1ccc2c(c1)CC/C(=C\c3ccc(cc3)Cl)/C2=O S15438 CN1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)Cl S15440 Cc1c(oc(n1)C)/C(=N\OC(=O)c2ccc(cc2Cl)Cl)/C SEW01653 Cc1ccc(n1c2ccc(cc2)/C=N/Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C SEW01685 Cc1ccc(n1c2ccc(cc2)/C=N/Nc3ccc(cc3F)F)C SEW01687 c1cc2c(cc1Cl)C(=C(CS2)/C=N/O)Cl SEW01690 CCOC(=O)/C(=C/1\CCc2c1cccc2)/C#N S14064 COc1ccc2c(c1)CCCC2(CC#N)C#N S14066 CC1(CC2(N(c3ccccc3C(=O)O2)C(=S)N1)C)C RJF01400 c1cc(cc(c1)OCc2nc(on2)c3ccsc3)C(F)(F)F SEW01741 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNC(=S)N S04374 Cc1cc(cc(c1)NC(=O)/C=C/C(=O)O)C S04381 Cc1ccc(cc1)NC(=S)NCCO S00591 c1cc(cnc1)C2N(C(=O)CS2)Cc3ccc(c(c3)Cl)Cl S07600 c1cc(cnc1)C2N(C(=O)CS2)Cc3ccc4c(c3)OCO4 S07606 Cc1ccc(cc1)N2C(=O)/C(=C/Nc3ccc(cc3)F)/C(=N2)C S13978 Cc1ccc(cc1)N/C=C/2\C(=NN(C2=O)c3ccc(cc3)C)C S13979 COc1cc(ccc1OC(=O)C2CC2)/C=N/NC(=O)Cn3nc(nn3)c4c(cccc4Cl)Cl RJF01301 C1CCC2(C1)C3CCC=C3C(=C(C2(C#N)C#N)N)C#N S04359 CC/C(=N\CCc1ccc(c(c1)OC)OC)/c2ccccc2O S04266 CCc1ccccc1n2c(=O)c3ccccc3[nH]c2=S S04273 c1ccc(cc1)c2ccc(cc2)OC(=O)Nc3ccc(cc3)Cl S08003 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3c(cccc3Cl)F S07615 c1cc2c(cc1CN3C(=O)C=CC3=O)OCO2 S04055 CSc1cccc(c1)NC(=S)Nc2cccc(c2)SC S04071 CCOC(=O)/C(=C/c1ccc(cc1)/C=C(/C(=O)OCC)\C#N)/C#N S08184 C=CCNC(=S)NCCO S01173 C/C(=C\c1ccccc1[N+](=O)[O-])/[N+](=O)[O-] S04302 CC1=CC2(C3C(C1C4C2C(=O)N(C4=O)c5ccc(cc5)OC)C(=O)N(C3=O)c6ccc(cc6)OC)C S13995 CN(C)c1ccc(c(c1C#N)F)/C=C(\C#N)/S(=O)(=O)C SEW01810 CC(C)(C)S(=O)(=O)/C(=C/c1ccc(c(c1F)C#N)N(C)C)/C#N SEW01811 Cc1c(c(on1)C(F)(F)F)C(=O)O/N=C(/c2ccc(cc2)Cl)\N SEW03107 c1csc(c1Br)C(=O)O SEW01838 CC(CNCc1ccc(cc1)Cl)(CSc2cccc(c2)Cl)O.Cl SEW03118 CN(c1c(cc(cn1)Cl)C(F)(F)F)NC2c3ccccc3C(=O)O2 SEW01847 COC(=O)c1cc(=O)n2c3ccccc3sc2c1C#N SEW02991 CC(c1ccc2cc(ccc2c1)OC)C(=O)NN S14047 CCOC(=O)/C(=C/1\CCCc2c1ccc(c2)OC)/C#N S14057 COC(=O)c1cc(=O)n2ccccc2c1C#N SEW02992 CC(C)(C)C(=O)n1cc2c(n1)-c3cc(ccc3SC2)Cl SEW01837 c1cc(ccc1C(=O)Oc2ccc3c(c2)OCC3=O)Cl SEW03738 c1cc(ccc1c2csc(n2)c3ccsc3)[N+](=O)[O-] SEW03741 c1ccc2c(c1)CCC(=C2Cl)C#N SEW01842 c1cc(c(c(c1)Cl)/C=C/[N+](=O)[O-])F S09275 Cc1ccc2c(c1)c(=O)oc(n2)/C=C/c3ccco3 S08685 CCOC(=O)c1c(oc2c1c(c(c(c2F)F)F)F)CS(=O)(=O)c3ccc(cc3)Cl SEW03290 c1ccc(c(c1)CC(=O)NC2(C(=O)c3ccccc3C2=O)O)Cl S14092 c1cc(cc(c1)Cl)/C=N/C(=C(\C#N)/N)/C#N S08283 COc1cc(cc(c1O)Br)/C=C(\C#N)/C(=O)OC S08288 COc1ccc(cc1)c2c(sc(c2c3ccc(cc3)OC)C(=O)N)C#N SEW03025 c1cc(ccc1CNCC(CO/N=C/C2=C(c3cc(ccc3OC2)Cl)Cl)O)Cl SEW02957 c1cc(ccc1CNCC(CSc2ccc(cc2)[N+](=O)[O-])O)Cl.Cl SEW02959 c1ccc(cc1)N/N=C/c2nc3ccccc3s2 SEW02961 CSCC(Cn1c(=O)ccc(n1)O)O S15390 c1ccc(c(c1)N2CCSCC2)OC(=O)Nc3ccc(cc3)Cl S09268 CCCc1ccc(cc1)NC(=O)CC2C(=O)N/C(=N\c3ccc(cc3)C4CCCCC4)/S2 S09688 CCc1cc(nc(n1)c2ccc(c(c2)Cl)F)O RJF01408 CCOC(=O)Cc1csc(n1)N SB00646 Cc1cc(nc(n1)NC(=O)C(C)(C)C)O RJF01423 COc1ccc(c(c1)[N+](=O)[O-])NC(=O)/C=C/C(=O)O S08735 CN(C)/C=C\1/C(=O)N(C(=S)S1)c2ccc(cc2)F S08743 CC(C)c1ccc(cc1)N2C(=O)/C(=C/N(C)C)/SC2=S S08745 C/C(=C\c1ccc(cc1)OC)/[N+](=O)[O-] S04334 c1ccc2c(c1)C(=O)N(C2=O)O S04335 Cc1c(c(on1)C(F)(F)F)C(=O)NNC(=O)c2cccc(c2)C(F)(F)F SEW03143 Cc1ccc(cc1)NC(=S)Nc2ccccc2F S00570 Cc1cccc(c1)c2nc3cc(ccc3o2)C S15553 CCCC1C/C(=C\c2ccc(cc2)C(F)(F)F)/C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/C1 S15559 COc1ccccc1NC(=S)NCCC(=O)O RJF01422 c1cc(c(cc1N2C(=O)CSC2=S)Cl)F S08870 Cc1cccc(c1C)NCN2C(=O)c3ccccc3C2=O S04401 Cc1c(cccc1Cl)Nc2nnc(s2)S S00903 Cn1c(n[nH]c1=S)C(F)(F)F SB00671 c1ccnc(c1)CCN2C(SCC2=O)c3cccnc3 S07605 CC(C)(C)c1ccc(cc1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl S08859 c1ccc(cc1)c2c(n3c(n2)SCC3)/C=N/c4cccc(c4)C(F)(F)F SEW03158 CC(C)(C)c1ccc(cc1)/N=C/c2c(nc3n2CCS3)c4ccccc4 SEW03160 COc1ccccc1Nc2nnc(s2)S S01002 c1ccc2c(c1)c(nnc2O)O S01027 COc1ccc-2c(c1)CCc3c2sc(c3)C(=O)OC SEW01844 c1c([nH]c(=O)[nH]c1=O)C(=O)O SB00661 c1ccc(c(c1)c2csc(n2)Nc3cccnc3)Cl SEW03074 c1ccc(c(c1)/C=N/Nc2nc3c(c4ccccc4[nH]3)nn2)O S09153 c1cc(cnc1)Nc2nc(cs2)c3ccc(cc3)F SEW03079 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3ccc(cc3F)F)C2=O S07852 CN1C/C(=C\c2sccc2)/C(=O)/C(=C/c3sccc3)/C1.Cl S07875 CC1(CC(=CC(=O)C1)Nc2ccc(cc2)F)C SEW02818 c1csc(c1)/C=N/N=C/c2sccc2 S09337 c1ccc(cc1)COc2ccccc2C=C(C#N)C#N S08664 Cc1ccc2c(c1)c(=O)oc(n2)c3cc4ccccc4o3 S08678 CC(=O)c1cc(cc2c1CCC2(C)C)C(C)(C)C SB01378 c1cc(sc1)C(=O)CC(c2ccsc2)C(=O)c3cccs3 SEW03760 CCCc1ccc(cc1)N2C(=O)C=CC2=O S09387 CC(C)C(=O)Nc1csc(c1c2ccccc2)C(F)(F)F SEW03203 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3cccc(c3)F)C2=O S09737 c1ccnc(c1)/N=C/c2cc(cc(c2O)Br)Br S00827 c1ccc(cc1)/C=N/C(=C(\C#N)/N)/C#N S08309 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)Nc3ccc(cc3Cl)Cl SEW02825 Cn1cc(c(n1)C(F)(F)F)c2ccccc2 SEW02858 c1cc2c(cc1Br)C3(C(=O)N2CN4CCCCC4)OCCO3 S13962 c1cnc2n(c1=O)COCS2 S13973 c1cc(c(cc1F)F)NC(=S)NCCNC(=S)Nc2ccc(cc2F)F RJF01304 COc1cc(cc(c1OC)OC)N2C(=O)C=C(C2=O)c3ccccc3 S09271 c1cc(ccc1C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-])F S14113 c1cc(ccc1C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-])Cl S14114 c1cc(ccc1C(c2cc3c(cc2O)OCO3)N4CCCCC4)C(F)(F)F S14116 c1ccc(cc1)CNC(=O)c2c(c3ccsc3s2)Cl SEW03331 c1cc(ccc1C(c2cc3c(cc2O)OCO3)N4CCCC4)C(F)(F)F S14118 c1cc(ccc1C2C(=Cc3cc(cc(c3O2)Cl)Cl)[N+](=O)[O-])F S14119 CC(C)c1ccc(cc1)NC(=S)NCCC(=O)O RJF01446 CCOC(=O)/C(=C/c1cc(c(c(c1)Br)O)OC)/C#N S08291 C=CC1C[N@@]2CC[C@H]1CC2C(c3ccnc4c3cccc4)O SB01387 CC(CS(=O)(=O)c1ccc(cc1)Cl)(CS(=O)(=O)c2ccc(cc2)Cl)O SEW03072 c1ccc(cc1)c2c(sc(c2c3ccccc3)C(=O)N)C#N SEW02912 c1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)Sc3ccccc3C(=O)O S15458 c1ccc-2c(c1)-c3cccc4c3c2ccc4 SB00542 c1ccc(cc1)C/C(=N/OC(=O)c2ccc(cc2)Cl)/C(F)(F)F SEW03745 c1c(cc(nc1O)O)C(=O)O SB00524 CCOC(=O)Cn1nc(nn1)c2cccc(c2)[N+](=O)[O-] RJF01448 COc1ccc2c(c1)sc(n2)/N=C/c3cc(cc(c3O)[N+](=O)[O-])[N+](=O)[O-] S00807 c1cc(sc1)C(=O)Oc2ccc3c(c2)OCC3=O SEW03740 c1c(c(c(cc1Cl)Cl)O)/C=N/N=C/c2c(c(cc(c2)Cl)Cl)O S01047 CC1(NC(=O)CS1)c2ccc(cc2)Br S08148 c1cc(cc(c1)NC(=O)CCSc2cccs2)C(F)(F)F SEW01771 c1ccc2c(c1)C(=O)N(C2=O)CN3CCC(CC3)CCCC4CCN(CC4)CN5C(=O)c6ccccc6C5=O S01038 c1ccc(cc1)OC(=O)c2cc3c(s2)-c4cc(ccc4SC3)Cl SEW01783 c1ccc(cc1)C2C(=NC(=C(N2)C#N)C(=O)N)c3ccccc3 S08313 c1ccc2c(c1)nc(s2)/C=N/Nc3cccc(c3)F SEW02979 Cc1ccccc1NC(=S)NNc2ccc(cc2)[N+](=O)[O-] S01162 Cc1ccc(cc1)S(=O)(=O)CC(C)(CS(=O)(=O)c2ccc(cc2)C)O SEW03101 Cc1c(c(on1)/C=C/c2cccn2S(=O)(=O)c3ccccc3Cl)[N+](=O)[O-] SEW03294 Cc1ccc(n1c2ccc(cc2)/C=N/c3ccc(cc3)Cl)C SEW01721 COC(=O)c1c(c2c(s1)-c3cc(ccc3SC2)Cl)NC(=O)c4ccccc4 SEW01774 c1ccc(cc1)c2cc(sc2C(F)(F)F)c3nnc(o3)c4cccc(c4)C(F)(F)F SEW02948 c1cc2c(cc1[N+](=O)[O-])C(=O)NC2=O SB00340 c1cc(ccc1/C=N/Nc2ccc(cc2)C(F)(F)F)C(F)(F)F SEW03758 c1cc(ccc1C#N)OCc2nc(on2)c3ccsc3 SEW01742 c1ccc2c(c1)c(=O)oc(n2)c3ccccc3F S08246 COc1ccc(cc1Br)/C=C(\C#N)/C(=O)OC S08287 Cc1c(oc(n1)C)c2ccnc(n2)c3ccc(cc3)C(F)(F)F SEW01747 c1cc(ccc1C=C(C#N)C#N)OCc2ccsc2C#N SEW03026 c1ccc(cc1)c2cn3c(n2)SCC3 SEW02949 CCSC(=S)c1c(nn(c1O)c2ccccc2)C S15536 c1ccc2c(c1)c(cc(=O)o2)NCCC3=CCCCC3 S14023 Cc1ccc2c(c1)nc(o2)c3cccc(c3)Cl S15555 CC(C)(C)c1ccc(cc1)NC(=S)NCCCCCCNC(=S)Nc2ccc(cc2)C(C)(C)C S08670 c1cc(ccc1/C(=N/OCc2nc(on2)c3ccsc3)/N)C(F)(F)F SEW01746 c1ccnc(c1)c2cccs2 SB00516 c1ccc(c(c1)c2ccccc2C(=O)O)C(=O)O SB00521 C1CNCCC1CCCC2CCNCC2 SB00537 Cc1c(cccc1Cl)/N=C/c2ccc(cc2)N(C)C S00618 c1ccc2c(c1)c(=O)oc(n2)/C=C/c3ccco3 S08684 c1ccc(c(c1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)N S08525 c1ccc2c(c1)C(=O)N(C2=O)CNc3ccc(cc3)Oc4ccc(cc4)Cl S01037 C[n+]1c(ccc2c1cccc2)/C=C/c3ccc(c(c3)Cl)Cl.[I-] S08178 COC(=O)c1cc2c(s1)-c3cc(ccc3OC2)F SEW01765 c1ccc(cc1)NC(=O)c2cc3c(s2)-c4cc(ccc4SC3)Cl SEW01782 Cc1c(c(on1)C(F)(F)F)C(=O)O/N=C(/c2cccc(c2)C(F)(F)F)\N SEW03108 c1cc2c(cc1F)C(=C(CO2)/C=N/O)Cl SEW01815 CN1C/C(=C\c2c(cccc2)Cl)/C(=O)/C(=C/c3c(cccc3)Cl)/C1.Cl S07776 c1ccc(cc1)c2cnc(o2)c3ccccc3 SB00840 c1cc(ccc1NC(=O)CSCC(=O)O)F S10509 CC1=CC(N=C(N1c2ccc(cc2)Cl)SCc3c(cccc3Cl)Cl)(C)C RJF01352 Cc1c2c(cc(=O)oc2[nH]n1)COC RJF01357 c1cc(cnc1)Nc2nc(cs2)c3ccc(cc3)Br SEW03077 Cc1ccc(cc1)c2csc(n2)Nc3cccnc3 SEW03078 Cc1nc(no1)c2ccccc2 SEW01809 c1cc(oc1)COC(=O)c2c(c3ccsc3s2)Cl SEW03341 c1cc(sc1/C=N/Nc2c(cc(cc2Cl)Cl)Cl)[N+](=O)[O-] S09284 c1ccc(cc1)C2C(=O)c3ccccc3C2=O SB00622 c1ccc2c(c1)CCC23CC(=O)N(C3=O)CN4CCSCC4 S14071 CCc1cc(=O)oc2c1ccc(c2)O RJF01426 c1ccc2c(c1)C3(C(=O)N2)OCCO3 S13949 Cc1cc(=O)n2c(n1)SCOC2 S13974 c1cc(cc(c1)[N+](=O)[O-])c2n[nH]nn2 RJF01427 c1cc(cc(c1)Br)c2csc(n2)Nc3cccnc3 SEW03080 COc1ccc(c(c1)OC)NC(=O)/C=C/C(=O)O S04289 Cc1cccc(c1NC(=S)NN)Cl S01088 COc1ccc(c(c1)OC)N2C(=O)C=CC2=O S04290 c1cc(ccc1C2CCCCC2)NC(=O)/C=C/C(=O)O S09388 CC(C)(C)C(=O)Cn1nc(nn1)c2cc(cc(c2)Cl)Cl RJF01375 c1cc(cc(c1)F)c2csc(n2)Nc3cccnc3 SEW03084 COc1ccc(cc1)c2csc(n2)Nc3cccnc3 SEW03089 c1ccc2cc(ccc2c1)C(=O)Cn3nc(nn3)c4cc(cc(c4)Cl)Cl RJF01379 CC1=CC(N=C(N1c2cc(cc(c2)Cl)Cl)SCc3c(cccc3Cl)F)(C)C RJF01383 COc1ccc(cc1)C(=O)C2CC2 SB00571 CCn1nc(nn1)c2cccc(c2)[N+](=O)[O-] RJF01436 c1cc(cc(c1)Cl)NC(=S)NCCNC(=S)Nc2cccc(c2)Cl RJF01312 Cc1ccc(cc1)c2ncns2 SEW01822 c1cc(c(cc1F)F)NC(=S)NCCCC(=O)O RJF01314 CC(C)(C)C(=O)CSc1nc2ccccc2c(=O)n1CC3CC3 RJF01316 C/C(=C\c1cccc(c1)[N+](=O)[O-])/[N+](=O)[O-] S04301 c1csc2c1/C(=N\Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)/CCS2 SEW01798 CCn1nc(nn1)c2cc(cc(c2)Cl)Cl RJF01384 CC1(C(=O)N(C(=O)N1)CNc2ccc(cc2)F)C S04331 Cc1cccc(c1C)N2C(=O)C=CC2=O S04400 Cc1c(c(on1)C(F)(F)F)C(=O)NNC(=O)c2ccccc2 SEW03142 CN(C)/C=C/1\COc2ccc(cc2C1=O)Cl SEW01817 c1cc(ccc1C(=O)n2cc3c(n2)-c4cc(ccc4SC3)Cl)Cl SEW01826 CSc1ccc(cc1)OC(=O)Nc2ccc(cc2)Cl S08004 c1ccc2cc(ccc2c1)OC(=O)Nc3ccc(cc3)Cl S08008 c1ccc(cc1)c2c(csc2C(F)(F)F)NC(=O)c3ccco3 SEW03193 c1cc(cc(c1)Cl)NC(=S)NN S01122 c1ccc(cc1)c2c(csc2C(F)(F)F)NC(=O)C(Cl)(Cl)Cl SEW03201 Cc1ccc(cc1NC(=S)NCCO)Cl S01132 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)c4c(cccn4)C(=O)O)C(F)(F)F SEW03851 c1ccc(c(c1)CC(=O)Nc2ccc(cc2)OC(F)(F)F)Cl S14087 CSc1c2ccccc2[nH]c1c3ccc(cc3)Cl SEW03033 CN(C)C(=O)c1cc(c(s1)C(F)(F)F)c2ccccc2 SEW03093 Cc1cc(ccc1NC(=S)NN)Cl S01078 c1ccc(cc1)c2c(csc2C(F)(F)F)N3C(=O)CSCC3=O SEW03131 c1ccc(cc1)c2c(c(sc2C(F)(F)F)C(=O)O)N SEW03132 CC(C)(C)Cc1nc(no1)C2(CC2)c3ccc(cc3Cl)Cl SEW03886 COc1cc(cc(c1OC)OC)C(CC#N)CC#N S08589 CCNCC(=O)Nc1c(cccc1C)C SEW03864 c1ccc(c(c1)C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-])Cl S14102 c1cc(c(cc1Cl)Cl)C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-] S14111 C/C(=N\NC(=S)N)/c1ccc(cc1)Br S04357 c1ccc2c(c1)c(=O)oc(n2)c3ccccc3NS(=O)(=O)c4ccc(cc4)Cl S08837 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2F)F)c3nnco3 SEW03920 CC(C)(C)c1ccc2c(c1)nc([nH]2)/C(=C\c3ccc(cc3)F)/NC(=O)c4ccccc4 S08591 CC1=NN(C(=O)C1)c2cccc(c2)Cl SB00654 c1ccc2c(c1)C(=O)OC3(N2C(=O)C4C3C5CC4C=C5)O S10554 COc1ccc(cc1)NC(=O)CC(CC(=O)O)c2cc(c(c(c2)OC)OC)OC S08597 COc1ccc(cc1)N2C(=O)CC(CC2=O)c3cc(c(c(c3)OC)OC)OC S08599 c1ccc(cc1)Oc2ccc(cc2)N3C(=O)CC(C3=O)Sc4ccccc4N S08786 C1CCC2(CC1)C3CCCC=C3C(=C(C2(C#N)C#N)N)C#N S04361 COC(=O)/C(=C/c1c(nc2n1CCS2)c3ccccc3)/C#N SEW03153 CSc1cccc(c1)N2C(=O)CC(CC2=O)c3c(cccc3Cl)Cl S08581 c1ccc(cc1)c2c(n3c(n2)SCC3)/C=N/c4ccc(cc4)Cl SEW03159 Cc1c(c(on1)C)C(=O)NCC(c2ccccc2)c3c[nH]c4c3cccc4 SEW04402 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)NCc3ccc(cc3)C(F)(F)F)C SEW04403 Cc1c(c(nc(n1)NC(=O)C)O)Oc2ccccc2 SPB04464 CC(CNCc1cccc(c1)Cl)(CSc2ccc(cc2)Cl)O.Cl SEW03102 CC(CNCc1ccc(cc1)Cl)(CSc2ccc(cc2)Cl)O SEW03103 Cc1c(c(on1)C(F)(F)F)c2nnc(o2)c3cccc(c3)C(F)(F)F SEW03157 c1ccc(c(c1)Nc2nnc(s2)S)F S00982 c1ccc(c(c1)CC(=O)Nc2cc(cc(c2)Cl)Cl)Cl S14090 Cc1c(c(nc(n1)SCc2ccccc2)O)Oc3ccc(cc3)Cl SPB04465 Cc1c(c(on1)C)S(=O)(=O)Nc2csc(c2c3ccccc3)C(F)(F)F SEW03247 Cc1c(c(on1)C(F)(F)F)c2nc(no2)c3ccccc3 SEW03121 COC(=O)C(Cc1ccccc1)NC(=O)C(CC(=O)O)N SB00761 Cc1ccc2c(c1)ccc(=O)o2 SB00764 COC(=O)c1ccc(s1)/C=C/c2cccc(c2)Cl SEW03929 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3ccc(cc3)C4CCCCC4)C2=O S09391 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3cccc(c3)C#N)C2=O S09402 COc1ccc(cc1)CNCC(CSc2ccc(cc2)OC)O.Cl SEW03139 Cc1cc(c(cc1C)[N+](=O)[O-])NC(=O)/C=C\C(=O)O S09503 CC(=O)c1ccc(cc1[N+](=O)[O-])C(F)(F)F SEW03261 c1ccc(c(c1)CC(=O)Nc2ccc(cc2)C(F)(F)F)Cl S14093 CC(C)(C)NC(=O)N1CCC(CC1)C(=O)c2ccccc2 SEW04336 c1cc(c(cc1Cl)Cl)C(CC(=O)O)CC(=O)O S08220 c1ccc(c(c1)C2NC(=O)CS2)F S08239 CC(CS(=O)(=O)c1ccc(cc1)OC)(CS(=O)(=O)c2ccc(cc2)OC)O SEW03123 CN(C)/C=N/C(=S)N1CCOCC1 SEW03921 CN(C)c1cc(cnc1/C(=N/O)/N)C(F)(F)F SEW03923 c1cc(sc1)c2ccc(s2)c3ccnn3C(=O)Nc4ccc(cc4)Cl SEW03181 CCCc1ccc(cc1)N2C(=O)CCC2=O S09473 CCOC(=O)c1cnc2c(c(sc2c1N3CCOCC3)C(F)(F)F)c4ccccc4 SEW03257 C=CCn1c(=O)c2ccccc2[nH]c1=S S01176 CCOc1cc(cnc1/C(=N/O)/N)C(F)(F)F SEW03899 c1cc(ccc1c2nc(cs2)c3cc(c(s3)Cl)Cl)Cl SEW03948 c1cc(ccc1c2nc(cs2)c3cc(c(s3)Cl)Cl)F SEW03949 Cc1ccc2c(c1)c(=O)oc(n2)c3ccccc3F S08245 CC(=O)c1ccc(cc1)NC(=O)C SB00534 c1cc2c(cc1Cl)-c3c(cc(s3)/C=N/NC(=S)N)CO2 SEW03059 c1cc(cc(c1)N2C(=O)CCC2=O)C#N S09472 C#Cc1cccc(c1)NC(=O)/C=C\C(=O)O S09440 C#Cc1cccc(c1)N2C(=O)C=CC2=O S09441 CC(=O)c1cc(cc(c1)OC(=O)C)OC(=O)C SB00663 C[C@H]1[C@@H]2CC[C@]3(C=CC(=O)C(=C3[C@H]2OC1=O)C)C SB01489 CC1=CC(=O)CC(C1(/C=C/C(=C/C(=O)O)/C)O)(C)C SB00645 CCOc1cc(cnc1C#N)C(F)(F)F SEW03898 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc(cc3)C4CCCCC4 S09399 c1cc(c(cc1F)F)N2C(=O)CSCC2=O S10508 c1cc(ccc1N2C(=O)CSCC2=O)F S10510 c1ccc(c(c1)N2C(=O)CCC2=O)Oc3ccc(cc3Cl)Cl S09531 c1ccc2c(c1)C(=O)N(C2=O)CNc3ccccc3Oc4ccc(cc4Cl)Cl S09533 CCOC(=O)c1cnc2c(c(sc2c1N3CCCC3)C(F)(F)F)c4ccccc4 SEW03258 Cc1c(c(on1)/C=C/c2ccco2)[N+](=O)[O-] SEW03259 c1ccc(cc1)c2c3c(c(ncn3)Sc4cccc(c4)C(F)(F)F)sc2C(F)(F)F SEW03272 CC(C)n1nc(nn1)c2cccc(c2)[N+](=O)[O-] RJF01450 c1ccc2c(c1)cccc2Nc3nnc(s3)S S00985 c1ccc(c(c1)C(F)(F)F)/N=C/c2cc(cc(c2O)Cl)Cl S00901 Cc1ccc(cc1NC(=S)NN)Cl S00902 c1ccc2c(c1)[nH]c(n2)S S00965 Cc1ccc(cc1Cl)N2C(=S)C(=N)N(C2=O)c3ccccc3 S08347 C/C(=N\O)/c1ccc(cc1)Sc2ccccc2 SEW03319 Cc1ccc(cc1)c2nc(cs2)c3cc(c(s3)Cl)Cl SEW03947 c1ccc2c(c1)nc(s2)S S08979 COc1ccc(cc1)c2nc3ccccc3c(=O)o2 S09010 c1ccc2c(c1)nc(s2)SCCC#N S09019 COC(=O)C/C(=C(/C(=C(/C#C)\c1ccccn1)/C(=O)OC)\C(=O)OC)/C(=O)OC SEW03190 Cc1nc(cs1)c2cc(c(s2)Cl)Cl SEW03950 c1ccc2c(c1)C=C(C(O2)c3ccccc3Cl)[N+](=O)[O-] S09109 c1ccc(cc1)C2C(=Cc3ccccc3O2)[N+](=O)[O-] S09121 c1ccc2c(c1)C=C(C(O2)c3cccs3)[N+](=O)[O-] S09141 COc1ccc(cc1)/C=C(/CC(=O)O)\C(=O)O SEW03196 Cc1ccc(cc1)N2C(=O)/C(=C\Nc3ccc(cc3)Cl)/C(=N2)C S13983 c1cc(cc(c1)Cl)N2CSC(=C(C#N)C#N)SC2 S08407 c1cc(ccc1N2C(=O)CC(CC2=O)c3ccc(cc3Cl)Cl)F S08423 c1ccc2c(c1)c3c([nH]2)nc(nn3)N/N=C/c4cc(cc(c4O)Br)Br S09154 CCOC(=O)c1c[nH]c2c(c(sc2c1=O)C(F)(F)F)c3ccccc3 SEW03167 c1cc(cc(c1)NC(=O)N2CCOC23CCCCC3)C(F)(F)F S08892 Cc1ccc(cc1)NC(=O)n2c(ccn2)c3ccc(s3)c4cccs4 SEW03177 c1cc(cc(c1)Cl)NC(=O)n2c(ccn2)c3ccc(s3)c4cccs4 SEW03178 CC(CC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)CC(=O)O S10537 c1cc(cc(c1)[N+](=O)[O-])c2nnn(n2)Cc3c(cccc3Cl)F RJF01445 CCc1cc2c(cc1C(=O)Cn3nc(nn3)c4cccc(c4)[N+](=O)[O-])C(CCC2(C)C)(C)C RJF01447 c1cc(n(c1)c2cc(cc(c2)Cl)Cl)/C=N/Nc3ccc(cc3)[N+](=O)[O-] SEW03065 c1cc(cc(c1)Cl)c2csc(n2)Nc3cccnc3 SEW03075 CC(C)(C)c1ccc(cc1)/C(=N/OCc2ccc(o2)C(=O)OC)/N SEW01762 Cc1c(snn1)C(=O)N2CCC(CC2)C(=O)c3ccccc3 SEW04348 CC(CC(=O)Nc1cc(cc(c1)Cl)Cl)CC(=O)O S10534 c1ccc(c(c1)N2C(=O)C=CC2=O)Oc3ccc(cc3Cl)Cl S09528 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccccc3Oc4ccc(cc4Cl)Cl S09529 C1CC2(CCC1=O)OCCO2 SB00697 CN(C)C(=S)Nc1ccccc1Oc2ccc(cc2Cl)Cl S09568 c1ccc(cc1)Oc2cccc(c2)/C=C/[N+](=O)[O-] S14125 c1cc(cc(c1)[N+](=O)[O-])c2nnn(n2)CC(=O)NN RJF01449 c1cc(ccc1C(=O)c2ccc(cc2)F)F SB00771 Cc1c(c(on1)/C=C/c2ccc(cc2)OCc3ccsc3C#N)[N+](=O)[O-] SEW03018 c1ccc(cc1)S(=O)(=O)/C(=C/c2cccn2c3cc(cc(c3)Cl)Cl)/C#N SEW03037 c1cc(c(c(c1)Cl)C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-])Cl S14104 CC(C)(C)c1ccc(cc1)/C=C/[N+](=O)[O-] S14124 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccc(cc2)Sc3ccccc3 SEW03327 c1ccc(cc1)CCN2C(=O)c3ccc(cc3C2=O)C(c4ccc5c(c4)C(=O)N(C5=O)CCc6ccccc6)(C(F)(F)F)C(F)(F)F SEW03882 CC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2cccc(c2)C(F)(F)F SEW04060 CCOC(=O)c1c(nc(s1)c2c(cc(cn2)C(F)(F)F)Cl)C SEW03799 CCOC(=O)c1csc(n1)c2c(cc(cn2)C(F)(F)F)Cl SEW03801 c1cc(ccc1NC(=O)O/N=C(/c2cc(c(c(c2)Cl)N)Cl)\N)OC(F)(F)F SEW03768 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)Nc3ccc(cc3)Cl SEW04335 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)Nc3ccc(cc3)SC(F)(F)F SEW04337 COc1cc(cc(c1OC)OC)C(CC(=O)O)CC(=O)O S08592 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C(C)(C)C S08629 c1cc2c(cc1Br)C3(C(=O)N2)OCCCO3 S13981 Cc1ccc(cc1)N2C(=O)/C(=C/Nc3ccc(cc3)OC(F)(F)F)/C(=N2)C S13982 C1CC1CN2C(=O)CSC2=S S10480 c1cc(cnc1)C2N(C(=O)CS2)CC3CC3 S10482 c1cc(c(cc1F)F)NC(=O)CSCC(=O)O S10507 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2ccccc2N3CC(OC(C3)C)C)C)C S08890 COc1ccc(cc1)C/N=C/c2ccnc(n2)SCc3ccc(cc3Cl)Cl SPB04469 CCOC(=O)c1ccc(cc1)n2c(nc3ccc(cc3c2=O)Br)C S08970 CCC1(C=CN(C(=S)N1)c2cccc(c2)C(F)(F)F)CC SEW04352 Cc1c(c(on1)C)C(=O)Nc2cc(ccc2OCC(F)(F)F)C(F)(F)F SEW04363 CC(CC(=O)Nc1ccc(cc1F)F)CC(=O)O S10544 Cc1cc(no1)N2C(=O)CC(CC2=O)C S10546 Cc1c(c(on1)C(F)(F)F)c2nc(no2)c3ccc(cc3)Cl SEW03120 c1ccc(cc1)/C(=N\NC(=O)Cc2ccccc2Cl)/C(=O)O S14078 COc1ccc(cc1OC)Cc2c3cc(c(cc3ccn2)OC)OC.Cl SB01383 CN(c1cc(ccn1)C(F)(F)F)NC(=O)CSCC(=O)O SEW03976 Cc1ccc(cc1)NC(=O)CC(C)CC(=O)O S10535 CC1CC(=O)N(C(=O)C1)Cc2ccc(cc2)Cl S10536 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)Nc3ccccc3 SEW04338 c1ccc(cc1)C(=O)C2CCN(CC2)c3c(cccn3)[N+](=O)[O-] SEW04343 CC1CC(=O)N(C(=O)C1)c2cc(cc(c2)Cl)Cl S10538 CC1CC(=O)N(C(=O)C1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F S10540 CC(CC(=O)Nc1cccc(c1)C#N)CC(=O)O S10543 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)c4ccccc4C(=O)O)C(F)(F)F SEW03852 c1cc(ccc1SCc2csc(n2)c3ccsc3)Cl SEW03848 CCc1cc(nc(n1)S)O RJF01407 CCc1ccccc1NC(=S)NCCO S04269 Cc1ccccc1NC(=S)NCCO S01069 c1c(c(sc1Br)c2c(cc(s2)Br)Br)Br SEW03993 COc1ccc(cc1)C(=O)C2CCNCC2.Cl SEW03999 CC(C)(C)c1ccc(cc1)C(=O)n2c3cc(ccc3oc2=S)Cl S09607 Cc1c(c(on1)C)C(=O)Nc2cc(ccc2SC)Cl SEW03895 CCc1ccccc1Nc2nnc(s2)S S04272 CCc1ccccc1n2c(=O)c3cc(ccc3[nH]c2=S)C S04274 CC(=O)NNC(=O)c1cc2c(s1)-c3cc(ccc3SC2)Cl SEW01795 c1cc(ccc1N2C(=O)c3ccc(cc3C2=O)C(c4ccc5c(c4)C(=O)N(C5=O)c6ccc(cc6)Cl)(C(F)(F)F)C(F)(F)F)Cl SEW03880 c1ccc(cc1)CNC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)NCc4ccccc4 S01143 c1ccc(cc1)c2[nH]c3ccc(cc3n2)S(=O)(=O)O SB01057 c1cc(ccc1c2nc(no2)C3(CC3)c4ccc(cc4Cl)Cl)OC(F)(F)F SEW03884 c1cc(sc1)c2nc(no2)C3(CC3)c4ccc(cc4Cl)Cl SEW03885 c1cc(cc(c1)C(F)(F)F)C2CC(=O)CC(=O)C2 SEW03371 CC(C)Oc1cccc(c1)NC(=O)C SEW03281 c1ccc(c(c1)N)Oc2ccc(cc2Cl)Cl.Cl SB00593 c1cc2c(cc1Cl)-c3c(c[nH]n3)CS2 SEW01823 c1cc2c(cc1Cl)C(=C(CO2)/C=N/O)Cl SEW01828 c1ccc(cc1)c2c(n3c(n2)SCC3)C=C(C#N)C#N SEW03151 CC(c1ccc2cc(ccc2c1)OC)C(=O)Nc3cc(cc(c3)Cl)Cl S14042 CC(CNCc1ccc(cc1)Cl)(CSc2ccccc2Cl)O.Cl SEW03124 COc1cc(c(c(c1)Cl)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC SEW04396 CN(c1cc(ccn1)C(F)(F)F)N2C(=O)c3ccccc3C2=O SEW03978 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)C(=O)c3ccccc3 SEW04344 c1cc(sc1)C(=NOc2ccc(cc2[N+](=O)[O-])C(F)(F)F)c3cccs3 SEW03990 c1ccc(c(c1)OCc2nnn(n2)CC(=O)NNC(=O)Nc3ccc(cc3)Cl)Cl SPB01565 c1cc(c(cc1/C=N/Nc2c(cc(cc2Cl)C(F)(F)F)Cl)Cl)F SEW04068 CCOC(=O)C(C(=O)OCC)N.Cl SB00700 c1ccc(cc1)CNC(=S)NCCO S01142 c1cc(sc1c2ccno2)S(=O)(=O)N SEW03870 CCOC(=O)c1cc(on1)/C(=N/NS(=O)(=O)c2ccc(c(c2)Cl)F)/C SPB04602 CN(C)/C=N/NC(=O)c1nc(no1)c2cccc(c2)n3cccc3 SPB01501 COc1ccc(cc1OC)CC(=O)NNC(=S)Nc2cccc(c2)F S09983 CS(=O)(=O)c1ccc(s1)C(=O)O SEW03813 c1cc(sc1)CC(=O)Nc2cc(ccc2OCC(F)(F)F)C(F)(F)F SEW04364 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)OCCOc3cc(ccn3)C(F)(F)F SEW04074 Cc1cc(n(n1)c2ccc(cc2)C(F)(F)F)C SEW03824 COc1ccc(cc1)NCC(CSc2ccc(cc2)OC)O SEW03147 Cc1ccc(cc1)N2C(=O)CC(CC2=O)c3cc(c(c(c3)OC)OC)OC S08600 c1ccc2c(c1)C(=O)N(C2=O)CN3CCSCC3 S09244 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCSCC2 S09262 Cc1c(c(on1)C)C(=O)Oc2ccc(cc2)c3c([nH]nn3)C#N SEW03775 CC(C)(C)CC(=O)Oc1ccc(cc1)c2c([nH]nn2)C#N SEW03776 c1ccc(c(c1)NC(=O)CSCC(=O)O)Cl S10513 c1ccc(c(c1)N2C(=O)CSCC2=O)Cl S10514 C(C(=O)O)SCSCC(=O)O S09904 CC1(OC(=O)C(=Cc2cc3ccccc3o2)C(=O)O1)C SEW03784 c1cc(ccc1NC(=O)CSCC(=O)O)Br S10515 c1ccc(cc1)C(=O)NC(CCCNC(=N)N)C(=O)O SB01487 Cc1ccsc1C=C(C#N)C#N S09708 Cc1c(c(c(c(n1)C)C(=O)OC)c2cccs2)C(=O)OC SEW04367 COc1cc(cc(c1O)Br)/C=C(\C#N)/C(=O)N S08616 Cc1ccc(cc1)C(=O)CC(c2ccc(cc2)OC)SCc3c(cccc3Cl)F S08662 COc1ccc(cc1)SCc2nc(sn2)Sc3ccc(cc3)OC SEW03174 c1cc(c(nc1)ON=C(c2cccs2)c3cccs3)[N+](=O)[O-] SEW03989 Cc1cs/c(=N\C)/n1/N=C/c2c(cccc2Cl)Cl SPB01520 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)/C(=C/c3cccc(c3)Cl)/C#N SEW03380 CS/C(=C(/C#N)\C(=O)c1cc(c(s1)C(F)(F)F)c2ccccc2)/Nc3ccccc3 SEW03445 CCOC(=O)c1csc(n1)c2cnccn2 SEW03456 CCOC(=O)c1cc(n(c1c2ccccc2)c3cccc(c3)[N+](=O)[O-])C SEW04478 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCC2 SEW04450 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCOCC2 SEW04453 CN(C)S(=O)(=O)c1c(c(sc1C(=O)OC)C(F)(F)F)c2ccccc2 SEW03472 Cc1ccccc1NS(=O)(=O)c2c(c(sc2C(=O)OC)C(F)(F)F)c3ccccc3 SEW03473 c1cc(cc(c1)C(F)(F)F)c2c(nc(s2)N)C(F)(F)F SEW03119 c1cc(oc1C(=O)O)[N+](=O)[O-] SB00607 Cc1c(c(nn1C)C(=O)NNC(=O)c2ccc(cc2)C(C)(C)C)Br SPB01527 c1ccc(c(c1)N)SC(C[N+](=O)[O-])c2ccc(cc2)Cl S09937 Cc1c(snn1)C(=O)/C(=C(\C)/NC)/C(=O)OC SPB01540 CCOc1nnc(n1c2ccccc2)SCC(=O)OCC SPB01541 Cc1cc(c(cc1Cl)C)S(=O)(=O)Cc2ccc(cc2Cl)[N+](=O)[O-] SPB01544 CCOC(CC(=O)NNC(=O)c1ccc(cc1)C(F)(F)F)OCC SPB04487 CCOC(=O)c1cc(on1)/C(=N/OC(=O)c2ccc(cc2)Cl)/C SPB04488 CN(C)/C=C(\C#N)/C(=O)OC S08794 c1cc(cc(c1)N2C(=O)C=CC2=O)C#N S09411 c1ccc2c(c1)NC(=O)CC(S2)c3ccc(cc3)C(F)(F)F SEW04037 c1cc(sc1)c2ccc(s2)c3cccs3 SEW04049 CCOC(=O)/C(=C/c1c2ccccc2cc3c1cccc3)/C#N S09747 C(CCC(=O)NN)CC(=O)NN SB01476 CCOC(=O)c1cc(on1)c2csc(n2)COc3ccc(cc3)Cl SPB04540 COc1cc(c(c(c1)Cl)NS(=O)(=O)c2cc(c(s2)Br)Br)OC SEW04397 c1ccc(cc1)C(CNC(=O)C(F)(F)F)c2c[nH]c3c2cccc3 SEW04404 Cc1ccc(n1CCN2CCN(CC2)S(=O)(=O)c3ccc(cc3F)F)C SEW04406 CS(=O)(=O)/C(=C/c1c(nc2n1CCS2)c3ccccc3)/C#N SEW03152 c1ccc(c(c1)NC(=O)/C=C\C(=O)O)Oc2ccc(cc2Cl)Cl S09527 c1ccc(cc1)c2cc(sc2C(F)(F)F)COC(=O)Nc3ccccc3 SEW03279 c1cc(cc(c1)Cl)C2CC(=O)CC(=O)C2 SEW03372 CSC(=C(C#N)C(=O)c1cc(c(s1)C(F)(F)F)c2ccccc2)SC SEW03444 c1ccc(cc1)c2c3c(c(ncn3)Oc4ccc(cc4)C(F)(F)F)sc2C(F)(F)F SEW03365 CC1=CC(=O)N(C1=O)c2ccc(c(c2)Cl)F S09920 CS(=O)(=O)Nc1csc(c1c2ccccc2)C(F)(F)F SEW03233 CSc1ccccc1NCN2C(=O)c3ccccc3C2=O S09615 Cc1cc(n(n1)c2ccc(cc2)NN=C3C(=O)CCCC3=O)C SEW04374 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3ccc(cc3)F)\C4CC4 SEW03283 c1cc(cc(c1)NC(=O)COCC(=O)O)C#N S10475 c1ccc(cc1)c2c(csc2C(F)(F)F)NS(=O)(=O)c3cc(c(s3)Br)Br SEW03231 c1(c(c(sc1Cl)Cl)Br)S(=O)(=O)N SEW03377 Cc1cc(n(n1)c2ccc(cc2)NN=C(C(=O)OC)C(=O)OC)C SEW04373 CN(C)/C=C/C(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCC(CC2)C(=O)c3ccccc3 SEW04368 c1cnc(cn1)c2nc(cs2)CC(=O)O SEW03463 c1cc(ccc1c2cc[nH]n2)Cl SEW03384 CCOc1ccc2c(cc(=O)oc2c1)C SB00763 c1nc(c2c3c(sc2n1)CCC3)N SEW04390 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)c3c(nns3)C)C(=O)OC SPB01547 CC\1=NN(C(=O)/C1=N\OC(=O)c2ccc(cc2)Cl)C SEW03425 CS(=O)(=O)/C(=C/c1cccn1S(=O)(=O)c2ccccc2)/C#N SEW03242 Cc1ccc2c(c1)nc([nH]2)S SB00799 CC(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F SB00811 COC(C(C#N)c1ccccc1)(C(F)(F)F)OC SEW03841 c1cc(ccc1C(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F)Cl SEW03952 COC(=O)c1ccc(o1)CO/N=C(/c2cc(c(c(c2)Cl)N)Cl)\N SEW03930 COC(=O)c1c(c(c(s1)C(F)(F)F)c2ccccc2)S(=O)(=O)N3CCCC3 SEW03484 COC(=O)c1cc(cc(c1)Br)Br SEW04137 Cc1cc(n(n1)c2ccc(cc2)N/N=C(/C#N)\S(=O)(=O)C)C SEW04372 c1cc(nc(c1)C(=O)O)C(=O)O SB01598 CCCc1ccc(cc1)NCN2C(=O)c3ccccc3C2=O S09425 C/C(=N\CCc1ccc(cc1)Cl)/c2ccccc2O S09757 CSC(=S)NNC(=O)c1ccc(cc1)C(F)(F)F SPB01552 CCCCCCCCCCCc1nnc(n1c2ccccc2C(F)(F)F)SCc3ccccc3 SPB01553 Cc1ccc(n1CCN2CCN(CC2)S(=O)(=O)c3cc(c(s3)Br)Br)C SEW04408 Cc1c(snn1)C(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F SEW03953 c1cnc(cc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3cc(c(s3)Cl)Cl SEW03957 CCS(=O)(=O)N1CCN(CC1)c2cc(ccn2)C(F)(F)F SEW03959 Cc1cc(n(n1)c2ccc(cc2)NN=C(C#N)C#N)C SEW04371 CCOC(=O)c1cc(on1)c2csc(n2)Nc3ccc(cc3)C SPB04530 CCOc1cc(cc(c1OCC)OCC)c2c3cc(c(cc3ccn2)OC)OC SB01639 COCc1cc(nc(n1)COc2ccc(cc2)Cl)O SPB01582 CCOC(=O)O/N=C(/c1ccccc1)\C(=O)c2ccccc2 SB01037 CC(C)(C)NS(=O)(=O)c1c(c(sc1C(=O)OC)C(F)(F)F)c2ccccc2 SEW03485 c1ccc(cc1)c2c(csc2C(F)(F)F)NC(=O)C(Cl)Cl SEW03200 CC(CC(=O)Nc1ccc(cc1)F)CC(=O)O S10549 CCOC(=O)c1c(oc2c1c(c(c(c2F)F)F)F)CSCc3ccc(cc3)Cl SEW03297 CCOC(=O)c1c(oc2c1c(c(c(c2F)F)F)F)CS(=O)c3ccc(cc3)Cl SEW03310 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F)Cl SEW03956 c1cc(ccc1CO/N=C(/c2cc(c(c(c2)Cl)N)Cl)\N)Cl SEW03926 CC1(OC(=O)C(=Cc2ccc(o2)CO)C(=O)O1)C SEW03791 CCOC(=O)Cc1csc(n1)c2c(cc(cn2)C(F)(F)F)Cl SEW03800 Cc1c(c(n(n1)c2cccc(c2)Cl)O)N=Nc3ccccc3 SEW04010 c1nc(c2c3c(sc2n1)CCCC3)N SEW04391 c1csc(c1Br)C(=O)N SEW03839 CCOC(=O)c1c(oc2c1c(c(c(c2F)F)F)F)CS(=O)(=O)Cc3ccc(cc3)Cl SEW03299 CC(C)(C)/C(=N/O)/c1cccs1 SEW04123 c1cc(ccc1CCN2C(=O)C=CC2=O)Cl S09759 c1cc(ccc1CCNC(=O)/C=C\C(=O)O)Cl S09758 CCCc1ccc(cc1)N2C(SCC2=O)c3cccnc3 S09415 c1cc(cnc1)C2N(C(=O)CS2)c3ccc(cc3)C4CCCCC4 S09416 COc1cc(c(c(c1)Cl)NC(=O)c2cccc(c2)C(F)(F)F)OC SEW04394 c1cc(ccc1Oc2cc(cnc2C#N)C(F)(F)F)Cl SEW03901 c1cc(ccc1CCn2c(=S)[nH]nn2)Cl S09767 c1ccc(c(c1)C(=O)NCCc2ccc(cc2)Cl)I S09776 CCC(C)c1ccc(cc1)NCN2C(=O)c3ccccc3C2=O S09426 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)C3CCC3 SEW04346 Cc1c(sc(n1)c2ccccc2)C(=O)NNC(=O)c3c(nns3)C SEW04124 Cc1c(c(on1)C)C(=O)NNC(=O)c2c(nc(s2)c3ccccc3)C SEW04126 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)O SB00915 CC(C)(C)OC(=O)NC(CC(=O)N)C(=O)O SB00924 c1ccc(cc1)C(=O)c2ccc(cc2)F SB01595 C#Cc1cccc(c1)NCN2C(=O)c3ccccc3C2=O S09444 c1c(c(sc1S(=O)(=O)N2CCCCC2)Br)Br SEW03416 c1ccc2c(c1)C=C(C(O2)c3ccc(cc3Cl)Cl)[N+](=O)[O-] S10607 C/C=C(\C)/C(=O)N1CCC(CC1)C(=O)c2ccccc2 SEW04347 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cc(ccc2OCC(F)(F)F)C(F)(F)F SEW04365 CCOC(=O)CCn1c2ccccc2n(c1=S)CCC(=O)OCC S10519 Cc1ccc(o1)C=C2C(=O)OC(OC2=O)(C)C SEW03782 c1cc(ccc1NC(=O)Nc2nc(cs2)c3cc(c(s3)Cl)Cl)Cl SEW03964 c1cc2c(cc[nH]2)cc1[N+](=O)[O-] SB01605 c1ccc(c(c1)OC/C(=N/O)/N)Cl SPB01570 c1ccc(cc1)C2=N/C(=C\c3c4ccccc4cc5c3cccc5)/C(=O)O2 S09749 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=N/Nc2c(cc(cc2Cl)C(F)(F)F)Cl SEW04067 c1ccc(cc1)C2=CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl S09212 CCCc1ccc(cc1)n2c(=S)[nH]nn2 S09678 CCCc1ccc(cc1)NC(=S)NC(=O)c2ccccc2 S09679 CCCNC(=O)O/N=C(/c1cc(c(c(c1)Cl)N)Cl)\N SEW03770 CN(c1cc(ccn1)C(F)(F)F)NC(=O)c2ccccc2C(=O)O SEW03975 CN(c1cc(ccn1)C(F)(F)F)N2C(=O)CSCC2=O SEW03979 c1cc(c(cc1C(F)(F)F)NC(=O)C(Cl)(Cl)Cl)OCC(F)(F)F SEW04362 c1cc(ccc1/C=N/Nc2c(cc(cc2Cl)C(F)(F)F)Cl)C(F)(F)F SEW03811 c1cc(ccc1C2CCCCC2)N3C(=O)CCC3=O S09471 COc1ccc(cc1)Nc2c(cc(cc2Cl)OC)Cl SEW03941 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSc4ccc(cc4)Cl)C(F)(F)F SEW03819 c1cc(ccc1C2CCCCC2)NC(=O)CC3C(=O)N/C(=N\c4ccc(cc4)C5CCCCC5)/S3 S09687 CC(C)(C)NC(=S)N1CCSCC1 S09240 c1cc(ccc1NC(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F)OC(F)(F)F SEW03972 CC(C)(C)NC(=O)NCC(c1ccc[nH]1)C(F)(F)F SEW04468 CCOC(CC(=O)NNC(=O)c1ccc(cc1)Cl)OCC SPB04486 c1ccc(cc1)N2C(SCC2=O)c3ccc(cc3)Cl S09497 CCc1ccc(o1)C=C2C(=O)OC(OC2=O)(C)C SEW03783 CCOC(=O)c1c(oc2c1c(c(c(c2F)F)F)F)CS(=O)Cc3ccc(cc3)Cl SEW03305 c1ccc(c(c1)C(=O)Nc2ccc(cc2F)F)I S09778 CC1(OC(=O)C(=Cc2ccc(s2)Cl)C(=O)O1)C SEW03792 CCOC(=O)c1c(oc2c1c(c(c(c2F)F)F)F)CS(=O)(=O)c3cccc(c3)C(F)(F)F SEW03309 c1cc(ccc1SCc2nc(sn2)Sc3ccc(cc3)Cl)Cl SEW03082 CC(=O)c1cc(sc1)[N+](=O)[O-] SEW03166 CC(CC(=O)NCc1ccc(cc1)Cl)CC(=O)O S10533 c1ccc(c(c1)C(=O)NN)O SEW04563 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(on2)C SEW04432 C1CN(CCC1C(=O)O)CCC(=O)O.Cl SEW04564 c1cc(ccc1S(=O)(=O)n2cc3c(n2)CCOC3)Cl SEW04566 Cc1ccc(cc1)N2C(=O)CC(=N2)C SB01050 Cc1c(c(on1)C)C(=O)OCc2ccc(o2)c3ccc(cc3F)F SEW04412 Cc1cc(c(cc1Cl)C)S(=O)(=O)Cc2ccc(cc2)NC(=O)NC(=O)c3ccccc3Cl SPB01505 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CCC(=O)O)C(F)(F)F SEW03814 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSc4ccc(cn4)C(F)(F)F)C(F)(F)F SEW03816 c1nc(c2c3c(sc2n1)CCCCC3)N SEW04081 C[C@@H]1CC[C@@H]2C13CCC(C(C3)C2(C)C)(C)O SB01465 c1ccc(cc1)C(=O)NC(=S)Nc2ccncc2 SEW04082 c1cc(sc1)c2ccc(s2)/C=C(/CC(=O)O)\C(=O)O SEW03211 CCOC(=O)c1cc(on1)c2csc(n2)N/N=C/c3ccc(cc3)Cl SPB04516 CCOC(=O)c1cc(on1)/C(=N/OC(=O)c2ccccc2)/C SPB04519 Cc1c(sc(n1)c2ccccc2)C(=O)NN SEW04110 c1ccc(cc1)NC(=O)Nc2ccc(cc2Br)C(F)(F)F SEW04112 c1cc(sc1C=C(C#N)C#N)Cl SEW03825 COc1ccc(cc1OC)CC(=O)NN S09954 Cc1ccc(cc1)N2C(=O)CC(CC2=O)C S10539 Cc1cc(no1)NC(=O)CC(C)CC(=O)O S10542 CC1CC(=O)N(C(=O)C1)c2ccc(cc2F)F S10545 Cc1ccsc1/C=C/2\C(=O)OC(=N2)c3ccccc3 S09712 c1cc(ccc1OC(=O)c2c(c3ccsc3s2)Cl)Cl SEW03340 COc1cc2c(c(c1OC)OC)C(=O)/C(=C/c3ccc(cc3Cl)Cl)/C2 SEW04094 c1cc2cc(ccc2nc1)C(=O)O CC04501 c1cc(ccc1NC(=S)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl)F SPB01666 Cc1ccc(cc1)SC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl SPB01669 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)Sc3ccc(cc3)Cl)Cl SPB01670 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/CSc2ccc(cc2)Cl)\N SPB01673 CCOC(=O)/C(=C/c1ccc(cc1)Br)/C#N S10270 c1cc(c(cc1C(F)(F)F)NN=C(C#N)C#N)OCC(F)(F)F SEW04461 Cc1ccc(cc1)S(=O)(=O)/C(=N/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-] SPB01512 Cc1ccc(cc1)S(=O)(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/[N+](=O)[O-] SPB01513 CCOC(=O)c1c(c(n(n1)C)C)Br SPB01516 COc1ccc(cc1OC)Cc2nnc(n2c3ccc(cc3)F)S S09973 Cc1ccc(cc1Cl)n2c(nnc2S)Cc3ccc(c(c3)OC)OC S09974 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)c3c(noc3C)C)C SEW04166 c1cc(ccc1N/N=C(/CC(=O)C(F)(F)F)\C(F)(F)F)[N+](=O)[O-] SEW04168 COc1ccc(cc1OC)Cc2nnc(n2CC=C)S S09977 COC(=O)c1c(c(c(s1)C(F)(F)F)c2ccccc2)S(=O)(=O)N3CCOCC3 SEW03401 CCOC(=O)c1cc(on1)c2csc(n2)COc3ccccc3 SPB04503 CCOC(=O)c1cc(on1)c2csc(n2)c3ccc(cc3)C(F)(F)F SPB04526 Cc1c(c(nn1C)C(=O)NNC(=O)c2cccs2)Br SPB01528 c1cc(ccc1C2CCCCC2)NC(=S)N S09668 Cc1c(c(on1)C)C(=O)Nc2c(cc(cc2Cl)OC)OC SEW04395 CCCCCCCCCCCc1nnc(n1c2ccccc2C(F)(F)F)SCc3ccc(cc3)Cl SPB01555 c1ccc(c(c1)OCc2n[nH]nn2)Cl SPB01556 c1ccc(cc1)Oc2ccc(cn2)/C=C/C(=O)O SEW04420 CCSc1ccc(cn1)/C(=N/O)/N SEW04427 c1cc(cnc1)c2ncc(c(n2)N)C#N SEW03387 CCOC(CC(=O)NNS(=O)(=O)c1ccc(cc1)Cl)OCC SPB04493 COc1ccc(c(c1)SCC(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F)OC SEW03817 CCOC(=O)c1cc(on1)/C(=N/OC(=O)c2ccc(cc2)C(C)(C)C)/C SPB04521 CCOC(=O)c1cc(n(c1c2ccccc2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C SEW04477 c1ccc(c(c1)OCc2nc(on2)C(=O)N/N=C/c3c(cccc3Cl)Cl)Cl SPB01584 c1ccc(c(c1)OCc2nnc(o2)c3ccc(c(c3)Cl)Cl)Cl SPB01591 c1ccc(c(c1)OCc2nnc(o2)c3cccs3)Cl SPB01592 COC(=O)c1cc(n(n1)c2ccc(cc2)C(F)(F)F)O SEW03488 CCOC(=O)C(=Cc1cc(c(o1)C)C)C(=O)OCC SEW03788 CC1(OC(=O)C(=Cc2ccc(o2)c3ccc(cc3F)F)C(=O)O1)C SEW03786 Cc1ccc(s1)C=C2C(=O)OC(OC2=O)(C)C SEW03790 COc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])/C(=N/O)/N SPB01643 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NCC(c3ccc[nH]3)C(F)(F)F SEW04469 c1ccc(cc1)c2nc(cs2)CC(=O)NN SEW04113 Cc1c(c(nc(n1)NC(=O)C)O)Oc2cccc(c2)C(F)(F)F SPB04462 CCn1c(cc(n1)C)C(=O)n2c(c(c(n2)C)Sc3nccn3C)C SPB04468 Cc1c(c(nc(n1)NC(=O)C)O)Oc2ccc(cc2Cl)Cl SPB04471 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCc2cccs2 SEW04434 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)/C(=N/Nc3ccc(cc3)C(F)(F)F)/C#N SEW03405 C/C(=N\OC(=O)Nc1cc(cc(c1)Cl)Cl)/c2ccc3cc(ccc3c2)OC SEW04537 CCCCCCCCCCCc1nnc(n1c2ccccc2C(F)(F)F)S SPB01551 Cc1ccc(cc1)Oc2c(nc(nc2O)N)C SPB04459 Cc1ccc(c(c1)NC(=S)NNC(=O)Cc2ccc(c(c2)OC)OC)C S09986 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)CSCC(=O)O)C SEW04181 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)CCC(=O)O)C SEW04182 CC1=CC(=O)c2ccccc2C1=O SB01122 Cc1ccc(cc1)Oc2c(nc(nc2O)SCc3ccc(cc3)Cl)C SPB04476 Cc1ccc(cc1)S(=O)(=O)Cc2csc(n2)N3CCOCC3 SEW03916 Cc1c(sc(n1)C)C(=O)NNC(=O)COc2ccc(cc2Cl)Cl SPB01608 C1C2CC(C1C=C2)NC(=S)NN SEW04211 c1c(ccc(c1)/C(=N/O)/N)/C(=N/O)/N SEW04220 CCOC(=O)c1cc(on1)c2csc(n2)CS(=O)(=O)Cc3cccc(c3)C(F)(F)F SPB04500 c1ccc(cc1)NC(=O)OCCOc2cc(ccn2)C(F)(F)F SEW04073 COc1cc(cc(c1OC)OC)C2CC(=O)Nc3ccccc3S2 SEW04087 c1cc(ccc1c2csc(n2)c3ccno3)Cl SPB04508 Cc1c(sc(n1)C)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F SPB01609 Cc1c([nH]cn1)C(=O)N/N=C/c2ccncc2 SPB01618 Cc1ccc(cc1)Oc2c(nc(nc2O)NC(=O)C)C SPB04463 c1cc(c(c(c1)F)C(=O)NNC(=O)c2c(cccc2F)F)F SEW04415 c1ccc(cc1)Oc2ccc(cn2)C#N SEW04418 C#Cc1cccc(c1)NC(=O)c2ccc(cc2Cl)Cl S09463 CCSc1ccc(cn1)C#N SEW04425 CCOC(=O)c1cc(on1)c2csc(n2)c3cccc(c3)Cl SPB04496 c1c(c(sc1Cl)c2c(cc(s2)Cl)Cl)Cl SEW04063 CCCCNC(=O)OCCOc1cc(ccn1)C(F)(F)F SEW04071 CCOC(=O)c1cc(n(c1c2ccccc2)c3cccc(c3Cl)Cl)C SEW04479 Cc1c(c(n(n1)C)C(=O)Nc2ccccc2Cl)[N+](=O)[O-] SPB01652 Cc1c(c(n(n1)C)C(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] SPB01653 Cc1c(c(n(n1)C)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] SPB01655 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)/C(=C/c3ccc(cc3)Cl)/C#N SEW03379 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N SEW03381 c1cc(c(cc1C(F)(F)F)NN=C2C(=O)CCCC2=O)OCC(F)(F)F SEW04463 Cc1ccc(cc1)C(=O)C2CCNCC2.Cl SEW04466 c1cc(ccc1S(=O)(=O)Cc2cc3c(o2)c(c(c(c3F)F)F)F)Cl SEW03436 c1cc(c(cc1Cl)Cl)NC(=O)N2CCCCC2 SEW04586 CC(=O)Oc1ccc(cc1)c2csnn2 SEW04471 c1nc(no1)CSC(=S)N2CCOCC2 SEW04474 Cc1c(sc(n1)c2cnccn2)C(=O)O CC19801 c1cc(cc(c1)F)NC(=S)N SEW04593 Cc1c(c(n(n1)C)C(=O)O)[N+](=O)[O-] SPB01647 Cc1c(cnc(n1)N)Sc2ccccc2 SPB04584 c1ccc(cc1)C(=O)/C(=C/c2cccn2S(=O)(=O)c3ccccc3)/C#N SEW03243 Cc1c(c(n(n1)C(=O)c2cccs2)c3c(nns3)C)C(=O)OC SPB01546 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)Sc3ccc(c(c3)Cl)Cl)Cl SPB01671 c1cc(ccc1C(=O)O/N=C(/CSc2ccc(cc2)Cl)\N)C(F)(F)F SPB01674 COc1cc2c(c(c1OC)OC)C(=O)/C(=C/c3c(cccc3Cl)F)/C2 SEW04093 c1cc(c(cc1OC(F)(F)F)Br)NC(=O)CCC(=O)O SEW04095 COc1c(cc(cc1Br)/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/N)Br SPB01648 c1cc(ccc1c2nc(cs2)C(=O)/C=C/N3CCOCC3)C(F)(F)F SPB04570 CN(C)/C=C/1\Cc2cc(c(c(c2C1=O)OC)OC)OC SEW04096 COc1cc(cc(c1OC)OC)CCC(=O)NNC(=O)c2ccc(cc2)Cl SEW04106 Cc1ccc(cc1)NS(=O)(=O)c2c(c(sc2C(=O)OC)C(F)(F)F)c3ccccc3 SEW03486 Cc1cc(nc(n1)c2csc(n2)C)OC SPB04542 C/C=C/C(C#C)OC(=O)c1ccccc1C(=O)O SB01654 CCOc1cc(cnc1c2nc(cs2)CC(=O)OCC)C(F)(F)F SEW03912 c1ccc(c(c1)C(=O)NCc2ccc(cc2)Cl)I S09784 c1cc(cnc1)C2N(C(=O)CS2)CCc3ccc(cc3)Cl S09785 c1ccc(cc1)C2=CC(=O)N(C2=O)c3cccc(c3)Cl S09579 CCOC(CC(=O)NNC(=O)Nc1cccc(c1)C(F)(F)F)OCC SPB04483 Cc1c(c(n(n1)C)C(=O)O/N=C(/c2ccc(cc2)C(C)(C)C)\N)[N+](=O)[O-] SPB01661 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)NC(=S)NCC3CC3)Cl SPB01665 CSc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccccc3 S10245 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)Br)/C(=O)O2 S10268 CCOC(=O)c1nc(no1)CS(=O)(=O)c2ccc(cc2)Cl SPB01712 CCOC(=O)c1cc(on1)/C(=N/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C SPB04608 Cc1c(sc(n1)C(=O)Oc2ccc(cc2)Cl)C(=O)Oc3ccc(cc3)Cl SEW04646 CSc1ccc(cc1)/C=C/[N+](=O)[O-] S10015 c1cc(c(cc1[N+](=O)[O-])Cl)CS(=O)(=O)c2ccc(cc2F)F SPB01607 Cc1c(c(on1)C)c2nc(no2)COc3ccc(cc3)/C=C(/C#N)\S(=O)(=O)C SEW03313 c1c(c(sc1S(=O)(=O)N2CCCC2)Br)Br SEW03417 CCSc1ccc(cn1)c2nc(on2)C(C)(C)C SEW04441 CCSc1ccc(cn1)c2nc(on2)c3cccc(c3)C(F)(F)F SEW04442 c1coc(c1)/C=C\2/C(=O)/C(=C/c3occc3)/COC2 SEW04543 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)C4CCCCC4 S09843 CC1=CC(=O)N(C1=O)c2ccc(cc2)C3CCCCC3 S09865 Cc1ncc2c(ncnc2n1)N SEW04080 Cc1cc(c(o1)C)C(=O)Nc2cc(c(c(c2)OC)OC)OC SEW04546 c1cc(c(c(c1)F)C(=O)NCCCNC(=O)c2c(cccc2F)F)F SEW04549 CC1=CC(=O)N(C1=O)c2ccc(cc2F)F S09873 C(CSCSCCC(=O)O)C(=O)O S09907 c1cc(ccc1c2cnc([nH]2)S)Cl SPB01507 C=CCSc1[nH]c(cn1)c2ccc(cc2)Cl SPB01510 C[C@@H](c1ccc2cc(ccc2c1)OC)C(=O)O SB01071 CCOC(=O)/C(=C\Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-] SPB01495 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)CSc3ccc(cc3)Cl SEW04353 C#CCSc1[nH]c(cn1)c2ccc(cc2)Cl SPB01511 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)C(F)(F)F SEW04078 c1cc(ccc1c2nnco2)O SEW04592 COc1cc(cc(c1OC)OC)C2C(=Cc3ccccc3O2)[N+](=O)[O-] S10606 Cc1ccc(cc1)C2C(=Cc3ccccc3O2)[N+](=O)[O-] S10608 c1ccc(cc1)N2C(=O)CC(=N2)N SB01062 Cc1cc(c(cc1Cl)C)SCc2ccc(cc2)[N+](=O)[O-] SPB01499 Cc1cc(c(cc1Cl)C)S(=O)(=O)Cc2ccc(cc2)[N+](=O)[O-] SPB01502 Cc1cc(c(cc1Cl)C)S(=O)(=O)Cc2ccc(cc2)N SPB01503 Cc1cc(cc(c1)c2nc(on2)C(C)(C)C)c3nc(on3)C(C)(C)C SEW04026 c1cc(ccc1C(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F)C(F)(F)F SEW03951 CC(C)(C)CC(=O)N1CCN(CC1)c2cc(ccn2)C(F)(F)F SEW03954 c1ccc2c(c1)ncc(n2)N3CCC(CC3)C(=O)N SEW04038 c1cc(sc1)C(=O)/C(=N/Nc2ccc(cc2)[N+](=O)[O-])/C(=O)C(F)(F)F SPB04446 c1cc(ccc1SCc2n[nH]nn2)Cl SPB01676 Cc1c(c(n(n1)c2cccc(c2)Cl)O)/N=N\c3cccc(c3)Cl SEW04009 COc1cc(cc(c1OC)OC)C2CC(=O)Nc3ccccc3S2(=O)=O SEW04088 CC(=O)Nc1ccc(cc1Br)OC(F)(F)F SEW04090 c1cc(c(cc1OC(F)(F)F)Br)NC(=O)/C=C\C(=O)O SEW04091 c1ccc2c(c1)ncc(n2)SCCOC(=O)c3cc(cc(c3)Cl)Cl SEW04018 CN(c1ccc(cc1)OC(F)(F)F)C(=S)NC(=O)c2ccccc2 SEW04098 CCCC(=O)c1ccc(cc1O)NC(=O)C SB01739 CC(C)(C)NC(=O)N1CCN(CC1)c2cc(ccn2)C(F)(F)F SEW03973 c1ccc(cc1)NC(=O)NCC(c2ccc[nH]2)C(F)(F)F SEW04458 c1ccc(cc1)C2=N/C(=C\c3cccc(c3)Br)/C(=O)O2 S10269 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(/COc2ccc(cc2)c3nnco3)\N SEW04637 Cc1c(c(on1)C)C(=O)O/N=C(/COc2ccc(cc2)c3nnco3)\N SEW04640 Cc1c(sc(c1C(=O)c2ccc(cc2)Cl)/N=C/N(C)C)C SPB01711 Cc1c([nH]cn1)C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] SPB01619 Cc1ccc(cc1)/C=C\2/C(=O)NC(=S)N2 S10178 Cc1ccc(cc1)C2C(=O)c3ccccc3C2=O S10188 c1cc(ccc1C(=O)O/N=C(\c2ncc(s2)[N+](=O)[O-])/N)Cl SPB01633 c1cc(ccc1CSC(=S)N2CCN(CC2)C(=S)SCc3ccc(cc3)F)F SEW04579 Cc1ccc(cc1)Nc2nnc(o2)Cc3ccc(c(c3)OC)OC S10087 COc1ccc(cc1OC)Cc2nnc(o2)Nc3ccc(cc3Cl)Cl S10089 COc1ccc(cc1)OCCC(=O)O SEW04596 c1cc(sc1)C(=O)OCCSc2ccc(cc2[N+](=O)[O-])C#N SEW04251 C1CCC(CC1)C2NC(CS2)C(=O)O S10018 Cc1ccc2c(c1)c(cc(n2)C3CCCCC3)C(=O)O S10022 c1ccc2c(c1)c(=O)oc(n2)C3CC3 S10046 COc1ccc(cc1)SCc2cc3c(o2)c(c(c(c3F)F)F)F SEW03433 c1cc(c(cc1N2C(=O)C3C4CC(C3C2=O)C=C4)Cl)F S10415 Cc1cc(no1)NC(=O)Cc2cc(cc(c2)F)F SEW04675 CN(C)/C=C\1/C(=O)NC(=N1)SCc2c(cccc2Cl)Cl S10200 c1cc(ccc1/C=C\2/C(=O)NC(=S)N2)C#N S10206 CCOC(=O)c1cc(on1)/C(=N/NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C SPB04603 COc1ccc(cc1)c2ccc(s2)/C=N/Nc3c(cc(cc3Cl)Cl)C(F)(F)F SEW04653 c1cc(cnc1)/C=N/NS(=O)(=O)c2ccc(c(c2)Cl)Cl S10055 CCOC(=O)c1cc(on1)/C(=N/Nc2ccc(cc2)[N+](=O)[O-])/C SPB04605 c1cc(cc(c1)C(F)(F)F)C2=CCNc3n2ncc3C(=O)N SB01723 Cc1c(c(n(n1)c2cccc(c2)Cl)O)/N=N\c3cccc(c3)C(F)(F)F SEW04008 c1ccc(cc1)C2C(=O)C(C(=O)C2=O)c3ccccc3 SB01688 c1ccc(cc1)C(=O)Nc2cccc(c2Cl)Cl SB01690 CCOC(=O)c1c(sc(n1)c2ccccc2)C(=O)C SPB04592 c1ccc(cc1)S(=O)(=O)C(C#N)/N=N/c2ccc3c(c2)COCO3 SEW03674 Cc1c(c(on1)C)C(=O)NCc2ccc(s2)SC SEW03649 c1cc(ccc1S(=O)(=O)Cc2nc(no2)c3ccsc3)Cl SEW03687 c1cc(ccc1C(=O)O/N=C(/CS(=O)(=O)c2ccc(cc2)Cl)\N)C(F)(F)F SPB01705 CC(C)(C)c1c(cno1)C(=O)Oc2ccc(cc2)[N+](=O)[O-] SEW04621 C/C(=N\OC(=O)C(C)(C)C)/c1ccc2cc(ccc2c1)OC SEW04530 c1ccc(cc1)CC(C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 SB00998 Cc1ccc(cc1)/C=N/NC(=O)Cc2ccc(c(c2)OC)OC S09960 COc1ccc(cc1OC)Cc2nnc(n2c3ccc(cc3)Cl)S S09965 Cc1cccc(c1OC(=O)C)C(=O)O SB01734 Cc1ccc(cc1)S(=O)(=O)ONCCN SB01735 c1ccc(cc1)SC(=O)c2ccc(cc2)C(F)(F)F SPB01694 Cc1c(c(n(n1)c2ccccc2)C)C(=O)NNC(=O)C(F)(F)F SEW04229 c1c(csc1/C=N/O)Br SEW04231 c1cc(ccc1S(=O)(=O)C/C(=N/OC(=O)c2cc(cc(c2)Cl)Cl)/N)Cl SPB01706 CC(C)(C)C(=O)N1CCCC1C(=O)O SEW04242 c1cc(ccc1NS(=O)(=O)c2ccc(c(c2)Cl)Cl)n3c(cc(n3)C(F)(F)F)C(F)(F)F SEW04240 Cc1c(sc(c1C(=O)c2ccc(cc2)Cl)N)C SPB01708 Cc1c(sc(c1C(=O)c2ccc(cc2)Cl)NC(=O)C)C SPB01709 c1cc(c(cc1C(=O)c2ccc(c(c2)Cl)F)Cl)F SEW04253 CC(C)(C)C(=O)O/N=C(/c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)OC)\N SPB01646 c1ccn(c1)c2cccc(c2)c3nc(on3)c4ccc(cc4)Cl SPB01686 c1ccc(c(c1)OCc2nnc(o2)c3ccc(cc3)C(F)(F)F)Cl SPB01593 c1cc(ccc1CCNc2n[nH]c(=S)s2)Cl S09769 COc1ccc(cc1)c2cc(c3ccccc3n2)C(=O)Nc4ccc(cc4Cl)I S09780 c1cc(c(c(c1)Cl)CSC(=S)N2CCN(CC2)C(=S)SCc3c(cccc3Cl)F)F SEW04578 COc1cc\2c(cc1OC)NC(=O)/C2=C\c3ccc(cc3)C(F)(F)F SEW04628 c1cc(ccc1S(=O)(=O)Cc2cc(cc(c2)F)F)Cl SEW04751 CC(C)(C)c1c(cno1)C(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N SEW04631 CC(C)(C)c1c(cno1)C(=O)O/N=C(/c2cccc(c2)Cl)\N SEW04632 c1cc(ccc1SCc2nnn(n2)CC(=O)NN)Cl SPB01678 C1CC1CN2CN(C(=S)SC2)CC3CC3 S10436 c1ccc2c(c1)cccc2NC(=O)CSCC(=O)O S10442 c1ccc2c(c1)cccc2N3C(=O)CSCC3=O S10443 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)N3C(=O)C=CC3=O)C SEW04188 COc1ccc(cc1OC)Cc2nnc(n2c3cccc(c3)C(F)(F)F)S S09990 Cc1ccc2c(c1)C(=O)OC3(N2C(=O)C4C3C5CC4C=C5)O S10556 CCOC(=O)c1cc(on1)c2csc(n2)Nc3ccc(cc3)Cl SPB04511 c1cc2c(cc1[N+](=O)[O-])c(n[nH]2)N SEW04668 c1cc(ccc1NC(=O)Cc2cc(cc(c2)F)F)Cl SEW04672 c1ccnc(c1)NC(=O)Cc2cc(cc(c2)F)F SEW04674 c1cc(c(nc1)Oc2ccc(cc2)c3nnco3)[N+](=O)[O-] SEW04601 c1cc(ccc1CSc2c(cc(cn2)C(F)(F)F)C(F)(F)F)C(F)(F)F SPB04666 c1cc(cc(c1)C(F)(F)F)CSc2c(cc(cn2)C(F)(F)F)C(F)(F)F SPB04667 CC(C)(C)c1c(cno1)C(=O)Nc2ccc(cc2)Cl SEW04616 CC(C)(C)c1c(cno1)C(=O)N2CCOCC2 SEW04619 CCOC(=O)c1nc(no1)Cc2ccc(cc2)[N+](=O)[O-] SPB01578 Cc1ccc(cc1C)Nc2nnc(o2)c3ccccc3N S10064 c1cc(ccc1C(=O)Sc2ccc(cc2)Cl)C(F)(F)F SPB01695 Cc1ccc(cc1)SC(=O)c2ccc(cc2)C(F)(F)F SPB01696 C/C(=N\OC(=O)Nc1ccc(cc1)OC(F)(F)F)/c2ccc3cc(ccc3c2)OC SEW04532 Cc1c(c(=O)n(c(n1)SCc2ccc(cc2)C(F)(F)F)C)Oc3cccc(c3)C(F)(F)F SPB04453 CCOC(=O)CSc1nnc(n1c2ccccc2)O SPB01539 Cc1c(c([nH]n1)c2c(nns2)C)C(=O)OC SPB01542 c1cc(ccc1n2c(cc(n2)C(F)(F)F)C(F)(F)F)N3C(=O)CSCC3=O SEW04529 CCOC(=O)c1nc(no1)COc2ccccc2Cl SPB01577 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)c3nnco3 SEW04608 c1ccc(cc1)c2c(nnc(n2)N)c3ccccc3 SB01743 c1ccc(c(c1)c2nnc(o2)COc3ccccc3Cl)Cl SPB01590 COc1c(c(cc(c1)/C=C\2/C(=O)/C(=C/c3cc(c(c(c3)OC)OC)OC)/COC2)OC)OC SEW04598 CCOC(=O)c1cc(on1)c2csc(n2)COc3ccccc3Cl SPB04504 COC(=O)c1c(c(c(s1)C(F)(F)F)c2ccccc2)S(=O)(=O)c3ccc(cc3)C(F)(F)F SEW03507 c1cc(ccc1C(=O)Nc2ccc(cc2Br)OC(F)(F)F)Cl SEW04115 Cc1c(sc(n1)c2ccccc2)C(=O)N/N=C/c3cc4ccccc4o3 SEW04116 COc1ccccc1CC/N=C/c2ccnc(n2)SCc3ccc(cc3Cl)Cl SPB04479 CCOC(CC(=O)NNC(=O)Nc1ccc(cc1)Cl)OCC SPB04482 CCOC(=O)/C(=C/c1ccc(cc1)C#N)/C#N S10003 COC(=O)/C(=C/c1ccc(cc1)C#N)/C#N S10004 C/C(=C\c1ccc(cc1)C#N)/[N+](=O)[O-] S10006 CCOC(=O)c1c(sc(n1)c2ccccc2)c3ccnn3C(=O)Nc4ccc(cc4)Cl SPB04633 c1ccc(c(c1)C(=O)NN)[N+](=O)[O-] S10034 CCOC(=O)c1cc(on1)c2csc(n2)Nc3c(cc(cc3C)C)C SPB04505 CCOC(=O)c1cc(on1)c2ccnn2S(=O)(=O)c3cccc(c3)C(F)(F)F SPB04641 c1cc(ccc1S(=O)(=O)Cc2ccc(cc2Cl)NC(=O)C(Cl)(Cl)Cl)Cl SPB01601 c1ccc(cc1)CN(Cc2cccs2)C(=O)CSCC(=O)O SEW03514 CCOC(=O)c1c(sc(n1)c2ccccc2)c3ccnn3C(=O)Nc4ccccc4 SPB04635 CN(C)/C=C/1\C(=O)NC(=N1)SCC#C S10198 c1ccc(cc1)C(=O)Nc2ccc(cc2Cl)Cl SB01689 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCSCC2 S10113 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccc3cc(ccc3c2)OC SEW04534 COc1cc(cc(c1OC)OC)/C=C/C2=NNC(=O)CC2 SEW04539 c1cc(cc(c1)Cl)/C=C\2/C(=O)NC(=S)N2 S10202 c1ccc(c(c1)C(=O)O/N=C(\c2ncc(s2)[N+](=O)[O-])/N)Cl SPB01634 CCOC(=O)c1cc(on1)c2csc(n2)N/N=C/c3ccccc3Cl SPB04515 CC(C)(C)c1[nH]c(nn1)Sc2ncc(s2)[N+](=O)[O-] SPB01621 c1c(sc(n1)/C(=N/O)/N)[N+](=O)[O-] SPB01632 COC(=O)C(=NNc1cc(ccc1OCC(F)(F)F)C(F)(F)F)C(=O)OC SEW04462 CCOC(=O)c1cc(on1)c2csc(n2)c3ccc(cc3)Cl SPB04495 Cc1cc(no1)NC(=O)CC(CC(=O)O)c2cc(c(c(c2)OC)OC)OC S10221 c1ccc(c(c1)C2C(=O)c3ccccc3C2=O)F S10129 Cc1cc(no1)N2C(=O)CC(CC2=O)c3cc(c(c(c3)OC)OC)OC S10222 CSc1ccc(s1)/C=N/c2ccc(cc2Cl)Cl SEW03616 Cc1ccc(cc1)/C=N/C(=C(/C#N)\N)/C#N S10154 c1cc(c(c(c1)F)C(=O)O)F SB01105 c1cc(ccc1C(F)(F)F)n2cnnc2S SPB01531 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)NC(=S)N3CCCCC3)Cl SPB01662 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)NC(=S)NN3CCOCC3)Cl SPB01664 c1ccc(cc1)SC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl SPB01668 c1ccn2c(c1)nc3c2cc(cc3[N+](=O)[O-])C(F)(F)F SEW04114 c1cc(ccc1CNS(=O)(=O)c2cc(c(s2)Br)Br)C(F)(F)F SEW03591 c1ccc2c(c1)CC(NC2)C(=O)O SB01676 c1cc(ccc1/C=N/C(=C(/C#N)\N)/C#N)C#N S10150 CCOC(=O)c1cc(on1)c2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl SPB04501 CCOC(=O)c1cc(on1)c2csc(n2)CS(=O)(=O)c3ccccn3 SPB04502 C/C(=N\NC(=O)N)/c1cccs1 S10160 c1ccc2c(c1)C(OC2=O)CC(=O)c3ccccn3 S10157 C/C(=N\NC(=O)N)/c1ccccn1 S10163 C/C(=N\NC(=O)N)/c1ccccc1O S10164 CCOC(=O)c1cc(on1)c2csc(n2)Nc3ccccc3 SPB04509 Cc1c(cn(n1)C(=O)c2ccc(cc2)Cl)c3ccc(cc3)OC SEW04108 Cc1nc(cs1)c2nc(cc(n2)N3CCCCC3)COC SPB04588 Cc1c(cn(n1)C(=O)c2cccs2)c3ccc(cc3)OC SEW04109 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)[N+](=O)[O-])C SEW04152 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)C(F)(F)F)C SEW04157 Cc1cccc(c1/C=N/NC(=O)Cc2csc(n2)c3ccccc3)Cl SEW04119 c1cc(c(cc1F)F)CNS(=O)(=O)c2cc(c(s2)Br)Br SEW03593 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2OC(F)(F)F)Cl SEW03600 COC(=O)/C(=C/c1ccc(s1)SC)/C#N SEW03575 c1ccc(cc1)c2nc(cs2)C(=O)NN SEW04122 C/C=C(\C)/C(=O)NNC(=O)c1c(nc(s1)c2ccccc2)C SEW04125 c1cc(oc1)C(=O)Nc2ccc(cc2OC(F)(F)F)Cl SEW03602 c1ccc(cc1)/C(=C(\C(F)(F)F)/Oc2ccccc2)/C#N SEW03609 c1c(c(ncn1)N)/C(=N/O)/N SEW03510 CN(C)/C=C/C(=O)c1cccnc1 SEW04052 C1(C(C(C(C(C1C(=O)O)C(=O)O)C(=O)O)C(=O)O)C(=O)O)C(=O)O SB01658 CN1CCC=C(C1)C(=O)OC.Br SB01660 c1ccc(c(c1)NC(=O)C2C3CC(C2C(=O)O)C=C3)Oc4ccc(cc4Cl)Cl S10400 Cc1cc(no1)N2C(SCC2=O)c3cccnc3 S10235 c1ccc(cc1)COC(=O)C(c2ccccc2)C(=O)O SB01143 CC(C)c1ccc(cc1)n2c(nnc2S)Cc3ccc(c(c3)OC)OC S09989 COc1ccc(cc1OC)Cc2nnc(n2c3cccc(c3)C(F)(F)F)SCC#C S09995 Cc1cc(c(o1)C)C(=O)NCc2ccco2 SEW04545 Cc1c(c(n(n1)c2ccccc2)C)C(=O)Nc3cccc(c3)C(F)(F)F SEW04193 COC(=O)/C(=C/c1cccc(c1)Br)/C#N S10275 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCCC2 SEW04451 c1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)C(=S)NC(=O)c3ccccc3 SEW04457 c1ccc(cc1)S(=O)(=O)/C(=N/Nc2cc(ccc2OCC(F)(F)F)C(F)(F)F)/C#N SEW04460 c1ccc(cc1)C(C[N+](=O)[O-])Sc2ccccc2N S09921 c1nc(no1)CSC(=S)N2CCSCC2 SEW04571 COc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C#N SPB01642 CC(C)(C)C(=O)Nc1cccc(c1C(=O)O)C(F)(F)F SEW03615 c1cc(ccc1COc2ccc(cc2)[N+](=O)[O-])C(F)(F)F SPB01836 CCn1c(cc(n1)C)C(=O)O SPB01840 c1cc(c(cc1Cl)Cl)CCC(=O)O SEW04678 c1ccc(c(c1)N)SCc2cc(cc3c2OCOC3)[N+](=O)[O-] SEW03617 CCOC(=O)Cn1nc(nn1)CSc2ccc(cc2)Cl SPB01677 CCOC(=O)c1cc(on1)c2csc(n2)CS(=O)(=O)C SPB04560 c1ccc(c(c1)c2cc(c3c(cc(cc3n2)C(F)(F)F)C(F)(F)F)C(=O)O)Br S10285 c1cc(c(cc1Cl)Cl)OCc2cc(cc3c2OCOC3)[N+](=O)[O-] SEW03625 CC\1=NN(C(=O)/C1=C\c2ccc(s2)SC)C SEW03626 c1cc(ccc1CC(=O)O)[N+](=O)[O-] SB00940 Cc1c(c(n(n1)c2cccc(c2)Cl)O)N=Nc3ccc(cc3)C(C)(C)C SEW04007 CSc1ccc(s1)C(=O)NC(=O)Nc2cccc(c2)C(F)(F)F SEW03636 CSc1ccc(s1)C(=O)Nc2ccc(cc2)Cl SEW03641 c1cc(ccc1C(=O)OCCSCc2cc(cc3c2OCOC3)[N+](=O)[O-])Cl SEW03620 c1c(cc(cc1Cl)Cl)NC(=O)CSc2c(cc(cn2)C(F)(F)F)C(F)(F)F SPB04533 c1ccc(cc1)NC(=O)CSc2c(cc(cn2)C(F)(F)F)C(F)(F)F SPB04534 Cc1ccc(cc1)c2csc(n2)c3cc(on3)C SPB04536 c1ccc(c(c1)NC(=O)c2cccs2)SCc3cc(cc4c3OCOC4)[N+](=O)[O-] SEW03623 CC(C)(C)c1nc2cccc(c2c(n1)c3ccc(cc3)C(F)(F)F)C(F)(F)F SEW03627 Cc1cc(no1)c2nc(cs2)c3ccc(cc3)Cl SPB04537 CCOC(=O)c1cc(on1)c2csc(n2)COc3cccc(c3)Cl SPB04541 COc1cc(cc(c1OC)OC)CCC(=O)NN SEW04105 CCOC(=O)c1c(nn(c1C)c2c(cccn2)[N+](=O)[O-])C SEW04520 c1cc(ncc1C(F)(F)F)N2CCNCC2 SEW04033 c1c(cnc(c1Cl)N2CCNCC2)C(F)(F)F SEW04036 COc1ccc(cc1OC)CC(=O)NNC(=S)Nc2cccc(c2)SC S09987 Cc1c(c(n(n1)c2ccccc2)C)C(=O)NNC(=O)c3ccc(cc3)Cl SEW04228 COc1cc2c(cc1OC)NC(=O)C2 SEW04570 Cn1cnnc1SCc2nc(no2)c3ccsc3 SEW03694 c1cc(cc(c1)C(F)(F)F)c2ccnc3n2ncc3C(=O)N SB01706 C[C@H](CCCC(C)C)[C@H]1CC(=O)C2=C3CC[C@H]4C[C@H](CC[C@@]4(C3CC[C@]12C)C)O SB01709 c1ccc(cc1)c2cnc(o2)c3ccc(cc3)c4ncc(o4)c5ccccc5 SB01212 C[C@H](CCCC(C)C)[C@H]1CC=C2[C@@]1(CC[C@H]3C2=CCC4[C@@]3(CC[C@@H](C4)OC(=O)c5ccccc5)C)C SB01710 Cc1c(c(n(n1)c2ccccc2)C)C(=O)Oc3ccc(cc3Cl)Cl SEW04195 Cc1c(snn1)C(=O)NCCNC(=O)c2c(nns2)C SEW04548 C[C@H](CCCC(C)C)[C@H]1CC[C@@H]2[C@@]1(CC[C@H]3C2=CC=C4[C@@]3(CC[C@H](C4)OC(=O)c5ccccc5)C)C SB01708 CC(C)(C(=O)O)Oc1ccc(cc1)Cl SB01597 c1cc(ccc1CO/N=C(/c2ccc(cc2)Cl)\C3CC3)[N+](=O)[O-] SB01643 c1cc(c(cc1Cl)Cl)CSc2c(cc(cn2)C(F)(F)F)C(F)(F)F SPB04669 Cc1cc(no1)c2nc(cs2)/C(=N/OC(=O)c3ccccc3)/C SPB04714 c1cc(ccc1SCc2csc(n2)c3ccno3)Cl SPB04676 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)N3C(=O)c4ccccc4C3=O)C SEW04189 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)/C=C\C(=O)O)C SEW04179 Cc1c(c(n(n1)C)C(=O)Nc2ccc(c(c2)Cl)F)[N+](=O)[O-] SPB01654 c1ccc(c(c1)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)C(F)(F)F)C(=O)O SEW04521 c1cc(ccc1NC(=O)/C=C/C(=O)O)n2c(cc(n2)C(F)(F)F)C(F)(F)F SEW04522 CCOC(=O)c1cc(on1)c2ccnn2C(=O)c3ccccc3 SPB04637 CCOC(=O)c1csc(n1)NC=C(C(=O)OCC)C(=O)OCC SEW03709 Cc1ccc(cc1)Sc2ccc(cc2)C(=O)c3ccccc3 SB01142 CCOC(=O)c1c(sc(n1)C)c2ccnn2C(=O)c3ccc(cc3)OC SPB04653 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)OC)C SEW04173 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NS(=O)(=O)c3c(noc3C)C)C SEW04176 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)C(F)(F)F SEW04224 c1ccc2c(c1)/C(=C/c3cc(cc(c3)F)F)/C(=O)N2 SEW04698 Cc1cc(ccc1NC(=C2C(=O)c3ccccc3C2=O)C#N)Cl S10175 Cc1c2c(c(nn(c2=O)c3ccc(cc3)Cl)C)on1 SPB04673 CCCS(=O)(=O)Cc1nnc(o1)c2ccc(cc2)C(C)(C)C SPB01844 c1cc(c(nc1)n2c(cc(n2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] SEW04528 c1cc(ccc1CS(=O)(=O)C2CS(=O)(=O)CC2O)Cl SEW03522 CCN(CC)c1ccc(cc1)Cc2ccc(cc2)N(CC)CC SB01693 Cc1c2c(c(=O)n(n1)c3c(cccc3Cl)Cl)nc(s2)C SPB04709 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)c3cccs3)C SEW04165 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)C(C)(C)C)C SEW04167 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=S)NC(=O)c3ccccc3)C SEW04818 Cc1nc(cs1)c2cc(no2)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB04739 c1cc(ccc1c2csc(n2)c3ccsc3)F SEW03734 CCOC(=O)c1csc(n1)c2c(ccs2)Br SEW03546 c1ccnc(c1)SCc2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl SPB01850 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)/N=C/c3ccc[nH]3 SEW04687 C1COCCN1Cc2c(snn2)Cl SEW03559 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)NNc2cnc3ccccc3n2 SEW03562 CC(C)(C)c1c(cno1)C(=O)O/N=C(/c2ccccn2)\N SEW04630 c1ccc(cc1)C(=O)c2ccc[nH]2 SEW04633 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)N3C(=O)CCC3=O)C SEW04205 c1ccc2c(c1)C(=O)C(=Cc3ccc(o3)c4ccc(cc4[N+](=O)[O-])C(F)(F)F)C2=O SEW04209 c1cc(ccc1COc2cc(cc(c2)Cl)Cl)C(F)(F)F SPB01835 COC(Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)c3ccc(cc3)Cl)OC SPB04886 CCOC(=O)c1c(noc1c2csc(n2)Nc3c(cc(cc3C)C)C)C SPB04698 c1cc2c(cc1OS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)c(co2)[N+](=O)[O-] SEW03547 CCOC(=O)c1csc(n1)c2c(nns2)C SEW03551 Cc1c(c(n(n1)C)C(=O)NNC(=O)c2cc(cc(c2)Cl)Cl)[N+](=O)[O-] SPB01720 Cc1c(c(n(n1)C)C(=O)N)[N+](=O)[O-] SPB01723 Cc1ccc(cc1)SC(=O)c2c(c(nn2C)C)[N+](=O)[O-] SPB01734 CC(C)(C)S(=O)(=O)CC(=S)N SPB04688 Cc1c(c(n(n1)c2ccccc2)C)C(=O)Oc3ccc(cc3)OC SEW04191 Cc1ccc(cc1)OC(=O)c2c(nn(c2C)c3ccccc3)C SEW04194 c1cc(ccc1CC(=O)O)OC(F)(F)F SB01807 CCOC(=O)c1cc(on1)/C(=N/Nc2ccccc2C(F)(F)F)/C SPB04606 c1cc(ccc1C(=O)NNC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F)Cl SPB04626 Cc1ccc(c(c1)Br)NC(=C2C(=O)c3ccccc3C2=O)C#N S10242 Cc1ccc(c(c1)Cl)NC(=C2C(=O)c3ccccc3C2=O)C#N S10243 c1ccc2c(c1)C(=O)C(=C(C#N)Nc3cccnc3)C2=O S10244 COC(Cn1c(nnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)c3ccc(cc3)Cl)OC SPB04887 c1cc(ccc1C(=O)Oc2ccc3c(c2)c(co3)[N+](=O)[O-])Cl SEW03542 c1ccc2c(c1)/C(=C/c3ccc(s3)c4cccs4)/C(=O)N2 SEW04666 Cc1c2c(c(=O)n(n1)c3ccc(cc3F)F)nc(s2)C SPB04718 Cc1c2c(c(=O)n(n1)c3ccc(cc3F)F)nc(s2)c4ccccc4 SPB04719 C/C(=N\NC(=O)N)/Cc1ccc(c(c1)OC)OC S10165 c1cscc1/C=C(\c2cc(cc(c2)F)F)/C(=O)O SEW04711 c1ccn(c1)c2cccnc2NNC(=O)Nc3ccc(cc3)OC(F)(F)F SEW04299 c1ccc(cc1)S(=O)(=O)Cc2ccc(cc2)F SEW03671 c1c(cc(cc1F)F)/C=N/NC(=O)N SEW04696 c1cc(c(cc1Cl)Cl)OCc2c(snn2)Cl SEW03524 Cc1cccc(c1Nc2nnc(o2)Cc3ccc(c(c3)OC)OC)C S10090 c1ccc2c(c1)/C(=C/c3ccc(cc3Cl)C(F)(F)F)/C(=O)N2 SEW04667 Cc1c(c(n(n1)C)C(=O)NNC(=O)COc2ccc(cc2Cl)Cl)[N+](=O)[O-] SPB01719 CCOC(=O)/C(=C(/Nc1ccc(cc1)Cl)\N=C(\c2ccc(cc2)C(F)(F)F)/N)/C#N SPB01770 Cc1c2c(c(=O)n(n1)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)nc(s2)C SPB04710 COc1cc(c(cc1OC)[N+](=O)[O-])C(=O)OC SB01833 CCCS(=O)(=O)Cc1nnc(o1)c2cc(cc(c2)Cl)Cl SPB01843 C/C(=N\OC(=O)c1cccc(c1)C(F)(F)F)/c2csc(n2)c3ccno3 SPB04694 Cc1cc(no1)c2nc(c(s2)C(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F)C SPB04748 c1ccc(c(c1)C2C(=O)c3ccccc3C2=O)Br S10277 c1ccc2c(c1)cccc2CC(=O)Nc3ccc(cc3)I S09993 Cc1nc(no1)c2ccc(cc2)c3nc(on3)C SEW04235 c1cc(cc(c1)Cl)N(CCO)CCO SB01823 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(o2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)/C#N SEW04210 CCCS(=O)(=O)Cc1nnc(o1)c2cccs2 SPB01845 COC(Cn1c(nnc1SC)c2ccc(cc2)Cl)OC SPB04890 c1cc(ccc1S(=O)(=O)Cc2nc(on2)c3cc(cc(c3)Cl)Cl)Cl SPB01865 CC(=O)OCCSc1ccc(cc1[N+](=O)[O-])C#N SEW04252 c1cc(sc1)/C=C/2\C(=O)NC(=S)N2 S10177 CC(C)(C)C(=O)NNC(=O)c1cc2c(s1)cc(cn2)C(F)(F)F SPB04630 CC(=O)Nc1ccc(cc1)OC(=O)c2cnoc2C(C)(C)C SEW04623 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)C2CS(=O)(=O)CC2O SEW03549 Cc1ccc2c(c1)[nH]c(=S)o2 S10307 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)N3C(=O)c4ccccc4C3=O SEW04795 CCn1c(c(c(n1)C)NS(=O)(=O)c2ccc(c(c2)Cl)F)C(=O)OC SPB01863 c1cc(ccc1c2nc(no2)CS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F SPB01864 c1ccc(c(c1)C(=O)NC(=O)NN2CCCCC2)C(F)(F)F SPB01791 c1ccc(c(c1)C(=O)NC(=O)NN2CCOCC2)C(F)(F)F SPB01792 COC(=O)c1ccc(o1)[N+](=O)[O-] SB01301 CCOC(=O)c1c(nc(s1)CS(=O)(=O)c2ccc(cc2)Cl)C SPB01750 c1cnccc1c2ncc(c(n2)N)C#N SEW03610 Cc1c(sc(n1)C)c2nnc(n2c3ccccc3C(F)(F)F)S SPB01701 COc1ccc(cc1OC)CC(=O)N/N=C/c2cccs2 S09961 Cc1nc(cs1)c2cc(no2)c3nc(no3)c4ccc(cc4)Cl SPB04737 COC(=O)c1ccc(n1c2ccc(cc2)F)/C=N/NC(=S)N SEW04816 CC(C)(C)C(=O)Nc1c(cccc1SC)OC(F)(F)F SEW03581 c1ccc(cc1)/C(=C(/C(F)(F)F)\Oc2ccc(cc2)C#N)/C#N SEW03587 Cc1ccc(cc1)C(=O)OCCSc2ccc(cc2[N+](=O)[O-])C#N SEW04250 CC(C)(C)c1ccc(cc1)C(=O)NNc2c(cccn2)n3cccc3 SEW04294 c1ccn(c1)c2cccnc2NNC(=O)c3ccco3 SEW04297 c1ccc2c(c1)NC(=O)CC(S2)c3cc(cc(c3)Cl)Cl SEW04267 Cc1c(c(n(n1)C)O)/N=N\c2ccc3c(c2)COCO3 SEW03673 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC(Cc3ccccc3)C(F)(F)F SEW03676 CC(C)(C)/C(=N\OC(=O)C(C)(C)C)/c1cccs1 SEW04154 c1cc(ccc1C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)C(F)(F)F)Cl SEW04226 c1cc(ccc1C(=O)OCCSc2ccc(cc2[N+](=O)[O-])C#N)Cl SEW04243 c1ccn(c1)c2cccnc2NNC(=O)Nc3ccc(cc3)Cl SEW04298 Cc1cc(c(nc1)SC)C#N SPB01722 c1cc(ccc1S(=O)(=O)CC(=S)N)Cl SPB01724 c1cc(ccc1c2nc(on2)Cc3cc(cc(c3)F)F)C(F)(F)F SEW04730 Cn1c(nnc1SCc2csc(n2)COc3ccc(cc3)OC)C(F)(F)F SPB01817 c1cc(ccc1NC(=O)O/N=C(/c2ncc(s2)[N+](=O)[O-])\N)Cl SPB01640 Cc1cc(no1)/N=C/c2ccccc2O S10227 Cc1cc(no1)N2C(=O)CCC2=O S10229 Cc1ccc(c(c1)n2c(nnc2S)Cc3ccc(c(c3)OC)OC)C S09991 c1cc(sc1)C(=O)N2CCCC2C(=O)O SEW04281 C=CCNC(=S)NNc1c(cccn1)n2cccc2 SEW04303 c1ccn(c1)c2cccnc2NNC(=O)c3ccc(cc3)Cl SEW04293 Cc1c(c(n(n1)C)C(=O)OC)[N+](=O)[O-] SPB01715 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)SCc3cc(cc4c3OCOC4)[N+](=O)[O-] SEW03621 Cc1nc(cs1)c2cc(no2)c3nc(no3)c4ccc(cc4)C(F)(F)F SPB04738 Cc1c2c(c(=O)n(n1)c3cccc(c3)C(F)(F)F)nc(s2)C SPB04741 Cc1c(c(c(c(c1C)C)S(=O)(=O)NNC(=O)c2c(nc(s2)c3ccccc3)C)C)C SEW04131 Cc1cc(no1)N2C(=O)C3C4CC(C3C2=O)C=C4 S10397 c1ccc(cc1)C/C(=N/OC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C(F)(F)F SEW03736 COC(Cn1c(nnc1SCC(=O)Nc2ccccc2)c3ccccc3)OC SPB04866 COC(Cn1c(nnc1SCc2ccc(cc2)Cl)c3ccc(cc3)Cl)OC SPB04871 c1ccc(cc1)CSC[C@H](C(=O)Nc2ccc(cc2)[N+](=O)[O-])N SB01229 c1ccc2c(c1)c(c[nH]2)C[C@@H](C(=O)O)N SB01750 CCCS(=O)(=O)/C(=C/c1ccc(s1)c2ccc(cc2)OC)/C#N SEW04648 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3ccco3 SEW04316 CC(=O)Cc1nc(sn1)NC SEW04134 Cc1c(c(on1)C)C(=O)O/N=C(/c2cccs2)\C(C)(C)C SEW04144 c1c(ccc(c1)Cl)/C=C\2/C(=O)/C(=C/c3ccc(cc3)Cl)/COC2 SEW04553 c1ccc(cc1)CC(C(F)(F)F)OC(=O)Nc2ccc(cc2)OC(F)(F)F SEW03729 CSc1ccc(s1)C(=O)O SEW03638 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2CC(OC)OC)c3ccc(cc3)Cl SPB04888 Cc1cc(no1)c2nc(c(s2)C(=O)NNS(=O)(=O)c3ccccc3)C SPB04727 Cc1cc(no1)c2nc(c(s2)C(=O)NNC(=O)NC(C)C)C SPB04733 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCC(CC3)C(=O)c4ccccc4 SEW04323 c1ccc2c(c1)NC(=O)CC(S2)c3ccc(cc3)OC(F)(F)F SEW04326 c1cc(c(nc1)N/N=C/c2ccc(cc2)O)[N+](=O)[O-] SEW04732 Cc1c(sc(n1)C)C(=O)NN SPB01606 Cc1c(c(n(n1)c2ccccc2)C)C(=O)Oc3ccccc3 SEW04196 C/C(=N\O)/c1csc(n1)c2ccno2 SPB04567 Cc1ccc(cc1Cl)n2c(nnc2S)Cc3c(oc4c3cccc4)C S10349 Cc1cc(no1)c2nc(cs2)C(=O)Nc3cc(on3)C SPB04724 c1ccn(c1)c2cccnc2NNC(=S)Nc3ccc(cc3)Cl SEW04301 c1cc(c(cc1C#N)[N+](=O)[O-])SCCOC(=O)Nc2cc(cc(c2)Cl)Cl SEW04311 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F SEW04314 c1cc(ccc1c2nnco2)OC/C(=N/OC(=O)c3ccc(cc3)Cl)/N SEW04634 c1cc(c(cc1Cl)Cl)NC(=O)CSc2c(cc(cn2)C(F)(F)F)C(F)(F)F SPB04661 Cc1c(c(n(n1)C)C(=O)Sc2ccccc2)[N+](=O)[O-] SPB01731 CC(CCC(=O)NCC(=O)[O-])C1CCC2C1(C(CC3C2C(CC4C3(CCC(C4)O)C)O)O)C.[Na+] SB01793 C[C@H](CCC(=O)O)[C@H]1CC[C@@H]2[C@@]1(CC[C@H]3[C@H]2C[C@H](C4=C[C@H](CC[C@]34C)O)O)C SB01794 COc1ccc(c(c1)NC(=O)c2ccc(s2)SC)OC SEW03655 CSc1ccc(s1)C(=O)NC(=O)Nc2ccc(cc2)Cl SEW03633 CCOC(=O)[C@H](Cc1ccccc1)N.Cl SB01138 c1ccc2c(c1)C(OC2=O)Nc3ccc(cc3Cl)C(F)(F)F SEW04665 c1c(cc(cc1Cl)Cl)NC(=O)COCC(=O)O S10462 c1cc(c(cc1C(=O)O)C(=O)O)C(=O)O SB01864 c1cc(cnc1)/C=N/Nc2c(cccn2)[N+](=O)[O-] SEW04726 c1cc(cc(c1)C(F)(F)F)/C=N/Nc2c(cccn2)[N+](=O)[O-] SEW04727 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)c3c(nns3)C)C SEW04170 c1cc(ccc1N/N=C(\C#N)/S(=O)(=O)c2ccsc2)Cl SEW03703 Cc1cc(no1)NC(=O)NC(=O)c2ccc(s2)SC SEW03634 c1c(c(nc(n1)O)O)Br SB01198 c1c(cc(cc1Br)Br)C#N SEW04145 CC(C)(C)OC(=O)N[C@@H](CCCNC(=N)N[N+](=O)[O-])C(=O)O SB01865 CC(C)(C)/C(=N\OC(=O)c1ccc(cc1)Cl)/c2cccs2 SEW04163 CC(C)(C)/C(=N\OC(=O)c1ccc(cc1)OC)/c2cccs2 SEW04164 c1ccc(cc1)c2cc(on2)c3csc(n3)c4ccc(cc4)C(F)(F)F SPB04863 Cc1c2c(c(=O)n(n1)c3ccc(c(c3)Cl)F)nc(s2)C SPB04705 CCOC(=O)/C(=C/c1ccccc1Sc2ccc(cc2)Cl)/C#N SPB01869 Cc1nc(cs1)c2cc(no2)c3nc(no3)c4ccc(cc4)C(C)(C)C SPB04740 Cc1c(c(n(n1)C)CO)[N+](=O)[O-] SPB01725 c1cc(ccc1c2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl)Cl SPB01729 c1nc(c(c(n1)O)[N+](=O)[O-])O SB01255 c1nc(no1)CSC(=S)N2CCCC2 SEW04569 Cc1c(c(n(n1)c2ccccc2)C)C(=O)Nc3ccccc3 SEW04197 Cc1c(c(n(n1)c2ccccc2)C)C(=O)Nc3ccc4c(c3)OCO4 SEW04198 C=CC(=O)Nc1ccc(cc1)OC(F)(F)F SEW03730 c1ccc(cc1)c2cc(on2)c3csc(n3)COc4cc(cc(c4)Cl)Cl SPB04885 Cc1ccc(cc1)S(=O)(=O)Cc2ccc(cc2)C(F)(F)F SPB01830 c1cnoc1C(=O)NNC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F SPB04629 Cc1c(n2ccccc2n1)c3ccn[nH]3 SPB04648 CCOC(=O)c1cc(on1)c2ccnn2C(=O)c3ccc(cc3)C SPB04639 c1cc(ccc1CS(=O)(=O)C/C(=N/O)/N)F SPB02050 COC(=O)CCCCCCCC(=O)Nc1ccc(cc1)C(F)(F)F SEW04980 c1cc(ccc1C(F)(F)F)NN=C(C#N)C#N SEW04981 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)Cl)Cc3cccnc3)C SPB01935 COC(Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)c3ccccc3)OC SPB04875 COC(Cn1c(nnc1SCC(=O)Nc2ccccc2)c3ccc(cc3)Cl)OC SPB04876 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl SPB04895 CS(=O)(=O)CC(=S)N SPB04681 Cc1ccc(cc1)n2c(=O)c3c(noc3c(n2)C)C SPB04679 Cc1c(c(n(n1)c2ccccc2)C)C(=O)O/N=C(/c3ccccc3)\N SEW04202 CCC(=O)c1ccc(cc1)c2ccccc2F SB01820 Cc1ccc(cc1)C(=O)NC(=N)c2cccs2 SPB07001 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F SEW04313 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3cccs3 SEW04315 Cc1c(c(on1)C)C(=O)N2CCC(CC2)C(=O)c3ccccc3 SEW04317 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3c(cccn3)n4cccc4 SEW04300 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3c(cccc3F)F SEW04322 CNC(=S)NNc1c(cccn1)n2cccc2 SEW04302 Cc1cc(cc(n1)C)c2ccsc2 SEW04304 Cc1ccc(cc1)NC(=S)NC(=N)C(C)C SPB07021 c1ccc(cc1)C(=N)NC(=O)c2ccc(nc2)OCC(F)(F)F SPB07022 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)/N=C\c3ccccc3O)C SEW04185 c1cc(c(c(c1)Cl)/C=C\2/C(=O)NC(=S)N2)F S10181 COc1ccc(cc1)C2C(=O)c3ccccc3C2=O S10187 c1ccc(c(c1)/C=C\2/C(=O)NC(=S)N2)Cl S10192 c1ccc(cc1)C(CC(=O)c2ccccc2)CC(=O)c3cccs3 S10068 Cc1c(sc(n1)c2ccc(s2)c3cccs3)c4ccnn4C(=O)C(C)(C)C SEW04868 c1cc(c(cc1/C(=N/O)/N)[N+](=O)[O-])Oc2ccc(cc2F)F SPB01976 Cc1c(sc(n1)c2ccc(s2)c3cccs3)c4ccnn4C(=O)c5cccc(c5)C(F)(F)F SEW04870 CCc1ccc(nc1NC(=O)c2c(nns2)C)C SEW04872 COc1cc(c(cn1)c2[nH]ncn2)C(F)(F)F SPB04783 c1cc(ccc1c2csc(n2)C3(CC3)c4ccc(cc4Cl)Cl)F SEW04882 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3ccco3 SEW04887 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)/N=C/c3ccc(cc3)OC SEW04690 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc3c(c2)c(co3)[N+](=O)[O-] SEW03536 CC(C(=O)NNC(=O)c1cc(c(c(c1)OC)OC)OC)Oc2ccc(cc2Cl)Cl SEW04663 c1cc(ccc1C(=O)CSc2[nH]nc(n2)C(F)(F)F)Cl SPB01758 CSc1ccc(s1)C=C(C#N)C#N SEW03574 c1ccnc(c1)SCc2[nH]nnn2 SPB01985 C=CCn1c(nnc1Sc2ncc(s2)[N+](=O)[O-])O SPB01986 c1cc(c(c(c1)Cl)/C=N\NC(=O)Cn2nc(nn2)C3CC3)Cl SPB01765 CC(C)(C)C(=O)CSc1nnc(n1c2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl SPB05817 CCCCCn1c(nnc1Sc2ncc(s2)[N+](=O)[O-])O SPB01987 CCOC(=O)c1csc(n1)Cc2c(cccc2Cl)Cl SPB02007 c1cc(ccc1c2csc3n2c(nn3)C(F)(F)F)Cl SPB01768 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)C3C4CC(C3C(=O)O)C=C4 SEW04739 Cc1c(sc(n1)C)c2nnc(n2C)S SPB01778 c1cc(ccc1SCc2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl)Cl SPB01848 CCOC(=O)c1cc(n(n1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C SPB01740 CCOC(=O)c1c(noc1c2csc(n2)COc3cccc(c3)Cl)C SPB04695 Cc1c(c(n(n1)c2ccccc2)C)C(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N SEW04204 COc1ccc(cc1)C/N=C/c2cc(c(c(c2)OC)OC)OC SEW04958 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2cc(no2)c3ccccc3 SPB04829 c1ccc(cc1)C(=O)CSc2c(c(c3c(n2)CCCC3)c4cccs4)C#N SPB07056 c1cc(cc(c1)S(=O)(=O)NNC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F)C(F)(F)F SPB04796 CCOC(=O)c1c(sc(n1)C)c2ccnn2S(=O)(=O)c3ccccc3C(F)(F)F SPB04762 C[C@H](CCC=C(C)C)[C@H]1CC[C@@]2([C@@]1(CCC3=C2CC[C@@H]4[C@@]3(CC[C@@H](C4(C)C)O)C)C)C SB01792 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)CSCC(=O)O SEW04691 c1cc(ccc1NC(=O)C2CC2)F SEW04208 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/c3cc(cc(c3)Cl)Cl SEW04272 c1ccc2c(c1)C(OC2=O)NNc3ccc(cc3Cl)C(F)(F)F SEW04712 CCOC(=O)c1c(sc(n1)C)c2ccnn2S(=O)(=O)c3cccc(c3)Cl SPB04778 c1cc(ccc1NC(=O)Cc2cc(cc(c2)F)F)F SEW04671 Cn1cc(c(n1)C2NN=C(S2)SCC(=O)Nc3ccccc3)Cl SPB07014 CC(C)(C)c1ccc(cc1)NC(=O)CSC2=NNC(S2)c3c(cn(n3)C)Cl SPB07018 COC(CNC(=S)NNC(=O)Nc1ccccc1)OC SPB04757 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)/N=C/c3cccc(c3OC)OC SEW04776 CNC(=S)NNC(=O)c1cccn1c2ccc(cc2)F SEW04782 C=CCNC(=S)NNC(=O)c1cccn1c2ccc(cc2)F SEW04783 Cc1ccc(cc-2c(cc(c12)C=C(C#N)C#N)C)C(C)C SEW04809 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)N3C(=O)CSCC3=O SEW04718 c1ccc(c(c1)N)SC(C[N+](=O)[O-])c2ccc3c(c2)OCO3 S10379 CSc1ccc(s1)/C=N/Nc2ccc(cc2Cl)Cl SEW03577 COc1ccc(cc1)NC(=O)Cc2cc(cc(c2)F)F SEW04673 c1cc(ccc1C(=O)NNC(=O)Cc2cc(cc(c2)F)F)Cl SEW04676 c1ccn(c1)c2cccc(c2)c3nc(cs3)CC(=O)NNC(=O)c4ccc(cc4)C(F)(F)F SPB01753 Cc1cc(no1)c2nc(cs2)C(=O)NN3CCCCC3 SPB04784 CCOC(=O)c1c(nn(c1C)c2c(cccn2)N)C SEW04720 COC(=O)c1cccn1c2ccc(cc2)Cl SEW04721 c1ccc(c(c1)Nc2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl)Cl SPB04898 c1cc(c(cc1Cl)Cl)c2cc(on2)c3csc(n3)COc4cc(cc(c4)Cl)Cl SPB04900 Cc1c2c(c(=O)n(n1)c3ccccc3C(F)(F)F)nc(s2)C SPB04708 CCOC(=O)c1c(noc1c2csc(n2)COc3ccc(cc3)Cl)C SPB04712 c1cc(ccc1C(=N)NC(=O)c2ccc(nc2)OCC(F)(F)F)Cl SPB07023 CSc1ccc(s1)/C=N/NC(=O)N SEW03578 Cc1ccc(cc1)C(=O)CSc2[nH]nc(n2)C(F)(F)F SPB01759 CSc1ccc(s1)C(=O)NC(=O)NCc2cccc(c2)Cl SEW03635 CCOC(=O)/C(=C(\Nc1ccccc1Cl)/SC)/C#N SPB01772 CCC1(c2cc-3n(c(=O)c2COC1=O)Cc4c3nc5ccccc5c4)O SB01929 c1cc(sc1)C(=N)NC(=O)c2cccs2 SPB07002 Cc1ccc(cc1)c2csc3n2c(nn3)C(F)(F)F SPB01769 CCOC(=O)/C(=C(/Nc1ccc(cc1)Cl)\N=C(/c2cccc(c2)C)\N)/C#N SPB01771 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=O)NC(C)C)C SEW04762 c1ccc(c(c1)NC(=S)NC2CC3CC2C=C3)SCc4cc(cc(c4)F)F SEW04767 c1cc(ccc1CS(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F SPB01829 Cc1c(snn1)C(=O)OCc2cc(cc(c2)F)F SEW04692 c1c(c(cc2c1NCNS2(=O)=O)S(=O)(=O)N)C(F)(F)F SB01887 Cc1c(sc(n1)C)C(=O)NNC(=O)Nc2ccc(cc2)Cl SPB01782 c1cnccc1c2ccncc2 SB01188 Cc1c2c(c(=O)[nH]n1)nc(s2)c3ccccc3 SPB04699 Cc1cc(no1)c2nc(cs2)C(=O)C SPB04706 c1ccc(cc1)c2[nH]cc(n2)/C=N/c3ccccc3n4cccc4 SEW04707 c1c(cc(cc1Cl)Cl)NN=C(C#N)C#N SEW04982 COc1ccc(c(c1)OC)NC(=O)CCCCCCCC(=O)OC SEW04983 CCOC(=O)c1c(sc(n1)C)c2ccnn2S(=O)(=O)c3ccc(cc3)C SPB04754 Cc1ccc(cc1)CSc2nccc(n2)c3c(nc4n3cccc4)C SPB04842 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(F)(F)F SPB04846 c1cc(sc1)C(=O)NNC(=O)c2csc(n2)c3ccc(c(c3)Cl)Cl SPB02058 Cc1ccc(cc1)NC(=O)Nc2ccc(cc2)C SEW04985 Cn1cc(c(n1)C2NN=C(S2)SCC(=O)c3ccc(cc3)Cl)Cl SPB07010 Cc1cc(no1)c2nc(c(s2)C(=O)NNC(=O)Nc3ccc(cc3Cl)Cl)C SPB04747 CS(=O)(=O)NNC(=O)c1cc2c(s1)cc(cn2)C(F)(F)F SPB04800 CCOC(=O)c1c(noc1/C(=N/OC(=O)Nc2cccc(c2)C(F)(F)F)/C)C SPB04809 c1ccnc(c1)SC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl SPB01890 Cc1ccc(cc1)C(=O)NNC(=S)NCC(OC)OC SPB04761 c1c(cc(cc1F)F)/C=N/NC(=S)N SEW04697 COc1cc(cc(c1OC)OC)C(C[N+](=O)[O-])Sc2ccccc2N S10375 CCOC(=O)Cc1csc(n1)CS(=O)(=O)c2ccc(cc2)Cl SPB01737 c1cc(ccc1c2nnc(o2)C3CC3)C(F)(F)F SPB01743 c1cnccc1c2ncc(c(n2)N)/C(=N/O)/N SEW03629 c1cc(ccc1COC(=O)c2ccc(o2)[N+](=O)[O-])C(F)(F)F SPB01822 c1cc(ccc1OCc2nc(on2)CSc3ccc(cc3)Cl)Cl SPB01815 c1cc(ccc1COC(=O)c2cc(cc(c2)Cl)Cl)C(F)(F)F SPB01820 c1c(cc(cc1Cl)Cl)NC(=O)C2C3CC(C2C(=O)O)C=C3 S10390 c1c(cc(cc1C(F)(F)F)NN=C(C#N)C#N)C(F)(F)F SEW04978 C/C(=N\NS(=O)(=O)c1ccccc1)/c2cc(no2)c3ccccc3 SPB04824 c1cc(n(c1)c2ccc(cc2)F)C(=O)C(F)(F)F SEW04716 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(C)C SPB04847 c1cc2c(cc1I)c3cc(ccc3o2)I SEW04798 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc(cc2)F)C(F)(F)F SPB01794 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)C/C(=N/O)/N SPB01795 Cc1ccc(cc1)SCc2ccc(cc2)C(F)(F)F SPB01825 c1cnccc1c2ncc(c(n2)N)C(=S)N SEW03631 CCOC(=O)c1cc(on1)c2ccnn2C(=O)c3ccc(cc3)C(F)(F)F SPB04624 Cc1cc(no1)c2nc(c(s2)C(=O)NNS(=O)(=O)c3ccc(cc3Cl)Cl)C SPB04749 c1ccc(cc1)NC2CCCCC2.Cl SB01939 c1ccc(c(c1)NN=C(C#N)C#N)OC(F)(F)F SEW04979 c1cc(ccc1NC(=S)N/N=C/c2c(nc3n2ccs3)Sc4ccc(cc4)Cl)Cl SPB05868 c1cc(ccc1C2SCCS2)OC/C(=N/O)/N SPB01882 CCn1c(cc(n1)C)/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/N SPB01884 CC(C)(C)c1ccc(cc1)C(=O)OCc2ccc(cc2)C(F)(F)F SPB01823 c1cc(ccc1CSc2ccc(cc2)Cl)C(F)(F)F SPB01824 c1cc(ncc1C(F)(F)F)c2nc(cs2)C(=O)NN SPB05836 c1cc(ccc1NC(=O)NNC(=O)c2csc(n2)c3ccc(cn3)C(F)(F)F)Cl SPB05837 c1cc(n(c1)c2ccc(cc2)F)C(=O)NNC(=O)Nc3ccc(c(c3)Cl)Cl SEW04803 c1ccc(cc1)NC(=O)NNC(=O)c2cccn2c3ccc(cc3)F SEW04804 Cn1c(nnc1SCc2ccc(cc2)C(F)(F)F)C(F)(F)F SPB01828 c1cc(ccc1N2C(=O)C3C4CC(C3C2=O)C=C4)F S10418 COC(=O)c1c(ccs1)N SB01239 Cc1ccc(o1)/C=C(/c2cc(cc(c2)F)F)\C(=O)O SEW04657 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/COc2ccc(cc2)C3SCCS3)\N SPB01886 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl SPB04843 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)NNC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F SPB04797 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)c4cccc(c4)C(F)(F)F SPB04841 c1cc(c(cc1CO)[N+](=O)[O-])Oc2ccc(cc2Cl)Cl SPB01893 COc1ccc(cc1)c2cc(sc2c3ccc(cc3)OC)C(=O)OC SEW04824 Cc1c(n(c(c1C#N)n2cccc2)CC3CC3)C SPB01901 Cc1ccc(cc1)CSc2nnc(n2CC(OC)OC)c3ccc(cc3)Cl SPB04872 c1c(cc(cc1C(F)(F)F)NC(=O)CSCC(=O)O)C(F)(F)F S10451 c1cc(c(cc1NC(=O)CSCC(=O)O)Cl)F S10453 Cc1cc(c(=S)[nH]c1)C#N SPB01714 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=O)CCC(=O)O)C SEW04737 Cc1cc(ccc1[N+](=O)[O-])OCc2cc(cc(c2)F)F SEW04747 Cc1cc(c(s1)C)/C=C(\C#N)/S(=O)(=O)c2ccccc2 SEW04278 c1c(cc(cc1Cl)Cl)N2C(=O)C3C4CC(C3C2=O)C=C4 S10391 c1cc(ccc1C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl)Cl SPB01894 CCOC(=O)c1c(c(n(c1NC(=O)c2ccc(cc2)Cl)Cc3ccccc3)C)C SPB01927 COC(=O)C(Cc1ccc(cc1Cl)Cl)Sc2ccc(cc2)Cl SEW04826 C/C(=N\OC(=O)c1ccccc1)/c2cc(no2)c3ccccc3 SPB04830 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2cc(no2)c3ccccc3 SPB04833 CC(=O)c1ccc(cc1)OCc2cc(cc(c2)F)F SEW04749 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)/N=C\c3ccc(cc3)F)C SEW04184 c1c(cnc2c1sc(c2)C(=O)NN)C(F)(F)F SPB04625 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F SPB04627 Cc1cc(no1)NC(=O)C2C3CC(C2C(=O)O)C=C3 S10396 c1cc(ccc1Sc2c(n3ccsc3n2)/C=N/NC(=S)N)Cl SPB05869 c1cc(sc1)c2ccc(s2)c3nc(cs3)c4ccc(cc4)[N+](=O)[O-] SEW04834 Cc1cc(c(s1)C)/C=C(\C#N)/C(=O)OC SEW04279 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3ccc(cc3)Cl SEW04318 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)C(=O)c3ccccc3 SEW04319 Cc1ccc(cc-2c(cc(c12)/C=N\Nc3ccc(cc3)[N+](=O)[O-])C)C(C)C SEW04847 c1cc(cc(c1)C(F)(F)F)c2ccnc3n2ncc3/C(=N/O)/N SEW04848 CN(C)/C=N/C(=S)c1ccc(s1)c2cccs2 SEW04850 c1cc(ccc1c2csc(n2)C3(CC3)c4ccc(cc4Cl)Cl)[N+](=O)[O-] SEW04880 c1ccc(cc1)CC(C(F)(F)F)OS(=O)(=O)c2ccc(cc2)Cl SEW03705 c1ccc(cc1)CC(C(F)(F)F)OS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW03706 c1cc(ccc1SC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl)Cl SPB01889 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)Cl)Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C SPB01914 Cc1c(n(c(c1C#N)NC(=O)c2cccs2)Cc3cccs3)C SPB01919 c1cc(c(cc1COC(=O)c2cc(cc(c2)Cl)Cl)[N+](=O)[O-])Oc3cc(cc(c3)Cl)Cl SPB01956 C/C(=N\OC(=O)c1cc(cc(c1)Cl)Cl)/c2cc(no2)c3ccccc3 SPB04834 C1CC1CNC(=O)/C=C/C(=O)O S10438 c1cc(ccc1S(=O)(=O)Cc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl)Cl SPB01961 CCOC(=O)NNC(=S)Nc1ccc(cc1Cl)Cl SPB01967 CCCCCNC(=S)NNC(=O)OCC SPB01969 CCOC(=O)NNC(=S)NCC=C SPB01970 c1cc(ccc1c2nnc(o2)c3ccc(cc3)[N+](=O)[O-])[N+](=O)[O-] SB01348 c1cc(ccc1c2nnc(o2)c3ccc(cc3)N)N SB01349 c1ccc(cc1)/C(=C(/C(F)(F)F)\Oc2ccc(cc2Cl)Cl)/C#N SEW03567 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)N)C SEW04161 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3ccc(cc3)C SEW04820 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnn3C(=O)Nc4ccccc4 SPB04978 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnn3C(=O)Nc4ccc(cc4)Cl SPB04979 Cc1ccc(cc-2c(cc(c12)/N=N\c3ccc(cc3)OC)C)C(C)C SEW04851 CCc1cccc(c1NC(=O)CSc2c(c(c3c(n2)CCCC3)c4cccs4)C#N)CC SPB07072 c1ccc(cc1)n2c(nnn2)S SB01352 COC(Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)c3ccc(cc3)Cl)OC SPB04878 Cc1cc(no1)c2nc(cs2)c3ccc(cc3)OC SPB04687 CCc1c([nH]c(c1C(=O)OC)C)C SP00051 COc1ccc(cc1)S(=O)(=O)NNC(=O)c2cccn2c3ccc(cc3)F SEW04805 COC(=O)c1ccc(n1c2ccc(cc2)F)C=C(C#N)C#N SEW04811 c1ccc(cc1)C(C2CCCCC2)O SEW04844 c1c(c(sc1S(=O)(=O)N2CCOCC2)Cl)Br SEW04935 Cc1c(n(c(c1C#N)n2cccc2)Cc3cccs3)C SPB01922 c1cc(ccc1/C=N/NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F SEW04942 c1cc(cc(c1)NC(=O)O/N=C(/c2ccc(cc2)Oc3c(cncc3Cl)Cl)\N)C(F)(F)F SPB07110 COc1ccc(cc1)NC(=O)O/N=C(/c2ccc(cc2)Oc3c(cncc3Cl)Cl)\N SPB07111 c1c(c(sc1S(=O)(=O)N2CCCC2)Cl)Br SEW04946 Cc1c(c(on1)C)C(=O)NNC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW04949 C/C(=N\Nc1c(cc(cn1)C(F)(F)F)Cl)/c2ccc(cc2)Oc3c(cncc3Cl)Cl SPB07115 COc1ccc(cc1OC)C/N=C/c2cc(c(c(c2)OC)OC)OC SEW04960 CCCCNC(=O)OCCSc1ccc(cc1[N+](=O)[O-])C#N SEW04308 c1cc(ccc1/C=C/C(=O)O)OC(F)(F)F SEW04310 c1cc(ccc1/C=N/Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F)OC(F)(F)F SEW04312 c1cc(ccc1C(=N)NC(=O)c2ccc(nc2)OCC(F)(F)F)C(F)(F)F SPB07024 COC(=O)c1ccc(n1c2ccc(cc2)F)/C=N/Nc3ccc(cc3)C(F)(F)F SEW04862 c1ccc(cc1)S(=O)(=O)Cc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl SPB01962 Cc1cc([nH]c1/C=C(\C#N)/C(=O)OC)C SEW04975 Cc1cc([nH]c1/C=C(\C#N)/S(=O)(=O)c2ccccc2)C SEW04976 Cc1cc([nH]c1/C=C(\C#N)/C(=O)c2cccs2)C SEW04977 Cc1cccc(c1NC(=O)n2c(ccn2)c3c(onc3c4ccccc4)C)C SPB05003 Cc1c(c(no1)c2ccccc2)c3csc(n3)N/N=C/c4c(cccc4Cl)Cl SPB05031 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)c4ccc(cc4)C(C)(C)C SPB05034 c1cc(ccc1C(=O)NNC(=O)c2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl)Cl SPB02060 CC(C)C(=O)NNC(=O)c1csc(n1)CS(=O)(=O)c2ccc(cc2)Cl SPB02061 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)Nc3ccc(cc3F)F)Cl SPB02065 c1cc(cc(c1)C(F)(F)F)c2ccnc3n2nc(c3)c4nc(cs4)c5ccc(cc5)Cl SEW04892 c1ccc(cc1)Cn2c(nnc2Sc3ncc(s3)[N+](=O)[O-])O SPB01974 c1ccc(c(c1)C(F)(F)F)n2c(nnc2Sc3ncc(s3)[N+](=O)[O-])O SPB01975 c1c(cc(cc1F)F)COC(=O)c2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-] SEW04694 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)O)Cl SP00061 c1ccc(cc1)C(c2ccncc2)O SEW04833 Cc1c(sc(n1)COc2ccc(cc2)C(C)(C)C)C(=O)NN SPB02078 CCOC(=O)c1cnc(nc1NNC(=O)c2ccc(cc2)Cl)C(F)(F)F SPB04944 c1cc(ccc1C2SCCS2)OCC(=S)N SPB01940 Cc1c(n2ccccc2n1)c3ccnn3C(=O)c4ccc(cc4)C(F)(F)F SPB04923 CN(C)/C=C/C(=O)c1cc(no1)c2ccccc2 SPB04924 c1cc(sc1)c2ccc(s2)c3nc(cs3)c4ccc(cc4)C(F)(F)F SEW04836 c1cc(sc1)c2ccc(s2)c3nc(cs3)c4ccc(c(c4)F)F SEW04837 c1c(cc(cc1F)F)COc2cc(cc(c2)Cl)Cl SEW04746 c1ccc(cc1)c2cc(on2)c3csc(n3)Nc4ccc(cc4)Cl SPB04883 c1ccc(c(c1)C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F SPB01793 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)Nc3cc(cc(c3)Cl)Cl)Cl SPB02071 Cc1c(n(c(c1C#N)NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cc3cccnc3)C SPB01937 c1cc(ccc1/C(=N/OC(=O)c2ccc(cc2)Cl)/N)Oc3ccc(cn3)C(F)(F)F SPB02980 Cc1c(n(oc1=O)C)C(=O)Oc2cc(cc(c2)Cl)Cl SPB02986 c1cc(c(cc1Cl)Cl)/C=N/O SPB04865 COc1ccc(cc1)OCC(=N)NC(=S)Nc2cccc(c2)C(F)(F)F SPB07027 COc1ccc(cc1)OCC(=N)NC(=S)Nc2ccc(cc2)Cl SPB07028 CCOC(=O)c1c(nc(s1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C SPB01851 CCOC(=O)c1c(nc(s1)Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])C SPB01852 CCOC(=O)c1c(nc(s1)COc2ccc(cc2)C(C)(C)C)C SPB02075 Cc1cc(cc(c1Cl)C)OCc2nc(on2)CSc3ccc(cn3)C(F)(F)F SPB02970 Cc1c(sc(n1)c2ccccc2)C(=O)Sc3ccc(cc3)Cl SPB02973 c1ccc(cc1)Cn2c(nnc2S)O SPB01971 COC(Cn1c(nnc1SCC(=O)c2ccccc2)c3ccccc3)OC SPB04857 c1cc(ccc1C2SCCS2)OCc3nc(cs3)C(=O)NN SPB02083 c1ccc(cc1)/C=N/Nc2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl SPB04956 c1ccc(cc1)c2cc(on2)c3ccnn3C(=O)c4ccccc4 SPB04963 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)CCC(=O)O SEW04839 CCOC(=O)c1cc(oc1C)c2cccc(c2)[N+](=O)[O-] SP00085 CCOC(=O)c1c(sc(n1)C)c2ccnn2S(=O)(=O)c3ccc(cc3Cl)Cl SPB04774 Cc1ccc(cc1[N+](=O)[O-])NC(=O)Cc2cc(cc(c2)F)F SEW04670 Cc1c(nc(nc1Sc2cccc(c2)C(F)(F)F)C(F)(F)F)C SPB04776 c1ccc(cc1)NC(=O)O/N=C(/c2ccc(cc2)Oc3c(cncc3Cl)Cl)\N SPB07108 c1cc(ccc1/C(=N/OC(=O)Nc2ccc(cc2)Cl)/N)Oc3c(cncc3Cl)Cl SPB07109 Cc1c(n(c(c1C#N)N)Cc2c(cccc2Cl)Cl)C SPB01965 Cc1ccc(cc1)SC(=O)c2c(nc(s2)c3ccccc3)C SPB02972 c1cc(ccc1c2csc(n2)COc3ccc(cc3)C4SCCS4)[N+](=O)[O-] SPB01943 CCOC(=O)c1c(nc(s1)COc2ccc(cc2)C3SCCS3)C SPB01944 c1cc(ccc1c2nc(on2)c3ccc(cc3)Cl)Oc4ccc(cn4)C(F)(F)F SPB02981 c1ccn(c1)c2cccc(c2)c3nc(cs3)CC(=O)NN SPB01751 c1cc(c(c(c1)Cl)/C=N/Nc2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl)Cl SPB04905 CN(C)c1ccc(c(c1C#N)F)C=C(C#N)C#N SEW04934 COC(=O)c1cc(=O)c2cc(ccc2[nH]1)C(F)(F)F SEW04940 c1cc(ccc1/C=N/NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl SEW04941 CC(=O)c1cc(no1)c2ccc(c(c2)Cl)Cl SPB04952 c1cc(sc1)c2ccc(s2)c3nc(cs3)c4ccc(cc4)Cl SEW04835 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)O SP00065 Cc1ccc(cc1)NC(=S)NC(=N)COc2ccccc2 SPB07029 COC(Cn1c(nnc1S)c2ccccc2)OC SPB04849 COC(Cn1c(nnc1SCc2ccc(cc2)Cl)c3ccccc3)OC SPB04851 Cc1c(sc(n1)COc2ccc(cc2)C(C)(C)C)C(=O)NNC(=O)c3ccc(cc3Cl)Cl SPB02080 CCOC(=O)c1csc(n1)COc2ccc(cc2)C3SCCS3 SPB02081 CCOC(=O)c1c(noc1c2csc(n2)COc3ccccc3)C SPB04693 COc1ccc(cc1OC)CNCc2cc(c(c(c2)OC)OC)OC SEW04968 Cc1ccc(cc-2c(cc(c12)/C=N\NC(=O)CCc3ccc(cc3)O)C)C(C)C SEW04830 Cc1ccc(cc-2c(cc(c12)/C=C(/C#N)\S(=O)(=O)C)C)C(C)C SEW04831 c1cc(sc1)c2ccc(s2)C(=S)N SEW04832 Cc1c(sc(n1)C)C(=O)O CC05801 Cc1cc(c(c(c1)C)Nc2nc(cs2)c3cc(no3)c4ccccc4)C SPB04882 COC(Cn1c(nnc1SCC(=O)Nc2ccc(cc2)C(F)(F)F)c3ccc(cc3)Cl)OC SPB04889 CCOC(=O)Nc1ccc(cc1OC)OC SEW04922 CCOC(=O)c1csc(n1)CS(=O)(=O)c2ccc(cc2)Cl SPB02013 CCC(=O)O/N=C(/c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2F)F)\N SPB01977 Cc1c(sc(n1)C)c2nnc(o2)c3ccc(cc3)Cl SPB02988 c1ccc(cc1)c2cc(on2)c3csc(n3)N/N=C/c4ccc(cc4)Cl SPB04894 Cc1cc(n(n1)C)/C(=N\O)/N SPB02000 Cc1cc(nc(c1C#N)SCc2nc(no2)COc3cccc(c3)C(F)(F)F)C SPB02969 c1ccc(cc1)/C=N/c2ccc(cc2)Cl SEW04901 CC(C)(C)c1csc(n1)c2cc3nccc(n3n2)c4cccc(c4)C(F)(F)F SEW04903 c1cc(cc(c1)C(F)(F)F)c2ccnc3n2nc(c3)c4nc(cs4)c5ccc(cc5)[N+](=O)[O-] SEW04904 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)Nc3ccc(cc3)Cl)Cl SPB02102 c1cc2c(cc1Cl)nc(s2)Sc3ncc(s3)[N+](=O)[O-] SPB02004 c1ccc(cc1)c2[nH]c(nn2)Sc3ncc(s3)[N+](=O)[O-] SPB02005 c1cc(ccc1c2[nH]c(nn2)Sc3ncc(s3)[N+](=O)[O-])Cl SPB02006 c1ccc(cc1)c2c(nc(c(n2)C#N)C#N)c3ccccc3 SEW04910 CC(=O)C(C(=O)C)Sc1nnnn1c2ccccc2 SPB05861 c1cc(ccc1/N=C/c2c(nc3n2ccs3)Sc4ccc(cc4)Cl)Cl SPB05863 c1cc(c(c(c1)Cl)Cc2nc(cs2)NC(=O)NNc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl SPB02046 Cc1cc(no1)/C=N/NS(=O)(=O)c2cccc(c2)C(F)(F)F SPB04787 Cc1cc(no1)/C=N/NS(=O)(=O)c2ccc(c(c2)Cl)F SPB04788 COc1ccccc1NC(=O)NNC(=S)NCC(OC)OC SPB04795 c1cc(ccc1/C=N/Nc2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl)Cl SPB04903 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=O)Nc3ccc(cc3)C)C SEW04763 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2[N+](=O)[O-])C#N SPB02026 c1cc(c(c(c1)Cl)Cc2nc(cs2)NC(=O)NN3CCOCC3)Cl SPB02043 Cn1cc(c(n1)C2NN=C(S2)SCC(=O)Nc3cccc(c3)Cl)Cl SPB07015 Cc1cc(ccc1OC)/C=N/Cc2cc(c(c(c2)OC)OC)OC SEW04988 c1cc(sc1)c2c3c(nc(c2C#N)SCC(=O)c4ccc(cc4)Cl)CCCC3 SPB07057 c1cc(sc1)c2c3c(nc(c2C#N)SCC(=O)c4ccc(c(c4)F)F)CCCC3 SPB07059 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)C/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/N SPB01797 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/CS(=O)(=O)Cc2cccc(c2)C(F)(F)F)\N SPB01798 c1cc(ccc1NC(=O)OCCSc2ccc(cc2[N+](=O)[O-])C#N)OC(F)(F)F SEW04296 COc1ccc(cc1OC)CNCc2ccc(c(c2)OC)OC SEW04964 Cc1c(c(no1)c2ccccc2)c3csc(n3)COc4ccccc4 SPB05000 Cc1c(c(no1)c2ccc(cc2Cl)Cl)C(=O)C SPB05001 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4ccc(cc4)C(C)(C)C SPB05014 Cc1ccc(cc1)S(=O)(=O)n2c(ccn2)c3c(onc3c4ccccc4)C SPB05016 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)c4ccc(cc4)Cl SPB05035 CNC(=S)N/N=C/c1c(nc2n1ccs2)Sc3ccc(cc3)Cl SPB05866 c1cc(ccc1C(=O)N/N=C(/c2cnccn2)\N)Cl SPB07144 c1cc(ccc1C#N)Oc2ccc(cn2)C(F)(F)F SPB02965 Cc1c(sc(n1)c2ccccc2)C(=O)Sc3ccc(cc3)C(F)(F)F SPB02971 c1cc(ccc1c2csc(n2)C3(CC3)c4ccc(cc4Cl)Cl)C(F)(F)F SEW04888 Cc1ccc(cc1)c2nnc(o2)COc3ccsc3C(=O)OC SPB07047 Cc1ccc(cc-2c(cc(c12)/C=N\Nc3c(cc(cc3Cl)Cl)C(F)(F)F)C)C(C)C SEW04810 CCOC(=O)c1c(noc1/C(=N\OC(=O)c2ccccc2)/C)C SPB04735 Cc1c(sc(n1)c2ccc(s2)c3cccs3)c4ccnn4C(=O)c5cccs5 SEW04867 COC(=O)/C=C(\C(=O)OC)/Oc1cccc(c1)C(F)(F)F SEW04873 COc1ccc(cc1)c2nnc(o2)COc3ccsc3C(=O)OC SPB07031 c1cc(sc1)c2c3c(nc(c2C#N)S)CCCC3 SPB07033 CCOC(=O)COc1cccc(c1)[N+](=O)[O-] SEW04874 c1cc(c(cc1Cl)Cl)C2(CC2)C(=S)N SEW04879 c1cc(c(cc1c2csc(n2)C3(CC3)c4ccc(cc4Cl)Cl)Cl)Cl SEW04883 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=O)c3ccccc3C(=O)O)C SEW04756 COc1c(ccc(c1)/C=C\2/C(=O)/C(=C/c3cc(c(cc3)O)OC)/COC2)O SEW04759 c1cc(sc1)c2c3c(nc4c2c(c(s4)C(=O)c5ccc(cc5)Cl)N)CCCC3 SPB07068 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3cccs3 SEW04821 c1ccc(cc1)C(=O)c2c(c3c(c4c(nc3s2)CCCC4)c5cccs5)N SPB07070 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)Cl)CC3CC3)C SPB01904 CC(C)NC(=O)O/N=C(\COc1ccc(cc1)C2SCCS2)/N SPB01905 Cc1c(n(c(c1C#N)NC(=O)c2cccs2)CC3CC3)C SPB01909 COC(Cn1c(nnc1SCC(=O)c2ccccc2)c3ccc(cc3)Cl)OC SPB04877 c1cc(c(cc1C(F)(F)F)Cl)NC(=O)NN SEW04909 COC(c1c(cc(c(n1)S)C#N)C(=O)OC)OC SPB04940 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=O)/C=C/C(=O)O)C SEW04753 COC(=O)c1ccc(n1c2ccc(cc2)F)/C=C\3/c4ccccc4NC3=O SEW04812 CCCCn1c(c(c(c1N)S(=O)(=O)c2ccccc2)C)C SPB01866 CCCS(=O)(=O)c1c(c(n(c1N)Cc2ccc(cc2)C(F)(F)F)C)C SPB01872 CCOC(=O)c1c(c(n(c1NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cc3ccccc3)C)C SPB01928 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl SPB04835 Cc1c(n2ccccc2n1)c3ccnc(n3)SCc4ccc(cc4)Cl SPB04836 Cc1csc(c1N)C(=O)OC SB01297 CC(=O)N1CCC(CC1)C(=O)c2ccc(cc2F)F SEW04268 c1ccc(c(c1)OCc2nc(cs2)C(=O)NNC(=O)c3ccc(cc3)Cl)Cl SPB02029 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)N3C(=O)C4C5CC(C4C3=O)C=C5 SEW04766 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2[N+](=O)[O-])/C(=N/OC(=O)c3cccs3)/N SPB02036 COc1ccc(cc1)/C=N/NC(=O)c2cccn2c3ccc(cc3)F SEW04779 c1cc(n(c1)c2ccc(cc2)F)C(=O)NNC(=S)Nc3ccc(c(c3)Cl)Cl SEW04781 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)Cl)Cc3cccs3)C SPB01917 CCC(=O)Nc1c(c(c(n1Cc2cccs2)C)C)C#N SPB01918 c1cc(cc(c1)Cl)S(=O)(=O)NNC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F SPB04799 Cc1c(nc(nc1NCc2ccc(cc2)OC)C(F)(F)F)C SPB04812 CCOc1ccc(cc1)C(C[N+](=O)[O-])Sc2ccccc2N S10369 c1cc(c(cc1/C(=N/O)/N)[N+](=O)[O-])Oc2ccc(c(c2)Cl)Cl SPB01939 c1ccc(c(c1)N)SC(C[N+](=O)[O-])c2c(cccc2Cl)F S10385 c1cc(cc(c1)C(F)(F)F)c2ccnc3n2ncc3C(=S)N SEW04891 c1ccc(cc1)/N=C/c2c(nc3n2ccs3)Sc4ccc(cc4)Cl SPB05862 Cc1ccc(cc1)/N=C/c2c(nc3n2ccs3)Sc4ccc(cc4)Cl SPB05864 Cc1c(c(no1)c2ccccc2)c3csc(n3)Nc4ccccc4Cl SPB05020 c1ccc(c(c1)NCN2C(=O)CCC2=O)OC(F)(F)F TL00406 COc1cccc(c1OC)/C=N/NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW04944 c1c(c(sc1S(=O)(=O)N2CCSCC2)Cl)Br SEW04945 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2c(cc(s2)Cl)Br SEW04948 Cc1c(n2ccccc2n1)c3ccnc(n3)S SPB04780 c1cc(ccc1OCc2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl)Cl SPB04920 c1ccc(cc1)CC(C(F)(F)F)OS(=O)(=O)c2cc(c(s2)Cl)Cl SEW03707 Cc1ccc(cc1)N/N=C(\C#N)/S(=O)(=O)c2ccsc2 SEW03715 COC(Cn1c(nnc1SCc2ccccc2)c3ccccc3)OC SPB04853 COC(Cn1c(nnc1SCc2ccccc2Cl)c3ccccc3)OC SPB04854 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)CC(=S)N SPB02010 Cc1ccc(cc1)CSc2c(c(c3c(n2)CCCC3)c4cccs4)C#N SPB07038 CCOC(=O)c1cnc(nc1Nc2ccccc2)C(F)(F)F SPB04763 CCOC(=O)c1cc(oc1C(F)(F)F)c2ccc(cc2)Cl SP00058 Cc1c(n(oc1=O)C)C(=O)Oc2ccc(cc2)Cl SPB02985 Cc1c(n(oc1=O)C)C(=O)Oc2cccc(c2)C(F)(F)F SPB02987 Cc1c(sc(n1)C)c2nnc(o2)c3ccc(cc3)C(F)(F)F SPB02989 c1cc(ccc1NCN2C(=O)CCC2=O)OC(F)(F)F TL00404 c1cc(ccc1c2nc(on2)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl)C(F)(F)F SPB03136 c1ccc(cc1)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4ccccc4 SPB05042 Cc1ccc(cc1)C(=O)N/N=C(/c2cnccn2)\N SPB07146 c1ccc(cc1)c2cc(on2)c3csc(n3)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB04939 Cc1c(n(c(c1C#N)NC(=O)c2cc(cc(c2)Cl)Cl)CC3CC3)C SPB01908 Cc1c(n(c(c1C#N)N)Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C SPB01911 Cn1c(nnc1SCc2csc(n2)COc3ccc(cc3)C4SCCS4)C(F)(F)F SPB02093 CCCCCn1c(nnc1SCc2csc(n2)COc3ccc(cc3)C4SCCS4)O SPB02094 COc1ccc(cc1)OC(=O)c2csc(n2)Cc3c(cccc3Cl)Cl SPB02106 c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cc(no3)c4ccc(cc4Cl)Cl SPB05072 CC(=O)Nc1ccc(cc1)C2NC(=NN2)c3cnccn3 SPB07138 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)Oc3cc(cc(c3)Cl)Cl)Cl SPB02107 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)NCc3cccs3)Cl SPB02109 Cc1nnc(o1)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl SEW04924 c1cc(c(c(c1NN=C(C#N)C#N)F)F)F SEW04994 c1cc(c(c(c1)Cl)Cc2nc(cs2)NC(=O)NCC3CC3)Cl SPB02113 Cc1cccc(c1NC(=O)n2c(ccn2)c3c(onc3c4ccc(cc4)Cl)C)C SPB04981 Cc1c(n(oc1=O)C)c2nc(no2)c3ccc(o3)[N+](=O)[O-] SPB02997 c1cc(ccc1C(=O)NNC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl SEW04953 COc1ccc(cc1)CNCc2ccc(cc2)OC SEW04956 COc1ccc(cc1)CNCc2cc(c(c(c2)OC)OC)OC SEW04962 CCOC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F SEW04920 Cc1cc(c(s1)C)C2CC(=O)Nc3ccccc3S2 SEW04325 c1c(cc(c(c1Cl)NN=C(C#N)C#N)Cl)C(F)(F)F SEW05092 CCOC(=O)c1csc(n1)CS(=O)(=O)Cc2ccc(cc2)F SPB02111 c1cc(c(cc1N2C(=O)CSCC2=O)Cl)F S10455 c1c(cc(cc1Cl)Cl)N2C(=O)CSCC2=O S10456 c1c(cc(cc1Cl)Cl)OCc2nc(cs2)C(=O)O SPB02119 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NNC(=O)c2csc(n2)COc3cc(cc(c3)Cl)Cl)C(F)(F)F SPB02123 CC(C)(C)c1ccc(cc1)c2nnn(n2)CC(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB02125 C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/c2cc(no2)c3ccccc3 SPB04818 Cc1ccc(cc1)NC(=O)c2csc(n2)Cc3c(cccc3Cl)Cl SPB02066 c1ccc(c(c1)NC(=O)c2csc(n2)Cc3c(cccc3Cl)Cl)Cl SPB02068 c1ccc2c(c1)n(c(=O)o2)Cc3ccc(cc3)Cl SPB03004 Cc1c(c([nH]n1)c2c(nns2)C)C(=O)N/N=C/c3ccc(s3)[N+](=O)[O-] SPB02135 CC(C)C(=O)NNC(=O)c1csc(n1)c2cccs2 SPB02136 c1cc(sc1)c2nc(cs2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB02138 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Sc3nnnn3c4ccccc4 SPB05880 c1cc(c(cc1S(=O)(=O)NNC(=O)c2csc(n2)COc3cc(cc(c3)Cl)Cl)Cl)Cl SPB02121 Cc1ccc(cc1C)c2cc(on2)c3csc(n3)COc4cccc(c4)Cl SPB04994 c1cc(sc1)c2nc(cs2)C(=O)NNC(=O)Nc3ccc(cc3)Cl SPB02139 Cc1c(c(n(n1)C)c2c(nns2)C)C(=O)OC SPB02142 CC(C)(C)c1csc(n1)c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F SPB03019 Cc1c(c(no1)c2ccccc2)c3ccnn3C(=O)NC(C)C SPB05008 Cc1c(c(no1)c2ccccc2)c3ccnn3C(=O)c4ccc(cc4)Cl SPB05010 Cc1c(c(n(n1)S(=O)(=O)c2ccc(cc2)Cl)C)Sc3nnnn3c4ccccc4 SPB05891 c1cc(cc(c1)NC(=O)c2csc(n2)Cc3c(cccc3Cl)Cl)C(F)(F)F SPB02070 CC(=O)CSc1nnc(n1C)C(F)(F)F SPB07064 CCCCNC(=O)NNC(=O)c1cccn1c2ccc(cc2)F SEW04801 CC(C)(C)C(=O)NNC(=O)c1ccc(o1)Oc2cc(cc(c2)Cl)Cl SPB03106 CC(C)(C)c1ccc(cc1)c2nc(on2)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl SPB03135 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4ccc(cc4)Cl SPB05006 CCOC(=O)c1cnc(nc1Nc2ccc(cc2)Cl)c3cccs3 SPB05884 CCOC(=O)c1cc(oc1C)c2ccc(cc2)Cl SP00057 COC(=O)CCCCCCCC(=O)Nc1ccc(cc1)Cl SEW04954 Cc1c(n(oc1=O)C)c2nc(no2)c3ccc(cc3)C(F)(F)F SPB02993 Cc1nc(no1)c2ccc(cc2)Oc3c(cc(cn3)C(F)(F)F)Cl SPB02999 Cc1c(sc(n1)c2ccccc2)c3nnnn3c4ccc(cc4)Cl SPB03024 c1cc(cc(c1)C(F)(F)F)c2ccnc3n2ncc3C#N SEW04841 c1cc(c(cc1Cl)Cl)c2cc(on2)c3csc(n3)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB04899 c1cc2c(cc1C(=S)N)CCO2 SP00108 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C=C/N(C)C SP00110 c1c(cc(cc1Cl)Cl)NC(=O)CSCC(=O)O S10452 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/Nc3ccc(cn3)Cl)/C#N SP00147 CC(C)(C)c1nnc(o1)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl SPB03110 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNC(=O)c3ccccc3 SPB03113 c1c(cc(cc1C(F)(F)F)N2C(=O)CSCC2=O)C(F)(F)F S10457 Cc1c(c(c([nH]1)C)C(=O)OC)c2cc[nH]n2 SP00120 Cc1c(c(c([nH]1)C)C(=O)OC)c2ccno2 SP00121 Cc1cc(c(o1)C)C(=O)CC#N SP00064 CSc1c(c(nc(n1)COc2ccccc2Cl)N)C#N SPB05894 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)NNC(=O)c2csc(n2)c3ccc(cn3)C(F)(F)F SPB05839 c1cc(ccc1S(=O)(=O)NNC(=O)c2csc(n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl SPB05842 COC(Cn1c(nnc1S)c2ccc(cc2)Cl)OC SPB04869 COC(Cn1c(nnc1SCc2ccccc2)c3ccc(cc3)Cl)OC SPB04870 COC(Cn1c(nnc1SCc2ccccc2Cl)c3ccc(cc3)Cl)OC SPB04873 c1ccc(cc1)Cn2c3ccccc3oc2=O SPB03005 c1ccc2c(c1)n(c(=O)o2)Cc3ccc(cc3)C(F)(F)F SPB03006 c1ccc2c(c1)n(c(=O)o2)Cc3cccc(c3)Cl SPB03007 CCOC(=O)c1csc(n1)c2ccc(cn2)C(F)(F)F SPB05832 Cc1c2cn[nH]c(=O)c2c(n1c3ccccc3)C SP00128 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/Nc3cccc(c3)OC(F)(F)F)/C#N SP00158 Cc1ccc(cc1)NC(=O)c2c(nc(s2)c3ccccc3)C SPB03010 Cc1c(sc(n1)c2ccccc2)C(=O)Nc3cccc(c3)C(F)(F)F SPB03012 c1ccc(cc1)c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F SPB03014 COC(=O)/C=C(\C(=O)OC)/Nc1ccc(cc1)[N+](=O)[O-] SEW04927 Cc1c(cc(o1)c2ccc(cc2)Cl)COC(=O)Nc3ccc(cc3)Cl SP00129 Cc1c(cc(o1)c2ccc(cc2)Cl)COC(=O)Nc3ccc(cc3)OC(F)(F)F SP00136 COc1ccc(cc1OC)C/N=C/c2ccc(c(c2)OC)OC SEW04959 Cc1ccc(cc1)CSc2nnc(n2CC(OC)OC)c3ccccc3 SPB04852 COC(=O)C(Cc1ccc(cc1Cl)Cl)S(=O)(=O)c2ccc(cc2)Cl SEW04827 Cc1ccc(cc-2c(cc(c12)/C=N\NC(=S)N)C)C(C)C SEW04829 Cc1cc(nc(c1C#N)SCc2nc(no2)c3ccc(cc3)OC(F)(F)F)C SPB03042 CCOC(=O)c1cnc(nc1Nc2ccc(cc2)C)c3cccs3 SPB05882 CCOC(=O)c1cnc(nc1Nc2cccc(c2)C(F)(F)F)c3cccs3 SPB05883 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)Sc3ccc(cc3)Br SPB03051 CSc1c(c(nc(n1)COc2ccccc2)N)C#N SPB05893 Cc1c(c(n[nH]1)C)Sc2nnnn2c3ccccc3 SPB05870 CSc1c(c(nc(n1)COc2ccccc2Cl)c3cccs3)C#N SPB05901 Cc1cccc(c1C)Cn2c(c(c(c2N)S(=O)(=O)c3ccccc3)C)C SPB02088 Cc1c(c(no1)c2ccccc2)C(=O)/C=C/N(C)C SPB04966 c1cc(c(cc1Nc2nc(cs2)C(F)(F)F)Cl)Cl SPB05914 CCOC(=O)c1csc(n1)c2cccs2 SPB02128 c1cc(sc1)c2nc(cs2)C(=O)NNC(=O)c3ccc(cc3)Cl SPB02137 Cc1c(c([nH]n1)c2c(nns2)C)C(=O)N/N=C/c3c(cccc3Cl)Cl SPB02134 c1cc(sc1)c2c3c(nc(c2C#N)SCC(=O)Nc4cc(cc(c4)Cl)Cl)CCCC3 SPB07071 Cc1cc(c(o1)C(F)(F)F)C(=O)/C(=C/Nc2cccc(c2)OC(F)(F)F)/C#N SP00166 COc1cccc(c1C(=O)NNC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC SEW04950 Cc1c(snn1)C(=O)NNC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW04951 c1cc(ccc1/C(=N/OC(=O)c2ccc(cc2)Cl)/N)Oc3c(cncc3Cl)Cl SPB07121 c1cc(ccc1/C(=N/O)/N)Oc2c(cc(cn2)C(F)(F)F)Cl SPB02968 CC(C)NC(=O)NNC(=O)c1cccc(c1)COc2ccc(cc2)C3SCCS3 SPB01994 Cc1c(nc(nc1NNC(=O)Nc2ccccc2)C(F)(F)F)C SPB04917 c1ccc(cc1)c2cc(on2)c3csc(n3)COc4ccc(cc4)Cl SPB04921 Cc1nc(cs1)CSc2nnc(n2Cc3ccccc3)O SPB02174 c1cc(ccc1S(=O)(=O)Cc2nc(cs2)C(=O)NN)Cl SPB02024 c1ccc(c(c1)OCc2nc(cs2)C(=O)NNC(=O)c3cccs3)Cl SPB02028 Cc1c(cc(o1)C(C)(C)C)C(=O)C(=C2SCCS2)C#N SP00153 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/Nc3ncccn3)/C#N SP00160 c1cc(ccc1CS(=O)(=O)CC#N)F SPB02049 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2[N+](=O)[O-])/C(=N/O)/N SPB02034 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2[N+](=O)[O-])/C(=N/OC(=O)C3CC3)/N SPB02037 Cc1cc(c(o1)C(F)(F)F)C(=O)/C(=C/Nc2ccc(cc2)Cl)/C#N SP00162 c1cc(c(c(c1)Cl)Cc2nc(cs2)NC(=O)Nc3cc(cc(c3)Cl)Cl)Cl SPB02020 c1cc(sc1)c2c3c(nc(c2C#N)SCc4ccc(cc4)Cl)CCCC3 SPB07036 c1cc(cc(c1)/N=C/c2c(nc3n2ccs3)Sc4ccc(cc4)Cl)C(F)(F)F SPB05865 c1ccc(cc1)CSc2c(c(c3c(n2)CCCC3)c4cccs4)C#N SPB07037 c1cc(ccc1C2SCCS2)OC/C(=N/OC(=O)c3ccc(cc3)Cl)/N SPB01887 c1cc(cc(c1)NC(=O)O/N=C(/CSc2ccc(cn2)C(F)(F)F)\N)C(F)(F)F SPB03064 CCOC(=O)c1cnc(nc1NNC(=O)c2ccccc2)C(F)(F)F SPB04943 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/c3ccccc3)/C#N SP00172 Cc1cc(cc(c1Cl)C)OC(=O)c2cc(nn2Cc3ccccc3)C(C)(C)C SPB03045 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Oc3cccc(c3)C(F)(F)F SPB03047 Cc1c(n2ccccc2n1)c3ccnn3C(=O)c4ccc(cc4)Cl SPB04925 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)C(=O)NN SPB02053 c1cc(sc1)C(=O)O/N=C(/CS(=O)(=O)Cc2ccc(cc2)F)\N SPB02054 Cc1c(n2ccccc2n1)c3ccnn3C(=O)C SPB04931 Cc1cc(ccc1NC(=O)COCC(=O)O)Cl S10464 c1cc(ncc1C(=O)NC(=N)c2cc(cc(c2)Cl)Cl)OCC(F)(F)F SPB07025 CCn1c(c(c(n1)C)Br)C(=O)NNC(=O)c2c(cc(cn2)C(F)(F)F)Cl SPB05924 CC(C)c1ccc(cc1)NC(=O)c2csc(n2)Cc3c(cccc3Cl)Cl SPB02104 c1cc(ccc1CS(=O)(=O)CC(=S)N)F SPB02110 CCOC(=O)c1csc(n1)COc2cc(cc(c2)Cl)Cl SPB02118 CC(C)(C)c1ccc(cc1)c2nnn(n2)CC(=O)NNS(=O)(=O)c3ccc(cc3)Cl SPB02124 c1ccc(cc1)NC(=O)O/N=C(/CSc2ccc(cn2)C(F)(F)F)\N SPB03066 Cc1c(sc(n1)c2ccc(cn2)C(F)(F)F)C(=O)NNC(=O)c3ccccc3C(F)(F)F SPB05917 c1cc(sc1)c2c3c(nc4c2c(c(s4)C(=O)c5ccc(c(c5)F)F)N)CCCC3 SPB07069 c1cc(ccc1/C=N/Nc2nc(cs2)C(F)(F)F)Cl SPB05919 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2csc(n2)COc3ccc(cc3)C4SCCS4)Cl SPB02112 c1cc(ccc1c2nc(on2)COc3ccc(cc3)Cl)OC(F)(F)F SPB03071 C#Cc1cccc(c1)NC(=O)CSc2c(c(c3c(n2)CCCC3)c4cccs4)C#N SPB07073 c1ccc(cc1)NC(=O)c2c(c3c(c4c(nc3s2)CCC4)c5cccnc5)N SPB07097 CCOC(=O)c1c(nc(s1)SCC(=O)c2ccc(cc2)Cl)C SPB01854 CCOC(=O)c1c(nc(s1)SCC(=O)c2ccc(cc2Cl)Cl)C SPB01855 CCCCCn1c(nnc1S)O SPB01983 COC(=O)c1cccc(c1)COc2ccc(cc2)C3SCCS3 SPB01990 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2c(c(c3c(n2)CCCC3)c4cccs4)C#N SPB07058 c1ccc(cc1)c2cc(on2)c3ccnn3C(=O)Nc4cccc(c4)Cl SPB05068 c1ccc2c(c1)nc3n2c(c(s3)C#N)N SEW05169 Cc1ccccc1N/C=C(\C#N)/C(=O)c2cc(oc2C(F)(F)F)C SP00168 COc1ccc(cc1)C/N=C/c2ccc(c(c2)OC)OC SEW04957 Cc1c(cc(o1)c2ccc(cc2)Cl)COC(=O)Nc3ccccc3 SP00134 Cc1c(cc(o1)c2ccc(cc2)Cl)COC(=O)Nc3cccc(c3)OC SP00135 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB03114 Cc1ccc(cc1C)c2cc(on2)c3csc(n3)COc4ccccc4Cl SPB04986 C/C(=N\NC(=S)NC(C)(C)C)/c1ccc(cc1)Oc2c(cncc2Cl)Cl SPB07118 C/C(=N\NC(=S)N)/c1ccc(cc1)Oc2c(cncc2Cl)Cl SPB07119 c1cc(ccc1C#N)NC(=O)Nc2ccc(cc2)C#N SEW04984 Cc1c(sc(n1)CS(=O)(=O)c2ccc(cc2)Cl)C(=O)O SPB02082 c1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2)Oc3c(cncc3Cl)Cl)\N SPB07120 CCOC(=O)Nc1ccc(cc1Cl)C(F)(F)F SEW04898 c1cc(ccc1/C=N/c2cc(cc(c2)Cl)Cl)C(F)(F)F SEW04900 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=O)Nc3cccc(c3Cl)Cl)C SEW04760 c1ccc(c(c1)OCc2nc(cs2)C(=O)NN)Cl SPB02023 c1cc(n(c1)c2ccc(cc2)[N+](=O)[O-])C(=O)C(F)(F)F SEW04764 Cn1cnnc1Sc2ccc(cn2)[N+](=O)[O-] SPB02048 CCOC(=O)c1cnc(nc1NNC(=O)c2ccc(cc2)C)C(F)(F)F SPB04945 c1cc(cc(c1)Cl)NC(=O)O/N=C(/CSc2ccc(cn2)C(F)(F)F)\N SPB03065 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/c3ccccc3Cl)/C#N SP00175 Cc1cccc(c1)/C=C(\C#N)/C(=O)c2cc(oc2C)c3ccc(cc3)Cl SP00177 Cc1cc(no1)N/C=C(\C#N)/C(=O)c2cc(oc2C)c3ccc(cc3)Cl SP00179 CCOC(=O)c1csc(n1)c2cccc(c2Cl)Cl SPB02051 Cc1cc(c(o1)C(F)(F)F)C(=O)/C(=C/Nc2cc(on2)C)/C#N SP00181 c1ccc(c(c1)C(=O)O/N=C(/CS(=O)(=O)Cc2ccc(cc2)F)\N)C(F)(F)F SPB02055 c1ccc(cc1)NC(=O)O/N=C(\COc2ccc(cc2)C3SCCS3)/N SPB01907 Cc1c(c(nc(n1)c2ccccc2OC)SCc3cccc(c3)C(F)(F)F)C(=O)C SPB05816 c1ccc(cc1)SC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl SPB01888 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnn3C(=O)c4ccc(cc4)Cl SPB04989 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnn3S(=O)(=O)c4ccc(cc4)Cl SPB04990 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnn3C(=O)NC(C)C SPB04977 CCOC(=O)c1cnc(nc1NNC(=O)c2ccno2)C(F)(F)F SPB04946 c1cc(ccc1c2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl)C(F)(F)F SPB04955 c1cc(ccc1C(=O)Sc2ccc(cc2)OC(F)(F)F)Cl SPB03075 CC(=O)n1c(ccn1)c2cc(no2)c3ccccc3 SPB04958 Cc1c(c(no1)c2ccccc2)C(=O)C SPB04960 CCn1c(c(c(n1)C)NC(=O)c2ccc(cc2)Cl)C(=O)OC SPB01858 COC(=O)c1c(ccs1)OCc2nnc(o2)c3ccc(cc3)F SPB07030 CCOC(=O)c1cc(on1)c2ccnn2S(=O)(=O)c3ccc(cc3Cl)Cl SPB04815 c1cc(ccc1/C(=N/OC(=O)Nc2ccc(cc2)Cl)/N)Oc3ccc(cn3)C(F)(F)F SPB02983 c1cc(sc1)S(=O)(=O)NCc2ccc3c(c2)CCO3 SP00206 Cc1cc(c(o1)c2ccccc2)/C(=N/OC(=O)c3ccccc3)/N SP00207 Cc1cccc(c1)NC(=S)NCc2ccc3c(c2)CCO3 SP00214 Cc1cc(no1)c2nc(no2)c3ccc(o3)[N+](=O)[O-] SPB03094 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3c(onc3c4ccc(cc4)Cl)C SPB04991 CC(=O)c1ccc(cc1)Oc2c(cncc2Cl)Cl SPB07096 c1cc(c(cc1c2cc(on2)c3csc(n3)COc4cc(cc(c4)Cl)Cl)Cl)Cl SPB04987 c1cc(cc(c1)Cl)OCc2nc(cs2)c3cc(no3)c4ccc(c(c4)Cl)Cl SPB04995 CCOC(=O)c1cc(on1)c2ccnn2S(=O)(=O)c3ccc(cc3)C SPB04816 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)O SB01884 Cc1c(c(no1)c2ccccc2Cl)C(=O)O SB01885 Cc1c(n2ccccc2n1)c3ccnn3C(=O)c4ccno4 SPB04926 c1cc(ccc1c2csc(n2)c3cnccc3C(F)(F)F)c4nc(on4)c5ccc(cc5)Cl SPB05959 c1ccc(c(c1)C(F)(F)F)n2c(nnc2SCC(=O)c3ccc(cc3)[N+](=O)[O-])O SPB02148 Cc1cccc(c1)C2NC(=NN2)c3cnccn3 SPB07136 c1cc(cnc1)C2NC(=NN2)c3cnccn3 SPB07137 Cn1c(nnc1SCC(=O)Nc2ccc(c(c2)Cl)F)C(F)(F)F SPB02152 c1ccc(cc1)Cn2c(nnc2SCC(=O)Nc3cc(cc(c3)Cl)Cl)O SPB02156 CCOC(=O)c1c(nc(s1)c2ccccc2)C SPB02157 Cc1c(cc(o1)c2ccccc2)c3cc[nH]n3 SP00100 CCOC(=O)Nc1cc(cc(c1)Cl)Cl SEW04919 Cc1c(cc(o1)C(C)(C)C)C(=O)/C(=C/Nc2ccc(cn2)Cl)/C#N SP00142 CCOC(=O)Nc1ccsc1C(=O)OC SEW04929 c1cc(cc(c1)NC(=O)O/N=C(/c2ccc(cc2)OC(F)(F)F)\N)C(F)(F)F SPB03034 Cc1cc(no1)C(=O)O/N=C(/c2ccc(cc2)C(C)(C)C)\N SPB03084 CCOC(=O)c1ccc(cc1)n2c(c(c(n2)C)C(=O)OCC)C SEW05142 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC(=O)Nc3cccc(c3)Cl SPB02149 Cc1c(c(n(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)C)C(=O)O SEW05007 COC(=O)c1cc(n(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)O SEW05011 CC(C)c1ccc(cc1)NC(=O)CSc2nc3c(s2)cc(cc3Cl)Cl SPB02169 Cc1nc(cs1)CSc2nnc(n2c3ccccc3)O SPB02172 Cc1ccccc1C(=O)Nc2cc(nn2C)c3cc(oc3C)C(C)(C)C SP00249 c1c(cc(c(c1Cl)n2c(c(cn2)C#N)N)Cl)C(F)(F)F SEW05022 CSc1c(c(n(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)N)C#N SEW05023 CSc1nc(n(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)N SEW05024 c1ccc(cc1)c2cc(on2)c3ccnn3S(=O)(=O)c4ccc(cc4)Cl SPB05052 c1ccc(c(c1)OCc2nc(cs2)c3cc(no3)c4ccc(c(c4)Cl)Cl)Cl SPB04983 c1cc(ccc1n2c(nnc2SCC#N)c3c(cc(cn3)C(F)(F)F)Cl)Cl SPB05819 c1cc(c(c(c1)Cl)/C=N/O)Cl SPB05820 c1cc(c(cc1F)F)NN=C(C#N)C#N SEW04995 Cc1cc(n(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)C SEW05005 c1cc(cc(c1)F)n2c(=O)[nH]nc2SCC(=O)Nc3cc(cc(c3)Cl)Cl SPB02165 c1cc(cc(c1)F)n2c(=O)[nH]nc2SCC(=O)Nc3ccc(cc3)Cl SPB02166 c1c(cc(cc1Cl)Cl)NC(=O)CSc2nc3c(s2)cc(cc3Cl)Cl SPB02168 CCOC(=O)c1c(c(on1)C)c2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl SPB05048 c1cc(sc1)c2nc(cs2)NC(=O)Nc3ccc(cc3)Cl SPB02196 c1ccc(c(c1)NC(=O)Nc2csc(n2)c3cccs3)Cl SPB02198 CC(C)(C)c1[nH]c(nn1)S SPB00159 CC(C)(C)c1[nH]c(nn1)SCC#C SPB00162 CC(C)(C)c1[nH]c(nn1)SCC=C SPB00163 c1cc(ccc1c2cc(c(o2)C(F)(F)F)COC(=O)Nc3ccc(cc3)OC(F)(F)F)Cl SP00145 c1ccc(cc1)NC(=O)OCc2cc(oc2C(F)(F)F)c3ccc(cc3)Cl SP00146 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NNS(=O)(=O)C SPB02131 Cc1nc(no1)c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F SPB02982 CCOC(=O)c1cnc(nc1Nc2ccccc2)c3cccs3 SPB05875 Cc1c(sc(n1)c2ccc(cn2)C(F)(F)F)C(=O)NN SPB05876 Cc1ccc(cc1)C(=O)C2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05122 CC(=O)OCC(=O)c1ccc(cc1)Br TL00561 Cc1c(sc(n1)c2ccc3c(c2)CCO3)C(=O)Nc4ccccc4 SP00243 Cc1c(sc(n1)c2ccc3c(c2)CCO3)C(=O)Nc4ccc(cc4)OC SP00245 Cc1ccccc1N/C=C(\C#N)/C(=O)c2cc(oc2C)c3ccc(cc3)Cl SP00159 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/c3cccs3)/C#N SP00178 CCOC(=O)c1c(nc(s1)c2ccc(cc2)C(F)(F)F)C SPB03021 c1cc(sc1)C(=O)O/N=C(/c2ccc3c(c2)CCO3)\N SP00190 c1cc(c(cc1C(F)(F)F)Cl)NC(=S)NN SEW05126 CCOC(=O)c1cnc(nc1O)c2cccs2 SPB05859 COc1ccc(cc1I)C(=O)OC TL00305 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnn3S(=O)(=O)c4cccc(c4)C(F)(F)F SPB05013 Cc1cc(c(o1)C(F)(F)F)C(=O)O CC00701 Cc1c(cc(o1)C(C)(C)C)C(=O)/C(=C/Nc2ncccn2)/C#N SP00154 Cc1ccc(cc1)/C=C(\C#N)/C(=O)c2cc(oc2C)c3ccc(cc3)Cl SP00176 c1cc(cc(c1)NC(=O)O/N=C(/c2c(cccc2Cl)Cl)\Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F SPB07166 c1cc(c(c(c1)Cl)/C(=N/OC(=O)c2ccc(cc2)Cl)/Nc3ccc(cc3)OC(F)(F)F)Cl SPB07168 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC(=O)Nc3ccc(c(c3)Cl)F SPB02150 c1cc(ccc1C2NC(=NN2)c3cnccn3)Cl SPB07135 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(F)(F)F SPB05938 CC(C)(C)c1ccc(cc1)OCc2ncc(c(n2)N)S(=O)(=O)c3ccccc3 SPB05978 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4ccccc4Cl SPB05062 CCOC(=O)Cc1n[nH]nn1 SEW05162 c1ccc(cc1)C(C#N)C(C#N)c2ccccc2 SEW05165 c1cc(ccc1C(=O)NCc2ccc3c(c2)CCO3)OC(F)(F)F SP00200 Cc1cc(c(o1)c2ccccc2)/C(=N/OC(=O)c3ccc(cc3)OC(F)(F)F)/N SP00203 CCOC(=O)c1csc(n1)COc2ccccc2Cl SPB02014 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2ncc(s2)c3ccc(cc3)Cl SPB02015 CC(C)c1ccc(cc1)NC(=O)Nc2csc(n2)Cc3c(cccc3Cl)Cl SPB02017 c1cc(ccc1c2cc(c(o2)C(F)(F)F)COC(=O)Nc3ccc(cc3)Cl)Cl SP00143 COc1ccc(cc1)C/N=C/c2ccc(cc2)OC SEW04955 c1ccc(c(c1)C(F)(F)F)n2c(nnc2Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F)O SPB02146 c1ccc(cc1)n2c(=O)[nH]nc2SCC(=O)c3ccc(cc3)Cl SPB02147 Cc1cc(n(n1)C(C)(C)C)C(=O)NNc2cc(ccc2Cl)C(F)(F)F SPB03145 Cc1ccc(cc1)C(=O)O/N=C(/CSc2ccc(cn2)C(F)(F)F)\N SPB03159 c1ccc(cc1)c2cc(on2)c3ccnn3S(=O)(=O)c4ccccc4 SPB05051 Cc1nc(no1)c2ccc3c(c2)CCO3 SP00194 c1cc(ccc1NC(=O)CC23CC4CC(C2)CC(C4)C3)Cl SEW05133 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3ccc(c(c3)Cl)Br SPB03056 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CC45CC6CC(C4)CC(C6)C5)C(F)(F)F SEW05152 COc1ccc(cc1)NC(=O)CC23CC4CC(C2)CC(C4)C3 SEW05153 CCOC(=O)c1ccc(cc1)n2c(c(cn2)C#N)N SEW05155 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)OC(F)(F)F SPB03002 Cc1ccc(cc1)CNc2c(c(nc(n2)C)C)Oc3ccc(cc3Cl)Cl SPB05822 CCOC(=O)CSc1nnc(n1c2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl SPB05823 c1cc(c(c(c1)Cl)CSc2ccc(cc2)OC(F)(F)F)Cl SPB03037 c1cc(c(c(c1)Cl)SCc2nc(no2)c3ccc(cc3)OC(F)(F)F)Cl SPB03040 CCOC(=O)c1c(nn(c1C)c2c(cc(cc2Cl)C(F)(F)F)Cl)C SEW05006 CC(C)S(=O)(=O)c1cnc(nc1N)C(F)(F)F SPB06001 CCC(=O)c1c(cc(cc1OC)OC)C(=O)OC TL00504 c1cc(ccc1S(=O)(=O)NCc2ccc3c(c2)CCO3)Cl SP00198 COC(=O)CCCCCCCC(=O)Nc1nccs1 SEW05138 c1cc(c(nc1)Oc2ccc(cc2)C3=NCCS3)C(F)(F)F SPB03126 c1cc(ccc1C2=NCCS2)Oc3cc(ccn3)C(F)(F)F SPB03127 Cc1ccc(cc1)NC(=O)c2cc(nn2Cc3ccccc3)C(C)(C)C SPB03055 c1cc(sc1)c2nc(sn2)NNC(=O)c3ccc(cc3)Cl SPB07141 c1c(cnc(c1Cl)NN2C3CSC2CS3)C(F)(F)F SPB05944 CC(C)(C)c1csc(n1)c2ccc(nc2)Oc3ccc(cc3)Cl SPB05985 Cc1csc(n1)c2ccc(nc2)Oc3ccc(cc3)Cl SPB05988 Cc1c(c(n(n1)C(=O)c2ccccc2)C)Sc3nnnn3c4ccccc4 SPB05879 c1ccc(cc1)OCC(=S)N SPB05907 CCOC(=O)c1cnc(nc1Sc2ccccc2)c3cccs3 SPB05906 c1cc(ccc1C(=O)N2CCCCC2)F TL00628 CCCCCn1c(nnc1SCc2c(sc(n2)c3ccccc3)C(=O)OCC)O SPB02193 Cc1cc(n(n1)C(C)(C)C)C(=O)O SPB03128 Cc1ccc(cc1)C(=O)C2CCN(CC2)S(=O)(=O)c3ccc(c(c3)Cl)Cl SEW05123 Cc1ccc(cc1)C(=O)C2CCN(CC2)S(=O)(=O)c3c(noc3C)C SEW05124 c1ccc(cc1)C(=O)O/N=C(/c2ccc3c(c2)CCO3)\N SP00189 c1cc(c(cc1C(F)(F)F)Cl)NC(=S)N2CCSCC2 SEW05146 c1cc(ccc1C(F)(F)F)S(=O)(=O)NCc2ccc3c(c2)CCO3 SP00204 Cc1cc(c(o1)C(F)(F)F)C(=O)/C(=C/Nc2ccccc2)/C#N SP00165 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/Nc3ccc(cc3)OC)/C#N SP00171 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)Cl)Sc3ncc(s3)[N+](=O)[O-] SPB07180 Cc1c(cc(o1)C(C)(C)C)C(=O)N SP00074 Cc1cc(c(o1)C(F)(F)F)C(=O)N SP00075 CCOC(=O)c1cc(oc1C)c2ccc(cc2)[N+](=O)[O-] SP00080 CC(=O)c1ccc(s1)C#N TL00354 c1ccc(cc1)c2cc(on2)c3ccnn3C(=O)Nc4cccc(c4)C(F)(F)F SPB05067 c1csc(c1Br)C=C(C#N)C#N SEW05121 Cc1c(c(no1)c2ccccc2)c3csc(n3)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB05022 c1ccc(cc1)C(=N)NC(=O)N2CCOCC2 SPB07195 CC(C)(C)c1ccc(cc1)C(=N)NC(=O)N2CCOCC2 SPB07197 c1cc(cc(c1)Cl)NC(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F SEW05147 c1ccc(cc1)SCC(=N)N.Cl SPB05877 c1cc(ccc1NC(=S)NCc2ccc3c(c2)CCO3)Cl SP00196 Cc1cc(no1)c2nc(no2)c3ccc(cc3)C(C)(C)C SPB03092 Cc1cc(no1)c2nc(no2)c3ccc(cc3)C(F)(F)F SPB03093 Cc1c2cn[nH]c(=O)c2c(n1Cc3cccs3)C SP00127 Cc1c(n(oc1=O)C)C(=O)Nc2ccsc2C(=O)OC SPB02995 CCOC(=O)c1ccc(cc1)Oc2c(cc(cn2)C(F)(F)F)Cl SPB03008 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F SPB03015 Cc1ccccc1NC(=O)NCc2ccc3c(c2)CCO3 SP00212 COc1ccc(cc1)C2(C(=C(N=C(N2)C(F)(F)F)SC)C#N)O SPB05892 CCC(=O)O/N=C(/c1ccc(c(c1)[N+](=O)[O-])Oc2cc(c(c(c2)C)Cl)C)\N SPB02038 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)NNc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl SPB02072 c1cc(sc1)C(=O)NCc2ccc3c(c2)CCO3 SP00201 CSC1=C(C(NC(=N1)C(F)(F)F)(c2cccs2)O)C#N SPB05873 Cc1ccccc1C(=O)NCc2ccc3c(c2)CCO3 SP00202 Cc1cc(c(o1)c2ccccc2)/C(=N/OC(=O)c3cccs3)/N SP00208 Cc1ccccc1C(=O)O/N=C(/c2cc(oc2c3ccccc3)C)\N SP00209 Cc1c(sc(n1)c2ccc(cn2)C(F)(F)F)C(=O)NNS(=O)(=O)c3ccccc3C(F)(F)F SPB05887 c1ccc(cc1)NC(=O)NCc2ccc3c(c2)CCO3 SP00210 CCOC(=O)c1cc(on1)CSc2nnc(n2c3ccccc3C(F)(F)F)O SPB02144 COC(Cn1c(nnc1SCC(=O)c2cccc(c2)C(F)(F)F)c3ccc(cc3)Cl)OC SPB04934 c1cc(c(cc1/C=N/O)Cl)Cl SPB04935 c1ccc(c(c1)/C=N/Nc2nc(cs2)c3cc(no3)c4ccc(cc4Cl)Cl)Cl SPB04938 c1ccc(cc1)c2cc(on2)c3ccnn3C(=O)c4ccc(cc4)C(F)(F)F SPB04962 CC(C)(C)c1ccc(cc1)C(=O)Sc2ccc(cc2)OC(F)(F)F SPB03078 CCOC(=O)c1c(nc(s1)c2ccccc2)CSc3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB02186 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNC(=O)N(C)C SPB00151 c1ccc2c(c1)c(=O)c(=NO)c2=O SPB00184 c1cc(c(c(c1)Cl)/C(=N/O)/N)Cl SPB00002 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(\c3c(cccc3Cl)Cl)/N SPB00005 c1cc(c(cc1C(F)(F)F)Cl)NC(=S)N SEW05128 Cc1nc(cs1)CSc2[nH]c(nn2)c3ccc(cc3)C(C)(C)C SPB02176 CN(C)/C=C/C(=O)c1cc(no1)c2ccc(cc2Cl)Cl SPB05038 c1ccc(cc1)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl SPB05043 c1cc(sc1)c2c3c(nc4c2c(c(s4)C(=O)Nc5cc(cc(c5)C(F)(F)F)C(F)(F)F)N)CCCC3 SPB07084 CC(C)(C)c1ccc(cc1)NC(=O)c2c(c3c(c4c(nc3s2)CCC4)c5cccnc5)N SPB07099 c1cc(sc1)C(=O)NNC(=O)c2csc(n2)COc3ccc(cc3)C4SCCS4 SPB02086 Cc1c(c(no1)c2ccccc2)c3csc(n3)Nc4ccc(cc4)Cl SPB05019 Cc1c(c(no1)c2ccccc2)c3csc(n3)COc4ccc(cc4)Cl SPB05024 Cc1c(c(no1)c2ccccc2)c3csc(n3)N/N=C/c4ccccc4 SPB05030 Cc1c(c(no1)c2ccccc2)c3csc(n3)N/N=C/c4ccccc4Cl SPB05032 CC(C)(C)c1ccc(cc1)OCc2nc(c(c(n2)SC)C#N)n3cccc3 SPB05931 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)C SP00096 Cc1ccc(cc1)SC(=O)c2c(nc(s2)c3ccc(cc3)C(F)(F)F)C SPB03050 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3ccc(cc3)Cl SPB03053 c1cc(ccc1C2SCCS2)OCc3nc(cs3)C(=O)NNC(=O)c4ccc(cc4)Cl SPB02087 Cc1c(n(c(c1S(=O)(=O)C(C)C)N)Cc2cccnc2)C SPB02090 Cc1ccc(cc1)/N=C/c2ccccc2 SEW04902 Cc1csc(c1NS(=O)(=O)c2ccc(cc2)OC(F)(F)F)C(=O)OC SPB02990 c1ccc(cc1)NC(=O)O/N=C(/c2ccc(cc2)OC(F)(F)F)\N SPB03033 c1ccc(cc1)S(=O)(=O)c2cnc(nc2N)COc3ccccc3Cl SPB05977 c1cc(oc1)C(C(=O)c2ccco2)O TL00464 Cc1c(n(oc1=O)C)c2nc(no2)c3ccc(cc3)C(C)(C)C SPB02998 c1cc(ccc1c2nc(on2)CSc3ccc(cc3)Br)OC(F)(F)F SPB03041 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Oc3ccc(cc3)Cl SPB03044 Cc1c(cc(o1)c2ccccc2)C(=O)/C(=C\c3ccc(cc3)[N+](=O)[O-])/C#N SP00226 c1cc(ccc1C(F)(F)F)NC(=S)NCc2ccc3c(c2)CCO3 SP00213 CC(=O)Nc1ccc(cc1[N+](=O)[O-])OC(F)(F)F TL00369 c1ccc(cc1)NC(=O)c2csc(n2)c3ccc4c(c3)CCO4 SP00247 COc1ccc(cc1OC)NC(=O)CCCCCCCC(=O)OC SEW04996 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)Sc2cccc(c2)Br SPB03080 c1ccc(cc1)S(=O)(=O)NCc2ccc3c(c2)CCO3 SP00205 COc1ccc(cc1)c2c(c(nc(n2)COc3ccccc3Cl)SC)C#N SPB05900 CCOC(=O)c1c(nc(s1)c2ccc3c(c2)CCO3)C SP00234 c1cc(cc(c1)NC(=O)NCc2ccc3c(c2)CCO3)C(F)(F)F SP00211 c1c(cc(cc1C(F)(F)F)Nc2nc(cs2)C(F)(F)F)C(F)(F)F SPB05912 Cc1ccc(cc1)Nc2nc(cs2)C(F)(F)F SPB05913 c1ccc(c(c1)/C=N/Nc2nc(cs2)C(F)(F)F)Cl SPB05918 c1cc2c(cc1c3nc(cs3)C(=O)O)CCO2 SP00242 Cc1nc(cs1)CSc2[nH]c(nn2)C(C)(C)C SPB02177 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)C(=O)O SPB02181 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNC(=O)C(C)(C)C SPB03116 COC(=O)c1c(ccs1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB04968 CCc1cc(ccc1NC(=O)C)Br TL00568 c1ccc(c(c1)C(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)O TL00544 c1cc(oc1C=C(C#N)C#N)c2c(cc(cc2Cl)C(F)(F)F)Cl SEW05115 c1ccc2c(c1)/C(=C/c3ccc(o3)c4c(cc(cc4Cl)C(F)(F)F)Cl)/C(=O)N2 SEW05116 CCOC(=O)c1c([nH]c(n1)SCC(=O)Nc2cc(cc(c2)Cl)Cl)C SPB02200 c1cc(c(c(c1)Cl)c2nc(on2)CN3CCOCC3)Cl SPB00093 C/C(=C(\C(=O)C)/Sc1nnc(s1)SC)/O SPB05942 c1cc2c(cc1/C(=N\O)/N)CCO2 SP00107 Cc1ccc(cn1)C(=S)N SPB05963 c1cc(ccc1C(=O)Nc2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl)Cl SPB05966 Cc1ccc(cc1C)c2cc(on2)c3csc(n3)COc4ccc(cc4)Cl SPB04996 CCOC(=O)Nc1ccc(cc1F)F SEW04913 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCC(CC3)C(F)(F)F SPB05951 Cc1c(sc(n1)c2cnccc2C(F)(F)F)C(=O)NN SPB05955 Cc1c(cc(o1)C(C)(C)C)C(=O)/C(=C/Nc2cccc(c2)OC(F)(F)F)/C#N SP00152 c1cc(ccc1C(F)(F)F)NC(=O)N2CCC(CC2)C(F)(F)F SPB05935 Cc1c(cc(o1)c2ccccc2)C(=O)/C=C/N(C)C SP00099 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/Nc3ccc(cc3)Cl)/C#N SP00156 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)c3cnccc3C(F)(F)F SPB06026 CSc1nc(cc(n1)Sc2[nH]c(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Sc4[nH]c(nn4)c5cc(cc(c5)C(F)(F)F)C(F)(F)F SPB07257 c1cc(oc1)CNC(=S)NNC(=O)c2ccc(cc2Cl)Cl SPB06033 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNc3c(cccc3Cl)Cl SPB00192 c1cc(ncc1C(=S)N)OCC(F)(F)F SPB05974 COc1ccc(cc1)CN(Cc2ccc(cc2)OC)C(=O)Nc3ccc(cc3)Cl SEW04989 COc1ccc(cc1)CN(Cc2ccc(cc2)OC)C(=O)c3cccs3 SEW04990 c1cc(cc(c1)F)n2c(=O)[nH]nc2S SPB02162 COC(=O)c1cnn(c1/C=N/NC(=S)Nc2ccc(cc2)Cl)c3ccc(cc3F)F SPB05141 CN(C)N/C(=N\O)/c1c(cccc1Cl)F SPB00107 CC(C)c1ccc(cc1)NC(=O)c2csc(n2)c3cccc(c3Cl)Cl SPB02189 CSc1nc(cc(n1)Sc2nnc(n2c3cccc(c3)C(F)(F)F)O)Sc4nnc(n4c5cccc(c5)C(F)(F)F)O SPB07259 c1ccc(cc1)CSc2nnc(s2)c3cnccn3 SPB07296 c1cc(ccc1N/N=C/c2ccc(o2)c3cc(ccc3Cl)C(F)(F)F)F SEW05257 c1cc(ccc1c2csc(n2)c3cnccc3C(F)(F)F)/C(=N/OC(=O)c4ccc(cc4)Cl)/N SPB05958 Cc1c(c(on1)C(F)(F)F)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N SEW05141 CC(C)C(=O)NNC(=O)c1csc(n1)c2c(cc(cn2)C(F)(F)F)Cl SPB05962 CCC(=O)Nc1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05964 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)OC SPB02201 COc1cc(cc(c1OC)OC)CNCc2cc(c(c(c2)OC)OC)OC SEW04993 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)N/N=C/c4ccccc4 SPB05063 c1c(cc(c(c1Cl)NN=C2C(=O)CCCC2=O)Cl)C(F)(F)F SEW05093 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB02190 c1cc(sc1)c2nc(cs2)NC(=O)Nc3ccc(cc3F)F SPB02197 CC(C)c1ccc(cc1)NC(=O)Nc2csc(n2)c3cccs3 SPB02199 Cc1nc(no1)c2ccc(cc2)c3csc(n3)c4cnccc4C(F)(F)F SPB05960 c1cc(ccc1c2cc(on2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl)Cl SPB05090 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)Nc2csc(n2)c3cccc(c3Cl)Cl)/N SPB02203 C#CCSc1nccc(n1)c2cc(no2)c3ccc(cc3Cl)Cl SPB05077 COC(c1c(cc(c(n1)SCC(=O)c2ccc(cc2)Cl)C#N)C(=O)OC)OC SPB05106 CC\1=NN(C(=O)/C1=N\Nc2c(cc(cc2Cl)C(F)(F)F)Cl)C SEW05094 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)COc4ccccc4 SPB05064 Cc1c(cc(o1)C(C)(C)C)C(=O)/C(=C/Nc2ccccc2)/C#N SP00149 Cc1ccccc1N/C=C(\C#N)/C(=O)c2cc(oc2C)C(C)(C)C SP00150 c1ccc(c(c1)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl)Cl SPB05085 c1ccc(c(c1)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(F)(F)F)Cl SPB05087 c1ccc(cc1)n2c(nnc2SCC(=O)N3CCC(CC3)C(F)(F)F)O SPB07229 COC(Cn1c(nnc1SCC(=O)Nc2ccc(cc2)C(F)(F)F)c3ccccc3)OC SPB05099 COC(c1c(cc(c(n1)SCC(=O)Nc2ccccc2)C#N)C(=O)OC)OC SPB05102 Cc1c(cc(o1)c2ccccc2)C(=O)/C(=C\c3cccc(c3)OC)/C#N SP00229 CC(C)(C)C(=O)CSc1c(cc(c(n1)C(OC)OC)C(=O)OC)C#N SPB05107 CCOC(=O)c1c(c(nc(n1)C)Sc2ccc(cc2)Cl)C SPB07208 c1ccc(cc1)NC(=O)Nc2ccccc2Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N SPB07237 c1ccc(cc1)NC(=O)O/N=C(/c2c(cccc2Cl)Cl)\Nc3ccc(cc3)OC(F)(F)F SPB07164 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)NN SPB03030 c1cc(cc(c1)n2c(nnc2SCC(=O)N3CCC(CC3)C(F)(F)F)O)C(F)(F)F SPB07231 CCCCCn1c(nnc1SCC(=O)N2CCC(CC2)C(F)(F)F)O SPB07232 Cc1c(cc(o1)c2ccccc2)C(=O)/C(=C\c3ccc(cc3)OC(F)(F)F)/C#N SP00220 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N SPB07233 CSc1nc(cc(n1)Sc2[nH]c(nn2)c3ccccc3)Sc4[nH]c(nn4)c5ccccc5 SPB07246 Cc1c(c(no1)c2c(cccc2Cl)Cl)N(C)C(=O)N3CCOCC3 SPB00047 Cc1cc2c(c(n1)Sc3ccc(cc3)Cl)C(=O)N(C2=O)SC(Cl)(Cl)Cl SPB00049 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cc(no3)c4ccccc4 SPB05045 c1cc(ccc1C(=O)Sc2ccc(cc2)OC(F)(F)F)C(F)(F)F SPB03077 Cc1cc(no1)NC(=O)CCCCCCCC(=O)OC SEW05137 CC(C)(C)c1nc2n(n1)c(cs2)c3ccc(cc3)Cl SPB00165 CCOC(=O)NNC(=S)Nc1cccc(c1)F SPB02159 CSc1nc(cc(n1)Sc2nnc(n2c3ccc(cc3)Cl)O)Sc4nnc(n4c5ccc(cc5)Cl)O SPB07243 CCOC(=O)c1c(c(nc(n1)C)Sc2ccccc2)C SPB07209 c1cc(ccc1C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)Cl SPB07281 c1cc(ccc1NC(=O)CSc2nc3c(s2)cc(cc3Cl)Cl)Cl SPB02167 Cc1nc(cs1)CSc2nnc(n2c3cccc(c3)F)O SPB02173 CC(C)(C)C(=O)O/N=C(/c1c(cccc1Cl)Cl)\Nc2ccc(cc2)OC(F)(F)F SPB07170 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)c3cnccc3C(F)(F)F SPB06027 CC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F TL00622 Cc1cc(no1)c2nnc(o2)c3cccc(c3)C(F)(F)F SPB03162 CCOC(=O)c1c(nc(s1)c2ccccc2)CSc3ccc(cc3)Cl SPB02160 c1cc(ncc1C(F)(F)F)Sc2[nH]c(nn2)C(F)(F)F SPB03179 c1cnc(cc1C(F)(F)F)Sc2[nH]c(nn2)C(F)(F)F SPB03180 CC(C)(C)c1cc(n(n1)C)C(=O)NNC(=O)c2cccc(c2)Cl SPB03166 CC(C)(C)c1cc(n(n1)C)C(=O)NNC(=O)c2ccccc2Cl SPB03167 c1ccc(cc1)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl SPB05044 CC(C)NC(=O)n1c(ccn1)c2cc(no2)c3ccccc3 SPB05071 c1cc(c(c(c1)Cl)/C(=N/OC(=O)Nc2ccc(cc2)Cl)/Nc3ccc(cc3)OC(F)(F)F)Cl SPB07165 COc1ccc(cc1)NC(=O)O/N=C(/c2c(cccc2Cl)Cl)\Nc3ccc(cc3)OC(F)(F)F SPB07167 c1cc(c(cc1C(F)(F)F)Cl)NC(=S)Nc2ccc(cc2Cl)C(F)(F)F SEW05143 Cn1c(nnc1SCC(=O)Nc2cccc(c2)Cl)C(F)(F)F SPB02151 Cc1c(sc(n1)c2cccnc2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB02183 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)C(=C3SCCS3)C#N SP00173 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/c3ccc(cc3)Cl)/C#N SP00174 Cc1c(c(no1)c2ccccc2)c3ccnn3S(=O)(=O)c4ccc(cc4)Cl SPB05017 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)N/N=C/c4ccccc4Cl SPB05065 c1cc(c(nc1)Sc2[nH]c(nn2)C(F)(F)F)C(F)(F)F SPB03181 c1ccc(cc1)c2cc(on2)c3ccnn3C(=O)Nc4ccccc4 SPB05070 CCOC(=O)c1cnc(nc1NNC(=O)C)c2cccs2 SPB06017 CCOC(=O)c1cnc(nc1NNC(=O)c2ccc(cc2)Cl)c3cccs3 SPB06018 c1cc(c(cc1Cl)Cl)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl SPB05074 Cc1cc(c(cc1Cl)C)S(=O)(=O)Cc2nc(no2)COc3c(cccc3Cl)Cl SPB03187 CSc1c(c(nc(n1)C(F)(F)F)N)C#N SPB06023 c1ccc(cc1)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(F)(F)F SPB05046 c1cc(ncc1C(F)(F)F)n2cncn2 SPB03171 c1cc(c(nc1)n2cncn2)C(F)(F)F SPB03172 c1cc(ccc1C(F)(F)F)NC(=O)CSc2nccc(n2)c3cc(no3)c4ccc(cc4Cl)Cl SPB05075 c1cc(ccc1/C(=N/OC(=O)N2CCOCC2)/N)Cl SPB07191 Cc1cc(no1)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N SPB03085 c1cc(c(c(c1)Cl)/C(=N/OC(=O)N2CCOCC2)/N)Cl SPB07194 c1ccc(c(c1)C(=N)NC(=O)N2CCOCC2)OC(F)(F)F SPB07196 COc1c(cc(cc1Br)C#N)Br SPB00194 c1ccc(c(c1)c2ccc(cc2)C(=O)Nc3cccc(c3)C(F)(F)F)F SEW05258 c1cc(c(c(c1)F)NC(=O)CC23CC4CC(C2)CC(C4)C3)F SEW05144 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)C)NC(=O)c3ccccc3 SP00233 c1cc(ccc1C(=O)CSc2nnc(s2)c3cnccn3)Cl SPB07301 Cc1cccc(c1)NC(=O)N/N=C(/c2cnccn2)\N SPB07266 CCOC(=O)c1csc(n1)c2ccc3c(c2)CCO3 SP00235 Cc1c(cc(o1)C(C)(C)C)c2cc([nH]n2)NS(=O)(=O)c3ccc(cc3)Cl SP00238 c1cc(oc1c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Oc4cc(cc(c4)Cl)Cl SPB03138 CCOC(=O)c1c(c(nc(c1Cl)C(C)(C)C)Sc2ccccc2)C#N SPB00053 Cc1cc(no1)C(=O)O/N=C(/c2ccc(o2)[N+](=O)[O-])\N SPB03086 c1cc(cc(c1)Cl)CNC(=O)CC23CC4CC(C2)CC(C4)C3 SEW05157 Cc1cc(n(n1)C(C)(C)C)C(=O)Oc2cccc(c2)C(F)(F)F SPB03141 Cc1ccc(cc1)c2csc(n2)c3ccc(nc3)Oc4ccc(cc4)Cl SPB05984 c1ccc(c(c1)c2ccc(cc2)C(=O)Nc3ccc(cc3)Cl)F SEW05259 c1ccc(c(c1)NC(=O)Nc2cccc(c2)C(F)(F)F)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N SPB07239 C/C(=N\NC(=S)NC(C)(C)C)/c1ccc(cc1)Oc2ncc(s2)[N+](=O)[O-] SPB07241 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC(C)C SPB00062 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N3CCCCC3 SPB00063 c1ccc(cc1)S(=O)(=O)N/N=C(/c2cnccn2)\N SPB07273 c1cnc(cn1)c2nnc(s2)SCC(=O)Nc3cc(cc(c3)Cl)Cl SPB07306 CC/C(=N\Nc1ccc(cc1)[N+](=O)[O-])/c2ccc(cc2)c3ccccc3F SEW05260 Cc1c(nc(s1)Nc2ccccc2)c3ccc(cc3)c4ccccc4F SEW05262 CC(C)(C)c1cc(n(n1)C)C(=O)Sc2cccc(c2)C(F)(F)F SPB03151 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccc(cc3)Cl SPB00067 c1cc(ccc1N/N=C/2\CCSc3c2cc(cc3)Cl)[N+](=O)[O-] SEW05168 c1ccc(c(c1)NC(=S)NCc2ccc3c(c2)CCO3)OC(F)(F)F SP00215 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)C)N SP00217 Cc1ccc(cc1)N/C=C(/C#N)\C(=O)c2cc(oc2C)c3ccccc3 SP00219 Cc1c(cnc(n1)COc2ccc(cc2)C(C)(C)C)S(=O)(=O)c3ccc(cc3)Cl SPB06044 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N3CCOCC3 SPB00064 CCN(c1ccccc1)C(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C SPB00065 CC(C)(C)c1cc(n(n1)C)C(=O)O SPB03149 Cc1c(c(no1)c2c(cccc2Cl)Cl)N(C)C(=O)N3CCCCC3 SPB00070 CC(C)NC(=O)Nc1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05981 CC(=O)Cn1c2ccccc2oc1=O SPB03221 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4ccc(cc4)C(F)(F)F SPB05007 c1cc(oc1)CNC(=S)NN SPB07149 CCOC(=O)CSc1c(n2ccsc2n1)/C=N/c3ccc(cc3)Cl SPB06045 c1cc(sc1)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 SPB07283 CC(C)(C)c1[nH]c(nn1)SCC(=O)c2ccc(cc2)[N+](=O)[O-] SPB00167 CC(C)S(=O)(=O)c1cnc(nc1N)COc2ccc(cc2)C(C)(C)C SPB05996 Cc1cc(no1)c2c(c(no2)C)C(=O)OC SPB03204 Cc1ccc(cc1)NC(=O)c2c(noc2c3cc(on3)C)C SPB03214 Cc1cc(no1)c2c(c(no2)C)C(=O)Nc3ccc(cc3)C(F)(F)F SPB03215 Cn1c(nnc1SC)c2ccccc2 SPB06057 c1ccc(c(c1)C(F)(F)F)n2c(nnc2Sc3ccc(cn3)C(F)(F)F)O SPB03224 CCOC(=O)c1ccc(cc1)N2C(=O)CC(=N2)C SEW05156 c1cc(ccc1N/N=C/c2ccc(o2)c3cc(ccc3Cl)C(F)(F)F)[N+](=O)[O-] SEW05256 Cc1cc(n(n1)C(C)(C)C)C(=O)NNc2ccc(cc2)C(C)C SPB03147 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cc(no3)c4ccccc4Cl SPB05086 c1cc(cc(c1)[N+](=O)[O-])NC(=O)c2csc(n2)c3ccc4c(c3)CCO4 SP00254 COc1c(cccn1)[N+](=O)[O-] SPB06058 Cc1c(cnn1CCC#N)Sc2ccc(cc2)Cl SPB06059 COC(c1c(cc(c(n1)SCC(=O)Nc2cc(cc(c2)Cl)Cl)C#N)C(=O)OC)OC SPB05104 CC(=O)Nc1ccc(cc1)OC(F)(F)F TL00595 c1cc(ccc1NC(=O)CSc2nccc(n2)c3cc(no3)c4ccc(cc4Cl)Cl)Cl SPB05076 c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cc(no3)c4ccc(cc4)Cl SPB05079 Cc1c2cn[nH]c(=O)c2c([nH]1)C SP00122 c1ccc(cc1)C(=O)NCc2ccc3c(c2)CCO3 SP00197 c1cc(ccc1NC(=O)NCc2ccc3c(c2)CCO3)Cl SP00199 CC(C)(C)c1ccc(cc1)OCc2nc(c(c(n2)SC)C#N)c3ccc(cc3)Cl SPB05899 Cc1c(cc(o1)c2ccccc2)C(=O)/C(=C\c3ccc(cc3)Cl)/C#N SP00227 Cc1c(cc(o1)c2ccccc2)C(=O)/C(=C\c3ccccc3[N+](=O)[O-])/C#N SP00228 c1ccc(c(c1)c2cc(on2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl)Cl SPB05089 CC(C)(C)c1ccc(cc1)c2[nH]c(nn2)SC SPB00120 CC(C)(C)c1ccc(cc1)c2[nH]c(nn2)SCC(=O)c3ccc(cc3)Cl SPB00122 c1ccc(cc1)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 SPB07289 c1cc(cc(c1)Cl)NC(=O)O/N=C(/c2ccno2)\N SPB03272 Cc1ccc(cc1)CSc2nnc(s2)c3cnccn3 SPB07297 c1cc(ccc1NC(=O)N/N=C(/c2cnccn2)\N)Cl SPB07265 Cc1cc2c(c(n1)Sc3ccc(cc3)Cl)C(=O)N(C2=O)Cc4ccc(cc4Cl)Cl SPB00048 CCOC(=O)c1c(c(nc(c1Cl)C(C)(C)C)Sc2ccccn2)C#N SPB00056 COC(c1c(cc(c(n1)SCC(=O)Nc2ccc(cc2)Cl)C#N)C(=O)OC)OC SPB05103 Cc1c(cc(o1)C(C)(C)C)c2cc([nH]n2)NC(=O)c3ccc(cc3)[N+](=O)[O-] SP00230 Cc1ccc(cc1)SC(=O)c2cc(on2)C SPB03096 c1cc(ccc1NC(=O)c2csc(n2)c3ccc4c(c3)CCO4)Cl SP00253 c1cc(c(=O)n(c1)CCC#N)C(F)(F)F SPB06060 COC(Cn1c(nnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)c3ccccc3)OC SPB05092 C#CCSc1nccc(n1)c2cc(no2)c3ccc(cc3)Cl SPB05100 C/C(=N\OC(=O)Nc1ccccc1)/Cn2c3ccccc3oc2=O SPB03244 CCc1nnc(s1)NS(=O)(=O)c2ccc(cc2)OC(F)(F)F SPB03246 CCOC(=O)c1cc(nc(c1C#N)Sc2ccc(cc2)Cl)c3ccc(cc3)Cl SPB00029 Cc1cc(no1)c2c(c(no2)C)C(=O)Sc3c(cccc3Cl)Cl SPB03254 Cc1cccc(c1NC(=O)NNC(=O)c2cc(nn2Cc3ccccc3)C(C)(C)C)C SPB03119 Cc1c(cc(o1)C(C)(C)C)C(=O)/C(=C/Nc2ccc(cc2)Cl)/C#N SP00148 c1cc(ccc1n2c(nnc2S)c3cnccc3C(F)(F)F)Cl SPB06016 c1cc(c(c(c1)Cl)c2nc(on2)CN3CCCCC3)Cl SPB00094 Cc1cc(no1)c2nnc(o2)c3cccc(c3)Cl SPB03161 c1ccc2c(c1)n(c(=O)o2)CC(=O)c3ccc(cc3)Cl SPB03165 c1ccc(cc1)C(=O)Cn2c3ccccc3oc2=O SPB03169 Cc1ccc(cc1)SC(=O)c2ccno2 SPB03178 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)N SPB03182 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNC(=O)Nc3cccc(c3)Cl SPB03120 Cc1[nH]c(c(c1/C=N/N=C/c2c(c([nH]c2C)C)C(=O)OC)C(=O)OC)C SP00123 Cc1c2cnn(c(=O)c2c([nH]1)C)Cc3ccc(cc3)Cl SP00124 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)O SPB03027 c1cc(cc(c1)Cl)NC(=O)O/N=C(/c2ccc(nc2)Oc3ccc(cc3)Cl)\N SPB05971 c1cc(ccc1NC(=O)N/N=C(/c2cnccn2)\N)OC(F)(F)F SPB07267 c1cc(ccc1S(=O)(=O)N/N=C(/c2cnccn2)\N)Cl SPB07272 c1ccc(c(c1)/C=N/NC(=O)c2nc(no2)c3ccc(cc3)OC(F)(F)F)Cl SPB03240 CC(=O)c1ccc(o1)c2ccccc2OC(F)(F)F SEW05203 CC(=O)N/N=C\1/c2cc(ccc2NC1=O)F SEW05213 c1ccc(cc1)NC(=O)NNC(=O)c2nc(no2)c3ccc(cc3)OC(F)(F)F SPB03243 c1cc(ccc1SCC(=N)N)Cl.Cl SPB06092 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNC(=O)Nc3cccc(c3)C(F)(F)F SPB03121 CC(C)(C)c1ccc(cc1)c2[nH]c(nn2)Sc3cc(nc(n3)SC)Sc4[nH]c(nn4)c5ccc(cc5)C(C)(C)C SPB07258 c1cc(sc1)c2[nH]c(nn2)SCC(=O)c3ccc(cc3)Cl SPB00139 c1ccc(c(c1)c2ccc(o2)/C=C/3\CSc4ccc(cc4C3=O)Cl)OC(F)(F)F SEW05190 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)NC(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N SPB02205 Cc1ccc(cc1)SCc2nc(nc(n2)SC)N SPB06116 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB02208 CCOC(=O)c1csc(n1)COc2ccc(cc2)OC SPB02212 c1cc(ccc1CC#N)Oc2ccc(cn2)C(F)(F)F SPB03122 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)C(F)(F)F SPB02153 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB05078 Cc1ccc(cc1)SC(=O)CCn2cccc(c2=O)C(F)(F)F SPB06111 c1cc(c(=O)n(c1)CCC(=O)Sc2ccc(cc2)Cl)C(F)(F)F SPB06112 CSc1nc(nc(n1)N)CSc2ccc(cc2)Cl SPB06114 COC(c1c(cc(c(n1)SCC#C)C#N)C(=O)OC)OC SPB05114 Cc1ccc(cc1)C(=O)CSc2nnc(n2C)C(F)(F)F SPB00208 Cn1c(nnc1SC(=O)Cc2cccc(c2)[N+](=O)[O-])C(F)(F)F SPB00210 COC(c1c(cc(c(n1)Sc2ncc(s2)[N+](=O)[O-])C#N)C(=O)OC)OC SPB05131 c1ccc2cc(ccc2c1)C(=O)CSc3[nH]c(nn3)C(F)(F)F SPB00211 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cc(no3)c4ccc(cc4)Cl SPB05081 c1cc(ccc1Oc2ccc(cn2)C(=S)N)Cl SPB05973 COC(c1c(cc(c(n1)Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C#N)C(=O)OC)OC SPB05119 CC(C)(C)c1ccc(cc1)C(=O)NNC(=S)Nc2ccc(cc2)Cl SPB00258 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc(cc3)Cl)S SPB00263 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc(cc3)Cl)SCC=C SPB00266 CCOC(=O)c1c(c(=O)[nH]c(n1)COc2ccccc2Cl)C SPB07214 C/C(=N\OC(=O)c1ccc(cc1)C(C)(C)C)/Cn2c3ccccc3oc2=O SPB03279 c1ccc(cc1)NC(=O)CSc2nnc(s2)c3cnccn3 SPB07308 CC(C)(C)c1ccc(cc1)NC(=O)CSc2nnc(s2)c3cnccn3 SPB07309 C/C(=N\Nc1cc(ccn1)C(F)(F)F)/c2ccc(cc2)Oc3ncc(s3)[N+](=O)[O-] SPB07216 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc(cc3)Cl)SCC#C SPB00267 Cc1ccc(cc1)/C(=N/OC(=O)c2c(nc(s2)C)C(F)(F)F)/N SPB07345 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNc3c(cc(cc3Cl)Cl)Cl SPB00272 Cc1ccc(cc1)C(=O)Nc2ccccc2Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N SPB07234 c1ccc(c(c1)NC(=O)c2cccs2)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N SPB07235 CCC(=O)Nc1ccccc1Sc2c(c(cc(n2)c3cccs3)C(F)(F)F)C#N SPB07236 c1cc2c(cc1F)/C(=N/Nc3ccc(cc3Cl)Cl)/C(=O)N2 SEW05214 CCOC(=O)c1csc(n1)c2ccc(cc2F)F SPB02254 Cc1c(sc(n1)c2cccs2)C(=O)NNC(=O)Nc3ccc(cc3)Cl SPB02261 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)c4ccc(cc4)[N+](=O)[O-] SPB05193 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SC SPB05194 c1ccc(c(c1)C(=O)O/N=C(/c2c(cccc2Cl)Cl)\Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F SPB07169 COC(=O)C/C(=N/Nc1c(cc(cc1Cl)C(F)(F)F)Cl)/C(=O)OC SEW05104 CCCCCn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)O SPB02154 c1cc(ccc1n2c(nnc2SCC(=O)N3CCC(CC3)C(F)(F)F)O)Cl SPB07230 CC/C(=N\OC(=O)CC12CC3CC(C1)CC(C3)C2)/c4ccc(cc4)c5ccccc5F SEW05237 Cc1c(n(c(c1S(=O)(=O)c2ccccn2)N)Cc3cccc(c3)Cl)C SPB02242 Cc1c(sc(n1)c2cccs2)C(=O)NNC(=O)c3ccc(cc3)Cl SPB02251 c1cc(ccc1/C(=N/OC(=O)Nc2ccc(cc2)Cl)/N)OCc3c(cc(cn3)C(F)(F)F)Cl SPB05172 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(F)(F)F SPB05187 Cc1ccc(cc1)S(=O)(=O)N/N=C(/c2cnccn2)\N SPB07274 c1ccc(c(c1)OC(F)(F)F)S(=O)(=O)N/N=C(/c2cnccn2)\N SPB07275 c1ccc(c(c1)c2ccc(cc2)C(=O)O)F SEW05200 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(C)C SPB00060 CCCCCn1c(nnc1SCC(=O)Nc2ccc(cc2)C(C)C)O SPB02155 CCOC(=O)c1c(c(nc(c1Cl)C(C)(C)C)Sc2ccc(cc2)C)C#N SPB00054 CCOC(=O)c1c(c(nc(c1Cl)C(C)(C)C)N2CCOCC2)C#N SPB00057 Cc1cc(n(n1)C(C)(C)C)C(=O)Oc2cccc(c2)Cl SPB03140 Cc1cc(n(n1)C(C)(C)C)C(=O)NNc2c(cccc2Cl)Cl SPB03146 CCOC(=O)c1c(nc(s1)c2cccs2)C SPB02246 c1cc(cc(c1)NC(=O)Cc2cc(sc2Br)Br)C(F)(F)F SPB02294 COC(=O)c1cnn(c1/C=N/NC(=S)N)c2ccc(cc2)Cl SPB05156 COc1ccc(cc1[N+](=O)[O-])C(=S)N SPB07324 COC(c1c(cc2c(c(sc2n1)C(=O)c3ccccc3)N)C(=O)OC)OC SPB05162 Cc1ccc(cc1F)/C(=N/O)/N SPB07338 Cc1nc(c(s1)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F SPB07348 Cc1ccc(cc1)NC(=O)CCn2cccc(c2=O)C(F)(F)F SPB06095 c1cc(ccc1/C(=N/OC(=O)c2ccc(nc2)OCC(F)(F)F)/N)OC(F)(F)F SPB06100 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)Cl)Sc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N SPB07238 c1cc2c(cc1F)C(=O)CCS2 SEW05178 c1ccc(cc1)c2cc(on2)c3ccnn3C(=O)c4ccno4 SPB05050 c1ccc(cc1)c2cc(on2)c3ccnn3S(=O)(=O)c4ccc(cc4)C(F)(F)F SPB05053 c1ccc(cc1)c2cc(on2)c3ccnn3S(=O)(=O)c4ccccc4Cl SPB05055 c1cc(ccc1SC(=O)c2ccno2)Cl SPB03176 c1ccc(cc1)SC(=O)c2ccno2 SPB03177 c1cc(ccc1NC(=S)N/N=C/c2c(cc(cn2)C(F)(F)F)Sc3ccc(cc3)Cl)Cl SPB06010 COC(=O)c1cnn(c1/C=N/NC(=S)Nc2ccccc2)c3ccc(cc3)Cl SPB05158 Cc1cc(no1)c2c(c(nn2c3cccc(c3)C(F)(F)F)C)C(=O)N4CCOCC4 SPB05209 c1cc(ccc1C(=O)CSc2nnc(o2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F)Cl SPB03390 Cc1cc(nn1c2c(cccc2Cl)Cl)C(=O)NNc3c(cccc3Cl)Cl SPB00297 Cc1cc(nn1c2c(cccc2Cl)Cl)NC(=O)NN3CCOCC3 SPB00301 Cc1nc(c(s1)C(=O)NNc2c(cc(cn2)Cl)C(F)(F)F)C(F)(F)F SPB07349 Cc1nc(c(s1)C(=O)NNc2cccc(n2)C(F)(F)F)C(F)(F)F SPB07350 Cc1ccc(cc1F)C(=N)N.Cl SPB07361 c1cc(ccc1c2csc(n2)c3ccc(nc3)n4cncn4)Cl SPB07278 c1cc(cc(c1)C(F)(F)F)c2csc(n2)c3ccc(nc3)n4cncn4 SPB07279 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)Cl SPB07365 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccc(cc3)C#N SPB07366 COc1ccc(cc1)OCc2ncc(s2)c3ccc4c(c3)OCCCO4 SPB07369 c1ccc(c(c1)NC(=O)Nc2cccc(c2)C(F)(F)F)Sc3ncc(s3)[N+](=O)[O-] SPB07181 c1ccc(cc1)S(=O)(=O)N/N=C/c2c(cc(cn2)C(F)(F)F)Sc3ccc(cc3)Cl SPB06013 Cc1ccc(cc1)CSc2nnc(n2C)c3csc(n3)C SPB02309 c1ccc(c(c1)C(=O)NNC(=O)Cn2nc(nn2)c3cccs3)Cl SPB02317 Cc1cccc(c1NC(=O)NNC(=O)c2c(c(on2)C)c3csc(n3)C)C SPB03397 CN(C)S(=O)(=O)Oc1cccc(c1OS(=O)(=O)N(C)C)F SEW05247 CC/C(=N\OC(=O)Nc1cc(cc(c1)Cl)Cl)/c2ccc(cc2)c3ccccc3F SEW05250 c1cc2c(cc1F)/C(=N/NC(=S)N)/C(=O)N2 SEW05220 Cc1c(sc(n1)c2cccs2)NC(=O)Nc3ccc(cc3)Cl SPB02270 Cc1c(c(on1)c2ccc(cc2)C(F)(F)F)C(=O)NNC(=O)Nc3ccc(cc3)Cl SPB02272 Cc1c(c(on1)c2ccc(cc2)C(F)(F)F)NC(=O)Nc3cc(cc(c3)Cl)Cl SPB02277 CC(C)(C)C(=O)N(Cc1ccc(cc1)OC)Cc2cc(c(c(c2)OC)OC)OC SEW05222 CSc1nc(cc(n1)Sc2nnc(n2c3ccccc3)O)Sc4nnc(n4c5ccccc5)O SPB07244 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SC SPB00245 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC=C SPB00246 Cc1ccc(cc1)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 SPB07282 c1ccc(c(c1)C(F)(F)F)n2c(nnc2Sc3c(cccn3)C(F)(F)F)O SPB03222 c1ccc(cc1)N/N=C\2/c3cc(ccc3NC2=O)F SEW05210 Cc1ccc(cc1)N/N=C\2/c3cc(ccc3NC2=O)F SEW05211 c1cc2c(cc1F)/C(=N/NC(=S)NC3CC4CC3C=C4)/C(=O)N2 SEW05212 CC1(OC(=O)C(=Cc2ccc(o2)c3cc(ccc3Cl)C(F)(F)F)C(=O)O1)C SEW05182 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)NC(=O)OCc3cc(cc(c3)Cl)Cl SPB02207 CCOC(=O)c1csc(n1)CS(=O)(=O)Cc2cccc(c2)C(F)(F)F SPB02224 CSc1nnc(s1)SCc2nc(cs2)c3ccc(cc3)[N+](=O)[O-] SPB02226 c1cc(ccc1c2cc(on2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(F)(F)F)Cl SPB05080 c1cc(sc1)C(=O)NNC(=S)N SPB00116 CC(C)(C)c1ccc(cc1)c2[nH]c(nn2)SCC#C SPB00118 c1cc(c(c(c1)Cl)OCc2nc(on2)CS(=O)(=O)c3ccc(cc3)Cl)Cl SPB03188 Cc1nnc(s1)NS(=O)(=O)c2ccc(cc2)OC(F)(F)F SPB03227 Cc1c(c(n(n1)C(C)(C)C)C(=O)Sc2cccc(c2)C(F)(F)F)Br SPB03228 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)NC(=O)O/N=C(/c3ccc(cc3)Cl)\N SPB02204 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)NN SPB02206 c1cc(ccc1c2csc(n2)c3cnccc3C(F)(F)F)/C(=N/OC(=O)Nc4ccc(cc4)Cl)/N SPB06049 CN(C)/C=C(\C#N)/c1ccc(cc1)Oc2ccc(cn2)C(F)(F)F SPB03232 CNC(=S)NNC(=O)c1ccccc1 SPB06035 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)NNC(=O)c3ccccc3Cl SPB02209 Cc1c(c(on1)c2ccc(cc2)C(F)(F)F)C(=O)NN SPB02211 Cn1c(nnc1SC)c2ccc(cc2Cl)Cl SPB06054 CC(=O)Nc1ccccc1[N+](=O)[O-] TL00610 COC(=O)c1cnn(c1/C=N/NC(=S)Nc2ccccc2)c3ccccc3 SPB05125 COC(=O)c1cnn(c1/C=N/NC(=S)Nc2ccc(cc2)Cl)c3ccccc3 SPB05126 Cc1cc(no1)C(=O)/C(=C(\C)/NC)/C(=O)OC SPB03189 c1cc(c(nc1)Sc2nnc(n2C3CCCCC3)O)C(F)(F)F SPB03195 c1cc(ncc1C(F)(F)F)Sc2nnc(n2C3CCCCC3)O SPB03197 c1cc(ccc1c2csc(n2)c3ccc(nc3)Oc4ccc(cc4)Cl)Cl SPB05983 CC(=O)Nc1ccc(cc1)OCC=C TL00510 Cc1ccc(cc1)c2nnc(n2C)S SPB06051 CC(C)(C)c1csc(n1)CS(=O)(=O)c2ccccn2 SPB02232 COC(c1c(cc(c(n1)SCC=C)C#N)C(=O)OC)OC SPB05116 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccccc3)SC SPB06053 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N/N=C/2\CCSc3c2cc(cc3)F SEW05299 CSc1nnc(n1Cc2ccco2)c3ccc(cc3Cl)Cl SPB06055 COC(c1c(cc(c(n1)SCc2ccc(cc2)Cl)C#N)C(=O)OC)OC SPB05118 CC(C)(C)NC(=S)N/N=C/c1c(cnn1c2ccccc2)C(=O)OC SPB05124 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3cc(c(c(c3)Br)OC)Br)\N SPB00199 c1ccc(cc1)NC(=O)O/N=C(/c2ccno2)\N SPB03271 CSc1cccc(c1)NC(=O)c2c(c3c(cc(nc3s2)c4cccs4)C(F)(F)F)N SPB07247 Cn1c(nnc1S)c2ccc(cc2Cl)Cl SPB06041 CCOC(=O)c1ccc(cc1)n2c(cc(n2)C)C SEW05154 c1cc2c(cc1F)/C(=N/Nc3c(cc(cn3)C(F)(F)F)Cl)/CCS2 SEW05300 c1cc2c(cc1F)/C(=N/NC(=S)NCC3CCCO3)/CCS2 SEW05301 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(C(C)C)C(C)C SPB00072 Cc1c(nc(s1)C)c2ccc(cc2)c3ccccc3F SEW05228 CC(C)(C)c1[nH]c(nn1)Sc2ccc(cn2)C(F)(F)F SPB03190 Cc1c(c(on1)c2ccno2)C(=O)OC SPB03206 c1ccc(c(c1)c2ccc(o2)/C=N/O)OC(F)(F)F SEW05191 CC(=O)c1ccc(o1)c2cc(ccc2Cl)C(F)(F)F SEW05192 c1cc(cc(c1)Cl)NC(=O)NNC(=O)c2nc(no2)c3ccc(cc3)OC(F)(F)F SPB03242 C1COCCN1C(=O)CC23CC4CC(C2)CC(C4)C3 SEW05159 COC(=O)Nc1cc(cc(c1)Cl)Cl TL00611 c1csc(n1)NC(=O)CC23CC4CC(C2)CC(C4)C3 SEW05164 COC(=O)C(=Cc1ccc(o1)c2cc(ccc2Cl)C(F)(F)F)C(=O)OC SEW05180 Cc1ccc(cc1)c2cc(c3cc(ccc3n2)F)C(=O)N SEW05223 c1cc(c(cc1C(F)(F)F)c2ccc(o2)C(C3C(=O)CCCC3=O)C4C(=O)CCCC4=O)Cl SEW05185 Cc1c(n(c(c1S(=O)(=O)c2ccccn2)N)Cc3ccc(cc3)C(F)(F)F)C SPB02245 Cc1c(n(c(c1C#N)N)Cc2cccc(c2)Cl)C SPB02252 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccco3)SCc4c(cccc4Cl)Cl SPB06068 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)N/N=C/c4c(cccc4Cl)Cl SPB05084 c1cc(cc(c1)C(F)(F)F)c2nnc(o2)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl SPB03112 CCOC(=O)c1c(nc(s1)c2ccccc2)CSc3ccccn3 SPB02185 Cc1ccc(cc1)SC(=O)c2c(noc2c3cc(on3)C)C SPB03255 c1ccn(c1)c2cccc(c2)c3nc(cs3)C(=O)NN SPB02236 c1ccc(cc1)S(=O)(=O)/C(=C/N2CCC(CC2)C(F)(F)F)/C#N SPB06081 CCc1ccccc1NC(=O)C TL00639 Cc1c(n(c(c1S(=O)(=O)c2ccccn2)N)Cc3ccccc3Cl)C SPB02240 Cc1c(n(c(c1S(=O)(=O)c2ccccn2)N)Cc3ccccc3)C SPB02241 CCCS(=O)(=O)c1c(c(n(c1N)Cc2cccc(c2)Cl)C)C SPB02244 c1cc(ccc1c2nc(on2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F)OC(F)(F)F SPB03263 Cc1cc(no1)c2c(c(no2)C)C(=O)Sc3ccccc3 SPB06061 Cc1cccc(c1NC(=O)n2c(c(cn2)C(=O)OC)C(OC)OC)C SPB05148 Cc1ccc(cc1)/N=C/c2c(cnn2c3ccc(cc3)Cl)C(=O)OC SPB05153 CC(=O)Nc1ccc(cc1OC(F)(F)F)Br TL00670 Cc1cc(no1)c2c(c(no2)C)C(=O)Sc3cccc(c3)C(F)(F)F SPB03256 Cc1cc(no1)c2c(c(no2)C)C(=O)Oc3ccc(cc3)Cl SPB03259 CCOC(=O)c1cc(nc(c1C#N)Sc2ccccc2)C SPB00033 CCOC(=O)c1cc(nc(c1C#N)Sc2ccc(cc2)C)C SPB00034 CCOC(=O)c1cc(nc(c1C#N)Sc2ccccn2)C SPB00035 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)Cl)Cc3cccc(c3)Cl)C SPB02257 Cc1c(sc(n1)c2cccs2)C(=O)NNC(=O)Nc3ccccc3 SPB02260 c1cc(c(c(c1)Cl)CSc2nnc(s2)c3cnccn3)Cl SPB07298 COC(c1c(cnn1C(=O)Nc2ccccc2)C(=O)OC)OC SPB05144 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N/N=C/c3c(cccc3Cl)Cl SPB00128 c1cc(cc(c1)NC(=O)O/N=C(/c2ccno2)\N)C(F)(F)F SPB03273 C/C(=N\OC(=O)c1ccc(cc1)Cl)/Cn2c3ccccc3oc2=O SPB03275 c1cc(c(c(c1)Cl)OCc2nc(on2)CSc3ccc(cc3)Cl)Cl SPB03186 c1cc(ccc1Sc2cc(cnc2/C=N/NC(=S)N)C(F)(F)F)Cl SPB06012 CC(=O)Nc1ccc(cc1OC(F)(F)F)C#N TL00674 C/C(=N\O)/c1ccc2cc(ccc2c1)OC TL00716 c1ccc(cc1)C(=O)CSc2nnc(s2)c3cnccn3 SPB07300 c1cc(cc(c1)C(F)(F)F)C(=O)CSc2nnc(s2)c3cnccn3 SPB07302 CSc1nc(cc(n1)Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)Sc4[nH]c(nn4)c5cc(cc(c5)Cl)Cl SPB07256 Cc1ccc(cc1)/C=N/OC(=O)c2c(noc2c3c(nns3)C)C SPB03402 Cc1c(c(on1)c2c(nns2)C)C(=O)Nc3ccc(cc3)OC SPB03403 c1cc(sc1)c2nc(cs2)CC(=O)NNC(=O)c3cccs3 SPB02331 c1cc(ccc1NC(=O)O/N=C(/COc2ccc(cc2Cl)Cl)\N)Cl SPB00379 CC(C)(C)C(=O)O/N=C(/COc1ccc(cc1Cl)Cl)\N SPB00385 Cc1ccc(cc1)/C=C/2\CSc3ccc(cc3C2=O)F SEW05288 Cc1ccc(cc1)OC/C(=N/OC(=O)c2cc(on2)C)/N SPB06134 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCCC2 TL00822 c1cc(c(=O)n(c1)CCC(=O)O/N=C(/c2ccc(cc2)Cl)\N)C(F)(F)F SPB06138 c1cc(cc(c1)Cl)/C(=N/OC(=O)CCn2cccc(c2=O)C(F)(F)F)/N SPB06140 c1cc(ccc1c2nc(on2)NC(=O)NN3CCCCC3)OC(F)(F)F SPB03294 C/C(=N\OC(=O)Nc1cccc(c1)Cl)/Cn2c3ccccc3oc2=O SPB03245 c1cc(ccc1OC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl)Cl SPB03248 CCOC(=O)N/N=C\1/c2cc(ccc2NC1=O)F SEW05221 Cc1cc(cc(c1Cl)C)OC(=O)c2cc(on2)C SPB03249 c1cc2c(cc1F)/C(=N/NC(=S)N)/CCS2 SEW05292 CSc1[nH]nc(n1)c2ccco2 SPB00319 C=C(CC(=O)N1CCOCC1)C(=O)N2CCOCC2 TL00857 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NN SPB00324 CCC(=O)O/N=C(/COc1ccc(cc1Cl)Cl)\N SPB00387 c1ccc(c(c1)C(=O)OCCOc2ccc(cc2Cl)Cl)Cl SPB00474 CSc1c(c(nc(n1)CSc2ccccc2)N)C#N SPB06235 Cc1ccc(cc1)SCc2nc(c(c(n2)SC)C#N)N SPB06236 CN(C)/C=C/1\CSc2ccc(cc2C1=O)F SEW05289 C/C(=N\O)/c1ccc2c(c1)C(CCC2(C)C)(C)C TL00729 CC/C(=N\OC(=O)c1cccs1)/c2ccc(cc2)c3ccccc3F SEW05234 CC/C(=N\OC(=O)NS(=O)(=O)c1ccc(cc1)C)/c2ccc(cc2)c3ccccc3F SEW05239 Cc1cc(no1)C(=O)Oc2ccc(cc2)Cl SPB03250 Cc1c(c(on1)c2ccc(cc2)C(F)(F)F)C(=O)NNC(=O)c3ccc(cc3)Cl SPB02218 c1c(cc(cc1Cl)Cl)NC(=S)N SEW05277 Cc1cc(no1)c2c(c(n[nH]2)C)C(=O)OC SPB03282 Cc1ccc(cc1)C(=O)n2c(c(c(n2)C)C(=O)OC)c3cc(on3)C SPB03286 CN(CCOC(=O)Nc1cccc(c1)Cl)c2ccc(cn2)C#N SPB06244 Cc1nc(cs1)C(=O)NNC(=O)Nc2ccc(cc2)Cl SPB02299 Cc1cc(no1)c2c(c(nn2c3ccccc3)C)C(=O)OC SPB03295 Cc1nc(cs1)c2nnc(n2C)SCc3c(cccc3Cl)Cl SPB02310 CC(C)(C)c1ccc(cc1)SC(=O)c2ccc(nc2)OCC(F)(F)F SPB06090 CSc1nnc(s1)SCC#N SPB02222 CSc1nnc(s1)SCC(=S)N SPB02223 CNC(=S)N/N=C/c1c(cnn1c2ccc(cc2F)F)C(=O)OC SPB05139 COC(=O)c1cnn(c1/C=N/NC(=S)N)c2ccc(cc2F)F SPB05140 CC(C)(C)NC(=S)NNC(=O)c1ccccc1 SPB00229 CCCCCCCCCCCCSCc1nc(no1)c2cc(c(c(c2)Br)OC)Br SPB00233 Cc1nc(cs1)C(=O)NNC(=O)Nc2ccccc2 SPB02298 c1ccc(cc1)c2nc(on2)c3ccc(nc3)OCC(F)(F)F SPB06105 Cc1c(sc(n1)c2cccs2)C(=O)NNS(=O)(=O)c3ccc(c(c3)Cl)F SPB02316 c1cc(sc1)c2nnn(n2)CC(=O)NNC(=O)c3ccc(cc3)Cl SPB02318 Cc1ccc(cc1)SCC(=N)N.Cl SPB06106 CCOC(=O)Cn1nc(nn1)c2cccs2 SPB02307 c1ccc(cc1)SC(=O)CCn2cccc(c2=O)C(F)(F)F SPB06110 CSc1nn(c(=S)s1)CSc2c(cccc2Cl)Cl SPB03311 Cc1c(sc(n1)c2cccs2)NC(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N SPB02311 CC(=O)Nc1ccccc1OC(F)(F)F TL00689 Cc1c(c(no1)C(=O)N(C)C)c2cc[nH]c(=S)n2 SPB03325 COc1c(cc(cc1Br)c2nc(on2)CSc3ccccc3)Br SPB00234 C1CC1CSc2nnc(s2)SCC(=O)N3CCC(CC3)C(F)(F)F SPB07225 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)SCC(=O)N3CCC(CC3)C(F)(F)F SPB07226 c1ccc(c(c1)c2ccc(cc2)C(=O)N)F SEW05230 CCC(c1ccc(cc1)c2ccccc2F)O SEW05231 CSc1nc(nc(n1)N)CSc2ccccc2 SPB06115 C1CCN(CC1)C(=O)CC#N TL00706 c1c(cnc(c1[N+](=O)[O-])O)Cl SPB06124 CCOC(=O)N1CCN(CC1)C2c3ccccc3-c4c2cccc4 SPB06126 CC(=O)Nc1ccc(cc1C(=O)O)[N+](=O)[O-] TL00682 Cc1cc(no1)C(=O)O/N=C(/COc2cccc(c2)Cl)\N SPB06131 Cc1cc(no1)C(=O)O/N=C(/COc2ccc(cc2Cl)Cl)\N SPB06132 Cc1cc(no1)C(=O)O/N=C(/COc2ccc(cc2)[N+](=O)[O-])\N SPB06135 CSc1[nH]c(nn1)C(F)(F)F SPB00212 CCN(CC)C(=O)O/N=C(/c1cc(c(c(c1)Br)OC)Br)\N SPB00220 Cc1cc(nc(n1)Cc2c(cccc2Cl)Cl)O SPB00314 c1cc(c(nc1)OCC(F)(F)F)C#N SPB07362 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3cccc(c3)C(F)(F)F SPB07363 c1cc(c(cc1Cl)Cl)NC(=O)Nc2ccno2 SPB03336 c1cc(ccc1NC(=O)Nc2ccno2)Cl SPB03337 c1cc(ccc1c2nc(on2)c3ccc(nc3)OCC(F)(F)F)Cl SPB06103 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N SPB02370 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C)Cc3ccsc3 SPB02379 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NNC(=O)C(Cl)(Cl)Cl SPB00360 CC(C)(C)C(=O)O/N=C(/c1c(cccc1Cl)Cl)\N SPB00363 CCOC(=O)C(C(=O)Nc1ccccc1)[N+](=O)[O-] SPB00364 c1cc(ccc1CSc2[nH]nc(n2)C(F)(F)F)Cl SPB00213 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NC(=O)NNc3c(cncc3Cl)Cl SPB00325 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)N/N=C/c3ccc(s3)[N+](=O)[O-] SPB00330 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)N/N=C/c3ccccn3 SPB00331 Cc1ccc(cc1)NC(=O)Nc2c(noc2c3ccc(cc3)C(F)(F)F)C SPB02275 CCOC(CC(=O)NNC(=S)NC)OCC SPB05181 c1ccc(c(c1)c2ccc(o2)C=C3C(=O)c4ccccc4C3=O)OC(F)(F)F SEW05188 CNC(=S)N/N=C/c1c(cnn1c2ccc(cc2)Cl)C(=O)OC SPB05155 CC(=O)Nc1nccc(n1)c2cc(no2)c3ccccc3 SPB05200 c1cc(c(cc1Cl)Cl)OC/C(=N/O)/N SPB00372 CC(=O)Nc1ccc2c(c1)CCCC2 TL00745 COC(=O)c1ccc(cc1)c2ccccc2F SEW05251 CC/C(=N\Oc1ccc(cc1[N+](=O)[O-])C(F)(F)F)/c2ccc(cc2)c3ccccc3F SEW05252 CCC(c1ccc(cc1)c2ccccc2F)Sc3ccccc3N SEW05253 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC#C SPB00247 Cc1c(sc(n1)c2cccs2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB02263 CCOC(=O)c1c(nc(s1)CS(=O)(=O)c2ccccn2)C SPB02265 c1cc(c(cc1Cl)Cl)CSc2[nH]nc(n2)C(F)(F)F SPB00214 c1ccc(cc1)/C(=N/OC(=O)CCn2cccc(c2=O)C(F)(F)F)/N SPB06137 c1cc(c(=O)n(c1)CCC(=O)O/N=C(/c2ccc(cc2)OC(F)(F)F)\N)C(F)(F)F SPB06139 Cc1ccc(cc1)CSc2[nH]c(nn2)C(F)(F)F SPB00216 CC(C)NC(=O)NNc1c(cccc1Cl)Cl SPB00349 Cc1nc(cs1)C(=O)NNC(=O)c2ccc(cc2)Cl SPB02303 Cc1nc(cs1)c2nnc(n2C)S SPB02306 Cc1c(c(no1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F)c3csc(n3)C SPB03387 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)O/N=C/c3ccc(cc3)Cl SPB02327 Cc1cc(no1)c2c(c(nn2c3ccccc3)C)C(=O)N4CCOCC4 SPB05214 CCOC(=O)c1csc(n1)C SPB02288 Cc1cc(no1)c2c(c(nn2c3ccccc3)C)C(=O)NN4CCOCC4 SPB05216 Cc1cc(no1)c2c(c(nn2c3ccc(c(c3)Cl)F)C)C(=O)NN4CCOCC4 SPB05219 CC(C)(C)c1ccc(cc1)C(=O)NN SPB00257 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc(cc3)Cl)SC SPB00264 Cc1c(c(on1)c2ccc(cc2)C(F)(F)F)C(=O)NNC(=O)Nc3ccccc3 SPB02273 Cc1c(nc(s1)c2ccc(cc2)Cl)c3ccc(cc3)c4ccccc4F SEW05204 CN(C)/C=C/C(=O)c1ccc(o1)c2cc(ccc2Cl)C(F)(F)F SEW05205 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC(C)(C)C SPB00068 CCOC(Cc1nnc(n1C)SCC(=O)Nc2ccc(cc2Cl)Cl)OCC SPB05198 c1cc(sc1)/C=N/Nc2ncc(s2)c3ccc4c(c3)OCCCO4 SPB07378 c1cc(ccc1/C=N/Nc2ncc(s2)c3ccc4c(c3)OCCCO4)C#N SPB07379 c1cc(ccc1NC(=O)Cc2cc(sc2Br)Br)Cl SPB02293 c1ccc(cc1)SCc2cc(=O)oc3c2ccc(c3)O SPB07383 Cc1c(c(no1)c2ccccc2)c3ccnc(n3)C SPB05202 Cc1c(c(no1)c2ccccc2)c3ccnc(n3)N SPB05204 Cc1c(c(no1)c2ccccc2)c3ccnc(n3)c4ccc(cc4)Cl SPB05205 c1ccc(cc1)c2cc(on2)c3ccnc(n3)c4ccc(cc4)Cl SPB05206 Cc1cc(no1)c2c(c(nn2c3cccc(c3)C(F)(F)F)C)C(=O)N4CCCCC4 SPB05208 Cc1nc(c(s1)C(=O)O/N=C(/c2ccc(cc2)Cl)\N)C(F)(F)F SPB07320 C/C(=N\O)/C(=O)c1ccc(cc1)c2ccccc2F SEW05226 Cc1ccc(cc1)NC(=O)c2c(noc2c3ccc(cc3)Cl)C SPB02291 c1ccc(c(c1)NC(=O)Cc2cc(sc2Br)Br)Cl SPB02292 CCOC(=O)C(C(=O)OCC)Nc1ccc(cc1)Cl SPB06294 CCOC(=O)C(C(=O)OCC)Nc1cccc(c1)Cl SPB06296 COc1cc\2c(cc1OC)NC(=O)/C2=C\c3cccs3 SEW05314 c1ccc(cc1)c2[nH]c(nn2)SCc3cc(=O)oc4c3ccc(c4)O SPB07388 CCO/C(=C(\C#N)/C(=S)N)/C SPB05311 Cc1c(c(on1)N)C(=S)N SPB05312 CN(c1ccccc1)C(=S)N TL00838 Cc1c(cnc(n1)COc2ccccc2Cl)S(=O)(=O)c3ccc(cc3)Cl SPB06043 CCOC(=O)CSc1c(n2ccsc2n1)/C=N/c3cc(cc(c3)Cl)Cl SPB06047 c1ccnc(c1)S(=O)(=O)Cc2nc(cs2)c3ccc(cc3)Cl SPB02231 CCCS(=O)(=O)c1c(c(n(c1N)Cc2ccccc2)C)C SPB02239 CC(C)(C)c1ccc(cc1)C(=O)NNC(=S)NC SPB00241 CC(C)(C)c1ccc(cc1)C(=O)NNC(=S)Nc2ccccc2 SPB00242 CC(C)(C)c1ccc(cc1)c2nnc(n2C)S SPB00243 Cc1c(c(no1)C(=O)NNC(=O)Nc2ccc(cc2)Cl)c3csc(n3)c4ccccc4 SPB03347 c1cc(ccc1Nc2ncc(s2)c3ccc4c(c3)OCCCO4)Cl SPB07372 Cc1c2cc(ccc2[nH]c1c3ccc(cc3)c4ccccc4F)OC SEW05261 Cc1ccc(cc1)NC(=O)c2c(c(on2)C)c3csc(n3)c4ccccc4 SPB03354 Cc1c(c(no1)C(=O)Nc2ccc(cc2)Cl)c3csc(n3)c4ccccc4 SPB03355 CCOC(=O)c1c(c(on1)C)c2csc(n2)COc3cc(cc(c3)Cl)Cl SPB03363 c1cc(ccc1/N=C/c2ccc(o2)c3cc(ccc3Cl)C(F)(F)F)Cl SEW05263 COC(c1c(cc(c(n1)SCC#N)C#N)C(=O)OC)OC SPB05129 c1cc(cc(c1)Cl)C(=O)NNC(=O)CCn2cccc(c2=O)C(F)(F)F SPB06157 CCSc1nnc(s1)N TL00786 Cc1c(c(nc(n1)c2ccccc2OC(F)(F)F)O)Cl SPB03321 CCOC(=O)c1c(c(on1)C)c2csc(n2)c3ccc(cc3)Cl SPB03327 Cc1c(c([nH]n1)COc2ccccc2)C(=O)OC SPB06167 c1cc(ccc1C(=O)O/N=C(/c2ccno2)\N)Cl SPB03303 Cc1cc(nc(n1)c2ccccc2OC(F)(F)F)O SPB03304 CCOC(=O)c1c(c(on1)C)c2csc(n2)CS(=O)(=O)Cc3cccc(c3)C(F)(F)F SPB03365 Cc1cc(n(n1)CC/C(=N/OC(=O)c2ccccc2)/N)C SPB06174 CCN(CC)C(=O)Nc1c(onc1c2c(cccc2Cl)Cl)C SPB00061 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(C)C3CCCCC3 SPB00066 Cc1cc(no1)c2c(c(no2)C)c3nc(no3)c4cccc(c4)C(F)(F)F SPB03268 c1cc(c(cc1C(F)(F)F)c2ccc(o2)C=C(C#N)C#N)Cl SEW05179 c1cc(ccc1/C=N/NC(=S)N)Cl SPB03332 C/C(=N\Nc1cccc(c1)C(F)(F)F)/c2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06285 c1ccc(cc1)C(=O)O/N=C/c2c(cc(cn2)C(F)(F)F)Sc3ccc(cc3)Cl SPB06287 Cc1c(nc(s1)c2ccc(cc2)F)CC(=O)OC SEW05311 c1cc(c(=O)n(c1)CCC(=S)N)C(F)(F)F SPB06169 c1cc(oc1)c2[nH]c(nn2)S SPB00315 Cc1nc(nc(n1)N)CSc2ccccc2 SPB06120 Cc1nc(nc(n1)N)CSc2ccc(cc2)Cl SPB06122 CCOC(=O)c1cc(n(n1)c2c(cc(cc2Cl)Cl)Cl)C SPB00322 Cc1cc(no1)C(=O)O/N=C(/COc2ccc(cc2)OC)\N SPB06133 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)N/N=C/N(C)C SPB00327 Cc1cc(no1)c2c(c(no2)C)C(=O)Nc3ccc(cc3)Cl SPB03211 Cc1cc(no1)c2c(c(no2)C)C(=O)Nc3cccc(c3)Cl SPB03213 c1cc(sc1)C(=O)O/N=C/c2c(cc(cn2)C(F)(F)F)Sc3ccc(cc3)Cl SPB06292 CCOC(Cc1nnc(n1C)SCC(=O)c2ccc(cc2Cl)Cl)OCC SPB05226 Cc1c(c(n(n1)c2cc(ccc2Cl)Cl)N)C(=S)N SPB06197 Cc1c(c(n(n1)c2ccccc2)N)C(=S)N SPB06198 Cc1c(c(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)C)Sc3ccc(cc3)Cl SPB06203 CCOC(Cc1nnc(n1C)SCC(=O)c2ccccc2)OCC SPB05227 Cc1nc(cs1)c2nnc(o2)S SPB02382 CC(C(=O)O/N=C(/c1c(cccc1Cl)Cl)\N)Oc2ccc(cc2Cl)Cl SPB00390 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)N/N=C/C(C)(C)C SPB00328 Cc1ccc(cc1)NC(=O)Nc2c(noc2c3cccs3)C SPB02336 c1cc(sc1)c2nc(cs2)COc3cc(cc(c3)Cl)Cl SPB02340 c1c(cc(c2c1sc(n2)N3CCC(CC3)C(F)(F)F)Cl)Cl SPB06073 CCOC(=O)/C(=C/Nc1cc(c(nc1)N(C)C)C(F)(F)F)/C#N SPB06078 CC(C)S(=O)(=O)/C(=C/N1CCC(CC1)C(F)(F)F)/C#N SPB06080 Cc1c(n(c(c1C#N)NC(=O)c2cccs2)Cc3cccc(c3)Cl)C SPB02255 CCOC(Cc1nnc(n1C)SCC(=O)c2cccc(c2)C(F)(F)F)OCC SPB05228 CC(=O)Nc1ccccc1NC(=O)C TL00809 CC(=O)Nc1cc(c(cc1NC(=O)C)Cl)Cl TL00810 c1cc(ccc1SCc2cc(=O)oc3c2ccc(c3)O)Cl SPB07384 CS(=O)(=O)Nc1ccccc1NS(=O)(=O)C TL00811 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCc3cc(=O)oc4c3ccc(c4)O SPB07386 CC(/C(=N/O)/N)Oc1ccc(cc1Cl)Cl SPB00391 c1cc(cc(c1)C(F)(F)F)/C=N/O SPB05234 CC/C(=N\OC(=O)c1cccc(c1)C(F)(F)F)/c2ccc(cc2)c3ccccc3F SEW05233 Cc1c(c(n(n1)c2ccccc2)N)c3nc(cs3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB06215 COC(c1c(cc2c(c(sc2n1)C(=O)c3ccc(cc3)Cl)N)C(=O)OC)OC SPB05250 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)C(C)(C)C)Cc3cccc(c3)Cl)C SPB02256 c1cc(sc1)c2[nH]c(nn2)SCc3cc(=O)oc4c3ccc(c4)O SPB07387 Cc1c(nc(s1)c2ccsc2)c3ccc(cc3)c4ccccc4F SEW05281 COC(=O)c1cc(ccc1N2CCCC2)[N+](=O)[O-] SEW05283 Cc1c(nc(s1)Nc2ccccc2N3CCOCC3)c4ccc(cc4)c5ccccc5F.Br SEW05285 c1cc2c(cc1F)C(=O)C(=O)N2CN3CCOCC3 SEW05287 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NNC(=O)C(C)(C)C SPB00362 c1cc(c(cc1Cl)Cl)c2cc(on2)c3ccnc(n3)N SPB05238 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCCCC2 TL00816 Cn1c(nnc1SCc2cc(=O)oc3c2ccc(c3)O)C(F)(F)F SPB07389 c1ccc(cc1)n2c(nnc2SCc3cc(=O)oc4c3ccc(c4)O)O SPB07392 Cc1ccc(cc1)C(=O)c2c(c3cc(c(nc3s2)C(OC)OC)C(=O)OC)N SPB05251 c1cc(ccc1n2c(nnc2SCc3cc(=O)oc4c3ccc(c4)O)O)Cl SPB07393 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCOCC2 TL00821 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3c(cccc3Cl)F SPB00142 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN=C(C)C SPB00131 C=CCSc1[nH]c(nn1)c2cccs2 SPB00136 CSc1[nH]nc(n1)c2cccs2 SPB00137 Cc1cc(nn1C(C)(C)C)C(=O)Nc2ccc(cc2)Cl SPB07504 Cc1cc(no1)c2nc(cs2)C(=O)/C=C/N(C)C SPB05270 Cc1cc(no1)c2c(c(nn2c3ccccc3)C)C(=O)Sc4ccccc4 SPB05277 Cc1cc(no1)c2c(c(nn2c3ccc(c(c3)Cl)F)C)C(=O)Sc4ccccc4 SPB05278 c1cc(c(c(c1)Cl)Cc2nc(cc(n2)O)C(F)(F)F)Cl SPB00346 Cc1c(c(no1)C(=O)N/N=C/c2c(cccc2Cl)Cl)c3csc(n3)C SPB03381 Cc1c(c(n(n1)C)C(=O)Sc2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] SPB03384 Cc1cc(no1)c2nc(cs2)c3ccnn3C(=O)Nc4cccc(c4)Cl SPB05279 CCC(=O)NNC(=O)c1cc(n(n1)c2c(cc(cc2Cl)Cl)Cl)C SPB00361 c1ccc2c(c1)c3c([nH]2)C(N(CC3)CN4c5ccc(cc5C(=O)C4=O)F)C(F)(F)F SEW05290 c1ccc(cc1)OCc2[nH]c(c/c(=N\c3ccc(cc3)Cl)/n2)O SPB06144 Cc1cc(nn1C(C)(C)C)C(=O)Sc2ccc(cc2)Cl SPB07501 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCc3cc(cc(c3)Cl)Cl SPB00435 COC(=O)c1cnn(c1C=C(C#N)C#N)c2ccc(cc2)Cl SPB05269 c1cc(ccc1SCc2cc(cc(c2)Cl)Cl)Cl SPB00451 c1c(cc(cc1Cl)Cl)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05253 CC(C)(C)c1csc(n1)c2ccc(nc2)N3CCC(CC3)C(F)(F)F SPB06250 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCc4ccccc4 SPB05255 Cc1c(c(no1)c2ccccc2)c3ccnc(n3)NC(=O)C SPB05257 c1cc(cc(c1)C(F)(F)F)c2cc(on2)c3ccnc(n3)N SPB05260 COC(=O)c1cnn(c1C=C(C#N)C#N)c2c(cccc2Cl)Cl SPB05266 Cc1ccc(cc1)SC(=O)c2c(noc2COc3ccccc3)C SPB06257 c1cc(ccc1C(=N)N)Cl.Cl SPB06264 c1ccc2c(c1)-c3ccccc3C2Sc4ccc(cn4)C(F)(F)F SPB06265 C#CCSc1[nH]c(nn1)c2cc(cc(c2)Cl)Cl SPB00416 COc1ccccc1c2nc(no2)CSc3ccccc3N SEW05240 c1ccc(c(c1)c2ccc(cc2)C#N)F SEW05243 c1cc(c(cc1OCC(F)(F)F)C(=O)NN)OCC(F)(F)F SPB03377 c1cc(ccc1c2nnc(o2)c3cnccc3C(F)(F)F)OC(F)(F)F SPB03478 c1ccc(c(c1)c2nnc(o2)c3ccccc3Cl)OC(F)(F)F SPB03483 c1ccc(cc1)c2csc(n2)c3ccc(nc3)N4CCC(CC4)C(F)(F)F SPB06247 c1cc(ccc1C(=O)NNC(=O)c2ccc(cc2)Cl)OC(F)(F)F SPB03438 CC(=O)Nc1ccc(cc1Cl)Br TL00885 CN(C)/C=C/C(=O)c1csc(n1)c2ccccc2 SPB03451 COc1ccc(cc1OC2CCCC2)C(=O)OC TL00897 Cc1cc(ccc1NC(=O)C)Cl TL00898 Cc1c(c(n(n1)c2cc(ccc2Cl)Cl)N)c3nc(cs3)C(C)(C)C SPB06217 CN(CCOC(=O)c1c(cccc1Cl)F)c2ccc(cn2)C#N SPB06218 CN(CCOC(=O)c1cc(cc(c1)Cl)Cl)c2ccc(cn2)C#N SPB06220 CN(CCOC(=O)c1ccc(cc1)OC(F)(F)F)c2ccc(cn2)C#N SPB06221 c1cc2c(cc1F)C(C(=O)N2)O SEW05246 Cc1c(sc(n1)c2cccs2)NC(=O)O/N=C(/c3ccc(cc3)Cl)\N SPB02313 Cc1c(sc(n1)c2cccs2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl SPB02315 c1cc(cc(c1)Cl)/C(=N/OC(=O)c2ccc(nc2)OCC(F)(F)F)/N SPB06098 c1cc(ccc1/C(=N/OC(=O)c2ccc(nc2)OCC(F)(F)F)/N)Cl SPB06099 c1cc(ccc1CC#N)OCc2c(cc(cn2)C(F)(F)F)Cl SPB06276 Cc1cc(cc(c1NC(=O)C)Cl)Cl TL00876 c1cc(c(nc1)Oc2ccc(cc2)F)C(=O)O TL00878 Cc1c(c(on1)c2c(nns2)C)C(=O)NC(=O)Nc3ccccc3 SPB03432 c1cc(cc(c1)S(=O)(=O)n2c(c(cn2)S(=O)(=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl)C(F)(F)F SPB05383 c1cc(sc1)C(=O)O/N=C(/Cc2ccc(cc2)[N+](=O)[O-])\N SPB00522 c1cc(c(c(c1)Cl)NNC(=O)c2cc(cc(c2)Cl)Cl)Cl SPB00524 Cc1cccc(c1)c2nc(on2)NC(=O)NNc3c(cccc3Cl)Cl SPB00528 Cc1c2c(nc(nc2sc1C(=O)c3ccc(cc3)Cl)c4ccc(cc4Cl)Cl)C SPB05389 Cc1cc(no1)c2c(c(nn2c3cccc(c3)C(F)(F)F)C)C(=O)Sc4ccccc4 SPB05291 CCOC(=O)c1c(c(on1)C)c2csc(n2)c3ccccc3 SPB03329 c1ccc(cc1)/C=N/NC(=S)N SPB03333 Cc1ccc(cc1)NC(=O)NC(=O)c2c(noc2c3c(nns3)C)C SPB03433 c1cc(ccc1C(=O)n2cc3c(n2)-c4cc(ccc4SC3)F)Cl SEW05351 Cc1ncc2c(n1)-c3cc(ccc3SC2)F SEW05363 c1cc(ccc1c2nc(cs2)c3ccc(cc3)Cl)OC(F)(F)F SPB03453 Cc1c(c(on1)c2cccs2)C(=O)NN SPB02333 Cc1c(c(on1)c2cccs2)C(=O)NNC(=O)c3c(cccc3F)F SPB02334 c1cc(ccc1c2nc(cs2)c3ccc(cc3)Br)OC(F)(F)F SPB03454 c1cc(c(c(c1)Cl)CSc2nnc(s2)SCc3cc(=O)oc4c3ccc(c4)O)Cl SPB07434 CC(C)(C)c1ccc(cc1)OCc2[nH]c(c/c(=N\c3ccccc3Cl)/n2)O SPB06146 c1ccc(cc1)c2nc(cs2)c3ccn[nH]3 SPB03525 Cc1ccc(cc1)C(=O)NNC(=O)Cc2csc(n2)c3csc(n3)C SPB03526 c1cc(oc1C(=O)OCc2cc(cc(c2)Cl)Cl)[N+](=O)[O-] SPB00439 Cc1c(nc(s1)c2ccc(cc2)Cl)CC(=O)OC SEW05303 Cc1c(c(on1)c2cccs2)C(=O)OC SPB02329 COC(=O)c1cc(c(nc1)Sc2ccc(cc2)Cl)[N+](=O)[O-] SPB07412 CCOC(=O)c1nc(no1)c2ccc(cc2)[N+](=O)[O-] SPB00494 c1cc(ncc1[N+](=O)[O-])Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl SPB00498 CC(C)(C)c1[nH]c(nn1)Sc2ccc(cn2)[N+](=O)[O-] SPB00500 Cc1ccc(cc1)Sc2c(cc(cn2)C(=O)OC)[N+](=O)[O-] SPB07413 CSc1nnc(s1)SCc2cc(=O)oc3c2ccc(c3)O SPB07431 c1ccc(c(c1)c2ccc(cc2)C(=O)NN)F SEW05305 CCCc1ccc(cc1)/C(=N/O)/C TL00858 c1cc(ccc1NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)Cl SPB07290 CCOC(=O)c1c(c(on1)C)c2csc(n2)N/N=C/c3ccccc3 SPB03343 c1ccc(cc1)OCc2ncc(s2)c3ccc4c(c3)OCCCO4 SPB07367 c1cc(ccc1OCc2ncc(s2)c3ccc4c(c3)OCCCO4)Cl SPB07368 c1cc2c(cc1c3cnc(s3)COc4cc(cc(c4)Cl)Cl)OCCCO2 SPB07370 COC(=O)c1cc(c(nc1)Sc2ccccc2NS(=O)(=O)C)[N+](=O)[O-] SPB07477 Cc1cc(no1)c2nc(cs2)c3ccnn3C(=O)Nc4ccccc4 SPB05280 CN(CCOC(=O)c1ccc(cc1)[N+](=O)[O-])c2c(cc(cn2)C(F)(F)F)Cl SPB06278 CCc1cccc(c1NC(=O)CSc2c(c(c3c(n2)CCC3)/C=C\c4ccccc4)C#N)CC SPB07457 C#Cc1cccc(c1)NC(=O)CSc2c(c(c3c(n2)CCC3)/C=C\c4ccccc4)C#N SPB07458 c1ccc(cc1)/C=C\c2c3c(nc(c2C#N)SCC(=O)c4ccccc4)CCC3 SPB07460 c1c(cc(cc1Cl)Cl)c2[nH]c(nn2)S SPB00410 c1cc(ccc1c2nnc(o2)c3ccc(cc3)Cl)OC(F)(F)F SPB03456 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)OC(F)(F)F)Cl SPB03459 c1cc(ccc1c2nnc(o2)c3ccc(cc3Cl)Cl)OC(F)(F)F SPB03460 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)Sc3ccc(cc3)Cl SPB02346 c1cc(cc(c1)Cl)c2nnc(o2)CSc3nnc(n3C4CCCCC4)O SPB07371 CC(=O)CSc1nnc(n1c2ccc(cc2)Cl)c3ccc(cc3)C(C)(C)C SPB00265 Cc1nc(cs1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F SPB02322 Cc1nc(cs1)C(=O)NNC(=O)c2c(cccc2F)F SPB02323 Cc1c(c(on1)c2ccc(cc2)C(F)(F)F)NC(=O)Nc3ccc(cc3)Cl SPB02276 Cc1cc(no1)c2nc(cs2)c3ccnn3S(=O)(=O)c4cccc(c4)C(F)(F)F SPB05283 c1ccc(cc1)CSc2c(c(c3c(n2)CCC3)/C=C\c4ccccc4)C#N SPB07452 CSc1c(c(c2c(n1)CCC2)/C=C/c3ccccc3)C#N SPB07454 c1ccc(cc1)/C=C\c2c3c(nc(c2C#N)SCC(=O)Nc4cc(cc(c4)Cl)Cl)CCC3 SPB07456 Cc1nc(cs1)c2nc(cs2)CC(=O)NNC(=O)c3ccc(cc3)Cl SPB03527 Cc1ccc(c(c1)C)c2csc(n2)N SEW05365 c1ccc(cc1)Sc2c(c(c(s2)Sc3ccccc3)[N+](=O)[O-])[N+](=O)[O-] SEW05367 c1cc(cc(c1)Cl)NC(=O)CSc2nc(nc(n2)O)c3ccc(cc3)Cl SPB02390 c1ccc(c(c1)c2nnc(o2)c3c(cccc3F)F)OC(F)(F)F SPB03533 COc1c(cc(cn1)C(=O)NNC(=O)c2cccs2)[N+](=O)[O-] SPB07439 c1cc(ccc1Sc2cc(cnc2/C=N/O)C(F)(F)F)Cl SPB06280 C/C(=N\Nc1ccccc1)/c2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06283 c1cc(sc1)/C=C/2\CSc3ccc(cc3C2=O)F SEW05304 Cc1c(c(on1)c2ccc(cc2)Cl)NC(=O)NN3CCCCC3 SPB02280 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl SPB05192 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl SPB05186 COC(c1c(cc2c(c(sc2n1)C(=O)c3cccc(c3)C(F)(F)F)N)C(=O)OC)OC SPB05252 c1cc2c(cc1c3cnc(s3)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)OCCCO2 SPB07375 C/C(=N\Nc1cc(ccc1Cl)Cl)/c2csc(n2)c3ccccc3 SPB03568 Cc1c(c(nc(n1)c2ccc(cc2)Cl)SCc3ccccc3)C(=O)C SPB05341 COC(=O)c1cc(c(nc1)Nc2ccc(cc2)Cl)[N+](=O)[O-] SPB07493 C/C(=N\Nc1ccc(cc1Cl)Cl)/c2csc(n2)c3ccc(nc3)OCC(F)(F)F SPB07490 CC(C)(C)c1ccc(cc1)C(=O)NNC(=S)NCCCOC SPB00446 c1c(cc(cc1Cl)Cl)CN2CCSCC2 SPB00448 c1ccc(c(c1)/C=N/Nc2ncc(s2)c3ccc4c(c3)OCCCO4)Cl SPB07377 c1c(cc(c(c1Br)OC(=O)c2cc(cc(c2)Cl)Cl)Br)C#N SPB00468 Cc1c(c(n(n1)CCC#N)C)Oc2ccc(cc2)Cl SPB06226 c1cc(ncc1C(=S)N)N2CCC(CC2)C(F)(F)F SPB06231 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3csc(n3)c4ccccc4 SPB03573 COC(=O)c1cc(c(nc1)Sc2ccccc2NS(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] SPB07487 c1cc(c(c(c1)Cl)CSc2[nH]c(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)F SPB00432 Cc1c(c(on1)c2c(nns2)C)C(=O)NC(=O)OCC#C SPB03436 Cc1c(c(n(n1)c2cc(ccc2Cl)Cl)N)c3nc(cs3)c4ccccc4 SPB06216 C/C(=C(/C#N)\C(=S)N)/NNc1ccccc1 SPB06183 Cc1cc(sc1c2ccc(cc2)c3ccccc3F)C(=O)OC SEW05282 Cc1c(c(on1)c2c(nns2)C)C(=O)O/N=C/c3cccc(c3)Cl SPB03404 Cc1c(c(n(n1)c2cc(ccc2Cl)C(F)(F)F)N)C(=S)N SPB06188 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC SPB06193 Cc1nccc(n1)c2cc(no2)c3ccc(cc3Cl)Cl SPB05222 c1cc(c(cc1Cl)Cl)OCCOC(=O)c2ccc(o2)[N+](=O)[O-] SPB00471 Cc1cc(no1)c2nc(no2)COc3ccc(cc3Cl)Cl SPB06148 Cc1cc(no1)c2nc(no2)COc3ccc(cc3)[N+](=O)[O-] SPB06149 Cc1c(c(on1)c2c(nns2)C)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N SPB03418 Cc1c(c(on1)c2c(nns2)C)c3nc(no3)c4ccc(o4)[N+](=O)[O-] SPB03421 CCOC(=O)c1c(c(on1)C)c2csc(n2)N/N=C/c3ccccc3Cl SPB03344 CCOC(CC(=O)NNC(=O)c1c(onc1c2c(cccc2Cl)Cl)C)OCC SPB06160 CC(=O)c1csc(n1)c2ccccc2 SPB03431 Cc1c(c(on1)c2c(nns2)C)C(=O)NC(=O)Nc3cc(cc(c3)Cl)Cl SPB03435 CN(CCOC(=O)Nc1ccccc1)c2ccc(cn2)C#N SPB06243 Cc1ccc(n1c2ccc(cc2)OC(F)(F)F)C SEW05265 Cc1c(c(on1)c2c(nns2)C)C(=O)Nc3cc(cc(c3)Cl)Cl SPB03370 c1cc(ccc1C(F)(F)F)NC(=S)N SEW05274 C/C(=C(/C#N)\C(=S)N)/NNc1ccc(cc1)[N+](=O)[O-] SPB06184 CCOC(CC(=O)NNC(=O)c1c(onc1c2ccccc2Cl)C)OCC SPB06159 CC(=O)Nc1ccc2c(c1)CCC2=O TL00757 Cc1ccc(cc1Cl)NC(=O)C TL00758 c1c(cnc(c1Cl)CSc2nnc(s2)SCC3CC3)C(F)(F)F SPB06233 CSc1c(c(nc(n1)CSc2ccc(cc2)Cl)N)C#N SPB06237 Cc1c(c(on1)C)C(=O)Sc2cccc(c2)C(F)(F)F SPB06166 Cc1cc(n(n1)CC/C(=N/OC(=O)c2ccccc2Cl)/N)C SPB06175 Cc1c(c(n(n1)CC/C(=N/OC(=O)c2ccccc2)/N)C)Oc3ccc(cc3)Cl SPB06239 Cc1c(c(n(n1)CC/C(=N/OC(=O)c2ccc(cc2)Cl)/N)C)Oc3ccc(cc3)Cl SPB06240 Cc1cc(no1)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)C(F)(F)F SPB06303 COc1cc\2c(cc1OC)NC(=O)/C2=C\c3ccc(cc3)OC(F)(F)F SEW05316 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)Cl)C SEW05318 COc1ccc(cc1)NC(=O)c2ccc(cc2)c3ccccc3F SEW05320 C/C(=C(/C#N)\C(=S)N)/NNc1cc(ccc1Cl)C(F)(F)F SPB06186 c1ccc(c(c1)c2nc(cc(n2)O)C(F)(F)F)OC(F)(F)F SPB03319 c1cc(ccc1c2c(cnn2S(=O)(=O)c3ccc(cc3Cl)Cl)S(=O)(=O)c4ccc(cc4)Cl)Cl SPB05382 c1cc(ccc1c2[nH]c(nn2)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl SPB00505 c1ccc(cc1)c2nc(on2)C(=O)NN SPB00508 Cc1cc(nn1C(C)(C)C)C(=O)Sc2cccc(c2)C(F)(F)F SPB07502 Cc1cc(nn1C(C)(C)C)C(=O)Sc2cccc(c2)Br SPB07503 Cc1cc(nn1C(C)(C)C)C(=O)Nc2ccc(cc2)C(C)(C)C SPB07506 c1c(cc(cc1Cl)Cl)C(=N)N.Cl SPB00407 Cc1c2c(onc2c(=O)[nH]n1)C SPB03409 CCOC(=O)c1c(c(on1)C)c2csc(n2)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB03361 CCOC(=O)c1c(c(on1)C)c2csc(n2)COc3ccc(cc3)Cl SPB03362 Cc1c(c(nc(n1)Cc2c(cccc2Cl)Cl)OC(=O)N(C)C)Cl SPB00333 CC/C(=N\Oc1ccc(cn1)C(F)(F)F)/c2ccc(cc2)c3ccccc3F SEW05275 c1ccc(c(c1)NC(=S)N)N2CCOCC2 SEW05276 c1cc(sc1)c2n[nH]nn2 SPB02301 Cc1ccc(cc1)SC(=O)c2cc(n(n2)c3c(cc(cc3Cl)Cl)Cl)C SPB02345 c1cscc1CC(=O)NN SPB02354 CC(=O)c1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05254 c1cnoc1NC(=O)NN2CCOCC2 SPB03341 Cc1cc(nn1C(C)(C)C)C(=O)Nc2cccnc2 SPB07507 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCc4ccc(cc4)Cl SPB05256 CC(=O)Nc1nccc(n1)c2cc(no2)c3cccc(c3)C(F)(F)F SPB05263 COC(=O)c1cc(c(nc1)Sc2ccc(cn2)C(F)(F)F)[N+](=O)[O-] SPB07449 c1ccc(cc1)/C=C\c2c3c(nc(c2C#N)SCc4ccc(cc4)Cl)CCC3 SPB07453 C=CCSc1c(c(c2c(n1)CCC2)/C=C/c3ccccc3)C#N SPB07455 Cc1c(c(n(n1)c2ccc(cc2)[N+](=O)[O-])N)C(=S)N SPB06187 c1ccc(cc1)c2csc(n2)CCn3cccc(c3=O)C(F)(F)F SPB06190 c1cc(c(=O)n(c1)CCc2nc(cs2)c3ccc(cc3)Cl)C(F)(F)F SPB06191 CCNC(=O)NNc1c(cccc1Cl)Cl SPB00348 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/Cn2c3ccccc3oc2=O SPB03276 Cc1c(c(n(n1)C)c2ccno2)C(=O)OC SPB03277 Cc1nccc(n1)c2cc(no2)c3cccc(c3)C(F)(F)F SPB05261 Cc1c(c(no1)C(=O)NN)c2csc(n2)C SPB03374 c1ccc(cc1)C(=O)CSc2nnc(o2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F SPB03389 CC(C)(C)C(=O)CSc1nnc(o1)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F SPB03393 Cc1c(c(on1)c2c(nns2)C)C(=O)O/N=C/c3ccc(cc3)Cl SPB03399 c1c(cc(cc1C(F)(F)F)NC(=S)N)C(F)(F)F SPB03351 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)SCc3cc(=O)oc4c3ccc(c4)O SPB07433 c1cc(c(cc1C(=O)NN)F)F SPB07437 Cc1c(c(on1)c2c(nns2)C)C(=O)ON=C(C)C SPB03400 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(o2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F SPB03405 Cn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])Cc3ccsc3 SPB02363 Cn1c(nnc1SCc2c(cccc2Cl)Cl)Cc3ccsc3 SPB02364 CC(=O)Nc1ccc(cc1OC(F)(F)F)Cl TL00814 c1ccc(c(c1)c2ccc(cc2)C(=O)N3CCOCC3)F SEW05272 c1cc(cc(c1)Cl)Nc2ncc(s2)c3ccc4c(c3)OCCCO4 SPB07373 CCOC(=O)C(=CNc1ccccc1OC(F)(F)F)C(=O)OCC TL00806 Cc1ccc(cc1)SCc2cc(=O)oc3c2ccc(c3)O SPB07382 c1cc2c(cc(=O)oc2cc1O)CSc3nnc(s3)SCC4CC4 SPB07432 c1cc(ccc1C(=O)NNC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl SEW05309 COc1cc(cc(c1OC)OC)/C=C\2/c3cc(c(cc3NC2=O)OC)OC SEW05315 COc1cc\2c(cc1OC)NC(=O)/C2=C\c3cccc(c3)C(F)(F)F SEW05317 c1ccc(c(c1)c2ccc(cc2)C(=O)Nc3ccc(cc3)C(F)(F)F)F SEW05321 c1ccc(c(c1)C(F)(F)F)NC(=O)CSc2nnc(o2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F SPB03406 CN(CCO)c1ccc(cn1)C#N SPB06209 CC(C)N(C(C)C)C(=O)c1ccc(cc1)c2ccccc2F SEW05322 CN(C)/C=C/C(=O)c1ccc2cc(ccc2c1)OC SEW05332 CCCCCn1c(nnc1SCc2c(cc(cn2)C(F)(F)F)Cl)O SPB06213 c1cc(ccc1C(=O)CSc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)Cl SPB00419 c1cc(c(c(c1)Cl)Cc2nc(no2)N)Cl SPB00336 c1cc(c(c(c1)Cl)c2nc(on2)C(=O)NN)Cl SPB00337 Cc1cc(c(c(c1)C)Nc2ncc(s2)c3ccc4c(c3)OCCCO4)C SPB07374 CNS(=O)(=O)c1ccc(cc1)[N+](=O)[O-] TL00824 Cc1c(nc(s1)N2CCOCC2)c3ccc(cc3)c4ccccc4F SEW05279 Cc1c(snn1)c2nc(c(s2)C)c3ccc(cc3)c4ccccc4F SEW05280 CC(C)(C)c1cc(nn1c2c(cc(cc2Cl)Cl)Cl)NC(=O)NN(C)C SPB00356 Cc1c(c(on1)COc2ccccc2)C(=O)O SPB06201 Cc1ccccc1Nc2c(cc(cn2)C(=O)OC)[N+](=O)[O-] SPB07494 c1ccc(cc1)c2nc(cs2)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl SPB03575 COC(=O)c1cc(c(nc1)Nc2cccc(c2)C(F)(F)F)[N+](=O)[O-] SPB07495 CC(C)(C)c1ccc(cc1)Nc2c(cc(cn2)C(=O)OC)[N+](=O)[O-] SPB07496 Cc1cc(nn1C(C)(C)C)C(=O)Sc2ccccc2 SPB07500 c1cc(ccc1C2=NCCS2)OCC#N SPB02431 COc1ccc(cc1)C(=O)O/N=C/2\CCSc3c2cc(cc3)F SEW05401 CC(C)NC(=O)O/N=C(\COc1ccc(cc1)C2=NCCS2)/N SPB02436 Cc1nc(cs1)c2nnc(n2C)SCC(=O)Nc3cc(cc(c3)Cl)Cl SPB02440 Cc1nc(cs1)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)C(C)C SPB02441 Cc1nc(cs1)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)Cl SPB02442 c1ccc(cc1)c2cc(nc(n2)Cc3c(cccc3Cl)Cl)O SPB00351 CC(C)(C)c1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)ONC(=O)c3ccccc3 SPB00352 c1cc(c(cc1Cl)Cl)CSc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl SPB00414 c1cc(c(cc1OCC(F)(F)F)c2nnc(o2)S)OCC(F)(F)F SPB03385 Cc1c(c(no1)C(=O)NNC(=O)c2ccc(cc2)Cl)c3csc(n3)C SPB03386 Cc1c(sc(n1)CS(=O)(=O)c2ccccn2)C(=O)NNC(=O)c3ccccc3 SPB02450 Cc1c(sc(n1)CS(=O)(=O)c2ccccn2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB02451 c1ccc(c(c1)C(F)(F)F)n2c(nnc2S)O SPB00559 Cc1nc(cs1)c2ccnc(n2)c3cc(cc(c3)Cl)Cl SPB03616 Cc1cc(no1)c2nnnn2c3ccc(cc3)F SPB03618 Cn1ccnc1SCC(=O)Nc2ccc(cc2)Cl SPB02459 c1cc(ccc1C2=NCCS2)OCC(=O)Nc3ccc(cc3)Cl SPB02467 Cc1ccc(cc1)SC(C)C(=O)c2ccc(c(c2)Cl)C XAX00014 Cc1c2c(onc2c(=O)n(n1)c3ccc(cc3)F)C SPB03608 Cc1ccc(cc1Cl)C(=O)C(C)S(=O)(=O)c2ccc(cc2)Cl XAX00017 Cc1ccc(cc1)S(=O)(=O)C(C)C(=O)c2ccc(c(c2)Cl)C XAX00018 c1ccc(cc1)C(=O)NCCSCc2c(cc(cn2)C(F)(F)F)Cl SPB06272 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2nc(no2)c3cccs3)Cl SPB00570 c1cc(sc1)c2nc(on2)C(=O)N/N=C/c3ccc(s3)[N+](=O)[O-] SPB00569 Cc1nc(cs1)c2nnc(n2c3cccc(c3)F)SCc4ccccc4 SPB02356 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N SPB02371 Cc1ccc(cc1Cl)c2c(sc(n2)n3c(ccc3C)C)C XAX00020 Cc1nc(cs1)c2nc(nc(n2)SC)N SPB03614 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Cl)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05465 c1cc(ccc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05466 Cc1ccc(cc1Cl)c2c(sc(n2)/N=C/N(C)C)C XAX00019 Cc1cc(nn1C(C)(C)C)C(=O)O/N=C(/c2cccc(c2)C(F)(F)F)\N SPB07516 c1cc(c(c(c1)Cl)CSc2nnc(o2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F)Cl SPB03413 Cc1c(c(on1)c2c(nns2)C)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB03419 COc1cc(ccc1N/N=C(\C#N)/C(=O)N)Cl XAX00021 CC(C)(C)c1ccc(cc1)/N=N/C2C(=NNC2=O)N XAX00023 c1cc(ccc1C2CCCCC2)C(=O)/C=C/C(=O)O XAX00025 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)C(F)(F)F)OC(F)(F)F SPB03465 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3Cl)Cl)OC(F)(F)F SPB03466 Cc1nc(cs1)c2nnc(o2)SCc3ccccc3Cl SPB02388 Cc1ccc(c(c1)C(=O)/C=C/C(=O)O)C XAX00030 CCOC(=O)c1nc(no1)c2cccc(c2)C SPB00502 Cn1c(nnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)Cc3ccsc3 SPB02381 Cc1cc(nn1C(C)(C)C)C(=O)O/N=C(/c2ccc(cc2)Cl)\N SPB07517 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2nc([nH]n2)c3cc(cc(c3)Cl)Cl SPB00506 Cc1cccc(c1)c2nc(on2)C(=O)NN SPB00509 CC(C)(C)c1ccc(cc1)c2[nH]nc(n2)Sc3c(cccn3)[N+](=O)[O-] SPB00512 Cn1c(nnc1SCc2c(cccc2Cl)F)c3csc(n3)c4cccs4 SPB02385 CSc1nnc(n1c2ccc(cc2)Cl)c3cnccc3C(F)(F)F SPB06224 CC(C)(C)c1ccc(cc1)c2nnc(n2CCCOC)SCC(=O)c3ccc(cc3)Cl SPB00456 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Oc3ccccc3 SPB05319 Cc1c(c(n(n1)C(=O)C)COc2ccccc2)C(=O)OC SPB06246 c1ccc(cc1)c2nc(cs2)c3ccnc(n3)SCc4ccccc4Cl SPB03468 Cn1c(cnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)c3ccc(cc3)Cl SPB02398 CC(C)c1ccc(cc1)NC(=O)CSc2ncc(n2C)c3ccc(cc3)Cl SPB02399 CCOC(=O)c1csc(n1)N/N=C/c2ccccc2Cl SPB02407 c1cc(ccc1c2cnn(c2N)c3c(cc(cn3)C(F)(F)F)Cl)Cl SPB06263 c1ccc2c(c1)-c3ccccc3C2Sc4[nH]c(nn4)N SPB06266 c1ccc2c(c1)c(c3ccccc3c2Sc4ccc(cc4)Cl)/C=N\O SEW05294 COC(=O)c1cc(c(nc1)Sc2ccccc2N)[N+](=O)[O-] SPB07470 c1ccc(c(c1)C(=O)NNC(=O)c2ccccc2Cl)OC(F)(F)F SPB03462 c1ccc(cc1)c2nc(cs2)c3ccnc(n3)SCc4ccc(cc4)Cl SPB03469 c1cc(ccc1NC(=O)NC(=O)c2ccc(nc2)Oc3ccc(cc3)Cl)Cl SPB06254 Cc1cccc(c1)/C(=N/O)/N SPB07589 c1cc(c(c(c1NN=C(C#N)C#N)C#N)Cl)Cl SEW05427 CCOC(=O)c1c(nc(s1)c2ccc(cc2)Cl)O SPB02472 Cc1cc(no1)c2nc(c(s2)c3nnc(n3C)SCC(=O)Nc4cc(cc(c4)Cl)Cl)C SPB05322 Cc1cc(no1)c2nc(c(s2)c3nnc(n3C)SCC(=O)Nc4ccc(cc4)C(C)C)C SPB05324 Cc1cc(no1)c2nc(c(s2)c3nnc(n3C)SCC(=O)Nc4ccc(cc4)Cl)C SPB05325 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)Cl)OC(F)(F)F SPB03489 Cc1ccc(c(c1)C)c2csc(n2)NC(=N)N SEW05388 CCOC(=O)c1c(c(on1)C)C(=O)CSc2c(c(c(c(n2)C)C)C)C#N SPB03490 CC(C)(C#C)NC(=O)c1ccc(cc1)c2ccccc2F SEW05386 Cc1nc(cs1)c2nnc(n2c3cccc(c3)F)S SPB02352 COc1c(cc(cn1)C(=O)NNC(=O)c2ccno2)[N+](=O)[O-] SPB07440 c1cc(ccc1c2nnc(o2)c3ccncc3)OC(F)(F)F SPB03503 c1ccc(c(c1)c2nnc(o2)c3cccnc3)OC(F)(F)F SPB03505 CCOC(=O)c1c(nc(s1)c2ccc(cc2)C(F)(F)F)O SPB02473 c1cc(oc1)CSC/C(=N/O)/N SPB02483 c1cc(ccc1S(=O)(=O)NNc2ccc(cc2F)F)Cl SPB00465 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCCOc3ccc(cc3Cl)Cl SPB00469 c1cc(c(cc1Cl)Cl)OCC(=O)Oc2c(cc(cc2Br)C#N)Br SPB00470 CC(=O)c1csc(n1)COc2ccc(cc2)Cl SPB03561 Cc1cc(no1)c2nnnn2c3cc(cc(c3)Cl)Cl SPB03621 Cc1nc(cs1)c2nc(cs2)c3ccnc(n3)SCC(=O)Nc4ccccc4C(F)(F)F SPB03627 Cc1nc(cs1)c2nc(cs2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl SPB03629 CC(=O)c1csc(n1)COc2ccc(cc2)OC SPB03562 CC(=O)c1csc(n1)Nc2ccccc2Cl SPB03566 Cc1nc(cs1)c2nnc(o2)SCc3ccc(cc3)C(F)(F)F SPB02387 c1ccc(c(c1)c2nnc(o2)c3cccc(c3)C(F)(F)F)OC(F)(F)F SPB03482 c1ccc(c(c1)c2nnc(o2)c3ccccc3F)OC(F)(F)F SPB03486 CC(C)c1ccc(cc1)NC(=O)COc2ccc(cc2)C3SCCS3 SPB02404 Cc1nc(cs1)c2nc(cs2)CC(=O)NNC(=O)Nc3cccc(c3)C(F)(F)F SPB03510 c1cc(ccc1C(=O)Sc2ccc(cc2)Cl)OC(F)(F)F SPB03511 COC(=O)c1cc(c(nc1)Sc2c(cccc2Cl)Cl)[N+](=O)[O-] SPB07450 COC(=O)/C(=C\c1ccccc1N2CCN(CC2)Cc3ccccc3)/C#N SEW05372 Cc1ccc(cc1)c2csc(n2)c3ccccc3 SEW05398 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)OCCOc3ccc(cc3Cl)Cl SPB00478 CC(C)(C)c1ccc(cc1)c2[nH]nc(n2)Sc3ccc(cn3)[N+](=O)[O-] SPB00499 Cc1c(snn1)C(=O)O/N=C/2\CCSc3c2cc(cc3)F SEW05380 c1ccc(c(c1)c2ccc(cc2)C(=O)N3CCCCCC3)F SEW05381 Cc1c(c(n(n1)S(=O)(=O)c2ccc(cc2)Cl)C)Oc3ccc(cc3)Cl SPB05332 c1ccc(c(c1)C(F)(F)F)n2c(nnc2Sc3cc(c(cn3)C(F)(F)F)C(F)(F)F)O SPB03534 c1cc(ccc1c2nc(nc(n2)SCC(=O)Nc3ccc(cc3)Cl)O)Cl SPB02391 CC(=O)c1csc(n1)COc2ccccc2 SPB03560 CC(=O)c1csc(n1)Nc2ccc(cc2)Cl SPB03565 COC(=O)c1cc(c(nc1)Sc2ccccc2NC(=O)c3cccs3)[N+](=O)[O-] SPB07473 Cc1cc(no1)c2nc(c(s2)c3nnc(n3C)S)C SPB05308 CCCCCCCCCCCc1nnc(n1c2ccccc2C(F)(F)F)SCC(=O)Nc3ccc(cc3)Cl SPB02432 Cc1c(c(nc(n1)c2ccc(cc2)C(F)(F)F)SCc3ccccc3)C(=O)C SPB05359 Cc1c2c(nc(nc2sc1C(=O)c3ccc(cc3)Cl)c4ccccc4)C SPB05365 CCCCCCCCCCCc1nnc(n1c2ccccc2C(F)(F)F)SCC(=O)Nc3ccc(cc3)C(C)C SPB02433 Cc1c(c(n(n1)C(=O)c2ccccc2)C)Oc3ccc(cc3)Cl SPB05315 Cc1c(c(n(n1)C(=O)C2CC2)C)Oc3ccc(cc3)Cl SPB05316 c1ccc(cc1)/C=C\c2c3c(nc(c2C#N)SCC(=O)c4ccc(cc4)C(F)(F)F)CCC3 SPB07463 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccccc2N3CCOCC3)/C#N SEW05389 Cc1nc(cs1)C(=O)NNC(=S)NCCCOC SPB02438 Cc1nc(cs1)c2nnc(n2CCCOC)SCC(=O)c3ccc(cc3)Cl SPB02446 COC(=O)c1cc(c(nc1)Sc2ccccc2NC(=O)c3ccc(cc3)Cl)[N+](=O)[O-] SPB07472 CC(C)C(=O)Nc1ccccc1Sc2c(cc(cn2)C(=O)OC)[N+](=O)[O-] SPB07475 Cc1ccc(cc1)C(=O)Nc2ccccc2Sc3c(cc(cn3)C(=O)OC)[N+](=O)[O-] SPB07474 Cc1c(c(no1)C(=O)NN)c2csc(n2)c3ccccc3 SPB03338 c1ccc(cc1)CN2CCN(CC2)c3ccccc3C=C(C#N)C#N SEW05346 COC(=O)c1cc2c(s1)-c3cc(ccc3SC2)F SEW05348 c1ccnc(c1)Sc2c(c(c(s2)Sc3ccccn3)[N+](=O)[O-])[N+](=O)[O-] SEW05440 Cc1c2c(nc(nc2sc1C(=O)c3ccccc3)c4ccccc4)C SPB05367 CC(=O)c1ccc(c(n1)S)C#N SPB05369 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2nc(no2)c3ccc(cc3)[N+](=O)[O-])Cl SPB00516 c1cc(ccc1C/C(=N/OC(=O)c2cc(cc(c2)Cl)Cl)/N)[N+](=O)[O-] SPB00521 CC(C)(C)c1ccc(cc1)c2n[nH]c(=S)n2CCCOC SPB00450 CC(C)(C)c1ccc(cc1)c2nc(on2)C(=O)N/N=C/c3c(cccc3Cl)Cl SPB00453 C/C(=C(/C#N)\C(=S)N)/NNc1c(cc(cn1)C(F)(F)F)Cl SPB06185 Cc1c(snn1)C(=O)OCCN(C)c2ccc(cn2)C#N SPB06219 c1cc2c(cc1F)-c3c(cno3)CS2 SEW05349 CC(C)(C)c1csc(n1)c2ccc(cc2)OC(F)(F)F.Br SPB03455 c1cc(ccc1c2nnc(o2)c3ccc(cc3)OC(F)(F)F)C(F)(F)F SPB03457 c1cc(ccc1C(=O)Nc2ccc(nc2)N3CCC(CC3)C(F)(F)F)OC(F)(F)F SPB06329 c1ccc(c(c1)c2nnc(o2)c3ccncc3)OC(F)(F)F SPB03506 Cc1ccc(cc1)Sc2c(c(c(s2)Sc3ccc(cc3)C)[N+](=O)[O-])[N+](=O)[O-] SEW05441 Cc1ccc(cc1)SC(=O)CCn2cc(ccc2=O)C(F)(F)F SPB06409 c1cc(ccc1C2SCCS2)OCC(=O)Nc3cc(cc(c3)Cl)Cl SPB02405 Cc1nc(cs1)c2ccc(cc2)/C(=N/OC(=O)c3ccc(cc3)C(F)(F)F)/N SPB02412 Cc1cc(no1)c2nnnn2c3ccc(cc3)C(F)(F)F SPB03620 c1ccn(c1)c2ccc(cc2)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05470 COc1ccc(cn1)[N+](=O)[O-] SEW05471 Cc1nc(cs1)c2nc(cs2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(C)C SPB03628 CC(=O)Nc1ccc2c(c1)CCC2 TL00752 CCCCc1ccc(cc1)C(=O)N TL00754 CC(C)c1ccccc1NC(=O)C TL00848 Cc1ccc(cc1)SC(=O)c2ccc(cc2)OC(F)(F)F SPB03512 Cc1cc(c(c(c1C)C(=O)/C=C/C(=O)O)C)C XAX00032 Cc1cc(no1)c2nnc(n2C)SCC(=O)c3ccc(cc3)Cl SPB06300 Cc1cc(no1)c2nnc(n2C)SCC(=O)c3ccccc3Cl SPB06302 Cc1nc(cs1)c2ccc(cc2)/C(=N/OC(=O)c3c(cccc3Cl)F)/N SPB02413 Cc1nc(cs1)c2nnc(o2)SCC(=O)c3ccccc3 SPB02415 CCOC(=O)c1cc(nc(n1)Sc2ccc(cc2)C)C SPB06307 c1cc(ccc1C(=O)Sc2ccc(cc2)C(F)(F)F)OC(F)(F)F SPB03513 c1ccc(c(c1)C(=O)Sc2c(cccc2Cl)Cl)OC(F)(F)F SPB03514 CCOC(=O)c1cc(nc(n1)Sc2ccc(cc2)Cl)C SPB06310 Cc1nc(cs1)c2nnc(o2)SCC(=O)c3ccc(cc3)Cl SPB02416 Cc1c(c(on1)C)c2c(c(no2)C)C(=O)NN SPB02417 Cc1c(c(n(n1)C(=O)c2ccccc2)C)Oc3ccccc3 SPB05317 c1ccc(c(c1)NC(=O)Nc2ccccc2Br)Br TL00797 Cc1nc(cs1)C(=O)NNC(=S)Nc2ccccc2C(F)(F)F SPB02344 CN(C)C(=O)n1c(nc(n1)c2cc(cc(c2)Cl)Cl)SC SPB00533 c1cc(cc(c1)Cl)n2c(=O)[nH]nc2S SPB00535 c1cc(ccc1NC(=O)Nc2cc(cc(c2)Cl)Cl)n3c(cc(n3)C(F)(F)F)C(F)(F)F SEW05433 c1cc(ccc1NC(=O)Nc2ccc(cc2F)F)n3c(cc(n3)C(F)(F)F)C(F)(F)F SEW05434 Cc1ccc(cc1)C(=O)NNC(=O)c2c(nc(s2)c3csc(n3)C)C SPB03518 C/C(=N\Cc1ccccc1)/c2ccccc2O XAX00033 Cc1cc(no1)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)C(C)C SPB06304 c1ccc(c(c1)C(=O)NN)OC(F)(F)F SPB03521 COc1ccccc1C(=O)O/N=C/c2c(cc(cn2)C(F)(F)F)Sc3ccc(cc3)Cl SPB06289 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)NC(=O)NN3CCOCC3 SPB00307 Cc1c(c(nc(n1)Cc2c(cccc2Cl)Cl)O)Cl SPB00312 c1cc(ccc1CSc2nnc(o2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F)[N+](=O)[O-] SPB03412 c1ccc(c(c1)CSc2nccc(n2)c3csc(n3)COc4cc(cc(c4)Cl)Cl)Cl SPB03658 c1cc(ccc1CSc2nccc(n2)c3csc(n3)COc4cc(cc(c4)Cl)Cl)Cl SPB03659 c1cc(c(cc1Cl)NNC(=O)C2CCCS2)Cl SPB03596 Cc1cc(no1)c2nnc(n2C)SCC(=O)Nc3ccccc3Cl SPB06305 CC(C)(C)c1[nH]c(nn1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F SPB00539 CSc1n[nH]c(=O)n1c2cccc(c2)Cl SPB00541 CSc1n[nH]c(=O)n1C2CCCCC2 SPB00542 c1cc(ccc1C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)C(F)(F)F)OC(F)(F)F SEW05428 Cc1cc(no1)c2nc(c(s2)c3nnc(n3C)SCC(=O)Nc4ccccc4)C SPB05326 C=CCSc1n[nH]c(=O)n1c2cccc(c2)Cl SPB00545 C=CCSc1n[nH]c(=O)n1C2CCCCC2 SPB00546 Cc1c(c(on1)c2c(nns2)C)C(=O)N SPB03414 CCOC(=O)c1c(c(on1)C)c2csc(n2)COc3ccccc3 SPB03373 c1ccc(cc1)/C=C\c2c3c(nc(c2C#N)SCC(=O)Nc4cccc(c4)C(F)(F)F)CCC3 SPB07459 Cc1cc(no1)c2nnc(n2C)SC SPB06336 CC(C)c1ccc(cc1)NC(=O)CSc2ncnc(n2)N SPB02428 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)Nc3ccc(cc3)Cl SPB07550 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)Nc3ccccc3 SPB07551 Cc1c2c(nc(nc2sc1C(=O)c3cccc(c3)C(F)(F)F)c4ccccc4)C SPB05393 Cc1cccc(c1)c2nc(on2)NC(=O)O/N=C/c3c(cccc3Cl)Cl SPB00529 CCOC(=O)c1c(n2c(s1)nc(n2)C(F)(F)F)C SPB05398 CN(C)S(=O)(=O)c1ccc(cc1)[N+](=O)[O-] TL00823 c1cc(ccc1N)S(=O)(=O)N2CCOCC2 TL00826 Cn1c(nnc1SCc2ccc(cc2)Cl)Cc3ccsc3 SPB02365 Cc1cc(n2c(n1)nc(n2)SCC(=O)Nc3cc(cc(c3)Cl)Cl)C SPB02424 c1cc(cc(c1)Cl)C(=O)NNC(=O)c2ccc(o2)Oc3ccc(cc3)C4SCCS4 SPB02427 Cc1c(sc(n1)CS(=O)(=O)c2ccccn2)C(=O)NNC(=O)c3c(cccc3Cl)F SPB02449 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05414 c1cc(ccc1S(=O)(=O)O/N=C/2\CCSc3c2cc(cc3)F)Cl SEW05371 c1ccc(cc1)CN2CCN(CC2)c3ccccc3/C=C/4\c5ccccc5NC4=O SEW05373 c1cc(ccc1N)Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW05382 c1cc(ccc1C/C(=N/O)/N)Oc2c(cncc2Cl)Cl SPB07554 Cc1ccc(cc1)c2csc(n2)NC(=N)N SEW05387 CCCCc1ccc(cc1)NC(=O)C TL00828 CCCCc1ccc(c(c1)C)NC(=O)C TL00829 Cc1c(c(nc(n1)c2cc(cc(c2)Cl)Cl)O)Cl SPB00427 CSc1[nH]c(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F SPB00429 C=CCSc1[nH]c(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F SPB00430 CC(C)(C)c1ccc(cc1)c2nnc(n2CCCOC)SCC(=O)NN SPB00581 CCOC(=O)c1cc(nc(c1C#N)Sc2ccccc2NC(=O)c3ccccc3)C SPB06415 CCOC(=O)c1cc(nc(c1C#N)Sc2ccccc2NC(=O)Nc3ccccc3)C SPB06418 CC(C)(C)c1ccc(cc1)CSc2nnc(n2Cc3ccco3)c4ccc(cc4)C(C)(C)C SPB00788 COCc1cc(nc(n1)Cc2c(cccc2Cl)Cl)O SPB00592 Cc1cccc(c1N/N=C(\C)/c2csc(n2)c3ccccc3)Cl SPB03567 Cc1cc(no1)c2c(c(no2)C)/C(=N/O)/N SPB03630 Cc1nc(cs1)c2nnc(n2CCCOC)SCC(=O)c3cccc(c3)[N+](=O)[O-] SPB02444 Cc1c(sc(n1)CS(=O)(=O)c2ccccn2)C(=O)NNC(=O)c3ccc(cc3)Cl SPB02448 c1cc(ccc1S(=O)(=O)Cc2nc(cs2)CSc3nnc(s3)SCC4CC4)Cl SPB02575 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)CS(=O)(=O)c3ccc(cc3)C(F)(F)F SPB02576 CC1(C2(CCC1(OC2=O)C(=O)N3CCSCC3)C)C SEW05473 c1cc(ccc1c2csc(n2)CS(=O)(=O)c3ccc(cc3)C(F)(F)F)Cl SPB02577 CC(C)n1c2ccccc2nc1Sc3ncc(s3)[N+](=O)[O-] SPB02582 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccco3)Sc4c(cccn4)[N+](=O)[O-] SPB00790 CCCSc1nnc(s1)N/C=N/O XAX00097 COc1cc(ccn1)C(=O)N SPB06368 Cc1cc(nc(n1)Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)C(=O)OC SPB06363 CCCCCCCCSc1nnc(s1)/N=C/N(C)C XAX00101 CC(C)(C)c1ccc(cc1)N/N=C(/C#N)\C(=O)N XAX00022 c1cc(oc1)CSC/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/N SPB02485 Cc1ccc(cc1)C(=O)/C=C/C(=O)O XAX00028 CCOC(=O)c1c(nc(s1)c2ccc(cc2)C)O SPB02495 COc1cc(cc(c1C(=O)N)C(F)(F)F)C(F)(F)F SEW05474 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)Cl)SCc3c(cc(cn3)C(F)(F)F)Cl SPB06378 CC(=O)Nc1ccc(c(c1)Cl)Br SPB06382 CC(=O)Nc1ccccc1C(F)(F)F SPB06386 Cc1c2c(ncnc2SCc3ccc(cc3)C(F)(F)F)on1 SPB05425 CN(C)/C=N/c1nnc(s1)SCc2ccc(cc2)Cl XAX00078 c1cc(ccc1CSc2nnc(s2)N)Cl XAX00081 CCCCCCSc1nnc(s1)/N=C/N(C)C XAX00102 CCOC(=O)/C(=C/c1ccc(c(c1)[N+](=O)[O-])N2CCCC2)/C#N XAX00103 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccc(cc2)C SPB07536 c1ccc(cc1)NC(=O)O/N=C(/Cc2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl)\N SPB06352 c1ccn(c1)c2nnc(s2)SCc3ccc(cc3)Cl XAX00079 Cc1cc(nn1C(C)(C)C)C(=O)O/N=C(/c2ccccc2)\N SPB07525 CC(C)(C)/C=N/NC(=O)c1nc(no1)c2ccc(cc2)C(C)(C)C SPB00462 COC(=O)c1cnn(c1/C=C(/C#N)\S(=O)(=O)c2ccccc2)c3ccc(cc3)Cl SPB05293 CCCSc1nnc(s1)N XAX00093 CCn1c(cc(n1)C)C(=O)NNC(=S)NCCCOC SPB02529 CCn1c(cc(n1)C)c2nnc(n2c3cccc(c3)C(F)(F)F)S SPB02532 CC(C)(C)c1ccc(cc1)NC(=O)CSc2nncn2C XAX00070 CC(C)(C)c1ccc(cc1)NC(=O)CSc2ccccn2 XAX00072 CC(=O)Nc1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05380 c1ccc(cc1)c2nc3n(n2)c(cs3)CC(=O)NN SPB00655 Cc1c(sc2c1c(nc(n2)c3ccc(cc3Cl)Cl)C)C#N SPB05388 CCOC(=O)c1cc(nn1Cc2ccc(cc2)C)C SPB07598 CCOC(=O)c1cc(nn1Cc2c(cccc2Cl)Cl)C SPB07600 CCOC(=O)c1cc(n(n1)Cc2c(cccc2Cl)Cl)C SPB07601 Cc1ccc(cc1)CSc2nnc(n2c3cccc(c3)Cl)OC(=O)N(C)C SPB00584 c1cc(ccc1CSc2nnc(s2)N)[N+](=O)[O-] XAX00083 CN(C)/C=N/c1nnc(s1)SCc2ccc(cc2)[N+](=O)[O-] XAX00084 CC(C)(C)c1ccc(cc1)C(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F SPB00666 CCOC(=O)c1cc(n(n1)Cc2cccc(c2)C(F)(F)F)C SPB07603 Cc1cccc(c1)c2nc(on2)C(=O)NNC(=O)C(Cl)(Cl)Cl SPB00514 c1cc(ccc1C(=O)O/N=C/2\CCSc3c2cc(cc3)F)Cl SEW05350 Cc1ccc(cc1)c2csc(n2)C SEW05368 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)OC(F)(F)F)F SPB03458 c1ccc(cc1)S(=O)(=O)n2c(c(cn2)S(=O)(=O)c3ccc(cc3)Cl)c4ccc(cc4)Cl SPB05381 CC(C)(C)c1ccc(cc1)c2[nH]c(nn2)SCc3ccccc3 SPB00575 Cc1ccc(cc1)CSc2[nH]c(nn2)c3ccc(cc3)C(C)(C)C SPB00576 CC(C)(C)c1ccc(cc1)c2[nH]c(nn2)SCc3ccc(cc3Cl)Cl SPB00577 CC(C)(C)c1ccc(cc1)c2nnc(n2C(=O)N(C)C)SCc3ccc(cc3Cl)Cl SPB00588 COc1c(cc(cn1)C(=O)NNC(=S)NC2CCCCC2)[N+](=O)[O-] SPB07580 c1ccc2c(c1)cccc2C/C(=N/OC(=O)c3ccc(cc3)Cl)/N SPB00828 Cc1ccc(cc1)CSc2nnc(n2C)c3cc(n(n3)c4ccc(cc4)[N+](=O)[O-])C SPB00831 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2csc(n2)c3ccccc3 SPB03587 COC(=O)c1cc(ccc1N2CCOCC2)NC(=S)NC(=O)c3ccccc3 SEW05450 CCn1c(cc(n1)C)c2nnc(n2c3ccccc3)SC SPB02503 CCOC(=O)c1c(nc(s1)c2ccccc2)CSc3nnc(n3C)C(F)(F)F SPB02517 Cc1cc(no1)c2c(c(no2)C)/C(=N/OC(=O)c3ccccc3)/N SPB03638 Cc1c(c(no1)C(=O)OC)c2cc[nH]n2 SPB03687 Cc1cc(cc(c1OC(=O)c2ccno2)Cl)Br SPB03690 CCCCCCSc1nnc(s1)N/C=N/O XAX00098 CCCCCCCCCCCCCCCCCCSc1nnc(s1)/N=C/N(C)C XAX00099 c1ccc(cc1)c2cc(on2)c3csc(n3)c4c(cc(cn4)C(F)(F)F)Cl SPB06453 c1cc(c(=O)n(c1)Cc2ccc(cc2)Cl)C(F)(F)F SPB06454 CCOC(=O)c1c(nc(s1)c2ccccc2)CSc3nnc(s3)SCC4CC4 SPB02512 Cc1c(sc(n1)COc2cccc(c2)Cl)C(=O)C SPB02514 Cc1c(sc(n1)COc2ccc(cc2)Cl)C(=O)C SPB02515 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccccc2Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07562 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)S SPB00668 c1c(cc(c(c1Cl)S(=O)(=O)N)Cl)C(F)(F)F SEW05430 c1cc(c(cc1CC(=O)NN)Cl)Cl TL00874 CCCCc1ccc(cc1)S(=O)(=O)N TL00879 CCCSc1nnc(s1)/N=C/N(C)C XAX00100 CCn1c(cc(n1)C)c2nnc(n2c3ccc(cc3)Cl)SCC(=O)c4ccccc4 SPB02506 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/Cc2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl)\N SPB06342 c1cc(ccc1C/C(=N/OC(=O)c2ccc(cc2)OC(F)(F)F)/N)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06344 CC(C)Nc1ccc(cc1[N+](=O)[O-])Cl SPB02520 c1cc(=O)n(cc1C(F)(F)F)CCC(=O)O SPB06384 Cc1c2c(nc(nc2sc1C(=O)c3cccc(c3)C(F)(F)F)c4ccc(cc4Cl)Cl)C SPB05390 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCc3ccccc3Cl SPB00599 C#CC1CCCCC1/N=C/c2cc(cc(c2O)Cl)Cl SEW05426 CC(=O)c1csc(n1)c2ccc(cc2)OC(F)(F)F SPB03583 c1cc(ccc1/C=N/NC(=S)N)C#N SPB02400 c1cc(sc1)/C=N/NC(=S)N SPB02402 c1cc(ccc1C2SCCS2)OCC(=O)Nc3ccc(cc3)Cl SPB02403 c1ccc(c(c1)C=C(C#N)C#N)N2CCOCC2 SEW05390 c1cc(ccc1C/C(=N/OC(=O)c2cc(cc(c2)Cl)Cl)/N)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06343 CCn1c(cc(n1)C)c2nnc(n2c3ccc(cc3)Cl)SC SPB02509 CCOC(=O)Cc1csc2n1nc(n2)c3ccccc3 SPB00650 Cc1cc(nn1C)C(=O)NN SPB00651 c1cc(ccc1NC(=O)Nc2ccc(nc2)N3CCC(CC3)C(F)(F)F)Cl SPB06331 c1cc(ccc1C(=O)CSc2nnc(s2)N)Cl XAX00087 CCOC(=O)c1c(c(on1)c2cccc(c2)[N+](=O)[O-])C#N SPB03643 CC(=O)c1csc(n1)COc2cc(cc(c2)Cl)Cl SPB03645 COc1c(c(ccn1)C(F)(F)F)C(=O)N SPB06361 CCOC(=O)c1c(nc(s1)c2ccc(cc2Cl)Cl)O SPB02521 Cc1c2c(ncnc2SCC(=O)C(C)(C)C)on1 SPB05414 COC(=O)c1cnn(c1/C=N/OC(=O)c2ccccc2)c3ccccc3 SPB05302 COC(=O)c1cnn(c1/C=N/OC(=O)c2ccc(cc2)Cl)c3ccccc3 SPB05303 c1cc(ccc1c2c(c[nH]n2)S(=O)(=O)c3ccc(cc3)Cl)Cl SPB05306 c1ccc(cc1)CC(C(=O)O)NCCC#N SEW05394 Cc1ccc(c(c1)C)c2csc(n2)c3ccc(cc3)Cl SEW05397 COc1c(cc(cn1)C(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F)[N+](=O)[O-] SPB07578 Cc1cc(no1)c2c(c(no2)C)COC(=O)c3ccccc3 SPB03650 Cc1ccc(cc1)c2csc(n2)c3ccc(c(c3)F)C SPB07588 c1ccc(c(c1)OCc2nc(cs2)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl)Cl SPB03694 CCOC(=O)c1cc(c(nc1C(F)(F)F)Nc2ccccc2)C#N SPB06430 CCOC(=O)c1cc(c(nc1C(F)(F)F)Nc2cccc(c2)Cl)C#N SPB06431 c1cnc(nc1c2csc(n2)COc3cc(cc(c3)Cl)Cl)S SPB03652 c1c(cc(c(c1Cl)S(=O)(=O)N2CCOCC2)Cl)C(F)(F)F SEW05431 C1CCC(CC1)n2c(nnc2S)O SPB00536 COC(=O)c1cc(c(nc1)Sc2ccccc2NS(=O)(=O)c3cccc(c3)C(F)(F)F)[N+](=O)[O-] SPB07476 Cc1ccc(cc1)NC(=O)Nc2ccccc2Sc3c(cc(cn3)C(=O)OC)[N+](=O)[O-] SPB07479 COC(=O)c1cc(c(nc1)Sc2ccccc2NC(=O)Nc3ccccc3)[N+](=O)[O-] SPB07481 Cc1c(c(nc(n1)c2ccc(cc2)C(F)(F)F)SCC#C)C(=O)C SPB05361 Cc1cc(no1)c2c(c(no2)C)C(=O)NNC(=O)C SPB03601 CC(C)(C)c1ccc(cc1)n2c(nnc2S)c3ccccc3Cl SPB00780 Cc1ccc(cc1)CSc2nnc(n2Cc3ccco3)c4ccc(cc4)C(C)(C)C SPB00786 Cc1c(cc(c(n1)/N=C/N(C)C)Br)Br XAX00107 Cc1cc(cnc1N/C=N/O)Br XAX00111 CC(=O)Nc1ccccc1F SPB06387 Cc1c(c(n(n1)c2ccc(cc2)OC(F)(F)F)c3c(nns3)C)C(=O)Sc4ccc(cc4)C(F)(F)F SPB05456 C/C(=N\c1ccc(cc1)C(F)(F)F)/CC(=O)C SEW05333 CC(=O)Nc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] SEW05335 c1cc2c(cc1F)/C(=N/O)/CCS2 SEW05340 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/Cc2ccc(cc2)[N+](=O)[O-])\N SPB00523 c1cc(ccc1NNC(=O)c2cc(cc(c2)Cl)Cl)I SPB00526 CSc1nc(c(c(n1)Sc2ccccc2)C#N)Sc3ccccc3 SPB07615 c1ccc(c(c1)N)SCc2cccc(c2F)Cl SEW05461 Cc1cc(no1)c2c(c(no2)C)C(=O)NNS(=O)(=O)c3ccccc3 SPB03604 CC(C)(C)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl XAX00064 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccco3)SCc4ccc(cc4)Cl SPB00787 c1ccc(c(c1)NC(=O)Nc2cccc(c2)Cl)SCc3c(cc(cn3)C(F)(F)F)Cl SPB06379 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)SCc3c(cc(cn3)C(F)(F)F)Cl SPB06380 Cc1c(c(n(n1)c2ccc(cc2)OC(F)(F)F)c3c(nns3)C)C(=O)OC SPB05452 Cc1c2c(ncnc2SCC(=O)Nc3ccccc3Cl)on1 SPB05457 CCOC(=O)c1cc(c(nc1C(F)(F)F)O)C#N SPB06401 CC(=O)c1csc(n1)CS(=O)(=O)Cc2cccc(c2)C(F)(F)F SPB03550 c1ccc(cc1)CSc2nnc(n2c3cccc(c3)Cl)O SPB00573 c1cc(c(c(c1)Cl)NNS(=O)(=O)c2ccc(c(c2)Cl)Cl)Cl SPB00527 C/C(=N\OC(=O)c1c(cccc1Cl)F)/c2csc(n2)c3ccccc3 SPB03581 Cc1cc(nn1C(C)(C)C)C(=O)Nc2cccc(c2)C(F)(F)F SPB07505 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)C(C)(C)C XAX00069 c1ccn(c1)c2nnc(s2)SCc3ccc(cc3)[N+](=O)[O-] XAX00082 CCOC(=O)CSc1nnc(s1)N XAX00085 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)Nc3ccc(cc3)C SPB07552 c1ccc(cc1)C(=O)CSc2[nH]c(nn2)c3ccccc3F SPB00633 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07560 CCOC(=O)NNC(=S)NC1CCCCC1 SPB00534 Cc1cc(no1)c2c(c(no2)C)C(=O)N/N=C/c3ccccc3 SPB03598 c1cc(ccc1/C(=N/OC(=O)C2CCCS2)/N)C(F)(F)F SPB03491 c1cc(sc1/C(=N/OC(=O)C2CCCS2)/N)[N+](=O)[O-] SPB03492 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCc3ccccc3 SPB00597 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCc3c(cccc3Cl)F SPB00600 Cc1ccc(cc1Cl)c2c(sc(n2)N/C=N/OC(=O)c3ccc(cc3)[N+](=O)[O-])C XAX00048 c1cc(ccc1CC#N)Oc2c(cncc2Cl)Cl SPB07553 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC(=O)c3ccc(cc3)Cl SPB00603 CC(C)(C)c1ccc(cc1)c2nnc(n2C)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F SPB00607 c1cc(ccc1C(=O)O/N=C/Nc2ncc(s2)c3ccc(s3)Br)[N+](=O)[O-] XAX00055 Cc1cc(no1)c2c(c(no2)C)C(=O)NNC(=O)c3ccccc3 SPB03600 COc1c(cc(cn1)C(=O)NNC(=S)Nc2ccccc2)[N+](=O)[O-] SPB07577 c1cc(ccc1Sc2c(c(c(s2)Sc3ccc(cc3)Cl)[N+](=O)[O-])[N+](=O)[O-])Cl SEW05442 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW05445 Cc1cc(no1)C(=O)NNC(=S)NC SPB06293 c1cc(ccc1C(=O)O/N=C/Nc2ncc(s2)c3ccc(s3)Br)Cl XAX00056 Cc1c(c(=N)n(nc1C(=O)Nc2ccccc2)c3ccc(cc3)C(C)(C)C)C#N XAX00059 CN(C)/C=N/c1ncc(s1)c2ccc(s2)Br XAX00060 CC(C)(C)c1ccc(cc1)OC/C(=N/O)/N SPB00821 c1cc(cc(c1)NC(=O)c2cccc(n2)C(F)(F)F)C(F)(F)F SPB06446 Cc1c(sc(n1)c2c(cc(cn2)C(F)(F)F)Cl)/C(=N/NC(=S)NC(C)(C)C)/C SPB06450 c1ccc(cc1)C(=O)O/N=C(/Cc2cccc3c2cccc3)\N SPB00827 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07571 C=CCNC(=S)Nc1ccc(cc1)Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW05467 COc1cc(cc(c1C(=O)NCc2cccs2)C(F)(F)F)C(F)(F)F SEW05475 CC(C)n1c2ccc(cc2nc1S)Cl SPB02586 Cc1ccc(cc1)NC(=O)CCn2cc(ccc2=O)C(F)(F)F SPB06411 CCOC(=O)c1cc(nc(c1C#N)Sc2ccccc2NC(=O)c3cccc(c3)C(F)(F)F)C SPB06417 C/C(=N\NC(=S)N)/c1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB06351 CC(C(=O)Nc1ccc(cc1)C(C)(C)C)N2CCCCC2 XAX00062 Cc1c(c(n(n1)S(=O)(=O)c2ccccc2)C)Oc3ccc(cc3)Cl SPB05333 Cc1ccc(cc1)CSc2nnc(n2c3cccc(c3)Cl)O SPB00548 c1ccc(c(c1)c2nnc(o2)c3ccc(cc3)OC(F)(F)F)C(F)(F)F SPB03531 c1ccc(cc1)C(=O)O/N=C(/Cc2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl)\N SPB06341 c1ccc(cc1)c2nc(cs2)c3ccnn3S(=O)(=O)c4ccc(cc4)Cl SPB03537 COc1cc(cc(c1C(=O)N2CCC(CC2)C(=O)c3ccc(cc3)Cl)C(F)(F)F)C(F)(F)F SEW05477 c1ccc(cc1)c2nc(cs2)c3ccnn3S(=O)(=O)c4ccc(cc4F)F SPB03539 C/C(=N\NC(=S)NC(C)(C)C)/c1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB06348 C/C(=N\NC(=S)Nc1ccccc1)/c2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06349 c1cc(ccc1C(=O)NNC(=O)C2CCCS2)Cl SPB03546 c1cc(ccc1C/C(=N/OC(=O)Nc2ccc(cc2)SC(F)(F)F)/N)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06355 COc1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05379 Cc1ccc(cc1)c2csc(n2)c3ccncc3 SEW05400 Cc1c(c(on1)C)C(=O)n2cc3c(n2)-c4cc(ccc4SC3)F SEW05402 COc1ccc(cc1)/C=N/c2ccc(cc2)OC SEW05326 c1c(cnc2c1CCCC2)C#N SEW05327 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)c3cccc(c3)C(F)(F)F SPB07547 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)Nc3cc(cc(c3)Cl)Cl SPB07549 CC(C(=O)Nc1ccc(cc1)C(C)(C)C)Sc2ccc(cc2)Cl XAX00068 Cc1cc(nn1c2ccc(cc2)C(C)C)C(=O)N/N=C/C(C)(C)C SPB00627 CC(C)(C)c1ccc(cc1)NC(=O)CSc2nccn2C XAX00073 Cc1c(c(nc(n1)C(F)(F)F)N2CCCCC2)Oc3ccccc3 SPB05405 Cc1c2c(ncnc2SCC(=O)Nc3cc(cc(c3)Cl)Cl)on1 SPB05408 Cc1ccc(c(c1)C)NC(=S)NNC(=O)c2cc(c(nc2)OC)[N+](=O)[O-] SPB07579 CCc1c(nc(s1)c2ccccc2)C(=O)OC SEW05422 Cn1c(nnc1S)Cc2ccsc2 SPB02360 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)c3ccc(cc3)Cl SPB07545 c1cc(ccc1C2SCCS2)Oc3ccc(o3)C(=O)NN SPB02421 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)c3ccccc3 SPB07546 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2NC(=O)c3cccs3 SPB07548 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)Cl)Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07568 c1ccc(c(c1)NC(=O)Nc2cc(cc(c2)Cl)Cl)Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07570 Cc1c(c(n(n1)c2ccccc2)c3c(nns3)C)C(=O)Sc4ccc(cc4)C(F)(F)F SPB05447 Cc1ccc(cc1)CSc2c3c(noc3ncn2)C SPB05424 c1ccc(c(c1)NC(=O)C2CC2)Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07572 Cc1ccc(c(c1)C)c2csc(n2)c3ccccc3 SEW05417 Cc1ccc(cc1)Sc2ccc(cc2/C=C\3/C(=O)NC(=S)S3)[N+](=O)[O-] XAX00138 Cc1c(c(no1)C(=O)OC)C(=O)/C=C/N(C)C SPB03709 Cc1c(c(no1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F)c3csc(n3)c4csc(n4)C SPB03713 C=CCSc1nnc(n1c2ccc(cc2)Cl)O SPB00728 Cc1c(c(no1)C(=O)N/N=C/c2ccccc2)c3csc(n3)c4csc(n4)C SPB03719 Cc1ccc(cc1)C(=O)n2c(ccn2)c3c(onc3C(=O)OC)C SPB03723 Cc1c(c(no1)C(=O)OC)/C(=N/OC(=O)c2c(cccc2F)F)/C SPB03725 Cc1ccc(cc1F)c2nc(cs2)c3ccccc3 SPB07585 Cn1ccnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl SPB02460 Cc1ccc(cc1F)c2nc(cs2)c3ccc(cc3)Cl SPB07586 Cc1ccc(cc1F)c2nc(cs2)c3cccc(c3)C(F)(F)F SPB07587 CC(C)c1ccc(cc1)NC(=O)Cn2cccc(c2=O)C(F)(F)F SPB06464 c1cc(c(=O)n(c1)CC(=O)c2ccc(cc2)Cl)C(F)(F)F SPB06465 c1cc(ccc1COc2ccc(cc2Cl)/C(=N/OC(=O)c3ccc(o3)[N+](=O)[O-])/N)Cl SPB00704 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3csc(n3)COc4ccccc4Cl SPB03680 CCOC(=O)c1cc(c(nc1C(F)(F)F)Oc2ccc(cc2)Cl)C#N SPB06473 c1cc(sc1)C2=NN(C(=O)CC2)CO XBX00032 Cc1nc(cs1)c2nc(cs2)c3ccnc(n3)SCc4ccc(cc4)Cl SPB03669 CC(=O)c1csc(n1)COc2ccccc2Cl SPB03670 c1c(cnc(c1C(F)(F)F)NN=C2C3CC4CC(C3)CC2C4)Cl SPB06481 COc1cc(c(cn1)c2nc(cs2)c3ccc(cc3)Cl)C(F)(F)F SPB06484 CCOC(=O)c1cc(n(n1)C)C SPB05352 Cc1nc(nc(n1)N)COc2ccccc2Cl SPB06371 CCOC(=O)c1cnc(nc1O)C SPB06372 CC(c1ccc(c(n1)S)C#N)(OC)OC SPB05368 CCOC(=O)c1c(cnn1C(=O)c2ccc(cc2)C(F)(F)F)Sc3ccccc3 SPB03686 Cc1cc(cc(c1Cl)C)OC(=O)c2ccno2 SPB03688 C/C(=N\NC(=O)Cc1cccs1)/C(=O)C XBX00020 CC(C)(C)OC(=O)Nc1ccc(cc1)OC SEW05518 c1ccc(cc1)C(=O)CSc2nccc(n2)c3csc(n3)COc4ccccc4Cl SPB03693 Cc1ccc(cc1)OC(=O)c2ccno2 SPB03696 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccc(cc2)Cl)C#N SPB06428 c1cc(sc1)C2=NNC(=O)CC2 XBX00035 c1ccc(cc1)C(=O)CCCCCC(=O)O XBX00039 CCOC(=O)c1cc(c(nc1C(F)(F)F)Nc2ccc(cc2)C)C#N SPB06432 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2[nH]c(nn2)c3ccccc3 SPB07540 Cc1cc(cnc1/N=C/N(C)C)Br XAX00108 Cc1c(cc(c(n1)N/C=N/O)Br)Br XAX00110 Cc1c(ccc(n1)N/C=N/O)Br XAX00112 c1ccc(cc1)C(=O)CSc2nnc(o2)Cc3ccsc3 SPB02524 CC(C)(C)c1ccc(cc1)NC(=O)OC(C)(C)C SEW05520 Cc1c(sc(n1)c2cccs2)c3ccnn3C(=O)C4CC4 SPB02622 Cc1c(sc(n1)c2cccs2)c3ccnn3C(=O)c4ccc(cc4)F SPB02624 CCOC(=O)c1c(c2ccc(nc2s1)C(=O)C)N SPB07718 Cc1ccc(cc1)CSc2n[nH]c(=O)n2C3CC4CC3C=C4 SPB07724 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Nc3cccc(c3)C(F)(F)F SPB07766 c1cc(ccc1Cc2nnc(s2)N/C=N/O)F XAX00121 C(CSc1nnc(s1)N)O XAX00123 CCn1c(cc(n1)C)c2nnc(n2CCCOC)S SPB02533 CCn1c(cc(n1)C)c2nnc(n2CCCOC)SCC(=O)Nc3ccccc3 SPB02534 CCOC(=O)CSc1nc2cc(ccc2n1C(C)C)Cl SPB02589 CCn1c(cc(n1)C)c2nnc(n2CCCOC)SCC(=O)c3ccccc3 SPB02535 Cc1c(c(n(n1)c2ccc(cc2)Cl)c3c(nns3)C)C(=O)N4CCOCC4 SPB05445 c1cc(ccc1C(=O)CSc2nnc(s2)N)F XAX00089 CCC(C)Cn1c(nnc1S)O SPB07591 c1cc(cc(c1)Cl)n2c(nnc2SCc3ccc(cc3Cl)Cl)O SPB00574 COc1ccc(cc1)C(=O)NC(=N)COc2ccccc2Cl SPB06424 CCOC(=O)c1c(nc(s1)c2ccccc2)CSc3nnc(s3)SC SPB02513 c1cc(ccc1CSc2nnc(s2)N)F XAX00120 CCNc1ccc(cc1[N+](=O)[O-])Cl SPB02522 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2nnc(o2)Cc3ccsc3 SPB02525 CN(C)/C=N/c1nnc(s1)SCc2ccc(cc2)F XAX00124 CC(=O)c1csc(n1)c2ccc(c(c2)[N+](=O)[O-])OC SPB07620 Cc1c(c(n(n1)c2ccccc2)c3c(nns3)C)C(=O)Oc4ccccc4 SPB05448 CCC(C)CNC(=S)NNC(=O)OCC SPB07590 Cc1ccc(cc1F)/C(=N/OC(=O)c2ccccc2)/N SPB07594 Cc1ccc(cc1F)/C(=N/OC(=O)c2ccc(cc2)C(C)(C)C)/N SPB07595 CN(C)C(=O)Oc1cc(nc(n1)Cc2c(cccc2Cl)Cl)COC SPB00601 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC(=O)c3ccccc3 SPB00602 Cc1ccc(cc1F)c2nc(cs2)C(=O)C SPB07619 Cc1c(c(n(n1)c2ccccc2)c3c(nns3)C)C(=O)O SPB05432 CC(=O)Nc1ccc(cc1)C#N SPB07621 CC(=O)Nc1ccc(cc1[N+](=O)[O-])C#N SPB07641 Cc1c(c(n(n1)c2ccccc2)c3c(nns3)C)C(=O)N4CCOCC4 SPB05446 CCn1c(cc(n1)C)c2nnc(n2c3ccccc3)SCc4ccccc4 SPB02504 Cc1cc(no1)c2c(c(no2)C)C(=O)NNC(=O)Nc3ccccc3 SPB03597 CCn1c(cc(n1)C)c2nnc(n2c3ccccc3)SCC(=O)c4ccccc4 SPB02505 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)Nc3cc(cc(c3)Cl)Cl SEW05486 c1cc(c(c(c1)F)S(=O)(=O)NCCSCc2c(cccc2Cl)F)F SEW05453 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)Nc3ccc(cc3)Cl SPB05421 CCOC(=O)CSc1[nH]c2ccc(cc2n1)C(F)(F)F SPB02527 CC(C)(C)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Br XAX00065 Cc1ccc(cc1)SC(C)C(=O)Nc2ccc(cc2)C(C)(C)C XAX00067 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)Oc3cccc(c3)C(F)(F)F SPB05550 c1c(cnc(c1Cl)NN=C2C3CC4CC(C3)CC2C4)C(F)(F)F SPB06480 c1cc(nc(c1)NN=C2C3CC4CC(C3)CC2C4)C(F)(F)F SPB06482 CC1(CC(CC(N1)(C)C)N2CCN(CC2)C3CC(NC(C3)(C)C)(C)C)C XBX00012 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)Nc3cccc(c3)Cl SPB05551 CC(C)(C)OC(=O)Nc1cc(c(c(c1)OC)OC)OC SEW05526 Cc1c(c(on1)N)c2nc(cs2)c3cccc(c3)C(F)(F)F SPB05485 Cn1cc2c(n1)-c3cc(ccc3SC2)Cl SEW05496 Cc1cc([nH]c1C=C2C(=O)CCCC2=O)C SEW05499 c1cc(c(c(c1)F)S(=O)(=O)NCc2cccs2)F SEW05454 c1cc(c(c(c1)F)S(=O)(=O)N2CCOCC2)F SEW05455 c1cc(c(c(c1)F)S(=O)(=O)Nc2ccc(cc2)Cl)F SEW05456 Cc1cc(no1)c2c(c(no2)C)C(=S)N SPB03635 c1ccc(cc1)NC(=O)Nc2ccccc2Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07569 c1ccc(c(c1)NC(=O)Nc2ccc(cc2F)F)Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07573 Cc1ccc(cc1)S(=O)(=O)Nc2nc(c(s2)C)c3ccc(c(c3)Cl)C XAX00043 Cc1ccc(cc1)SCc2nc(c(c(n2)SC)C#N)c3ccccc3 SPB06404 CCn1c(cc(n1)C)c2nnc(n2c3cccc(c3)C(F)(F)F)SCc4ccccc4 SPB02538 CCn1c(cc(n1)C)c2nnc(n2c3cccc(c3)C(F)(F)F)SC SPB02540 Cc1ccc(c(c1)C)OC(=O)c2c(c(nn2C)C)[N+](=O)[O-] SPB02545 CCOC(=O)CSc1c(ccc(n1)C(=O)C)C#N SPB05486 Cc1c(c(n(n1)C)C(=O)Oc2ccc(cc2)Cl)[N+](=O)[O-] SPB02547 Cc1c(c(n(n1)C)C(=O)NNC(=O)c2csc(n2)C)[N+](=O)[O-] SPB02550 CC(=O)c1ccc(c(n1)SCC(=O)c2ccc(cc2)C#N)C#N SPB05489 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)SCc4ccccc4 SPB00679 CCOC(=O)c1c(nc(s1)c2cccc(c2)C(F)(F)F)O SPB02551 CCn1c(cc(n1)C)C(=O)Sc2ccccc2Cl SPB02556 CCn1c(cc(n1)C)C(=O)Sc2cccc(c2)Cl SPB02557 CCn1c(cc(n1)C)C(=O)Sc2ccc(cc2)C SPB02558 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)SCc4ccccc4Cl SPB00684 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccco3)S SPB00779 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccccc2SCc3c(cc(cn3)C(F)(F)F)Cl SPB06375 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])/C=C/3\C(=O)NC(=S)S3)Cl XAX00149 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)SCC#C SPB00678 CCn1c2ccccc2nc1SCC(=O)OCC SPB02562 Cc1c(c(n(n1)c2ccc(cc2)OC(F)(F)F)c3c(nns3)C)C(=O)O SPB05453 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)Sc4ccc(cc4[N+](=O)[O-])C(F)(F)F SPB00683 Cc1c(c(on1)N)c2nc(cs2)c3ccc(cc3Cl)Cl SPB05464 CC(=O)c1ccc2c(c(sc2n1)C(=O)Nc3ccccc3)N SPB05465 c1ccc2c(c1)-c3ccccc3C2c4ccncc4 SPB06366 c1ccc(cc1)C2(CCOCC2)O SEW05476 c1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)SCc3c(cc(cn3)C(F)(F)F)Cl SPB06374 CCCCCCCCSc1nnc(s1)N XAX00092 Cc1c(c(n(n1)C)C(=O)Oc2cc(cc(c2)Cl)Cl)[N+](=O)[O-] SPB02544 CCn1c(cc(n1)C)C(=O)Oc2ccc(cc2)C SPB02563 c1ccc(cc1)NC(=O)Nc2ccccc2SCc3c(cc(cn3)C(F)(F)F)Cl SPB06377 c1cc(=O)n(cc1C(F)(F)F)CCC#N SPB06383 CCOC(=O)c1c(nc(s1)c2cccc(c2)Cl)O SPB02494 CC(C)(C)/C=N/NC(=O)c1nc(no1)c2c(cccc2Cl)F SPB00724 CSc1nnc(n1c2ccc(cc2)Cl)O SPB00727 c1cc(ccc1n2c(nnc2SCC#N)O)Cl SPB00729 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Nc3ccc(cc3)C SPB07767 Cc1c(c(on1)N)c2nc(cs2)c3ccc(cc3)OC SPB05463 c1ccnc(c1)c2nc(cc(n2)O)N SPB05469 CCCCCCSc1nnc(s1)N XAX00095 CCCCCCCCCCCCCCCCCCSc1nnc(s1)N XAX00094 Cc1cc(no1)c2nnc(n2C)SCC(=O)Nc3ccccc3 SPB06306 Cc1ccc(cc1)Sc2c(c(nc(n2)SC)Sc3ccc(cc3)C)C#N SPB07616 COc1cccc(c1)Sc2c(c(nc(n2)SC)Sc3cccc(c3)OC)C#N SPB07617 Cc1c2ccccc2nc(c1C#N)Sc3[nH]c(nn3)c4cc(cc(c4)Cl)Cl SPB07762 CC(C)NC(=O)O/N=C(/CSc1nccn1C)\N SPB02697 c1ccc2c(c1)n(c(=O)o2)CCC(=O)Nc3ccc(cc3)Cl SPB02701 Cc1ccc(cc1)Sc2c(c(c3ccccc3n2)C)C#N SPB07729 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3Cl SPB07730 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3 SPB07732 Cc1c2ccccc2nc(c1C#N)SCc3ccc(cc3)C(C)(C)C SPB07733 Cc1cc(n(n1)Cc2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3Cl)Cl SPB07772 Cc1cc(nn1C)C(=O)NNc2c(cc(cc2Cl)Cl)Cl SPB00661 CC(C)(C)c1ccc(cc1)c2nnc(n2C(=O)N(C)C)SCc3ccccc3 SPB00586 CC(C)(C)c1ccc(cc1)c2nnc(n2CCCOC)SCC(=O)NNC(=O)C(Cl)(Cl)Cl SPB00591 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)Oc4ccc(cc4)Cl SPB05509 Cc1cc(nn1C)C(=O)N/N=C/C(C)(C)C SPB00656 c1ccc(cc1)CN2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])Sc4ccc(cc4)Br)/SC2=S XAX00155 Cc1cc(nn1C)C(=O)O/N=C/c2c(cccc2Cl)Cl SPB00662 c1cc(c(cc1C2SCCS2)[N+](=O)[O-])Sc3ccc(cn3)C(F)(F)F XAX00159 c1cc(c(cc1C2SCCS2)[N+](=O)[O-])SC3CCCCC3 XAX00160 c1cc(oc1)CSc2ccc(cc2[N+](=O)[O-])C3SCCS3 XAX00161 C#CCSc1n[nH]c(=O)n1c2cccc(c2)Cl SPB00543 Cc1cc(no1)c2c(c(no2)C)C(=O)NNC(=O)NC SPB03606 Cc1cc(no1)c2c(c(no2)C)C(=O)NNS(=O)(=O)C SPB03605 c1cc(cnc1)c2[nH]c(nn2)S SPB00555 CCOC(=O)NNC(=S)Nc1ccccc1C(F)(F)F SPB00553 COC(=O)c1cc(ccc1N2CCOCC2)n3cccc3 SEW05500 Cc1cc([nH]c1C=C2C(=O)OC(OC2=O)(C)C)C SEW05501 COc1ccc(cc1)C(=O)NNC(=O)c2c(cc(cc2OC)C(F)(F)F)C(F)(F)F SEW05505 COCCCNC(=S)NNC(=O)c1c(cc(cc1OC)C(F)(F)F)C(F)(F)F SEW05510 CCOC(=O)NNC(=S)Nc1ccc(cc1)C(C)(C)C SPB07665 COc1cc(cc(c1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(F)(F)F SEW05478 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2ccc(cc2)Cl SPB07691 Cc1c(nc(s1)c2ccc(cc2)Cl)CC(=O)O SEW05487 Cc1c(nccn1)c2ccnn2C(=O)Nc3cc(cc(c3)Cl)Cl SEW05485 CC(C)(C)c1cc(n(n1)C)C(=O)Sc2ccc(cc2)Cl SPB07702 CC(C)(C)c1cc(n(n1)C)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N SPB07698 CN(C)/C=C/C(=C(/C#N)\C(=O)N)/c1ccc(cc1)Cl SEW05489 c1ccc(c(c1)C(=O)NNC(=O)c2c(cccc2F)F)OC(F)(F)F SPB03524 c1ccc(cc1)c2nc(cs2)c3ccnn3C(=O)c4ccc(cc4)F SPB03530 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3NC(=O)Nc4cc(cc(c4)Cl)Cl SPB07748 C/C(=N\OC(=O)c1ccccc1)/c2csc(n2)COc3ccc(cc3)Cl SPB03773 Cc1ccc(cc1)N/C=C(\C#N)/C(=O)c2cc(on2)C(C)(C)C SPB03783 Cc1c2ccccc2nc(c1C#N)SCc3cccc(c3)C(F)(F)F SPB07753 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccc(cc2)C)C#N SPB06427 CC(C)n1c2ccc(cc2nc1SCC(=O)Nc3ccc(cc3)Cl)C(F)(F)F SPB02567 Cc1c(sc(n1)COc2cccc(c2)Cl)c3ccnn3C(=O)C SPB02573 CC(C)(C)OC(=O)Nc1ccc(cc1)Cl SEW05525 Cc1ccc(cc1)NC(=O)c2c(n3c(s2)nc(n3)C(F)(F)F)C SPB05552 CCOC(=O)c1c(nc(s1)c2ccccc2)OC SPB02596 CC(C)n1c2ccc(cc2nc1SCC(=O)Nc3cc(cc(c3)Cl)Cl)Cl SPB02595 CC(=O)c1ccc(c(n1)SCC(=O)Nc2ccc(cc2)C(F)(F)F)C#N SPB05480 CC(C)(C)c1ccc(cc1)OC/C(=N/OC(=O)C(C)(C)C)/N SPB00832 CCOC(=O)c1cc(nc(n1)Sc2ccccc2Cl)C SPB06308 c1ccc(c(c1)N)SCc2c(cc(cn2)C(F)(F)F)Cl SPB06356 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2cccc(c2)OC SPB07537 Cc1c(c(no1)C(=O)NN)c2csc(n2)c3csc(n3)C SPB03708 c1cc(ccc1COc2ccc(cc2Cl)C#N)Cl SPB00697 CC(C)(C)C(=O)O/N=C(/c1ccc(c(c1)Cl)OCc2ccc(cc2)Cl)\N SPB00703 c1cc(ccc1/C=N/O)OC(F)(F)F SPB05555 CC1=C(SCCO1)C(=O)Nc2ccc(cc2)F XBX00014 CC1=C(SCCO1)C(=O)Nc2ccc(cc2Cl)Cl XBX00016 c1ccc(cc1)C(CC(=O)c2cccs2)C#N XBX00018 CC(C)NC(=O)O/N=C(/COc1ccc(cc1)C(C)(C)C)\N SPB00836 c1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)C3SCCS3 SPB00837 c1cc(ccc1Sc2ccc(cc2/C=C/3\C(=O)NC(=S)S3)[N+](=O)[O-])Cl XAX00152 Cc1c(c(no1)C(=O)NNC(=O)Nc2cccc(c2)Cl)c3csc(n3)c4csc(n4)C SPB03717 c1cc2c(cc1F)C(=O)CCS2(=O)=O SEW05415 Cc1c2c(ncnc2SCC(=O)c3ccc(cc3)Cl)on1 SPB05415 c1ccc(cc1)C(=O)Nc2ccccc2Sc3c(cc(cn3)[N+](=O)[O-])C(F)(F)F SPB07561 Cc1nc(cs1)c2nc(on2)C(=O)NN SPB02682 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)O/N=C(/c4cccc(c4)C(F)(F)F)\N SPB05530 CCCOc1ccc(cc1)NC(=O)C SEW05639 CCOC(=O)c1cc(c(nc1C(F)(F)F)Oc2ccc(cc2)C)C#N SPB06475 Cc1nc(cs1)/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/N SPB02656 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)O/N=C(/c4ccc(cc4)Cl)\N SPB05535 CCOC(=O)/C(=C\c1ccc(cc1)[N+](=O)[O-])/[N+](=O)[O-] SPB00688 c1cc(nc(c1)NN=C2CCSCC2)C(F)(F)F SPB06460 c1ccc(cc1)NC(=O)Cn2cccc(c2=O)C(F)(F)F SPB06461 c1cc(cc(c1)Cl)NC(=O)Cn2cccc(c2=O)C(F)(F)F SPB06462 CS(=O)(=O)CS(=O)(=O)NCc1cccs1 SEW05555 c1cc(ccc1c2cnc(o2)SCC(=O)c3ccc(cc3)Cl)Cl SPB02675 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)NNC(=O)c4ccc(cc4)Cl SPB05525 Cc1ccc(cc1)Cn2c(cc(n2)C(=O)Nc3ccccc3)C SPB07776 Cc1ccc(cc1)Cn2c(cc(n2)C(=O)Sc3cccc(c3Cl)Cl)C SPB07778 c1cc(n(c1)c2ccc(cc2)Cl)C=C(C#N)C#N SEW05640 Cc1c(c(no1)c2cccc(c2Cl)Cl)C(=O)C SPB05643 Cc1c(c(n[nH]1)C)Sc2nc3ccccc3s2 SPB07709 Cc1c(sc(n1)c2cccs2)/C(=N\NC(=S)NC3CCCCC3)/C SPB02601 c1cc(ccc1S(=O)(=O)NN)Cl SPB02602 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)NNC(=O)c4cccc(c4)C(F)(F)F SPB05523 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)c4nc(no4)c5cccc(c5)C(F)(F)F SPB05531 c1ccc(c(c1)OCc2nc(cs2)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl)Cl SPB03679 CC1=C(C(C(=C(O1)N)C#N)c2ccco2)C(=O)C XBX00009 c1ccc(cc1)NC2=CC(CC2=O)N3CCN(CC3)c4ccccc4 XBX00010 CC1=C(SCCO1)C(=O)Nc2ccccc2OC XBX00015 CC1=C(SCCO1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F XBX00017 CCOC(=O)/C=C(\c1ccccc1)/Nc2ccccc2SC SPB00809 Cc1cc(nn1Cc2c(cccc2Cl)Cl)C(=O)SCc3ccccc3 SPB07786 Cc1c(c(no1)c2ccccc2)C(=O)O/N=C(/c3csc(n3)C)\N SPB02733 Cc1c(sc(n1)c2cccs2)c3ccnc(n3)SCc4ccc(cc4)Cl SPB02619 c1cc(c(cc1[N+](=O)[O-])/C=C\2/C(=O)NC(=S)S2)Sc3ccc(cn3)C(F)(F)F XAX00168 CSc1nnc(n1c2cccc(c2)C(F)(F)F)O SPB00731 CCCSc1ccc(c(c1)/N=C(/NCCS(=O)(=O)O)\NC(=O)OC)[N+](=O)[O-] XBX00004 Cc1c2ccccc2[nH]c(=O)c1C#N SPB07716 CC(C)(C)C(=O)O/N=C(/Cc1cccc2c1cccc2)\N SPB00830 CN(C)C(=O)Oc1nnc(n1c2ccc(cc2)Cl)SCC=C SPB00742 CC(C)(C)c1ccc(cc1)n2c(=O)[nH]nc2SCc3ccc(cc3)Cl SPB07720 Cc1cc(no1)C(=O)NC(=N)c2ccc(cc2)Cl SPB06443 Cc1c(c(n(n1)C)C(=O)Sc2ccc(cc2)C(F)(F)F)[N+](=O)[O-] SPB02536 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)N3CCCCC3 SPB05540 CC(=O)C(C(=O)C)Sc1[nH]c(nn1)C(F)(F)F SPB05544 CC(=O)C(C(=O)C)Sc1nc2ccccc2s1 SPB07708 Cc1ccc(cc1)c2csc(n2)N/N=C(/C)\c3csc(n3)c4ccccc4.Br SPB03742 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)[N+](=O)[O-] SEW05572 CCN(CC)c1ccc(c(n1)N(CC)CC)[N+](=O)[O-] SEW05573 c1cc(nc(c1[N+](=O)[O-])SCCO)SCCO SEW05575 Cc1c(sc(n1)COc2ccccc2Cl)c3ccnc(n3)N SPB02651 Cc1c(sc(n1)n2cccc2)C(=O)N/N=C/c3ccccc3Cl SPB02692 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)C#N SPB06498 C1CC(C(C(C1)(CO)CO)O)(CO)CO XBX00089 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)Sc3ccccc3 SPB05541 Cc1c(c(n(n1)C)C(=O)Sc2ccc(cc2Cl)Cl)[N+](=O)[O-] SPB02537 CC(C)n1c2ccc(cc2nc1SCC(=O)O)Cl SPB02591 CCn1c2ccc(cc2nc1SCC(=O)O)Cl SPB02593 CC(C)n1c2ccc(cc2nc1SCC(=O)Nc3ccc(cc3)Cl)Cl SPB02594 c1cc(nc(c1[N+](=O)[O-])N2CCCC2)N3CCCC3 SEW05566 c1cc(nc(c1[N+](=O)[O-])N2CCCCC2)N3CCCCC3 SEW05567 CC(C)Cc1ccc(cc1)C(C)C(=O)N2CCN(CC2)c3ccccc3OC SEW05604 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)NC(=O)Nc4ccccc4 SPB05528 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)c4nnc(o4)c5cccc(c5)C(F)(F)F SPB05527 Cc1c(sc(n1)n2cccc2)C(=O)NN SPB02690 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2)C3SCCS3 SPB00848 c1cc(ccc1C2SCCS2)OC(=O)c3ccc(cc3)Cl SPB00851 Cc1c2ccccc2nc(c1C#N)Sc3ccccn3 SPB07735 COC(=O)C(CC(=O)c1cccs1)c2ccccc2 XBX00022 CC(CC#N)C(=O)c1ccccc1 XBX00023 Cc1c(=O)[nH]c2ccccc2n1 XBX00029 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)Sc3ccc(cc3F)F SPB05564 Cc1ccc(c(c1F)C)S(=O)(=O)Oc2ccc(cc2)C3SCCS3 SPB00839 Cc1c2c(ncnc2SCc3ccc(cc3)Cl)on1 SPB05423 Cc1c(c(nc(n1)C(F)(F)F)Sc2ccccc2Cl)Oc3ccccc3.CO SPB05426 CC(C)NC(=O)O/N=C(/Cc1cccc2c1cccc2)\N SPB00844 c1ccc(cc1)C(=O)Oc2ccc(cc2)C3SCCS3 SPB00846 Cc1ccc(cc1)C(=O)CSc2nc3cc(ccc3n2C(C)C)C(F)(F)F SPB02739 CC(C)n1c2ccc(cc2nc1SCC(=O)c3cccc(c3)[N+](=O)[O-])C(F)(F)F SPB02740 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])Sc2[nH]c(nn2)N SPB00949 CCn1c(cc(n1)C)C(=O)Sc2ccc(cn2)C(F)(F)F SPB03838 Cc1cc(no1)C(=O)/C(=C/c2ccc(cc2)OC)/C#N SPB03798 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)Oc3ccccc3Cl SPB05548 Cc1ccc(cc1)OC(=O)c2c(n3c(s2)nc(n3)C(F)(F)F)C SPB05549 c1cc(ccc1C(F)(F)F)NC(=S)NN SPB07687 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2csc(n2)COc3ccc(cc3)Cl SPB03772 c1ccc(cc1)OC(=O)Nc2ccc(cc2Cl)C(F)(F)F SEW05480 c1cc(ccc1C#N)Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW05481 CC(C)c1ccc(cc1)NC(=O)CSc2nc3cc(ccc3n2C(C)C)C(F)(F)F SPB02565 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2nnc(s2)SCc3cccc(c3)C(F)(F)F)C#N SPB06518 Cc1cc(nn1c2ccc(cc2)[N+](=O)[O-])c3nnc(n3C)S SPB00807 CC(C)(C)c1nc(no1)c2cc(ccc2NC(=O)C(C)(C)C)Cl SPB00815 CC(C)(C)c1ccc(cc1)OC/C(=N/OC(=O)N(C)C)/N SPB00834 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3NC(=O)c4ccccc4 SPB07744 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3NC(=O)c4cccs4 SPB07745 Cc1ccc(cc1F)/C(=N/OC(=O)c2cc(n(n2)Cc3c(cccc3Cl)Cl)C)/N SPB07788 Cc1c2ccccc2nc(c1C#N)SCc3c(cccc3Cl)F SPB07734 CC(C)Sc1nnc(n1c2cccc(c2)C(F)(F)F)O SPB00867 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)O/N=C/c3ccc(cc3)OC SPB05561 CC(C)n1c2ccc(cc2nc1SCC(=O)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F SPB02566 CC(C)n1c2ccccc2nc1SCC(=O)O SPB02568 COc1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05458 c1cc(c(c(c1)Cl)/C(=N/OS(=O)(=O)c2ccc(c(c2)Cl)Cl)/C#N)Cl SPB00640 Cc1c2ccccc2nc(c1C#N)Sc3n[nH]c(=O)n3C4CCCCC4 SPB07739 c1ccc(cc1)/C=N/NC(=S)Nc2ccccc2F SPB07740 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3N SPB07741 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3NC(=O)c4ccc(cc4)Cl SPB07742 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05608 Cc1nc(cs1)/C(=N/OC(=O)c2c(cccc2Cl)F)/N SPB02655 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2[nH]c(nn2)C(F)(F)F)C#N SPB06497 Cc1c(nc(nc1Sc2[nH]c(nn2)c3ccccc3)C(F)(F)F)C SPB06501 c1ccc(cc1)NC(=O)O/N=C(/Cc2cccc3c2cccc3)\N SPB00840 Cc1c2ccccc2nc(c1C#N)SCc3ccc(cc3)Cl SPB07751 c1cc(c(cc1c2cc(on2)c3csc(n3)c4ccc(cn4)C(F)(F)F)Cl)Cl SPB06452 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(\C#N)/c3c(cccc3Cl)Cl SPB00641 Cc1c(sc(n1)c2cccs2)c3ccnc(n3)C SPB02641 Cc1c(n(c(c1S(=O)(=O)C(C)C)N)Cc2ccc(cc2Cl)Cl)C SPB02642 c1cc(c(c(c1)Cl)C(=O)Oc2ccc(cc2)C3SCCS3)F SPB00847 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)O/N=C/c3ccc(cc3)OC(F)(F)F SPB05559 c1cc(ccc1c2nc(on2)CSc3nc([nH]n3)N)Cl SPB00854 CC(=O)N(CC(=O)O)c1ccccc1C(=O)O SEW05508 Cc1cc([nH]c1C=C2C(=O)NC(=S)NC2=O)C SEW05512 Cc1ccc(cc1)C(=O)Nc2ccccc2Sc3c(c(c4ccccc4n3)C)C#N SPB07743 COc1cc(cc(c1C(=O)Oc2ccc(cc2)Cl)C(F)(F)F)C(F)(F)F SEW05513 Cc1cc(n(n1)Cc2cccc(c2)C(F)(F)F)C(=O)Nc3ccc(cc3)C4CCCCC4 SPB07773 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3Cl)Cl)C(=O)C1)C XAX00140 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])/C=C/3\C(=O)NC(=S)S3 XAX00145 CCn1c(cc(n1)C)C(=O)Sc2ccc(cc2Cl)Cl SPB02559 CCOC(=O)c1csc(n1)c2cccc(c2)C(F)(F)F SPB02560 CC(=O)Nc1cc(nc(n1)c2ccccn2)O SPB05562 Cc1c(sc(n1)COc2ccccc2Cl)C(=O)C SPB02599 CC(C)(C)c1cc(n(n1)C)C(=O)O/N=C(/c2ccccc2)\N SPB07700 CC(C)(C)c1cc(n(n1)C)C(=O)O/N=C/c2ccccc2 SPB07701 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2nnc(s2)SCC3CC3)C#N SPB06519 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2nnc(s2)SC)C#N SPB06520 CCOC(=O)c1c(nc(s1)c2ccccc2)CSc3nccn3C SPB02751 CCn1c(cc(n1)C)C(=O)NNC(=O)c2ccccc2Cl SPB02753 c1cc(ccc1Sc2ccc(cn2)C#N)Cl SEW05587 CCOC(=O)c1cnc(nc1Sc2[nH]c(nn2)c3cccs3)C(F)(F)F SPB06521 c1cc([nH]c1)C(=O)NNC(=O)Nc2cc(cc(c2)Cl)Cl SEW05637 c1ccc(cc1)NC(=O)NNC(=O)c2ccc[nH]2 SEW05638 CN(C)/C=N/NC(=O)Cc1csc2n1nc(n2)c3ccccc3 SPB00692 CC(=O)c1ccc2c(c(sc2n1)C(=O)Nc3cc(cc(c3)Cl)Cl)N SPB05466 CC(=O)c1ccc2c(c(sc2n1)C(=O)Nc3ccc(cc3)C(F)(F)F)N SPB05467 c1ccc(cc1)C(=O)CN2C(=O)CCC2=O SPB00702 c1ccc(cc1)C(=O)CNC(=O)CCC(=O)O SPB00706 Cc1c(c([nH]n1)c2cccs2)C(=O)N/N=C/c3ccc(s3)[N+](=O)[O-] SPB00948 Cc1cc(nn1Cc2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)C(C)(C)C SPB07783 Cc1cc(nn1Cc2c(cccc2Cl)Cl)C(=O)Sc3ccc(cc3)OC SPB07784 Cc1cc(nn1Cc2c(cccc2Cl)Cl)C(=O)O/N=C(/c3cccc(c3Cl)Cl)\N SPB07789 COC(=S)Nc1ccccc1Cl SEW05584 CCCCNC(=O)n1c(ccn1)c2c(nc(s2)c3cccs3)C SPB02626 c1ccc(cc1)Sc2ccc(cn2)C#N SEW05586 c1cc(c(cc1/C=C/2\C(=O)NC(=S)S2)[N+](=O)[O-])Sc3ccc(cn3)C(F)(F)F XAX00167 c1ccc(c(c1)OCc2nc(cs2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl)Cl SPB03678 c1ccc(c(c1)OCc2nc(cs2)c3ccnc(n3)SCC(=O)Nc4cccc(c4)Cl)Cl SPB03681 CCCCCCCCSc1nnc(s1)N/C=N/O XAX00096 Cc1ccc(cc1)CSc2nnc(n2c3ccc(cc3)C(C)(C)C)c4ccccc4Cl SPB00795 c1c(cnc(c1Cl)C(=S)N)C(F)(F)F SPB05587 Cc1c(c(n[nH]1)C)Sc2ccc(cc2)Cl SPB07713 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)NC(=O)O/N=C(\c4ccccc4)/N SPB05588 Cc1c(c(no1)c2ccccc2)C(=O)NNc3c(cc(cn3)C(F)(F)F)Cl SPB06486 Cc1cc(nn1Cc2c(cccc2Cl)Cl)C(=O)Sc3ccccc3Cl SPB07785 c1cc(ccc1/C=N/NC(=O)Nc2ccc(cc2Cl)C(F)(F)F)C(F)(F)F SEW05551 c1cc(c(cc1Cl)Cl)C2CC=CCC2C(=O)O SEW05553 Cc1ccc(cc1)OC(=O)c2c(n3c(s2)nc(n3)c4ccc(cc4)Cl)C SPB05510 c1cc2c(cc1F)/C(=N/NC(=S)N)/CCO2 SEW05543 Cc1c(c(no1)C(=O)NNC(=O)c2ccccc2)c3csc(n3)c4csc(n4)C SPB03711 c1ccc(cc1)Oc2ccc(cn2)/C=C(\C#N)/S(=O)(=O)c3ccccc3 SEW05539 CCOC(=O)c1cc(nc(c1C#N)Sc2ccccc2NC(=O)Nc3ccc(cc3)Cl)C SPB06419 c1cnoc1C(=O)Oc2cc(cc(c2)Cl)Cl SPB03697 CC(=O)c1csc(n1)c2ccc(cc2)C(F)(F)F SPB03698 Cc1cc(no1)c2c(c(no2)C)c3nc(on3)C SPB03633 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNc3cccc(n3)C(F)(F)F SPB06487 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNc3cccc(n3)C(F)(F)F SPB06488 c1ccc(c(c1)C(F)(F)F)n2cnnc2S SPB07694 CC(C)(C)c1cc(n(n1)C)C(=O)Oc2ccc(cc2)C(F)(F)F SPB07699 CC(=O)Nc1ccc(cc1)OC(=O)c2cccc(n2)C(F)(F)F SPB06493 CC(C)(C)c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)F)c4ccccc4Cl SPB00797 CC(C)(C)c1cc(n(n1)C)C(=O)O/N=C/c2c(cccc2Cl)Cl SPB07703 Cc1c(sc(n1)COc2ccccc2Cl)c3ccnc(n3)SCc4ccc(cc4)Cl SPB02609 Cc1c(sc(n1)c2cccs2)c3ccnc(n3)S SPB02613 c1ccc(cc1)C(=O)Cn2cccc(c2=O)C(F)(F)F SPB06466 CCOC(=O)c1cc(c(nc1C(F)(F)F)Oc2ccccc2)C#N SPB06474 Cc1cc(no1)c2c(c(no2)C)C(=O)NC(=O)Nc3ccccc3 SPB03636 CC1=C(SCCO1)C(=O)Nc2ccccc2 XBX00001 c1ccc(cc1)COc2ccc3c(c2)cc[nH]3 XBX00005 CC1=C(S(=O)CCO1)C(=O)Nc2ccccc2 XBX00006 c1ccc(cc1)C2(C(=O)NC(=O)N2)C3CCC3 XBX00048 Cc1c(c(no1)C(=O)N/N=C/c2cccs2)c3csc(n3)c4csc(n4)C SPB03720 Cc1c(c(no1)C(=O)N/N=C/c2ccc(cc2)Cl)c3csc(n3)c4csc(n4)C SPB03721 Cc1cc(n2c(n1)nc(n2)Sc3ccc(cn3)[N+](=O)[O-])C SPB00943 Cc1cc(n2c(n1)nc(n2)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F)C SPB00944 Cc1c(sc(n1)COc2ccccc2Cl)C(=O)/C=C/N(C)C SPB02606 Cc1nc(cs1)/C(=N/O)/N SPB02633 Cc1ccc(cc1)Cn2cccc(c2=O)C(F)(F)F SPB06456 c1cc(c(=O)n(c1)Cc2cc(cc(c2)Cl)Cl)C(F)(F)F SPB06457 Cc1ccc(cc1)Cn2c(cc(n2)C(=O)O/N=C(/c3cccc(c3)C(F)(F)F)\N)C SPB07780 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3NC(=O)Nc4cccc(c4)C(F)(F)F SPB07763 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Nc3ccccc3Cl SPB07765 CS(=O)(=O)CS(=O)(=O)Nc1cccc(c1)OC(F)(F)F SEW05556 c1cc(c(cc1F)F)c2nc(cs2)C(=O)N SPB02702 c1cc(c(cc1F)F)c2nc(cs2)C#N SPB02703 Cc1c(sc(n1)COc2ccccc2Cl)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl SPB02704 Cc1cc([nH]c1C=C2C(=O)NC(=O)NC2=O)C SEW05497 Cc1cc(no1)NC(=O)c2c(cc(cc2OC)C(F)(F)F)C(F)(F)F SEW05504 Cc1c(sc(n1)c2csc(n2)C)C(=O)NNC(=O)Nc3ccccc3 SPB03648 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Sc3cccc(c3)C(F)(F)F SPB07771 Cc1ccc(cc1)Cn2c(cc(n2)C(=O)Nc3ccc(cc3)Br)C SPB07775 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C3SCCS3 XAX00162 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2[nH]c(nn2)C(C)(C)C)C#N SPB06499 Cc1c(c(n(n1)C)C(=O)Nc2ccccc2)[N+](=O)[O-] SPB07817 Cc1ccc(cc1)/C(=N/OC(=O)c2cc(n(n2)Cc3c(cccc3Cl)Cl)C)/N SPB07787 Cn1c(nnc1Sc2ccc(c(n2)Sc3nnc(n3C)C(F)(F)F)[N+](=O)[O-])C(F)(F)F SEW05582 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])/C=C/3\C(=O)NC(=S)S3 XAX00165 CC(=O)c1ccc(c(n1)SCC(=O)Nc2ccccc2Cl)C#N SPB05481 CC(=O)c1ccc(c(n1)SCC(=O)Nc2cc(cc(c2)Cl)Cl)C#N SPB05482 CC(=O)CSc1c(ccc(n1)C(=O)C)C#N SPB05483 C/C(=N\Nc1cc(ccc1Cl)Cl)/c2csc(n2)COc3ccc(cc3)Cl SPB03767 CC(C)(C)c1ccc(cc1)n2c(=O)[nH]nc2SCc3ccc(c(c3)Cl)Cl SPB07719 C=CCSc1nnc(n1c2cccc(c2)C(F)(F)F)O SPB00732 COc1cc(cc(c1C(=O)O)C(F)(F)F)C(F)(F)F SEW05446 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C3SCCS3)Cl XAX00164 Cc1c2ccccc2nc(c1C#N)Sc3cccc(c3)C(F)(F)F SPB07731 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)Nc3ccc(cc3)OC(F)(F)F SEW05530 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C3SCCS3)Br XAX00166 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)Nc3ccccc3C(F)(F)F SEW05531 Cc1c(c(no1)C(=O)NNC(=O)c2ccc(cc2)Cl)c3csc(n3)c4csc(n4)C SPB03712 c1ccc(cc1)Oc2ccc(cn2)/C=C\3/c4ccccc4NC3=O SEW05540 Cc1c(c(no1)C(=O)OC)/C(=N/OC(=O)c2ccc(cc2)Cl)/C SPB03714 CC(C)(C)c1cc(no1)C(=O)/C(=C/c2ccc(cc2)OC)/C#N SPB03770 c1cc(nc(c1)C(F)(F)F)C(=O)Oc2cc(cc(c2)Cl)Cl SPB06492 COc1ccc(cc1)Nc2ccc(c(n2)Nc3ccc(cc3)OC)[N+](=O)[O-] SEW05576 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3cccc(c3)C(F)(F)F SEW05449 CCn1c(cc(n1)C)c2nnc(n2c3ccccc3)SCC(=O)Nc4ccccc4 SPB02502 CC(C)(C)c1ccc(cc1)OCC(=N)NC(=O)c2ccc(cc2)OC(F)(F)F SPB06422 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)SC SPB00676 CC(C)(C)c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)c4ccccc4Cl SPB00796 CCOC(=O)c1c(cnn1C(=O)Nc2cccc(c2)Cl)Sc3ccccc3 SPB03702 Cc1c(c(no1)C(=O)OC)c2ccnn2C(=O)c3ccc(cc3)Cl SPB03722 Cc1c(c(no1)C(=O)OC)c2ccnn2C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB03724 CS(=O)(=O)CS(=O)(=O)Nc1cc(cc(c1)Cl)Cl SEW05534 Cc1c(sc(n1)c2ccccc2)C(=O)O SPB03749 c1c(cnc(c1Cl)NN=C2CCSCC2)C(F)(F)F SPB06458 c1ccc2c(c1)/C(=C/c3cccn3c4ccc(cc4)Cl)/C(=O)N2 SEW05650 CCCOc1ccc(cc1)NC(=O)c2ccccc2C(=O)O SEW05653 c1ccc(cc1)C(C#N)N(CCO)CCO XBX00114 COC(=O)c1c(ccs1)NC(=O)c2ccno2 SPB03853 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(c3c(nc(nc3s2)c4ccccc4OC)C)C SPB05577 Cc1ccc(cc1)SC(=O)c2c(n3c(s2)nc(n3)C(F)(F)F)C SPB05542 Cc1cccc(c1OC(=O)c2cc(nn2C)C(C)(C)C)Cl SPB07707 Cc1c(sc(n1)c2cccs2)C(=O)/C=C/N(C)C SPB02608 CCn1c(cc(n1)C)c2nnc(o2)SCc3ccc(cc3)C(F)(F)F SPB02765 Cc1ccc(cc1)C(=O)O/N=C(/c2ccc(cn2)C(F)(F)F)\N SPB05629 COC(c1c(cnc(n1)SCC#C)C(=O)O)OC SPB05669 c1ccc2c(c1)ccc(c2/N=N/c3ccccc3OC(F)(F)F)O SEW05571 Cc1c(c(on1)C)C(=O)Nc2ccc(nc2N3CCOCC3)N4CCOCC4 SEW05610 CCn1c(c(c(n1)C)Br)C(=O)Sc2ccc(cc2)OC SPB02768 CCn1c(c(c(n1)C)Br)C(=O)Oc2ccc(cc2)Cl SPB02774 Cc1c(sc2n1nc(n2)C(F)(F)F)c3ccn[nH]3 SPB05631 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2ccc[nH]2 SEW05656 c1ccc(cc1)C2C(=NC(=O)N2)c3ccccc3 XBX00119 CCOC(=O)c1c(nc(s1)c2ccccc2)OCc3c(cccc3Cl)Cl SPB02718 COC(=O)c1cc(=O)n2c(nnc2s1)c3cc(cc(c3)Cl)Cl SPB05608 c1c(c[nH]c1C(=O)NN)Br SEW05620 Cc1c(sc(n1)COc2ccccc2Cl)c3ccnc(n3)SCC#C SPB02611 Cc1c(sc(n1)c2cccs2)c3ccn[nH]3 SPB02612 CS/C(=N\C#N)/NCCO XBX00002 Cc1ccc(cc1)CSc2n[nH]c(=O)n2c3ccc(cc3)C(C)(C)C SPB07721 COC(c1c(cnc(n1)SCc2ccc(cc2)Cl)C(=O)O)OC SPB05671 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)NC(=O)Nc4ccc(cc4Cl)Cl SPB05583 CC(C)Sc1n[nH]c(=O)n1c2ccc3c(c2)OCCO3 SPB07906 CC(C)OC(=O)Nc1ccc(cc1)Cl SPB07910 CC(C)(C)C(=O)N1CCN(CC1)C2c3ccccc3-c4c2cccc4 SPB06565 c1ccn(c1)c2cccc(c2)C3=NC(=O)C(S3)CC(=O)O SPB02674 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(/c3csc(n3)C)\N SPB02734 c1c(cc(cc1Cl)Cl)/C(=N/O)/N SPB05592 CC(C)OC(=O)Nc1cc(cc(c1)Cl)Cl SPB07912 Cc1cc(no1)C(=O)NNC(=O)c2c(onc2c3ccccc3)C SPB02786 Cc1cc(no1)C(=O)NNC(=O)c2c(onc2c3ccccc3Cl)C SPB02787 CCOC(=O)NNC(=S)Nc1ccc(cc1)OCc2ccccc2 SPB07852 CC(C)n1c2ccc(cc2nc1SCC(=O)c3ccc(cc3)Cl)C(F)(F)F SPB02741 c1cc2c(cc1Cl)sc(n2)N3CCOCC3 SEW05618 c1cc(ccc1CSc2n[nH]c(=O)n2C3CC4CC3C=C4)Cl SPB07723 CN(C)C(=O)Oc1nnc(n1c2cccc(c2)C(F)(F)F)SCC=C SPB00744 CC(C)(C)c1ccc(cc1)C(=O)NNC(=S)NCc2ccco2 SPB00772 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccco3)SC SPB00783 Cc1cc(n2c(n1)nc(n2)Sc3c(cccn3)[N+](=O)[O-])C SPB00942 Cc1cc(cc(c1)OCCC#N)C XBX00211 CN(C)NC(=O)CCC(=O)O XBX00214 Cc1cc(n2c(n1)nc(n2)Sc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C SPB00945 C/C(=N\NC(=S)N)/c1ccc(cc1)OCCCOc2ccc(cc2)/C(=N/NC(=S)N)/C SEW05565 c1ccc(cc1)c2csc(n2)c3cccc(c3)n4cccc4 SPB01090 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Sc3ccc(cn3)C(F)(F)F SPB03906 COC(=O)c1cccn1S(=O)(=O)c2ccc(cc2)Cl SEW05624 COC(=O)c1cc(=O)n2c(nnc2s1)c3ccccc3 SPB05603 CCOC(=O)c1c(n2c(s1)nc(n2)C(F)(F)F)CSc3nnc(n3C)C(F)(F)F SPB05602 c1cc(ccc1/C=c/2\c(=O)n3c(s2)nc(n3)c4ccc(cc4)Cl)Cl SPB05604 Cc1c(nc(nc1Sc2[nH]c(nn2)c3cccs3)C(F)(F)F)C SPB06503 c1ccc(c(c1)c2ccc(c(n2)Sc3ccccc3N)[N+](=O)[O-])N SEW05581 c1ccc2c(c1)cccc2C/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N SPB00841 CCOc1ccccc1NC(=O)O/N=C(/Cc2cccc3c2cccc3)\N SPB00842 c1ccc2c(c1)n(c(=O)o2)CCC(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N SPB02713 CC1(C(=O)NC(=O)N1)C2CC2 XBX00046 CC(C)c1ccc(cc1)NC(=O)CSc2ncc(o2)c3ccc(cc3)Cl SPB02672 c1cc(cc(c1)NC(=O)CSc2nnc(n2c3ccc(cc3)Cl)c4ccc(nc4)OCC(F)(F)F)C(F)(F)F SPB06606 c1ccc2c(c1)n(c(=O)o2)CCc3nc(no3)c4ccc(cc4)C(F)(F)F SPB02716 CC(C)(C)c1ccc(cc1)c2nc(on2)CCn3c4ccccc4oc3=O SPB02717 c1ccc2c(c1)ccc(c2CN3CCCCC3)O XBX00103 CC1=N/C(=C\c2cccc(c2)[N+](=O)[O-])/C(=O)O1 XBX00090 CCOC(=O)NNC(=S)Nc1ccc2c(c1)OCCO2 SPB07853 c1ccc(cc1)CN(CCC#N)CN2C(=O)c3ccccc3C2=O SW00045 CC(C)Nc1ccc(cc1[N+](=O)[O-])C(F)(F)F TG00008 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCC(=O)c4ccccc4)c5ccco5 SPB07908 c1ccnc(c1)c2ccc(c(=O)[nH]2)C#N SPB07833 c1cc(ccc1CSc2[nH]nc(n2)N)Cl SPB00856 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)NC(=O)O/N=C(\c4ccc(cc4)OC(F)(F)F)/N SPB05589 c1cc(ccc1CSc2ncc(o2)c3ccc(cc3)Cl)C(F)(F)F SPB02678 c1cc(c(c(c1)Cl)CSc2ncc(o2)c3ccc(cc3)Cl)Cl SPB02679 Cc1cc(n2c(n1)nc(n2)SC)C SPB00860 COc1ccc(cc1)n2c(nnc2S)c3ccc(cc3)OC(F)(F)F SPB03795 CCOC(=O)c1c(nc(s1)c2ccccc2)OCc3ccccc3Cl SPB02724 c1ccc(cc1)C2CC(=NNC2=O)c3cccs3 XBX00031 CCCCCn1c(=O)[nH]nc1Sc2c(c(c3ccccc3n2)C)C#N SPB07752 CC(C)(C)c1cc(no1)C(=O)/C(=N/Nc2ccccc2)/C#N SPB03785 Cc1ccc(cc1)N/N=C(\C#N)/C(=O)c2cc(on2)C(C)(C)C SPB03786 C/C(=C(\C(=O)c1ccc(cc1Cl)Cl)/C(=O)OC)/NC SPB00905 CN(C)/C=N/NS(=O)(=O)c1ccc(c(c1)Cl)Cl SPB00873 CN(C)C(=O)Oc1ccc(cc1)C2SCCS2 SPB00877 Cc1ccc(cc1)C2CC=CCC2[N+](=O)[O-] SEW05616 CC(C)(C)c1cc(no1)C(=O)/C(=N/Nc2ccc(cc2)Cl)/C#N SPB03788 c1ccc(c(c1)NC(=S)NNC(=O)c2ccc(cc2)OC(F)(F)F)Cl SPB03792 CC(C)(C)C(=O)Nc1ccccc1Sc2ccc(c(n2)Sc3ccccc3NC(=O)C(C)(C)C)[N+](=O)[O-] SEW05589 c1ccc(c(c1)NC(=O)C(Cl)(Cl)Cl)Sc2ccc(c(n2)Sc3ccccc3NC(=O)C(Cl)(Cl)Cl)[N+](=O)[O-] SEW05590 Cc1c(c(no1)C(=O)OC)/C(=N/OC(=O)Nc2ccccc2)/C SPB03728 Cc1c(c(no1)C(=O)OC)/C(=N/OC(=O)Nc2ccc(cc2)Cl)/C SPB03729 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Nc3ccc(cc3)Cl SPB07764 CC(C)c1ccc(cc1)n2c(nnc2SCc3c(cccc3Cl)F)c4ccc(cc4)C(C)(C)C SPB01085 c1cc(c(nc1)SCC(=O)c2ccc(cc2)Cl)C(F)(F)F SPB03888 COC(c1c(cnc(n1)SCc2c(cccc2Cl)Cl)C(=O)O)OC SPB05670 Cc1ccc(cc1)N/N=C(\C#N)/C(=O)c2cc(nn2C(C)(C)C)C SPB03808 CN1CN(C(=S)SC1)C XBX00215 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3S SPB07854 c1ccc(cc1)CSc2[nH]nc(n2)N SPB00866 c1ccc2c(c1)nc3n2CC(CS3)O SPB00879 c1ccc2c(c1)nc3n2CC(CS3)OC(=O)c4ccc(o4)[N+](=O)[O-] SPB00880 COc1ccc(c(n1)OC)NC(=O)Nc2ccc(cc2)OC(F)(F)F SEW05628 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2ccccc2OC SPB07693 c1ccc(cc1)C(=O)CCCCCCCCC(=O)O XBX00045 c1ccc(cc1)C(=O)Cc2cccc(c2)CC(=O)c3ccccc3 XBX00053 c1cc(ccc1S(=O)(=O)c2ccc(cn2)C#N)Cl SEW05598 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(nc2N3CCOCC3)N4CCOCC4 SEW05601 Cc1c(c(on1)C)C(=O)N2CCN(CC2)c3ccccc3OC SEW05602 CC\1(C2CCC(C2)/C1=C/CC(=O)O)C XBX00219 CCOc1ccccc1CCC(=O)O XBX00227 Cc1c(snn1)c2nc(cs2)/C(=N/O)/C SPB03847 c1ccc(cc1)C(=O)Cc2ccc(cc2)CC(=O)c3ccccc3 XBX00054 C1CCC(CC1)(C#N)NNC2(CCCCC2)C#N XBX00088 CCOC(=O)c1cnc(nc1Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)C(F)(F)F SPB06523 COc1ccc(c(n1)OC)NS(=O)(=O)c2ccc(cc2)Cl SEW05641 c1ccc2c(c1)ccc(c2CN3CCOCC3)O XBX00104 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCC(=O)c4ccc(cc4)C#N)c5ccco5 SPB07909 CCn1c(cc(n1)C)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F SPB02755 CC(C)(C)c1nc(no1)c2ccc(cn2)C(F)(F)F SPB05634 CCOC(=O)c1cnc(nc1O)COc2ccc(cc2)C(C)(C)C SPB05636 Cc1ccc(cc1)Cn2c(cc(n2)C(=O)O/N=C(/c3ccccc3)\N)C SPB07779 CN(C)/C=N/NS(=O)(=O)c1ccccc1 SPB00872 c1cc(c(c(c1)Cl)CSc2[nH]nc(n2)N)Cl SPB00858 c1cc(c(c(c1)Cl)CSc2[nH]nc(n2)N)F SPB00859 c1cc(cc(c1)n2c(nnc2S)c3ccc(cc3)OC(F)(F)F)C(F)(F)F SPB03823 c1cc(ccc1CSc2c(cc(cn2)C(F)(F)F)Cl)Cl SPB03825 CCOC(=O)Cc1csc(n1)c2ccc(cc2F)F SPB02719 c1ccc(cc1)C(=O)N2C=Cc3ccccc3C2C#N XBX00102 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)NC(=O)NNc4ccc(cc4)OC(F)(F)F SPB05662 Cc1c(sc(n1)n2cccc2)C(=O)N/N=C/c3ccc(cc3)Cl SPB02691 Cc1ccc(cc1)SC(=O)c2cc(nn2Cc3cccc(c3)C(F)(F)F)C SPB07774 CN(c1c(cccn1)[N+](=O)[O-])NS(=O)(=O)CS(=O)(=O)C SEW05535 CC1(OC(=O)C(=Cc2ccc(nc2)Oc3ccccc3)C(=O)O1)C SEW05541 Cc1ccc(cc1)Cn2c(cc(n2)C(=O)Sc3ccc(cc3)NC(=O)C)C SPB07777 CC(=O)Nc1ccccc1Sc2ccc(c(n2)Sc3ccccc3NC(=O)C)[N+](=O)[O-] SEW05588 Cc1cc(nn1Cc2c(cccc2Cl)Cl)C(=O)Nc3ccccc3C(F)(F)F SPB07781 c1cc2c(cc1Cl)/C(=N/NC(=S)N)/CCS2 SEW05542 CC/C(=N\NC(=O)OCC)/c1ccc(cc1)c2ccccc2F SEW05547 CCOC(=O)N/N=C(/c1c(cccc1)c2c(cccc2)/C(=N/NC(=O)OCC)/C)\C SEW05548 CC(C)(C)c1cc(no1)C(=O)/C(=N/Nc2cccc(c2)Cl)/C#N SPB03787 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)NC(=O)O/N=C(\c4ccc(cc4Cl)Cl)/N SPB05623 c1ccc(cc1)/C=c/2\c(=O)n3c(s2)nc(n3)c4ccc(cc4)Cl SPB05609 Cc1c(sc2n1nc(n2)C(F)(F)F)/C(=N/O)/C SPB05610 CCOC(=O)c1c(nc(s1)c2ccccc2)OCc3ccc(cc3)Cl SPB02723 c1ccc(c(c1)NC(=O)c2cccs2)Sc3ccc(c(n3)Sc4ccccc4NC(=O)c5cccs5)[N+](=O)[O-] SEW05591 c1cc(ncc1C#N)N2CCOCC2 SEW05595 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2ccccc2 SPB07690 Cc1c(snn1)C(=O)O/N=C(\COc2ccc(cc2)C3SCCS3)/N SPB02638 Cc1ccc(cc1)C(=O)Sc2c(cc(cn2)C(F)(F)F)Cl SPB03818 CC(C)(C)c1cc(no1)C(=O)/C=C\2/NC(=O)CS2 SPB03822 CC(=O)Nc1ccc(c(c1)OC)/C=N/NC(=S)N XBX00144 CC(C)n1c2ccc(cc2nc1SCC(=O)NNC(=O)c3ccc(cc3)Cl)C(F)(F)F SPB03896 COc1ccc2c(c1)c(c3ccccc3n2)N XBX00150 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)CC2=NC(=O)CS2 SPB05633 c1cc([nH]c(=O)c1C#N)c2ccncc2 SPB07835 COCc1cc(nc(n1)c2ccc(cn2)C(F)(F)F)O SPB05678 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2c(onc2C(=O)OC)C SPB03715 Cc1cccc(c1NC(=O)NNC(=O)c2c(c(on2)C)c3csc(n3)c4csc(n4)C)C SPB03718 CC(C)n1c2ccc(cc2nc1Sc3ncc(s3)[N+](=O)[O-])C(F)(F)F SPB02620 CCn1c(cc(n1)C)c2nnc(o2)c3ccccc3Cl SPB02762 CN(C)/C=N/NC(=O)c1ccccc1Cl SPB00869 CC(C)Sc1nnc(n1c2ccccc2)OC(=O)N(C)C SPB00870 Cc1c(sc2n1nc(n2)C(F)(F)F)/C(=N/OC(=O)Nc3ccccc3)/C SPB05617 c1cc(cc(c1)C(F)(F)F)C(=O)Sc2c(cccn2)C(F)(F)F SPB03900 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4ccccc4OC SEW05607 CCc1ccc(cc1)NCN2C(=O)c3ccccc3C2=O XBX00272 C/C(=N\NC(=O)c1ccncc1)/Cc2ccccc2 XBX00286 CSc1cccc(c1)NC(=O)CSc2nnc(n2c3ccc(cc3)Cl)c4ccc(nc4)OCC(F)(F)F SPB06607 c1ccc2c(c1)n(c(=O)o2)CCC#N SPB02694 CC(C)n1c2ccc(cc2nc1Sc3ncc(s3)[N+](=O)[O-])Cl SPB02621 Cc1c2cc(ccc2sc1c3csc(n3)c4c(cc(cn4)C(F)(F)F)Cl)Cl SPB06478 c1cc(ccc1C2SCCS2)OS(=O)(=O)c3ccc(c(c3)Cl)Cl SPB00838 Cc1c(c(no1)C(=O)NNS(=O)(=O)c2ccc(cc2)Cl)c3csc(n3)c4csc(n4)C SPB03727 CSc1nc(nc(n1)N)COc2ccccc2Cl SPB05666 COc1ccc(cc1)OCc2nc(nc(n2)SC)N SPB05667 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5cccs5 SPB06562 c1cc2c(cc1F)c(c3c(n2)CCCCC3)C(=O)O SEW05649 Cc1c(c(on1)N(C(=O)C)C(=O)C)c2nc(cs2)c3ccc(cc3)OC SPB05605 c1cc(cc(c1)Cl)NC(=O)CSc2c(cc(cn2)C(F)(F)F)Cl SPB03834 Cc1ccc(cc1Cl)NC(=O)OC(C)C SPB07913 CCn1c(cc(n1)C)c2nnc(o2)SCc3c(cccc3Cl)Cl SPB02767 Cc1cccc(c1NC(=S)N2CC(OC(C2)C)C)Cl SW00009 Cc1cccc(c1NC(=S)Nc2cccc(c2)C(F)(F)F)Cl SW00010 CN(C)Cc1c2ccccc2ccc1O XBX00115 c1ccc(cc1)C2=NN=C(NN2)c3ccccc3 XBX00117 Cc1c(sc2n1nc(n2)C(F)(F)F)/C(=N/OC(=O)c3ccccc3)/C SPB05611 c1ccc(c(c1)N2C(=O)/C(=C\c3ccc(c(c3)[N+](=O)[O-])SC4CCCCC4)/SC2=S)Cl XAX00156 CC(=O)c1ccc(c(n1)SCC(=O)c2ccccc2)C#N SPB05484 c1cc(c(nc1)SCc2ccc(cc2)Cl)C(F)(F)F SPB03886 Cc1ccc(cc1)CSc2c(cccn2)C(F)(F)F SPB03887 c1cc(cc(c1)C(F)(F)F)C(=O)CSc2c(cccn2)C(F)(F)F SPB03889 c1cc(c(nc1)SCC#N)C(F)(F)F SPB03892 c1cc([nH]c1)C(=O)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW05648 CC(=NNC(=O)NCc1ccccc1)C XBX00145 c1ccc2c(c1)n(c(=O)o2)CCC(=O)Sc3c(cc(cc3Cl)Cl)Cl SPB02721 c1cc(ccc1c2nnc(o2)CSc3nnc(s3)SCC4CC4)Cl SPB02781 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl SEW05614 Cc1cccc(c1NC(=S)NCCc2ccccn2)Cl SW00013 CCOC(=O)c1cnc(nc1O)c2ccccn2 SPB05487 CC1C/C(=N\NC(=S)N)/c2cc(ccc2S1)Cl SEW05544 c1cc2c(cc1Cl)/C(=N/NC(=S)N)/CCO2 SEW05545 CCC(CC)(c1cc(c(c(c1)C)O)C)c2cc(c(c(c2)C)O)C XBX00099 c1ccc(cc1)C(C#N)N2CCCCC2 XBX00107 c1cc(c(cc1F)F)c2nc(cs2)/C(=N\OC(=O)C3CC3)/N SPB02709 c1ccc2c(c1)n(c(=O)o2)CCC(=O)O/N=C(/c3ccc(cc3)Cl)\N SPB02712 c1cc(sc1)C(=O)O/N=C(/c2cc(c(c(c2)Cl)N)Cl)\N SEW05564 CC(C)OC(=O)Nc1ccc(c(c1)Cl)Cl SPB07911 Cc1c(snn1)c2nc(cs2)/C(=N/OC(=O)c3ccc(cc3)Cl)/C SPB03850 Cc1c(noc1NC(=O)Cn2nc(nn2)c3cccc(c3)C(F)(F)F)C SPB03951 COC(c1c(cnc(n1)S)C(=O)O)OC SPB05672 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3csc(n3)C)\N SPB02735 CCOC(=O)c1cnc(nc1O)COc2ccc(cc2)OC SPB05646 CC(=O)c1ccc(cc1)OCCCOc2ccc(cc2)C(=O)C SEW05552 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)O/N=C/c4ccc(cc4Cl)Cl SPB05515 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)NNC(=O)C SPB05522 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)C SPB05545 c1cc(ccc1C(=O)NC(=N)c2ccc(cn2)C(F)(F)F)OC(F)(F)F SPB06628 COc1ccccc1NC(=S)N SPB06629 c1ccc2c(c1)[nH]c(n2)C(C(C(C(c3[nH]c4ccccc4n3)O)O)O)O XBX00163 c1cc(ccc1c2cc(c3cc(ccc3n2)Br)C(=O)O)Br XBX00165 c1cc(c(c(c1)Cl)NC(=S)N)Cl SPB06631 Cc1ccccc1NC(=S)N SPB06632 c1cc(c(cc1F)F)NC(=S)N SPB06633 c1ccc(c(c1)NC(=S)N)Br SPB06634 CC(C)C(=O)Nc1ccc(cc1)c2ccccc2 XBX00169 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4ccc(cc4F)F SPB06643 Cc1c(sc(n1)COc2ccccc2Cl)c3ccnc(n3)SCC(=O)c4cccc(c4)[N+](=O)[O-] SPB02705 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)Cn3cc(ccc3=O)C(F)(F)F SPB06531 COC(=O)c1c(ccs1)/N=N/c2c3ccccc3ccc2O SEW05658 CCOC(=O)c1cc(nn1C(C)(C)C)CSc2nnc(n2c3ccccc3)O SPB03941 CC(C)c1ccc(cc1)NC(=O)Cn2c3c(cccn3)oc2=O SPB06592 c1cc(cc(c1)C(F)(F)F)C(=O)NC(=N)c2ccc(cn2)C(F)(F)F SPB06627 c1cc(ccc1C(=O)Oc2ccc(cc2C3SCCS3)Br)Cl SPB00956 c1cc(ccc1C(=O)CSc2[nH]c(nn2)N)Cl SPB01057 c1cc(ccc1c2cnn(c2N)c3cc(cc(c3)Cl)Cl)Cl SPB01061 c1cc(c(cc1Br)C2SCCS2)OC(=O)c3ccc(o3)[N+](=O)[O-] SPB00957 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc(cc2C3SCCS3)Br SPB00960 CC(C)(C)C(=O)O/N=C(/c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)C3SCCS3)\N SPB00979 CC(C)(C)c1[nH]c(nn1)SCc2nc(no2)c3cccc(c3)n4cccc4 SPB01075 CCn1c(cc(n1)C)c2nnc(o2)SCC(=O)c3ccc(cc3)C SPB02758 CCn1c(cc(n1)C)c2nnc(o2)SCC(=O)c3cccc(c3)[N+](=O)[O-] SPB02759 c1ccc(c(c1)OCC(=N)N)Cl.Cl SPB05621 COc1ccc(c(n1)OC)NC(=O)Nc2cccc(c2Cl)Cl SEW05627 CCOC(=O)Cn1cc(ccc1=O)Cl XBX00236 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCCCC2 XBX00243 c1ccc(cc1)NC(=O)c2cccc(c2)Cn3cc(ccc3=O)C(F)(F)F SPB06691 Cc1c(c(nc(n1)c2ccc(cc2)C(F)(F)F)O)Oc3ccc(cc3Cl)Cl SPB04096 CCOC(=O)CC1=CSC2=NCCN12 SPB01009 c1ccc2c(c1)ccc(c2C3SCCS3)OC(=O)c4ccc(o4)[N+](=O)[O-] SPB01018 c1ccc(c(c1)C(F)(F)F)NC(=S)NN SPB07863 C=CCSc1n[nH]c(=O)n1c2ccc(cc2)OCc3ccccc3 SPB07901 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2nc(no2)c3ccc(o3)[N+](=O)[O-])Cl SPB00928 c1cc(c(c(c1)F)C(=O)NNC(=O)c2ccc(nc2)Oc3ccc(cc3)Cl)F SPB03957 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Sc3nnc(n3C)C(F)(F)F SPB03960 Cc1c(c(n(n1)C(=O)c2ccccc2OC)C)Sc3nnc(n3C)C(F)(F)F SPB03962 c1cc(c(c(c1)Cl)CS(=O)c2ccc(cn2)C(F)(F)F)Cl SPB03871 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NNC(=S)NC SPB03920 Cc1ccc(cc1)C(=O)O/N=C(/CSc2c(cccn2)C(F)(F)F)\N SPB03922 c1ccc(cc1)NC(=O)CSc2ccc(cn2)C(F)(F)F SPB02816 c1cc(c(c(c1)Cl)CN2CCC(C(=C2)C(=O)N)C(F)(F)F)Cl SPB06576 Cc1cc(n(c(=O)c1C#N)Cc2ccccc2)C SPB06578 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(n3C)S SPB03926 CCCCCn1c(nnc1SCc2cc(nc(n2)C34CC5CC(C3)CC(C5)C4)O)O SPB03929 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(n3C)SCC=C SPB03931 COc1ccc(c(n1)OC)NC(=O)Nc2cccc(c2)C(F)(F)F SEW05629 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Sc3ccccc3 SPB07768 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Sc3ccc(cc3)Cl SPB07769 Cc1ccc(cc1)Cn2c(cc(n2)C)C(=O)Sc3ccc(cc3)C SPB07770 c1cc(ccc1OCc2nc(cs2)c3ccnc(n3)N)Cl SPB03864 c1cc(ccc1C(=O)Oc2ccc(cc2C3SCCS3)[N+](=O)[O-])Cl SPB01051 CCOC(=O)c1cnc(nc1O)COc2ccccc2Cl SPB05690 CCOC(=O)c1csc(n1)c2csc(n2)C SPB02806 c1coc(c1)/C(=N\O)/C(=N/O)/c2occc2 XBX00255 c1cc(c(cc1)O)/N=C/C=N/c2c(cccc2)O XBX00256 Cc1ccc(cc1)/C(=N/OC(=O)c2cccc(n2)C(F)(F)F)/N SPB06513 c1ccc2c(c1)[nH]c(=O)c(n2)c3cccs3 XBX00041 c1ccc2c(c1)[nH]c(=O)c(n2)c3ccc(s3)Br XBX00043 CCOC(=O)Cc1c(c(sc1C(=O)OCC)N)C#N SEW05594 c1ccc(cc1)S(=O)(=O)c2ccc(c(n2)S(=O)(=O)c3ccccc3)[N+](=O)[O-] SEW05596 Cc1ccc(cc1)c2nnc(o2)CSc3nnc(n3c4ccccc4C(F)(F)F)O SPB02803 Cc1c(sc(n1)c2ccccc2)c3nnc(o3)C4CC4 SPB02808 c1ccc(cc1)NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05664 Cc1ccc(cc1Cl)NC(=S)NNC(=O)c2ccc[nH]2 SEW05668 Cc1nc(cs1)C(=S)N SPB02802 c1cc(ccc1c2nnc(o2)CSc3nnc(n3C4CCCCC4)O)Cl SPB02794 c1ccc(cc1)c2nnc(o2)CSc3nnc(n3C4CCCCC4)O SPB02796 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=N)c3ccccc3 SPB06671 COc1ccc(cc1)Nc2[nH]c(nn2)NC(=O)Nc3ccc(cc3)Cl TG00130 CC(C)NC(=O)Nc1[nH]nc(n1)Nc2ccc(cc2)Cl TG00133 CSc1nnc(n1Cc2ccco2)c3cc(nc(c3)OCC(F)(F)F)OCC(F)(F)F SPB06675 Cc1nc(cs1)/C(=N/OC(=O)Nc2cccc(c2)C(F)(F)F)/N SPB02667 Cc1cc(no1)c2nnc(o2)c3ccc(cc3)Cl SPB02791 Cc1cc(no1)c2nnc(o2)c3ccc(cc3)C(F)(F)F SPB02790 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(n3C)SCC(=O)C(C)(C)C SPB03948 Cc1ccc(cc1)C(=O)NNC(=O)c2c(=O)ccn(n2)c3ccc(cc3)F SPB04041 c1cc(c(cc1Cl)Cl)NC(=S)N SPB06630 c1cc(cc(c1)NC(=O)NC(=O)c2ccc(cc2)OC(F)F)C(F)(F)F SPB05700 Cc1c(c(nc(n1)c2ccc(cn2)C(F)(F)F)N3CCCCC3)Cl SPB05704 Cc1c(c(on1)C)C(=O)NNC(=O)c2ccc[nH]2 SEW05677 c1cc(ccc1C(=S)N)F SEW05679 Cc1c2c(nc(nc2sc1C(=O)NNC(=O)Nc3cccc(c3)C(F)(F)F)c4ccccc4OC)C SPB05579 CC(C)Sc1n[nH]c(=O)n1c2ccc(cc2)OCc3ccccc3 SPB07904 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2[nH]nc(n2)N SPB00887 c1cc(ccc1C2SCCS2)Oc3ccc(cn3)[N+](=O)[O-] SPB00897 c1ccc(cc1)/C=C/2\CCc3ccccc3C2=O TL00083 CN(C)c1ccc(cc1)SC#N TL00118 c1ccc(cc1)C(=N)NC(=O)c2cccc(c2)Cn3cc(ccc3=O)C(F)(F)F SPB06710 c1cc(cc(c1)C(=O)NC(=N)c2ccc(cc2)C(F)(F)F)Cn3cc(ccc3=O)C(F)(F)F SPB06712 Cn1c(cnc1SC)c2ccc(cc2)Cl TG00106 c1ccc(cc1)N/C(=N\C#N)/Oc2ccccc2 TG00119 c1ccc(cc1)O/C(=N/C#N)/Nc2cccc(c2)Cl TG00122 c1ccc(cc1)Nc2nc([nH]n2)N TG00124 c1cc(c(c(c1)Cl)CSc2nnc(o2)c3ccc(nc3)OCC(F)(F)F)Cl SPB06669 c1cc(ccc1C(=O)Sc2c(cc(cn2)C(F)(F)F)Cl)Cl SPB03811 CCOC(=O)/C(=N\Nc1cc(cc(c1)Cl)Cl)/C(=O)CSc2nnc(n2C)C(F)(F)F SPB03966 CCOC(=O)c1cnc(nc1O)c2ccc(cn2)C(F)(F)F SPB05681 Cc1c(c(nc(n1)SCc2ccc(cc2)Cl)O)Oc3ccc(cc3)Cl SPB03977 CC(C)c1ccc(cc1)n2c(nnc2SCC#C)c3ccc(cc3)C(C)(C)C SPB01080 c1cc(ccc1NC(=S)NNS(=O)(=O)c2ccc(cc2)Cl)Cl SPB00994 c1cc(ccc1c2cs/c(=N/NS(=O)(=O)c3ccc(cc3)Cl)/n2c4ccc(cc4)Cl)Cl SPB01002 CC(C)(C)C(=O)OCCN(C)c1nc2cc(ccc2s1)Cl TG00094 CN(CCOC(=O)c1ccc(cc1)Cl)c2nc3cc(ccc3s2)Cl TG00097 Cc1c(c(nn1C)C(=O)Sc2cccc(c2Cl)Cl)[N+](=O)[O-] SPB03817 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccccc3Cl)C SPB00951 c1cc(ccc1NC(=S)NC(=O)c2ccc(o2)[N+](=O)[O-])Cl SPB00989 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2n[nH]c(=O)n2Cc3ccccc3)C#N SPB06554 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3c(cccc3Cl)F)C SPB00952 Cc1ccc(cc1)CSc2c(cc(cn2)C(F)(F)F)Cl SPB03826 c1cc(c(c(c1)Cl)CSc2c(cc(cn2)C(F)(F)F)Cl)Cl SPB03827 c1cc(ccc1CSc2c(cc(cn2)C(F)(F)F)Cl)[N+](=O)[O-] SPB03828 c1cc(sc1)C(=O)Oc2ccc(cc2C3SCCS3)Br SPB00958 c1cc(c(nc1)SCC(=O)Nc2ccc(cc2)Cl)C(F)(F)F SPB03884 CNC(=S)NNC(=O)c1ccc[nH]1 SEW05645 c1cc(ccc1OCC(CO)O)Cl XBX00167 c1ccc(c(c1)C(=O)c2cc(cc(c2)Cl)Cl)C(=O)O XBX00171 CC(C(=O)O)NCc1ccccc1 XBX00173 Cc1cc(n(n1)C(C)(C)C)C(=O)/C(=N/Nc2ccc(cc2)Cl)/C#N SPB03809 Cc1cc2cc(ccc2s1)Cl XBX00175 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SC/C(=N/OC(=O)c3ccc(cc3)Cl)/N SPB00980 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2n[nH]c(=O)n2c3cccc(c3)C(F)(F)F)C#N SPB06555 CSc1nnc(s1)S TL00146 c1ccc(cc1)/C(=C\c2cccc(c2)[N+](=O)[O-])/C(=O)O XBX00106 c1ccc(c(c1)C(C#N)O)[N+](=O)[O-] XBX00108 c1ccc2c(c1)n(c(=O)o2)CCC(=O)O SPB02696 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2csc(n2)COc3ccc(cc3)Cl SPB03774 c1cc([nH]c1)C(=O)N/N=C/c2ccc(cc2)C(F)(F)F SEW05646 Cc1cc(n2c(n1)nc(n2)S)C SPB00852 CC(C)(C)c1ccc(cc1)c2nc(on2)CSc3nc([nH]n3)N SPB00855 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SC/C(=N/O)/N SPB00972 c1cc(c(nc1)N2CCC(CC2)C(F)(F)F)NC(=O)Nc3cc(cc(c3)Cl)Cl SPB06550 CCO.c1cc(c(nc1)N2CCC(CC2)C(F)(F)F)NC(=O)Nc3ccc(cc3)SC(F)(F)F SPB06551 CCOC(=O)c1cc2c(c(sc2nc1C(F)(F)F)C(=O)OCC)N SPB06585 Cc1c(sc2n1nc(n2)C(F)(F)F)/C(=N/OC(=O)c3cc(cc(c3)Cl)Cl)/C SPB05612 Cc1cccc(c1NC(=S)N2CCCC2)Cl SW00015 Cc1cccc(c1)NC(=S)N2CCCCC2 SW00024 c1cc(ccc1C2SCCS2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F SPB00902 CC(C)(C)c1cc(no1)C(=O)/C(=C/Nc2ccccc2)/C#N SPB03782 c1ccc(cc1)CN2CCC(C(=C2)C(=O)N)C(F)(F)F SPB06574 Cc1ccccc1CN2CCC(C(=C2)C(=O)N)C(F)(F)F SPB06575 Cc1c(c(nc(n1)C)O)Oc2cccc(c2)C(F)(F)F SPB04088 Cc1c(c(nc(n1)C)O)Oc2ccc(cc2Cl)Cl SPB04089 c1ccc(c(c1)C(=O)NNC(=O)c2c(=O)ccn(n2)c3ccc(cc3)F)Cl SPB04042 c1ccc(cc1)Cn2c3c(cccn3)oc2=O SPB06588 CCN(c1ccccc1)C(=S)Nc2c(cccc2Cl)C SW00016 Cc1cccc(c1)NC(=S)N2CCCCC2C SW00020 Cc1cccc(c1)NC(=S)N2CCC(CC2)C SW00022 CC(C)(C)C(=O)NNC(=O)c1ccc[nH]1 SEW05678 c1cc2c(cc1n3c(=O)[nH]nc3S)OCCO2 SPB07855 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl SPB07907 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(nc2OC)OC SEW05642 CCCCCCCCCCCCCCCCCC1N=CCN1CCO XBX00259 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Sc3c(cccn3)C(F)(F)F SPB03905 COc1ccc(cc1)CCC(=O)c2ccc(cc2OC)OC XBX00261 CC(C)CN(CC(C)C)CN1C(=O)c2ccccc2C1=O XBX00263 Cc1cc(n(c(=O)c1C#N)CC(=O)Nc2ccc(cc2)C(C)C)C SPB06582 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)NC(=O)NNc4ccccc4 SPB05660 Cc1cccc(c1NC(=S)N2CCOCC2)Cl SW00008 Cc1cccc(c1NC(=S)NCC2CCCO2)Cl SW00011 Cc1cccc(c1NC(=S)NCc2ccncc2)Cl SW00014 CN(C)c1ccc(c(c1)Cl)/C=C\2/c3ccccc3NC2=O SEW05681 CCn1c(c(c(n1)C)Br)C(=O)Sc2ccc(cc2)C(F)(F)F SPB02770 CCn1c(c(c(n1)C)Br)C(=O)Sc2c(cc(cc2Cl)Cl)Cl SPB02771 c1cc(c(c(c1)Cl)COc2ccc(cc2)C3SCCS3)Cl SPB00913 CS(=O)(=O)CS(=O)(=O)NCc1ccc(cc1)Cl SEW05557 CS(=O)(=O)CS(=O)(=O)NNc1c(cc(cn1)C(F)(F)F)Cl SEW05558 Cc1c(c(nn1C)C(=O)Sc2ccc(cc2)Br)[N+](=O)[O-] SPB03814 c1cc(c(nc1)N2CCN(CC2)C(=S)Nc3ccc(cc3)F)C(F)(F)F SEW05665 c1cc(c(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(c(c3)Cl)Cl)C(F)(F)F SEW05667 CCn1c(c(c(n1)C)Br)C(=O)O SPB02757 Cc1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2c(c(oc2N)C)C SEW05669 c1ccc(cc1)C2=N/C(=C/c3cc(cc(c3)Cl)Cl)/C(=O)O2 SEW05673 CCn1c(cc(n1)C)c2nnc(o2)c3ccc(cc3)C(F)(F)F SPB02761 CCn1c(cc(n1)C)c2nnc(o2)c3ccc(cc3)C SPB02763 c1ccc(cc1)C(=O)NC(=N)c2ccc(cn2)C(F)(F)F SPB06625 c1cc(ccc1C(=O)NC(=N)c2ccc(cn2)C(F)(F)F)Cl SPB06626 Cc1ccc(cc1)SC(=O)c2c(c(n(n2)C)C)[N+](=O)[O-] SPB03815 c1ccc2c(c1)c3cc(ccc3cc2Br)[N+](=O)[O-] XBX00122 Cc1cc(cc(c1O)C)C2(CCCCC2)c3cc(c(c(c3)C)O)C XBX00124 CC(C)(C)c1ccc(cc1)OCC(=N)N.Cl SPB05615 Cn1c(nnc1SCc2ccc(cc2)Cl)c3ccc(nc3)OCC(F)(F)F SPB06611 Cc1c(sc(n1)CCn2cccc(c2=O)C(F)(F)F)C(=O)C SPB06614 c1cc(c(cc1NC(=S)N2CCN(CC2)C(=S)Nc3ccc(c(c3)Cl)Cl)Cl)Cl XBX00160 Cc1c(sc(n1)CCn2cccc(c2=O)C(F)(F)F)/C(=N/Nc3c(cccc3Cl)Cl)/C SPB06616 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccccc2NC(=O)c3ccccc3C(F)(F)F)C#N SPB06620 c1ccc(cc1)COc2ccc(cc2)C3SCCS3 SPB00911 Cn1c(nnc1SCc2ccc(cc2)C(F)(F)F)c3ccc(nc3)OCC(F)(F)F SPB06612 c1cc(ccc1CN2CCC(C(=C2)C(=O)N)C(F)(F)F)Cl SPB06573 CC(C)n1c2ccc(cc2nc1SCC(=O)NNC(=O)c3c(cccc3F)F)C(F)(F)F SPB03904 Cc1c(c(no1)c2ccccc2)C(=O)Sc3ccc(cn3)C(F)(F)F SPB03907 Cc1cc(no1)C(=O)NNC(=O)c2c(onc2c3c(cccc3Cl)Cl)C SPB02788 CCOC(=O)N1CCN(CC1)c2ccccc2OC SEW05625 c1ccc(cc1)CN(CCC#N)C(=S)Nc2cccc(c2)C(F)(F)F SW00041 Cc1nc(cs1)c2nnc(o2)c3ccc(cc3)C(F)(F)F SPB02746 CC(C)(C)c1ccc(cc1Cn2nc(nn2)c3cccc(c3)C(F)(F)F)c4ncon4 SPB03943 Cc1nccc(n1)c2c(=O)ccn(n2)c3ccc(cc3)F SPB04025 CNc1c(cc(cn1)C(F)(F)F)[N+](=O)[O-] SPB04036 CN(C)NC(=O)NC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)Cl SPB01159 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)NC(=O)NN3CCOCC3)Cl SPB01160 CCOC(=O)/C(=N\Nc1ccc(cc1)C(F)(F)F)/C(=O)CSc2nnc(n2C)C(F)(F)F SPB03967 CCOC(=O)/C(=N\Nc1ccccc1Cl)/C(=O)CSc2nnc(n2C)C(F)(F)F SPB03968 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)O)Oc3ccc(cc3)Cl SPB03983 c1ccc(cc1)O/C(=N/C#N)/Nc2ccc(cc2)Cl TG00120 COc1ccc(cc1)N/C(=N/C#N)/Oc2ccccc2 TG00123 c1ccc2c(c1)nc3n2c(=O)/c(=C\c4ccc(cc4)[N+](=O)[O-])/s3 TG00076 COc1ccc(c(n1)OC)NS(=O)(=O)c2c(cc(s2)Cl)Br SEW05644 Cc1ccc(cc1)c2nnc(o2)c3csc(n3)C SPB02747 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)C4SCCS4 SPB00915 CC(=NN(C)c1c(cccn1)[N+](=O)[O-])C SEW05560 c1cc(nc(c1[N+](=O)[O-])N2CCOCC2)N3CCOCC3 SEW05561 Cc1c(c(nc(n1)COc2ccccc2)O)Cl SPB05686 c1ccc2c(c1)nc3n2c(=O)/c(=C\c4ccc(cc4)Cl)/s3 TG00080 Cn1c(cnc1SCC=C)c2ccc(cc2)Cl TG00107 CCOC(=O)c1cnc2nc(nn2c1N)SC BTB08391 Cn1c(nnc1Sc2cnc(nc2c3ccc(cc3)Cl)SCC(=O)c4ccc(cc4)Cl)C(F)(F)F SPB04202 Cn1c(nnc1Sc2cnc(nc2c3ccc(cc3)Cl)SCc4ccc(cc4)Cl)C(F)(F)F SPB04203 CCOC(=O)c1c(nc(s1)c2cccc(c2)n3cccc3)C SPB01122 CCOC(=O)Cn1nc(nn1)c2ccc(cc2)C(C)(C)C SPB01123 c1cc(ccc1C(=O)NNC(=O)c2c(=O)ccn(n2)c3ccc(cc3)F)C(F)(F)F SPB04043 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4ccccc4OC SPB06640 c1cc(sc1)c2cc(nc3n2ncn3)C(F)(F)F SPB01147 c1cc(oc1)Cn2c(nnc2S)c3cc(nc(c3)OCC(F)(F)F)OCC(F)(F)F SPB06655 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccccc2NC(=O)Nc3ccc(cc3)Cl)C#N SPB06622 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccccc2NC(=O)Nc3cccc(c3)C(F)(F)F)C#N SPB06623 Cc1ccc(cc1)S(=O)(=O)OCC(C)(C)COS(=O)(=O)c2ccc(cc2)C XBX00225 CSc1cc(nc(c1C#N)O)c2ccco2 SPB01137 CCOC(=O)C1=C(NC(=C(C1C)C(=O)OCC)C)C XBX00199 CCOC(=O)C(=CNc1cccc(n1)C)C(=O)OCC XBX00202 CCOC(=O)c1c(sc(n1)c2ccccc2)C(=O)OCC XBX00205 Cc1ccc(cc1[N+](=O)[O-])I SEW05708 c1ccc2c(c1)ccc(c2C3SCCS3)OC(=O)c4cccs4 SPB01017 c1c(oc(c(c1=O)O)CO)CO XBX00210 Cc1ccc(cc1)C(=O)CSc2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)F SPB02830 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SC/C(=N/OC(=O)c3cccs3)/N SPB00982 CC(C)c1ccc(cc1)n2c(nnc2S)c3ccc(cc3)C(C)(C)C SPB01078 CC(C)c1ccc(cc1)n2c(nnc2SCC=C)c3ccc(cc3)C(C)(C)C SPB01079 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccc3ccccc3c2C4SCCS4 SPB01015 c1ccc2c(c1)ccc(c2C3SCCS3)OC(=O)c4ccc(cc4Cl)Cl SPB01016 COC(c1cc(nc(n1)SCC(=O)Nc2ccc(cc2)C(F)(F)F)O)OC SPB05730 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2ccc(cn2)C(F)(F)F SPB02846 c1cc(c(c(c1)Cl)Cl)/C=N/O SPB01023 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2ccc(cn2)C(F)(F)F SPB02853 c1cc(ccc1C(=O)Sc2ccc(cn2)C(F)(F)F)C(F)(F)F SPB02838 Cc1cc(no1)NC(=O)c2ccc(cc2)CSCc3c(cccc3Cl)Cl SPB01029 Cc1ccc(cc1)C(=O)Sc2ccc(cn2)C(F)(F)F SPB02839 c1cc(ccc1CSc2ccc(cn2)C(F)(F)F)Cl SPB02840 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)N)Cl SPB01153 Cc1c(c(n(n1)CC(=O)Nc2cccc(c2)SC)C)Oc3ccccc3 SPB06604 Cc1cc(no1)NC(=O)c2ccc(cc2)CSCc3ccc(cc3)Cl SPB01028 CCCCCc1ccc(cc1)c2[nH]c(nn2)SCC(=O)C SPB01044 CCCCCc1ccc(cc1)c2[nH]c(nn2)SCC(=O)c3ccc(cc3)Cl SPB01046 CCCCCc1ccc(cc1)c2[nH]c(nn2)SCC(=O)c3ccc(cc3)[N+](=O)[O-] SPB01047 c1ccc2c(c1)n(c(=O)o2)CCC(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB02847 c1cc(cc(c1)Cl)NC(=O)O/N=C(/CSc2c(cccn2)C(F)(F)F)\N SPB03918 c1cc(cc(c1)NC(=O)O/N=C(/CSc2c(cccn2)C(F)(F)F)\N)C(F)(F)F SPB03919 c1ccc2c(c1)n(c(=O)o2)CCC(=O)NNC(=O)c3ccc(cc3)Cl SPB02850 c1cc(c(cc1C#N)[N+](=O)[O-])Oc2ccc(cc2F)F SPB01152 c1cc(c(nc1)SC/C(=N/OC(=O)c2ccc(cc2)Cl)/N)C(F)(F)F SPB03921 c1cc(c(nc1)SC/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/N)C(F)(F)F SPB03923 Cc1cc(no1)C(=O)O/N=C(/CSc2c(cccn2)C(F)(F)F)\N SPB03924 Cn1ccnc1Sc2cnc(nc2c3ccccc3)SCc4ccc(cc4)Cl SPB04199 CN(C)/C=C/C(=O)c1c(=O)ccn(n1)c2ccc(cc2)Cl SPB04002 CCOC(=O)c1c(=O)c(cn(n1)c2ccccc2Cl)Sc3nnc(n3C)C(F)(F)F SPB04011 c1ccc(c(c1)C(F)(F)F)n2c(nnc2SCc3cc(nc(n3)C45CC6CC(C4)CC(C6)C5)O)O SPB03927 Cc1cc(n(c(=O)c1C#N)CC(=O)Nc2ccccc2)C SPB06581 Cc1cc(n(c(=O)c1C#N)CC(=O)Nc2cccc(c2)Cl)C SPB06584 c1cc2c(nc1)n(c(=O)o2)Cc3ccc(cc3)Cl SPB06587 C=CCn1c(nnc1SCc2cc(nc(n2)C34CC5CC(C3)CC(C5)C4)O)O SPB03933 COC(=O)c1ccc(nc1)Oc2cccc(c2)C(F)(F)F SPB03938 Cc1ccccc1NC(=O)c2cccc(c2)Cn3cc(ccc3=O)C(F)(F)F SPB06693 Cc1ccc(cc1)SCC(=O)c2ccc(cc2)Cl SPB04106 Cc1c(c(nc(n1)c2ccc(cc2)C(F)(F)F)OC(=O)N(C)C)Oc3ccc(cc3Cl)Cl SPB04102 Cc1c(c(nc(n1)C)Sc2cccc(c2)C(F)(F)F)Oc3ccc(cc3Cl)Cl SPB04104 c1cc(c(cc1C(F)(F)F)NC(=S)N)Cl SPB06701 CCOc1ccc(cc1)CCC(=O)O XBX00229 COC(c1cc(nc(n1)SC)O)OC SPB05719 c1ccc(cc1)/C=C/C=C/C=C/c2ccccc2 XBX00233 COC(c1cc(nc(n1)SCc2ccc(cc2)Cl)O)OC SPB05722 CCOC(=O)Cn1nc(nn1)c2ccc(cn2)C(F)(F)F SPB05723 c1ccc(cc1)C(=O)CSc2[nH]c(nn2)N SPB01056 Cc1c(c(nc(n1)c2ccc(cn2)C(F)(F)F)N3CCOCC3)Cl SPB05705 Cc1c(oc(c1S(=O)(=O)/C(=C/c2cc(cc(c2)Cl)Cl)/C#N)N)C SEW05685 CC(C)(C)c1cc(n(n1)C)C(=O)N2CCC(CC2)C(F)(F)F SPB06646 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCOc3ccccc3 SPB06650 c1ccc(cc1)SC(=O)c2cccc(c2)Cn3cc(ccc3=O)C(F)(F)F SPB06695 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCOc3ccccc3 SPB06651 Cc1c(c(no1)c2ccccc2)C(=O)NCCOc3ccccc3 SPB06652 Cc1ccc(cc1)/C(=N/OC(=O)c2cccc(c2)Cn3cc(ccc3=O)C(F)(F)F)/N SPB06704 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)Nc3cccnc3 SPB03953 c1ccc(cc1)c2cc(=O)[nH]c3c2cccc3 XBX00298 CCOC(=O)CC(=O)CSc1nnc(n1C)C(F)(F)F SPB03954 c1cc(ccc1C(=O)NNC(=O)c2ccc(nc2)Oc3ccc(cc3)Cl)Cl SPB03956 Cc1ccc(cc1)C(=O)CCC(=O)O TL00153 Cc1ccc(cc1)Sc2c(c(nc(n2)C)C)Oc3ccc(cc3Cl)Cl SPB04067 c1(nc(=S)ss1)N TL00112 COC(c1c(cnc(n1)SCC(=O)Nc2cccc(c2)Cl)C(=O)O)OC SPB05737 c1ccc(cc1)CNC(=S)Nc2ccc(c(c2)Cl)Cl XBX00245 c1ccc(cc1)CNC(=S)Nc2ccc(cc2)Br XBX00246 COC(c1c(cnc(n1)SCC(=O)Nc2ccc(cc2)C(F)(F)F)C(=O)O)OC SPB05738 c1cc(ccc1NC(=O)CSc2ccc(cn2)C(F)(F)F)Cl SPB02818 CC(C)c1ccc(cc1)n2c(nnc2SCc3ccccc3Cl)c4ccc(cc4)C(C)(C)C SPB01082 COc1ccc(cc1)C(=O)c2ccc(cc2)F XBX00254 c1cc(ccc1C(=O)CCC(=O)O)F TL00155 C1CC1CSc2nnc(s2)S TL00159 c1ccn(c1)c2cccc(c2)c3nc(cs3)c4ccc(cc4)Cl SPB01088 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)NC(=O)N3CCCC3)Cl SPB01163 Cc1c(c(nc(n1)N)O)Oc2ccc(cc2)Cl SPB03993 c1cc(ncc1C(F)(F)F)Sc2ncc(s2)[N+](=O)[O-] SPB02854 Cc1c(c(nc(n1)c2cc(cc(c2)Cl)Cl)O)Oc3ccc(cc3)Cl SPB03989 Cc1c(c(nc(n1)COc2ccc(cc2)C(C)(C)C)O)Cl SPB05687 Cc1c(c(nc(n1)COc2ccccc2Cl)O)Cl SPB05688 CC(C)c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Cl)c4ccc(cc4)C(C)(C)C SPB01083 CC(C)c1ccc(cc1)n2c(nnc2Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F)c4ccc(cc4)C(C)(C)C SPB01087 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4ccccc4Br SPB06707 c1ccc(cc1)NC2CC(=O)C(=C2)Nc3ccccc3 XBX00322 c1cc(c(cc1C#N)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl SPB01097 c1cc(ccc1c2nnn(n2)CC(=O)Sc3ccc(cc3F)F)C(F)(F)F SPB03949 COC(=O)c1c(ccs1)NC(=O)Cn2nc(nn2)c3cccc(c3)C(F)(F)F SPB03952 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4ccccc4F SPB06708 c1cc(ncc1C#N)OCC(F)(F)F SPB05790 c1ccc(cc1)n2c(c(cn2)c3ccc(cc3)Cl)N SPB01060 C#CCSc1nnc(s1)S TL00164 c1cc(ccc1c2cnn(c2N)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl SPB01062 CN(C)c1nc(=S)ss1 TL00165 CCCC(CC(=O)O)(c1ccccc1)C(=O)O XBX00296 c1cc(oc1)Cn2c(nnc2SCc3ccc(cc3)Cl)c4cc(nc(c4)OCC(F)(F)F)OCC(F)(F)F SPB06678 c1cc(ccc1c2nnc(o2)CSc3nnc(n3C4CCCCC4)O)[N+](=O)[O-] SPB02797 c1ccc2c(c1)nc(s2)NC=C(C#N)C#N BTB08385 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)Nc3ccc(cc3)SC(F)(F)F)C(F)(F)F BTB08363 Cn1ccnc1Sc2cnc(nc2c3ccc(cc3)Cl)SCC(=O)c4ccc(cc4)Cl SPB04197 c1c(cc(c(c1Br)O)Br)C2SCCS2 SPB01187 c1cc(c(cc1C(=O)N)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl SPB01189 c1cc(ccc1Oc2ccc(cn2)C(=O)N)Cl SPB05792 c1cnc(nc1)NC=C(C#N)C#N BTB08387 c1ccc2c(c1)C(=O)N(C2=O)Oc3ccc(c(c3)[N+](=O)[O-])[N+](=O)[O-] XBX00332 c1ccc(cc1)CSc2nnc(o2)c3ccc(nc3)OCC(F)(F)F SPB06667 CCOC(=O)CS/C(=C(/C#N)\C(=O)OCC)/Nc1ccccc1C(F)(F)F SEW05688 Cc1c(c(nc(c1/N=N/c2cc(cc(c2)Cl)Cl)C)SCc3ccccc3)C#N SPB06730 Cc1c(c(nc(c1/N=N/c2cc(cc(c2)Cl)Cl)C)SC)C#N SPB06731 Cc1c(c(nc(c1/N=N/c2ccccc2)C)SCc3ccccc3Cl)C#N SPB06733 CCN(CC)c1cc(cc(c1)Cl)Cl SEW05690 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC#N SPB00967 c1cc(ccc1NC(=O)CSc2c(cc(cn2)C(F)(F)F)Cl)Cl SPB03832 CC(C)(C)c1cc(no1)C(=O)/C=c\2/[nH]c(=O)/c(=C/c3ccc(cc3)Cl)/s2 SPB03836 c1cc(ccc1C2SCCS2)Oc3ccc(cc3[N+](=O)[O-])C#N SPB00968 c1cc(ccc1C2SCCS2)Oc3ccc(cc3[N+](=O)[O-])/C(=N/O)/N SPB00970 CCCCCCCCCCCc1nnc(n1C)SC(=O)N(C)C SPB01444 CC(C)(C)C(=O)OCc1nc(cs1)c2cc(no2)c3ccc(c(c3)Cl)Cl SPB06659 c1cc(ccc1c2nc(no2)c3c(cn[nH]3)Br)Cl SPB02864 Cc1c(c(nc(n1)COc2ccc(cc2)OC)O)Cl SPB05689 c1cc(ccc1C(=O)NC(=O)Nc2ccc(cc2)F)C(F)(F)F SPB01454 CS/C(=N\C#N)/N1CCC(CC1)C(=O)c2ccccc2 SEW05724 Cc1c(c(no1)c2ccccc2)C(=O)NC(=N)c3ccc(cc3)Cl SPB06673 Cc1nc(cs1)C(=O)N/N=C/c2c(c[nH]n2)Cl SPB02868 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2csc(n2)CSc3nnc(s3)SCC4CC4 SPB02867 c1cc(cc(c1)NC(=S)Nc2cccnc2N3CCC(CC3)C(F)(F)F)C(F)(F)F SPB06558 CC(C)c1ccc(cc1)NC(=O)CSc2c(cccn2)C(F)(F)F SPB03885 CCOC(=O)c1nc(no1)c2ccc(o2)[N+](=O)[O-] SPB00925 c1ccc(cc1)C(=O)c2c(=O)ccn(n2)c3ccc(cc3)Cl SPB04029 c1cc(ccc1C(=O)NNC(=O)c2c(=O)ccn(n2)c3ccc(cc3)F)Cl SPB04040 c1ccc2c(c1)nc3n2c(=O)/c(=C\c4cccc(c4Cl)Cl)/s3 TG00083 CSc1nnc(s1)SCc2nc(cs2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB02866 CN(C)/C=C/C(=O)c1c(=O)ccn(n1)c2ccc(cc2)F SPB02819 CCCCNC(=O)n1ccc(n1)c2c(=O)ccn(n2)c3ccc(cc3)F SPB02821 C#CCN1C(=O)c2ccccc2C1=O XBX00270 CSc1nnc(s1)SCc2csc(n2)c3ccc(cc3)C(F)(F)F SPB02870 c1cc(ccc1/C(=N\OC(=O)c2ccno2)/N)C(F)(F)F SPB02874 CCOC(=O)c1cc(on1)C(=O)CSc2ccc(cn2)C(F)(F)F SPB05696 c1ccc2c(c1)c(c[nH]2)/C=N\O XBX00284 c1cc(ccc1CS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl SPB03860 c1cc(ccc1CS(=O)(=O)c2ccc(cn2)C(F)(F)F)[N+](=O)[O-] SPB03861 Cc1c(snn1)c2nc(cs2)/C(=N/Nc3ccccc3C(F)(F)F)/C SPB03867 Cc1cc(n(c(=O)c1C#N)Cc2ccc(cc2)Cl)C SPB06579 c1cc(ncc1C(F)(F)F)C(=N)N.Cl SPB05657 Cc1c(sc2n1nc(n2)C(F)(F)F)c3ccnc(n3)c4ccccc4 SPB05658 c1cc(ccc1n2c(nnc2S)c3ccc(nc3)OCC(F)(F)F)Cl SPB06599 c1ccc(c(c1)S(=O)(=O)NNC(=O)c2c(=O)ccn(n2)c3ccc(cc3)F)Cl SPB04048 Cc1c(c(nc(n1)c2ccc(cn2)C(F)(F)F)Sc3ccc(cc3)Cl)Cl SPB05707 Cn1c(nnc1S/C(=C/N(C)C)/C(=O)c2ccc(cc2)Cl)C(F)(F)F SPB04116 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=S)Nc3ccc(cc3C)Br SEW05716 Cc1c(c(n(n1)C)C(=O)Sc2ccc(cn2)C(F)(F)F)[N+](=O)[O-] SPB04053 CN(C)/C=N/NC(=O)c1c(=O)c(cn(n1)c2cccc(c2)Cl)Sc3ccc(cc3)Cl SPB04054 CN(C)Cc1coc2ccccc2c1=O.Cl SPB05713 CN(C)/C=C(/C(=O)c1ccc(cc1)Cl)\Sc2ccc(cc2)Cl SPB04113 Cc1ccc(cc1)S/C(=C\N(C)C)/C(=O)c2ccc(cc2)Cl SPB04114 c1ccc(cc1)NC(=O)Cn2c3c(cccn3)oc2=O SPB06591 c1cc(c(nc1)Sc2[nH]c(nn2)N)[N+](=O)[O-] SPB00886 Cc1cc(n2c(n1)nc(n2)SCc3ccc(cc3)Cl)O SPB00882 C/C(=C(\C(=O)c1ccc(cc1)Cl)/C(=O)OC)/NC SPB00904 Cn1c(nnc1S)c2ccc(nc2)OCC(F)(F)F SPB06600 c1cc(c(nc1)Oc2ccc(cc2)C3SCCS3)[N+](=O)[O-] SPB00898 c1cc(ccc1C2SCCS2)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] SPB00900 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05717 c1c(cc(c(c1Cl)S(=O)(=O)NC(=N)N)Cl)C(F)(F)F SEW05694 COC(=O)c1cccn1S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW05696 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=S)Nc3cccc(c3)Cl SEW05718 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=S)Nc3ccc(cc3Cl)Cl SEW05719 Cc1c(c(=O)n2c(csc2n1)c3ccc(cc3)Cl)Oc4ccc(cc4)Cl SPB04119 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccccc2N)C#N SPB06605 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3ccc(nc3)OCC(F)(F)F SPB06608 CCn1c(c(c(n1)C)Br)C(=O)Oc2ccc(cc2)C SPB02775 CCn1c(cc(n1)C)c2nnc(o2)SCC(=O)Nc3ccc(cc3)C(C)C SPB02776 c1ccc(c(c1)C=Nc2ccc(c(c2)Cl)Cl)O XBX00198 c1cc(ccc1c2csc(n2)c3cnccc3C(F)(F)F)Cl SPB05768 c1cc(ccc1C#N)c2csc(n2)c3cnccc3C(F)(F)F SPB05769 CN(C)c1ccc(c(c1)Cl)/C=N/Nc2cc(ccc2Cl)Cl SEW05701 c1cc(c(c(c1)Cl)Cl)/C(=N/OC(=O)C(Cl)Cl)/N SPB01113 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=S)NCC2CCCO2 SEW05699 Cc1c(c(nc(c1/N=N/c2cc(cc(c2)Cl)Cl)C)SCC(=O)c3cccc(c3)F)C#N SPB06743 Cc1ccc(c(c1)C)NCN2C(=O)c3ccccc3C2=O XBX00271 c1ccc(cc1)N(CCO)CCO XBX00274 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)O XBX00275 CN(C)c1ccc(c(c1)Cl)/C=N/Nc2cnc3ccccc3n2 SEW05700 c1ccc(cc1)c2nc(c(o2)N)C#N SEW05707 CCOC(=O)C(Cc1ccccn1)(c2ccccc2)C(=O)OCC.Cl XBX00204 c1cc(sc1/C=N/NC(=O)c2nc(no2)c3ccc(o3)[N+](=O)[O-])[N+](=O)[O-] SPB00929 c1cc(c(c(c1)Cl)COc2ccc(cc2)[N+](=O)[O-])Cl SPB00933 Cc1ccc(cc1)CS(=O)(=O)c2ccc(cn2)C(F)(F)F SPB03862 c1ccc2c(c1)CCN2c3ccc(cc3)[N+](=O)[O-] XBX00320 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CN2C(=O)c3ccccc3C2=O XBX00326 C=CC(=O)NC(C(NC(=O)C=C)O)O XBX00280 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)OC SEW05705 c1cc(oc1CSC(=N)N)[N+](=O)[O-].Br XBX00327 CCO/C(=N/Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/C XBX00331 Cn1cncc1CC2COC(=O)C2C(c3ccccc3)O XBX00287 c1cc(c(cc1/C(=N/O)/N)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl SPB01099 c1ccnc(c1)OCCOc2ccccn2 XBX00134 CC(C)(C)c1ccc(cc1)C(=O)C2CC2 XBX00136 c1ccc2c(c1)[nH]c(n2)/C(=C/Nc3cccc(c3)C(F)(F)F)/C#N BTB08364 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=S)Nc3ccc(cc3)F SEW05715 CSc1cc(nc(c1C#N)O)c2ccc(cc2)Cl SPB01136 c1ccc(cc1)c2c(nc3cc(ccc3n2)[N+](=O)[O-])c4ccccc4 XBX00337 CN(C)/C=C/C(=O)c1c(=O)ccn(n1)c2ccc(cc2)C(F)(F)F SPB04003 CC(C)(C)C\1=NN(C(=O)/C1=C/N(C)C)c2ccccc2 BTB07065 CCOC(=O)c1c(=O)c(cn(n1)c2ccccc2Cl)Sc3ccc(cc3)Cl SPB04013 c1cc2c(nc1)n(c(=O)o2)CC(=O)c3ccc(cc3)Cl SPB06636 c1ccc(cc1)S(=O)(=O)/C(=C/c2cccn2c3ccc(cc3)Cl)/C#N SEW05651 COC(=O)CSc1ccc(c(n1)SCC(=O)OC)[N+](=O)[O-] SEW05657 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06817 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2ccc(cc2C3CCCCC3)Cl BTB07144 c1cc(ccc1Cn2ccnc2c3ccc(cc3)C(F)(F)F)[N+](=O)[O-] SPB01487 c1cc(ccc1NC(=O)Nc2ccc(nc2)Sc3ccc(cc3)Cl)SC(F)(F)F BTB08355 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)O)C(F)(F)F BTB07082 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)O)Cl BTB07083 Cc1cccc(c1C(=O)O)NC(=O)C(F)(F)F BTB07153 COc1ccc(cc1OC)/C=C(\C#N)/c2ccc(cc2)O BTB07084 Cc1ccc(cc1)Sc2ccc(cn2)NC(=O)Nc3ccc(cc3)SC(F)(F)F BTB08356 Cc1ccccc1Nc2nc(cs2)c3c(onc3c4ccc(cc4Cl)Cl)C SPB06644 c1cc(cc(c1)C(=O)Nc2ccc(cc2)Cl)Cn3cc(ccc3=O)C(F)(F)F SPB06692 c1ccc(c(c1)N)Sc2c(cc(c(n2)Sc3ccccc3N)C(F)(F)F)C(F)(F)F SEW05687 c1c(cc(cc1Cl)Cl)/C=N/O SEW05689 CN(C)c1ccc(cc1)/C=C/c2ccccc2 XBX00220 c1ccc2c(c1)n(c(=O)o2)CCC(=O)NC(=N)c3ccc(cc3)Cl SPB06758 c1cc(ccc1NC(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl)Cl SPB06812 CC(C)(C)NC(=O)NNC(=O)c1c(ccs1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB06814 Cc1ccc(cc1)Cn2nc(nn2)c3cc(c(c(c3)Br)OC)Br SPB01481 Cc1cccc(c1C)Oc2ccc(cn2)[N+](=O)[O-] BTB07175 Cc1cccc(c1)C(=O)Nc2ccnc3n2nc(n3)SC BTB08419 CN(C)/C=N/NC(=O)COc1ccc(cc1)SC(F)(F)F BTB08357 Cc1ccc(cc1)S(=O)(=O)NNC(=O)COc2ccc(cc2)SC(F)(F)F BTB08358 c1cc(ccc1OCC(=O)NNS(=O)(=O)c2cc(ccc2Cl)Cl)SC(F)(F)F BTB08359 c1cc(ccc1C(=O)O/N=C(/c2ccc(nc2)OCC(F)(F)F)\N)Cl SPB05796 CN(C)c1ccc(c(c1)O)/C=N/NC(=S)N XBX00222 Cc1c(c(on1)C)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW05691 Cc1ccc(cc1)CSc2ccc(cn2)C(F)(F)F SPB02842 CCCCCc1ccc(cc1)c2[nH]c(nn2)S SPB01039 CCCCCc1ccc(cc1)c2[nH]c(nn2)SCC#C SPB01040 Cc1cc(ccc1Oc2ccc(cn2)[N+](=O)[O-])Cl BTB07177 CCCCN1C(C(=O)N(C1=O)c2nnc(s2)C(C)(C)C)c3ccc(c(c3)Cl)Cl BTB08403 Cc1ccc(cc1)CSc2cc3c(cc2[N+](=O)[O-])C(=O)NC3=O BTB08408 CCCCn1c(cn(c1=O)c2nnc(s2)C(C)(C)C)CSCc3ccc(cc3)Cl BTB08405 COc1cccc(c1C(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl)OC BTB07244 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2ccc(nc2)Oc3cccnc3)Cl BTB07230 Cc1c(c(nc(n1)C)OC)Oc2ccc(cc2Cl)Cl SPB04069 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(/c2ccc(nc2)OCC(F)(F)F)\N SPB05798 CSc1nc2nccc(n2n1)N BTB08400 CCOC(=O)C1=C(NC(=C(C1/C=C/c2ccccc2)C(=O)OCC)C)C XBX00342 CCOC(=O)C1=C(NC(=C(C1c2cccc(c2)[N+](=O)[O-])C(=O)OCC)C)C XBX00343 CCCCCc1ccc(cc1)c2[nH]c(nn2)SCc3ccccc3Cl SPB01043 CCCCCc1ccc(cc1)c2[nH]c(nn2)SCC(=O)c3ccccc3 SPB01045 Cc1ccc(cc1)C(=O)CSc2ccc(cn2)C(F)(F)F SPB02844 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(n3C)SCc4ccccc4 SPB03932 COC(=O)c1ccc(nc1)Oc2ccc(cc2)Cl SPB03936 CCOC(=O)c1c(=O)c(cn(n1)c2cccc(c2)Cl)Sc3ccc(cc3)Cl SPB04014 c1cc(ccc1S(=O)(=O)n2ccc(c2)c3cnc4cc(c(cc4n3)Cl)Cl)Cl BTB07251 c1ccc2c(c1)ncc(n2)c3ccn(c3)S(=O)(=O)c4ccc(cc4)Cl BTB07253 c1(nc(nc(n1)S)S)N TL00238 Cc1c(c(nc(n1)S)O)Oc2ccc(cc2)F SPB04175 Cc1ccc(cc1)S(=O)(=O)n2c(c(cn2)Sc3ccc(cc3)Cl)c4ccc(cc4)Cl SPB04186 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl)C#N SPB06802 Cc1c(sc2n1nc(n2)C(F)(F)F)c3csc(n3)c4ccc(cc4)Cl SPB05725 Cc1ccc(cc1)C(=O)/C(=C/N(C)C)/Sc2ccc(cn2)C(F)(F)F SPB04019 Cc1ccc(cc1)c2c(c[nH]n2)Sc3ccc(cn3)C(F)(F)F SPB04020 C/C(=C(\C(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C(=O)OC)/NC SPB01171 c1cc(ccc1C#N)Oc2nc3cc(ccc3s2)Cl SPB01177 CCN(CC)C(=O)Oc1nnc(n1c2ccc(cc2)Cl)SC(C)C SPB01185 Cc1cc(no1)C(=O)N SPB04068 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CC4(CC3CC(C4)(C)C)C SPB04174 c1cc(ccc1C(=O)CSc2ccc(cn2)C(F)(F)F)Cl SPB02845 c1ccc2c(c1)n(c(=O)o2)CCC(=O)NNC(=O)c3cccc(c3)Cl SPB02849 COC(c1cc(nc(n1)SCC#C)O)OC SPB05720 c1cc2c(cc1[N+](=O)[O-])cc(c(=O)o2)C(=O)O BTB07074 c1cc(ccc1CC#N)OS(=O)(=O)c2cc(cc(c2)Cl)Cl BTB07097 COc1c(cc(cc1Br)c2nnn(n2)Cc3ccc(cc3)[N+](=O)[O-])Br SPB01482 CCOC(=O)/C(=C\Nc1ccc(cc1)F)/[N+](=O)[O-] SPB01494 c1cc(ccc1NC(=O)Nc2ccc(nc2)Sc3ccc(cc3)Cl)OC(F)(F)F BTB08353 c1cc(ncc1c2nnc(o2)S)OCC(F)(F)F SPB06656 CC(C)(C)C(=O)OCc1nc(cs1)c2cc(no2)c3ccccc3 SPB06657 Cc1ccc(cc1C)c2cc(on2)c3csc(n3)COC(=O)C(C)(C)C SPB06658 Cc1cc(no1)c2nnc(o2)c3ccc(cn3)C(F)(F)F SPB05742 c1cc(c(c(c1)I)C(=O)O)F TL00162 c1cc(c(c(c1)Cl)COc2ccc(cc2)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N)F BTB07094 c1cc(cnc1)Oc2ccc(cn2)NC(=O)c3ccc(cc3)C(F)(F)F BTB07224 c1cc(c(c(c1)Cl)CSc2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)F)Cl SPB02825 Cc1ccc(cc1)CSc2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)F SPB02826 c1cc(ccc1CSc2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)F)C(F)(F)F SPB02827 Cc1ccc(cc1)C(=O)CSc2nc(cc(n2)O)C(OC)OC SPB05729 c1ccn(c1)c2cccc(c2)/C(=N/OC(=O)C(Cl)Cl)/N SPB01069 c1ccn(c1)c2cccc(c2)C(=S)N SPB01074 c1cc(ccc1CC#N)OS(=O)(=O)c2ccc(cc2)Cl BTB07095 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)CC#N BTB07096 Cc1ccc(cc1)SCC(=O)Nc2ccc(c(c2F)F)F BTB08439 c1ccc(cc1)c2c(=S)ssc2SCC(=O)Nc3ccc(c(c3F)F)F BTB08441 c1cc(cnc1)Oc2ccc(cn2)NC(=O)c3ccc(cc3)Cl BTB07225 c1cc(c(c(c1)Cl)Sc2cc3c(cc2[N+](=O)[O-])C(=O)NC3=O)Cl BTB08406 c1cc(ccc1CSc2cc3c(cc2[N+](=O)[O-])C(=O)NC3=O)Cl BTB08407 CN(C)c1cc(cc(c1)Cl)Cl SEW05711 c1ccc(cc1)NC(=O)Oc2ccc(cc2)CC#N BTB07087 c1cc(ccc1/C(=C/c2ccc(cc2Cl)Cl)/C#N)O BTB07090 CCO/C=N/c1c(nc(o1)c2ccccc2)C#N SEW05731 C/C(=N\O)/c1ccn(c1)S(=O)(=O)c2ccc(cc2)Cl BTB07130 COc1cccc(c1C(=O)NC(=O)Oc2c(cccc2F)F)OC BTB07135 Cc1ccc(cc1)Sc2nc(ns2)c3cccs3 SPB06936 Cc1ccc(cc1)Oc2c(nc(nc2O)C)C SPB04087 Cc1ccc(cc1)Oc2c(nc(nc2OC(=O)N(C)C)C)C SPB04090 c1cc(ccc1n2ccc(=O)c(n2)c3ccnc(n3)S)F SPB02824 CS(=O)(=O)Nc1ccc(cc1)/C(=N/O)/N SPB06756 c1cc(ccc1C(=O)Sc2ccc(cn2)C(F)(F)F)Cl SPB02832 Cc1ccc(cc1)C(=O)C2CCN(CC2)C(=S)NCC=C SEW05725 COc1ccc(cc1)Oc2ccc(cc2)[N+](=O)[O-] SEW05726 CN(C)/C=C(\C#N)/c1ccc(cc1)OCc2ccc(c(c2)Cl)Cl BTB07066 Cc1cc(no1)/C(=N/OC(=O)c2cccc(c2)Cl)/N SPB04135 c1cc(ccc1c2c(c[nH]n2)Sc3ccc(cc3)Cl)Cl SPB04137 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C)Cn3cc(ccc3=O)C(F)(F)F SPB06687 c1ccc(c(c1)NC(=S)N)F SPB06700 Cc1ccn2c(c1)ncc2[N+](=O)[O-] XBX00318 CCOC(=O)c1cc(ccc1Oc2ccc(cc2)SC(F)(F)F)[N+](=O)[O-] BTB08366 CN(C)c1ccc(c(c1)Cl)/C=N/Nc2c(cc(cc2Cl)C(F)(F)F)Cl SEW05692 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=S)N SEW05693 c1ccc(cc1)CSc2nnc(o2)c3cccc(n3)C(F)(F)F SPB06737 c1cc(cc(c1)C(=O)O/N=C(/c2ccc(cc2)Cl)\N)Cn3cc(ccc3=O)C(F)(F)F SPB06705 COCCCn1c(nnc1SCC#C)c2ccc(cc2)C(F)(F)F SPB01438 COc1cc(ccc1Oc2ccc(cn2)[N+](=O)[O-])CC=C BTB07119 CC(C)Oc1ccccc1Oc2ccc(cn2)[N+](=O)[O-] BTB07120 Cc1cc(c([nH]1)C)C(=O)OC SP00004 CCOC(=O)c1ccc(cc1)n2cccc2 SEW05729 c1ccc2c(c1)ncc(n2)n3c(=O)c(c(cn3)N4CCOCC4)Cl SEW05730 c1cc(ccc1c2csc(n2)CSc3nnc(s3)SCC4CC4)[N+](=O)[O-] SPB02865 Cc1nc(cs1)C(=O)N/N=C/c2c(c[nH]n2)Br SPB02869 c1ccc(cc1)C(C(=O)O)n2cccc2 SEW05732 Cc1c(c(c([nH]1)C)C(=O)OC)C(=O)C SP00007 Cc1c(c(c([nH]1)C)C(=O)OC)/C=N/O SP00009 c1ccc(cc1)C(=O)C2CCN(CC2)C=C(C#N)C#N SEW05736 c1cc(nc(c1)C(F)(F)F)c2nnc(o2)SCc3ccc(cc3)Cl SPB06738 Cc1c(c(nc(c1/N=N/c2ccccc2)C)SCC(=O)Nc3cccc(c3)SC)C#N SPB06740 c1ccc2c(c1)n(c(=O)o2)CCc3nnc(o3)c4cccc(c4)Cl SPB02858 c1c(cc(cc1Br)Br)C(=S)N SEW05752 C#CCOC(=O)NC(=O)c1ccc(cc1)C(F)(F)F SPB01455 c1ccc2c(c1)n(c(=O)o2)CCc3nnc(o3)c4ccc(cc4)Cl SPB02859 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)Sc2ccc(cn2)C(F)(F)F SPB02860 CSc1nnc(s1)SCc2nc(cs2)c3ccc(c(c3)Cl)Cl SPB02871 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)Nc2ccc(cc2)C(F)(F)F SPB02909 c1cc(sc1)C(=O)N2CCC(CC2)C(=O)c3ccc(cc3F)F SEW05737 c1cc(ccc1c2nc(cs2)C(=O)NN)C3SCCS3 SPB02810 c1cc(ncc1C(F)(F)F)/C(=N/OC(=O)c2c(cc(cn2)C(F)(F)F)Cl)/N SPB05697 Cc1nc(cs1)c2nc(cs2)C(=O)NNS(=O)(=O)C SPB02814 c1cc(ncc1C(F)(F)F)SCC(=O)Nc2cc(cc(c2)Cl)Cl SPB02817 c1cncc(c1C(F)(F)F)C(=S)N SPB05766 c1cc(ccc1/C(=N/O)/N)OC(F)(F)F SPB02881 CC(C)c1ccc(cc1)NC(=O)CSc2ncc(c(n2)C(OC)OC)C(=O)O SPB05743 c1ccc(cc1)NC(=O)NC(=O)c2ccc(cc2)OC(F)F SPB05699 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)NCC(=O)c2ccc(cc2)Cl SPB02900 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)Nc2cc(cc(c2)Cl)Cl SPB02903 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NS(=O)(=O)c3ccc(cc3)C)F BTB08462 COCc1c(cc(c(n1)S)C#N)C(=O)OC SPB04228 c1cc(cnc1)CNC(=O)c2ccc(cc2[N+](=O)[O-])Cl BTB07297 c1ccc2c(c1)n(c(=O)o2)CCC(=O)NC(=N)c3ccc(cc3)C(F)(F)F SPB06759 Cc1cc(no1)C(=O)N/N=C/c2c(c[nH]n2)Cl SPB02875 Cc1cccc(c1NC(=O)O/N=C(\C)/c2c(n3c(s2)nc(n3)C(F)(F)F)C)C SPB05703 COC(=O)C(=C(NC(=O)N)SC)C(=O)OC SPB05745 CCCCN1C(C(N(C1=O)c2nnc(s2)C(C)(C)C)O)c3ccc(cc3)C BTB08422 c1cc(ccc1NC(=O)Nc2ccc(nc2)Oc3ccc(cc3Cl)Cl)SC(F)(F)F BTB08360 CC(=O)Nc1ccc(cc1C(F)(F)F)I TL00261 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(nc2)Oc3cccnc3 BTB07222 Cc1c2c(c(sc2nc(c1/N=N/c3cc(cc(c3)Cl)Cl)C)C(=O)Nc4cccc(c4)C#C)N SPB06748 c1ccc(cc1)c2c3ccccc3[nH]c(=O)n2 XBX00299 CC(C)(C)NC(=O)N1CCN(CC1)c2ccc(cn2)C#N SPB06787 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C#N)Cl SPB06790 CS(=O)(=O)N1CCN(CC1)c2ccc(cn2)C#N SPB06791 c1cc(c(cc1c2c(c(=O)c3c(cc(cc3o2)O)O)O)O)O XBX00307 c1cc(ccc1NC(=O)NNC(=O)c2c(=O)ccn(n2)c3ccc(cc3)F)Cl SPB04060 CC(C)NC(=O)NNC(=O)c1c(=O)ccn(n1)c2ccc(cc2)F SPB04063 CCOC(=O)CSc1nc2cc(cnc2n1C)C(F)(F)F SPB04065 Cc1ccc(c(c1)Oc2ccc(cn2)NC(=O)Nc3ccc(cc3)SC(F)(F)F)C BTB08361 Cn1ccnc1Sc2c[nH]c(=S)nc2c3ccc(cc3)Cl SPB04191 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4cc(ccc4Cl)C(F)(F)F SPB06721 CC(C)(C)NC(=O)O/N=C(/c1ccc(cc1)NS(=O)(=O)C)\N SPB06774 c1cc(ncc1C#N)N2CCN(CC2)C(=O)C3CC3 SPB06783 CCOC(=O)c1cc(n(c1C)c2ccccc2)C SP00019 CC(C)S(=O)(=O)c1c(csc1SC)N SP00041 CCOC(=O)c1cc(n(c1C)c2ccccc2)C(C)(C)C SP00039 C/C(=N\NC(=O)N)/c1ccc(cc1)OC SEW05744 Cc1c(sc(n1)CCn2cccc(c2=O)C(F)(F)F)/C(=N/Nc3ccc(cc3F)F)/C SPB06617 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccccc2NC(=O)c3ccccc3)C#N SPB06618 c1cc(nc(c1[N+](=O)[O-])Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05709 Cc1cc(c(n1C)C)C(=O)O CC08601 c1ccc2c(c1)n(c(=O)o2)Cc3cccc(c3)C#N SPB06722 c1ccc(cc1)Nc2c(c(=O)[nH]c(=O)[nH]2)C#N SPB05760 COc1ccc(cn1)C(=S)N SPB05765 CCn1c(c(c(n1)C)[N+](=O)[O-])c2nnnn2c3ccc(cc3)C(F)(F)F SPB02923 CC1(CCC(c2c1cc3c(c2)C(CCC3(C)C)(C)C)(C)C)C TL00204 c1ccc(cc1)c2nc3c(ncnc3o2)N SEW05740 c1cc(ccc1C(F)(F)F)n2c(nnn2)c3ccno3 SPB02926 c1cc(ccc1Cn2c(c(cn2)Br)/C=N/NC(=O)Cc3cc(sc3Br)Br)Cl SPB02946 Cc1c(sc(n1)c2ccccc2)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N SPB02947 CC(=O)c1ccn(c1)S(=O)(=O)c2ccc(cc2)Cl BTB07122 c1ccc(c(c1)c2nc(c(o2)N)C#N)OC(F)(F)F SEW05747 CC(=O)/C(=C\N(C)C)/Sc1ccccn1 SPB04125 CCCNC(=S)N1CCC(CC1)C(=O)c2ccc(cc2)C SEW05720 Cc1c(c(no1)c2ccccc2)C(=O)NC(=N)c3ccc(cc3)C(F)(F)F SPB06674 c1ccc(cc1)CSc2nnc(n2Cc3ccco3)c4cc(nc(c4)OCC(F)(F)F)OCC(F)(F)F SPB06677 c1csc(n1)NC=C(C#N)C#N BTB08384 c1cc(ccc1NC(=S)NNC(=O)COc2ccc(cc2)SC(F)(F)F)F BTB08378 c1cc(sc1)c2nc(cs2)Cc3nnc(o3)c4ccc(cc4)Cl SPB02942 c1ccc2c(c1)n(c(=O)o2)CCC(=O)Oc3cccc(c3)Cl SPB02945 c1cc(ccc1Oc2ccc(cn2)C(F)(F)F)Oc3ccc(cn3)[N+](=O)[O-] SEW05742 Cc1ccc(cn1)/C(=N/Nc2nc(cs2)C(C)(C)C)/C.Br BTB07264 c1cc(ccc1CNS(=O)(=O)c2c(cc(cc2Cl)C(F)(F)F)Cl)C(F)(F)F SEW05722 c1ccnc(c1)NNC(=O)NC(=O)c2ccc(cc2)C(F)(F)F SPB01463 C/C(=C(/C(=O)c1ccc(cc1)C(F)(F)F)\C(=O)OC)/NC SPB01465 COC(=O)c1cc(ccc1Oc2ccc(c(n2)Oc3ccc(cc3C(=O)OC)Cl)[N+](=O)[O-])Cl SEW05741 CN1CCN(CC1)c2ccccc2/C=C(/C#N)\S(=O)(=O)C SEW05745 c1cc(c(cc1F)F)C(=O)C2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05746 CC(C)(C)C(=O)O/N=C(/c1ccc(c(c1)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl)\N SPB01102 Cc1c(c(nc(n1)c2ccccc2)OC(=O)N(C)C)Oc3cccc(c3)C(F)(F)F SPB04078 c1csc(c1OCc2c(cc(cn2)C(F)(F)F)Cl)C(=O)NN SPB06770 CS(=O)(=O)Nc1ccc(cc1)/C(=N/OC(=O)Nc2ccccc2)/N SPB06771 Cc1ccc(cn1)/C(=N/Nc2nc(cs2)c3ccc(cc3)Cl)/C BTB07265 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)SC(F)(F)F BTB08442 c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cn3)C#N SPB06784 Cc1ccc(cc1)Oc2c(nc(nc2O)c3ccccc3)C SPB04073 Cc1c(c(nc(n1)c2ccccc2)O)Oc3ccc(cc3Cl)Cl SPB04075 CC(=O)Nc1ccc(cc1C(F)(F)F)[N+](=O)[O-] TL00253 CC(=O)Nc1ccc(cc1C(F)(F)F)C#N TL00263 Cc1c(c(nc(n1)c2ccccc2)OC(=O)N(C)C)Oc3ccc(cc3Cl)Cl SPB04079 c1ccc(cc1)C(=O)c2c(=O)ccn(n2)c3cccc(c3)Cl SPB04028 Cc1c(c(nc(n1)C)N2CCCCC2)Oc3ccc(cc3Cl)Cl SPB04082 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4ccc(cc4Cl)Cl SPB06641 c1(nc(=N)nc(s1)S)N TL00237 Cn1c2c(cc(cn2)C(F)(F)F)nc1SCc3ccccc3 SPB04052 c1cc(cc(c1)Cl)NC(=O)NNC(=O)c2c(=O)ccn(n2)c3ccc(cc3)F SPB04061 CCOC(=O)c1c(c2c(c(c(nc2s1)C)/N=N/c3ccccc3)C)N SPB06753 Cn1c(nnc1SCC(=O)Nc2cccc(c2)Cl)Cn3cc(ccc3=O)C(F)(F)F SPB06754 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)Sc2ccc(cc2)C(F)(F)F SPB04064 Cn1c2c(cc(cn2)C(F)(F)F)nc1SCC(=O)O SPB04066 c1ccc(cc1)C(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06815 CS(=O)(=O)Nc1ccc(cc1)/C(=N/OC(=O)c2ccccc2Cl)/N SPB06764 c1cc(cc(c1)Cl)OC/C(=N/OC(=O)CCn2cc(ccc2=O)C(F)(F)F)/N SPB06766 c1cc(ccc1NC(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl)SC(F)(F)F SPB06874 Cc1cc(no1)/C(=N/OC(=O)Nc2ccccc2)/N SPB04163 c1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccc(c(c2F)F)F BTB08468 Cc1ccc(cc1)S(=O)(=O)CC(=O)Nc2ccc(c(c2F)F)F BTB08469 c1ccc(cc1)c2nnc(o2)Cc3cc(sc3Br)Br SPB02951 Cc1c(sc(n1)c2ccccc2)c3nc(no3)c4ccc(cc4)C(F)(F)F SPB02957 Cn1c(nnc1Sc2cnc(nc2c3ccc(cc3)Cl)S)C(F)(F)F SPB04168 CN(C)/C=C(\C(=O)Nc1ccc(c(c1F)F)F)/S(=O)(=O)c2ccc(cc2)Cl BTB08475 COc1ccc(cc1)N2C(=O)C=CC2=O BTB07155 c1cc(c(cc1F)F)Oc2ccc(cn2)[N+](=O)[O-] BTB07167 c1cc(ccc1Oc2ccc(cn2)[N+](=O)[O-])Br BTB07170 c1ccc(c(c1)COc2ccc(cc2)/C(=N/O)/N)F SPB01466 CCOC(=O)C(=CNc1ccc(nc1)Oc2cccnc2)C(=O)OCC BTB07237 COc1cccc(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OC BTB07242 COc1cccc(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC BTB07243 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl SPB05814 COC(c1ccnc(n1)SCC(=O)Nc2cc(cc(c2)Cl)Cl)OC SPB04262 CC(=O)c1cccn1S(=O)(=O)c2ccccc2 BTB07161 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Br)Br)Br)OC)[N+](=O)[O-] BTB07574 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)C)C#N SPB06808 Cc1cc(no1)c2nc(on2)c3ccccc3 SPB04275 COc1ccc(cc1)Oc2ccc(cn2)[N+](=O)[O-] BTB07173 c1ccc(c(c1)NC(=O)c2cccs2)Sc3c(cncc3Cl)Cl SPB06902 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)Cl)Sc3c(cncc3Cl)Cl SPB06903 CCCCn1c(cn(c1=O)c2nnc(s2)C(C)(C)C)CSc3ccccn3 BTB08404 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCNCC2)C#N SPB06796 CN(C)/C=C(\C(=O)Nc1ccc(c(c1F)F)F)/S(=O)(=O)c2ccccc2 BTB08491 CSc1c(cccn1)C2=N/C(=C\c3ccc(cc3)C(F)(F)F)/C(=O)O2 BTB08778 CCCCCC(=O)O/N=C(\C)/c1ccn(c1)S(=O)(=O)c2ccc(cc2)Cl BTB07141 c1cc(ccc1NC(=O)N/N=C(/c2ccc(cn2)C(F)(F)F)\N)Cl SPB06895 c1cc(c(cc1Cl)Sc2ccc(cn2)N)Cl BTB07162 c1cc(ccc1Oc2ccc(cn2)[N+](=O)[O-])F BTB07165 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)N BTB08806 c1cc(ccc1Sc2ccc(cn2)N)Cl BTB07168 c1ccc(cc1)NC(=O)N/N=C(/c2ccc(cn2)C(F)(F)F)\N SPB06896 CC(C)(C)NC(=O)N/N=C(/c1ccc(cn1)C(F)(F)F)\N SPB06898 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)Sc3c(cncc3Cl)Cl SPB06899 c1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)Sc3c(cncc3Cl)Cl SPB06901 CC(C)c1cc(cc(c1)Oc2ccc(cn2)[N+](=O)[O-])C(C)C BTB07169 Cn1c2c(cc(cn2)C(F)(F)F)nc1S SPB04045 Cc1ccc(cc1)Oc2c(nc(nc2OC(=O)N(C)C)c3ccccc3)C SPB04077 Cc1c2c(onc2c(=O)n(n1)c3ccc(cc3)Cl)C SPB04295 Cc1c2c(onc2c(=O)n(n1)c3ccccc3C(F)(F)F)C SPB04297 Cc1ccc(cc1)NC(=O)c2cc(on2)c3cccs3 SPB04301 Cc1c2c(c(=O)[nH]nc2c3ccccc3)no1 BTB08875 Cc1ccc(c(n1)[N+](=O)[O-])OC(=O)c2c(c3ccccc3s2)Cl BTB07321 Cc1ccc(cc1)Oc2c(cccn2)C(=O)N BTB08807 c1cc(cc(c1)NC(=O)N/N=C(/c2ccc(cn2)C(F)(F)F)\N)C(F)(F)F SPB06897 Cc1ccc(c(n1)[N+](=O)[O-])OCc2ccc(c(c2)Cl)Cl BTB07290 Cc1cc(no1)/C(=N\OC(=O)Nc2ccc(cc2)Cl)/N SPB04164 c1cc(nnc1NCCO)NCCO BTB07274 Cc1ccc(cn1)/C(=N/N=C(\N=C\N(C)C)/SCc2cc(cc3c2OCOC3)F)/C BTB07270 CS(=O)(=O)n1c(c(cn1)Sc2ccc(cc2)Cl)c3ccc(cc3)Cl SPB04205 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3ccccc3)C#N SPB06805 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3ccccc3Cl)C#N SPB06806 CS(=O)(=O)Nc1ccc(cc1)/C(=N/OC(=O)c2cccc(c2)C(F)(F)F)/N SPB06762 Cc1ccc(c(n1)[N+](=O)[O-])OC(=O)c2cccs2 BTB07322 Cc1c(sc(n1)c2ccccc2)c3nc(no3)c4ccc(o4)[N+](=O)[O-] SPB02956 Cc1c(sc(n1)c2ccccc2)c3nc(no3)c4ccc(cc4)C(C)(C)C SPB02958 CCCCN1C(C(N(C1=O)c2nnc(s2)C(C)(C)C)O)c3ccc(c(c3)Cl)Cl BTB08423 Cc1cc(no1)/C(=N/OC(=O)Nc2cccc(c2)C(F)(F)F)/N SPB04165 c1cc(c(c(c1NC(=O)CSc2nnc(s2)N)F)F)F BTB08428 Cn1c(nnc1Sc2c[nH]c(=S)nc2c3ccccc3)C(F)(F)F SPB04192 COC(c1ccc(c(n1)SCc2ccc(cc2)Cl)C#N)OC SPB04266 c1cc(cc(c1)NC(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F SPB06813 c1cc(ccc1C(=O)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F)Cl SPB06831 c1cnc(nc1)Sc2cnc(nc2c3ccc(cc3)Cl)SCC(=O)c4ccc(cc4)Cl SPB04323 Cc1ccc(cc1)CSc2c(ccc(n2)C(OC)OC)C#N SPB04328 c1cc(ccc1COc2ccc(cc2)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N)Cl BTB07091 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl)C(F)(F)F BTB07092 Cc1ccc(cc1)COc2ccc(cc2)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N BTB07093 Cc1c(c(on1)C)C(=O)N2CCC(CC2)C(=O)c3ccc(cc3F)F SEW05738 C/C(=N\NC(=O)c1ccccc1)/c2ccccc2O BTB08523 c1cc2cccnc2c(c1)S(=O)(=O)Nc3ccc(nc3)Oc4ccc(cc4)F BTB08527 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)C#N SPB06807 c1ccc(c(c1)NC(=O)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F)Cl SPB06826 Cc1ccc(cn1)/C(=N/NC(=S)N)/C BTB07184 Cc1c(cnn1C(=O)c2ccccc2)Sc3ccc(cc3)Cl SPB04122 Cc1c(cnn1C(=O)c2ccc(cc2)Cl)Sc3ccc(cc3)Cl SPB04123 CCOC(=O)c1cc(n(c1C)Cc2ccncc2)C SP00029 COCc1c(cc(c(n1)SCC(=O)OC)C#N)C(=O)OC SPB04251 Cc1c(c(nc(n1)C)NCc2ccc(cc2)Cl)Oc3ccc(cc3Cl)Cl SPB04080 c1cc(c(cc1Cl)C2CCCCC2)Oc3ccc(cn3)[N+](=O)[O-] BTB07146 CNc1nc(ns1)c2cccs2 SPB06924 c1cc(ccc1C(=NOC(=O)c2ccc(c(c2)Cl)Cl)c3ccc(cc3)F)F BTB07191 c1ccc(cc1)/C=C/S(=O)(=O)c2ccc(c(c2)Cl)F BTB08483 Cc1cc(no1)/C(=N/OC(=O)c2ccno2)/N SPB04172 Cn1c(nnc1Sc2cnc(nc2c3ccccc3)SCc4ccc(cc4)Cl)C(F)(F)F SPB04201 c1cc(ccc1c2c(cnn2S(=O)(=O)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl)Cl SPB04204 c1ccc(c(c1)/C=N/c2ccc(cc2)Cl)OC(F)F BTB08522 Cc1ccc(cc1)S(=O)(=O)n2c(c(cn2)Sc3ccc(cc3)Cl)C SPB04208 Cc1c(c(nc(n1)C)NCc2ccc(cc2)OC)Oc3ccc(cc3Cl)Cl SPB04081 Cc1cc(no1)/C(=N/OC(=O)c2c(nns2)C)/N SPB04170 c1cc(cc(c1)C(=O)Sc2ccc(cc2)Cl)Cn3cc(ccc3=O)C(F)(F)F SPB06696 c1cc(cc(c1)C(=O)Sc2cccc(c2)C(F)(F)F)Cn3cc(ccc3=O)C(F)(F)F SPB06698 c1ccc(cc1)NC(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06811 Cc1ccc(c(n1)[N+](=O)[O-])OC(=O)c2c(nn(n2)c3ccccc3)C BTB07315 Cc1cccc(c1)C2NC(=NN2)c3ccc(cn3)C(F)(F)F SPB06888 c1ccc(cc1)COc2cccc(c2)CC#N BTB07332 COc1cccc(c1OC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)OC BTB07579 Cc1ccc(c(n1)[N+](=O)[O-])OS(=O)(=O)c2ccc(cc2)F BTB07316 c1cc(ccc1NC(=O)NNC(=O)c2csc(n2)c3c(cc(cn3)C(F)(F)F)Cl)Cl SPB05809 CCCSc1ccc2c3c1cccc3C(=O)N(C2=O)c4ccccc4 BTB11678 c1cc(c(cc1F)F)Oc2ccc(cn2)N BTB07203 CC(C)(C)c1ccc(cc1)C(=O)Sc2ccc(cn2)C(F)(F)F SPB02837 CS(=O)(=O)Nc1ccc(cc1)/C(=N/OC(=O)c2cccs2)/N SPB06763 c1cc(ncc1C#N)N2CCNCC2 SPB06765 Cc1ccc(cc1)OC/C(=N/OC(=O)CCn2cc(ccc2=O)C(F)(F)F)/N SPB06767 c1cc(ccc1NC(=O)CSc2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)F)Cl SPB02855 CC(=O)Nc1ccc(cc1)C2NC(=NN2)c3ccc(cn3)C(F)(F)F SPB06890 c1cc(ccc1CSCC(=O)Nc2nnc(s2)SCC(=O)Nc3ccc(c(c3F)F)F)Cl BTB08501 Cc1ccc(cc1)C(=O)/C(=C\N(C)C)/Sc2ccc(cc2)C SPB04130 Cc1cc(no1)c2nc(on2)c3c(nns3)C SPB04222 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2cc(ccc2Oc3ccc(cc3)OC)[N+](=O)[O-])/N BTB08511 c1cc(ccc1[N+](=O)[O-])OC/C(=N/OC(=O)CCn2cc(ccc2=O)C(F)(F)F)/N SPB06769 Cc1ccc(cc1)NC(=O)O/N=C(/c2ccc(cc2)NS(=O)(=O)C)\N SPB06772 CN1CCN(CC1)c2ccccc2/C=N/NC(=O)c3cccnc3 SEW05748 c1cc(cc(c1)NC(=O)N2CCN(CC2)c3c(cncc3Cl)Cl)C(F)(F)F SPB06850 COc1ccc(cc1)Oc2ccc(cc2C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N)[N+](=O)[O-] BTB08512 c1cc(cc(c1)Cl)NC(=O)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F SPB06827 Cc1c(sc(n1)c2cccs2)c3cc(n[nH]3)SC SPB02889 c1ccc(c(c1)NC(=O)NC(=O)c2ccno2)Cl SPB02896 c1cc(ccc1NC(=O)NC(=O)c2ccno2)F SPB02897 c1cc(ccc1n2ccc(=O)c(n2)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl)F SPB02856 c1ccc(cc1)SCC(=O)Nc2ccc(c(c2F)F)F BTB08440 c1ccc(cc1)S(=O)(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06819 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl SPB06821 Cc1c(n(oc1=O)C)C(=O)NNc2c(cccc2Cl)Cl SPB02891 Cc1ccc(cc1)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F SPB06829 CSc1nnc(o1)c2ccc(cn2)C(F)(F)F SPB06830 CCCCCC(=O)O/N=C(\C)/c1cc[nH]c1 BTB07181 CC(=O)c1ccc(cc1)Oc2ncc(s2)[N+](=O)[O-] SPB02901 CC(C)Oc1ccccc1Oc2ccc(cn2)N BTB07183 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)Nc2ccc(cc2)Cl SPB02902 Cc1cc(no1)C(=O)N/N=C/c2c(c[nH]n2)Br SPB02876 c1cc(c(c(c1)Cl)c2cc(on2)CSc3nnc(n3C4CCCCC4)O)Cl SPB02883 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)SCc3cc(no3)c4c(cccc4Cl)Cl SPB02884 Cc1c(sc(n1)c2cccs2)C(=O)C=C(SC)SC SPB02885 COC(=O)c1ccc(cc1NS(=O)(=O)c2ccc(cc2)Cl)Cl BTB08453 c1cc(ccc1S(=O)(=O)CC(=O)Nc2ccc(c(c2F)F)F)Cl BTB08459 CC(=O)Nc1nnc(s1)SCC(=O)Nc2ccc(c(c2F)F)F BTB08460 C/C(=N\OC(=O)c1cccc(c1)F)/c2cc[nH]c2 BTB07182 c1cc(ccc1Oc2ccc(cn2)N)Br BTB07205 c1cc(ccc1C(=NOC(=O)C(Cl)(Cl)Cl)c2ccc(cc2)F)F BTB07207 c1cc(cc(c1)Cl)NC(=O)NNC(=O)c2csc(n2)c3cnccc3C(F)(F)F SPB05784 Cc1cc(ccc1Cl)Oc2ccc(cn2)N BTB07209 CC(C)c1cc(cc(c1)Oc2ccc(cn2)N)C(C)C BTB07210 c1cc(c(cc1C(=O)Nc2nnc(s2)SCC(=O)Nc3ccc(c(c3F)F)F)Cl)Cl BTB08431 c1cc(ccc1Oc2ccc(cn2)C#N)Cl SPB05789 c1cc(ccc1Oc2ccc(cn2)/C(=N/O)/N)Cl SPB05791 c1cc(cc(c1)C(=O)Nc2cccc(c2)C(F)(F)F)Cn3cc(ccc3=O)C(F)(F)F SPB06694 CC(=O)/C(=C\N(C)C)/Sc1nnc(n1C)C(F)(F)F SPB04126 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4cc(ccc4Cl)OC SPB06709 c1cc(ccc1N2CCCCCCC2)[N+](=O)[O-] XBX00316 c1ccn(c1)S(=O)(=O)c2ccc(cc2)Cl BTB07116 Cc1ccc(nn1)NNC(=O)Nc2ccc(cc2)Cl BTB07301 Cc1ccc(c(n1)[N+](=O)[O-])OS(=O)(=O)c2c(c(sc2Cl)Cl)Br BTB07328 CCOC(=O)c1c(c(c(=N)n(n1)c2ccc(cc2)C(C)(C)C)C#N)C BTB08886 c1cc(c(nc1)Sc2ccc(cc2)Cl)C(=O)N BTB08808 CC(C)(C)C1=NN2C(=N)CC(=O)N=C2S1 BTB08811 C1C(=N)N2C(=NC1=O)SC(=N2)C(F)(F)F BTB08812 Cc1cccc(n1)NC(=O)c2ccc(cc2N)Cl BTB07303 CC(=O)Nc1c(cccn1)OC(=O)C BTB07311 CS(=O)(=O)Nc1ccc(cc1)/C(=N/OC(=O)c2ccc(cc2)Cl)/N SPB06761 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)c3ccccc3)C#N SPB06792 CC1CCCN(C1)c2ccc(cc2)[N+](=O)[O-] XBX00315 Cn1c(c2c(n1)CCCC2)N(C)S(=O)(=O)c3ccc(cc3)Cl BTB07105 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3ccc(cc3)/C(=C/c4ccc(cc4)C(F)(F)F)/C#N BTB07112 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)/C(=C/c4ccc(cc4)C(F)(F)F)/C#N BTB07115 C#CCOC(=O)NC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl SPB01190 c1ccc(c(c1)S(=O)(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl)Cl SPB06820 Cc1cc(no1)/C(=N/OC(=O)c2ccccc2Cl)/N SPB04134 Cc1c(cc(o1)C(C)(C)C)C(=O)O SP00043 Cc1c(cc(o1)c2ccccc2)C(=O)O CC14901 c1cc(sc1)C(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl SPB06867 CS(=O)(=O)NNC(=O)c1c(ccs1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB06822 c1cc(ncc1C(F)(F)F)c2nnc(o2)S SPB06824 c1ccc(cc1)NC(=O)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F SPB06825 CS(=O)(=O)Nc1ccc(cc1)/C(=N/OC(=O)Nc2ccc(cc2)C(F)(F)F)/N SPB06773 Cc1c(sc(n1)c2ccccc2)C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N SPB02948 Cc1cc(c(cc1Cl)C)S(=O)(=O)Oc2ccc(cc2)CC#N BTB07098 c1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cn3)C#N SPB06781 Cc1c(snn1)C(=O)N2CCN(CC2)c3ccc(cn3)C#N SPB06782 c1cc(ccc1NC(=O)N2CCN(CC2)c3ccc(cn3)C#N)Cl SPB06785 C/C(=N\OC(=O)c1cc2ccccc2s1)/c3cc[nH]c3 BTB07179 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2cc[nH]c2 BTB07180 c1cc(cc(c1)NC(=O)N2CCN(CC2)c3ccc(cn3)C#N)C(F)(F)F SPB06786 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C#N SPB06788 c1ccc(c(c1)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C#N)Cl SPB06789 c1ccn(c1)c2cc(c(cc2Cl)NC(=O)c3ccc(cc3)Cl)Oc4ccc(cc4)Cl BTB07558 Cc1ccc(cn1)/C(=N/O)/C BTB07185 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)c3ccc(cc3)Cl)C#N SPB06793 Cn1c(c2c(n1)CCCC2)N(C)C(=O)Nc3ccccc3 BTB07099 Cn1c(c2c(n1)CCCC2)N(C)C(=O)Nc3ccc(cc3)Cl BTB07100 Cc1c(c(nc(c1/N=N/c2cc(cc(c2)Cl)Cl)C)SCC#C)C#N SPB06732 Cc1c(c(nc(c1/N=N/c2ccccc2)C)SCC(=O)Nc3ccccc3Cl)C#N SPB06739 Cc1ccccc1/N=N/c2c(c(c(nc2C)SCC(=O)Nc3cc(cc(c3)Cl)Cl)C#N)C SPB06741 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccn(c2)S(=O)(=O)c3ccccc3 BTB07124 CCCCCC(=O)O/N=C(\C)/c1ccn(c1)S(=O)(=O)c2ccccc2 BTB07126 CC(C)(C)C(=O)ON=C(c1ccc(cc1)F)c2ccc(cc2)F BTB07198 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cccc2F)F)OC)[N+](=O)[O-] BTB07589 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2ccn(c2)S(=O)(=O)c3ccccc3 BTB07125 c1ccc(cc1)S(=O)(=O)n2ccc(c2)c3cnc4cc(c(cc4n3)Cl)Cl BTB07133 Cc1ccc(c(n1)[N+](=O)[O-])OCc2c(cccc2Cl)F BTB07288 Cc1ccc(cc1)COc2ccc(nc2[N+](=O)[O-])C BTB07289 CCOC(=O)CNC(=O)c1cccnc1Sc2ccc(cc2)C BTB08779 c1ccc(cc1)NC(=S)NNC(=O)COc2ccc(cc2)SC(F)(F)F BTB08369 c1ccc(cc1)N2C(=O)c3cccc4c3c(ccc4Sc5ccccc5)C2=O BTB11679 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl)Cl SPB06876 c1cc(ccc1NC(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl)Cl SPB06877 Cc1ccc(cc1)C(=O)/C(=C\N(C)C)/Sc2ccc(cc2)Cl SPB04129 c1cc(cc(c1)C(=O)O/N=C(/c2cccc(c2)C(F)(F)F)\N)Cn3cc(ccc3=O)C(F)(F)F SPB06706 COC(=O)c1c(=O)[nH]c(nc1SC)c2ccccc2 BTB08846 Cc1ccc(c(n1)[N+](=O)[O-])OS(=O)(=O)c2ccc(cc2)Cl BTB07318 CCOC(=O)c1cc(n(c1C)c2ccccc2)c3ccccc3 SP00040 COc1ccc(cc1)C(=O)Nc2ccccc2Sc3c(cncc3Cl)Cl SPB06900 c1ccc(cc1)NC(=O)Nc2ccccc2Sc3c(cncc3Cl)Cl SPB06905 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)Cl)Sc3c(cncc3Cl)Cl SPB06907 CC(C)(C)C(=O)N1CCN(CC1)c2nc3ccc(cc3s2)Cl SPB06869 CCOC(=O)/C(=C/Nc1ccc(nc1)Oc2cccnc2)/C#N BTB07231 CCCCN1C(C(=O)N(C1=O)c2nnc(s2)C(C)(C)C)c3ccc(c(c3)C)Cl BTB08413 CCCCN1C(C(=O)N(C1=O)c2nnc(s2)C(C)(C)C)c3ccc(cc3)F BTB08414 Cc1ccc(cn1)/C(=N/N=C(\N=C\N(C)C)/SCc2ccc(cc2Cl)Cl)/C BTB07267 c1cc(cc(c1)C(=O)NC(=N)c2ccc(cc2)Cl)Cn3cc(ccc3=O)C(F)(F)F SPB06711 Cc1ccc(cc1)n2c(=O)c3c(c(n2)C)c(on3)C SPB04296 COc1ccc(c(c1C(=O)NC(=O)Nc2nc(nc(n2)OC)OC)OC)[N+](=O)[O-] BTB07597 c1cc(sc1)CNc2ccc(cn2)[N+](=O)[O-] BTB07601 Cc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)C BTB07609 Cc1c2c(onc2c(=O)n(n1)c3cc(ccc3Cl)C(F)(F)F)C SPB04298 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)C(OC)OC SPB04261 CSc1nnc(n1CCNC(=O)Nc2cccc(c2)Cl)SC BTB07618 Cc1c(c(nc(n1)c2cccc(c2)OC)SCc3ccccc3)C(=O)C SPB05812 Cc1cc(no1)c2nc(on2)c3cccs3 SPB04183 CCOC(=O)c1cc(nn1C(=O)c2ccccc2)c3cccs3 SPB04185 Cn1ccnc1SCC(=O)c2ccc(cc2)Cl BTB08489 c1ccc(cc1)/C=C/c2c(=O)nc([nH]n2)c3ccccc3 BTB11706 COc1ccc(cc1)c2cc3c(s2)nc(nn3)c4ccccc4 BTB11716 Cc1c2c(onc2c(=O)n(n1)c3ccc(cc3F)F)C SPB04284 Cc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)[N+](=O)[O-])OC)C BTB07719 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OC)Cl)[N+](=O)[O-] BTB07724 c1ccc(c(c1)C(=O)O)SCCC(=O)O BTB11506 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OC)Br BTB07623 c1cc(cc(c1)C(F)(F)F)C(=O)N/N=C(/c2ccc(cn2)C(F)(F)F)\N SPB06885 c1ccc(cc1)c2c(=S)ssc2SCC(=O)Nc3ccc(cc3)Cl BTB08456 Cc1ccc(nn1)NNC(=O)NC(=O)c2c(cccc2Cl)F BTB07302 Cc1ccc(c(n1)[N+](=O)[O-])OS(=O)(=O)c2cc(c(s2)Br)Br BTB07326 C/C(=N\O)/c1ccn(c1)S(=O)(=O)c2ccccc2 BTB07123 COc1ccc(c(c1C(=O)NC(=O)Oc2c(cc(cc2Cl)F)Cl)OC)[N+](=O)[O-] BTB07580 Cc1c2c(onc2c(=O)n(n1)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C SPB04283 c1cc(ccc1C(=O)OC2=C(CCN(c3c2ccc(c3)Cl)S(=O)(=O)c4ccc(cc4)Cl)C#N)Cl BTB08604 c1ccc(cc1)c2cc3c(s2)nc(nn3)c4ccccc4 BTB11714 CC(C)(C)c1ccc(cc1)C(=O)OC2=C(CCN(c3c2ccc(c3)Cl)S(=O)(=O)c4ccc(cc4)Cl)C#N BTB08607 COc1nc(nc(n1)OC)Nc2ccccc2 BTB08898 CC(=O)c1ccccc1C(=O)c2ccccc2 BTB08538 Cc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccccc3N(CC=C)S(=O)(=O)c4ccc(cc4)Cl BTB08796 Cc1cccc(c1C)Oc2ccc(cn2)N BTB07213 c1cc(c(cc1Cl)C2CCCCC2)Oc3ccc(cn3)N BTB07221 Cc1ccc(c(n1)[N+](=O)[O-])OS(=O)(=O)c2cc(sc2Cl)Cl BTB07327 c1ccc(c(c1)N)N2C(=O)c3cccc4c3c(ccc4)C2=O BTB11682 Cc1ccc(cc1)S(=O)(=O)N(CC=C)c2ccccc2C3=N/C(=C\c4ccc(cc4)Cl)/C(=O)O3 BTB08797 Cc1ccc(cc1)S(=O)(=O)N(CC=C)c2ccccc2C3=N/C(=C\c4cccc(c4)Cl)/C(=O)O3 BTB08798 COc1ccc(c(c1C(=O)OC)OC)NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)[N+](=O)[O-])OC BTB07730 Cc1cccc(c1)n2c(c(cn2)C#N)N BTB07731 Cc1ccc(c(n1)[N+](=O)[O-])OS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB07317 c1ccc(cc1)c2nc3c(cc(s3)c4ccc(cc4)Cl)nn2 BTB11717 CCOC(=O)c1cc(c(nc1C)S)C#N SPB04231 c1cc(ccc1CC#N)Oc2ccc(cn2)[N+](=O)[O-] BTB07337 C=CCN(c1ccccc1C2=N/C(=C\c3ccc(cc3)Cl)/C(=O)O2)S(=O)(=O)c4ccc(cc4)Cl BTB08792 c1ccc(cc1)NC(=O)Nc2ccc(nc2)Oc3cccnc3 BTB07226 COc1ccc(cc1)C(c2ccccc2)(c3ccccc3)OC[C@@H]4[C@H](C[C@@H](O4)n5ccc(nc5=O)NC(=O)c6ccccc6)O BTB14112 c1cc(ccc1/N=C/c2cc(cc(c2O)Cl)Cl)OC(F)(F)F BTB08525 COc1ccc(cc1)Oc2ccc(cc2C(=O)NNC(=O)c3ccc(cc3Cl)Cl)[N+](=O)[O-] BTB08518 COc1ccc(cc1)Oc2ccc(cc2C(=O)NNC(=O)c3cccc(c3)OC)[N+](=O)[O-] BTB08520 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)Oc3cccnc3 BTB07232 c1cc(cnc1)Oc2ccc(cn2)N(S(=O)(=O)c3ccc(cc3)Cl)S(=O)(=O)c4ccc(cc4)Cl BTB07234 c1ccc2c(c1)nc(s2)SCC(=O)Nc3ccc(cc3)Br BTB14121 c1cc(ccc1c2nnc(o2)Cc3cc(sc3Br)Br)Cl SPB02949 Cc1ccc(c(n1)[N+](=O)[O-])Oc2c(cccn2)[N+](=O)[O-] BTB07277 Cc1ccc(c(n1)[N+](=O)[O-])Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB07283 Cc1ccc(c(n1)[N+](=O)[O-])Oc2ccc(cc2)[N+](=O)[O-] BTB07284 Cc1ccc(cc1)S/C(=C/N(C)C)/C(=O)C SPB04124 Cn1ccnc1Sc2cnc(nc2c3ccccc3)SCC(=O)c4ccc(cc4)Cl SPB04212 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)OC)[N+](=O)[O-] BTB07573 CC(C)SCC(=O)Nc1ccc(cc1)C(=O)C BTB14119 Cc1cc(c(c(c1)C)NC(=O)NC(=O)c2c(ccc(c2OC)Cl)OC)C BTB07638 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OC)Cl BTB07650 COC(c1ccc(c(n1)SCc2ccccc2)C#N)OC SPB04331 COc1c(cc(c(c1C(=O)O)OC)Cl)[N+](=O)[O-] BTB07671 c1ccn(c1)c2cc(c(cc2Cl)N)Oc3ccc(cc3)Cl BTB07554 Cc1cc(no1)c2nc(on2)c3cc(on3)C SPB04213 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)c3c(nns3)C)C#N SPB06794 COc1ccc(cc1)Oc2ccc(cc2C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F)[N+](=O)[O-] BTB08519 Cc1cc(no1)/C(=N/OC(=O)c2cc(on2)C)/N SPB04211 CC(=O)c1ccc(cc1)NC(=O)CSc2nccn2C BTB14117 c1cnc(nc1)Sc2cnc(nc2c3ccc(cc3)Cl)SCc4ccc(cc4)Cl SPB04324 CC(C)(C)C(=O)OC[C@@H]1[C@H](C[C@@H](O1)n2cnc3c2nc[nH]c3=O)O BTB14105 COC(c1ccc(c(n1)SCC(=O)Nc2ccccc2)C#N)OC SPB04359 COC(c1ccc2c(c(sc2n1)C#N)N)OC SPB04361 COC(c1ccc2c(c(sc2n1)C(=O)OC)N)OC SPB04362 c1cc(ccc1c2c(cnn2C(=O)Nc3ccc(cc3)Cl)Sc4ccc(cc4)Cl)Cl SPB04209 c1cc(ccc1C(=O)NNC(=O)c2c(ccs2)OCc3c(cc(cn3)C(F)(F)F)Cl)Cl SPB06816 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccn(c2)S(=O)(=O)c3ccc(cc3)Cl BTB07140 c1cc(cc(c1)C(F)(F)F)C(=O)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F SPB06833 CC(=O)C(C(=O)C)Sc1ncccn1 SPB04335 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)OC)Cl BTB07637 COc1ccc(c(c1C(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl)OC)Cl BTB07643 c1cc(ccc1c2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl)Cl SPB04434 c1cc(cc(c1)N/N=C(/C(=O)c2cccs2)\C(=O)C(F)(F)F)C(F)(F)F SPB04438 COc1c(cc(c(c1C(=O)N)OC)Cl)[N+](=O)[O-] BTB07697 COc1ccc(c(c1C(=O)O)OC)Cl BTB07592 c1cc(cnc1)Oc2ccc(cn2)NC(=O)Nc3ccc(cc3)Cl BTB07227 Cc1ccc(c(n1)[N+](=O)[O-])OCc2c(cccc2Cl)Cl BTB07278 c1cc(ccc1SCC(=O)NCC(=O)O)Cl BTB14099 c1cc(sc1)c2cc(no2)C(=O)Nc3ccc(cc3)Cl SPB04302 c1cc(sc1)c2cc(no2)C(=O)N3CCCCC3 SPB04303 CC(C)NC(=O)c1cc(on1)c2cccs2 SPB04304 CCOC(CC(=O)NN)OCC SPB04333 c1ccc(cc1)OCC(=O)N SPB04334 COC(c1ccc(c(n1)SCC(=O)c2ccccc2)C#N)OC SPB04337 Cc1cc(c(c(c1)C)NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)C BTB07576 c1ccc(c(c1)N)Sc2c(cncc2Cl)Cl SPB06878 COc1ccc(cc1)Oc2ccc(cc2C(=O)NCC(=O)O)[N+](=O)[O-] BTB08828 Cc1ccc(cn1)/C(=N/Nc2nc(cs2)c3ccccc3)/C.Br BTB07263 Cc1ccc(cn1)/C(=N/N=C(\N)/SCc2cc(cc3c2OCOC3)F)/C BTB07269 COC(c1ccc(c(n1)SCC#N)C#N)OC SPB04354 COC(c1ccc(c(n1)SCC(=O)c2ccc(cc2)Cl)C#N)OC SPB04356 c1cc(ccc1C(=O)/C=C/Sc2ccc(cc2)Cl)Br BTB11774 c1cc(c(c(c1)Cl)S/C=C/C(=O)c2ccc(cc2)Br)Cl BTB11775 c1ccc2c(c1)cccc2C(=O)/C=C/Sc3ccc(cc3)Cl BTB11778 COc1cccc(c1C(=O)NC(=O)Nc2c(cccc2OC)OC)OC BTB07245 Cc1cccc(c1NC(=O)NC(=O)c2c(cccc2OC)OC)C BTB07246 Cc1ccc(cc1)SCC(=O)Nc2nnc(s2)SCC(=O)Nc3ccc(c(c3F)F)F BTB08503 c1cc(sc1)C(=O)N/N=C(/c2ccc(cn2)C(F)(F)F)\N SPB06886 c1cc(ccc1C2NC(=NN2)c3ccc(cn3)C(F)(F)F)Cl SPB06887 Cc1cc(no1)/C(=N/OC(=O)c2ccc(cc2)Cl)/N SPB04127 Cc1ccc(cc1)S(=O)(=O)n2c(c(c(n2)C)Sc3ccc(cn3)C(F)(F)F)C SPB04351 Cc1c(c(n(n1)S(=O)(=O)c2ccc(cc2)Cl)C)Sc3ccc(cn3)C(F)(F)F SPB04352 CC(C)(C)c1ccc2c(c1)OCCOCCOCCOCCO2 BTB11765 c1cc2c(cc1N)OCCOCCOCCOCCO2 BTB11767 c1ccc(cc1)C(=O)/C=C/Sc2ccc(cc2)Cl BTB11769 COc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC)OC BTB07700 c1ccc(cc1)CSC2=NNC(S2)c3ccccn3 SPB06980 CSC1=NNC(S1)c2ccccn2 SPB06981 Cc1cc(cc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC)C)Br BTB07677 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)OC)Cl)Cl BTB07678 CSc1c(c(nc(n1)c2ccccc2)Sc3ccccn3)C#N BTB08925 Cc1nc(c(c(n1)Sc2cccc(c2)C(F)(F)F)C#N)SC BTB08928 c1ccc(c(c1)OC(F)(F)F)S(=O)(=O)N2CCN(CC2)c3c(cncc3Cl)Cl SPB06852 Cc1c(c(nc(n1)S)O)Oc2cccc(c2)C(F)(F)F SPB04215 Cc1ccc(cc1)Oc2c([nH]c(=S)[nH]c2=O)C SPB04216 c1c(cnc(c1C(=O)O)O)Cl SPB06836 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cccc2Cl)Cl)OC)Cl)Cl BTB07689 Cn1cc(c(n1)C2NN=C(S2)S)Cl SPB06972 COc1ccc(c(c1C(=O)OC)OC)NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC BTB07695 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC)Br)[N+](=O)[O-] BTB07699 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cccc2Cl)Cl)OC)Cl)[N+](=O)[O-] BTB07714 COc1ccc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC)Cl BTB07645 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Br)Br)Br)OC)Cl BTB07651 CCOC(=O)c1c(=O)c(cn(n1)c2ccc(cc2Cl)Cl)Sc3c(c(c(c(n3)C)C)C)C#N SPB04443 c1cc(c(cc1F)F)c2nc(cs2)C(=O)NN SPB02259 C#Cc1cccc(c1)NC(=O)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F SPB06828 c1cc(ccc1CSc2nccc(n2)/C=N/OC(=O)c3ccc(cc3)C(F)(F)F)Cl SPB04325 CC(=O)C(=NNc1ccc(cc1)OC(F)(F)F)C(=O)C SPB02907 c1cc(ccc1C(=NOC(=O)c2ccc(cc2)F)c3ccc(cc3)F)F BTB07193 c1cc(cnc1)Oc2ccc(cn2)[N+](=O)[O-] BTB07195 c1cnoc1C(=O)Nc2cc(cc(c2)Cl)Cl SPB02915 CSc1c(c(nc(n1)c2ccccc2)Nc3ccc(cc3)C(F)(F)F)C#N BTB08945 CC(=O)OCc1ccccc1Sc2ccccc2C(=O)Nc3ccccc3 BTB11500 CNC(=O)c1ccccc1Sc2ccc(cc2C(=O)O)Cl BTB11503 COc1ccc(c(c1C(=O)OC)OC)NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC BTB07713 Cc1ccccc1c2[nH]c(nn2)S BTB14101 CCOC(=O)c1ccc(cc1)NC(=O)COc2c(c(c(c(c2F)F)F)F)F BTB14129 Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2NS(=O)(=O)c3ccc(cc3)C)Sc4ccc(cc4)Cl)[N+](=O)[O-] BTB08547 c1cc(ccc1N/N=C(/C#N)\C(=S)N)OC(F)(F)F SPB02912 CCCCNC(=O)n1c(cc(n1)SC)c2c(nc(s2)c3cccs3)C SPB02913 c1cc(sc1)c2cc(c(c(n2)SCc3csc(n3)c4cccs4)C#N)C(F)(F)F SPB02920 Cc1cc(cc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)C)Br BTB07626 Cc1cc(nc(n1)NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)C BTB07628 COc1ccc(c(c1C(=O)N)OC)Cl BTB07633 Cc1ccccc1S(=O)(=O)N(CC=C)c2ccccc2C(=O)NCC(=O)O BTB08841 CCO/N=C(\C)/c1ccc(nc1)C.Cl BTB07272 CN(C)/C=C/1\C(=O)OC(=N1)c2cc(ccc2Oc3ccc(cc3)OC)[N+](=O)[O-] BTB08830 c1ccc(cc1)OCC(=O)Nc2ccc(cc2)C(=O)O BTB14126 CC(=O)c1ccccc1C(=O)c2ccc(cc2)Cl BTB08543 CN(C)/C=C/C(=O)c1ccccc1C(=O)c2ccccc2 BTB08544 COC(=O)c1ccc(cc1N(CCCC#N)S(=O)(=O)c2cccc(c2)C(F)(F)F)Cl BTB08554 c1cc(ccc1NC(=O)N2CCN(CC2)c3c(cncc3Cl)Cl)Cl SPB06849 CS(=O)(=O)N1CCN(CC1)c2c(cncc2Cl)Cl SPB06854 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Sc3ccc(cn3)C(F)(F)F SPB04348 CCn1c(cc(n1)C)C(=O)n2c(c(c(n2)C)Sc3ccc(cn3)C(F)(F)F)C SPB04349 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(/c2ccc(nc2)Oc3ccc(cc3)Cl)\N SPB05797 c1ccc2c(c1)OCC(O2)CO CC01509 COCc1c(cc2c(c(sc2n1)C(=O)OC)N)C(=O)OC SPB04247 Cc1ccc(cc1)C(=O)CSc2nnc(n2C)SCC(=O)c3ccc(cc3)C BTB08550 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)SCC(=O)c3ccc(cc3)Cl BTB08552 CCOC(=O)c1cc2c(c(sc2nc1C)C(=O)OCC)N SPB04249 c1cc(oc1)C(=O)N2CCN(CC2)c3c(cncc3Cl)Cl SPB06846 Cc1c(c(n(n1)C(=O)C)C)Sc2ccc(cn2)C(F)(F)F SPB04345 COC(c1ccc2c(c(sc2n1)C(=O)Nc3ccc(cc3)C(F)(F)F)N)OC SPB04343 c1ccc(cc1)NC(=O)N2CCN(CC2)c3c(cncc3Cl)Cl SPB06848 c1cc(sc1)c2nc(cs2)CC(=O)NNC(=O)c3ccc(cc3)Cl SPB02941 c1ccnc(c1)C2NN=C(S2)SCc3ccc(cc3)Cl SPB06966 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)NNC(=O)c2ccc(cc2)Cl SPB02961 CCOC(=O)c1cc(nn1Cc2ccc(cc2)Cl)C SPB06778 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl)C(F)(F)F SPB06872 CS(=O)(=O)N1CCN(CC1)c2nc3ccc(cc3s2)Cl SPB06873 c1cc(sc1)c2nc(sn2)Sc3ccc(cc3)Cl SPB06937 c1cc(sc1)C(=O)NC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl SPB06942 c1cnoc1c2nnnn2c3cc(cc(c3)Cl)Cl SPB02925 c1cc(ccc1n2c(nnn2)c3ccno3)Cl SPB02927 c1ccc(cc1)S(=O)(=O)N/N=C(/c2ccc(cn2)C(F)(F)F)\N SPB06963 c1ccc(c(c1)OC(F)(F)F)S(=O)(=O)N/N=C(/c2ccc(cn2)C(F)(F)F)\N SPB06964 CC1(CN(C1=O)N(C)c2cnn(c(=O)c2Cl)c3ccc(cc3Cl)Cl)C BTB08855 Cc1ccc(cc1)n2c(=O)c(c(cn2)N(C)N3CC(C3=O)(C)C)Cl BTB08856 Cc1ccc(nn1)NNC(=O)c2ccc(cc2)Cl BTB07299 Cc1ccnc(c1)NC(=O)c2ccc(cc2[N+](=O)[O-])Cl BTB07300 c1cc(ccc1C(=O)N2CCN(CC2)c3ccc(cn3)C#N)Cl SPB06780 c1cc(ccc1C(=O)ON=C(c2ccc(cc2)F)c3ccc(cc3)F)C(F)(F)F BTB07189 c1cc(ccc1C(=NOC(=O)c2ccc(cc2)Cl)c3ccc(cc3)F)F BTB07192 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-])C(F)(F)F BTB07108 CC(C)(C)NC(=O)N1CCN(CC1)c2nc3ccc(cc3s2)Cl SPB06875 Cn1c(=O)c(c(cn1)N(C)NC(=O)Nc2ccccc2)Cl BTB07351 CC(C)(C)c1cc(c(cc1OS(=O)(=O)c2ccc(cc2)Cl)C(C)(C)C)OS(=O)(=O)c3ccc(cc3)Cl BTB07352 CC(C)(C)c1cc(c(cc1OS(=O)(=O)c2ccc(cc2)C(F)(F)F)C(C)(C)C)OS(=O)(=O)c3ccc(cc3)C(F)(F)F BTB07353 CC(C)(C)c1ccc(cc1)COc2cccnc2N/C=N/O BTB08616 COc1ccc(c(c1C(=O)O)OC)Br BTB07593 Cc1nc(nc(n1)NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)C BTB07594 Cc1cc(nc(n1)NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)C BTB07596 Cc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Cl)OC)Cl BTB07644 Cn1ccnc1S(=O)(=O)CC(=O)OC BTB08458 c1ccc(cc1)c2c(=S)ssc2SCC(=O)Nc3cccc(c3)C(F)(F)F BTB08455 Cc1cccc2c1c(=O)oc(n2)c3cc(ccc3Oc4ccc(cc4)OC)[N+](=O)[O-] BTB08533 C/C(=N\NC(=O)c1ccc(cc1)C(C)(C)C)/c2ccccc2O BTB08537 CCn1c(cc(n1)c2cccs2)C(=O)Nc3ccccc3 SPB04238 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)C(F)(F)F BTB07109 c1cc2cccc(c2c(c1)SCC(=O)O)Cl BTB08836 C=CCN(c1ccccc1C(=O)NCC(=O)O)C(=O)c2ccc(cc2)Cl BTB08837 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nc3ccccc3o2 BTB14124 CCOC(=O)c1ccc(cc1)NC(=O)COc2ccccc2 BTB14125 Cc1ccc(nn1)N(C)/N=C/c2ccc(cc2Cl)Cl BTB07309 c1c(cnc(c1Br)N)Br BTB07310 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(nc2[N+](=O)[O-])C BTB07314 Cc1cc(cc(c1Cl)C)Oc2ccc(cn2)NS(=O)(=O)c3cccc4c3nccc4 BTB08528 CCOC(=O)c1cc(c(nc1c2ccccc2)SC)C#N SPB04232 CCn1c(cc(n1)c2cccs2)C(=O)N(C)C SPB04236 CCOC(=O)CSc1c(cc(c(n1)c2ccccc2)C(=O)OCC)C#N SPB04244 c1ccc(c(c1)N)N2C(=O)c3cccc4c3c(ccc4Cl)C2=O BTB11684 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC)Cl)[N+](=O)[O-] BTB07728 c1ccc(cc1)C(=O)n2c(c(cn2)Sc3ccc(cc3)Cl)c4ccc(cc4)Cl SPB04158 c1cc(ccc1c2c(cn(n2)C(=O)c3ccc(cc3)Cl)Sc4ccc(cc4)Cl)Cl SPB04159 CC(C)(C)c1ccc(cc1)Oc2cc3c(cc2[N+](=O)[O-])C(=O)NC3=O BTB08417 CCOC(=O)c1cc(c(nc1c2ccccc2)S)C#N SPB04229 c1ccc(cc1)/C=C/S(=O)(=O)c2ccc(cc2F)F BTB08481 c1cc(ccc1NC(=O)/C=N/O)Cl BTB08482 CN(C)/C=C(/C(=O)Nc1ccc(c(c1F)F)F)\Sc2nnc(s2)N BTB08484 CCn1c(cc(n1)c2cccs2)C(=O)NC(C)C SPB04237 CN(C)CCNc1cc(nc2c1cccc2)c3ccccc3.Br.Br BTB14087 COc1ccc(cc1OC)S(=O)(=O)N(CCCC#N)c2cc(ccc2C(=O)OC)Cl BTB08495 c1c(cc(cc1Cl)Cl)S(=O)(=O)Oc2cc(cnc2)Cl BTB07406 CN(C)/C=N/c1c(cccn1)OCc2ccc(c(c2)Cl)Cl BTB08580 CCOC(=O)c1cnc2c(ccc(c2c1Sc3cccc(c3)C(F)(F)F)F)F BTB08661 c1cc(sc1)C(=O)Oc2cc(cnc2)Cl BTB07418 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3cc(cnc3)Cl BTB07417 c1cc(c(nc1)Sc2ccc(cc2)Cl)C3=N/C(=C\c4ccc(cc4)Cl)/C(=O)O3 BTB08787 c1cnn(c1)c2cnn(c(=O)c2Cl)c3ccc(cc3Cl)Cl BTB08601 CCOC(=O)c1cnc2c(ccc(c2c1Sc3ccccc3)F)F BTB08660 Cc1c(c(n(n1)C(=O)Nc2cccc(c2)C(F)(F)F)C)Sc3ccc(cn3)C(F)(F)F SPB04367 COc1ccc(cc1)Oc2ccc(cn2)NC(=O)Cc3cccs3 BTB08686 c1cc(ccc1C2=NN(C(=O)CC2)c3ccc(cc3)[N+](=O)[O-])F BTB08570 c1ccc(cc1)c2cc(c3ccccc3n2)N BTB14090 c1ccc(c(c1)CCO)S(=O)c2ccccc2C(=O)O BTB11528 CNC(=O)c1ccccc1S(=O)c2ccc(cc2C(=O)O)Cl BTB11531 CNC(=O)c1ccccc1S(=O)c2ccc(cc2C(=O)O)[N+](=O)[O-] BTB11532 CN1CCN(CC1)c2cc(nc3c2cccc3)c4ccccc4.Br.Br BTB14089 c1cc(ccc1CSc2c(ccc(n2)/C=N/c3ccc(cc3Cl)Cl)C#N)Cl SPB04383 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Sc3nccn3C SPB04385 CN1C(=O)c2cccc3c2c(ccc3)S14c5ccccc5C(=O)O4 BTB11533 Cc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2C(=O)OC)Cl BTB08464 c1cc(ccc1CC#N)OCc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB07333 c1ccn(c1)c2cc(c(cc2Cl)NC(=O)NC(=O)c3c(cccc3Cl)Cl)Oc4ccc(cc4)Cl BTB07556 c1ccn(c1)c2cc(c(cc2Cl)NC(=O)c3ccc(cc3)C(F)(F)F)Cl BTB07561 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)Cc3cccs3 BTB08687 Cc1ccc(cc1)C(=O)n2c(c(c(n2)C)Sc3nccn3C)C SPB04391 Cc1ccc(cc1)/N=C/c2ccc(c(n2)SC)C#N SPB04402 CSc1c(ccc(n1)/C=N/c2ccc(cc2Cl)Cl)C#N SPB04401 CC(=O)Nc1ccc(cc1)C(F)(F)F BTB07343 Cn1c(=O)c(c(cn1)N(C)/N=C/c2ccc(cc2)Cl)Cl BTB07344 Cn1c(=O)c(c(cn1)N(C)NC(=O)c2ccc(cc2)Cl)Cl BTB07346 CC(C)(C)c1cc(c(cc1OS(=O)(=O)c2cc(cc(c2)Cl)Cl)C(C)(C)C)OS(=O)(=O)c3cc(cc(c3)Cl)Cl BTB07360 c1ccc(cc1)NC(=O)CSC2=NNC(S2)c3ccccn3 SPB06987 Cc1ccc(cc1)S(=O)(=O)N(CC=C)c2ccccc2C3=N/C(=C\c4ccccc4C)/C(=O)O3 BTB08800 c1cc2c(cc1Br)c(cc(=O)o2)O BTB14073 Cc1cccc(c1)/C=C\2/C(=O)OC(=N2)c3ccccc3N(CC=C)S(=O)(=O)c4ccc(cc4)Cl BTB08803 c1cc2/c(=N\N)/nc3n(c2nc1)ccs3 BTB08467 c1cc(cc(c1)Cl)NC(=O)Nc2ccc(nc2)Oc3cc(cnc3)Cl BTB07791 CCOC(=O)c1c(c(c(c(c1F)F)S(=O)(=O)C)F)F BTB08571 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2cc(c(c(c2)C(C)(C)C)O)C(C)(C)C BTB14040 c1cc(c(nc1)Sc2ccc(cc2)Cl)C3=N/C(=C\c4ccc(cc4)C(F)(F)F)/C(=O)O3 BTB08785 Cc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3cccnc3Sc4ccc(cc4)Cl BTB08786 CC(C)c1ccc(cc1)NC(=O)CSC2=NNC(S2)c3ccccn3 SPB06988 CCc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)CC BTB07610 CC(=O)OCc1ccccc1Sc2ccccc2C(=O)NCc3ccccc3 BTB11498 CCOC(=O)c1cnn(c1C)c2ccc(c(c2)Cl)Cl BTB08594 CC(=O)CC(=O)Nc1nccs1 BTB11736 c1cc(c(nc1)Sc2ccc(cc2)Cl)C(=O)NCC(=O)O BTB08780 c1cc(c(nc1)Oc2ccc(cc2)Cl)C3=N/C(=C\c4ccc(cc4)C(F)(F)F)/C(=O)O3 BTB08781 Cc1c(c(n(n1)C(=O)C2CC2)C)Sc3ncccn3 SPB04373 Cc1cc(n2cnnc2n1)OCC(=O)c3ccc(cc3)C(F)(F)F BTB08805 CCNC(=O)c1ccccc1Sc2ccccc2CO BTB11495 CNC(=O)c1ccccc1Sc2ccccc2[N+](=O)[O-] BTB11497 c1ccnc(c1)SCc2ccc(cc2)[N+](=O)[O-] BTB14092 Cn1cnnc1SCc2ccc(cc2)[N+](=O)[O-] BTB14093 COc1cc(c(cc1OC)Br)CCNC(=O)c2ccccc2Cl BTB14115 COc1cc(c(cc1OC)Br)CCNC(=O)c2ccc(cc2)Cl BTB14116 c1ccc(cc1)/C=C/C(=O)Nc2ccccc2 BTB11744 CCOC(=O)/C(=N/Nc1ccc(cc1Cl)Cl)/C(=O)CSc2ccc(cn2)C(F)(F)F SPB04426 Cc1ccc(cc1)n2c(c(cn2)C#N)N BTB07634 COc1ccc(c(c1NC(=O)NC(=O)c2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC)Cl BTB07636 c1ccc2c(c1)nc(o2)SCc3ccc(cc3)[N+](=O)[O-] BTB14098 CC(C)(C)c1cc(c(cc1OC(=O)c2ccc(cc2)Cl)C(C)(C)C)OC(=O)c3ccc(cc3)Cl BTB07347 c1ccc(cc1)c2cc(c3ccccc3n2)N4CCOCC4 BTB14085 CN(C)CCNc1cc(nc2c1cccc2)c3ccccc3 BTB14086 C/C=C/CC(=O)NCC(=O)N BTB14113 COc1cc(c(cc1OC)Br)CCNC(=O)c2cccc(c2)Cl BTB14114 CN(C)c1ccc2c3c1cccc3C(=O)N(C2=O)c4[nH]c5ccccc5n4 BTB11699 CC(C)(C)OC(=O)C(C)(C)S(=O)(=O)c1ccc(cc1)Cl BTB08903 CNC(=O)c1ccccc1S(=O)c2cccc3c2c(ccc3)C(=O)OC BTB11513 Cn1c(=O)c(c(cn1)S(=O)(=O)Cc2ccccc2)Cl BTB07373 Cc1ccc(cc1)Sc2c(cccn2)C3=N/C(=C\N(C)C)/C(=O)O3 BTB08823 Cc1cc2c(cc1C)nc(cn2)c3ccn(c3)S(=O)(=O)c4ccc(cc4)Cl BTB07252 CN(C)/C=C\1/C(=O)OC(=N1)c2cccnc2Oc3ccc(cc3)Cl BTB08824 CC(=O)Nc1ccc(cc1Br)C(F)(F)F BTB07356 Cc1c(cnn1c2ccccc2)C(=O)O CC15501 c1cc(ncc1N/C=N/O)Oc2cc(cnc2)Cl BTB07792 CCOC(=O)CC(=O)CSc1nnc(s1)NC(=O)c2ccc(cc2)Cl BTB07804 CC(C)(C)c1cc(c(cc1Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C(C)(C)C)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB07359 CC(C)(C)c1cc(cc(c1)C(=O)Oc2cc(cnc2)Cl)C(=O)Oc3cc(cnc3)Cl BTB08635 Cc1ccc(cc1)Sc2c(cccn2)C(=O)NCC(=O)O BTB08791 C=CCN(c1ccccc1C2=N/C(=C\c3cccc(c3)Cl)/C(=O)O2)S(=O)(=O)c4ccc(cc4)Cl BTB08793 CN(c1cnn(c(=O)c1Cl)c2ccc(c(c2)Cl)F)NC(=O)c3ccc(cc3)C(F)(F)F BTB08818 Cc1ccc(cc1)S(=O)(=O)n2c(c(c(n2)C)Sc3nccn3C)C SPB04392 CC(C)(C)C(=O)Nc1ccn(c(=O)n1)[C@H]2C[C@@H]([C@H](O2)COC(=O)C(C)(C)C)O BTB14106 CC(C)(C)C(=O)OC[C@@H]1[C@H](C[C@@H](O1)n2cnc3c2ncnc3N)OC(=O)C(C)(C)C BTB14108 COc1ccc(c(c1)OC)NC(=O)C(c2ccccc2)C(=O)Nc3ccc(cc3OC)OC BTB11814 COC(=O)c1ccccc1Sc2cccc3c2c(ccc3)C#N BTB11494 CC(C)(C)c1cc(cc(c1)C(=O)NCc2cccs2)C(=O)NCc3cccs3 BTB08643 CSc1c(c(nc(n1)c2ccccc2)Sc3ccccc3)C#N BTB08917 Cn1c(=O)c(c(cn1)N(C)NS(=O)(=O)c2ccc(cc2)C(F)(F)F)Cl BTB07369 Cc1cc(n(n1)c2ccccc2)OC(=O)c3ccccc3 BTB07659 COc1c(cc(c(c1C(=O)N)OC)Br)[N+](=O)[O-] BTB07683 c1cc(ccc1C(=O)NC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl SPB06940 Cc1ccc(cc1)C(=O)NC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl SPB06941 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC)Cl)Cl BTB07685 COc1c(cc(c(c1C(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl)OC)Cl)Cl BTB07687 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3cc(nn3c4ccccc4)C(F)(F)F BTB07629 Cc1c(nn(n1)c2ccccc2)C(=O)c3c(nn(c3O)c4ccccc4)C(C)(C)C BTB07630 C1CC1C2=NN3C(=N)CC(=O)N=C3S2 BTB08810 CCOC(=O)CNC(=O)c1ccccc1N(CC=C)S(=O)(=O)c2ccc(cc2)C BTB08814 COC(=O)C(=C(SC)SC)C#N BTB08843 c1c(cncc1Cl)Oc2cc(c(cc2[N+](=O)[O-])Br)Oc3cc(cnc3)Cl BTB08840 Cn1c(=O)c(c(cn1)N(C)NC(=O)Nc2ccc(cc2)Cl)Cl BTB07378 CN(C)/C=C\1/C(=O)OC(=N1)c2cccnc2SC BTB08820 Cc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2)Cl BTB11783 CC(C)(C)c1cc(cc(c1)C(=O)Oc2cccnc2)C(=O)Oc3cccnc3 BTB08637 COc1c(cc(c(c1C(=O)N)OC)Cl)Cl BTB07674 Cc1cc(c(c(c1)C)NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC)C BTB07679 c1ccnc(c1)S(=O)(=O)CCOC(=O)c2cccc(c2)Cl BTB08941 CSc1c(c(nc(n1)c2ccccc2)SC)C#N BTB08942 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)Cl)Cl BTB07680 Cc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC)C BTB07681 c1cn(c(=O)nc1N)[C@H]2CC[C@H](O2)CO BTB14103 c1ccc(cc1)/C=C/CSc2ccccn2 BTB14134 CCOC(=O)Cc1csc(n1)NC(=O)CSc2nccn2C BTB14130 c1cc(c(cc1C(=O)CSC#N)F)F BTB08658 CC(C)(C)c1cc(cc(c1)C(=O)Nc2cccnc2)C(=O)Nc3cccnc3 BTB08632 CC(=O)Oc1ccc2c(c1)oc(c(c2=O)Oc3ccc(cc3)Cl)C(F)(F)F BTB11798 CCCCCCCCCCCCCCNC(=O)CSc1ccccn1 BTB14136 CN(C)/C=N/c1ccc(nc1)Oc2cc(cnc2)Cl BTB07673 Cc1ccc(cc1)C(=O)NN(C)c2cnn(c(=O)c2Cl)c3ccc(c(c3)Cl)F BTB08817 COc1ccc(cc1)Oc2ccc(cn2)NS(=O)(=O)c3cccc4c3nccc4 BTB08529 C/C(=N\NC(=O)c1ccc(cc1)Cl)/c2ccccc2O BTB08531 Cc1ccc(cc1)Oc2c(cccn2)C3=N/C(=C\N(C)C)/C(=O)O3 BTB08825 C/C(=N\NC(=O)c1ccc(cc1)C(F)(F)F)/c2ccccc2O BTB08532 c1ccc(cc1)/C(=N/Nc2ccc(cc2)[N+](=O)[O-])/CCC(=O)O BTB08536 Cc1c(c2cc(ccc2n1C(=O)c3ccc(cc3)Cl)OC)CC(=O)OCC(=O)OCc4ccccc4 BTB11728 CC(=O)Nc1ccc(nc1)Oc2cc(cnc2)Cl BTB07789 CCn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br BTB11853 c1ccc(cc1)Cn2c3ccc(cc3c4c2ccc(c4)Cl)Cl BTB11854 Cc1c(c(no1)C(=O)NNS(=O)(=O)c2ccc(cc2)Cl)c3csc(n3)COc4ccccc4 SPB04416 Cc1c(c(nc(n1)SCc2ccc(cc2)C(F)(F)F)O)Oc3cccc(c3)C(F)(F)F SPB04420 c1cc2c(cc1Br)OCCOCCOCCOCCO2 BTB11766 Cc1c(c(c(=O)n(c1c2ccccc2)c3ccccc3)c4ccccc4)O BTB11829 Cc1ccc(cc1)n2c(=O)c(c(cn2)N(C)/N=C/c3ncc(n3C)[N+](=O)[O-])Cl BTB08857 Cc1ccc(cc1)n2c(=O)c(c(cn2)N(C)n3cccc3)Cl BTB08859 COC(c1ccc2c(c(sc2n1)C(=O)c3ccc(cc3)Cl)N)OC SPB04338 c1ccc2c(c1)c(=O)n3c(n2)CCC(=O)N3 BTB11750 CCOC(=O)/C(=C/c1ccccc1)/C#N BTB11751 c1cc2c(cc1[N+](=O)[O-])OCCOCCOCCO2 BTB11764 Cc1c(c(n(n1)C(=O)C2CC2)C)Sc3ccc(cn3)C(F)(F)F SPB04346 Cc1ccc(cc1)C(=O)n2c(c(c(n2)C)Sc3ccc(cn3)C(F)(F)F)C SPB04347 c1ccc(cc1)Cn2c3ccc(cc3c4c2ccc(c4)Br)Br BTB11855 CC(C)(C)c1cc(cc(c1)C(=O)Nc2ccsc2C(=O)OC)C(=O)Nc3ccsc3C(=O)OC BTB08634 c1cc(cc(c1)Cl)C(=O)Nc2ccc(nc2)Oc3cc(cnc3)Cl BTB07672 CC(=O)NC(=O)c1cccc2c1c(ccc2)I BTB11552 Cc1cccc(c1)NC(=O)C(C(F)(F)F)C(F)(F)F BTB14192 COC(=O)/C(=C(\NC(=O)c1ccccc1)/SC)/C#N BTB08844 Cc1ccc(cc1)C(=O)c2c(c3ccc(nc3s2)C(OC)OC)N SPB04339 c1cc(ccc1C(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl)Cl SPB06866 CC(=O)N1CCN(CC1)c2nc3ccc(cc3s2)Cl SPB06868 Cc1ccc(cc1)C(=O)CSc2c(ccc(n2)C(OC)OC)C#N SPB04357 CCCCCCCCCCCCCCOC(=O)C(C)O BTB14123 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2F)Cl)F BTB11792 c1cc(ccc1/C(=N/Nc2ccc(cc2)[N+](=O)[O-])/CCC(=O)O)F BTB08564 c1cc(ccc1C(F)(F)F)S(=O)(=O)Nc2ccc(nc2)Oc3ccc(cc3)F BTB07430 Cc1ccc(cc1)S(=O)(=O)N2CCN(CCN(CCN(CC2)S(=O)(=O)c3ccc(cc3)C)S(=O)(=O)c4ccc(cc4)C)S(=O)(=O)c5ccc(cc5)C BTB14158 CN(c1cnn(c(=O)c1Cl)c2cc(cc(c2)Cl)Cl)NC(=O)c3ccc(s3)Cl BTB08887 Cn1cnnc1SCC(=O)Nc2nc(cs2)CC(=O)O BTB14132 CCCCCCCCCCCCCCNC(=O)CSc1nncn1C BTB14135 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)Cl)Cl BTB11782 c1cc(ccc1S(=O)(=O)Oc2cc(cnc2)Cl)Cl BTB07407 COC(c1ccc(c(n1)SCC(=O)Nc2ccc(cc2)C(F)(F)F)C#N)OC SPB04358 c1ccc(c(c1)OC(F)(F)F)S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl SPB06871 CC(C)(C)c1cc(c(cc1OC(=O)c2ccc(cc2)C(F)(F)F)C(C)(C)C)OC(=O)c3ccc(cc3)C(F)(F)F BTB07348 CC(C)(C)c1ccc(cc1)C(=O)Oc2cc(c(cc2C(C)(C)C)OC(=O)c3ccc(cc3)C(C)(C)C)C(C)(C)C BTB07349 C/C(=N\NC(=O)/C=C/C(=O)O)/c1ccc(cc1)[N+](=O)[O-] BTB11748 CCOC(=O)C(=CNc1ccc(nc1)Oc2cc(cnc2)Cl)C(=O)OCC BTB07787 CC(C)n1c2ccccc2c3c1cccc3 BTB11846 Cc1cccc(c1)COc2cccnc2N BTB08566 Cc1ccc(cc1)S(=O)(=O)N(CCCC#N)c2cc(ccc2C(=O)OC)Cl BTB08567 c1ccn(c1)c2c3cccnc3ccc2[N+](=O)[O-] BTB07795 c1cc2c(cc1[N+](=O)[O-])OCCOCCOCCOCCO2 BTB11763 c1cc(ccc1c2ccc(=O)n(n2)c3ccc(cc3)[N+](=O)[O-])F BTB08574 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NS(=O)(=O)c3ccc(cc3)C)[N+](=O)[O-] BTB08583 Cc1ccc(cc1)C(=O)/C=C/Sc2ccc(cc2)Cl BTB11770 CN(C)/C=N/c1ncccn1 BTB08921 Cc1ccc(cc1)C(=O)/C=C/Sc2ccc(cc2)Br BTB11771 CC(C)(C)c1cc(c(cc1OC(=O)c2ccc(cc2Cl)Cl)C(C)(C)C)OC(=O)c3ccc(cc3Cl)Cl BTB07350 CC(C)SCC(=O)NCC(=O)OC BTB14122 Cc1ccc(nn1)N(C)NC(=O)Nc2ccc(cc2)Cl BTB07305 COc1ccc(cc1OC)S(=O)(=O)Nc2cc(ccc2C(=O)OC)Cl BTB08461 CC(C)CCn1c2ccccc2c3c1cccc3 BTB11849 C1[C@@H]([C@H]1C(=O)NN)C(=O)NN BTB14035 c1cc(ccc1SCc2cc(=O)[nH]c(=O)[nH]2)Cl BTB08913 Cc1ccc(cc1)CSc2cnc(nc2C)C SPB04407 CNC(=O)c1cccc2c1c(ccc2)S(=O)c3ccccc3 BTB11525 Cc1nc(c(c(n1)Sc2ccccc2)C#N)SC BTB08923 c1cc(cc(c1)Cl)C(=O)OCCS(=O)(=O)c2ccc(cn2)[N+](=O)[O-] BTB08915 Cc1nc(c(c(n1)Sc2ccccn2)C#N)SC BTB08916 c1cc(ccc1C(=O)/C=C/Sc2ccc(cc2)Br)Cl BTB11772 Cn1c(=O)c(c(cn1)N(C)NC(=O)c2cccs2)Cl BTB07345 CC(C)(C)OC(=O)C(C)(C)Sc1ccc(cc1)Cl BTB08901 COC(=O)c1ccc(cc1NS(=O)(=O)c2cccc(c2)C(F)(F)F)Cl BTB08463 CC(=O)c1ccccc1C(=O)c2ccc(cc2)C(F)(F)F BTB08540 COC(=O)c1ccc(cc1N(CCCC#N)S(=O)(=O)c2ccc(cc2)Cl)Cl BTB08541 CC(=O)c1ccccc1C(=O)c2ccc(cc2)C(C)(C)C BTB08545 c1ccc(cc1)C2=NN(C(=O)CC2)c3ccc(cc3)[N+](=O)[O-] BTB08546 CCOC(=O)c1c(c(c(=N)n(n1)c2ccc(cc2)C)C#N)C BTB08885 c1cc2cccc(c2c(c1)CO)S(=O)c3cccc4c3c(ccc4)C(=O)O BTB11520 COc1ccc(c(c1C(=O)NC(=O)Nc2c(c(c(c(c2F)F)F)F)F)OC)[N+](=O)[O-] BTB07590 Cc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3cccnc3SC BTB08777 c1ccc-2c(c1)Cc3c2ccc(c3)C(=O)c4ccccc4Br BTB11872 c1ccc(cc1)Nc2c(cc(cn2)[N+](=O)[O-])[N+](=O)[O-] BTB11873 CCc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)CC BTB07582 COc1ccc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)[N+](=O)[O-] BTB07583 Cc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)C BTB07584 c1cc(cc(c1)Cl)C(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08623 CCOC(=O)c1c(c(c(=N)n(n1)c2ccc(cc2)Cl)C#N)C BTB08899 Cn1c2ccccc2nc1N3C(=O)c4cccc5c4c(ccc5)C3=O BTB11695 c1cc(ccc1[N+](=O)[O-])OCC#N SPB04268 Cc1cc(no1)c2nc(on2)C(C)(C)C SPB04274 Cc1c2c(onc2c(=O)n(n1)c3cccc(c3)C(F)(F)F)C SPB04272 CC(C)(C(=O)OC)S(=O)(=O)c1ccc(cn1)C(F)(F)F BTB09015 c1cc(ccc1C(F)(F)F)S(=O)(=O)Oc2cc(cnc2)Cl BTB07404 c1cc(c(cc1Cl)Cl)n2c(c(cn2)C#N)N BTB07761 CC(=O)Nc1nnc(s1)SCC#N BTB07769 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)Cl)Br BTB11786 CC(C)NC(=O)/C(=N/C(C)C)/C(F)(F)F BTB14222 c1cc(c(nc1)Oc2cc(cnc2)Cl)[N+](=O)[O-] BTB07419 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3cccc(c3)C(F)(F)F BTB07770 COC(=N)NC(=S)Nc1ccccc1 SPB06994 c1ccc(c(c1)C(=O)O)SCC(=O)O BTB07338 Cc1cccc(c1C)Oc2ccc(cn2)/N=C/c3ncc(n3C)[N+](=O)[O-] BTB07425 Cn1c(nnc1SCC(=O)Nc2ccccc2)SCC(=O)Nc3ccccc3 BTB08559 Cc1c2c(onc2c(=O)[nH]n1)/C=C/c3ccc(cc3)C(F)(F)F BTB08999 Cc1c(c(c(=O)n(n1)C)N)c2cc([nH]n2)c3ccsc3 BTB09005 CNC(=O)c1ccccc1S(=O)c2cccc3c2c(ccc3)CO BTB11517 c1ccc(cc1)C(=O)Nc2nnc(s2)SCC#N BTB07763 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cn1)C BTB14236 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1F)F BTB14239 c1cc(ncc1C(F)(F)F)S(=O)(=O)CCNC=C(C#N)C#N BTB07998 CC(C)OC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccccc1C(=O)O BTB14242 CCC(=O)N1C2CC(C1(C(F)(F)F)C(F)(F)F)C=C2 BTB14245 Cc1c(c(n(n1)c2ccccc2)O)C(=O)c3cccnc3SC BTB07773 C=CCN(c1ccccc1C2=N/C(=C\c3ccccc3Cl)/C(=O)O2)S(=O)(=O)c4ccc(cc4)Cl BTB08794 Cc1ccc(cc1)S(=O)(=O)n2c(c(c(n2)C)Sc3ncccn3)C SPB04376 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccccc1F BTB14233 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC)Br)Cl BTB07751 CCCN(CCC)S(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)N(CCC)CCC BTB11875 CCOC(=O)C1=C(CC(=C(C1)N)C(=O)OCC)N BTB09095 c1cc(sc1c2csc(n2)N)Br BTB09097 Cc1c(c(no1)C(=O)NNS(=O)(=O)c2ccc(cc2)Cl)c3csc(n3)COc4ccc(cc4)Cl SPB04417 c1ccc(cc1)C(=O)OCCSc2ccccn2 BTB08930 c1ccc(cc1)C2CC(=O)c3c2cccc3 BTB14149 Cc1c(c(n(n1)S(=O)(=O)c2ccc(cc2)Cl)C)Sc3nccn3C SPB04393 c1cc(ncc1Cl)SCCO BTB08976 CN(C)c1c(c(nc(n1)c2ccccc2)c3ccccc3)C#N BTB08980 Cc1ccc(cc1)S(=O)(=O)NC(C(=O)OC)(C(F)(F)F)O BTB14202 CCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[NH2+][O-] BTB11881 CCCCn1c2ccccc2c3c1cccc3 BTB11847 CCOC(=O)CC(=O)CSc1c(c(c(c(n1)C)C)C)C#N SPB04411 c1ccc(cc1)Cn2c3ccccc3c4c2cccc4 BTB11848 CCOC(=O)/C(=N/Nc1ccc(cc1Cl)Cl)/C(=O)CSc2c(c(c(c(n2)C)C)C)C#N SPB04425 CCOC(=O)/C(=N/Nc1ccccc1)/C(=O)CSc2ccc(cn2)C(F)(F)F SPB04427 c1ccc(cc1)NNC(=S)SCC(=O)c2ccc(cc2)Cl BTB07847 Cc1ccc(cc1)S(=O)(=O)Oc2cc(cnc2)Cl BTB07405 CCOC(CN(c1ccc(cc1)F)C(=O)c2ccc(cc2)C(F)(F)F)OCC BTB07873 CC(=O)O.CN1C(=O)c2cccc3c2c(ccc3)[S+]1c4cccc5c4c(ccc5)C(=O)[O-] BTB11547 Cc1c(nn(n1)c2ccccc2)C(=O)Oc3cc(nn3c4ccccc4)C(=O)OC BTB07774 CSc1nnc(n1CCNC(=O)c2cccc(c2)Cl)SC BTB07617 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cccc2F)F)OC)Br BTB07627 CCn1c2ccc(cc2c3c1ccc(c3)Br)Br BTB11852 Cc1cc(ccc1Cl)c2csc(=S)n2Nc3ccccc3 BTB07844 CNC(=O)c1cccc2c1c(ccc2)S(=O)c3ccccc3CO BTB11519 Cc1cc(cc(c1NC(=O)NC(=O)c2c(cccc2OC)OC)C)Br BTB07452 c1ccc2c(c1)cc(s2)C(=O)Oc3cc(cnc3)Cl BTB07408 c1ccc(cc1)NC(=S)Nc2ccccc2 BTB07414 c1ccc(cc1)Sc2c(cccn2)C(=O)O BTB08722 c1cc(c(c(c1)Cl)Cl)SCC(=O)O BTB08713 CCOC(=O)c1cnn(c1C)c2ccc(cc2)Cc3ccc(cc3)n4c(c(cn4)C(=O)OCC)C BTB08717 COc1ccc(cc1)Oc2ccc(cc2C(=O)NCC(=O)OC)[N+](=O)[O-] BTB08720 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Sc3ncccn3 SPB04365 Cc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccccc3N(CC=C)S(=O)(=O)c4ccc(cc4)C BTB08801 CN(C)/C=C\1/C(=O)OC(=N1)c2cccnc2Sc3ccc(cc3)Cl BTB08822 CNC(=O)c1ccccc1S(=O)c2cccc3c2c(ccc3)C(=O)NC BTB11522 COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccc(cc3)[N+](=O)[O-])Cl BTB07508 CCOC(=O)C(C(F)(F)F)(NC(=O)C)NS(=O)(=O)c1ccccc1 BTB14176 CCOC(=O)c1cnc2c(c1O)c(no2)C BTB08703 Cc1cc(c2ccccc2n1)N/C=N/O BTB09126 CCOC(=O)CNC(=O)c1ccccc1N(CC=C)C(=O)c2ccccc2Cl BTB08761 c1ccc(cc1)Sc2cccc3c2c(ccc3)C#N BTB11507 CNC(=O)c1cc(ccc1Sc2ccccc2)[N+](=O)[O-] BTB11508 CCOC(=O)c1ccccc1Sc2ccccc2C(=O)OC BTB11509 CC1=NN(C(=O)C1CCO)c2ccc(cc2)Cl BTB07498 CCOC(=O)CNC(=O)c1cc(ccc1Oc2ccc(cc2)OC)[N+](=O)[O-] BTB08826 Cn1c(cnc1/C=C(\C#N)/C(=O)Nc2ccc(cc2)F)[N+](=O)[O-] BTB07385 COC(c1ccc(c(n1)SCC(=O)c2ccc(cc2)C#N)C#N)OC SPB04400 c1ccc(c(c1)N2C(=O)c3cccc4c3c(ccc4)C2=O)O BTB11688 c1ccc2c(c1)ncc(n2)c3ccc(s3)Br BTB08704 c1c(cc(c(c1Cl)SCC(=O)O)Cl)Cl BTB08711 c1cc-2c(cc1S(=O)(=O)N3CCCCCC3)Cc4c2ccc(c4)S(=O)(=O)N5CCCCCC5 BTB11902 Cc1cccc(c1)S(=O)(=O)N(CC=C)c2ccccc2C(=O)NCC(=O)O BTB08767 c1ccc(cc1)C(=O)Nc2nnc(s2)C(F)(F)F BTB09129 CNC(=O)c1cccc2c1c(ccc2)[S+]3c4ccccc4CO3.[Cl-] BTB11543 CCNC(=O)c1ccccc1Sc2ccccc2COC(=O)C BTB11499 Cc1cccc(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)C BTB07481 Cn1c(cnc1/C=N/c2ccc(nc2)Oc3ccc(cc3)OC)[N+](=O)[O-] BTB07423 CC(=O)OCCS(=O)(=O)c1ccc(cn1)C(F)(F)F BTB08647 c1ccc2c(c1)c3ccccc3c4c2nc(nn4)N5CCOCC5 BTB11719 CCOC(=O)/C(=C/Nc1nnc(s1)SCC#N)/C#N BTB07781 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)OCC#C BTB14246 CCCCCCCOCC(Cn1c2ccccc2c3c1cccc3)O BTB11858 CC(C)CCOCC(Cn1c2ccccc2c3c1cccc3)O BTB11859 CCCN(CCC)S(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)N(CCC)CCC BTB11903 CCN(CC)S(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)N(CC)CC BTB11904 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)/N=C/c3cc(cc(c3O)Cl)Cl BTB07893 CN1C(=O)c2cccc3c2c(ccc3)[S+]1c4ccccc4C(=O)O.[Cl-] BTB11545 Cc1nc(c(c(n1)SC)C#N)Nc2ccccc2 BTB08947 c1ccc(cc1)OS(=O)(=O)c2ccc-3c(c2)C(=O)c4c3ccc(c4)S(=O)(=O)Oc5ccccc5 BTB11876 CCCN(CCC)C(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[NH2+][O-] BTB11880 CC(=O)NC(=O)CCSc1ccccc1C(=O)NC(=O)C BTB11505 Cn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br BTB11861 C(#N)c1c(c(c(c(c1Cl)Cl)Cl)Cl)C#N BTB14154 c1cc(sc1)C(=O)/C(=N/Nc2ccc(cc2Cl)Cl)/C(=O)C(F)(F)F SPB04437 c1ccc(cc1)N/N=C(/C(=O)c2cccs2)\C(=O)C(F)(F)F SPB04440 Cc1ccc(cc1)Sc2c(cccn2)C(=O)O BTB08723 CCOC(=O)CNC(=O)c1ccc(cc1)Cl BTB08724 c1cc(c(cc1F)Cl)SCC(=O)O BTB08730 c1ccn(c1)c2ccc(nc2)Oc3cc(cnc3)Cl BTB07816 COC(=O)CNC(=O)c1cccnc1Sc2ccccc2 BTB08744 c1cc2c(cc1Br)c3cc(ccc3n2CC(CO)O)Br BTB11835 COc1ccc(c(c1)Sc2c(cccn2)C(=O)O)OC BTB08732 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)O BTB08733 COc1ccc(c(c1C(=O)OC)OC)N/C=N/O BTB07819 COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccccc3)Cl BTB07507 c1ccc(c(c1)CO)S(=O)c2cccc3c2c(ccc3)C(=O)O BTB11518 Cn1c(cnc1/C=C(\C#N)/C(=O)Nc2ccc(cc2OC)OC)[N+](=O)[O-] BTB07386 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)C(=O)O BTB08827 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2Cl)Cl)Br BTB11789 CC(C)(C)c1cc(c(c(c1)Br)OS(=O)(=O)c2ccc(cc2)Cl)Cl BTB07516 CC(C)(C)c1cc(c(c(c1)Br)OS(=O)(=O)c2cc(ccc2OC)Br)Cl BTB07517 CCOC(=O)/C(=C/Nc1ccc(c(c1OC)C(=O)OC)OC)/C#N BTB07809 CN(C)S(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)N(C)C BTB11905 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2cc(cc(c2)C(C)(C)C)C(=O)NNC(=O)c3ccc(cc3)C(C)(C)C BTB08642 C(C#N)Sc1nnc(s1)N BTB07735 CCc1c(c(c(=O)n(c1c2ccccc2)c3ccccc3)c4ccccc4)O BTB11803 c1ccc(cc1)NC(=O)C(C(F)(F)F)C(F)(F)F BTB14190 Cn1c(cnc1/C=N/N(C)c2cnn(c(=O)c2Cl)c3ccccc3)[N+](=O)[O-] BTB08861 CCOC(=O)C(=CNc1ccc(cn1)C(=O)O)C(=O)OCC BTB08863 COC(=O)CNC(=O)c1cccnc1Sc2ccc(cc2)Cl BTB08741 Cc1ccc(cc1)Oc2c(cccn2)C(=O)NCC(=O)OC BTB08743 CCOC(=O)CNC(=O)c1cccnc1SC BTB08725 COC(=O)CNC(=O)c1cccnc1Oc2ccccc2 BTB08726 CCOC(=O)CNC(=O)c1cccnc1Oc2ccccc2 BTB08727 Cc1cnc(c(n1)C)N BTB07911 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2ccc(c(c2F)F)F)Cl BTB07912 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2ccc(c(c2F)F)F)[N+](=O)[O-] BTB07914 Cc1nc(c(c(n1)SC)C#N)Nc2ccc(cc2Cl)Cl BTB08948 CC(=O)NNC(=O)c1ccccn1 BTB14006 Cc1ccccc1NC(=O)C(C(F)(F)F)C(F)(F)F BTB14191 CSc1c(c(=O)[nH]c(n1)c2ccccc2)C#N BTB08867 CN(C)/C=C(\C#N)/Sc1nnc(s1)n2cccc2 BTB07783 c1ccc(cc1)Oc2c(cccn2)C(=O)NCC(=O)O BTB08728 c1ccc(cc1)NNC(=S)SCC(=O)c2cccc(c2)[N+](=O)[O-] BTB07833 c1ccc(cc1)NNC(=S)SCC(=O)c2ccc(c(c2)Cl)Cl BTB07834 CN(C)/C=N/c1c(cnn1c2ccccc2)C#N BTB07492 CN(C)/C=N/c1c(cnn1c2ccc(c(c2)Cl)F)C#N BTB07493 CN(C)/C=N/c1c(cnn1c2ccc(cc2)[N+](=O)[O-])C#N BTB07494 c1cc(cc(c1)S(=O)(=O)OC2=C(CCN(c3c2ccc(c3)Cl)S(=O)(=O)c4ccc(cc4)Cl)C#N)C(F)(F)F BTB08612 c1cc(cc(c1)Cl)/C=N/c2ccc(nc2)Oc3cc(cnc3)Cl BTB07817 Cc1[nH]c(=O)c(c(n1)SC)C#N BTB08869 CC(=O)O.CNC(=O)c1cccc2c1c(ccc2)S(=O)c3cccc4c3c(ccc4)C(=O)O BTB11514 COC(=O)c1ccccc1S(=O)c2cccc3c2c(ccc3)CO BTB11516 c1ccc(c(c1)NC(=O)CC(=O)Nc2ccccc2OC(F)(F)F)OC(F)(F)F BTB11813 c1ccc2c(c1)c3ccccc3n2CN4CCCCC4 BTB11844 c1cc(c(cc1C(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl)Cl BTB08620 CC(=O)N[C@@H]1[C@H]([C@@H]([C@H](O[C@@H]1OCc2ccccc2)CO)O)O BTB11574 Cc1cn(c(=O)[nH]c1=O)[C@H]2C[C@@H]([C@H](O2)COC(=O)C(C)(C)C)OS(=O)(=O)C BTB11575 c1ccnc(c1)C2NN=C(S2)SCC(=O)c3ccc(cc3)Cl SPB06984 c1ccnc(c1)C2NN=C(S2)SCC(=O)c3cccc(c3)F SPB06985 CC(C)(C)C(=O)CSC1=NNC(S1)c2ccccn2 SPB06986 CNC(=O)Nc1ccc(nc1)Oc2cc(cnc2)Cl BTB07814 c1ccnc(c1)C2NN=C(S2)SCC(=O)Nc3ccc(cc3)C(F)(F)F SPB06989 Cn1cc(c(n1)C2NN=C(S2)SC)Cl SPB06992 CC(=O)C(=CNc1ccc(nc1)Oc2cc(cnc2)Cl)C(=O)C BTB07818 CN(c1cnn(c(=O)c1Cl)c2ccccc2)n3cccc3 BTB08858 c1cc(ccc1C(=O)/C=C/Nc2ccc(cc2)Cl)F BTB11784 CC(C)(C)OC(=O)C(C)(C)S(=O)(=O)c1ccc(cn1)C(F)(F)F BTB08906 Cc1ccc(cc1)SCc2cc(=O)[nH]c(=O)[nH]2 BTB08909 CCOC(=O)C(=CNc1ccc(c(c1OC)C(=O)OC)OC)C(=O)OCC BTB07807 COc1ccc(c(c1C(=O)OC)OC)NC=C(C#N)C#N BTB07808 Cc1cc2c(cc1Cl)c(=O)cco2 BTB14161 c1cc(sc1)C(=N)NC(=O)c2ccc(cc2)Cl SPB06999 c1ccc(c(c1)C(=O)N)Sc2ccccc2C(=O)N BTB11492 c1ccc(c(c1)C(=O)O)Sc2ccccc2[N+](=O)[O-] BTB11496 c1cc(ncc1NC(=O)/C=C/C(=O)O)Oc2cc(cnc2)Cl BTB07815 c1cc(cc(c1)Cl)C(=O)OCCS(=O)(=O)c2c(cccn2)C#N BTB08960 Cn1c(cnc1/C=C(\C#N)/C(=O)Nc2ccccc2)[N+](=O)[O-] BTB07383 c1ccc(cc1)c2[nH]c3c(c(n(n3)c4ccccc4)N)c(=O)n2 BTB08970 Cn1c(cc(=O)n(c1=O)C)N2CCOCC2 BTB08972 COc1c(cc(c(c1C(=O)N)OC)Br)Cl BTB07739 c1ccn(c1)c2nnc(s2)SCC#N BTB07764 CCOC(=O)c1cnn(c1C)c2ccccc2 BTB08591 Cc1c2c(onc2c(=O)n(n1)C)C SPB04371 c1cc(cc(c1)Cl)C(=O)OCCSc2c(cccn2)C#N BTB08954 CCOC(=O)CNC(=O)c1ccccc1NCC=C BTB08756 CCOC(=O)CNC(=O)c1ccccc1N(CC=C)C(=O)c2cccc(c2)C BTB08758 CC1=NC(=C(/C(=C(\C#N)/C(=O)OC)/N1)C#N)SC BTB08965 c1cc(cc(c1)Cl)C(=O)OCCS(=O)(=O)c2c(cccn2)C(F)(F)F BTB08962 CC1=NC(=C(C(=C(C#N)C#N)N1)C#N)SC BTB08968 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NC(=O)NC(=O)c3c(cccc3Cl)Cl BTB07897 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NS(=O)(=O)c3ccc(cc3)C BTB07900 Cn1c(=O)c(c(cn1)N(C)NS(=O)(=O)c2ccc(cc2)Cl)Cl BTB07368 c1cc(ccc1Oc2ncc(c(n2)N)C#N)Cl BTB08600 CCOC(=O)C1=C(N(C(=O)NC1c2ccccc2)C)C BTB11822 CCOC(Cn1c2ccccc2c3c1cccc3)OCC BTB11839 c1cc2c(cc1Br)c3cc(cc(c3[nH]2)Br)Br BTB11841 CSc1nc2c(=S)[nH]c(=S)[nH]c2s1 BTB14034 c1ccc2c(c1)c3ccccc3n2CC(CO)O BTB11842 CCOC(=O)CNC(=O)c1ccccc1N(CC=C)C(=O)c2cccc(c2)Cl BTB08759 Cc1cc(c2ccccc2n1)/N=C\N(C)C BTB09124 CCN(c1ccccc1)C(=O)C(Cc2ccccc2)C(=O)N(CC)c3ccccc3 BTB11811 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NS(=O)(=O)c3ccc(cc3)Cl BTB07901 CCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB11882 Cn1c(nnc1SCc2c(cccc2Cl)F)S BTB08609 c1cc(cc(c1)Cl)NC(=O)CC(=O)Nc2cccc(c2)Cl BTB11826 Cc1ccc(cc1)S(=O)(=O)OC2=C(CCN(c3c2ccc(c3)Cl)S(=O)(=O)c4ccc(cc4)Cl)C#N BTB08613 CCOC(=O)c1cc(on1)C(=O)C SPB04430 c1ccc2c(c1)nc(s2)S/C=C/C(=O)c3ccc(cc3)Cl BTB11781 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)SCC(=O)Nc3ccc(cc3)Cl BTB08560 Cc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)Cl BTB07585 c1cc(c(nc1)N)OCc2ccc(c(c2)Cl)Cl BTB08561 CC(C)c1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)C(C)C BTB07586 Cc1cc(c(c(c1)C)NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)C BTB07613 c1cc(cc(c1)C(F)(F)F)C(=O)OC2=C(CCN(c3c2ccc(c3)Cl)S(=O)(=O)c4ccc(cc4)Cl)C#N BTB08606 c1cc(c(c(c1)Cl)C(=O)OC2=C(CCN(c3c2ccc(c3)Cl)S(=O)(=O)c4ccc(cc4)Cl)C#N)F BTB08608 c1ccc2c(c1)c(c3c(n2)CCCC3)N.Cl BTB14162 CCOC(=O)c1cc(cc(c1)C(=O)OCC)CO BTB14164 CC(C)(C)c1ccc(cc1)CSc2nnc(n2C)S BTB08610 Cc1ccc(cc1)C(=O)c2ccc(cc2)C BTB14169 CN(C)/C=N/c1c(cnn1c2ccc(cc2)Cl)C#N BTB07495 c1cc(c(c(c1NC(=O)Cc2ncon2)F)F)F BTB07949 c1c(cnc(c1Cl)N/C=N/O)C(F)(F)F BTB07974 c1cc(c(nc1)NCc2ccc(cc2)Cl)[N+](=O)[O-] BTB07546 c1ccc2c(c1)c3ccccc3n2CC(COC4CCCCC4)O BTB11857 CCOC(=O)c1c[nH]c2c(ccc(c2c1=O)F)F BTB07839 c1ccc(cc1)Nn2c(csc2=S)c3cccc(c3)[N+](=O)[O-] BTB07843 CN(c1ccc(cc1)C(C(=O)OC)(C(F)(F)F)O)C(=O)Nc2ccc(c(c2)Cl)F BTB14225 CCOC(=O)C(=CNc1ccc(cc1)C(C(=O)OCC)(C(F)(F)F)O)C(=O)OCC BTB14229 Cn1c(cnc1/C=N/c2ccc(nc2)Oc3ccc(cc3)F)[N+](=O)[O-] BTB07426 c1ccc(cc1)C(=O)OCCS(=O)(=O)c2ccccn2 BTB08944 COc1ccc(c(n1)Sc2ccc(cc2)Cl)N BTB09163 c1ccc(cc1)C(=O)c2cccc(c2)[N+](=O)[O-] BTB09114 Cc1cccc(c1)Nc2ccc(cc2[N+](=O)[O-])Cl BTB14027 c1cc(ccc1C(=O)NCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl BTB07995 CCOC(=O)/C(=C\Nc1cc(cc2c1nccc2)OC)/C#N BTB09243 C1=C(C(=O)C=C(C1=O)Cl)Cl BTB14373 CSc1nc(c(s1)N)C(=O)N BTB14032 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1OC)NC(=O)c2ccco2 BTB14307 CNc1ncc(c(n1)c2ccccc2)c3nnnn3c4ccccc4 BTB11591 c1ccc2c(c1)c3ccccc3n2CC4CS4 BTB11869 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NC(=O)C BTB07894 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1)NC(=O)c2ccco2 BTB14298 Cc1cc(cc(c1O)CN2CCCCC2)/N=N/c3ccc(cc3)Cl BTB11599 Cc1cc(cc(c1O)CN2CCOCC2)/N=N/c3ccc(cc3)Cl BTB11600 Cc1cc(cc(c1O)CN2CCCC2)/N=N/c3ccc(cc3)Cl BTB11601 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)Cl)NC(=O)c2ccco2 BTB14303 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C)NC(=O)c2ccco2 BTB14305 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)OC)NC(=O)c2ccco2 BTB14306 Cc1ccc(cc1)S(=O)(=O)OC[C@@H]2[C@H]([C@H]([C@@H](O2)OC)OS(=O)(=O)c3ccc(cc3)C)OS(=O)(=O)c4ccc(cc4)C BTB11979 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1F)F)NC(=O)c2ccco2 BTB14311 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1Cl)NC(=O)c2ccco2 BTB14312 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)Oc2ccccc2)OC(=O)C)OC(=O)C)OC(=O)C BTB11984 CC(C)(C)c1cc(cc(c1)C(=O)NNC(=O)c2ccc(cc2Cl)Cl)C(=O)NNC(=O)c3ccc(cc3Cl)Cl BTB08650 CC(C)(C)c1cc(cc(c1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F BTB08651 C=CCn1c2ccc(cc2c3c1ccc(c3)Br)Br BTB11840 Cc1cc(cc(c1O)CN2CCCC2)/N=N/c3ccc(cc3)OC BTB11603 c1cc(c(nc1)Oc2ccc(cc2F)F)[N+](=O)[O-] BTB08013 COC(=O)c1cc2ccccc2s1 BTB07526 CC(=O)NC(c1ccc(cc1)Cl)n2ccnc2 BTB11619 CC1(OC[C@@H](O1)[C@H]([C@H]([C@@H]2COC(O2)(C)C)O)O)C BTB11983 CC(C)S[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O)O)O BTB11985 c1ccc2c(c1)c(c(s2)C(=O)N)Cl BTB07540 c1ccnc(c1)CNc2c(cccn2)[N+](=O)[O-] BTB07545 c1ccn(c1)c2cc(c(cc2Cl)NC(=O)c3ccc(cc3)Cl)Cl BTB07551 CCCn1c2ccccc2c3c1cccc3 BTB11845 C#CCn1c2ccccc2nn1 BTB14152 Cc1ccc(cc1)CCC(=O)O BTB14159 CCCCCCCCOc1ccc(cc1)c2ccc(cc2)C(=O)O BTB14160 Cc1ccc(cc1)C(=O)Oc2cccc3c2cc[nH]3 BTB07881 CCOC(CN(c1ccc(cc1)F)C(=O)c2ccc(cc2)[N+](=O)[O-])OCC BTB07877 c1cc(c(nc1)Oc2ccc(cc2F)F)N BTB08015 c1cc(c(nc1)Oc2ccc(cc2)F)N BTB08016 CC1=Nc2ccc3ccccc3c2C1(C)C BTB14062 CCOC(=O)N1CCCN=C1SC BTB07942 CCOC(=O)/C(=C/Nc1ccc(cc1F)O)/C#N BTB07945 CC(=O)C(C(=O)NC)Sc1nnc(s1)N BTB09058 c1cc(c(cc1Cl)Cl)C(=O)NN BTB08025 COc1cc(ccc1OCc2ccccc2)CC(=O)O BTB14066 c1cc(cc(c1)Cl)CSC2=NCCN2.Cl CD00383 CN(C)/C=N/c1nc([nH]n1)Sc2c(cccn2)[N+](=O)[O-] BTB08002 c1cc2c(cc[nH]2)c(c1)OS(=O)(=O)c3ccc(cc3Cl)Cl BTB07887 CCCSc1ccc(c(c1)NC(=O)c2c(nn(n2)c3ccccc3)C)[N+](=O)[O-] BTB07889 c1cc2c(cc[nH]2)c(c1)OC(=O)c3ccc(cc3)C(F)(F)F BTB07880 c1ccc2c(c1)ncc(n2)c3cccs3 BTB08701 c1cc2c(cc1C(=O)CSc3ccc(cc3Cl)Cl)CCC(=O)N2 BTB09229 c1ccc(cc1)N(C(=O)c2ccc(cc2)Cl)n3c(csc3=S)c4cccc(c4)[N+](=O)[O-] BTB07858 Cc1cc(cc(c1O)CN2CCCCC2)/N=N/c3ccc(cc3)OC BTB11602 Cc1ccc(cc1)C(=O)N(c2ccccc2)n3c(csc3=S)c4cccc(c4)[N+](=O)[O-] BTB07859 c1cc(c(nc1)Oc2ccc(cc2)F)[N+](=O)[O-] BTB08014 c1cnccc1C=C2C(=O)NC(=O)NC2=O CD00385 CCOC(=O)CC(=O)CSc1nnc(s1)N BTB07522 Cc1c(c(c(=O)n(n1)C)NC(=O)c2ccc(cc2)F)c3cc([nH]n3)c4ccsc4 BTB09013 c1cc(c(nc1)Oc2ccc(cc2)Cl)C3=N/C(=C\c4ccc(cc4)Cl)/C(=O)O3 BTB08768 c1cc-2c(cc1S(=O)(=O)N)Cc3c2ccc(c3)S(=O)(=O)N BTB11897 CN1C(=O)c2ccccc2[S+]1c3cccc4c3c(ccc4)C(=O)O.[Cl-] BTB11546 CCCN(CCC)S(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)N(CCC)CCC)C2=O BTB11894 c1cc(c(cc1Cl)Cl)SCC(=O)O BTB08747 Cc1nc(c(c(n1)SC)C#N)N(C)C BTB08997 Cc1c2c(onc2c(=O)n(n1)C)/C=C/c3ccsc3 BTB09000 CCOC(CN(c1ccc(cc1)F)S(=O)(=O)c2cc(cc(c2)Cl)Cl)OCC BTB07870 CCOC(CN(c1ccc(cc1)F)S(=O)(=O)c2ccc(cc2F)F)OCC BTB07871 CCOC(CN(c1ccc(cc1)F)C(=O)c2ccc(cc2)F)OCC BTB07874 Cc1ccc(cc1)C(=O)COc2cc(nc3n2cnn3)C BTB08754 CCOC(=O)CNC(=O)c1cccnc1Oc2ccc(cc2)Cl BTB08760 c1ccc2c(c1)c3ccccc3n2CO BTB11860 c1cc2c(cc[nH]2)c(c1)OS(=O)(=O)c3ccc(cc3F)F BTB07886 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NC(=O)c3ccc(c(c3)Cl)F BTB07902 c1cc(c(cc1[N+](=O)[O-])C(=O)O)Oc2cc(cnc2)Cl BTB07905 Cc1cnc(c(n1)C)NS(=O)(=O)c2ccccc2 BTB07908 c1cc-2c(cc1S(=O)(=O)N3CCOCC3)Cc4c2ccc(c4)S(=O)(=O)N5CCOCC5 BTB11900 c1ccnc(c1)SCCOC(=O)c2cccc(c2)Cl BTB08936 Cc1ccc(cc1)S(=O)(=O)N2CCCC2 BTB08938 Cc1ccc(cc1)S(=O)(=O)N2CCCCC2 BTB08939 c1cc2c(cc[nH]2)c(c1)OC(=O)c3c(cccc3F)F BTB07888 c1cc(cc(c1)Cl)C(=O)OCCS(=O)(=O)c2c(cccn2)Cl BTB09003 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ncccn1 BTB14232 c1ccc(cc1)n2c(=O)c(c(cn2)Oc3ccccc3)Cl BTB09007 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)NCC(=O)O BTB08763 C=CCN(c1ccccc1C(=O)NCC(=O)O)S(=O)(=O)c2ccccc2 BTB08764 c1ccc(cc1)CSc2c(cccn2)[N+](=O)[O-] BTB14070 Cc1nc(c(c(n1)N(C)C)C#N)Nc2ccc(cc2Cl)Cl BTB08991 Cc1c(c(on1)C)C(=O)Sc2ccc(cn2)C(F)(F)F SPB04435 c1ccc(c(c1)C(=O)O)S(=O)c2cccc3c2c(ccc3)CO BTB11515 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)Cl BTB14235 CCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB11883 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2c(cc(cn2)C(F)(F)F)Cl)Cl BTB07964 COC(=S)Nc1ccccc1 BTB11637 CN1C(=O)c2ccccc2S13c4cccc5c4c(ccc5)C(=O)O3 BTB11534 Cn1c(=O)c2c(cn1)N(N=C(S2)SC)C BTB09061 CCOC(=O)C1c2ccccc2Oc3c1cccc3 BTB10308 c1cc(c(cc1n2c(c(cn2)C#N)N)Cl)F BTB07486 c1cc(sc1)CC(=O)NCc2ccc(cc2)C(F)(F)F BTB08689 Cc1ccc(cc1)Oc2c(cccn2)C(=O)O BTB08735 Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl BTB11833 CN(C)/C=N/c1c(cc(cn1)C(F)(F)F)Cl BTB07972 COc1ccc(cc1Br)C=C2C(=O)NC(=O)NC2=O CD00382 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NC(=O)c3ccc(cc3)C(C)(C)C BTB07903 Cc1cc(n(n1)c2ccc(cc2)[N+](=O)[O-])O BTB09186 Cc1cnc(c(n1)C)NC(=O)Nc2ccccc2 BTB07909 Cc1c(c(c(=O)[nH]n1)N)c2cc([nH]n2)c3ccsc3 BTB09033 COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccc(cc3)Cl)Cl BTB07509 c1cc(ccc1NC(=O)Nc2c(cc(cn2)C(F)(F)F)Cl)Cl BTB07962 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2c(cc(cn2)C(F)(F)F)Cl)F BTB07963 COc1ccc(cc1)Oc2c(cnn(c2=O)c3ccc(c(c3)Cl)F)Cl BTB07510 CCOC(=O)CC(=O)CSc1nnc(s1)NC(=O)c2ccc(cc2)C BTB07805 c1cc2cnccc2c(c1)[N+](=O)[O-] BTB07826 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2Br)C(C)(C)C)Cl BTB07511 CC(C)(C)c1cc(c(c(c1)Br)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl BTB07514 CC(=O)C(=CNc1c(cc(cn1)C(F)(F)F)Cl)C(=O)C BTB07971 CCOC(=O)/C(=C/Nc1c(cc(cn1)C(F)(F)F)Cl)/C#N BTB07973 CC(C)(C(=O)Oc1ccc(cc1)Cl)S(=O)(=O)c2ccc(cn2)C(F)(F)F BTB09029 Cc1c2c(onc2c(=O)[nH]n1)/C=C/c3ccc(c(c3)Cl)Cl BTB09032 c1cc(c(c(c1NC(=O)CC#N)F)F)F BTB07906 CCOC(=O)C(C(F)(F)F)(Nc1nc2ccccc2s1)NC(=O)c3cccnc3 BTB14257 Cc1cccc(n1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2 BTB14261 c1ccc(cc1)c2cc(ccc2Oc3ccc(cn3)[N+](=O)[O-])Oc4ccc(cn4)[N+](=O)[O-] BTB08678 c1ccc(cc1)c2cc(ccc2Oc3c(cccn3)[N+](=O)[O-])Oc4c(cccn4)[N+](=O)[O-] BTB08679 CC(=O)C(=CNc1ccc(c(c1OC)C(=O)OC)OC)C(=O)C BTB07810 Cc1c(c(n[nH]1)c2ccc(cc2O)O)Oc3ccccc3 BTB11556 Cc1ccc(c(c1)C(=O)O)I BTB11559 CSc1c(c(nc(n1)c2ccccc2)Nc3ccc(cc3Cl)Cl)C#N BTB08963 c1cc(cnc1)CNc2c(cc(cn2)C(F)(F)F)Cl BTB07985 COC(=O)C1=NN(C(=O)C1)c2cccc(c2)C(F)(F)F BTB07825 CCOC(=O)C(=CNc1cc(ccc1F)F)C(=O)OCC BTB07830 c1c(c(cc(c1Br)C(=O)O)Br)C(=O)O BTB11564 c1cc(cnc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)F BTB14259 c1ccc(c(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2)F BTB14260 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)N4CCCCC4 BTB11886 CNC(=O)c1ccccc1S(=O)c2ccccc2 BTB11523 c1cc(cnc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)Cl BTB14262 CCCCN(CCCC)S(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)N(CCCC)CCCC BTB11889 CCN(CC)S(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)N(CC)CC)C2=O BTB11890 c1c(cc(c-2c1C(=O)c3c2c(cc(c3)S(=O)(=O)N4CCCCC4)[N+](=O)[O-])[N+](=O)[O-])S(=O)(=O)N5CCCCC5 BTB11891 c1ccc(cc1)c2[nH]c3c(c([nH]n3)N)c(=O)n2 BTB08967 c1ccc(cc1)C(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08617 c1ccc(cc1)n2c(=O)cc(c3c2CCCC3)O BTB11567 Cc1cc(n2c(n1)nc(n2)SC)O BTB11569 CCOC(=O)/C(=C/Nc1cc(ccc1F)F)/C#N BTB07831 CSC1=C(C(=C(C#N)C#N)NC(=N1)c2ccccc2)C#N BTB08975 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)N4CCOCC4 BTB11887 CCCCN(CCCC)C(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB11888 CCOC(=O)C1=C(N(C(=O)NC1c2ccccc2Cl)C)C BTB11959 Cc1cc(c(cc1Sc2cc(c(cc2C)Oc3ccc(cn3)[N+](=O)[O-])C(C)(C)C)C(C)(C)C)Oc4ccc(cn4)[N+](=O)[O-] BTB07496 CCOc1cc(ccc1O)C=C2C(=O)NC(=O)NC2=O CD00388 c1ccc(c(c1)Oc2ccc(cn2)N)F BTB08017 CC(C)c1ccc(cc1)NC(=S)NC(=N)OC SPB06996 CCc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2F)Cl BTB11791 Cc1c(nn(n1)c2ccccc2)C(=O)OCCC3C(=NN(C3=O)c4ccc(cc4)Cl)C BTB07506 c1cc(ccc1C(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)C(F)(F)F BTB08619 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccn2 BTB14274 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)Cc2ccccc2 BTB14278 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2F)F)NC(=O)c3cccs3 BTB09175 C/C=C(/C(=C/C)/c1ccccc1)\c2ccccc2 BTB14415 COc1ccc(c2c1C(=O)c3ccccc3C2=O)OC BTB14416 Cc1ccc(cc1)C(=O)O/N=C(/CC(=O)Nc2ccc(c(c2F)F)F)\N BTB07940 CCOC(=O)c1c(c(c(n1c2ccc(cc2Cl)Cl)/N=C/N(C)C)C#N)C BTB09080 CN(C)/C=N/c1cc(c(cc1Cl)n2cccc2)Cl BTB07552 Cc1cc(n2cnnc2n1)OCC(=O)c3cccc(c3)C(F)(F)F BTB08755 CCOC(=O)c1c(c2c(ncnc2n1c3ccccc3)/N=C\N(C)C)C BTB09119 c1ccc(cc1)c2c(c(c(n(c2=O)c3ccccc3)c4ccccc4)Cl)O BTB11805 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccc(c(c1F)F)F BTB14284 COc1ccc2ccccc2c1C3Nc4ccccc4C(=O)N3 BTB14013 CCOC(=O)/C=C/C(=O)[O-].[K+] BTB14020 CC(=O)Nc1ccc(cc1C(=O)O)OC BTB11557 Cc1ccc(cc1)C2=NC(N=C(O2)N3CCOCC3)(C(F)(F)F)C(F)(F)F BTB14293 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)Cl)NC(=O)Cc2ccccc2 BTB14295 CCOC(=O)/C(=N\OC)/c1csc(n1)NC(=O)c2c(nn(n2)c3ccccc3)C BTB08602 Cn1c(nnc1SCc2ccc(c(c2)Cl)Cl)S BTB08603 c1cc(ccc1S(=O)(=O)N2CCC(=C(c3c2cc(cc3)Cl)OS(=O)(=O)c4ccc(cc4)Cl)C#N)Cl BTB08605 CC(C)(C)c1ccc(cc1)C(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08618 CC(C)(C)c1ccc(c(c1)Cl)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB07488 COc1ccc(c(c1C(=O)N)OC)[N+](=O)[O-] BTB07490 CC(C)(C(=O)O)Oc1ccc(cc1)C#N BTB09159 Cc1c(cc(c(=O)[nH]1)C#N)c2csc(n2)c3ccccc3 BTB09160 c1ccc(c(c1)NC(=O)C(Cl)Cl)F CD04828 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2C(F)(F)F)Cl BTB14292 Cn1cc(c(n1)N)C(=O)Nc2ccc(c(c2F)F)F BTB07946 c1cc(c(cc1Cl)C(=O)O)I BTB11561 COC(=O)c1ccncc1C(=O)O BTB07951 c1cnc(c(n1)C(=O)O)C(=O)O BTB07953 CC1=C(C(NC(=O)N1)c2ccccc2)C(=O)C BTB11828 c1cc2c(cc1Cl)c3cc(ccc3[nH]2)Cl BTB11831 c1c(cc(c2c1c3cc(cc(c3[nH]2)Br)Br)Br)Br BTB11832 CCOC(=O)CC(=O)CSc1nnc(s1)NC(=O)c2c(cccc2F)F BTB07806 CCOC(CN(c1ccc(cc1)F)C(=O)c2ccc(cc2)C)OCC BTB07876 Cc1c(cc(c(n1)Sc2ccc(cc2)OC)C#N)c3csc(n3)C BTB09221 Cc1c(c(c(=O)n(n1)C)N)c2cc([nH]n2)c3ccc(c(c3)Cl)Cl BTB09053 CCC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cccc(c1)Cl BTB14248 c1ccc(cc1)CN(Cc2ccccc2)c3ccccc3 BTB14339 Cc1ccc(cc1)C(=O)/C=C(/C(=O)NNC(=O)c2cc(nc3c2cccc3)C)\O BTB14343 CC(=CC(=O)Nc1ccc(cc1F)Oc2cc(ccc2Cl)C(F)(F)F)C BTB08062 CCOC(=O)c1c(cc(cc1Cl)C)N2CCCC2 CD04805 c1cc(c(cc1C(F)(F)F)NC(=O)C(Cl)Cl)Cl CD04821 COc1cccc(c1)c2nnc(o2)c3cc(ccc3Oc4cc(cnc4)Cl)[N+](=O)[O-] BTB08055 COc1ccc(cc1)/N=N/c2ccc(c(c2)CN3CCCCC3)O BTB11596 Cc1c2c(onc2c(=O)n(n1)C)/C=C/c3ccc(c(c3)Cl)Cl BTB09049 Cc1ccc(cc1)c2cc(n[nH]2)c3c(nn(c(=O)c3N)C)C BTB09051 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Cl)C(=O)OCC)C)C BTB14328 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)O)C(=O)OCC)C)C BTB14329 Cc1ccc(cc1)NC(=O)N(c2ccccc2)C3=NCC(S3)(C)C BTB14283 CC(=O)OC1CC2CCC1N(C2=O)Cc3ccccc3 BTB14333 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(n2)C BTB14291 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)F)NC(=O)Cc2ccccc2 BTB14294 c1cc(ccc1/C=C\2/C(=O)NC(=O)N2)OC(=O)c3ccc(cc3Cl)Cl BTB08066 c1ccc(cc1)C(=O)Oc2ccc(cc2)/C=C\3/C(=O)NC(=O)N3 BTB08068 c1ccc(cc1)Nn2c(csc2=S)c3ccc(c(c3)Cl)Cl BTB07845 c1ccc(cc1)C(=O)N(c2ccccc2)n3c(csc3=S)c4cccc(c4)[N+](=O)[O-] BTB07856 c1ccc(cc1)N(C(=O)c2ccc(cc2)C(F)(F)F)n3c(csc3=S)c4cccc(c4)[N+](=O)[O-] BTB07857 CC(=O)NC(c1ccccc1)n2cncn2 BTB11615 c1cc(ccc1/N=N/c2ccc(c(c2)CN3CCCCC3)O)Cl BTB11593 CCOC(=O)c1ccc(cc1)N/C(=C(/C#N)\C(=O)OCC)/SC BTB12055 CCOC(=O)/C(=C(\N(C)C)/SC)/C#N BTB12057 Cc1ccc(cc1)S(=O)(=O)/N=C(/N(C)C)\SC BTB12060 CCOC(=O)C1=C(N(C(=O)NC1c2ccc3c(c2)OCO3)C)C BTB11953 c1cc(ccc1/C=C\2/C(=O)NC(=O)N2)OS(=O)(=O)c3ccc(cc3F)F BTB08064 c1cc(ccc1/C=C\2/C(=O)NC(=O)N2)OS(=O)(=O)c3ccc(cc3)Cl BTB08065 Cn1c(c2c(n1)CCCC2)N(C)C(=O)CSc3ccc(cn3)C(F)(F)F BTB09208 CC(=O)Oc1cc2c(c3c1cccc3)oc(=O)s2 BTB11964 Cc1c(cc(c(n1)Sc2ccccc2)C#N)c3csc(n3)C BTB09218 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@H](O1)OC2[C@H](O[C@H]([C@@H]([C@H]2OC(=O)C)OC(=O)C)OC(=O)C)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C BTB11977 COc1ccc(cc1)/N=N/c2ccc(c(c2)CN3CCOCC3)O BTB11597 c1ccc2c(c1)c(c[nH]2)CCO BTB14321 CCOC(=O)C1=C(NC(=O)NC1c2cccc3c2cccc3)C BTB11954 CN(C)Cc1ccc(o1)CSCCNC(=O)Nc2ccccc2 BTB08081 c1ccc(cc1)/C=C/C(=O)Nc2cccnc2Oc3ccccc3F BTB08112 Cc1c(cc(c(=O)[nH]1)C#N)c2csc(n2)C BTB09214 c1ccc(cc1)C(=O)NNC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08117 CN(C)CC(Cn1c2ccccc2c3c1cccc3)O BTB12226 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)C(=O)CSc2nnc(n2c3ccccc3)Nc4ccccc4 BTB14414 Cn1c(c2c(n1)CCCC2)N(C)C(=O)CSc3ccccn3 BTB09205 CC(=O)C(C(=O)NC)Sc1nnc(s1)NC(=O)c2ccc(cc2)Cl BTB09064 CCOC(=O)c1c(c2c(=O)[nH]cnc2n1c3ccccc3)C BTB09066 CC(C)(C)c1cc(c(c(c1)Br)OS(=O)(=O)c2cc(cc(c2)Cl)Cl)Cl BTB07518 c1cc(c(c(c1NC(=O)C/C(=N/O)/N)F)F)F BTB07938 COc1ccc(cc1)OCC(CN)O BTB12133 Cc1cc(cc(n1)S(=O)(=O)CCOC(=O)c2cccc(c2)Cl)C(F)(F)F BTB09085 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ncccn2 BTB14275 c1cc(ncc1C(F)(F)F)SCC(=O)O BTB08102 c1cc(ccc1c2nnc(o2)c3cc(ccc3Oc4cc(cnc4)Cl)[N+](=O)[O-])C(F)(F)F BTB08056 Cc1c(cc(c(n1)Sc2cccc(c2)C(F)(F)F)C#N)c3csc(n3)C BTB09219 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NC(=O)Nc3ccccc3 BTB07891 CCOC(=O)c1c(c(c(n1c2ccc(cc2)C)n3cccc3)C#N)C BTB09076 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C)NC(=O)c2ccco2 BTB14301 CCOC(=O)COc1ccc2c3ccccc3c(=O)oc2c1 BTB14371 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)c2ccco2 BTB14309 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1F)NC(=O)c2ccco2 BTB14310 CC1(OC2C(OC(C2O1)n3cnc4c3nc[nH]c4=O)CO)C BTB14375 CN(C)/C=N/c1nc([nH]n1)Sc2c(cccc2Cl)[N+](=O)[O-] BTB07999 Cn1c(=O)c2c(cn1)N(N=C(S2)SCc3ccc(cc3Cl)Cl)C BTB09089 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(c(c1F)F)F BTB07910 CC(C)(C(=O)Nc1ccccc1)S(=O)(=O)c2ccc(cn2)C(F)(F)F BTB09023 Cc1ccc(cc1)/C=C/c2c3c(n[nH]c(=O)c3no2)C BTB09031 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)[N+](=O)[O-] BTB07544 c1cc(c(nc1)NCc2cccs2)[N+](=O)[O-] BTB07547 CCOC(=O)C(C(F)(F)F)(Nc1ccccn1)NC(=O)c2ccco2 BTB14304 CCOC(=O)C(=c1sc(=C(C#N)C(=O)OCC)s1)C#N BTB12101 COC(=O)CS(=O)(=O)c1ccc(cn1)C(F)(F)F BTB08115 COC(=O)c1cc(=O)nc2n1C3[C@H](O2)C([C@H](O3)CO)O BTB11661 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)c2[nH]nnn2)OC(=O)C)OC(=O)C)OC(=O)C BTB11666 c1ccc(c(c1)[N+](=O)[O-])O[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)CO)O)O)O BTB11976 COc1ccc(cc1)C(=O)/C=C/Sc2c(cc(cn2)C(F)(F)F)Cl BTB12035 Cc1ccc(cc1)C2=NC(N=C(O2)N3CCCCC3)(C(F)(F)F)C(F)(F)F BTB14276 CCOC(=O)C(C(F)(F)F)(Nc1nc2ccccc2s1)NC(=O)Cc3ccccc3 BTB14277 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)Cc2ccccc2 BTB14279 CN(C)c1c(c(nc(n1)c2ccccc2)Nc3ccc(cc3Cl)Cl)C#N BTB08994 c1ccn(c1)c2cc(c(cc2Cl)N/C=N/O)Cl BTB07553 CCOC(=O)CNC(=O)c1ccccc1N(CC=C)C(=O)c2ccc(cc2)Cl BTB08774 c1cc2c(c3c(n2O)CCCC3)c4c1non4 BTB14048 c1cc(ccc1[N+](=O)[O-])O[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)CO)O)O)O BTB11973 c1cc(ccc1[N+](=O)[O-])O[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)CO)O)O)O BTB11974 CCOc1ccc(cc1C=C2C(=O)NC(=O)NC2=O)Br CD00430 C1CC23CC(=O)CC2(C1)CC(=O)C3 BTB14425 CC(=O)Nc1ccc(cc1)OCCOc2ccc(cc2)NC(=O)C BTB12138 CC(=O)Nc1c(cc(cn1)C(F)(F)F)Cl BTB07969 CC1(c2ccccc2N(C13C=Cc4cc(ccc4O3)O)C)C BTB14058 c1cc(cc(c1)CC#N)CC#N BTB14061 c1cc(cc(c1)Cl)C(=O)NC2CN3CCC2CC3 BTB14063 CCOC(=O)c1c(c(c(n1c2ccc(cc2)C)NC(=O)c3ccc(cc3Cl)Cl)C#N)C BTB09107 c1ccc(cc1)S(=O)(=O)NC(=S)NC2CCCCC2 BTB12074 COC(=O)c1ccc(cc1)c2ccc(cc2)C(=O)OC BTB09118 Cc1c(cc(c(n1)Sc2ccc(cc2Cl)Cl)C#N)c3csc(n3)C BTB09222 Cc1c(cc(c(n1)Oc2ccc(cc2)C(F)(F)F)C#N)c3csc(n3)C BTB09226 c1ccc(cc1)Nc2nc-3c(s2)Cc4c3cccc4.Br CD00350 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)Cc2cccs2)/N BTB08695 c1cc(c2c(c1N)C(=O)c3c(ccc(c3C2=O)O)N)O BTB14385 Cn1c2cnn(c(=O)c2c(n1)SCc3ccc(cc3Cl)Cl)C BTB09103 CCOC(=O)c1c(c(c(n1c2ccccc2)NC(=O)C(C)(C)C)C#N)C BTB09105 Cn1c2cnn(c(=O)c2c(n1)S(=O)(=O)Cc3ccc(cc3Cl)Cl)C BTB09106 CC(=S)[C@@H]([C@H]([C@@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C BTB12007 Cc1cc(n(n1)c2nc(cs2)c3ccc(cc3)Br)C BTB12016 c1ccc(cc1)c2nc\3c(n2O)CCC/C3=N/O BTB13060 c1cc(ncc1C(F)(F)F)SCCNC=C(C#N)C#N BTB07923 Cc1ccc(cc1)C(=O)OCCSc2ccc(cn2)C(F)(F)F BTB07925 c1cc(sc1)CC(=O)O/N=C(/c2ccc(cc2)Cl)\N BTB08692 c1cc(ncc1C(F)(F)F)S(=O)(=O)CCO BTB07931 c1cc(ccc1C(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl BTB07935 Cc1cc(on1)/N=C/N(C)C BTB08698 CCOC(=O)/C(=C/Nc1cc(no1)C)/C#N BTB08705 Cc1cc(n2c(n1)nc(n2)SC)OC BTB08708 CCOC(=O)/C(=N\Nc1c(cccc1Cl)Cl)/c2csc(n2)N BTB09041 CC(=O)/C=C\c1ccc(cc1)O[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C BTB12005 C[C@]12CC=C([C@]1(CC=C2C#N)C)C#N BTB14407 c1ccc(cc1)c2ccc(=O)on2 BTB13079 CC(C)(C)n1c(cc(n1)c2ccccc2)O CD04815 c1cc(ccc1C(=O)OCCSc2ccc(cn2)C(F)(F)F)Cl BTB07926 c1cc(ccc1C(=O)NCCSc2ccc(cn2)C(F)(F)F)Cl BTB07927 Cc1ccc(cc1)/C=C/c2c3c(nn(c(=O)c3no2)C)C BTB09047 Cc1c2c(onc2c(=O)n(n1)C)/C=C/c3ccc(cc3)C(F)(F)F BTB09048 c1ccc(cc1)COC(=O)NC(C(F)(F)F)(C(F)(F)F)OCc2ccccc2 BTB14249 COc1ccc(cc1)Oc2ccc(cn2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F BTB07428 c1cc(cnc1)C2=NC(N=C(O2)N3CCOCC3)(C(F)(F)F)C(F)(F)F BTB14268 C[C@@]12[C@@](C(=O)C=C1)(C(=O)C=C2)C BTB14410 Cn1c(=O)cc(c2c1n(c(=O)n(c2=O)c3ccccc3)c4ccccc4)Nc5ccccc5 BTB13074 Cn1c2c(c(c(c1=O)[N+](=O)[O-])O)c(=O)n(c(=O)n2C)C BTB13075 CC(=O)c1ccc2c(c1)OCCO2 BTB12187 c1ccc2c(c1)C(c3ccccc3O2)C4C(=O)c5ccccc5C4=O BTB12190 c1cc2c(cc1Br)c3cc(cc(c3n2CC(CN4CCCCCC4)O)Br)Br BTB12220 CCN(CC)CC(Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl)O BTB12223 CCOC(=O)c1cnc2c(ccc(c2c1Oc3cccnc3)F)F BTB08680 CCOC(=O)c1cnc2c(ccc(c2c1Oc3cc(cnc3)Cl)F)F BTB08681 CC(=O)NCc1ccccc1S(=O)c2ccccc2C(=O)O BTB11526 c1cc(ccc1[N+](=O)[O-])O[C@@H]2[C@@H]([C@H]([C@@H]([C@H](O2)CO)O)O)O BTB11991 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/C(=O)Nc2ccc(c(c2F)F)F BTB07913 CCCCCCCCCCN(CCCCCCCCCC)S(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)N(CCCCCCCCCC)CCCCCCCCCC BTB12214 CCOC(=S)NC(C)(C)C BTB14402 CCOC(=O)C1=C(NC(=C(C1c2ccc(c(c2)OC)O)C(=O)OCC)C)C BTB14330 CCOC(=O)C1=C(NC(=C(C1c2ccco2)C(=O)OCC)C)C BTB14332 CCOC(=O)c1cccc(c1)[N+](=O)[O-] BTB09265 c1ccc(cc1)S[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)CO)O)O)O BTB11990 CCCCCCCCCCc1ccc(cc1)c2ccccc2 BTB10314 CCOC(=O)c1c(c(c(n1c2ccccc2)NC(=O)c3ccccc3)C#N)C BTB09101 CN(C)/C=N/c1nc([nH]n1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB08000 c1ccc2cc(ccc2c1)c3csc(n3)N.Br CD00379 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1)NC(=O)c2cccnc2 BTB14258 CCOC(=O)/C(=C\Nc1cc2cccnc2c(c1)OC)/C#N BTB09249 COc1ccc(c(n1)S(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] BTB09154 Cc1ccc(c(c1)NC(=O)C)OC(C)(C)C(=O)OC(C)(C)C BTB09157 c1ccc(cc1)n2c(=O)nc3n(c2=O)c4ccccc4s3 BTB12009 CCN(CC)C(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB11885 c1c(cc(c-2c1C(=O)c3c2c(cc(c3)S(=O)(=O)N4CCCCCC4)[N+](=O)[O-])[N+](=O)[O-])S(=O)(=O)N5CCCCCC5 BTB11893 CCCCN(CCCC)S(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)N(CCCC)CCCC)C2=O BTB11895 c1ccn2c(c1)nc(n2)c3cccc(c3)C(F)(F)F BTB12020 Cc1ccc(cc1)Sc2c(cccn2)C(=O)NCC(=O)OC BTB08742 COC(=O)CNC(=O)c1cccnc1Oc2ccc(cc2)Cl BTB08745 COc1ccc(c(c1)SCC(=O)O)OC BTB08746 CCOC(=O)c1c(c(c(n1c2ccccc2)NC(=O)c3ccc(cc3Cl)Cl)C#N)C BTB09104 c1cc(cc(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2)C(F)(F)F BTB14263 c1cc(cc(c1)Cl)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2 BTB14265 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)O[C@@H]([C@@H](COC(=O)C)OC(=O)C)[C@H]([C@@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C BTB12003 COc1cccc(c1)CC(=O)N BTB09254 c1ccc(cc1)N/N=C/C(=N\Nc2ccccc2)/[C@@H]([C@H]([C@@H](CO)O)O[C@H]3[C@@H]([C@H]([C@@H]([C@H](O3)CO)O)O)O)O BTB12004 Cc1cccc(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2 BTB14266 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccc2F BTB14271 c1cc(ccc1c2nnc(o2)c3cc(ccc3Oc4cc(cnc4)Cl)[N+](=O)[O-])Cl BTB08051 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3cc(ccc3Oc4cc(cnc4)Cl)[N+](=O)[O-] BTB08052 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)F BTB14272 Cn1c2ccccc2c(c(c1=O)c3ccccc3)O BTB11565 CCN(CC)S(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)N(CC)CC BTB11901 c1ccc(cc1)C2(C(=O)c3cc(ccc3NC2=O)Cl)F BTB11952 CCCC1=C(C(=O)NC1)c2ccccc2 BTB09311 CCOC(=O)C1=C(C(=O)N(C1)c2ccccc2)N BTB09312 c1cc([nH]c1)/C=C(\C#N)/C(=O)Nc2ccc(c(c2F)F)F BTB07915 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])NN=C2CCCCC2 BTB09139 C=CCN(c1ccccc1C(=O)NCC(=O)O)S(=O)(=O)c2ccccc2Cl BTB08769 C=CCN(c1ccccc1C(=O)NCC(=O)O)S(=O)(=O)c2ccc(cc2)Cl BTB08770 CSc1c(cccn1)C2=N/C(=C\c3ccc(cc3)Cl)/C(=O)O2 BTB08776 CC(C)(C)SCCNC(=O)C(C)(C)S(=O)(=O)c1ccc(cn1)C(F)(F)F BTB09140 CC(=O)Nc1ccc(cc1)S(=O)(=O)N BTB11566 Cc1cn(c(=O)[nH]c1=O)[C@@H]2C[C@H]([C@@H](O2)COS(=O)(=O)C)OS(=O)(=O)C BTB11576 c1ccc(cc1)C(=O)Nc2ccccc2[N+](=O)[O-] BTB11949 c1cc(ccc1/C=C\2/C(=O)NC(=O)N2)OS(=O)(=O)c3cc(cc(c3)Cl)Cl BTB08060 CCOC(=O)/C(=C/Nc1nc(cs1)c2cc(c(=O)[nH]c2C)C#N)/C#N BTB09209 c1cc(ccc1C(=O)O/N=C(/C=C/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N)Cl CD04804 c1cc(cc(c1)S(=O)(=O)NNC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F)C(F)(F)F BTB08129 CN(c1ccccc1)/N=C/Cc2nnnn2c3ccc(cc3)Cl BTB14344 CC(=O)OC[C@@H]([C@H]([C@H]([C@@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C BTB11995 CC(=O)O[C@@H]1[C@H](O[C@H]([C@@H]([C@H]1OC(=O)C)OC(=O)C)OC(=O)C)COC(c2ccccc2)(c3ccccc3)c4ccccc4 BTB11993 CC1(C2CCC1(/C(=N/OC(=O)c3ccc(cc3)[N+](=O)[O-])/C2)C)C BTB10347 c1cc(ccc1CSC2=NCCN2)C#N.Br CD00410 c1cc2c(cc1Cl)c3cc(ccc3n2CC(CN4CCCCCC4)O)Cl BTB12250 COc1ccc(c(c1OC)Cl)C(=O)O BTB09259 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=C/c2nc(on2)CN3CCCC3 CD04850 CCCCCCNc1ccc(cc1)C(=O)O BTB10317 Cc1cc(cc(c1OC(=O)Nc2ccccc2)C)c3c4ccccc4c(=O)n(n3)C BTB08294 CCCCCCCCCCN(CCCCCCCCCC)S(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)N(CCCCCCCCCC)CCCCCCCCCC BTB12204 c1ccc(cc1)C2c3ccccc3CC(=O)N2 BTB12202 c1cc2c(cc1C3=CSC4=NCCN34)CCC(=O)N2 BTB09263 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccc(c2C(=O)Nc3cc(ccc3Cl)C(F)(F)F)F BTB09177 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)/C=C\3/C(=O)NC(=O)N3 BTB08071 CN(C)Cc1ccc(o1)CSCCNC(=O)Nc2ccc(c(c2)Cl)Cl BTB08079 CN(C)Cc1ccc(o1)CSCCNC(=O)Nc2ccc(cc2)Cl BTB08080 c1ccc(cc1)/C=C/C(=O)Nc2ccc(nc2)Oc3ccccc3F BTB08109 Cn1c(cc(n1)O)C(F)(F)F BTB09194 c1cc(ccc1SCSc2ccc(cc2)Cl)Cl CD05015 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)c4ncccn4 BTB14511 COC(=O)c1ccccc1S(=O)(=O)N2CCN(CC2)c3ncccn3 BTB14513 c1ccc(c(c1)N)Nc2c(cn(c(=O)n2)Cc3ccc(cc3)Cl)C#N BTB08232 Cc1cccc(c1N=C=Nc2c(cccc2C)C)C BTB14421 CN(C)CCCNC(=O)c1c(cccc1F)NC(=O)c2cccs2 BTB09179 Cn1c2ccccc2c(c(c1=O)[N+](=O)[O-])O BTB12121 Cc1ccc(c2c1CCC2)Oc3c(cccn3)N BTB09397 c1cc(ccc1OC(=O)/C=C/c2cc(ccc2Sc3ccc(cn3)C(F)(F)F)[N+](=O)[O-])Cl BTB09423 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08124 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08125 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)C=C(C#N)C#N BTB08140 CS(=O)(=O)NNC(=O)CS(=O)(=O)c1ccc(cn1)C(F)(F)F BTB08127 c1ccc(cc1)CS(=O)(=O)Oc2c(=O)c3ccccc3oc2c4ccccc4 BTB14499 CCCCCCCCCc1c(c2ccccc2[nH]c1=O)O BTB12125 COc1ccccc1N2C(=O)C3C(N(OC3C2=O)c4ccc(cc4)Cl)c5ccc(cc5)O BTB14348 CC(=C)C(=O)Nc1cccnc1Oc2ccccc2F BTB08131 c1cc(c(c(c1)Cl)C(=O)N2CCN(CC2)c3ncccn3)Cl BTB14507 c1cc2cccc(c2c(c1)S(=O)(=O)[O-])Cl.[Na+] BTB09071 CCOC(=O)c1c(c(c(=N)n(n1)c2ccc(cc2Cl)Cl)C#N)C BTB09073 CCOC(=O)c1c(c(c(n1c2ccc(cc2)C)N)C#N)C BTB09074 CCSc1ncc(c(n1)c2ccccc2)c3nnnn3c4ccccc4 BTB12040 c1cc2c(cc1Br)c3cc(ccc3n2CC(CN4CCCCC4)O)Br BTB12229 c1cc(ccc1SCc2nc(no2)/C=C/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl CD04849 c1cc(cc(c1)[N+](=O)[O-])C(=O)N2CCN(CC2)c3ncccn3 BTB14504 Cc1cc(c(cc1Cl)C)S(=O)(=O)N2CCN(CC2)c3ncccn3 BTB14505 CC(=O)NNC(=O)CS(=O)(=O)c1ccc(cn1)C(F)(F)F BTB08128 CC(C)(C(=O)NCC(=O)OC)Oc1ccc(cc1)C#N BTB09277 CCOC(=O)c1ccc(c(c1Cl)OC)OC BTB09278 CCOC(=O)C1=C(C(=O)N(C1)C2CCCCC2)O BTB09300 C[n+]1c(ccc2c1cccc2)/C=C/c3ccc(cc3)N(C)C.[I-] BTB10323 CC[n+]1ccccc1/C=C/c2ccc(cc2)N(C)C.[I-] BTB10324 Cn1c2ccccc2nc1C(F)(F)F BTB14437 c1ccc2c(c1)ccc(c2O)CN3CCOCC3 BTB12142 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)CCC(=O)OC BTB12143 CCOC(=O)/C(=C(\Nc1ccc(cc1)OC)/SC)/C#N BTB12054 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)c2cccnc2 BTB14281 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C(F)(F)F)NC(=O)c2cccnc2 BTB14282 CC(C)CCN(CCC(C)C)CC(Cn1c2ccc(cc2c3c1ccc(c3)Br)Br)O BTB12251 c1ccc(c(c1)N)Nc2c(cn(c(=O)n2)Cc3cccs3)C#N BTB08248 c1cc(ccc1[N+](=O)[O-])Oc2ccc(c(c2)C(=O)O)C(=O)O BTB14469 Cc1ccc(cc1)S(=O)(=O)N=C(SC)SC BTB12061 c1cc(sc1)C(=O)N2CCN(CC2)c3ncccn3 BTB14503 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)c3ncccn3)C(F)(F)F BTB14506 c1ccc(cc1)/C=N/NC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08122 CCCCCCCCCO[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)CO)O)O)O BTB11968 c1ccc(cc1)/C=C/C(=O)Nc2ccc(nc2)Oc3ccc(cc3)F BTB08111 CCCCCCCCCCCCO[C@H]1[C@@H]([C@H](C([C@H](O1)CO)O[C@@H]2[C@@H]([C@H]([C@@H]([C@H](O2)CO)O)O)O)O)O BTB11969 Cc1cc([nH]n1)C(F)(F)F BTB14053 COc1ccc2c(=O)cc(oc2c1)c3ccccc3OC BTB14493 CCc1c(c(c(=O)n(c1c2ccccc2)c3ccccn3)c4ccccc4)O BTB12108 c1ccc(cc1)Oc2ccc(cc2)OS(=O)(=O)c3ccc(cc3)F BTB14508 c1cnc(nc1)N2CCN(CC2)C(=O)C3CCCCC3 BTB14510 c1ccc(cc1)/C(=N/OC(=O)c2cccs2)/O CD04997 c1ccc(cc1)c2cc(n[nH]2)C(=O)NN BTB14347 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)c4ncccn4 BTB14509 c1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)C#N BTB14512 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2ccc(cc2)[N+](=O)[O-] BTB14514 c1cc(ccc1C2(CCNCC2)O)Cl BTB09284 C[n+]1ccccc1/C=C/c2ccc(cc2)N(C)C.[I-] BTB10321 CC1=C(C(C(=O)N1)CC(=O)OC)C(=O)OC BTB09299 CC1(C=C(C(N1)(C)C)C(=O)N)C BTB14057 c1ccc(cc1)C2(c3ccccc3-c4c2cccc4)O BTB14462 CCCCSc1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])SCCCC)C2=O BTB12211 COc1ccc(c(c1OC)Cl)C(=O)OC BTB09269 Cn1c2cnn(c(=O)c2c(n1)SC)C BTB09090 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)C(=O)Nc4ccc(cc4)Cl BTB08142 CC(=O)CSc1ccc(cn1)C(F)(F)F BTB08149 CCCCCCCCCc1c(c2ccccc2n(c1=O)C)O BTB12120 CCOC(=O)c1c(cc(nc1O)C)O BTB12129 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)C(c3ccccc3)c4ccccc4 BTB08155 c1cc(ccc1Oc2ccc(cn2)NS(=O)(=O)CS(=O)(=O)Nc3ccc(nc3)Oc4ccc(cc4)F)F BTB08146 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)CCC(=O)O BTB12144 CC1(CC2=C(C(C3=C(O2)CC(CC3=O)(C)C)c4ccc(cc4)Br)C(=O)C1)C BTB14354 CC1=C(C(NC(=O)N1)c2ccco2)C(=O)C BTB14358 COc1cc(c(c(c1)OC)[N+](=O)[O-])OC BTB09099 Cc1c(c(c(cn1)Cl)N)Cl BTB14386 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)O)c3ccccc3 BTB08175 CCOC(=O)C1C(N(C(=O)C1=O)C)c2ccccc2 BTB09305 CCc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2)C(=O)C BTB12038 CCOC(=O)c1c(c([nH]c1C)C(=O)OCC)C BTB09314 c1cc(ccc1/C=C\2/C(=O)NC(=O)N2)OC(=O)c3ccc(c(c3)Cl)F BTB08067 CC(=O)c1ccc(cc1)N/C=C/C(=O)c2ccc(cc2)F BTB12039 CN(C)/C=C(/c1nnnn1c2ccc(cc2)OC)\C(=O)c3ccc(cc3)Cl BTB12042 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)N2CCCCC2)OC(=O)C)OC(=O)C)OC(=O)C BTB12093 Cc1ccc(cc1)N[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C BTB12090 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Nc2ccc(cc2)Br)OC(=O)C)OC(=O)C)OC(=O)C BTB12091 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)c2ccco2 BTB14300 c1cc(ccc1C(=O)/C=C/Sc2cc(ccc2Cl)Cl)Br BTB12032 CCOC(=O)/C(=C(\NC)/SC)/C#N BTB12056 Cc1cc(cc(c1OS(=O)(=O)c2ccccc2OC(F)(F)F)C)c3c4ccccc4c(=O)n(n3)C BTB08286 CC(C)(C)c1nnc(s1)NC(=O)Nc2ccc(cc2)OC(F)(F)F BTB08287 c1cc(ncc1C(F)(F)F)S(=O)(=O)CC(=O)NN BTB08116 c1cc(ccc1n2c(=O)n3c(n2)NCCC3)F BTB08269 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2ccc(cc2)OC(F)(F)F BTB08292 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)cccn3 BTB12021 c1cc2c(cc1CCCC(=O)O)OCCO2 BTB13064 Cc1ccc(cc1)/N=C/c2ccccc2O BTB13067 Cn1c2c(c3c(c1=O)cc4ccccc4n3)c(=O)n(c(=O)n2c5ccccc5)c6ccccc6 BTB13069 c1cc(ccc1/C(=C/C=C(C#N)C#N)/Sc2cc(ccc2Cl)Cl)Cl BTB12027 Cc1cc(cc(c1OCC(=O)OC)C)c2c3ccccc3c(=O)n(n2)C BTB08290 c1cc(cc(c1)C(F)(F)F)C(=O)CSc2ccc(cn2)C(F)(F)F BTB08151 CC(=C1C2C=CC1c3c2cccc3)C BTB14374 COc1ccccc1c2cc(=O)c3ccccc3o2 BTB14495 c1cc(c(nc1)Oc2ccc(cc2)/C(=C/c3ccc(cc3)C(F)(F)F)/C#N)[N+](=O)[O-] BTB08159 C1CSC(=C2C=CC=C2)S1 BTB14389 CCCCCCCCCCN(CCCCCCCCCC)S(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)N(CCCCCCCCCC)CCCCCCCCCC)C2=O BTB12205 Cc1c(cc(c(n1)NCc2ccccc2)C#N)c3csc(n3)C BTB09273 CCc1c(c([nH]c1C)C(=O)OCC)C BTB09309 CC1=C(C(C(=O)N1)CC(=O)O)C(=O)C BTB09310 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)S(=O)(=O)c4cc(ccc4Cl)Cl BTB08153 c1cc(cc(c1)NC(=O)CSc2ccc(cn2)C(F)(F)F)C(F)(F)F BTB08178 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)O)c3cccc(c3)Cl BTB08181 Cc1ccc(cc1)S(=O)(=O)NC(=S)Nc2ccccc2 BTB12073 c1cc(ccc1Sc2ccc(cc2C#N)[N+](=O)[O-])Cl BTB08185 c1ccc(cc1)NC(=O)N(CCC#N)Cc2ccco2 BTB08198 CC1=C(C(C(=O)N1)CC(=O)O)C(=O)OC BTB09316 c1cc(oc1)C=C2C(=O)NC(=O)NC2=O CD00394 C(CS(=O)(=O)O)NC(=N)N BTB09138 c1cc(ccc1c2ccc(cc2)C(=O)N)C(=O)N BTB09150 c1cc(ccc1/C=N\NC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl BTB08119 CC(C)(C(=O)NCCSc1ccccc1)S(=O)(=O)c2ccc(cn2)C(F)(F)F BTB09142 CC(C)(C)SCC(=O)c1ccc2c(c1)CCC(=O)N2 BTB09245 CCOC(=O)c1c(c(c([nH]1)C)C)C BTB09339 c1cc2c(cc1C3=CSC4=NCCCN34)CCC(=O)N2 BTB09343 c1ccc(cc1)/C=C/C(=O)Nc2ccc(nc2)Oc3ccc(cc3F)F BTB08108 COc1ccc(cc1)N[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)COCc3ccccc3)OCc4ccccc4)OCc5ccccc5)OCc6ccccc6 BTB12092 c1ccc(cc1)C2=CCC3C2CC=C3c4ccccc4 BTB14456 c1ccc(cc1)NC(=O)NNC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB08120 COc1ccc(c(c1OC)Cl)C(=O)N BTB09270 c1ccc2c(c1)C(=O)c3c(cc(c(c3C2=O)N)S(=O)(=O)O)N BTB14338 COc1ccc(c(c1OC)Cl)/C=C/C#N BTB09274 c1cc(ccc1/C=N/NC(=N)N)Cl BTB11997 c1ccc2c(c1)C(=CC(=O)C2=O)Nc3ccccc3O BTB13061 c1ccc(cc1)/C=C/C(=O)Nc2cccnc2Oc3ccc(cc3F)F BTB08114 c1ccc(cc1)SCC(=O)c2ccc3c(c2)CCC(=O)N3 BTB09244 c1cc(ccc1NC(=O)Nc2cc(ccn2)C(F)(F)F)OC(F)(F)F BTB08316 c1cc(ccc1NC(=O)NNC(=O)CS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl BTB08121 COc1cccc(c1)CC(=O)NN BTB09260 CC(=O)Nc1cccc(c1)OCCCNC(=O)C2CCCCC2 BTB14515 c1ccc(cc1)NC(=O)Nc2nc3ccccc3s2 BTB12023 c1ccc(cc1)OS(=O)(=O)c2cc3c(c(c2)[N+](=O)[O-])-c4c(cc(cc4[N+](=O)[O-])S(=O)(=O)Oc5ccccc5)C3=O BTB11896 CN(C)S(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)N(C)C BTB11898 c1cc-2c(cc1S(=O)(=O)N3CCCCC3)Cc4c2ccc(c4)S(=O)(=O)N5CCCCC5 BTB11899 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)F)NC(=O)c2cccnc2 BTB14296 CCCCCCC(=O)c1ccc(cc1)Br BTB13062 Cc1ccc(c2c1CCC2)OC(C)(C)C(=O)O BTB09368 CC1(CN(C(=S)N(C1=O)C(=O)c2ccc(cc2)Cl)c3ccccc3OC)C BTB08257 c1ccc(cc1)c2c(=S)ssc2SCC(=O)c3ccccc3 BTB08263 c1ccc(cc1)Sc2ccc(cc2C#N)[N+](=O)[O-] BTB08184 Cc1ccc2c(c1[N+](=O)[O-])cccn2 BTB10313 c1ccc-2c(c1)Cc3c2nc(s3)Nc4cc(c(cc4Cl)Cl)Cl.Br CD00351 c1cc(ccc1CSC2=NCCCN2)C#N.Br CD00461 c1cc(oc1)CN(CCC#N)S(=O)(=O)c2cc(cc(c2)Cl)Cl BTB08200 c1ccc(cc1)NC(=N)SCc2ccc(cc2)Br.Br CD00406 Cc1ccc(cc1)S(=O)(=O)NN=C2C[C@]3([C@@](C2)(CC(=NNS(=O)(=O)c4ccc(cc4)C)C3)C)C BTB14445 c1ccnc(c1)/C(=N/OC(=O)c2c(cccc2F)F)/N CD04831 CC(C)c1cc(c2ccccc2n1)c3ccccc3 BTB14477 c1ccc2c(c1)-c3c(cccc3C(=O)N)C2=O BTB13068 c1cc(ccc1NC(=O)/C=C/c2cc(ccc2Sc3ccc(cn3)C(F)(F)F)[N+](=O)[O-])Cl BTB09378 Cc1ccc(c2c1CCC2)OC BTB09379 CC1(CN(C1=O)C(=S)Nc2ccccc2OC)C BTB08204 Cc1cc(c(c2c1CCC2)OC)C#N BTB09395 CC(C)(C)c1cc2[nH]c(=N)[nH]c(=N)n2n1 BTB09381 COn1c2ccc3c(c2c4c1CCCC4)non3 BTB14049 c1ccc2c(c1)CC(N2)C(=O)O BTB14322 COc1ccc(c(n1)S(=O)(=O)c2ccccc2)[N+](=O)[O-] BTB09155 CCOC(=O)C(C(F)(F)F)(Nc1cccc(n1)C)NC(=O)c2cccnc2 BTB14254 c1ccc(cc1)CCCC(c2ccc(cc2)Cl)(c3ccc(cc3)Cl)O BTB12164 Cc1c(cc(c(n1)SCCNC(=O)c2ccc(cc2Cl)Cl)C#N)c3csc(n3)C BTB09484 c1ccc(cc1)CSc2ccc(cc2C#N)[N+](=O)[O-] BTB08186 CCCCCCCCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB13107 c1ccc(cc1)NC2=CC(N(C2=O)c3ccccc3)c4ccc(cc4)[N+](=O)[O-] BTB12160 CN1C2CCC1CC(=NOC(=O)c3ccco3)C2.Cl BTB14524 COC(=O)c1cc2ccccc2cn1 BTB09392 c1ccc(cc1)OC(=O)/C=C/c2cc(ccc2Sc3ccc(cn3)C(F)(F)F)[N+](=O)[O-] BTB09394 c1cc(cc(c1)Cl)C=C2C(=O)NC(=O)NC2=O CD00401 c1ccc2cc(ccc2c1)OCCC#N BTB09593 CC(C)(C)c1ccc(cc1)C(=O)Nc2nnc(s2)Sc3ccc(cc3C#N)[N+](=O)[O-] BTB08338 c1ccc2c(c1)[nH]c(n2)/C(=C/Nc3ccc(cc3)OC(F)(F)F)/C#N BTB08343 c1ccnc(c1)SCC(=O)c2ccc(cc2)OCc3ccc(cc3)[N+](=O)[O-] BTB09524 Cc1c2cc(c(=O)[nH]c2ccn1)C#N BTB09364 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 BTB14543 c1cc(sc1)C(C(=O)c2cccs2)O BTB09372 CCCCN(CCCC)CC(Cn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br)O BTB12254 c1ccc(cc1)c2c(=S)ssc2Sc3ccc(cn3)[N+](=O)[O-] BTB08239 c1cc(oc1)C=C2C(=O)NC(=S)NC2=O CD00509 CC1(C2CCC1(/C(=N/OC(=O)c3ccc(cc3)Cl)/C2)C)C BTB10345 CC(C)(C)NCC(Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl)O BTB12248 Cc1cc(n(n1)c2ccc(c(c2)Cl)Cl)O BTB09184 Cc1ccc(cc1)n2c(cc(n2)C)O BTB09185 CC(=C(C#N)C#N)c1ccccc1 BTB12102 Cc1c2c(c(sc2nc(n1)c3ccccc3)C(=O)C)N BTB09460 CC(=O)c1ccc(cc1)OCc2ccc(c(c2)Cl)Cl BTB09463 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N(C)S(=O)(=O)c3ccc(cc3)C BTB12199 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 BTB14533 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)c4ccco4 BTB14535 CC1(CC1C(=O)NN)C(=O)NN BTB14473 c1ccc(cc1)/C=N/C(c2ccccc2)C(c3ccccc3)NC(=O)c4ccccc4 BTB14474 CC(C)(C)c1ccc(cc1)C(=O)NCCSC(=O)c2ccc(cc2)C(C)(C)C BTB09429 COc1ccccc1C2C(CC(=O)O2)C(=O)O BTB09413 CN(c1ccc(cc1)Br)c2nc(=O)c3cccnc3s2 BTB08225 c1ccc(cc1)NC(=O)/C=C/c2cc(ccc2Sc3ccc(cn3)C(F)(F)F)[N+](=O)[O-] BTB09391 Cc1cc(n2c(n1)ncn2)O BTB10447 CCOC(=O)CC(=O)c1cccc(c1)[N+](=O)[O-] BTB10448 CN1C2CCC1CC(C2)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl BTB14568 Cc1cc(cc(c1OC(=O)c2ccc(cc2)[N+](=O)[O-])C)c3c4ccccc4c(=O)n(n3)C BTB08282 c1ccc(cc1)C2CC(=O)NC(=S)N2c3ccc(cc3)OC(F)(F)F BTB08296 c1c2c(cc(c1[N+](=O)[O-])Sc3nnc(s3)N)C(=O)NC2=O BTB08297 CC(C)CCN(CCC(C)C)S(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)N(CCC(C)C)CCC(C)C BTB12206 CC(=C)C(=O)Nc1ccc(nc1)Oc2ccc(cc2)F BTB08135 CC(=C)C(=O)Nc1cccnc1Oc2ccc(cc2)F BTB08136 CCOC(=O)C(=CN1CCC(CC1)C(c2ccccc2)c3ccccc3)C(=O)OCC BTB08138 COCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB12261 c1cc2c3c(c1)c(c(c(=O)n3CCC2)[N+](=O)[O-])O BTB09424 c1cc(c(nc1)Oc2ccc(cc2)Cl)[N+](=O)[O-] BTB09538 COc1ccc(cc1)Oc2c(cccn2)[N+](=O)[O-] BTB09539 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2ccc(cc2)C(C)(C)C BTB14526 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)OCc3ccccc3)c4ccccc4 BTB08187 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)OCc3ccccc3)c4cccc(c4)Cl BTB08189 CC(C)(C)NCC(Cn1c2ccccc2c3c1cccc3)O BTB12224 CCN(CC)CC(Cn1c2ccccc2c3c1cccc3)O BTB12225 c1ccc-2c(c1)Cc3c2c(ccc3)C(=O)N4CCCCC4 BTB13111 CCOC(=O)C/C(=N/Nc1ccccc1)/C(F)(F)F BTB09396 CC1(C2CCC(C2)(C1NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl)C)C BTB14552 Cc1cc(c(cc1Cl)C)S(=O)(=O)NC2C(C3CCC2(C3)C)(C)C BTB14553 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2cccc3c2cccc3 BTB14516 CN(C)/C=C(/c1nnnn1c2ccccc2)\C(=O)c3ccccc3Cl BTB12044 CCOC(=O)[C@@H](Cc1ccccc1)NS(=O)(=O)c2ccc(cc2)C BTB14453 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2ccc(cc2)C#N BTB14527 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)OC)c3ccccc3 BTB08183 c1cc(ccc1COc2ccc(cc2)C3SCCS3)[N+](=O)[O-] BTB09466 CCCCOS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)OCCCC BTB12213 c1cc(ccc1SCC(=O)Nc2ccc(c(c2F)F)F)Cl BTB08235 CC1(C2CCC(C2)(C1NS(=O)(=O)c3ccccc3C(=O)OC)C)C BTB14551 c1c2c(cc(c1N)Cl)C(=O)NC2=O BTB08300 CC(C)CCN(CCC(C)C)S(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)N(CCC(C)C)CCC(C)C BTB12207 CN1C2CCC1CC(=NOC(=O)c3ccc(cc3)Cl)C2.Cl BTB14521 CC(C)CCn1c2ccc(cc2c3c1ccc(c3)Cl)Cl BTB12237 c1ccc2c(c1)NC(O2)C3Nc4ccccc4O3 BTB14464 c1cc2c(cc1Br)c3cc(ccc3n2CC(CN4CCCCCC4)O)Br BTB12249 c1cc(ccc1NC(=O)CCC(=O)O)S(=O)(=O)N BTB12147 COC(=O)CCC(=O)Nc1ccc(cc1)S(=O)(=O)N BTB12148 CCCN(CCC)CC(Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl)O BTB12221 CC(C)(CNC(=S)Nc1ccccc1OC)C(=O)O BTB08226 c1cc(ccc1CSCC(=O)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl)Cl BTB09520 CCN(CC)C(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB13124 COc1ccccc1C2[C@@H](CC(=O)O2)C(=O)Nc3nnc(s3)C(F)(F)F BTB09431 CC1(C2CCC(C2)(C1NC(=O)c3cccs3)C)C BTB14558 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)OCc3ccccc3)c4ccc(c(c4)Cl)Cl BTB08190 CCOc1ccc(cc1)/N=c\2/c(c(ss2)SC)c3ccccc3 BTB08191 CSc1c(/c(=N/c2ccc(cc2)Cl)/ss1)c3ccccc3 BTB08192 COc1ccc(cc1)n2c3c(cccn3)c(=O)[nH]c2=S BTB08213 c1cc(c(cc1F)F)Oc2ccc(cn2)NS(=O)(=O)CS(=O)(=O)Nc3ccc(nc3)Oc4ccc(cc4F)F BTB08137 c1ccc(cc1)C2CCCC(C2=O)c3ccccc3 BTB14359 c1ccc(cc1)c2c(=S)ssc2SCC(=O)c3ccc(c(c3)F)F BTB08262 COc1ccccc1C2[C@H](CC(=O)O2)C(=O)Nc3nncs3 BTB09427 c1cc(ccc1C(=O)NCCSC(=O)c2ccc(cc2)F)F BTB09428 Cc1cc(c2ccccc2n1)SC BTB09602 CC1=C(C(C(=C(N1)C)C(=O)C)c2cccc(c2)[N+](=O)[O-])C(=O)C BTB09597 CCOC(=O)CSCC(=O)c1ccc(cc1)OCc2ccc(cc2)[N+](=O)[O-] BTB09525 c1cc(ccc1C(=O)COc2ccc(cc2)[N+](=O)[O-])OCc3ccc(c(c3)Cl)Cl BTB09527 c1cc(ccc1C(=O)CSCc2ccc(cc2Cl)Cl)OCc3ccc(c(c3)Cl)Cl BTB09529 CCCCN(CCCC)C(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB13126 c1cc2c(cc1c3csc(n3)N/C=N/O)CCC(=O)N2 BTB09432 c1cc-2c(cc1[N+](=O)[O-])C(=C(C#N)C#N)c3c2c(cc(c3)[N+](=O)[O-])C(=O)N4CCCCCC4 BTB13128 c1cc2c(cc1Cl)c(cc(=O)o2)O BTB14361 CCOC(=O)CNc1c(=O)[nH]c(=O)[nH]n1 BTB14365 CS(=O)(=O)NCc1ccc(cc1)Cl BTB08166 CS(=O)(=O)NCc1ccccc1 BTB08167 CN1C2CCC1CC(C2)NS(=O)(=O)c3ccc(cc3)F BTB14567 c1cc(ccc1NC(=O)Nc2nnc(s2)C(F)(F)F)OC(F)(F)F BTB08288 CC(C)(CCSc1ccc(cn1)[N+](=O)[O-])O BTB08289 Cc1cc(cc(c1OC(=O)Nc2ccc(cc2)OC(F)(F)F)C)c3c4ccccc4c(=O)n(n3)C BTB08295 c1ccc(c(c1)[N+](=O)[O-])OCCOc2ccccc2[N+](=O)[O-] BTB12337 CCOC(=O)Cc1c(c([nH]c1C(=O)OCC)C)C(=O)OCc2ccccc2 BTB10373 Cc1c(c(c([nH]1)C(=O)OCc2ccccc2)CCC(=O)OC)C(=O)OC(C)(C)C BTB10374 c1ccc(c(c1)N)Nc2c(cn(c(=O)n2)Cc3ccc(c(c3)Cl)F)C#N BTB08242 c1cc2c(=O)[nH]c(=S)n(c2nc1)c3ccc(cc3)Br BTB08215 CC1(C2CCC1(C(C2)N)C)C BTB10381 Cc1ccc(cc1)N(CC=C)c2nc(=O)c3cccnc3s2 BTB08216 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CSc4ccc(cc4)Cl BTB09505 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CSc4ccccn4 BTB09506 CCOC(=O)c1c(c(c([nH]1)Cc2c(c(c([nH]2)C(=O)OCC)C)C)C)C BTB09301 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)c2n[nH]nn2)OC(=O)C)OC(=O)C)OC(=O)C BTB12047 CC(=O)Nc1ccc(c(c1)C(=O)CC(=O)c2ccccc2)O BTB14487 c1cc2c(cc1Br)c3cc(cc(c3n2CC(CN4CCCCC4)O)Br)Br BTB12222 CC(C)(C)c1nnc(s1)N2C(=O)C(N(C2=O)C)c3ccccc3 BTB08273 C1CCC(CC1)N2CC(=C(C2=O)O)C(=O)N BTB09317 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C)C CD04933 c1ccc(c(c1)Oc2c(cccn2)[N+](=O)[O-])F BTB08077 Cn1c2ccccc2nc1c3ccccc3 BTB14439 c1ccc(cc1)/C=C/C=N/NC(=S)N BTB11629 c1ccc(cc1)Oc2ccc(cc2)OS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl BTB14500 Cc1c(c(=O)n(n1C)c2ccccc2)/N=C/3\C=CC(=O)C(=C3)C BTB12196 c1ccc2c(c1)c3ccccc3n2CC(CN4CCCCC4)O BTB12246 c1ccc(cc1)c2c(=S)ssc2SCC(=O)c3cccc(c3)[N+](=O)[O-] BTB08264 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)c4cccc5c4cc[nH]5 BTB14547 CS(=O)(=O)N(Cc1ccc(cc1)Cl)c2c(cc(cn2)C(F)(F)F)Cl BTB08168 c1ccc(cc1)NC(=O)c2cccc3c2-c4ccccc4C3 BTB14448 c1ccc(cc1)/N=c/2\[nH]c(=N)[nH]c(=O)n2c3ccccc3 BTB11634 c1ccc(cc1)CC(C#N)C(=O)O BTB11640 CCCN(c1ccc(cc1)C)c2nc(=O)c3cccnc3s2 BTB08212 c1ccc(cc1)S(=O)(=O)NCc2cccnc2 BTB08164 c1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)Cl BTB08165 c1c2c(cc3c1c(=O)n(c3=O)CCO)c(=O)n(c2=O)CCO BTB12197 c1ccc(cc1)S(=O)(=O)N(Cc2ccc(cc2)Cl)c3c(cc(cn3)C(F)(F)F)Cl BTB08169 CN1C2CCC1CC(C2)NS(=O)(=O)c3ccc(cc3)C#N BTB14570 CN1C2CCC1CC(C2)NS(=O)(=O)c3cccc(c3)C(F)(F)F BTB14571 CC(C)(C)c1ccc(c(c1)/C(=N/O)/c2ccccc2)O BTB10339 c1cc(c(c(c1)F)C(=O)ON=C(c2cccs2)c3cccs3)F BTB10341 CCCCNC(=O)Nc1nnc(s1)C(C)(C)C BTB08301 Cc1cc(cc(c1OCC(=O)NNC(=O)Nc2ccc(cc2)Cl)C)c3c4ccccc4c(=O)n(n3)C BTB08304 CCOC(=O)CSCC(=O)c1ccc(cc1)OCc2ccc(c(c2)Cl)Cl BTB09562 c1cc(ccc1C(=O)COc2ccc(cc2)Cl)OCc3ccc(c(c3)Cl)Cl BTB09563 c1ccc2c(c1)c3c([nH]2)-c4c(non4)CC3 BTB14393 CC1(CN(C1=O)C(=S)Nc2ccc(cc2F)F)C BTB08205 c1ccc(cc1)NCCNc2ccccc2 BTB09325 CC1=C(C(=O)NC1)c2ccccc2 BTB09329 CC1(C(=O)N(C(C(=O)N1O)(C)C)O)C BTB14396 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)OC)c3ccc(c(c3)Cl)Cl BTB08174 c1cc(c(c(c1)Cl)C=C2C(=O)NC(=O)NC2=O)Cl CD00395 CC(=O)NC(CO)C(=O)c1ccc(cc1)[N+](=O)[O-] BTB09353 Cc1c(nnn1c2ccccc2C#N)C(=O)C CD05121 Cc1c(nnn1c2cc(ccc2Cl)C(F)(F)F)C(=O)C CD05124 Cc1cccc(c1)NC(=O)N2CCN(CC2)c3cccc4c3cc[nH]4.Cl BTB14563 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)Nc4ccc(c(c4)Cl)Cl.Cl BTB14564 CCOC(=O)N1CCCN=C1NNc2cc(ccc2C)F BTB08245 CCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB13103 CCCCCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB13106 COc1ccccc1C2[C@@H](CC(=O)O2)C(=O)Oc3cccc(c3)C(F)(F)F BTB09434 CC1=C(C(N(C1)C(=O)C)O)C#N BTB09333 CC(C)CCN(CCC(C)C)CC(Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl)O BTB12252 Cc1c(cc(c(n1)SCCNS(=O)(=O)c2ccc(cc2Cl)Cl)C#N)c3csc(n3)C BTB09494 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)CCC(=O)O)C BTB12149 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc(cc3)NC(=O)CCC(=O)O BTB12151 CN(C)c1c(cc(cc1F)C#N)F CD04944 CCOC(=O)C1=C(C(=O)N(C1)Cc2ccccc2)O BTB09318 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl BTB14544 CCOC(=O)NC1=Nc2ccccc2NC=C1C#N BTB08207 c1cc2c3c(c1)c4c(c(cc(=O)o4)O)c(=O)n3CCC2 BTB09370 CC1(C2CCC1(/C(=N/OC(=O)c3c(cccc3F)F)/C2)C)C BTB10344 CCCCN(CCCC)CC(Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl)O BTB12228 CCCSc1nc(=O)c2cccnc2n1c3ccc(cc3)OC BTB08221 c1cnc(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)Cl BTB14502 c1cc(c(cc1Cl)NC(=O)CC2C(=O)N=C(S2)NC3CC4CC3C=C4)Cl CD04888 c1cc(ccc1NC(=O)CC2C(=O)N=C(S2)NC3CC4CC3C=C4)Cl CD04889 C1C2(CSC(=N2)N)N=C(S1)N CD04932 Cc1ccc(cc1)S(=O)(=O)N(CCC#N)Cc2ccco2 BTB08199 COc1ccc(cc1OC)S(=O)(=O)N(CCC#N)Cc2ccco2 BTB08201 CC1(CN(C1=O)C(=S)Nc2cccc(c2)Cl)C BTB08203 CCOC(=O)[C@H](Cc1ccccc1)NS(=O)(=O)c2ccc(cc2)C BTB14452 CCCN(CCC)CC(Cn1c2ccccc2c3c1cccc3)O BTB12242 CCN(CC)CC(Cn1c2ccc(cc2c3c1ccc(c3)Br)Br)O BTB12244 c1ccc2c(c1)c3ccccc3n2CC(CN4CCCCCC4)O BTB12247 CSC(=C(C#N)C#N)NCC=C BTB12104 COc1cc(ccc1O)C=C2C(=O)NC(=O)NC2=O CD00387 c1ccc2c(c1)c(c(s2)C(=O)Oc3ccc(cc3)/C(=C/c4ccc(cc4)C(F)(F)F)/C#N)Cl BTB08160 c1cc(oc1)CN(CCC#N)C(=O)Nc2ccc(cc2)OC(F)(F)F BTB08196 c1cc(oc1)CN(CCC#N)C(=O)Nc2ccc(cc2)Cl BTB08197 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)c4cccs4 BTB14534 CC1=CC(=O)C(=CC1=O)CCC2=CC(=O)C(=CC2=O)C BTB14447 CC(C)(C)NCC(Cn1c2ccc(cc2c3c1ccc(c3)Br)Br)O BTB12236 c1cc2c(cc1Br)c3cc(ccc3[nH]2)Br BTB12239 Cc1cc(cc(c1OC(=O)c2ccc(cc2)Cl)C)c3c4ccccc4c(=O)n(n3)C BTB08279 c1ccc(cc1)COc2cccc(c2)C=C3C(=O)NC(=O)NC3=O CD00389 CN(C)c1ccc(cc1)C=C2C(=O)NC(=O)NC2=O CD00391 CC1(CN(C(=S)NC1=O)c2ccccc2OC)C BTB08209 CC(C)(C)NC(=O)/C=C/c1cc(ccc1Sc2ccc(cn2)C(F)(F)F)[N+](=O)[O-] BTB09390 CN(C)CC(Cn1c2ccc(cc2c3c1ccc(c3)Cl)Cl)O BTB12232 c1cc2c(cc1Cl)c3cc(ccc3n2CC(CN4CCOCC4)O)Cl BTB12233 CCN(CC)C(=O)c1c(c(c([nH]1)C)C)C BTB09341 c1ccc(cc1)OC(=O)c2cc(cc3c2-c4ccc(cc4C3=O)[N+](=O)[O-])[N+](=O)[O-] BTB12260 c1cc(cc(c1)NC(=O)CSc2c(c(c(c(c2F)F)C(=O)O)F)F)C(F)(F)F BTB08337 c1cc(cc(c1)[N+](=O)[O-])C(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 BTB14536 Cc1cc(ccc1Oc2c(cccn2)[N+](=O)[O-])Cl BTB09540 c1c(cnc(c1Cl)O)C(F)(F)F BTB09546 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)c4ccc(cc4)Cl BTB14539 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCCC(C2)C CD00639 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)NC4CCCCC4 BTB13181 CCOC(=O)/C(=C/Nc1cccnc1Oc2ccc(c3c2CCC3)C)/C#N BTB09503 CN(C)c1c(cc(cc1F)C(=O)NCc2ccccc2)F CD05092 CN(Cc1ccccc1)Cc2nc(no2)/C=C/c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04856 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)S(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F BTB08154 c1ccc(cc1)CNS(=O)(=O)c2ccccc2 BTB08156 CSc1c(/c(=N/c2ccc(cc2)OC(F)(F)F)/ss1)c3ccccc3 BTB08193 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2ccc(cc2)Cl BTB14528 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])Cl)Cl CD05115 c1cc(oc1)C(=O)/C(=C/c2ccc(s2)[N+](=O)[O-])/C#N CD05196 c1ccc2c(c1)c(nc3n2nnc3C(=O)N4CCOCC4)N CD05125 c1cc(oc1)C(=O)/C(=C/c2cccs2)/C#N CD05204 CCOC(=O)C(=CNc1cccnc1Oc2ccc(c3c2CCC3)C)C(=O)OCC BTB09502 c1cc(ccc1C(=O)OC2CN3CCC2CC3)Cl BTB14606 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)F)NC(=O)OCC BTB13195 CCOC(=O)C(C(F)(F)F)(NCc1ccccc1)NC(=O)OCC BTB13197 c1cc(ccc1NC(=O)Nc2cc(cnc2)C(F)(F)F)OC(F)(F)F BTB08317 Cc1cc2[nH]c(=N)[nH]c(=N)n2n1 BTB09383 c1cc2c(cc1Br)c3cc(cc(c3n2CC(CN4CCOCC4)O)Br)Br BTB12258 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)N4CCCCCC4 BTB12259 CCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB13115 CCCCCc1cnc(nc1)c2ccc(cc2)C#N BTB09572 COc1cc(ccc1N2CCCC2)[N+](=O)[O-] BTB09574 c1cc(ccc1N/N=C(\C#N)/C(=S)N)Cl CD04975 CCC1(CCCCN(C1=O)C)c2cccc(c2)OC(=O)Nc3ccc(cc3)OC(F)(F)F BTB14605 COc1ccc(cc1OC)CCNC(=O)c2cccs2 BTB14608 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)OCC BTB13199 COc1ccccc1N2CCN(CC2)Cc3ccc4ccccc4c3 BTB14598 COc1ccccc1C2CCN(CC2)Cc3ccc(cc3Cl)Cl BTB14599 c1cc(ccc1S(=O)(=O)CS(=O)(=O)c2ccc(cc2)Cl)Cl CD05017 COc1ccccc1C2CCN(CC2)Cc3ccc(c(c3)Cl)Cl BTB14601 Cc1c(cccc1[N+](=O)[O-])NCC(=O)N(c2ccccc2)C3CCCCC3 BTB14607 COc1ccccc1N2CCN(CC2)Cc3cccc4c3cccc4 BTB14614 CC1(C2CCC1(C(C2)NC(=O)c3cccc(c3)C(F)(F)F)C)C BTB10383 c1cc(ccc1COc2ccc(cc2)c3csc(n3)N)[N+](=O)[O-] BTB09523 c1cc(ccc1c2csc(n2)N)OCc3ccc(c(c3)Cl)Cl BTB09526 c1cc(ccc1COc2ccc(cc2)C(=O)CSCc3ccc(cc3Cl)Cl)[N+](=O)[O-] BTB09528 CN1C2CCC1CC(=NOC(=O)C3CCCCC3)C2.Cl BTB14522 CN1C2CCC1CC(=NOC(=O)c3ccc(cc3)[N+](=O)[O-])C2.Cl BTB14523 CC(C)(C)c1ccc(cc1)OC(=O)C2c3ccccc3Oc4c2cccc4 BTB10397 CC(=O)Nc1ccccc1OCCOc2ccccc2NC(=O)C BTB12338 c1cc(oc1)/C(=N/OC(=O)c2cccs2)/O CD05019 c1cc(ccc1SCC#CCSc2ccc(cc2)Cl)Cl CD05018 COc1ccccc1C2CCN(CC2)Cc3ccccc3Cl BTB14600 c1ccc2cc(ccc2c1)OC(=O)C3c4ccccc4Oc5c3cccc5 BTB10400 c1c(cnc(c1Cl)/N=C/N2CCOCC2)C(F)(F)F BTB10406 CCCCCCCC\1CCC/C1=N/OC(=O)c2cccc3c2cccc3 BTB10387 CC(C)(C)c1cc2cc(cc3c2c(c1)CC3)C(C)(C)C BTB10389 c1c(cnc(c1Cl)/N=C/N2CCCCC2)C(F)(F)F BTB10408 CN(C)CC1COC(=O)C1=O.Cl BTB10411 Cc1c(c(=O)n(n1C)c2ccccc2)N=C3C=C(C(=O)C(=C3)C(C)C)C(C)C BTB12194 c1ccc(cc1)OS(=O)(=O)c2ccc-3c(c2)Cc4c3ccc(c4)S(=O)(=O)Oc5ccccc5 BTB12209 Cn1c(c(c2ccc(cc2c1=O)[N+](=O)[O-])C#N)N BTB12296 c1cc(ccc1c2nc(on2)CN3CCOCC3)Cl CD02881 c1cc(ccc1c2nc(on2)CN3CCCC3)Cl CD02883 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)CC#N CD02893 Cc1c(c(c(c(c1C)C)CSc2nnc(n2C)/C(=C/c3cccs3)/C#N)C)C CD02899 CN1CCN(CC1)/C=N/c2c(cc(cn2)C(F)(F)F)Cl BTB10407 CC1CCN(CC1)Cc2nc(no2)c3ccc(cc3)Cl CD02910 COCCCNC(=S)N/N=C/c1ccc2ccccc2c1 CD02912 c1cc(ccc1F)S(=O)(=O)NOc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] BTB09584 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)COc2ccc(cc2)SC(F)(F)F BTB08349 c1cc(cc(c1)F)NC2=NC(=O)C(S2)CC(=O)Nc3cc(ccc3Cl)Cl CD04894 c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3 CD04897 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2ccc(cc2)F BTB14529 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 BTB14531 c1ccc(cc1)C(=O)CSc2c(c(sn2)SCC(=O)c3ccccc3)C#N CD00464 Cc1ccc(cc1)n2c3c(cccn3)c(=O)nc2SC BTB08217 CCCCCCCCCCOC(=O)c1cc(cc\2c1-c3ccc(cc3/C2=N\O)[N+](=O)[O-])[N+](=O)[O-] BTB13158 c1c(cnc(c1Cl)C(=O)NNC(=O)c2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F BTB09622 COc1cccc(c1O)/C=N/CCCC2C=NNC2=O CD02895 Cc1ccccc1NC(=S)NNC(=O)c2ccccc2n3cccc3 CD03000 c1ccc(c(c1)NC(=O)CC2C(=O)N=C(S2)NC3CC4CC3C=C4)Cl CD04887 COc1ccc(cc1)NC(=O)C(Cl)Cl CD04890 Cc1cc(cc(c1O)C)C(=O)c2ccccc2C(=O)OC BTB08277 c1ccc2c(c1)C(c3ccccc3O2)C(=O)Oc4ccc(cc4)Br BTB10395 CCOc1ccc(cc1)C=C2C(=O)NC(=O)NC2=O CD00434 CCOc1ccccc1C=C2C(=O)NC(=O)NC2=O CD00456 Cc1ccc(n1c2cccc(c2)[N+](=O)[O-])C BTB10409 c1cc(ccc1c2ccc(o2)C(=O)O)Cl BTB13086 c1cc(ccc1c2ccc(o2)C(=O)O)[N+](=O)[O-] BTB13087 c1cc(cc(c1)C(F)(F)F)C(c2ccc(cc2)C(F)(F)F)O BTB13088 Cc1cc(c(c(c1)O)CN(C)C)C BTB10412 Cc1cc(cc(c1OS(=O)(=O)c2cc(ccc2Cl)Cl)C)c3c4ccccc4c(=O)n(n3)C BTB08283 c1ccc2c(c1)[nH]c(n2)C(C#N)C(=O)c3ccco3 BTB12316 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2C)c3c4ccccc4c(=O)n(n3)C)C BTB08284 COc1cccc(c1OC)C=C2C(=O)NC(=S)NC2=O CD00550 c1cc(c(cc1C=C2C(=O)NC(=S)NC2=O)O)O CD00553 CCCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB13105 COCCCNC1=NC(=O)C(S1)CC(=O)Nc2ccc(cc2)Cl CD04879 COCCCNC1=NC(=O)C(S1)CC(=O)Nc2ccccc2Cl CD04885 COc1cc(cc(c1OC)OC)C=C2C(=O)NC(=S)NC2=O CD00556 CCOc1ccc(cc1C=C2C(=O)NC(=S)NC2=O)Br CD00558 c1cc(ccc1C=C2C(=O)NC(=S)NC2=O)O CD00569 CC(=O)Nc1c(cc(cc1F)Br)F CD04908 c1ccc(cc1)/C=C/C=C2C(=O)NC(=S)NC2=O CD00513 c1ccc2c(c1)C(=CC(=O)C2=O)Nc3ccc(cc3)O BTB13089 c1ccc2c(c1)C(=CC(=O)C2=O)Nc3cccc(c3)O BTB13090 Cc1cc(cc(c1OCC(=O)NNC(=O)Nc2ccccc2)C)c3c4ccccc4c(=O)n(n3)C BTB08303 Cc1cc(cc(c1OCC(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F)C)c3c4ccccc4c(=O)n(n3)C BTB08305 CCCN(CCC)CC(Cn1c2ccc(cc2c3c1ccc(c3)Br)Br)O BTB12240 Cc1cc(cc(c1OCC(=O)NNC(=O)c2ccc(cc2)Cl)C)c3c4ccccc4c(=O)n(n3)C BTB08307 c1cc(ccc1COc2ccc(cc2)/C=C\3/C(=O)NC(=S)S3)[N+](=O)[O-] BTB09456 c1cc(c(cc1C(=O)Nc2nnc(s2)Sc3ccc(cc3C#N)[N+](=O)[O-])Cl)Cl BTB08339 c1cc(ccc1OCC(=O)NN)SC(F)(F)F BTB08347 c1cc(ccc1C(=O)NNC(=O)COc2ccc(cc2)SC(F)(F)F)Cl BTB08348 CC(=O)c1ccc(cc1)OCc2ccc(cc2)[N+](=O)[O-] BTB09465 c1cc(ccc1C2SCCS2)OCc3ccc(c(c3)Cl)Cl BTB09467 C#CCSc1nc(=O)c2cccnc2n1c3ccc(cc3)Br BTB08218 CCc1cc2c(cc1C(=O)CSc3c(c(sn3)SCC(=O)c4cc5c(cc4CC)C(CCC5(C)C)(C)C)C#N)C(CCC2(C)C)(C)C CD00469 CNc1c(cccn1)[N+](=O)[O-] BTB09509 Cc1nc(c(o1)c2ccccc2)c3ccc(cc3)[N+](=O)[O-] BTB09510 c1cc(sc1)C(=O)C2CC(=O)OC2 BTB09515 c1cc(ccc1C(=O)NNC(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl BTB09578 C1C2C3[C@H](C4C2C5C1C3[C@@H](C45)O)O BTB12413 CN1C2C[C@@H](CC1CC2)NC(=O)Nc3c(cc(cc3)F)F.Cl BTB14597 Cc1ccc(cc1)CN2CCC(CC2)c3ccccc3OC BTB14602 COc1ccccc1C2CCN(CC2)Cc3ccc4ccccc4c3 BTB14604 CN1C2C[C@@H](CC1CC2)NC(=O)Nc3ccc(cc3)Cl.Cl BTB14594 Cc1cc(cnc1Sc2ccc(cc2)Cl)[N+](=O)[O-] BTB09626 COc1ccc(cc1)NC(=O)c2ccc(o2)CSc3ccc(cc3)Cl CD05024 CC1(C2CCC(C2)(C1NS(=O)(=O)c3ccc(cc3)C#N)C)C BTB14554 CCNc1ccc(cc1)C(=O)O BTB10315 c1ccc(c(c1)N)SCc2nc(no2)/C=C/c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04854 CCCCN1CC(=C(C1=O)O)C(=O)OCC BTB09319 Cc1ccc(cc1)S(=O)(=O)NCC(=O)OCc2ccccc2 BTB09327 CC1(C2CCC(C2)(C1NC(=O)c3ccc(cc3)[N+](=O)[O-])C)C BTB14559 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)Nc4ccc(cc4)Cl.Cl BTB14566 CCOc1c(c(c([nH]1)/C=C\2/C(=C(C(=N2)OCC)CC(=O)OC)C(=O)OC)C(=O)OC)CC(=O)OC BTB09334 C1[C@H](C2C3C1C4C[C@@H](C2C4C3)O)O BTB12414 CN(C)c1c(cc(cc1F)C(=O)N)F CD04945 c1cc-2c(cc1[N+](=O)[O-])C(=NO)c3c2ccc(c3)[N+](=O)[O-] BTB13145 c1cc-2c(cc1Br)C(=NN)c3c2ccc(c3)Br BTB13148 CCOCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB13149 Cc1ccc(c(c1)[N+](=O)[O-])OS(=O)(=O)c2cc(ccc2OC)OC CD05028 c1ccc2c(c1)C(=O)N(S2(=O)=O)CCCCN3C(=O)c4ccccc4S3(=O)=O BTB10348 c1ccnc(c1)SC/C=C/CSc2ccccn2 CD05103 CN(C)c1c(cc(cc1F)C(=O)NCCc2ccc(c(c2)OC)OC)F CD05093 CN(C)c1c(cc(cc1F)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F CD05094 c1cc(ccc1CO)OCc2ccc(c(c2)Cl)Cl BTB09519 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)C4CCCCC4 BTB14550 CC1(C2CCC(C2)(C1NC(=O)c3cccc(c3)[N+](=O)[O-])C)C BTB14555 CC1(C2CCC(C2)(C1NC(=O)C3CCC3)C)C BTB14556 c1cc(ccc1SC/C=C/CSc2ccc(cc2)Cl)Cl CD05099 CC(C)(C)c1ccc(cc1)NS(=O)(=O)c2ccc(c(c2)OC)OC CD05112 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])Cl CD05118 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)Nc4ccc(cc4)Br.Cl BTB14562 CC1CCC(C(C1)NC(=O)c2cccc3c2cccc3)C(C)C BTB10377 CC1CCC(C(C1)N(Cc2ccccc2)C(=O)c3cccc4c3cccc4)C(C)C BTB10379 CC1(C2CCC1(C(C2)NC(=O)c3ccc(cc3)Cl)C)C BTB10382 c1cc(ccc1C(=O)CSc2c(c(sn2)SCC(=O)c3ccc(cc3)[N+](=O)[O-])C#N)[N+](=O)[O-] CD00466 c1cc(ccc1NC(=O)c2ccc(o2)CSc3ccc(cc3)Cl)F CD05023 c1ccc2c(c1)C(=O)N(S2(=O)=O)CCCCCN3C(=O)c4ccccc4S3(=O)=O BTB10384 Cn1c2ccccc2nc1SC BTB14440 CN(C)CC(Cn1c2ccc(cc2c3c1ccc(c3)Br)Br)O BTB12241 c1ccc2c(c1)c3ccccc3n2CC(CN4CCOCC4)O BTB12245 Cc1cc(cc(c1OCC(=O)NNS(=O)(=O)c2cc(ccc2Cl)Cl)C)c3c4ccccc4c(=O)n(n3)C BTB08312 CCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB12272 C/C(=N/O)/CCc1ccc(c(c1)OC)OCc2ccc(cc2Cl)Cl BTB11052 CN1C2C[C@@H](CC1CC2)NC(=O)Nc3ccc(cc3)OC(F)(F)F.Cl BTB14593 CN(C)Cc1cc(c(cc1O)CN(C)C)O BTB10421 CCOC(=O)N1CCCN=C1NNc2cc(ccc2OC)Cl BTB08252 CC1(CN(C(=NC1=O)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)c3ccccc3OC)C BTB08256 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)S(=O)(=O)c4cccc(c4)C(F)(F)F BTB08152 CN(C)C(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB13108 COc1ccccc1C2[C@@H](CC(=O)O2)C(=O)NN BTB09516 CC1(CN(C(=S)N(C1=O)C(=O)c2cccc(c2)C(F)(F)F)c3ccccc3OC)C BTB08259 c1ccc(cc1)c2c(=S)ssc2SCC(=O)c3ccc(cc3)Cl BTB08261 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=C/c2nc(on2)CN3CCCCC3 CD04866 CC1CCC(C(C1)NC(=O)c2cccc(c2)C(F)(F)F)C(C)C BTB10454 CCCCCC(=O)c1ccc-2c(c1)Cc3c2cccc3 BTB10460 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)C#N BTB10463 c1cc(ccc1c2csc(n2)C/C(=N/O)/N)F CD03006 Cc1c(c(c(c(c1C)C)CSc2nnc(n2C)/C(=C/c3c(cccc3Cl)Cl)/C#N)C)C CD02898 CC(=O)n1c2ccc(cc2c3c1ccc(c3)Br)Br BTB12230 CC(C)CCN(CCC(C)C)CC(Cn1c2ccccc2c3c1cccc3)O BTB12231 CCN(CC)CC(Cn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br)O BTB12256 c1cc2c(cc1Br)c3cc(ccc3n2CC(CN4CCOCC4)O)Br BTB12257 CC(C=C1C(=O)NC(=S)NC1=O)c2ccccc2 CD00618 c1ccc-2c(c1)Cc3c2c(ccc3)C(=O)N4CCOCC4 BTB13112 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)OC(=O)c4ccc(cc4)C#N BTB10467 c1cc(ccc1C(=O)CSc2c(c(sn2)SCC(=O)c3ccc(cc3)F)C#N)F CD00491 c1ccc(cc1)C2(C(=O)c3ccccc3N(C2=O)c4ccccc4)[N+](=O)[O-] BTB10445 CCOC(=O)c1cc2cc(cc(c2oc1=O)Br)Br BTB09656 CN(C)NC(=S)Nc1ccc(cc1)S(=O)(=O)N2CCCCC2 CD00589 COc1cc(c(c(c1)OC)C=C2C(=O)NC(=S)NC2=O)OC CD00594 Cc1cc(ccc1Cl)C(=O)CSc2c(c(c(c(c2F)F)C(=O)O)F)F BTB08328 c1cc(c(cc1[N+](=O)[O-])C#N)Sc2nnc(s2)N BTB08332 CCSc1c(cccn1)C(=O)NOc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] BTB09587 c1cc(ccc1NC(=O)NNC(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl BTB09589 c1ccc(cc1)CNc2cccc(c2)[N+](=O)[O-] BTB09591 c1ccc(cc1)CNC(=O)c2cccc-3c2C(=O)c4c3cccc4 BTB13174 c1cc(ccc1N/N=C(\C#N)/C(=S)N)F CD04960 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)c4ccc(cc4Cl)Cl BTB09497 c1cc(ccc1C#N)NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00586 CCCCCOc1ccc(cc1)c2ccc(cc2)Br BTB09576 CC(C)c1ccc(cc1)/N=C/c2ccc(cc2)NC(=O)C CD00634 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCC(CC2)C CD00638 CCCN(CCC)C(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB13125 c1ccc\2c(c1)-c3ccc(cc3/C2=N\O)I BTB13161 C[C@@]12CCC(=O)[C@@]1(CCC2=O)C BTB14444 c1cc(c(c(c1NC(=O)CCCC(=O)O)F)F)F BTB14708 Cc1ccc(c(c1)Br)OC(=O)c2cccc(c2)[N+](=O)[O-] BTB14574 Cc1ccc(c(c1)Br)OC(=O)c2ccc(cc2)[N+](=O)[O-] BTB14575 c1ccc(cc1)CNC(=O)c2c(cc(cn2)C(F)(F)F)Cl BTB09535 c1cc(c(nc1)Oc2ccc(cc2Cl)Cl)[N+](=O)[O-] BTB09537 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)[N+](=O)[O-] BTB09541 Cc1ccc(c(c1)Br)OS(=O)(=O)c2ccc(cc2)Cl BTB14580 c1ccc2c(c1)-c3cccc(c3C2=O)C(=O)N4CCCCCC4 BTB13173 Cn1c(cc(=O)n(c1=O)C)Nc2ccccc2 BTB13233 CCNC(=O)c1c(onc1c2c(cccc2Cl)Cl)C CD05280 c1ccc(cc1)Oc2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl BTB14631 c1cc(ccc1C(=O)OC2CN3CCC2CC3)[N+](=O)[O-] BTB14638 Cc1ccc(cc1)C(=O)OC2CN3CCC2CC3 BTB14639 Cc1ccc(c(c1)Br)OC(=O)c2ccc(cc2)Cl BTB14577 Cc1ccc(c(c1)Br)OS(=O)(=O)c2cc(c(cc2C)Cl)C BTB14579 Cc1cccc(c1C)Oc2c(cccn2)N BTB09636 c1ccc(cc1)C(=O)OC2CN3CCC2CC3 BTB14642 Cc1ccc(c(c1)Br)OS(=O)(=O)c2ccc(cc2)C#N BTB14582 COc1ccccc1N2CCN(CC2)Cc3ccccc3Cl BTB14587 c1ccc(c(c1)N)SC/C=C/CSc2ccccc2N CD05102 c1ccc(cc1)OCC#CC#CCOc2ccccc2 CD05104 CC(C)(C)c1ccc(cc1)NS(=O)(=O)c2cc(ccc2OC)OC CD05113 COc1ccc(cc1C=C2C(=O)NC(=O)NC2=O)Br CD00428 c1cc(cc(c1)[N+](=O)[O-])C=C2C(=O)NC(=O)NC2=O CD00431 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC2CC3CCC(C2)N3C BTB14572 Cc1ccc(c(c1)Br)OC(=O)c2ccc(cc2)C(C)(C)C BTB14573 c1c2c(cc3c1OCCO3)nc([nH]2)S BTB10427 COc1cc(nc(n1)N)OC BTB09643 Cn1c2c(c3c(c1=O)cc4cc(ccc4n3)OC)c(=O)n(c(=O)n2C)C BTB14651 c1cc(ccc1COc2ccc(cc2)C3SCCS3)F BTB09558 c1cc(ccc1C(=O)CSCc2ccc(c(c2)Cl)Cl)OCc3ccc(c(c3)Cl)Cl BTB09559 COC(=O)c1cccc2c1[nH]cc2 BTB12321 c1ccc2c(c1)-c3cccc(c3C2=O)N BTB12322 Cn1c(=O)cc(c2c1n(c(=O)n(c2=O)c3ccccc3)c4ccccc4)N5CCOCC5 BTB14653 c1cc2cccc(c2c(c1)C(=O)O)Br BTB12326 c1cc2c(cc1C=C3C(=O)NC(=S)NC3=O)OCO2 CD00608 c1ccc2c(c1)C(c3ccccc3O2)C(=O)Oc4ccc(cc4)Sc5ccc(cc5)OC(=O)C6c7ccccc7Oc8c6cccc8 BTB10392 COc1ccc(cc1COC(=O)C2c3ccccc3Oc4c2cccc4)Br BTB10391 CCCc1ccccc1NCc2cccc3c2cccc3 BTB14615 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C)NC(=O)OCC BTB13193 c1cc(=O)oc2c1cc(cc2)[N+](=O)[O-] BTB12331 c1cc(ccc1CO)OCc2ccc(cc2)[N+](=O)[O-] BTB09554 c1cc(ccc1COc2ccc(cc2)c3csc(n3)N)F.Br BTB09555 COc1cc(c(c(c1)OC)/C=C/2\c3ccccc3NC2=O)OC CD00750 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)Cl)NC(=O)c2cccc(c2)Cl BTB13210 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)F)NC(=O)c2cccc(c2)Cl BTB13213 c1cc(sc1)C(=O)CC#N CD05218 c1cc(sc1)/C=C(\C#N)/C(=O)c2cccs2 CD05220 c1ccnc(c1)SCC(=O)c2ccc(cc2)OCc3ccc(cc3)F BTB09565 Cc1cccc(c1C)Oc2c(cccn2)[N+](=O)[O-] BTB09567 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)c2cccc(c2)Cl BTB13215 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)OC(F)(F)F)NC(=O)c2cccc(c2)Cl BTB13217 c1ccc(cc1)c2ccc(cc2)OC(=O)C3c4ccccc4Oc5c3cccc5 BTB10393 c1ccc2c(c1)C(c3ccccc3O2)C(=O)Oc4cc(c(cc4Cl)Cl)Cl BTB10396 Cc1nc2c3ccccc3ccc2s1 BTB12365 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCCOC CD05284 COC(=O)/C(=C\Nc1ccc(nc1)Sc2cc(ccc2Cl)Cl)/NC(=O)c3ccccc3 BTB09697 CC(c1ccc2ccccc2c1)O BTB10505 c1cc(sc1)C2C(=C(OC(=C2C#N)N)c3cccs3)C#N CD05223 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)OC(=O)c4ccc(cc4)CCC BTB10470 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCCCC2 CD00640 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCCC2 CD00641 CN(C)c1c(cc(cc1F)c2[nH]nnn2)F CD05059 COc1cccc(c1)NC(=S)Nc2ccc(cc2)O CD00688 c1ccc(cc1)c2cc(on2)c3ccccc3 BTB10419 CC(C)(CCO)NC(=S)Nc1cccc(c1)OC CD00692 c1cc(cc(c1)NC(=S)Nc2cccc(c2)C(F)(F)F)C(F)(F)F CD00691 COCCCNC(=S)NNC(=S)Nc1cccc(c1)C(F)(F)F CD02874 CCOC(=O)CSCC(=O)c1ccc(cc1)OCc2ccc(cc2)F BTB09615 CC1(c2ccccc2-c3c1cccc3)C BTB10506 CN(C)c1c(cc(cc1F)/C(=N/O)/N)F CD05056 c1ccc(c(c1)NC(=O)Nc2ccc(o2)CSc3ccc(cc3)Cl)F CD05070 COc1cccc(c1)NC(=S)NC(Cc2ccccc2)c3ccccc3 CD00686 COc1cccc(c1)NC(=S)NCCO CD00687 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1F)F)F)NC(=O)c2cccc(c2)Cl BTB13218 Cc1ccc(cc1)C2NC(C(S2)(C)C)C(=O)O BTB12364 Cc1c(snn1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05404 Cc1c(cc(c(n1)SCCC(=O)OC(C)(C)C)C#N)c2csc(n2)C BTB09620 Cc1cc(c(c(c1)O)/C(=N/Cc2ccccc2)/C)C CD04918 Cc1ccc(c(c1)Br)OS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl BTB14581 CCCCOC(=O)c1cc(cc\2c1-c3ccc(cc3/C2=N\O)[N+](=O)[O-])[N+](=O)[O-] BTB13143 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)C(=O)C BTB10474 CCCCCCCCc1ccc-2c(c1)Cc3c2cccc3 BTB10476 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCOCC2 CD00642 c1ccc(cc1)c2ccc(cc2)C(=O)c3ccccc3 BTB10516 c1ccc2c(c1)c(c(c(=O)o2)C(c3ccc(cc3)[N+](=O)[O-])c4c(c5ccccc5oc4=O)O)O BTB10438 COc1ccc(cc1OC)CCNC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00587 CCC(CC)(C#C)/N=C/c1cc(ccc1OCC)Br CD00607 C1COC2(O1)C3C4CC5C3[C@@H](C6C5C4C26)O BTB12422 c1ccc2c(c1)-c3cccc(c3C2=O)C(=O)N4CCCCC4 BTB13169 CCN(CC)C(=O)c1cccc-2c1C(=O)c3c2cccc3 BTB13170 c1cc(sc1)C(=NOC(=O)c2ccc(cc2)[N+](=O)[O-])c3cccs3 BTB10457 c1cc(cnc1)NC(=O)c2ccc(o2)CSc3ccc(cc3)Cl CD05029 c1cc(ccc1SCc2ccc(o2)C(=O)N3CCOCC3)Cl CD05031 c1cc(ccc1SCc2ccc(o2)C(=O)Sc3ccc(cc3)Cl)Cl CD05037 CCCCOC(=O)c1cc(cc\2c1-c3ccc(cc3/C2=N\N)[N+](=O)[O-])[N+](=O)[O-] BTB13144 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)Nc3c(cccc3F)F)C)C CD04938 CCN(CC)C(=S)Sc1c(c(sn1)SC(=S)N(CC)CC)C#N CD00517 CCc1cc2c(cc1c3cnc(s3)Nc4ccccc4)C(CCC2(C)C)(C)C.Br CD00527 c1c(cc(c-2c1C(=O)c3c2c(cc(c3)C(=O)N)[N+](=O)[O-])[N+](=O)[O-])C(=O)N BTB13166 COC(=O)c1cccc-2c1C(=O)c3c2cccc3 BTB13171 Cn1c2c(c3c(cc4cc(ccc4n3)F)c(=O)n2c5ccccc5)c(=O)n(c1=O)C BTB13227 COc1cc(c(cc1OC)NC(=O)c2c(cc(cn2)C(F)(F)F)Cl)C(=O)O BTB09629 CCCCNC(=S)Nc1cccc(c1)OC CD00708 CC(C)(C)NC(=O)NCCc1ccc(c(c1)OC)OC CD00717 COc1ccc(cc1OC)C=C2C(=O)NC(=S)NC2=O CD00609 c1ccc2c(c1)cccc2C=C3C(=O)NC(=S)NC3=O CD00622 CC(c1ccccc1)NC(=O)NC(C)(C)C CD00723 CCCCCCCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB13099 Cc1cc(cc(c1OC(=O)c2ccc(cc2)C(F)(F)F)C)c3c4ccccc4c(=O)n(n3)C BTB08280 Cc1ccc(cc1)C(=O)Oc2c(cc(cc2C)c3c4ccccc4c(=O)n(n3)C)C BTB08281 c1c(cc(c2c1[nH]c(=O)c(=O)[nH]2)Br)C(F)(F)F BTB09703 CCN(CC)CCN(C)CC1c2ccccc2Oc3c1cccc3.C(=O)(C(=O)O)O.C(=O)(C(=O)O)O BTB10676 Cc1cc(ccc1Oc2c(cccn2)N)Cl BTB09630 COc1ccc(cc1)C(=O)/C(=C/c2cccs2)/C#N CD05294 CSc1ccc(cc1NC(=O)c2ccco2)Cl CD05296 CSc1ccc(cc1NC(=O)C(F)(F)F)Cl CD05302 Cc1c(nnn1c2cccc(c2Cl)Cl)C(=O)C CD05148 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)C)C)NC(=O)OCC BTB13200 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1Cl)NC(=O)OCC BTB13202 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C(F)(F)F)NC(=O)OCC BTB13203 c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3cccc4c3cccc4 BTB14610 c1cc(ccc1CCNC(=O)c2ccc(cc2)Cl)O BTB12398 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)C BTB10681 Cc1ccc(cc1)S(=O)(=O)c2c(cc(cc2C)C)C BTB10685 c1ccc(c(c1)C(=O)N)OCCOc2ccccc2C(=O)N BTB12339 COc1ccc(c(c1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)OC CD05134 COc1ccc(c(c1)Sc2ccc(cc2[N+](=O)[O-])Cl)OC CD05137 c1ccc(cc1)/C(=C/C(=O)c2ccc3c(c2)OCCO3)/C(=O)c4ccccc4 CD05160 c1cc(ccc1OCCOc2ccc(cc2)Cl)Cl BTB12345 COc1ccc(cc1)OCCOc2ccc(cc2)OC BTB12347 c1cc(c(cc1Cl)OCCOc2cc(ccc2Cl)Cl)Cl BTB12348 C1C2CC3CC1CC(C2)C3=C(C(=O)O)C(=O)O BTB12435 Cc1nc(cs1)c2ccc(cc2)OCc3ccc(c(c3)Cl)Cl BTB09522 C1C2C3CC4C2C5C1C3CC5O4 BTB12416 Cc1cc(cc(c1OCC(=O)NNC(=O)c2ccc(cc2Cl)Cl)C)c3c4ccccc4c(=O)n(n3)C BTB08308 c1cc(cc(c1)C(F)(F)F)CSCC(=O)c2ccc(cc2)OCc3ccc(cc3)F BTB09564 CCCCCCCc1cnc(nc1)c2ccc(cc2)C#N BTB09568 CCCCCc1ccc(cc1)c2ccc(cc2)Br BTB09573 CC(C)/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2ccccc2 BTB08314 c1cc(ccc1C(=O)CSc2c(c(sn2)SCC(=O)c3ccc(cc3)Br)C#N)Br CD00480 COc1ccccc1OCCOc2ccccc2OC BTB12340 COc1cccc(c1)OCCOc2cccc(c2)OC BTB12342 c1cc(c(cc1Br)Br)OCCOc2ccc(cc2Br)Br BTB12344 CC1(OC(=O)C2(C3C4C5CC6C4C2C7C6C5C73)C(=O)O1)C BTB12419 c1ccnc(c1)NC=C(C#N)C#N CD00521 c1ccc\2c(c1)-c3ccc(cc3/C2=N\O)[N+](=O)[O-] BTB13157 COc1ccc(cc1OC)S(=O)(=O)Oc2ccc(cc2)[N+](=O)[O-] CD05026 CCC(C#N)(c1ccccc1)c2ccc(cc2)[N+](=O)[O-] BTB09571 c1ccc(cc1)C(=O)c2ccc3c(c2)OCCCO3 BTB10432 Cc1ccc(c(c1)[N+](=O)[O-])OS(=O)(=O)c2ccc(c(c2)OC)OC CD05032 c1ccc(cc1)C(c2ccccn2)N.Cl.Cl BTB10358 CC1(C(NC(S1)c2ccc(cc2)[N+](=O)[O-])C(=O)O)C BTB12372 c1cc(ccc1SCc2ccc(o2)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl CD05079 CN(C)c1c(cc(cc1F)C(=O)Nc2ccc(cc2)OC)F CD05095 c1cc(ccc1COc2ccc(cc2[N+](=O)[O-])C3SCCS3)F BTB09613 CC(C)(C)NC(=O)NC(C)(C)C#C CD00711 COc1ccc(c(c1)S(=O)(=O)Oc2ccc(cc2)[N+](=O)[O-])OC CD05027 COc1ccc(cc1OC)CCNC(=O)c2ccc(o2)CSc3ccc(cc3)Cl CD05030 c1ccc(cc1)S(=O)(=O)Cc2cc(ccc2[N+](=O)[O-])C(=O)O BTB10424 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)S(=O)(=O)c4cc(c(cc4Cl)Cl)Cl BTB14541 Cc1cc(c(cc1Cl)C)S(=O)(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 BTB14542 COc1ccc(c(c1)S(=O)(=O)Oc2ccc(cc2)C#N)OC CD05034 C#CCOC(=O)c1ccc(o1)CSc2ccc(cc2)Cl CD05036 Cc1ccc(c(c1)Br)OS(=O)(=O)c2ccc(cc2)NC(=O)C BTB14585 COc1ccccc1N2CCN(CC2)Cc3ccc(cc3Cl)Cl BTB14586 CC(=O)c1ccc(c(c1)CSc2nnc(s2)SCc3cc(ccc3OC)C(=O)C)OC CD02942 CC1(OC(=O)C(=C2C3CC4CC(C3)CC2C4)C(=O)O1)C BTB12432 c1cc(sc1)C=C2C(=O)NC(=O)NC2=O CD00800 COc1cccc(c1)NC(=S)NC2CCCCCCCCCCC2 CD00716 CCOC(=O)c1c(nc(s1)N)C.Cl BTB10693 CC(C)(C)NC(=O)NCc1ccncc1 CD00727 CC(C)(C)NC(=O)NCc1cccnc1 CD00728 Cc1ccc(c(c1)Br)OS(=O)(=O)c2cccc(c2)C(F)(F)F BTB14583 c1ccc(c(c1)C2C(C2(C#N)C#N)(C#N)C#N)Cl CD02963 c1cc(ccc1NC(=O)NNC(=O)COc2ccc(cc2)SC(F)(F)F)Cl BTB08352 COCCCNC(=S)NNC(=S)Nc1cccc(c1)SC CD02871 Cc1ccc(cc1)CN2CCN(CC2)c3ccccc3OC BTB14590 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)C/C(=N/O)/N CD02984 c1cc(ccc1c2nc(on2)CN3CCCCC3)Cl CD02882 Cc1cccc(c1C(=O)O)NC(=O)C BTB09608 c1ccc(cc1)Oc2ccc(cc2)OC(=O)c3ccc(cc3)N BTB14630 c1cc(ccc1c2cnc(s2)Nc3cc(cc(c3)Cl)Cl)Cl BTB14688 COc1cccc(c1)c2cnc(s2)Nc3ccc(cc3)F BTB14690 COc1ccc(cc1)C2C(C2(C#N)C#N)(C#N)C#N CD02965 CCc1cc2c(cc1c3csc(n3)C/C(=N/O)/N)C(CCC2(C)C)(C)C CD02966 CC(C)OC(=O)c1ccc(cc1)[N+](=O)[O-] BTB10453 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)N)C CD02985 COc1ccccc1N2CCN(CC2)Cc3cccc(c3)[N+](=O)[O-] BTB14591 Cn1c(=O)ccc(n1)c2ccccc2 BTB12373 c1ccc(cc1)c2cccnn2 BTB12377 CC1(C2CCC(C2)(C1NCC(=O)N(c3ccccc3)C4CCCCC4)C)C.Cl BTB14624 Cc1nc2c(o1)c3c(n(c2=O)C)n(c(=O)n(c3=O)C)C BTB14684 c1c([nH]cn1)CCN2C(=O)CCC2=O BTB12383 c1c([nH]cn1)CCN2C(CCC2=O)O BTB12384 Cn1c2ccccc2nc1C(C#N)C(=O)c3ccccc3I BTB12309 c1ccc2c(c1)c(c(c(=O)[nH]2)/C=N/C(=O)N)O BTB12393 COCCCNC(=S)N/N=C/c1ccccc1Cl CD02914 CN(C)c1ccc(cc1)/C=N/NC(=S)NCCCOC CD02917 c1cc(ccc1COc2ccc(cc2)C(=O)CSCc3ccc(c(c3)Cl)Cl)F BTB09614 CN1C2CCC1CC(C2)NC(=O)c3ccc(cc3)[N+](=O)[O-] BTB10455 c1cc(sc1)C(=NOC(=O)c2ccc(cc2)Cl)c3cccs3 BTB10456 CC(C)c1ccc(cc1)C=C2C(=O)NC(=S)NC2=O CD00611 C(C#N)Sc1c(c(sn1)SCC#N)C#N CD00507 Cc1ccc(cc1F)NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00575 c1cc(ccc1NC(=S)Nc2ccc3c(c2)OCO3)S(=O)(=O)N4CCCCC4 CD00578 Cn1c2ccccc2nc1C(C#N)C(=O)c3ccccc3Br BTB12310 COc1cc(ccc1O)C=C2C(=O)NC(=S)NC2=O CD00512 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C)NC(=O)OCC BTB13194 c1cc(ccc1c2nc(on2)CSc3nnc(s3)SCc4nc(no4)c5ccc(cc5)Cl)Cl CD02944 c1cc-2c(cc1[N+](=O)[O-])C(=NN)c3c2ccc(c3)[N+](=O)[O-] BTB13146 c1cc-2c(cc1Br)C(=NO)c3c2ccc(c3)Br BTB13147 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/NCc3ccccc3)/C(=O)N2C BTB14678 CCCCC1C(=O)N(N(C1=O)c2ccccc2)c3ccccc3 BTB12395 COc1ccc(cc1Br)C=C2C(=O)NC(=S)NC2=O CD00508 COc1ccc(cc1)C=C2C(=O)NC(=S)NC2=O CD00510 c1c(cc(c(c1F)NC(=O)C(Cl)Cl)F)Br CD04956 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3ccc(cc3)F)/C(=O)N2C BTB14659 Cn1c2ccccc2c(cc1=O)O BTB12329 CCOc1ccc(cc1OC)C=C2C(=O)NC(=S)NC2=O CD00792 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3cc(cc(c3)Cl)Cl)/C(=O)N2c4ccccc4 BTB14666 c1ccc(cc1)C(=O)/C(=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)/C#N CD05192 CN(C)c1ccc(cc1)/C=C(\C#N)/C(=O)c2ccco2 CD05207 c1cc(oc1)C(=O)/C(=C/c2ccc3c(c2)OCO3)/C#N CD05208 c1ccc2c(c1)NC(=O)C(S2)CC(=O)Nc3ccccc3Cl BTB14756 CS/C(=C(/C#N)\C(=O)c1ccco1)/Nc2cc(ccc2Cl)Cl CD05212 CSc1ccc(cc1NC=C(C#N)C#N)C(F)(F)F CD05229 COc1ccc(cc1)C2C3C(C(=O)N(C3=O)Cc4ccccc4)ON2c5ccccc5 BTB14761 Cc1cc(nc2n1nnn2)c3ccccc3 BTB14762 c1cc(ccc1COc2ccc(cc2[N+](=O)[O-])C3SCCS3)[N+](=O)[O-] BTB09612 Cc1c(cc(c(n1)SCCNS(=O)(=O)c2ccc(cc2)C(C)(C)C)C#N)c3csc(n3)C BTB09544 c1c(c(=O)[nH]c2c1C(=O)CCC2)C#N BTB09549 CC(=O)c1ccc(cc1)OCc2ccc(cc2)F BTB09553 CCCCCCCC\1CCC/C1=N\OC(=O)c2cccs2 BTB10539 c1ccc(cc1)Nc2ccc(cc2)/N=N/c3ccccc3 BTB10542 c1ccc(cc1)C2/C(=C/c3ccc(cc3)Br)/C(=O)c4ccccc4O2 BTB13253 CCOC(=O)C(C(F)(F)F)(NCc1ccc(cc1)F)NC(=O)OCC BTB13198 c1ccc2c(c1)C(C(=O)N2)(C(F)(F)F)O BTB10550 COc1ccc(cc1)/C=C\2/C(Oc3ccccc3C2=O)c4ccccc4 BTB13256 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1F)F)F)NC(=O)OCC BTB13207 c1cc(cc(c1)C(F)(F)F)c2nc3c(cc(cn3n2)C(F)(F)F)Cl BTB10553 CCOc1ccccc1/C=C/2\c3ccccc3NC2=O CD00754 c1ccc2c(c1)/C(=C\c3ccc(cc3)F)/C(=O)N2 CD00755 COc1ccccc1N2CCN(CC2)Cc3ccc(c(c3)Cl)Cl BTB14588 Cn1c2c(c3c(c1=O)cc4cc(ccc4n3)OC)c(=O)n(c(=O)n2c5ccccc5)c6ccccc6 BTB14650 CC1(C(NC(S1)c2ccc(cc2Cl)Cl)C(=O)O)C BTB12367 COc1ccccc1N2CCN(CC2)Cc3ccccc3F BTB14589 COc1ccc(cc1)NC(=S)NCCCC2C=NN=C2O CD02928 c1cc([nH]c1)C=C2C(=O)NC(=O)NC2=O CD00861 c1cc2c(cc1Cl)[nH]c(=O)c(=O)[nH]2 BTB09743 c1ccc(cc1)S(=O)(=O)N=C(NN)NN CD03087 CC(C)c1ccc(cc1)/C=C\2/C(Oc3ccccc3C2=O)c4ccccc4 BTB13258 CCN(CC)CCN(C)C(=O)C1c2ccccc2Oc3c1cccc3.C(=O)(C(=O)O)O.C(=O)(C(=O)O)O BTB10677 c1cc(oc1)C2C(=C(OC(=C2C#N)N)c3ccco3)C#N CD05250 c1cc(cc(c1)Cl)N/N=C(\C#N)/C(=O)c2ccco2 CD05253 c1ccnc(c1)Sc2ccc(cn2)[N+](=O)[O-] BTB09633 CCC(C)(C)NC(=S)Nc1cccc(c1)OC CD00700 c1ccc(c(c1)CO)Sc2ccccc2CO BTB12327 CCc1ccc2c(c1)cc3c(n2)c4c(n(c(=O)n(c4=O)C)C)n(c3=O)c5ccccc5 BTB14658 CCOc1ccccc1C=C2C(=O)NC(=S)NC2=O CD00623 CCCCCCCC\1CCC/C1=N/OC(=O)c2ccc(cc2)[N+](=O)[O-] BTB10538 COc1ccc(cc1OC)CC/N=C/c2ccc3c(c2)OCO3 CD00663 CN(C)CCCNC(=S)Nc1cccc(c1)OC CD00701 COc1cccc(c1)NC(=S)Nc2cccc(c2)O CD00706 CC1CCC(C(C1)N)C(C)C.Cl BTB10558 Cc1ccc(cc1)NC(=O)c2cc(cc3c2-c4ccc(cc4C3=O)[N+](=O)[O-])[N+](=O)[O-] BTB13186 c1cc2cn[nH]c2cc1/N=C/c3cc(ccc3O)Cl CD00636 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)OC(=O)C4CCC(CC4)CCC BTB10483 c1cc(sc1)C=C2C(=O)NC(=S)NC2=O CD00801 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N/N=C/c2cccs2 CD00809 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1)NC(=O)OCC BTB13192 CC1CC(CC(C1)(C)C)NC(=S)Nc2cccc(c2)OC CD00707 C1C2C3C4C1C5C2C6C3C4C5(O6)C[N+](=O)[O-] BTB12417 c1ccc(cc1)/C=C/C=C(\C#N)/C(=S)N CD02950 c1c(cc(c(c1/C=C(\C#N)/C(=S)N)O)Cl)Cl CD02951 c1cc(ccc1CO)OCc2ccc(cc2)F BTB09617 CCCCCCc1ccc-2c(c1)Cc3c2cccc3 BTB10488 CC(=O)c1ccc-2c(c1)Cc3c2cccc3 BTB10491 c1ccc-2c(c1)Cc3c2ccc(c3)C(=O)c4ccc(cc4)Br BTB10465 CCCCC(=O)c1ccc-2c(c1)Cc3c2ccc(c3)CCc4ccc(cc4)Br BTB10468 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)OC(=O)c4ccc(cc4)OCCC BTB10469 c1ccc(cc1)C2/C(=C/c3ccc(cc3Cl)Cl)/C(=O)c4ccccc4O2 BTB13254 c1cnc(cc1C(F)(F)F)O BTB09682 Cc1c(nnn1c2c(cccc2F)F)C(=O)C CD05144 Cc1cc(c(c(=O)[nH]1)[N+](=O)[O-])O BTB12408 C1C2C3C4C1C5C2C6C3C4C5(O6)C(C(=O)O)(F)F BTB12411 c1cc(ccc1c2csc(n2)C/C(=N/O)/N)Cl CD02946 COc1cc(cc(c1OC)OC)/C=C(\C#N)/C(=S)N CD02948 COc1ccc(cc1)/C=C(\C#N)/C(=S)N CD02962 Cc1cc2cc3c(nc2cc1C)n(c(=O)n(c3=O)C)C BTB14679 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)OC(=O)c4ccc(cc4)OCCCCC BTB10471 c1ccc(cc1)C(Cn2ccccc2=N)O BTB10420 c1ccc(cc1)C(C(=O)c2ccccc2)SC#N BTB10422 CSc1ccc(c(c1)CS(=O)(=O)c2ccccc2)[N+](=O)[O-] BTB10423 c1ccc(c(c1)C(F)(F)F)NC(=S)Nc2cccc(c2)C(F)(F)F CD00702 Cc1c(nnn1c2cccc(c2)C#N)C(=O)C CD05147 COc1cnn(c(=O)c1Cl)c2ccccc2 BTB09683 c1ccc(c(c1)C(=O)O)n2cccc2 CC34301 CN(C)/C=N/c1nc(cc(n1)OC)OC BTB09678 c1ccc2c(c1)/C(=C\c3c(cccc3Cl)Cl)/C(=O)N2 CD00995 C1CCN(CC1)C/C(=N/O)/N CD05169 c1ccc(cc1)c2ccc(cc2)c3csc(n3)N4CCOCC4.Br CD01171 Cc1c(nn(n1)c2ccccc2)C(=O)ON3C(=O)C4C5C=CC(C4C3=O)O5 BTB09739 c1ccc2c(c1)/C(=C\c3ccc(c(c3)Cl)Cl)/C(=O)N2 CD00751 CS(=O)(=O)O[C@H]1[C@@H](Oc2ccccc2C1=O)c3ccccc3 BTB13243 C1C2C3C4C1C5C2C6C3C4C5O6 BTB12415 CN(C)CCCNC(=S)Nc1cccc(c1)C(F)(F)F CD00703 c1cc(ccc1C=C2C(=O)NC(=O)NC2=O)F CD00732 CC(C)c1ccc(cc1)/C=C/2\c3ccccc3NC2=O CD00749 c1c(ccc(c1)/N=C/c2cc(c(cc2)O)O)Cc3ccc(cc3)/N=C/c4cc(c(cc4)O)O CD01000 c1ccc2c(c1)/C(=C\c3cccs3)/C(=O)N2 CD00821 CC1CN(CC(O1)C)C(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00831 CCC(CC)(C#C)NC(=O)c1c(onc1c2ccccc2Cl)C CD00843 CC1(CC2=C(C(C3=C(O2)CC(CC3=O)(C)C)c4cc(cc(c4O)Cl)Cl)C(=O)C1)C CD03380 COc1cccc(c1)NC(=S)Nc2ccc(cc2Cl)Br CD00709 C1C2C3C4C1C5C2C6C3C4C5C6(CO)CO BTB12418 c1cc(c(cc1CSc2nnc(s2)SCc3ccc(c(c3)Cl)Cl)Cl)Cl CD02958 c1cc(oc1)/C=N/NC(=S)NC2CC3CCC2C3 CD03012 COCCCNC(=S)N/N=C/c1ccc(cc1)OC CD02913 CCCCCCCc1ccc-2c(c1)Cc3c2ccc(c3)Br BTB10492 COC(=O)/C(=C\Nc1ccc(nc1)Sc2ccc(cc2)Cl)/NC(=O)c3ccccc3 BTB09696 COc1ccc(cc1)C(=O)/C(=N/Nc2cccc(c2Cl)Cl)/C#N CD05418 Cn1c2c(c3c(c1=O)cc4ccc(cc4n3)F)c(=O)n(c(=O)n2C)C BTB14665 c1ccc(cc1)CCNC(=O)Oc2ccc(cc2)Cl BTB13274 CC(C)(C)NC(=O)Oc1ccc(cc1)Cl BTB13275 COc1ccc(cc1)OC(=O)NCCc2ccccc2 BTB13278 c1ccc(cc1)S(=O)(=O)/N=C/2\NCC3CCCC3N2 CD03056 c1cc(cnc1)C=C2C(=O)NC(=S)NC2=O CD00916 Cn1c2ccccc2c3c(c1=O)c(cc(=O)o3)O BTB12394 COCCCN(Cc1cc(c(c(c1)OC)OC)OC)C(=S)Nc2cccc(c2)Cl CD03075 c1ccc2c(c1)ccc3c2-c4c(ccc5c4cccc5)CC3 BTB10671 COC(C(=O)N)(C(F)(F)F)F BTB12427 COc1ccccc1C2CCN(CC2)Cc3cccc4c3cccc4 BTB14611 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)OCC BTB13204 COc1cc(cc(c1OC)OC)/C=C/2\c3ccccc3NC2=O CD00902 COc1ccc(cc1)c2cc(c(nn2)c3ccccc3)c4ccccc4 CD05157 COc1cc(nc(n1)N/C=N/O)OC BTB09686 CCOc1cnn(c(=O)c1Cl)c2ccccc2 BTB09693 COc1ccc(cc1CN2CCOCC2)C(=O)/C=C(/c3ccccc3)\C(=O)c4ccccc4 CD05164 COc1ccc(cc1CN2CCOCC2)c3cc(c(nn3)c4ccccc4)c5ccccc5 CD05165 c1cnccc1C(=N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05166 c1ccc2c(c1)cccc2OCCOc3cccc4c3cccc4 BTB12349 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)F)F)NC(=O)OCC BTB13206 c1cc(cc(c1)[N+](=O)[O-])C(=O)OC2CN3CCC2CC3 BTB14621 C=C(CN1CCN(CC1)CC(=C)C#N)C#N CD05172 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)OC(=O)C4CCC(CC4)CCCCC BTB10478 CC(c1cccc2c1cccc2)O BTB10484 c1cc2c(cc1S(=O)(=O)[O-])[nH]c(n2)S.[Na+] BTB12361 c1cc(c(cc1CS(=O)(=O)Cc2ccc(c(c2)Cl)Cl)Cl)Cl CD05378 c1ccc(c(c1)C(=O)/C(=N/Nc2ccc(cc2)F)/C#N)Cl CD05434 COc1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)F)/C#N CD05435 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)SCc3cccc(c3)C(F)(F)F CD05386 COc1ccc(cc1)/C(=C/c2c[nH]nc2)/C#N BTB09692 c1cc(c(cc1/C=N/NC(=S)NC2CC3CCC2C3)Cl)Cl CD03011 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=S)NCCCOC CD02918 CC(=O)CC(c1ccccc1[N+](=O)[O-])c2c(c3ccccc3oc2=O)O BTB10436 COc1ccc(cc1)NC(=O)CSc2ncccn2 BTB14699 COCCCNC(=S)N/N=C/c1ccc(cc1)O CD02915 CC(C)(C)NC(=O)c1cccc2c1-c3ccccc3C2=O BTB13182 Cc1ccc(cc1C)NC(=O)c2c(cc(cc2CC(C)(C)C(=O)O)C)C CD03145 CC1(OC(=O)C(=NNc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)O1)C CD05367 CC(=O)C(=NNc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(=O)C CD02999 CN(CCC#N)c1ccc(cc1)C=C2C(=O)NC(=O)NC2=O CD01011 c1ccc(cc1)c2ccc(=O)[nH]n2 BTB10629 c1cc(sc1)C(=O)CCC(=O)O BTB10644 CCC(CC)(c1ccccc1c2ccccc2C(CC)(CC)O)O BTB10653 c1ccc(c(c1)/C=N/NC(=S)NC2CC3CCC2C3)O CD03007 Cc1c(snn1)C(=O)NCc2c(cccc2Cl)F CD05408 c1ccc(c(c1)N)SCc2nc(no2)c3ccc(cc3)Cl CD03140 c1cc(cc(c1)C#N)CSc2nnc(s2)SCc3cccc(c3)C#N CD02941 CCOC(C(=O)N)(C(F)(F)F)F BTB12428 c1ccc(cc1)N2C(=NC3(N2)CCCCC3)S CD03187 CCOc1cc(c(cc1OCC)OCC)C=C2C(=O)NC(=O)NC2=O CD00906 CC(=CC(=O)Oc1ccc(cc1)n2c(nnn2)SCC=C)C BTB09665 c1cc(ccc1/C=N/NC(=S)NC2CC3CCC2C3)O CD03008 c1ccc(cc1)OC(=O)N2CCCC2 BTB13284 c1cc(cc(c1)/N=C/c2cccnc2)C(F)(F)F CD00923 Cc1ccc(c2c1CCC2)OC(C)(C)C(=O)Nc3ccc(nc3)Sc4cc(ccc4Cl)Cl BTB09674 c1cc(ccc1C(=O)c2ccc(cc2)F)[N+](=O)[O-] BTB09677 COC(=O)c1c(c2ccccc2[nH]c1=O)O BTB14682 CCc1cc2c(cc1c3csc(n3)CC#N)C(CCC2(C)C)(C)C CD02904 c1ccc(cc1)/C=C(\C#N)/C(=O)N BTB09600 c1c2cc(c(=O)oc2c(cc1Br)Br)C(=O)O BTB09657 COc1ccc(cc1)/C=N/NC(=S)N[C@H]2CC3CCC2C3 CD03199 CCOc1ccc(cc1OC)C=C2C(=O)NC(=O)NC2=O CD00790 c1ccc2c(c1)nc3n2c(=O)/c(=C\c4cccc(c4)[N+](=O)[O-])/s3 BTB14753 CCOc1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)C(C)(C)C BTB14696 c1cc(cc(c1)C(F)(F)F)c2nc3c(cc(cc3Cl)Cl)c(=O)o2 BTB14703 CC(C)(C)NC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB12456 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05389 c1cc(sc1)c2nc3c(cc(cc3Cl)Cl)c(=O)o2 BTB14704 C1COC2(O1)C3C4CC5C3C(=O)C6C5C4C26 BTB12423 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Oc2ccc(cc2)Oc3ccccc3 BTB14634 c1ccc(cc1)Oc2ccc(cc2)OS(=O)(=O)c3cccc(c3Cl)Cl BTB14635 CCC(C)c1ccc(cc1)NC(=O)CSc2ccccn2 BTB14697 Cc1nnc(s1)SCC(=O)Nc2ccc3c(c2)OCCO3 BTB14700 Cn1c2c(c3c(c1=O)cc4c(n3)cc(cc4Cl)Cl)c(=O)n(c(=O)n2c5ccccc5)c6ccccc6 BTB14648 COC(=O)c1cccnc1Oc2ccccc2 BTB09746 Cc1c(onc1/N=C/N(C)C)C BTB09685 c1ccc2c(c1)C(=O)N(C2=O)c3cccc(c3)[N+](=O)[O-] BTB10701 CC1N=C(N2N1C(=NC2C)S)S CD03103 c1cc(ccc1CSc2ccc(cc2)Cl)C#N CD03112 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N/N=C/c2ccncc2 CD00812 CCOC(=O)c1cc(n[nH]c1=O)c2ccc(s2)Br BTB09723 CCOc1ccc(cc1)C=C2C(=O)NC(=S)NC2=O CD00551 Cc1c(c(c(c(c1C)C)CSC(=N)CC#N)C)C.Cl CD02923 c1cc(ccc1CSc2nnc(s2)SCc3ccc(cc3)Cl)Cl CD02932 Cn1c(=O)cc(c2c1n(c(=O)n(c2=O)c3ccccc3)c4ccccc4)N5CCCCC5 BTB14654 c1ccc(cc1)CCN2CC(CN(C2)CCc3ccccc3)C#N CD05179 c1ccc(cc1)C(=O)/C(=C/c2cccs2)/C#N CD05189 Cc1ccc2c(c1)c(cc(n2)C)C BTB10702 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1)NC(=O)c2cccc(c2)Cl BTB13209 c1cc(ccc1CON2C(=O)C3C4C=CC(C3C2=O)O4)OC(F)(F)F BTB09747 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C(F)(F)F)NC(=O)c2cccc(c2)Cl BTB13216 C=CCOC(=O)C(CC(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 BTB13319 COc1ccc(cc1)/C=C/2\c3ccccc3NC2=O CD00756 c1ccc(c(c1)/C=C/2\c3ccccc3NC2=O)Cl CD00757 COc1ccc(c(c1)C(=O)/C(=C/c2cccs2)/C#N)Br CD05259 c1cc(oc1)C(=O)/C(=N/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N CD05270 Cc1c(snn1)C(=O)Oc2ccc(cc2)[N+](=O)[O-] CD05438 Cc1c(snn1)C(=O)N2CCc3c(c4cc(ccc4[nH]3)F)C2 BTB13387 COc1ccccc1C2CCN(CC2)C(=O)c3ccco3 BTB13388 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)Nc2cccc(c2)SC)C CD03034 c1ccnc(c1)/C=N/NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD03041 c1cc(c(c(c1)Cl)CNC(=S)Nc2ccc(cc2)Cl)F CD05450 c1cc(c(c(c1)Cl)CSC(=C(C#N)C#N)SCc2c(cccc2Cl)F)F CD05451 c1cc(c(c(c1)Cl)CNC(=O)c2ccc(cc2)Cl)F CD05457 c1cc(ccc1CON2C(=O)C3C4C=CC(C3C2=O)O4)[N+](=O)[O-] BTB09749 COc1ccc(cc1)C(c2ccc(cc2)OC)NC(=O)CCC(C(=O)O)NC(=O)OCc3ccccc3 BTB13323 Cc1nc2ccccc2c(=O)n1c3ccc(c(c3F)F)F BTB14710 CCCCCc1ccc-2c(c1)Cc3c2ccc(c3)Br BTB10533 c1ccnc(c1)/C=N/NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03262 c1c(cc(cc1C(F)(F)F)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD03264 c1ccc(cc1)C(=O)CC(c2cccc(c2)Cl)Sc3ccccc3N BTB14874 Cc1cccc(c1)OC(=O)NC BTB13280 COc1ccc(cc1Br)c2ccccc2 BTB14799 CC(C)NC(=O)Oc1ccccc1 BTB13267 c1ccc(cc1)OC(=O)N2CCCCC2 BTB13283 c1ccc2c(c1)c(nc3n2nnc3c4ccc(cc4)Br)N CD05128 COCCCNC(=S)N/N=C/c1ccc2c(c1)OCO2 CD02916 c1ccc2c(c1)c(c[nH]2)C=C3C(=O)NC(=S)NC3=O CD00825 Cc1nc(cn1C(C)C)[N+](=O)[O-] BTB09767 CCOC(CSc1c(nc2ccccc2n1)SCC(OCC)OCC)OCC BTB14803 CC(C)NC(=O)Oc1cccc(c1)Cl BTB13281 CNC(=O)Oc1cccc2c1cccc2 BTB13282 CN1C2C[C@@H](CC1CC2)NC(=O)CSCc3ccc(cc3)Cl BTB14829 CC1C(OCCN1C(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3)c4ccccc4 CD00921 c1cc(ccc1[N+](=O)[O-])OC(=O)N2CCCCC2 BTB13287 CC1=C(C(=O)C(=C(C1=O)Br)C)Br BTB14806 COc1cc(c(cc1SC)OC)SC BTB14807 COc1ccc(c(c1)CCCc2cc(ccc2OC)OC)OC BTB14810 CC1CN/C(=N/S(=O)(=O)c2ccccc2)/N1 CD03057 c1ccc(cc1)n2c3c(c(on3)c4ccc(cc4)[N+](=O)[O-])c(=O)n(c2=O)c5ccccc5 BTB14655 CC(c1ccccc1c2ccccc2C(C)O)O BTB10593 c1ccnc(c1)C=C2C(=O)NC(=O)NC2=O CD00917 CC(=O)c1ccc(cc1)c2ccc(cc2)C(=O)C BTB09791 CN1C2C[C@@H](CC1CC2)NC(=O)CS(=O)(=O)c3ccccc3 BTB14831 COc1ccc(cc1)c2coc3ccccc3c2=O BTB12551 c1cc-2c(cc1Br)C(=O)c3c2ccc(c3)Br BTB13291 CN1C2C[C@@H](CC1CC2)NC(=O)CSc3sc(nn3)N BTB14837 Cn1c2c(cc3ccc(cc3n2)Cl)c(=O)n(c1=O)C BTB14660 c1ccc2c(c1)/C(=C\c3cccc(c3)[N+](=O)[O-])/C(=O)N2 CD00752 c1ccc2c(c1)/C(=C\c3ccc(cc3)Cl)/C(=O)N2 CD00759 c1cc(oc1)CNC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00773 CC(c1ccc(cc1)SCC(=O)N[C@H]2CC3N(C(C2)CC3)C)(C)C BTB14826 CN1C2C[C@@H](CC1CC2)NC(=O)CSCc3c(cc(cc3)Cl)Cl BTB14828 Cc1coc2c(c1=O)cc(cc2Cl)Cl BTB12539 CC(=O)c1ccc(c(c1)CS(=O)(=O)Cc2cc(ccc2OC)C(=O)C)OC CD05373 CN(C)c1ccc(cc1)/C=C(\C#N)/C(=O)c2ccccc2Cl CD05375 c1ccc(c(c1)C(=O)/C(=C/c2cccs2)/C#N)Cl CD05376 COC(=O)c1cccc(c1)CS(=O)(=O)C CD05649 c1ccc(cc1)S(=O)(=O)N=C(NNC(=O)c2cccc(c2)Cl)NNC(=O)c3cccc(c3)Cl CD03173 Cc1ccc(cc1)S(=O)(=O)O.C=CCOC(=O)[C@H](Cc1ccc(cc1)O)N BTB10720 c1c(cc(cc1C(F)(F)F)N2CCCC2)C(F)(F)F CD03289 CC1(c2ccccc2-c3c1cccc3)O BTB10680 CN(C)c1ccc(cc1)CC2c3ccccc3NC2=O CD01045 Cc1nc(cn1CCC(=O)C)[N+](=O)[O-] BTB09772 CC1(CN=C(S1)N(c2ccc(cc2)Cl)C(=O)Nc3ccccc3)C BTB13189 CC1(CN=C(S1)N(c2ccc(c(c2)Cl)F)C(=O)Nc3ccccc3)C BTB13190 c1cc(cc(c1)NC(=S)NCCCC2C=NN=C2O)C(F)(F)F CD02920 c1ccc(cc1)C2/C(=C/c3cccc(c3)Cl)/C(=O)c4ccccc4O2 BTB13250 c1ccc(cc1)C2/C(=C\c3ccc(cc3)Cl)/C(=O)c4ccccc4O2 BTB13251 COc1ccccc1c2coc3ccccc3c2=O BTB12546 COc1ccc(cc1)CSC2=C(C(=O)NC3(S2)CCCCC3)C#N CD01332 COc1cc(cc(c1OC)OC)C2N=C(C(=C(S2)SC)C#N)O CD01334 CSC1=C(C(=O)NC(S1)c2cccc3c2cccc3)C#N CD01335 c1ccc2c(c1)cccc2/C=N/NC(=S)N[C@H]3CC4CCC3C4 CD03198 c1cc(ncc1[N+](=O)[O-])N/N=C/c2cc(cc(c2O)Cl)Cl CD01177 CC1CN(CC(O1)C)c2ccc(cn2)[N+](=O)[O-] CD01197 COc1ccc(cc1OC)CCNC(=O)c2nc3ccccc3c(=O)n2n4cccc4 CD03353 CC(C)CCN(CCC(C)C)S(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)N(CCC(C)C)CCC(C)C)C2=O BTB12446 COCCCN(Cc1cc(c(c(c1)OC)OC)OC)C(=S)Nc2cccc(c2)SC CD03078 COc1ccc(c(c1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl)OC CD05139 CNc1nnc(s1)C(F)(F)F CD05460 c1cc(cc(c1)C(F)(F)F)Cc2cccc(c2)C(F)(F)F CD03080 c1ccc(cc1)C2c3ccccc3C(=O)O2 BTB10637 Cc1ccc(cc1Cl)NC(=O)c2c(nns2)C CD05495 CCNS(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)NCC)C2=O BTB13361 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O CD05388 c1cc(cc(c1)C(F)(F)F)C(=O)ON=C(c2cccs2)c3cccs3 BTB10714 c1ccc2c(c1)nc(c3n2ccc3)SCc4csc(n4)c5ccc(cc5)Cl CD03391 c1ccc-2c(c1)NC(c3n2ccc3)c4cccnc4 CD03393 CC(=O)NCc1c(cccc1Cl)F CD05339 CC1(OC(=O)C(=Cc2cccs2)C(=O)O1)C CD05350 c1ccc(c(c1)N)SCc2csc(n2)c3ccc(cc3)Cl CD03342 CC(C)(C)c1ccc(cc1)/C=C/C(=O)NCCc2c[nH]c3c2cccc3 BTB14723 c1ccc(cc1)C2=NN3C(C2)c4ccccc4OC3c5cccc(c5)[N+](=O)[O-] BTB14754 CC(C)(C)c1cc(c(c(c1)C(C)(C)C)NC)C(C)(C)C BTB14758 Cc1c(snn1)C(=O)Nc2cccc(c2)[N+](=O)[O-] CD05498 c1ccc(cc1)CN(Cc2ccccc2)C(=O)c3cc(cc4c3-c5ccc(cc5C4=O)[N+](=O)[O-])[N+](=O)[O-] BTB12455 CCOC(=O)c1cccc2c1-c3ccccc3C2=O BTB12457 C1CCCCCC(C(CCCC1)CCC#N)O BTB09773 C1CCCCCC(=O)C(CCCC1)CCC#N BTB09775 c1cc(c(cc1C2C(C2(C#N)C#N)(C#N)C#N)Cl)Cl CD02973 CC1(OC(=O)C(=Cc2ccc[nH]2)C(=O)O1)C CD05351 c1ccc(cc1)COC(=O)c2cc(cc3c2-c4ccc(cc4C3=O)[N+](=O)[O-])[N+](=O)[O-] BTB13358 c1c(cc(c-2c1C(=C(C#N)C#N)c3c2c(cc(c3)S(=O)(=O)N)[N+](=O)[O-])[N+](=O)[O-])S(=O)(=O)N BTB13360 CC(C)CCOS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)OCCC(C)C BTB12453 CC1(OC(=O)C(=Cc2ccc(o2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)C(=O)O1)C CD05528 CC(C)OC(=O)c1cccc2c1-c3ccccc3C2=O BTB12459 c1ccc(cc1)c2ccsc2c3ccccc3 BTB10743 c1ccc(cc1)S(=O)(=O)N=C(NNC(=S)Nc2ccc(cc2)F)NNC(=S)Nc3ccc(cc3)F CD03276 c1ccc(c(c1)NC(=O)/C=C/C(=O)O)SCCC#N CD03377 CCCCn1cc(nc1C)[N+](=O)[O-] BTB09768 c1ccc2c(c1)C(C(=O)N2)Cc3cccs3 CD01046 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2)c3ccccc3 BTB10683 CN(C)c1ccc(cc1)/C=C\2/C(Oc3ccccc3C2=O)c4ccccc4 BTB13259 CC(C)CCNC(=O)Oc1ccccc1 BTB13269 COc1ccc(c(c1)Sc2ccc(cc2)[N+](=O)[O-])OC CD05140 c1c(cc(cc1C(F)(F)F)[N+](=O)[O-])Cc2cc(cc(c2)[N+](=O)[O-])C(F)(F)F CD03098 CC1(OC(=O)C(=Cc2ccc(o2)c3ccccc3[N+](=O)[O-])C(=O)O1)C CD05529 c1ccc(cc1)n2cnnc2S BTB12614 c1c(ccc(c1)S(=O)(=O)c2ccc(cc2)/N=C/c3cc4c(cc3)OCO4)/N=C/c5cc6c(cc5)OCO6 CD00932 c1cc(ccc1OC(=O)N2CCCCC2)Cl BTB13286 CCOc1ccc(cc1)NC(=O)N BTB13290 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)S(=O)(=O)Cc3cccc(c3)C(F)(F)F CD05391 CC1=C(c2ccc(cc2S1(=O)=O)Cl)Cl BTB14691 CN(C)CCCNS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F CD05416 c1ccc2c(c1)[nH]c(n2)S(=O)(=O)O BTB12616 CN1C(=O)C(=CNc2ccc(cc2Cl)Cl)C(=O)N(C1=O)C BTB12619 c1ccc(cc1)C2(c3ccccc3-c4c2cccc4)c5ccccc5 BTB10694 COC(=O)c1cccc2c1c(ccc2)c3cccc4c3c(ccc4)C(=O)OC BTB10698 c1cc(cnc1)Nc2nc(cs2)c3ccc(cc3)[N+](=O)[O-].Br CD01133 COC(=O)/C(=C\Nc1ccc(nc1)Oc2cc(cnc2)Cl)/NC(=O)c3ccccc3 BTB09695 c1ccc(cc1)C2=C(C(=O)NC2=O)N BTB12461 c1cc(ccc1NC(=S)NCc2ccncc2)S(=O)(=O)N3CCCCC3 CD00733 c1ccc(cc1)C(c2ccccc2)N3CC(C3)O.Cl BTB10697 c1ccc(cc1)c2ccc(cc2)/C=C/3\c4ccccc4NC3=O CD00742 c1ccc(cc1)COC(=O)NC(Cc2ccc(cc2)O)C(=O)NN BTB13337 c1ccc2c(c1)C(=O)N(C2=O)c3ccc(cc3)[N+](=O)[O-] BTB10700 c1c(cc(cc1C(F)(F)F)NC(=S)N/N=C/c2cc(cc(c2O)Cl)Cl)C(F)(F)F CD03254 COc1cccc(c1O)/C=N/NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03258 CCOc1cc(c(c(c1)OCC)/C=N/O)OCC CD00933 c1cc(cnc1)CNC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00735 CC(=O)CSc1c(c(sn1)SCC(=O)C)C#N CD00738 c1ccc2c(c1)/C(=C\c3ccco3)/C(=O)N2 CD00746 CC(C)c1ccc2c(c1)CCC3C2(CCCC3(C)CNC(=O)NC(C)(C)C)C CD00894 c1ccc(c(c1)CC#N)c2ccccc2CC#N BTB10562 COc1c(c(ccc1)/C=N/c2cc(cc(c2)C(F)(F)F)/N=C/c3c(c(ccc3)OC)O)O CD03241 CCC(CC)(C#C)NC(=S)NCCc1ccccc1 CD00818 CCOc1ccc(cc1OC)/C=C/2\c3ccccc3NC2=O CD00822 c1ccc2c(c1)c(c[nH]2)/C=C/3\c4ccccc4NC3=O CD00823 CSc1[nH]c(=O)c(c(n1)c2cccs2)C#N BTB12621 Cc1cc(c2ccccc2n1)SCC(=O)OC BTB09645 Cc1nc(c(o1)c2ccccc2)c3ccc(cc3)NC(=O)C(C)(C)C BTB09651 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2C(=O)OC)I)C BTB14685 Cc1cc(ccc1Br)NCn2c3ccccc3nn2 BTB14686 c1ccc(cc1)CNC(=O)CC2C(=O)Nc3ccccc3S2 BTB14764 Cc1nc(c(o1)c2ccccc2)c3ccc(cc3)NC(=S)Nc4cccc(c4)C(F)(F)F BTB09659 CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc(c(c2)Cl)F BTB14694 CC(C)(C)C(=O)/C=C/1\C(=O)Nc2ccc(cc2N1)[N+](=O)[O-] BTB13303 CC(C)(C)c1ccc(cc1)/C=C/C(=O)Nc2ccc3c(c2)OCO3 BTB14695 c1cc(ccc1CN(Cc2ccc(cc2)Cl)OC(=O)c3ccc(cc3Cl)Cl)Cl CD05736 c1cc2c(c(c1)F)c(nc3n2nnc3C#N)N CD05745 CC1(CC(=O)C(=NNc2cccc(c2C#N)F)C(=O)C1)C CD05788 Cc1cccc(c1NC(=O)c2c(nns2)C)C CD05497 c1ccn(c1)c2cccc(c2C#N)F CD05646 C[C@@]1(C[C@]1(C)C(=O)NN)C(=O)NN BTB14787 C1COCCN1CC(CN2CCOCC2)C#N CD05230 c1ccc(c(c1)CO)c2ccccc2CO BTB10526 CCCCCCCCc1ccc-2c(c1)Cc3c2ccc(c3)Br BTB10532 c1ccc(cc1)C(=O)c2ccc-3c(c2)Cc4c3cccc4 BTB10537 Cc1cc(c(cc1CNC(=N)NC(=S)N)C)CNC(=N)NC(=S)N.Cl.Cl CD03118 CCCOc1ccccc1NC(=O)CC2C(=O)Nc3ccccc3S2 BTB14768 c1cc(oc1)/C=C(\C#N)/C(=O)c2ccco2 CD05248 COc1ccc(c(c1)C(=O)CC#N)Br CD05258 CN(C)c1ccc(cc1)/C=C(\C#N)/C(=O)c2cc(ccc2Br)OC CD05260 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2cccc(c2)C(F)(F)F CD05370 c1ccc2c(c1)c(c[nH]2)C=C3C(=O)NC(=O)NC3=O CD00824 CN(C)c1ccc(c(c1)Cl)/C=C(\C#N)/C(=O)c2cccs2 CD05225 Cc1cc(c(c(c1NC(=O)C)[N+](=O)[O-])[N+](=O)[O-])C BTB10524 CCc1ccc-2c(c1)Cc3c2cccc3 BTB10530 c1ccn(c1)c2c(c(c(c(c2Cl)Cl)Cl)Cl)Cl CD03282 CC(=CC(=O)ON1C(=O)C2C3C=CC(C2C1=O)O3)C BTB09736 c1cc(sc1C(=O)ON2C(=O)C3C4C=CC(C3C2=O)O4)Cl BTB09738 c1cc(c(c(c1)Cl)CSCC(=O)Nc2ccc(cc2)Cl)F CD05342 CC1(OC(=O)C(=Cc2ccc(cc2)N(C)C)C(=O)O1)C CD05357 COc1ccccc1/C=C\2/C(Oc3ccccc3C2=O)c4ccccc4 BTB13255 Cc1ccc(cc1)/C=C\2/C(Oc3ccccc3C2=O)c4ccccc4 BTB13257 c1cc(c(c(c1)Cl)CN2CCN(CC2)Cc3c(cccc3Cl)F)F CD05364 CC(=O)c1ccc(c(c1)CSCc2cc(ccc2OC)C(=O)C)OC CD05371 c1ccc(cc1)CC(=O)c2ccc(cc2)O BTB12517 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(cc(c3)OC)C(F)(F)F CD03033 COc1ccc(c(c1)/C=C/2\c3ccccc3NC2=O)OC CD00661 CCCCCCCC(=O)c1ccc-2c(c1)Cc3c2cccc3 BTB10531 c1ccc(cc1)COC(=O)CCC(C(=O)O)NC(=O)OCc2ccccc2 BTB13322 CC1(OC(=O)C(=Cc2c(cccc2Cl)F)C(=O)O1)C CD05358 CC(C)(C)OC1CC(N(C1)C(=O)OCc2ccccc2)C(=O)O BTB13324 COc1cccc(c1O)/C=N/NC(=S)NC2CC3CCC2C3 CD03009 c1cc(ccc1NC(=S)NN)S(=O)(=O)N2CCCCC2 CD03020 CN1C2C[C@@H](CC1CC2)/N=C\c3ccccc3.Cl.Cl BTB14839 CN1C2C[C@@H](CC1CC2)NCc3ccccc3.Cl.Cl BTB14840 Cc1ccc(c(c1Nc2ccccc2C(=O)O)C)[N+](=O)[O-] BTB10803 COc1ccc(cc1)[C@H]2[C@@H](C(=O)c3ccccc3O2)OS(=O)(=O)C BTB14845 CCOc1ccc(cc1)/C=N/NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03261 c1ccc(cc1)Cc2coc3ccccc3c2=O BTB12533 c1ccc(cc1)CSc2c(c(c(s2)C(=O)c3ccccc3)N)C(=O)N CD01352 COc1cccc(c1)NC2=C(C(=O)NC(S2)c3ccc(cc3)[N+](=O)[O-])C#N CD01357 c1ccc(c(c1)C(=O)NCc2cccnc2)N CD01358 c1ccc(cc1)COc2ccccc2Cc3coc4ccccc4c3=O BTB12541 Cc1cccc(c1)NC2=C(C(=O)NC(S2)c3ccc(c(c3)OC)O)C#N CD01361 COc1cccc(c1)NC2=C(C(=O)NC(S2)c3cccc(c3O)OC)C#N CD01362 Cc1cccc(c1)NC2=C(C(=O)NC3(S2)CCCC3)C#N CD01363 COc1ccccc1C2CCN(CC2)C(=O)c3ccc(cc3)Cl BTB13421 CC(C)(C)c1ccc(cc1)Oc2cnn(c(=O)c2Cl)c3ccccc3 BTB09715 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2C(=O)NCc3cccnc3 CD01366 c1ccc(c(c1)C(=O)NCc2cccnc2)NC(=O)c3ccc(cc3)Cl CD01367 c1ccc2c(c1)c(c(s2)NC(=O)c3ccccc3C(=O)NCc4cccnc4)Cl CD01368 c1ccc(cc1)OC(=O)NC2CCCCC2 BTB13268 COc1ccc(cc1)/C(=C/c2c[nH]c(n2)c3ccccc3)/C#N BTB09757 CCNC(=O)Oc1ccccc1 BTB13270 c1ccc(cc1)NC(=O)Oc2ccccc2 BTB13271 c1ccc2c(c1)C(C(=O)N2)Cc3ccc(cc3)Cl CD01039 COc1ccc(cc1OC)CCN2C(C(CCC2=O)C(=O)O)c3cc(c(c(c3)OC)OC)OC CD01041 Cc1ccc(cc1)C=C2C(=O)NC(=O)NC2=O CD01081 COc1ccccc1C2CCN(CC2)C(=O)c3cccc4c3cccc4 BTB13418 CCC1(CCCCN(C1=O)C)c2cccc(c2)OC(=O)C3CCCCC3 BTB13424 COc1ccc(cc1OC)CCNC(=S)Nc2cccc(c2)C(F)(F)F CD01085 c1ccn(c1)c2ccc(cc2)Cl CD03747 COc1ccccc1/C=C/2\c3ccccc3NC2=O CD00999 CCCCNS(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)NCCCC BTB13350 CN(C)c1ccc(c(c1C#N)F)Br CD05677 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)ONC(=O)C CD05331 c1cc(c(c(c1)Cl)CN2CCOCC2)F CD05333 COc1ccc(c(c1)CCCCc2cc(ccc2OC)OC)OC BTB14811 CN1C2C[C@@H](CC1CC2)NC(=O)CSc3ccc(cc3)F BTB14823 c1ccc(cc1)Nc2[nH]c(=O)c(c(n2)c3cccs3)C#N BTB12626 c1ccnc(c1)/C=N/NC(=S)NC2CC3CC2C=C3 CD01476 COc1ccc-2c(c1)N3C(c4ccccc4C3=O)c5n2ccc5 CD03466 COc1ccc-2c(c1)NC(c3n2ccc3)c4cc(cc(c4O)Cl)Cl CD03467 c1ccc2c(c1)ccc(c2C3c4cccn4-c5ccccc5N3)O CD03470 Cc1ncc(n1CCO)[N+](=O)[O-] BTB09707 c1cc(ncc1[N+](=O)[O-])NCc2ccncc2 CD01201 c1ccn(c1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03278 c1ccn(c1)c2c(c(cc(c2Cl)Cl)Cl)Cl CD03281 C/C(=N\O)/c1cc(ccc1O)[N+](=O)[O-] BTB12600 c1ccc(cc1)[C@H]2[C@@H](C(=O)c3ccccc3O2)OS(=O)(=O)c4ccc(cc4)Br BTB14848 c1ccc(cc1)C(=O)/C=C/2\C(=O)Nc3ccc(cc3N2)[N+](=O)[O-] BTB13302 CC1N=C(N2N1C(=NC2C)SCc3ccc(cc3)Cl)SCc4ccc(cc4)Cl CD03237 c1ccc2c(c1)c3ccccc3n2CC(CN4CCN(CC4)CC(Cn5c6ccc(cc6c7c5ccc(c7)Cl)Cl)O)O BTB13370 CCCC(=O)Oc1c[nH]c2c1cccc2 BTB13373 c1ccc2c(c1)cccc2C(=O)N3CCc4c(c5cc(ccc5[nH]4)F)C3 BTB13386 CCCCCCc1ccc(cc1)C(=O)CCC(=O)O BTB09812 CCCCCc1ccc(cc1)C(=O)CCC(=O)O BTB09813 c1cc2c(cc1Cl)c(=O)cco2 BTB12537 CC(C)NC(=S)N1CCCN2C1c3ccccc3C2=O CD01304 Cc1cc(c(cc1OC)CCCCCCc2cc(c(cc2OC)C)OC)OC BTB14815 COc1ccc(c(c1)CCCCCc2cc(ccc2OC)OC)OC BTB14816 c1ccnc(c1)Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03424 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)Nc3cccc(c3)C(F)(F)F BTB14777 Cc1ccc-2c(c1)NC(c3n2ccc3)c4cc(cc(c4O)Cl)Cl CD03453 c1cc(ccc1C(C#N)N2CCOCC2)O BTB09801 c1c(cc(c(c1/C=N/NC(=S)N[C@H]2CC3CC2C=C3)O)Br)Br CD03251 CCNc1ccc(cc1)[N+](=O)[O-] BTB13398 CCC(=O)c1ccc(cc1O)NC(=O)C BTB12512 CNC(=S)N/N=C/c1ccc(cc1)N(C)C CD01315 CC1(CC2=C(Cc3cccc(c3O2)OC)C(=O)C1)C CD03290 c1c(cc(cc1C(F)(F)F)NC(=O)C(Cl)(Cl)Cl)C(F)(F)F CD03308 CN1C(=O)C(=Cc2ccccc2)C(=O)N(C1=O)C BTB12474 Cc1cc(nc(n1)SCC(=O)Nc2ccc(c(c2OC)C(=O)OC)OC)C BTB09823 c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)NN)O BTB12485 c1ccc2c(c1)c(=O)c(cs2)Cc3ccc(cc3)Cl BTB14854 c1ccc2c(c1)c(=O)c(cs2)Cc3ccc(cc3)Br BTB14856 c1c(c(sc1C(=O)O)Br)Br BTB12603 c1cc(ccc1NC(=O)C2C3C=CC(C2C(=O)O)O3)[N+](=O)[O-] BTB09721 c1cc(ccc1C=C2C(=O)NC(=S)NC2=O)Cl CD00896 c1cc(sc1)c2c(c(=O)[nH]c(n2)S)C#N BTB09782 c1ccc-2c(c1)NC(c3n2ccc3)c4cc(cc(c4O)Cl)Cl CD01485 CCOC(=O)NC(=S)NNC(=O)c1cccnc1 CD01495 c1cc2c(c(c1)Cl)c(n[nH]2)N CD05676 c1ccc2c(c1)C(c3ccccc3O2)C(=O)N BTB09916 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)Nc3cccc(c3)C(F)(F)F BTB14783 c1c(cc(cc1C(F)(F)F)NNc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD03243 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3c(cccc3Cl)F CD05503 C(C(C(=O)O)Sc1nnc(s1)S)C(=O)O BTB12608 c1cc(ncc1)/C=N/c2ccc(cc2)Cc3ccc(cc3)/N=C/c4ncccc4 CD00949 CC(C)(C)c1ccc2cc(c(cc2c1)C#N)C#N BTB13381 c1ccc(cc1)CCNC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00955 c1cc(ccc1NC(=S)N2CCCC2)S(=O)(=O)N3CCCCC3 CD00962 c1cc2c(cc1F)c3c([nH]2)CCN(C3)C(=O)C4CCCCC4 BTB13384 c1cc2c(cc1F)c3c([nH]2)CCN(C3)C(=O)c4ccc(cc4Cl)Cl BTB13385 CC(=O)Nc1cc(ccc1OC)OC BTB13405 CC1CCCN(C1)C(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00963 c1cc(ccc1NC(=S)N2CCOCC2)S(=O)(=O)N3CCCCC3 CD00964 Cc1nc(cn1CCC#N)[N+](=O)[O-] BTB09769 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NCCCN2CCOCC2)C(F)(F)F CD05572 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)SC3=NC(N4N3C(N=C4SC(=O)c5c(onc5c6c(cccc6Cl)Cl)C)C)C CD05575 c1ccc(cc1)/C=C/C=N/c2ccc(cc2)Cc3ccc(cc3)/N=C/C=C/c4ccccc4 CD00985 c1ccc(cc1)COC(=O)CCC(=O)c2ccccc2 BTB10786 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)ONC(=O)c3ccccc3 CD05602 CCC(C#N)(c1ccccc1)c2ccc(cc2)N BTB10688 c1ccc(cc1)n2c(=O)c(c(cn2)Oc3cccc(c3)C(F)(F)F)Cl BTB09699 C1CCCCCC(=O)C(CCCC1)CCC(=O)O BTB09776 c1ccc2cc(c(cc2c1)C(=O)NN)O BTB10690 COc1cccc(c1)NC(=S)NCCc2ccc(c(c2)OC)OC CD01086 CC(=O)C(C#N)c1cccc(c1)OC BTB10788 c1ccc(cc1)CC(=O)C(c2ccccc2)C(CC(=O)c3ccccc3)c4ccccc4 BTB14800 c1ccc2c(c1)/C(=C\c3ccc(cc3)[N+](=O)[O-])/C(=O)N2 CD01270 c1ccn(c1)c2ccc(cc2)[N+](=O)[O-] CD03723 c1ccc(c(c1)C2=NCCCN2)C(=O)N/N=C/c3ccc(cc3)[N+](=O)[O-] CD01272 Cc1cccc(c1NC(=S)NNC(=O)c2ccccc2C3=NCCCN3)C CD01278 COc1cc(c(cc1Br)OC)CCCCCc2cc(c(cc2OC)Br)OC BTB14813 COc1ccc(c(c1)CCCCCCc2cc(ccc2OC)OC)OC BTB14814 c1ccc(cc1)/C=C/S(=O)(=O)N CD01301 COC(=O)/C(=C\Nc1ccc(nc1)Oc2ccc(cc2F)F)/NC(=O)c3ccccc3 BTB09701 C(CCN)C[C@@H](C(=O)O)NC(=O)C(F)(F)F BTB13344 CNS(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)NC)C2=O BTB13346 c1cc(c(cc1F)NC(=O)CCCC(=O)O)F BTB14709 c1ccc2c(c1)nnn2CNc3ccc(c(c3F)F)F BTB14712 C/C(=N\NC(=O)CC#N)/C(=O)C BTB10692 CCNS(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)NCC BTB13348 CCCCNS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)NCCCC BTB13349 CC(C)CCNS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)NCCC(C)C BTB13351 c1ccc(c(c1)C(=O)NCCNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl CD03722 c1c(cc(c2c1[n+](c(s2)C(=O)NN)[O-])[N+](=O)[O-])C(F)(F)F CD03736 Cc1ccc-2c(c1)NC(c3n2ccc3)c4ccc(cc4)C(=O)O CD03469 CC1N=C(N2N1C(=NC2C)SCc3c(cccc3Cl)F)SCc4c(cccc4Cl)F CD05574 Cc1c(c(n(n1)C(=O)c2cc(c(c(c2)OC)OC)OC)C)/N=N/c3ccc(cc3)Cl CD01514 CCC(=O)c1ccc(cc1OC)OC BTB12500 CN(C)C(=S)c1ccccc1 CD03238 CC1N=C(N2N1C(=NC2C)SCC(=O)c3ccc(cc3)F)SCC(=O)c4ccc(cc4)F CD03239 c1ccc-2c(c1)CC(Cc3c2cccc3)C(=O)O BTB10588 CC1(c2ccccc2-c3ccccc3C(=O)O1)C BTB10589 Cc1ccnc(c1)NC(=O)CSc2ccccn2 CD03477 COc1ccc(c(c1)C(=O)/C(=N/Nc2ccc(cc2)F)/C#N)Br CD05436 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD05437 c1ccc(c(c1)NC(=O)c2c(cccc2Cl)F)SCc3cccc(c3)C(F)(F)F CD05439 COc1ccc(c(c1OC)Cl)/C=N/OC(=O)c2cccs2 BTB09833 c1ccc2c(c1)c(=O)[nH]c(n2)CN3CCCCC3 CD03525 Cc1cc(c(c(c1)C)NC(=O)CSCc2c(cccc2Cl)F)C CD05452 c1cc(c(c(c1)Cl)COc2ccc(cc2)[N+](=O)[O-])F CD05455 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NOC(=O)c3cccs3 CD05466 c1ccc2c(c1)c(nc(n2)CSc3ccccn3)O CD03537 c1ccc(cc1)CN2CCC(CC2)Nc3cccc(c3C#N)F CD05692 c1ccc(cc1)CNS(=O)(=O)c2cc3c(c(c2)[N+](=O)[O-])-c4c(cc(cc4[N+](=O)[O-])S(=O)(=O)NCc5ccccc5)C3=O BTB13353 c1ccc(cc1)CNS(=O)(=O)c2cc3c(c(c2)[N+](=O)[O-])-c4c(cc(cc4[N+](=O)[O-])S(=O)(=O)NCc5ccccc5)C3=C(C#N)C#N BTB13355 CCNS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)NCC BTB13356 CC1(NN(C(=N1)S)c2ccccc2)C CD03248 c1ccc(cc1)COC(=O)c2cc(cc3c2-c4ccc(cc4C3=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB13359 Cc1c(snn1)C(=O)Nc2ccccc2 CD05494 Cc1c(snn1)C(=O)NC2CCCCC2 CD05496 Cc1ccc(cc1)C(=O)O/N=C/c2ccc(c(c2Cl)OC)OC BTB09834 c1ccc2c(c1)nc(c(n2)c3ccccn3)c4ccccn4 BTB10706 CN1C2CCC1CC(C2)NC(=O)c3c(cccc3F)F BTB09838 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Br)Sc3ccccc3N BTB14877 CN1C2CCC1CC(=NO)C2.Cl BTB10716 c1ccc(cc1)C(=CCCC=C(c2ccccc2)c3ccccc3)c4ccccc4 BTB10718 CCOC(=O)/C(=N/Nc1cc(cc(c1)C)C)/C BTB09841 CN1C2CCC1CC(C2)NC(=O)c3cccc(c3)C(F)(F)F BTB09844 c1ccc(cc1)CNC(=O)C(CC(=O)O)C2=CCCCC2 BTB09731 c1c(cc(cc1C(F)(F)F)NC(=O)C(CC(=O)O)C2=CCCCC2)C(F)(F)F BTB09732 c1ccc(cc1)C2/C(=C/c3ccccc3Cl)/C(=O)c4ccccc4O2 BTB13249 CC1CCC(N1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C CD03327 c1ccnc(c1)SCc2csc(n2)c3ccc(cc3)Cl CD03337 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=C(\C(=O)NN)/NC(=O)c4ccc(cc4Cl)Cl BTB14881 c1ccc(cc1)c2c(c(=O)[nH]c(n2)N/N=C/c3ccco3)C#N BTB12630 Cc1c2c(n(n1)c3ccccc3)OC(=C(C2c4ccc(cc4)Br)C#N)N BTB14885 c1ccc(cc1)CNC(=O)/C(=C\c2cn(nc2c3ccccc3)c4ccccc4)/NC(=O)c5ccccc5 BTB14886 c1ccc(cc1)COC(=O)N2C3CC3NC2=O BTB14792 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N CD05279 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(C)C CD05283 CCN(CC)CCNC(=O)c1c(onc1c2c(cccc2Cl)Cl)C CD05285 c1cc(c(c(c1)Cl)Cl)N/C=N/c2cccc(c2Cl)Cl CD05298 Cc1ccc(cc1)S(=O)(=O)N/N=C/C(=O)O BTB10555 c1ccc2c(c1)nc(c3n2ccc3)SCc4c(cccc4Cl)Cl CD03388 c1ccc2c(c1)nc(c3n2ccc3)SCc4nc(no4)c5ccc(cc5)Cl CD03392 c1cc(sc1)/C=N/Nc2[nH]c(=O)c(c(n2)c3ccc(cc3)Cl)C#N BTB12633 CN1C2C[C@@H](CC1CC2)NC(=O)CS(=O)(=O)c3c(cc(cc3)F)F BTB14836 COc1ccc(cc1OC)S(=O)(=O)NCc2c(cccc2Cl)F CD05507 COc1ccc(c(c1)S(=O)(=O)NCc2c(cccc2Cl)F)OC CD05508 COc1ccc(cc1)C(=O)Cc2ccccc2 BTB12518 Cc1nnc(s1)n2cccc2 CD03286 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)SCCC(=O)O BTB14865 Cc1ccc2c(c1)nnc3n2c(=O)[nH]n3 BTB10878 CC1N=C(N2N1C(=NC2C)SC)SC CD03228 CCn1cc(nc1C)[N+](=O)[O-] BTB09705 CC(=O)Nc1ccc(c(c1)Cl)OC BTB10813 CSC1=C(C(=O)NC(S1)c2cccs2)C#N CD01345 CS(=O)(=O)O[C@H]1[C@@H](Oc2ccccc2C1=O)c3ccc(cc3)Br BTB14847 c1ccc2c(c1)c(=O)c(cs2)Cc3ccc(cc3)[N+](=O)[O-] BTB14858 c1cc2c(cc1Cl)nnc3n2c(=S)[nH]n3 BTB10871 c1ccc2c(c1)C(=O)C(=O)N2CCC#N BTB12649 CC(C)CC1(CCCCC1)C/C(=N/NC(=O)N)/C BTBG00002 Cc1ccc(cc1)S(=O)(=O)OCC2CC(C=C2)COS(=O)(=O)c3ccc(cc3)C BTBG00099 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD05605 c1cc(c(c(c1)F)C#N)NCc2cccnc2 CD05632 Cc1coc2ccccc2c1=O BTB12529 COc1cc(nc(n1)N/C=C/2\C(=O)OC(=N2)c3ccccc3)OC BTB09726 CN(CCC#N)c1ccc(cc1)C=C2C(=O)NC(=S)NC2=O CD01010 CC(C)(C)C(=O)Nc1ccccc1C(=O)NCc2cccnc2 CD01370 Cc1cc(n(n1)c2c(c(c(nn2)c3ccccc3)c4ccccc4)c5ccccc5)C BTB13493 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=O)Nc3ccc(cc3)F CD05928 CCc1ccc(cc1)C(=O)O BTB09873 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C(=N/c3ccccc3)/N4CCCC4 CD06193 c1ccc(cc1)S(=O)(=O)/N=C(\NNC(=S)Nc2cc(ccc2Cl)Cl)/N3CCCC3 CD03644 c1cc(ccc1C2CCCCC2)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03594 c1ccc(cc1)S(=O)(=O)/N=C(\NNC(=S)NCc2ccco2)/N3CCCC3 CD03645 CCOC(=O)C(c1ccccc1)C(c2ccccn2)Nc3ccc(c(c3)Cl)Cl CD03656 Cc1ccccc1C(=O)Nc2ccccc2C(=O)NCCc3ccc(c(c3)OC)OC CD01381 c1cc(c(c(c1)Cl)CSc2nnc(s2)N)F CD05854 c1ccc(cc1)C2COc3ccccc3C2=O BTB12542 COc1ccc2c(c1)occ(c2=O)c3ccccc3 BTB12549 CCOC(=O)C(c1ccccc1)C(c2ccccn2)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD03620 c1ccc(c(c1)n2cccc2)SCc3cccc(c3)C(F)(F)F CD03625 CCOC(=O)C(C(c1ccsc1)NC(=S)N)C(=O)C(F)(F)F BTB09803 CCCCCCCc1ccc(cc1)C(=O)CCC(=O)O BTB09808 CCOC(=O)C(=Cc1c[nH]c2c1cccc2)C(=O)OCC BTB10789 CCCCCCCCc1ccc(cc1)C(=O)CCC(=O)O BTB09811 CCCc1ccc(cc1)C(=O)CCC(=O)O BTB09815 CSc1nnc(s1)n2cccc2 CD05860 CCN(c1ccccc1)S(=O)(=O)c2cc(ccc2N)[N+](=O)[O-] BTB13390 CCOc1cc(c(cc1[N+](=O)[O-])OCC)N2CCOCC2 BTB13392 c1ccc(cc1)c2c(nc3ccccc3n2)Nc4cccc(c4)Cl BTB12623 c1ccc(cc1)Oc2c(cccn2)C(=O)ON3C(=O)C4C5C=CC(C4C3=O)O5 BTB09740 c1cc(ccc1c2nnc(o2)c3ccc(cc3)NC(=O)C(Cl)Cl)NC(=O)C(Cl)Cl BTB09742 Cc1cc(n(c(=O)c1C#N)C)C BTB09800 c1ccc(cc1)NN/C(=N/S(=O)(=O)c2ccccc2)/NN CD03626 c1ccc2c(c1)C(C(=O)N2)Cc3ccc(cc3)/N=C/c4cc(cc(c4O)Cl)Cl CD01296 COC1=CC(=O)C=C(C1=O)OC CD01312 CNC(=S)N/N=C/c1cccnc1 CD01313 CSC1=C(C(=O)NC(S1)c2ccc(cc2)Cl)C#N CD01333 CCc1cc2c(cc(=O)oc2cc1OCC(=O)Nc3cccc(c3)C)C BTB14905 c1ccc2c(c1)-c3ccccc3C2(CCC#N)CCC#N BTB12648 c1cc(c(c(c1)Cl)C#N)NCc2cccs2 CD05979 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCOCC3 CD05603 CCOC(=O)CSc1nnc(s1)S BTB12605 CCOC(=O)CCSc1nnc(s1)S BTB12606 c1cc(c(c(c1)Cl)CON2C(=O)C3C4C=CC(C3C2=O)O4)F BTB09748 c1ccc(c(c1)N)SCc2cc(cc3c2OCOC3)Cl CD03406 CC1(CC2=C(C(C3=C(O2)CC(CC3=O)(C)C)c4cccc(c4O)OC)C(=O)C1)C CD03417 COc1cc(cc(c1)n2cccc2)C(F)(F)F CD03423 Cc1ccc(cc1)c2cccc(n2)c3ccc(cc3)C BTB09879 c1cc(sc1C(=O)O)Br BTB12643 CC(=O)CC(=O)NCc1ccccc1 BTB13412 Cc1ccn2c(c1)nc(c2C(=O)N/N=C/c3ccccc3)C BTB13437 CC(=O)c1ccc(c(c1)[N+](=O)[O-])OCc2ccc(cc2)F BTB09854 Cn1cc2c(=O)[nH]nnc2n1 BTB12666 c1ccc(c(c1)SCc2c(cccc2Cl)F)Br CD05546 CC(=O)c1cccc(c1)NC(=O)CCN2C(=O)c3ccccc3C2=O BTB14784 CCc1ccc(cc1)C(=O)CCC(=O)O BTB09816 c1ccc(cc1)c2cccc(n2)c3ccccc3 BTB09880 Cc1ccc(cc1)/N=N/N(C)C BTB14901 Cc1ccc(cc1)C(=O)O/N=C(\C)/c2cc(cc3c2CCC3(C)C)C(C)(C)C BTB09920 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=O)NCCCN(C)C CD05932 CCOC(=O)/C(=C/N(c1ccccc1)/N=C/c2ccccc2)/C#N BTB12656 COc1ccc(c(c1OC)Cl)/C=C/2\C(=O)NC(=S)N2 BTB09821 c1cc(c(c(c1)Cl)C(=O)ONC(=O)c2ccc(c(c2)Cl)Cl)F CD05562 COc1ccc(c(c1)C(=O)ONC(=O)c2ccc(c(c2)Cl)Cl)Br CD05563 c1cc(sc1)CN(CN2C(=O)CCC2=O)CN3C(=O)CCC3=O CD06015 c1ccc2c(c1)C(=O)c3c(ccc(c3C2=O)O)[N+](=O)[O-] BTB13481 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)NN BTB10781 Cc1cc(n(n1)c2ccccc2)N BTB13482 c1ccn(c1)c2c(cccc2Cl)F CD05946 c1c(cc(c2c1C=C3CCCCC3(O2)N4CCCC4)Cl)Cl CD03667 CN1C2CCC1CC(C2)NC(=O)Cc3ccccc3F BTB09836 CC(C)CC1(CCCCC1)/C(=N/NC(=O)N)/C BTBG00046 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)Cl)Cl CD03478 c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)S(=O)(=O)c3ccc(cc3)NC(=S)NC(=O)c4ccccc4 CD01259 c1ccc(c(c1)C(=O)NCCCN2CCOCC2)NC(=O)c3cccc(c3)[N+](=O)[O-] CD01436 COC(=O)c1ccc(cc1)CS(=O)(=O)C CD05666 CCOC(=O)Nc1c(noc1C)C CD05618 c1ccc(cc1)COC(=O)NC(Cc2c[nH]cn2)C(=O)NN BTB13334 C/C(=C\C(=O)NCc1ccccc1)/C(=O)O BTB13484 c1ccc(cc1)Cc2c(c3ccccc3oc2=O)O BTB13487 C/C(=N\O)/CC1(c2ccccc2NC1=O)O BTB10800 COC(=O)CCC(CCC(=O)OC)(C(=O)OC)C(=O)OC BTBG00039 CC(=O)NC1=C(CC(CC1)C(=O)OC)C(=O)OC BTBG00040 c1ccc(cc1)CN2CC3CC(C2C3)C#N BTBG00043 COC(=O)C1CCC(=O)C(C1)C(=O)OC BTBG00047 C1C2CC3CC1C(C(C2)C3=O)C(=O)O BTBG00049 c1cc(ccc1C2=NNC(=O)CC2)Br BTB10814 c1ccc(c(c1)C(=O)NCc2cccnc2)NC(=O)c3ccco3 CD01369 COc1cc2cccnc2c(c1)NC(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB12669 c1cc(c(c(c1)F)C#N)N2CCCC2 CD05628 c1cc(c(c(c1)Cl)CSc2ccc(cc2)Br)F CD05547 CC(C)(C)c1ccc(cc1)C(=O)ONC(=O)c2ccc(c(c2)Cl)Cl CD05564 c1ccc(cc1)CN2CC3CCC2[C@H](C3)O BTBG00045 c1c(cc(cc1C(F)(F)F)NC(=S)NCCN2CCNC2=O)C(F)(F)F BTB12689 c1ccc2c(c1)C(=O)N(C(N2)c3cc(cc(c3O)Cl)Cl)Cc4cccnc4 CD01377 C/C(=N\Nc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])/c2ccc(c(c2)CC#N)OC CD03815 C=CCNC(=O)N1CC(C1)Oc2ccc(cc2)Cl BTB13414 c1cc(oc1)C(=O)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03565 Cc1ccc(cc1)S(=O)(=O)NC(=N)NCCCC(C(=O)O)NC(=O)OCc2ccccc2 BTB13329 CC(C)(C)Oc1ccc(cc1)CC(C(=O)O)NC(=O)OCc2ccccc2.C1CCC(CC1)NC2CCCCC2 BTB13331 COc1ccc(cc1)/C=N/c2ccc(cc2)Cc3ccc(cc3)/N=C/c4ccc(cc4)OC CD00973 COc1ccc(cc1)/C=N/c2ccc(cc2)O CD00977 CC(=C)n1c2ccccc2[nH]c1=O BTB10777 CN(C)c1ccc(c(c1C#N)F)/C=N/O CD06017 CCOC(=O)C1CC2CN(CC(C1)C2=O)S(=O)(=O)c3ccc(cc3)C BTBG00001 C1CC2CCC1CC2C(=O)O BTBG00024 CCOC(=O)/C(=N/Nc1ccc(cc1F)F)/C BTB09842 c1ccnc(c1)CCNc2cccc(c2C#N)F CD05638 c1ccc2c(c1)c(c(s2)C(=O)O/N=C(/c3c(cccc3Cl)Cl)\N)Cl CD03677 c1ccc(cc1)COC(=O)NC(CCCNC(=N)N[N+](=O)[O-])C(=O)O BTB13332 CCOC(=O)/C(=C/c1ccc(c(c1F)C#N)N(C)C)/C#N CD06019 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C(F)(F)F CD03572 c1ccn2cc(nc2c1)c3ccc(cc3)Br BTB09825 Cc1nc(cs1)c2ccc(cc2)OCc3ccc(cc3)F BTB09849 c1cc(ccc1COc2ccc(cc2)/C=C\3/C(=O)NC(=S)S3)F BTB09850 c1ccc2c(c1)C3=NCCCN3C2=O CD01206 CCCCCCCCCCc1ccc(cc1)C(=O)C BTB09790 Cc1ccc(cc1)SCC(=O)N[C@H]2CC3N(C(C2)CC3)C BTB14825 c1cc(c(c(c1)F)C#N)NCCO CD05667 CN(C)CCCNc1cccc(c1C#N)Cl CD05672 c1cc(c(c(c1)Cl)C#N)N2CCCC2 CD05669 COc1ccccc1C2CCN(CC2)C(=O)c3ccccc3 BTB13422 CN1C2C[C@@H](CC1CC2)NC(=O)CSc3c(cc(cc3)F)F BTB14827 COc1ccc(c(c1OC)Cl)/C=N/OC(=O)c2ccc(cc2Cl)Cl BTB09830 COc1cc(cc(c1OC)OC)/C=N/NC(=O)c2ccccc2N CD01424 CN(C)c1ccc(cc1)/C=N/Nc2ccc(cn2)[N+](=O)[O-] CD01178 c1ccnc(c1)C(=N)NNC(=O)c2ccncc2 CD01221 c1ccnc(c1)C(=N)NNC(=O)c2ccco2 CD01222 c1ccnc(c1)c2[nH]nc(n2)c3ccncc3 CD01230 CCSc1[nH]c2ccccc2n1.Cl.Cl BTB13462 CN(C)c1ccc(cc1)C(=O)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03568 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)N CD05470 c1cc2c(nc1)nc(c(n2)O)O BTB09826 COc1ccc(c(c1OC)Cl)/C=N/OC(=O)c2ccc(cc2)C(F)(F)F BTB09831 c1ccc(cc1)c2c(snn2)C(=O)O CC21501 Cc1cc(c(c(c1)C)NC(=O)CS(=O)(=O)Cc2c(cccc2Cl)F)C CD05482 c1cc(ncc1[N+](=O)[O-])N2CCC=CC2 CD01198 C1C=CC2C1C3CC2C(C3)NC(=S)N CD01203 Cc1ccn2c(c1)nc(c2C(=O)N/N=C/c3ccc(cc3)OC)C BTB13441 CSC(=S)Nc1ccc(cc1)Br BTB13455 c1c(cc(c-2c1C(=O)c3c2c(cc(c3)S(=O)(=O)NC4CCCCC4)[N+](=O)[O-])[N+](=O)[O-])S(=O)(=O)NC5CCCCC5 BTB13367 CC(=O)Nc1ccc(cc1)NC(=S)SC BTB13456 C=CCNC(=O)N1CCc2c(c3cc(ccc3[nH]2)F)C1 BTB13383 c1cc(oc1/C=C(\C#N)/C(=O)O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05534 c1cc(c(cc1Cl)Cl)/C=N/OCC(=O)NNC(=O)c2ccc(cc2Cl)Cl CD06202 COc1ccc(cc1)CC(=O)c2ccc(cc2O)OC BTB12526 CN1C2CCC1CC(C2)NC(=O)Cc3ccccc3OC BTB09845 c1ccc(c(c1)n2cccc2)[N+](=O)[O-] CD03294 c1ccc(cc1)C(=O)NOC(=O)c2ccccc2 BTB10705 COc1ccc(c(c1OC)Cl)/C=N/OC(=O)c2ccc(cc2)Cl BTB09832 COc1ccc(c(c1OC)Cl)CSCC(=O)Nc2ccc(c(c2)Cl)F BTB09848 c1ccc(cc1)Nc2nnc(n2c3ccccc3)SCC(=O)O BTB13459 c1ccc2c(c1)nnc3n2c(=O)[nH]n3 BTB10863 c1ccc-2c(c1)NNc3n2c(=O)[nH]n3 BTB10864 CC(C)(C)c1ccc(cc1)S/C(=C/C(=O)O)/C(=O)O BTB09989 Cc1ccc(cc1)S(=O)(=O)NC(CO)C(=O)OC BTB12677 Cc1cccn2c1nc(c2C(=O)N/N=C/c3ccccc3[N+](=O)[O-])C BTB13435 c1ccc(c(c1)C(=O)NCCCN2CCOCC2)NC(=O)c3ccc(cc3)Cl CD01400 COc1ccc(c(c1OC)Cl)CSCC(=O)c2ccc(c(c2)Cl)Cl BTB09847 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3ccccc3OC BTB13419 CC(=C/C(=N/Nc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])/C)C CD03822 COc1cccc(c1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC CD03839 c1cc(ccc1c2nc(cs2)CN3CCOCC3)Cl CD03315 CCOc1ccc(cc1OC)C(CC(=O)c2ccccc2)Sc3ccccc3N BTB14875 Cc1cc2cc(ccc2[nH]1)OC BTB13426 Cc1c(cc2c(c1/N=C/c3cc(cc(c3O)Cl)Cl)C(CC2(C)C)(C)C)/N=C/c4cc(cc(c4O)Cl)Cl CD03871 COc1ccc(cc1)Nc2c(nc3ccccc3n2)c4ccccc4 BTB12625 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=O)NCc3ccc(cc3)Cl CD05929 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=O)NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C CD05930 c1ccc(c(c1)C(=O)NCCc2ccccn2)N CD01388 Cc1csc(c1c2ccccc2)c3ccccc3 BTB10740 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2C(=O)NCCc3ccccn3 CD01392 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)NC2CC3CC2C=C3 CD01405 c1ccc(cc1)c2c(nc3ccccc3n2)c4ccccc4 BTB14869 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=O)OCC#C CD05935 C/C(=N\Nc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])/c2cccnc2 CD03843 c1cc(c(c(c1)Cl)C#N)N2CCOCC2 CD05675 c1c(cc(cc1C(F)(F)F)NC(=O)CC#N)C(F)(F)F CD03206 CNS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)NC BTB13363 c1ccc(cc1)/C=C/C=N/NC(=O)CS(=O)(=O)Cc2cccc(c2)C(F)(F)F CD03885 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC(=O)c3c(cccc3Cl)Cl CD05883 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N3CCCC3=O CD05887 CCOC(=O)C(c1ccccc1)C(c2ccccn2)Nc3ccccc3 CD03634 C/C(=N\Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/c2ccccc2 BTB12704 c1ccc2c(c1)ccnc2NC(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB12705 c1ccc(cc1)COc2cc(cc(c2OCc3ccccc3)OCc4ccccc4)[N+](=O)[O-] BTB10049 c1ccc(cc1)c2cccc(c2)c3ccccc3 BTB10963 c1ccc2c(c1)C3c4ccccc4C2C(C3C(=O)O)C(=O)O BTBG00146 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=S)N3CCOCC3 CD05943 CCn1c2ccccc2c(c(c1=O)c3ccccc3)O BTB10848 COc1ccc(cc1OC)CCNc2ccc(cc2[N+](=O)[O-])Cl CD01594 COc1cccc2c1OC3(CCCCC3C2C[N+](=O)[O-])N4CCOCC4 CD01412 c1cc(ccc1c2csc(n2)N3CCOCC3)[N+](=O)[O-].Br CD01165 c1cc(ccc1CSc2nnc(s2)SCc3ccc(cc3)Br)Br CD01420 c1ccc(c(c1)N)n2cccc2 CD01423 c1ccc2c(c1)c3ccccc3n2CCC#N BTB12647 Cc1ccc(n1CCn2c(ccc2C)C)C BTB12650 c1ccc(cc1)/C(=N/O)/CNC(c2ccccc2)(c3ccccc3)c4ccccc4 BTBG00061 C/C(=N\Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/c2ccc(c(c2)CN3CCOCC3)OC CD03754 CN(C)C(=O)c1cccc2c1-c3ccccc3C2=O BTB10968 CNC(=O)c1cccc2c1-c3ccccc3C2=O BTB10974 c1cc(c(c(c1)Cl)/C(=N/OC(=O)c2ccc(cc2)[N+](=O)[O-])/N)Cl CD03678 c1ccc(c(c1)n2cccc2)SCc3ccc(cc3)Cl CD03612 c1cc(sc1)CNC(=O)CC#N CD05988 Cc1c(c(c(c(c1C)C)C(=O)c2cc(c(c(c2)OC)OC)OC)C)C CD01713 Cc1c(c(c(c(c1C)C)CSCC(=O)N/N=C/c2ccncc2)C)C CD01714 Cc1c(c(c(c(c1C)C)CSCC(=O)N/N=C/c2ccc(c(c2)Cl)Cl)C)C CD01719 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCC(=O)c3ccccc3 CD06043 c1ccc(cc1)CSCC(=O)O CD04055 Cc1c(c(c(c(c1C)C)C(C)O)C)C CD01740 c1cc(ccc1CC#N)NC(=O)c2ccc(cc2)Cl CD01745 c1ccc(cc1)S(=O)(=O)/N=C(/NN)\N2CCCC2 CD03618 COc1ccc(c(c1OC)Cl)/C=C/2\C(=O)OC(=N2)c3ccccc3 BTB09819 c1cc(cc(c1)F)C2(CCCCC2)O BTB12754 c1ccc(cc1)/C=C/c2nc(no2)c3ccc(cc3)Cl CD04012 CC(=O)NNC(=O)c1cccnc1 CD04013 COc1cccc(c1C(=O)NNC(=O)c2cccnc2)OC CD04023 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2nnc(s2)SCC(=O)c3cccc(c3)[N+](=O)[O-] CD01417 c1cc(oc1c2nnc(s2)N)[N+](=O)[O-] BTB10020 Cc1ccc(cc1)/C=N/NC(=O)c2c(nc3n2ccc(c3)C)C BTB13439 Cc1c(c(c(cn1)CSc2ccc(cc2)Cl)CO)O CD04095 CCOC(=O)C(CCC(=O)O)(CCC(=O)O)C(=O)C BTBG00032 CC(C)(C)C#CC(C#CC(C)(C)C)(C#CC(C)(C)C)O BTBG00034 COc1ccc(c(c1OC)Cl)C=C2C(=O)NC(=O)NC2=O BTB09820 c1cc(ccc1C(=O)O)S(=O)(=O)N BTB13399 CC12CCC(CC1)(CC2)C(C)(C)O BTBG00137 CCNS(=O)(=O)c1ccc(cc1)C BTB12698 C/C(=N\O)/CCc1ccc(c(c1)OC)O BTB09937 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)C)C)NC(=O)c2cccc(c2)Cl BTB13580 CCOC(=O)C(Cc1cccc(c1)C(=O)OC)NC(=O)c2ccccc2 BTB09994 CC(C)(C)/C(=N/O)/c1ccccc1 BTBG00062 C1CC2C(CCCC2=O)/C(=N/O)/C1 BTBG00068 c1cc(c(cc1Cl)Cl)/C=C/2\C(=O)NC(=S)S2 BTB10821 c1ccc(cc1)COc2ccc(cc2Cl)[N+](=O)[O-] BTB10824 c1cc(nc(c1)CSC2=NCCS2)CSC3=NCCS3 BTB14891 CSC1=N/C(=C/c2ccco2)/C(=O)N1 BTB12638 CSC1=N/C(=C/c2cccs2)/C(=O)N1 BTB12639 CS/C(=N\c1ccccc1)/Nc2ccccc2 BTB09958 COC(=O)C1CC2(CC(C1=O)(CC(C2=O)C(=O)OC)C(=O)OC)C(=O)OC BTBG00054 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCCN(C)C)C)C CD06110 CC1(CC2=C(C(C(=C(O2)N)C#N)c3cn(nc3c4ccccc4)c5ccccc5)C(=O)C1)C BTB14882 c1ccc2c(c1)[nH]c(n2)c3cccs3 BTB10837 Cc1c(snn1)c2nc(on2)CS(=O)(=O)c3ccc(cc3)Cl CD05771 c1cc(c(c(c1)F)C#N)NN=C(C#N)C#N CD05773 c1cc(c(c(c1)Cl)CNCc2c(cccc2Cl)F)F CD05798 Cc1c2c(n(n1)c3ccccc3)OC(=C(C2c4ccc(cc4)Cl)C#N)N BTB14884 C1CC(C(C1)NC(=S)NC2CC3CC2C=C3)CNC(=S)NC4CC5CC4C=C5 CD01579 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2N3CCCCC3 CD01583 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)N3CCCCC3 CD01587 CCOC(=O)c1cc(=O)c2c(cccc2o1)O BTB09948 CN(C)c1cccc2c1c(ccc2)N(C)C BTB09871 c1cc(sc1)CNC=C(C#N)C#N CD05982 CC(C)c1ccc(cc1)NC(=S)OC CD03931 c1ccc(cc1)c2c(c(=O)[nH]c(n2)N/N=C/c3cccs3)C#N BTB12632 COC(=O)c1cccc2c1-c3ccccc3C2=O BTB10905 c1ccc(c(c1)C(=O)NCCCN2CCOCC2)N CD01395 c1cc(c(c(c1)F)C(=O)Nc2cccc(n2)NC(=O)c3c(cccc3F)F)F CD03958 c1ccc(cc1)NC(=S)Nc2ccccc2n3cccc3 CD01527 c1cc(sc1)C/N=C/c2cccs2 CD06070 C1CC(=O)C(C(=O)C1)CCC#N BTBG00003 CCCCN1C(=O)c2cccc3c2c(ccc3N)C1=O BTB10776 Cc1cc(=O)oc2c1ccc(c2)N BTB10779 c1ccc2c(c1)c(=O)[nH]c(n2)CSc3ccccc3N CD03535 CCCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB10910 Cc1ccn2c(c1)nc(c2C(=O)N/N=C/c3ccc(cc3)Cl)C BTB13438 COc1cccc2c1[nH]c(cc2=O)C(=O)OC BTB10048 CCCCCCCCc1ccc(cc1)C(=O)O BTB09861 CS/C(=N\c1ccccc1C(F)(F)F)/N2CCCC2.I CD06210 CCCCCCc1cc2c(cc(=O)oc2cc1O)C BTB10067 c1cnccc1C(=O)NNC(=S)NC2CC3CC2C=C3 CD01403 c1cc(cnc1)C(=O)NNC(=S)NC2CC3CC2C=C3 CD01404 c1ccc2c(c1)C3NCCCN3C2=O CD01280 c1ccc(c(c1)C2=NCCCN2)C(=O)NNC(=S)Nc3cccc(c3)C(F)(F)F CD01277 c1ccc(c(c1)C2=NCCCN2)C(=O)NNC(=S)Nc3ccccc3Cl CD01279 Cc1ccc(cc1[N+](=O)[O-])Br BTB09868 c1ccn(c1)Cc2cccs2 CD06058 c1ccc(cc1)N2c3ccccc3C(=O)C(C2=O)(Cl)Cl BTB13508 CN(C)c1ccc(cc1)C(=O)N/N=C/c2cc(c(c(c2)OC)OC)OC CD01793 Cc1cc(c(c(=O)o1)C(=O)/C=C/N(C)C)O BTB10069 C1C2C=CC1C(C2C(=O)O)C(=O)O BTBG00141 C1CC2CCC(C1)C(C2C(=O)O)C(=O)O BTBG00142 c1ccc2c(c1)[nH]c(n2)SCc3cccc(n3)CSc4[nH]c5ccccc5n4 BTB14890 CCOC(=O)CO/N=C/c1c(cccc1Cl)Cl CD06115 c1ccc(cc1)/C(=N\O)/C2CC3CCC2CC3 BTBG00007 Cc1c(c(c(c(c1C)C)COC(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C)C)C CD06041 CCOC(=O)C(CCC#N)(CCC#N)C(=O)C BTBG00015 Cc1ccc(cc1)S(=O)(=O)N2CCCC2=O BTB12682 Cc1ccc(cc1)S(=O)(=O)NN=C2C3CC4CC(C3)CC2C4 BTB12680 COc1ccc(cc1OC)CCNC(=O)c2ccccc2/N=C/c3cc(cc(c3O)Cl)Cl CD01372 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNC(=O)CO/N=C/c3ccc(cc3Cl)Cl CD06111 c1ccc(cc1)CN2C(SCC2=O)c3cn(nc3c4ccccc4)c5ccccc5 BTB14883 Cc1ccc(cc1)S(=O)(=O)OCC(C)(C)C BTB12747 Cc1ccc2c(c1)nnc3n2cnn3 BTB10873 c1ccc(c(c1)C(=O)NCCc2ccccn2)NC(=O)c3ccc(c(c3)Cl)Cl CD01435 c1ccc2c(c1)c(c(s2)C(=O)NNC(=O)/C=C/C(=O)O)Cl CD01471 c1cc(ccc1Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])I CD03591 c1cc(c(c(c1)F)C#N)NCc2cccs2 CD05980 c1ccc(cc1)CN2C3CCC(C2=O)CC3O BTBG00038 c1ccc(c(c1)NC(=S)Nc2ccc(c(c2)Cl)Cl)SCc3cc(cc4c3OCOC4)Cl CD03797 COC(=O)/C(=C/C(=O)c1ccc(cc1)Cl)/Nc2ccccc2 BTB13534 Cc1c2c(n(n1)c3ccccc3)OC(=C(C2c4ccccc4)C#N)N BTB12667 c1ccc(c(c1)NC(=O)c2c(cccc2F)F)NC(=O)c3c(cccc3F)F CD03954 c1cc(ccc1c2nc(c3c4c(sc3n2)CCCCC4)N)Cl CD01512 CCOC(=O)CCc1ccc(cc1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03595 c1cc(cc(c1)NC(=S)Nc2ccc(c(c2)Cl)Cl)C(F)(F)F CD03979 c1ccc2c(c1)c(nc(n2)CN3CCOCC3)O CD03523 CC(=O)c1ccc(c(c1)n2cccc2)Cl CD03532 COC12CCC(CC1)C(C2)(C#N)O BTBG00029 c1ccc(c(c1)C(=O)N)NC(=O)CN2CCOCC2 CD03540 c1cc(c(c(c1N2CCCCC2)C(=O)O)N3CCCCC3)[N+](=O)[O-] CD03548 CC(=O)c1ccc(c(c1)[N+](=O)[O-])OCc2ccc(c(c2)Cl)Cl BTB09855 CCCCCCN(CCCCCC)c1ccc(cc1)C(=O)O BTB09858 Cc1ccc(cc1)S(=O)(=O)NCCCCCC(=O)O BTBG00084 Cc1ccc(cc1)S(=O)(=O)OCC23CC4CC(C2)CC(C4)C3 BTBG00085 CCCCCCc1ccc(cc1)C(=O)O BTB09862 CC(=O)C1CCc2cc(ccc2C1=O)OC BTB10051 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)Sc3ccccc3N BTB14876 Cc1ncc(n1CCOC(=O)c2ccc(cc2Cl)Cl)[N+](=O)[O-] BTB14879 C1CC(C2CC1C(C2)C(=O)O)O BTBG00035 Cc1ccc(cc1)S(=O)(=O)OC2C3CCCC2CN(C3)C BTBG00036 c1ccc(cc1)C(=O)CCCCCCCCC(=O)c2ccccc2 BTBG00037 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)NC(=O)CCC(C(=O)O)NC(=O)OCC4c5ccccc5-c6c4cccc6 BTB10799 C[C@H](C(=O)OCc1ccccc1)N.Cl BTB13569 Cc1ccc(cc1)S(=O)(=O)O.C[C@@H](C(=O)OCc1ccccc1)N BTB13570 c1cc(cc(c1)Cl)C(=O)NNC(=O)CO/N=C/c2c(cccc2Cl)Cl CD06198 c1cc(c(c(c1)Cl)/C=N/OCC(=O)NNC(=O)c2ccc(cc2)Cl)Cl CD06205 COc1ccc2c(c1)nnc3n2c(=O)[nH]n3 BTB10883 Cc1ccc(cc1)S(=O)(=O)N(C)C BTB12748 CC1CC(C(CC1C)C(=O)O)C(=O)O BTBG00086 CC1C[C@H](C(CC1C)C(=O)O)C(=O)O BTBG00091 CCC(CC)(C#C)NC(=O)/C=C\C(=O)O CD01472 c1ccc(cc1)C2(C(=O)NC(=O)N2)c3ccccc3 BTB14870 c1ccc2c(c1)[nH]c(n2)CCS(=O)(=O)CCc3[nH]c4ccccc4n3 BTB13449 CCOC(=O)CS(=O)(=O)C(c1ccccc1)S(=O)(=O)CC(=O)OCC BTB13450 COc1ccc(cc1)C(SCC(=O)O)SCC(=O)O BTB13451 CC(C)(C)NS(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)NC(C)(C)C)C2=O BTB13365 c1ccc-2c(c1)Cc3c2c(ccc3)C(=O)O BTB10913 c1ccc(cc1)C(CCC#N)(CCC#N)C#N BTB12645 c1ccc(cc1)c2ccccc2c3ccccc3 BTB10962 C1CC(CC=C1)C(C#N)N2CCOCC2 BTB12651 c1ccc2c(c1)C/C(=C/C3CCC=CC3)/C2=O BTB12653 c1ccc(cc1)C(CC(=O)C2CC2)Nc3ccccc3 BTB13464 c1ccc(cc1)COc2cccc(c2OCc3ccccc3)CCC#N BTB09977 c1ccc(cc1)C2C3CC4CC(C3)CC2C4 BTBG00048 COC(=O)C1C(NC(C(S1(=O)=O)C(=O)OC)c2ccccc2)c3ccccc3 BTB13461 C/C(=C\1/C(=O)OC(=N1)c2ccccc2)/Nc3ccccc3 BTB12671 c1cc(c(c(c1)F)C#N)NC(=O)c2ccc(cc2Cl)Cl CD05867 Cc1c(c(n(n1)C(=O)c2ccc(cc2)[N+](=O)[O-])C)/N=N/c3ccc(cc3)Cl CD01518 Cc1csc(n1)NC(=N)N.Cl CD01619 CCNc1cc(=N)n(c2c1c(c(s2)C(=O)OCC)N)CC CD03752 c1ccc(cc1)c2c(c3ccccc3n(c2=O)c4ccccc4)O BTB13518 c1ccc(cc1)c2ccccc2S(=O)(=O)c3ccc(c(c3)Cl)Cl BTB13465 Cc1ccc(cc1)S(=O)(=O)NNc2c(c(c(nn2)c3ccccc3)c4ccccc4)c5ccccc5 BTB13527 c1ccc(cc1)C(=O)/C=N/Nc2ccc(cc2)Cl BTB10833 Cn1c2ccccc2nc1c3cccs3 BTB10838 c1ccc(c(c1)NC(=S)NNC(=S)NC2CC3CC2C=C3)Cl CD01407 CC1(OC(=O)C(=Cc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)O1)C CD05530 CCNc1c(c(nn1c2ccccc2)C)[N+](=O)[O-] BTB13521 CC1CCCCN1CCCNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB12703 CC(=O)NC1CCC(CC1C(=O)OC)C(=O)OC BTBG00028 c1cc(oc1C=C2C(=O)NC(=S)NC2=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04081 CC(C)(C(=O)O)C(C)(C)NC(=O)OC BTBG00109 c1ccc(cc1)CCNC(=S)NNC(=S)NC2CC3CC2C=C3 CD01408 COc1ccccc1NC(=S)NNC(=S)NC2CC3CC2C=C3 CD01410 C(C#N)Sc1nnc(s1)SCC#N CD01419 C/C(=C\1/c2ccccc2NC1=O)/CCc3ccc(cc3)OC CD01544 CCOC(=O)C1CCN(CC1)C(=S)NC2CC3CC2C=C3 CD01563 c1ccc(cc1)c2c3c([nH]nc3N/N=C/4\C(=O)N=C5C=CC=CN5C4=O)nnc2c6ccccc6 BTB13496 c1ccc\2c(c1)CSC/C2=N\Nc3ccc(cc3[N+](=O)[O-])S(=O)(=O)N CD04214 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccccc3N4CCCCC4 CD01584 Cc1c(nc(o1)c2ccccc2)CC(=O)O BTB09929 COc1ccc2c(c1)c(ccn2)C(=O)C3CC4CCN3C(C4)C=C BTB09931 c1ccc(cc1)c2cc(n(n2)CCC#N)O CD05719 c1ccc2c(c1)nnc3n2c(=S)[nH]n3 BTB10862 COc1cc(c(cc1OC)[N+](=O)[O-])CC(=O)O CD01521 COc1cc(c(cc1OC)[N+](=O)[O-])CC(=O)OC CD01523 COc1ccc(cc1O)[C@H]2CC(=O)c3c(cc(cc3O2)O)O BTB12807 c1ccc\2c(c1)CSC/C2=N\OCc3c(cccc3Cl)Cl CD04230 CC(=O)Nc1c(cccc1F)F CD04232 CCOC(=O)c1c(c(c(n1c2ccccc2)C(=O)OCC)O)O BTB10028 Cc1cc(c(cc1N2Cc3ccccc3C2)C)/N=N/c4ccc(cc4)Br BTB11013 CCCc1c2c(cc3c1oc(cc3=O)C(=O)OCC)CCCC2 BTB10009 c1ccc(cc1)NC2=CC(CC2=O)N3CCCCC3 BTB10021 c1cc(ccc1[N+](=O)[O-])OC2CCC3CCC2C3 BTB12709 COc1ccc(cc1)NC(=O)CSCC(=O)N CD01698 CC(C(=O)c1ccccc1)N2CCOCC2.Br BTB12700 c1c(cc(cc1C(F)(F)F)NCCC#N)C(F)(F)F CD04233 Cc1cc(ccc1n2c(=O)c3ccccc3nc2Sc4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Br CD04236 Cc1ccc2c(c1S(=O)(=O)O)sc(n2)c3ccc(cc3)N BTB13613 Cc1c(c(c(cn1)CSc2ccccc2N)CO)O CD04096 CC(C)(C)c1cc2c(=O)cc(oc2c(c1)C(C)(C)C)C(=O)O BTB10109 C1CC2C=CC1CC2C(=O)O BTB12713 c1cc2c(cc1C(=O)CCC(=O)O)OCCCO2 BTB12796 CC(=O)c1cc2c(cc1Br)OCCO2 BTB12797 CC(=O)NC(CCCNC(=N)N)C(=O)O BTB13542 CC(=O)N[C@@H](CC(=O)N)C(=O)O BTB13544 CC(C)NC(=S)NNC(=S)NC1CC2CC1C=C2 CD01409 c1cc(oc1/C=N/Nc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04105 c1cc(ccc1N2CCC(=O)N2)Cl BTB10095 Cc1c(cc2c(c1N)C(CC2(C)C)(C)C)NC(=S)Nc3ccc(cc3)OC CD03896 c1ccc(c(c1)N)NC(=O)c2c(cccc2F)F CD03905 CC(=O)c1ccc-2c(c1)Cc3c2ccc(c3)C(=O)C BTB10893 c1cc(ccc1C23CC4CC(C2)CC(C4)C3)OCC(CN5CCCCC5)O.Cl BTB12794 c1cc(ccc1C(=O)N(CC#N)CC#N)Cl CD06274 c1cc(cc(c1)Cl)C(=O)N(CC#N)CC#N CD06275 c1cc-2c(cc1Br)Cc3c2ccc(c3)Br BTB10903 c1cc2c(cc1N)OCCCO2 BTB12798 CC(=O)c1cc2c(cc1Br)OCCCO2 BTB12799 CC1(OC(=O)C(=Cc2ccc(cc2Cl)Cl)C(=O)O1)C CD06279 c1cc(c(cc1F)F)NCN2C(=O)CCC2=O CD06292 CC(C)/C(=N\O)/c1ccc(cc1)OC BTBG00075 CNC(=O)NCc1c(cccc1Cl)F CD06055 c1ccc-2c(c1)Cc3c2c(ccc3)C#N BTB10886 C/C(=N\O)/C(=C)c1ccccc1 BTBG00181 CS/C(=N\c1ccc(cc1)Cl)/NCc2ccco2.I CD06257 Cc1ccc(cc1OC)/C=N/NC(=S)NC2CC3CC2C=C3 CD01757 c1cc(c(c(c1)F)C(=O)NNC(=O)c2cccnc2)F CD03999 c1cc(ccc1/C=N/NC(=S)NC2CC3CC2C=C3)[N+](=O)[O-] CD01760 c1cc(sc1)/C=N/NC(=S)NC2CC3CC2C=C3 CD01771 CN(C)c1ccc(cc1)C(=O)NN CD01774 c1ccc(cc1)CC(=O)c2cccs2 BTB12887 Cc1c(c(c(c(c1C)C)C=C2C(=O)OC(OC2=O)(C)C)C)C CD06090 c1ccc(cc1)CNC(=O)/C(=C\c2cn(nc2c3ccccc3)c4ccccc4)/NC(=O)c5ccc(cc5Cl)Cl BTB14880 CCCCCCCCN1C(=O)c2cccc3c2c(ccc3/N=N\c4ccc(cc4)N(CC)CC)C1=O BTB10943 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NN=C(C(=O)C)C(=O)C CD03973 CC(=O)Nc1ccc(cc1)CC#N BTB10998 c1cc(c(c(c1)F)C(=O)O/N=C(/c2ccc(cc2)Cl)\N)F CD04007 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(cc2Cl)Cl)Cl CD06128 c1ccc2c(c1)c3c([nH]2)CNC(C3)C(=O)O BTB10915 Cn1c2ccccc2c3c1ccc(c3)[N+](=O)[O-] BTB12828 c1ccc2c(c1)nc(s2)c3cccs3 BTB10835 c1ccc(cc1)/C=C/c2cccs2 BTB10836 Cc1nnc(n1c2ccccc2)S BTB12615 c1ccc(cc1)n2c(=O)cc(c(n2)C(=O)N)O BTB12617 c1ccc(cc1)c2cc3ccccn3c2 BTB12618 c1ccc(cc1)c2c(nc3ccccc3n2)Nc4ccc(cc4)Cl BTB12624 COC(=S)Nc1ccc(cc1)F CD03993 CC(=O)c1c(ccc(c1O)C(C)(C)C)OCc2ccccc2 BTB10000 c1cc-2c(cc1[N+](=O)[O-])C(=C(C#N)C#N)c3c2ccc(c3)[N+](=O)[O-] BTB10966 CC(=O)c1ccc(cc1OCc2ccccc2)OC BTB10072 CC(C)C[C@H](C(=O)O)NC(=O)C BTB13549 CC(C)C[C@@H](C(=O)O)NC(=O)C BTB13550 CC(CSC(=O)C)C(=O)O BTB13552 c1cc(c(cc1Cl)Cl)C(=O)N(CC#N)CC#N CD06293 C1C2CC(C1C=C2)NC(=S)NNC(=O)CC#N CD01610 c1cc(ccc1c2csc(n2)NC(=N)N)[N+](=O)[O-].Br CD01617 CC(CCC(C)OC(=O)c1ccccc1C(=O)O)OC(=O)c2ccccc2C(=O)O CD03934 c1ccc(cc1)/C=C/C=N/NC(=S)NC2CC3CC2C=C3 CD01759 C1C2CC(C1C=C2)NC(=S)NNC(=S)NC3CC4CC3C=C4 CD01411 c1ccc(cc1)C(=O)CSc2nnc(s2)SCC(=O)c3ccccc3 CD01416 c1ccc(cc1)COc2c(c(oc2C(=O)O)C(=O)O)OCc3ccccc3 BTB10004 CCCc1cc(c(c2c1oc(cc2=O)C(=O)OCC)O)[N+](=O)[O-] BTB10102 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(cc2Cl)Cl)F CD06127 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)O BTB10912 Cn1c2ccccc2c(c(c1=O)Cc3ccccc3)O BTB13517 c1ccc(cc1)Nc2ccc(c(n2)Nc3ccccc3)[N+](=O)[O-] BTB12822 Cc1c(c(sc1C#N)C(=O)N)C CD06066 CC(=O)NC(Cc1ccccc1)C(=O)O BTB13558 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OCC=C BTB10041 c1c(cc(cc1C(F)(F)F)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD06116 c1ccnc(c1)CCNC(=O)/C(=C/c2ccc[nH]2)/C#N CD01686 c1cc2c(cc1[N+](=O)[O-])c3cc(ccc3[nH]2)[N+](=O)[O-] BTB12827 CCN(CC)CCCNS(=O)(=O)c1c(c(c(c(c1C)C)C)C)C CD06144 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])c2ccc(cc2[N+](=O)[O-])C(F)(F)F CD04256 c1ccc2c(c1)-c3cccc(c3C2=O)C(=O)O BTB12831 C/C(=N\Nc1c(c(c(nn1)c2ccccc2)c3ccccc3)c4ccccc4)/c5ccccc5 BTB13523 c1ccc(cc1)c2c(c(nnc2c3ccccc3)NNS(=O)(=O)c4ccccc4)c5ccccc5 BTB13526 CCCCCCCCCCCCCCCCCC(=O)c1cccs1 BTB12888 c1cc2c(cc1Cl)nnc3n2c(=O)[nH]n3 BTB10872 CC(=O)N/N=C/c1ccccc1 BTB12720 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)Nc2ccccc2Cl)C)C CD01694 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)NCCc2ccccc2)C)C CD01697 Cc1ccc(cc1C)NC(=S)N/N=C/2\CSCc3c2cccc3 CD04244 CC1(CC(=O)C(=NNc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C(=O)C1)C CD04261 COc1cccc(c1NC(=O)c2c(cccc2F)F)OC CD04267 CCC(C)(C)/C(=N/O)/c1ccccc1 BTBG00064 c1cc(sc1)CNC(=O)c2cccs2 CD06419 c1cc(sc1)CNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD06420 Cc1cc(=O)oc2c1ccc(c2C(=O)C)O BTB09970 CC(C)(C(CC(=O)c1ccccc1)c2ccccc2)[N+](=O)[O-] BTB12712 c1ccc(c(c1)/C=N/NC(=S)NC2CC3CC2C=C3)Cl CD01475 COc1ccc(cc1)C2c3cccn3-c4ccccc4N2 CD01487 Cc1ccc(cc1)C2=C(C(=O)C(=C2c3ccc(cc3)Cl)c4ccccc4)c5ccccc5 CD01491 Cc1cc(c(c2c1C(=O)C(C2)(C)C)C(=O)Nc3cccc(c3)C(F)(F)F)C CD01507 c1ccc(cc1)n2c(c(sc2=S)C#N)N CD01509 c1ccc(cc1)/C=C/C(=O)O/N=C(/c2ccc(cc2)Cl)\N CD04005 c1cc(ccc1C(=O)OCC#Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] CD04251 C/C=C(/c1ccccc1)\C(=O)O BTBG00057 CS/C(=N\c1cccc(c1)C(F)(F)F)/N2CCCC2.I CD06244 CCCc1cc(=O)c2ccc(cc2o1)OC/C(=N/O)/C BTB09972 COc1cc(c(cc1OC)Br)CCC#N BTB09973 Cc1ccc(cc1)S(=O)(=O)NCc2cccs2 CD06405 COc1cccc(c1O)/C=N/NC(=O)C2CCCN(CC2)C(=S)NNC3CC4CC3C=C4 CD03637 c1cc(c(c(c1)F)c2nc(no2)c3ccc(cc3)Cl)F CD04006 CSc1cccc(c1)NC(=S)NN/C(=N\S(=O)(=O)c2ccccc2)/N3CCCC3 CD03646 c1ccc(cc1)S(=O)(=O)/N=C(\NNC(=S)Nc2cccc(c2)C(F)(F)F)/N3CCCC3 CD03647 CC1CC(CC(C1)(C)C)NC(=O)/C(=C/c2ccc[nH]2)/C#N CD01688 CS/C(=N\c1ccccc1F)/N2CCCCC2.I CD06262 c1ccc(c(c1)C(=O)NCc2cccs2)Cl CD06369 CN(C)C(=S)SCc1ccccc1C(=O)Oc2c(cccc2Cl)Cl CD06367 Cc1cc(c(cc1N2Cc3ccccc3C2)C)/N=N/c4ccc(cc4)C(=O)C BTB11015 COc1cc(c(c(c1OC)Cl)C#N)[N+](=O)[O-] BTB09918 C/C(=N\OC(=O)c1cccs1)/c2cc(cc3c2CCC3(C)C)C(C)(C)C BTB09919 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2cc(cc3c2CCC3(C)C)C(C)(C)C BTB09921 Cc1c(cccc1OCc2ccccc2)[N+](=O)[O-] BTB09953 CCn1c2ccc(cc2c(=O)cc1C(=O)OC)OC BTB09952 Cc1ccc(c(c1)C)NC(=S)NNC(=O)CCOc2ccc(cc2)OC CD01777 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCCN2CCCCC2C)C)C CD06145 Cc1ccc(cc1[N+](=O)[O-])OCc2ccccc2 BTB09965 C1CC2CCC1CC2C(=O)N BTBG00135 c1cc(cnc1)C(N2CCOCC2)N3CCOCC3 CD04143 c1cc(oc1/C=C/C(=O)O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04150 CN(CC(=O)Nc1ccccc1)C(=O)c2ccccc2 BTBG00066 CCCc1c(cc(cc1[N+](=O)[O-])C(=O)O)[N+](=O)[O-] BTB10008 Cc1cccc(c1N/C(=N/C(C)(C)CO)/SC)C.I CD06208 CC(C)CCOC(=O)C1(CC2(C1)COC(OC2)c3ccccc3)C(=O)OCCC(C)C BTBG00016 CC1(C2CCC1(/C(=N/O)/C2)C)C BTB09928 c1cc(c(c(c1N2CCCC2)C#N)Cl)Br CD05678 COc1ccc(cc1OC)/C=C/2\C(=O)NC(=N2)SC BTB12637 c1cc(oc1)/C=N/OCCC#N BTB12644 c1ccc2c(c1)/C(=N/O)/C(=O)N2 BTB09934 c1cc(cc(c1)C(F)(F)F)CN(Cc2cccc(c2)C(F)(F)F)O CD05724 c1cc(ccc1CN(Cc2ccc(cc2)Cl)O)Cl CD05732 c1cnccc1c2nc(c3c4c(sc3n2)CCCCC4)N CD01510 c1cc(oc1/C=C(\C#N)/C(=S)N)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04135 CCCc1c(ccc2c1oc(cc2=O)C(=O)OCC)OCC=C BTB10010 CC(=O)c1ccc(cc1NC(=O)C)OC BTB10012 Cc1cc(=O)oc2c1ccc(c2)O BTB10013 CC(c1ccccc1)/N=C(/Nc2ccc(cc2)Oc3ccc(cc3)Cl)\SC.I CD06264 CCNC(=O)c1cccc2c1-c3ccccc3C2=O BTB10975 CN(C)C(=O)c1cccc2c1-c3ccccc3C2 BTB10979 c1ccc(c(c1)N)Nc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03704 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2)C)C CD01699 CCC(=O)c1c(c(c(c(c1C)C)C)C)C CD01702 c1cc(ccc1NC(=O)CSCC(=O)N)F CD01705 c1cc([nH]c1)/C=C(\C#N)/C(=O)N2CCCCC2 CD01689 CCOC(=O)CSCc1c(c(c(c(c1C)C)C)C)C CD01690 CCCc1ccc(c2c1oc(cc2=O)C(=O)OCC)OCc3ccccc3 BTB10006 CCOC(=O)c1c(c(c(o1)C(=O)OCC)O)O BTB10007 Cc1ccccc1NS(=O)(=O)c2ccc-3c(c2)Cc4c3ccc(c4)S(=O)(=O)Nc5ccccc5C BTB13631 COc1ccc(cc1)/N=C(/N2CCOCC2)\SC.I CD06280 c1cc(sc1)C(=O)N(CC#N)CC#N CD06286 c1ccn(c1)c2ccc(cc2F)F CD06289 Cc1c(c(c2c(c1C)[nH]c(n2)C)C)C CD04407 COc1cccc(c1C(=O)Nc2cc(cc(c2)OC)C(F)(F)F)OC CD03863 Cc1c(c(c(c(c1C)C)CSCC(=O)Nc2ccc(cc2)OC)C)C CD01677 c1cc(ccc1c2ccc(cc2)S(=O)(=O)c3ccc(c(c3)Cl)NS(=O)(=O)c4ccc(cc4)Cl)S(=O)(=O)c5ccc(c(c5)Cl)NS(=O)(=O)c6ccc(cc6)Cl BTB13470 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Cl BTB13472 c1ccc(cc1)NC(=N)Nc2ccccc2 BTB13475 c1cc([nH]c1)/C=C(\C#N)/C(=O)NCC2CCCO2 CD01687 CC(C)(C)C1=CC(=O)C=C(C1=O)C(C)(C)C BTB09891 Cc1ccc(c(n1)N)[N+](=O)[O-] BTB13479 c1cc2c(cc1F)c3c([nH]2)CCNC3 BTB13480 C#CCOc1c(cccc1Cl)Cl CD06185 c1ccc(cc1)C(=N)NC(=S)Nc2ccc(c(c2)Cl)Cl CD04311 CCC1CCCN(C1)S(=O)(=O)c2ccc(cc2)C BTB12762 CC(=NOc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])C BTB12764 CCOC(=O)c1ccc(cc1)n2nc(nn2)/C=C/C=C/N3CCOCC3 BTB12773 c1cc(cc(c1)C(F)(F)F)CO/N=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04188 c1cc(c(c(c1)F)C(=O)OCC#Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F CD04289 c1ccc(cc1)C(=N)NC(=S)Nc2cc(ccc2Cl)Cl CD04301 CC1(CC2(CCCCC2)C(=O)O1)C BTBG00067 C/C(=N\NC(=O)N)/CC(C)(C)C BTBG00070 COc1cccc(c1[N+](=O)[O-])C(=O)OC BTB10054 CC/C(=N\NS(=O)(=O)c1ccc(cc1)C)/c2ccco2 BTB10066 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N CD03848 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NC(=O)c3c(cccc3OC)OC CD03862 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2cc(c(c(c2)C(F)(F)F)N)C(F)(F)F CD04181 CCOC(=O)N1CCC(=NNc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])CC1 BTBS00011 c1ccc(cc1)/N=N\c2c(ccc3c2c(=O)cc(o3)C(=O)O)O BTB10045 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2cccnc2 CD02019 CCOC(=O)c1cc(=O)c2ccc(cc2o1)O BTB10085 Cc1cc(=O)oc2c1ccc(c2)OC(=O)C BTB10086 CC1(CC1(Br)Br)c2ccccc2 BTB12880 c1ccc\2c(c1)CSC/C2=N\Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD04220 CC(=O)c1ccc(c(c1)CO/N=C/2\CSCc3c2cccc3)OC CD04226 CN(C)c1ccc(cc1)C2Nc3ccccc3S2 CD01597 c1ccc2c(c1)NC(S2)c3cc(ccc3O)Br CD01598 Cc1c(cc2c(c1N)C(CC2(C)C)(C)C)NC(=S)Nc3cccc(c3)SC CD03891 c1cc2c(c(c1)C(=O)O)-c3ccc(cc3C2)I BTB13664 CC(=O)Nc1ccc(cc1)/C=N/NC(=O)CSCc2c(cccc2Cl)Cl CD01966 COc1cc(cc(c1OC)OC)/C=N/NC(=O)CSCc2c(cccc2Cl)Cl CD01971 c1cc(c(cc1)O)/C=N/CCC/N=C/c2c(cccc2)O CD06394 CCOC(=O)C/C(=C(\C#N)/C(=O)OCC)/N CD04091 Cc1c(c(c(cn1)CSc2ccccn2)CO)O CD04092 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2cc(c(c(c2)C(F)(F)F)[N+](=O)[O-])C(F)(F)F CD04166 CC(=O)C(=NNc1ccc(cc1)OC)C(=O)C CD01863 COc1ccc(cc1)OCCC(=O)NNC(=S)Nc2cccc(c2)OC CD01769 COc1ccc(cc1)OCCC(=O)NNC(=S)NC2CC3CC2C=C3 CD01770 CCCCCCCCCCCCCCCCCC(=O)CCN(C)C BTB12892 c1cc2c(cc1Cl)Nc3c(cc(cc3O2)[N+](=O)[O-])[N+](=O)[O-] BTB11001 COC(=O)/C=C/c1cn(c(=O)[nH]c1=O)C2C(C(CO2)CO)O BTBS00021 c1cc(ccc1N/N=C(\C#N)/C(=O)NCC2CCCO2)F CD01870 c1ccc(cc1)/C(=N\O)/C(=N/O)/c2ccccc2 BTB11003 CCCCCCCCOc1ccc(cc1)c2ccc(cc2)Br BTB11004 COC(=O)CO/N=C/c1ccc(cc1Cl)Cl CD06078 Cc1ccc(cc1)S(=O)(=O)O[C@@H]2CC3C[C@@H](C2C3)C(=O)OC BTBG00171 c1ccc2c(c1)CCC(C2)C(=O)O BTB10042 c1ccc2c(c1)cccc2NS(=O)(=O)c3ccc-4c(c3)Cc5c4ccc(c5)S(=O)(=O)Nc6cccc7c6cccc7 BTB13627 C[C@@H](C(=O)Nc1ccc(cc1)[N+](=O)[O-])N.Cl BTB13574 Cc1c(c(c2c(c1C)nc(c(n2)C)C)C)C CD04432 C1CCC(=NNC(=S)NC2CC3CC2C=C3)C1 CD01772 CCC1(c2ccccc2NC(O1)/C=C/c3ccccc3)c4ccccc4 CD01778 COc1ccc(cc1)OCCC(=O)N/N=C/C=C/c2ccccc2 CD01788 CN(C)c1ccc(cc1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl CD01790 CN(C)c1ccc(cc1)C(=O)N/N=C/c2ccc(c(c2)OC)O CD01794 CC(=O)N[C@@H](CCCCNC(=O)OCc1ccccc1)C(=O)O BTB13566 CC(=C(c1ccc(cc1)N(C)C)C(=O)OC)C BTBG00176 CCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB10904 CCCCCCCCCCN(CCCCCCCCCC)C(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] BTB10908 c1ccc(cc1)c2nc(=S)c3c(n2Cc4ccccn4)CCCC3 CD03943 CCCCCCCCCCCCCC#CC(C(CO)N)O BTBG00201 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)F)F)NC(=O)c2cccc(c2)Cl BTB13582 Cc1c(nc2cc(c(cc2n1)Cl)Cl)C CD04449 c1c(cc(c(c1C2Nc3cc(c(cc3N2)Cl)C(F)(F)F)O)Cl)Cl CD04455 C/C(=N/OC(=O)c1ccc(cc1)[N+](=O)[O-])/c2cc(cc3c2CCC3(C)C)C(C)(C)C BTB10088 COc1cc(c(cc1C(F)(F)F)[N+](=O)[O-])OC CD04530 CCOC(=S)SCc1c(cccc1Cl)F CD06437 c1ccc2c(c1)Nc3c(cc(cc3O2)[N+](=O)[O-])[N+](=O)[O-] BTB10997 CCOC(=O)C1=C(NC(=C(C1c2ccc(s2)[N+](=O)[O-])C(=O)OCC)C)C CD04172 c1cc(c2c(c1)oc(cc2=O)C(=O)O)O BTB09995 CCCc1c(ccc2c1oc(=O)cc2C)SC(=O)N(C)C BTB10079 c1ccc2c(c1)-c3c(cccc3C(=O)N4CCCCCC4)C2=O BTB10973 CC(C)CCNC(=O)c1cccc2c1-c3ccccc3C2=O BTB10977 c1ccc(cc1)NC(=O)c2cccc3c2-c4ccccc4C3=O BTB10978 c1ccc2c(c1)C(CC2=O)C(=O)O BTB10091 COc1ccc(cc1)C23CC4CC(C2)CC(C4)C3 BTBG00203 CN(C)c1ccc(cc1)C(=O)NNC(=O)c2ccc(cc2)Cl CD01805 Cc1c(c(c(c(c1C)C)CSCC(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)C)C CD01804 CC1(COC(=N1)c2ccc(cc2)C(=O)OC)C BTB10089 c1cc(c(cc1Cl)Cl)/C=N/OCC(=O)NN CD06081 Cc1c(c(c(c(c1C)C)CSCC(=O)N/N=C/c2cc(c(c(c2)OC)OC)OC)C)C CD01796 c1c(cc(c-2c1C(=C(C#N)C#N)c3c2c(cc(c3)S(=O)(=O)N4CCCCC4)[N+](=O)[O-])[N+](=O)[O-])S(=O)(=O)N5CCCCC5 BTB10981 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)Nc2cccc(c2)OC)C)C CD01701 CC(=O)N[C@@H]1[C@H]([C@H]([C@H](OC1O)CO)O)O BTB13540 CC(C)c1ccc(cc1)/C(=N/O)/C(C)C BTBG00177 C1C2CC3(CC1(CC(C2)(C3)Br)Br)Br BTBG00179 CSc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD04464 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)c2cccc(c2)Cl BTB13586 CCOC(=O)C1=C(NC(=C(C1c2ccc(o2)c3c(cccc3F)F)C(=O)OCC)C)C CD06423 Cc1c(c(c(c(c1C)C)/C=N/OC(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C)C)C CD06100 C/C(=N\O)/C(=O)Nc1ccccc1 BTBG00175 CCOC(=O)C12CCC(CC13SCCS3)(C4(C2)SCCS4)C(=O)OCC BTBG00106 c1cc(cnc1)CNc2ccc(cc2Cl)Cl CD06243 Cc1c(c(c(c(c1C)C)CC2CCC(C2=O)Cc3c(c(c(c(c3C)C)C)C)C)C)C CD01744 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)Cl)NC(=O)c2cccc(c2)Cl BTB13579 CN(C)c1ccc(cc1)C(=O)NNC(=S)NC2CC3CC2C=C3 CD01828 CC(=O)NC(c1ccccc1)C(=O)O BTB13561 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=O)c2ccc(cc2Cl)Cl)C)C CD01831 Cc1c(c(c(c(c1C)C)CSCC(=O)N/N=C/c2ccc(cc2)[N+](=O)[O-])C)C CD01797 Cc1c(c(no1)c2ccccc2Cl)C(=O)N CD01799 CCOC(=O)C(C(F)(F)F)(NCc1ccccc1)NC(=O)c2cccc(c2)Cl BTB13584 Cc1c(c(c(c(c1C)C)CSCC(=O)N/N=C/C=C/c2ccccc2)C)C CD01715 COc1cc(cc(c1OC)OC)C(=O)Nc2ccc(cc2)CC#N CD01730 COc1cc(cc(c1OC)OC)C(=O)Nc2ccc(cc2)/C(=C/c3ccc4c(c3)OCO4)/C#N CD01733 C/C(=C/C(=O)[O-])/C(=C\c1cccnc1)/C(=O)[O-].[Na+].[Na+] BTB12918 c1cc(ccc1C(=O)NNC(=O)CO/N=C/c2ccc(cc2Cl)Cl)Cl CD06212 COc1ccc(cc1)/N=C(/Nc2cccc(c2)C(F)(F)F)\SC.I CD06245 CN(C)c1ccc(cc1)C(=O)NNC(=S)Nc2cc(ccc2Cl)Cl CD01833 Cc1cc(c(cc1I)C)I BTB13663 COc1ccc(cc1)C23CC4CC(C2)CC(C4)(C3)O BTBG00210 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NCCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD04342 Cc1ccc(cc1)NC(=O)N(c2ccc(c(c2)Cl)F)C3=NCC(S3)(C)C BTB13595 c1ccc(cc1)N2CC(=O)N(C2=O)c3ccccc3 BTB11141 Cc1ccc(cc1)S(=O)(=O)c2c(c(c(c(c2C)C)C)C)C CD01883 CCOC(=O)C(C(F)(F)F)(Nc1cc(on1)C)NC(=O)c2cccc(c2)Cl BTB13587 CCOC(=O)C(C(F)(F)F)(Nc1nc2ccccc2s1)NC(=O)c3cccc(c3)Cl BTB13588 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cccnc2 CD04020 CCOC(=O)C(C(F)(F)F)(Nc1cc(ccc1OC)Cl)NC(=O)OCC BTB13600 c1cc(ccc1C(=O)c2cc3c(cc2Br)OCCCO3)Br BTB12836 c1cc(c(c(c1)F)NC(=O)C(F)(F)F)F CD04247 c1ccc\2c(c1)CSC/C2=N\NC(=S)Nc3cc(ccc3Cl)Cl CD04243 c1ccc(cc1)C2=CC(=O)OC(O2)c3ccc(cc3)[N+](=O)[O-] BTB13535 c1ccc(c(c1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04343 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)C CD06502 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccc(cc3Cl)Cl CD06503 c1ccc2c(c1)nc(c(=O)n2c3ccc(cc3)Cl)O BTB10142 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)O)C)C CD02018 CCC(C)/C(=N\O)/c1ccccc1 BTBG00207 CCOC(=O)C1(CCC(=NO)CC1)C(=O)OCC BTBG00183 c1ccc(cc1)COc2c[nH]c(cc2=O)CO BTB10143 C1C(=O)N=C2C=CC=CN2C1=O BTBG00194 CS/C(=N\S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/N2CCCCCC2 CD04389 c1cc(cc(c1)Cl)C(=O)NCc2cccs2 CD06330 c1ccc(cc1)/C(=N/O)/CN2CCCCC2 BTBG00113 CCCCN(C(C)C)S(=O)(=O)c1ccc(cc1)C BTBG00117 CC(=O)N[C@@H](CCCNC(=N)N)C(=O)O BTB13543 CC(=O)NC(CCC(=O)O)C(=O)O BTB13546 C1CC2C(CC1C2C(=O)O)O BTBG00114 c1ccc(cc1)C2OCC3(CC(C3C(=O)O)C(=O)O)CO2 BTBG00120 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NC(=N)N)C(F)(F)F CD06326 c1cc(sc1)CNC(=O)c2ccc(cc2Cl)Cl CD06365 CCOc1ccc(cc1)N2Cc3cc(ccc3N=C2)OCC BTB12725 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)n3cccc3 CD03831 c1ccnc(c1)c2[nH]c(nn2)CC#N CD04123 CC(C(=O)O)(C(F)(F)F)O BTB12864 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])ON=C2CCCC2 BTB12767 c1cc(cnc1)C(=O)NNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl CD04011 CCN(c1ccc(cc1)/N=N/c2ccc(cc2)[N+](=O)[O-])C(C)C BTB11017 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccnc3 CD01650 COc1ccc(cc1OC)CCNC(=O)/C(=C/c2ccc[nH]2)/C#N CD01682 c1cc([nH]c1)/C=C(\C#N)/C(=O)NCc2ccncc2 CD01683 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])c2ccc(o2)/C=N/NC(=S)N CD04357 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])c2ccc(o2)/C=N/NC(=O)N CD04358 c1cc(oc1/C=N/O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04126 c1ccnc(c1)NCN2C(=O)CCC2=O CD04506 CC(C)c1ccc(cc1)NCN2C(=O)CCC2=O CD04507 c1ccc(cc1)c2c(nnn2c3c(cccc3F)F)C(=O)O CD04518 c1c(cc(c(c1[N+](=O)[O-])N2CCCC2)[N+](=O)[O-])C(F)(F)F CD04014 CCC12CC3CC(C1)CC(C3)(C2)Br BTBG00225 CC(CCc1ccc(c(c1)OC)O)NCc2ccccc2 BTB09927 CN1C2CCC1CC(C2)NC(=O)c3ccc(cc3)Cl BTB09933 C/C(=N\OC(=O)c1c(cccc1F)F)/c2cccnc2 CD04157 CCOC(=O)C1=C(NC(=C(C1c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)OCC)C)C CD04170 CC(=O)c1ccc(c(c1)CO/N=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)OC CD04175 c1cc(sc1)C(=NO)c2cccs2 BTB09936 COc1ccc(cc1OC)CCNC(=O)/C(=N/Nc2ccc(cc2)F)/C#N CD01871 CC(=O)C(=NNc1ccc(cc1)F)C(=O)C CD01876 Cc1ccc(cc1)S(=O)(=O)OCC23CCC(CC2)C=C3 BTBG00157 COc1ccc(cc1)c2cc(=O)c3ccccc3o2 BTB10082 CCCc1c(ccc2c1oc(cc2=O)C(=O)OCC)N BTB10084 CC(C)(C)C(=O)Nc1cccc(c1)OC BTB10151 CN(C)C(=S)SCc1ccc(cc1)C(=O)Oc2c(cccc2Cl)Cl CD06363 c1ccnc(c1)C(=N)NS(=O)(=O)c2ccc(c(c2)Cl)Cl CD06366 c1ccc2c(c1)cccc2NS(=O)(=O)c3ccc-4c(c3)C(=O)c5c4ccc(c5)S(=O)(=O)Nc6cccc7c6cccc7 BTB13628 c1cc2cccc3c2c(c1)CCC3=O BTB12784 C1C2C=CC1[C@H]([C@H]2C(=O)O)C(=O)O BTB12787 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])ON=C2CCCCC2 BTB12761 c1cc(ccc1c2ccc(cc2)C(C(F)(F)F)(C(F)(F)F)O)C(C(F)(F)F)(C(F)(F)F)O BTB12860 CCCCOc1ccc(cc1)c2ccc(cc2)C#N BTB12792 C/C(=N\NC(=S)Nc1cccc(c1)C(F)(F)F)/c2cc(cc(c2O)Cl)Cl CD03804 CC(=O)C(CCC(=O)OC)(CCC(=O)OC)C(=O)OC BTBG00153 CC1(C2C1C3(CCC2CC3)CO)C BTBG00154 CC(C)CC(C)c1cc(nc2n1c3ccccc3n2)N BTB12778 Cc1c(c(no1)c2ccccc2)C(=O)N CD03844 c1ccc\2c(c1)CSC/C2=N\Nc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD04213 c1ccc\2c(c1)CSC/C2=N\OC(=O)c3ccccc3Cl CD04224 c1cc(cnc1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD04228 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C#CCN2CCCCC2.Cl CD04316 COc1cccc(c1C(=O)Nc2ccc(cc2)F)OC CD01880 c1ccc2c(c1)c(=O)n(c(n2)Sc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])c4ccc(c(c4)Cl)Cl CD04234 c1ccc2c(c1)c(=O)n(c(n2)Sc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])c4ccc(cc4)F CD04235 C/C(=N\OC(=O)c1cccc(c1)C(F)(F)F)/c2cccnc2 CD04158 Cc1c(snn1)C(=O)ON=C(c2cccs2)c3cccs3 BTB12782 c1ccc(cc1)/C(=N\c2ccccc2)/c3ccc(cc3)Cl CD03883 c1c(cc(cc1C(F)(F)F)S(=O)(=O)N=C2NCCCN2)C(F)(F)F CD04217 CNC(=S)NNC(=O)CSCc1c(cccc1Cl)Cl CD01993 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2cc(cc(c2)Cl)Cl)C)C CD06593 CN(/C=C/C=C(/c1ccccc1)\[N+](=O)[O-])c2ccccc2 BTB11105 c1ccc(cc1)c2cc3cccc4c3c(c2)C(=C4c5ccccc5)c6ccccc6 BTB11108 CN(/C=C/C=C/C=C1c2ccccc2-c3c1cccc3)c4ccccc4 BTB11110 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(c(c2)OC)OC CD01999 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)NC(=O)C CD02004 CCCC(CCC)C(C(=O)O)C(=O)OCC BTB13669 CCCc1ccc(cc1NC(=O)C)OC BTB10205 CCOC(=O)c1c([nH]c2c1cc(cc2)OCC=C)C BTB10131 CCN(CC)C(=O)c1cccc2c1-c3ccccc3C2=O BTB10969 CCCN(CCC)C(=O)c1cccc2c1-c3ccccc3C2=O BTB10970 Cc1cc(c2c(c1)-c3ccccc3CC2)C#N BTB11124 CC(=O)c1c(cc(c(c1OCc2ccccc2)C(=O)C)OCc3ccccc3)OCC=C BTB10137 CN(C)C=C1C(=C(C(=C1c2ccccc2)c3ccccc3)c4ccccc4)c5ccccc5 BTB11096 c1ccc(cc1)CC(=O)c2cc3c(cc2Br)OCCO3 BTB12835 c1ccc(cc1)C(=O)c2cc3c(cc2Br)OCCCO3 BTB12837 c1cc2c(cc1C(=O)CCC(=O)O)OCCO2 BTB12838 CC(=O)C(=NNc1ccc(c(c1)Cl)Br)C(=O)C CD01946 c1cc(c(c(c1)Cl)CSCC(=O)NN)Cl CD01950 CC(=O)C(=NNc1ccc2c(c1)OCO2)C(=O)C CD01891 COc1cccc(c1C(=O)NCCc2ccccn2)OC CD01892 c1cc(c(c(c1)F)C(=O)Nc2c(cccc2F)F)F CD04240 c1ccc2c(c1)-c3c(cccc3C(=O)N4CCCCC4)C2=O BTB10971 c1ccc2c(c1)-c3c(cccc3C(=O)N4CCOCC4)C2=O BTB10972 Cc1cc(c(c(c1)C)CO/N=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C CD04189 c1ccc(cc1)C2=C(C(=C(C2=C/C=C/C=C/N3CCCCC3)c4ccccc4)c5ccccc5)c6ccccc6 BTB11100 C=CCSc1nc2ccccc2c(=O)n1c3ccc(c(c3)Cl)F CD06724 CC(C)c1ccc(cc1)NN=C2C(=O)NC(=O)NC2=O CD01923 c1ccnc(c1)SCC(=O)Nc2c(cccc2F)F CD04312 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NN CD01963 COc1c(c(sc1C(=O)O)C(=O)O)OC BTB10060 c1c(cc(c(c1/C=N/NC(=S)NC2CC3CC2C=C3)O)Cl)Cl CD01758 Cc1cc(cc(c1/C=C\2/C(=O)NC(=O)N2)C)O BTBS00039 CC(=O)/C=C\c1cc[n+](cc1)C.[I-] BTB12919 C/C(=C/C(=O)[O-])/C(=C\c1ccncc1)/C(=O)[O-].[Na+].[Na+] BTB12921 c1ccc(cc1)C(=N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04302 c1ccc(c(c1)N)SCC(=O)Nc2c(cccc2F)F CD04305 c1cc(c(c(c1)F)NC(=O)CSc2ccc(cc2)Cl)F CD04306 c1cc(c(cc1NC(=O)C2CCC2)F)F CD01921 c1cc(c(c(c1)Cl)CSc2nnc(s2)SCc3c(cccc3Cl)Cl)Cl CD01932 c1cc(sc1)C(=O)ON=C2CCCCCCCCCCC2 BTB11032 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCc2ccc(c(c2)OC)OC)C)C CD06506 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)N(C)C)/C#N CD06512 Cc1c(c(c(c(c1C)C)S(=O)(=O)NC(C)(C)C#C)C)C CD06627 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)C CD06595 Cc1ccc(cc1)S(=O)(=O)O.C[C@H](C(=O)OCc1ccccc1)N BTB13571 CC(=O)Nc1cccc(c1[N+](=O)[O-])[N+](=O)[O-] BTB11167 Cc1c(c(c(c(c1C)C)CC#N)C)C CD00059 CCN(CC)c1ccc(cc1)/N=N/c2ccc(cc2)Br BTB11026 CCNc1ccc(cc1)/N=N/c2ccc(cc2)Br BTB11027 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2ccc(cc2Cl)Cl)C)C CD06594 CCOC(=O)c1ccc(c(c1O)C(=O)C)OCC(COc2ccc(c(c2C(=O)C)O)C(=O)OCC)O BTB10167 c1cc2c(cc1C(=O)CC3(c4cc(ccc4NC3=O)Br)O)OCO2 BTBT00007 CN1C(=O)C(C(=O)N(C1=O)C)C(=O)c2ccc(cc2)[N+](=O)[O-] BTB12848 CCCc1cc(=O)c2c(ccc(c2o1)OC)O BTB10063 COc1ccc(c2c1c(=O)cc([nH]2)C(=O)O)OC BTB10064 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2ccc(cc2)[N+](=O)[O-])C)C CD06485 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3cccs3 CD06540 c1ccc(cc1)C(Cn2ccnc2)NC(=S)Nc3ccc(cc3Cl)Cl BTBS00070 CC(C)(CCCCC(C)(C)C(=O)O)C(=O)O BTBS00081 c1cc2c(cc1Br)C(C(=O)N2)(C3CCCCC3=O)O BTBT00008 CCC/N=C(\C)/c1c(cc(oc1=O)C)O BTB12846 c1cc(c(cc1Cl)Cl)NC=C2C(=O)NC(=O)NC2=O BTB12847 c1ccc(c(c1)C2NCC(O2)c3ccc(cc3)[N+](=O)[O-])Cl BTB12942 CCOC(=O)c1ccc(cc1)C(=S)N2CCCC2 BTB10173 Cc1c(c(c(c(c1C)C)S(=O)(=O)N2CC(CC(C2)C)C)C)C CD06493 CC(=O)c1c(c(c2c(c1OC)cco2)OC)O BTB09981 Cc1cc2cc(c(c(c2c(c1)O)O)C(=O)C)C BTB09985 COc1cc(c(cc1OC)CO)CC(=O)N/N=C/C=C/c2ccccc2 CD01931 COc1ccc(cc1)C2NCC(O2)c3ccc(cc3)[N+](=O)[O-] BTB12947 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C#CCN2CCOCC2.Cl CD04318 CCCCCCCOc1ccc(cc1)C(=O)CCC(=O)O BTB10250 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCc2ccccn2)C)C CD06602 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2ccc(cc2F)F)C)C CD06603 c1ccc(cc1)c2ccc(cc2)C(=O)CC3(c4cc(ccc4NC3=O)Br)O BTBT00011 c1cc(sc1)/C=C(\C#N)/c2ccc(cc2)NC(=O)c3ccc(cc3)Cl CD01765 Cc1c(c(c(c(c1C)C)C(c2ccccc2)O)C)C CD01737 c1cc(ncc1[N+](=O)[O-])N2CCCC2 CD04421 CCN(CC)c1ccc(cc1)C2NCC(O2)c3ccc(cc3)[N+](=O)[O-] BTB12940 C(C(=O)O)C(C(=O)O)(F)F BTB12859 c1ccc(cc1)NC=c2c(=O)c3cccc4c3c(c2=O)ccc4 BTB11195 COc1ccc(cc1OC)CCNC(=O)Cc2cc(c(cc2CO)OC)OC CD01889 CSc1ncc(c(n1)C(=O)O)Cl BTB10252 c1cc2c(cc1C(=O)/C=C\3/c4cc(ccc4NC3=O)Br)OCO2 BTBT00050 Cc1c(c(c(c(c1C)C)C(=O)c2ccc(cc2)Cl)C)C CD01820 c1cc(ccc1C(=O)c2cc3c(cc2Br)OCCO3)Br BTB12949 COc1ccccc1C(=O)c2cc3c(cc2Br)OCCO3 BTB12950 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)Sc2ccc(cc2)Cl)C CD04581 c1ccc(cc1)c2cc(n(n2)CCC#N)N CD06631 c1ccc2c(c1)c(=O)n(c(n2)S)c3ccc(cc3F)F CD06633 Cc1c(c(c2c(c1C)[nH]c(n2)S)C)C CD04425 CC(=O)N[C@@H](CCSC)C(=O)O BTB13553 CCCCC(C(=O)O)NC(=O)C BTB13554 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=O)c2ccc(cc2)Cl)C)C CD01815 CCCC[C@@H](C(=O)O)NC(=O)C BTB13555 Cc1c(c(c(c(c1C)C)C(=O)c2ccc(cc2)NC(=O)c3ccc(c(c3)Cl)Cl)C)C CD01909 CC(C)c1ccc(cc1)NN=C(C(=O)C)C(=O)C CD01910 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=O)c2cc(c(c(c2)OC)OC)OC)C)C CD01816 CN(C)c1ccc(cc1)C(=O)NNC(=O)/C=C/c2ccc3c(c2)OCO3 CD01819 CN(C)c1ccc(cc1)C(=O)NNC(=O)COc2ccccc2 CD01821 CNC(=S)NNC(=O)c1ccc(cc1)N(C)C CD01830 CCn1c2ccc(cc2c(=O)cc1C(=O)O)OCC=C BTB10169 CCN(c1ccccc1)C(=N)SC.I BTB10196 CCOC(=O)C(C(F)(F)F)(NC(=O)c1cccc(c1)Cl)OCc2ccc(cc2)F BTB13591 c1c(c(=O)[nH]c(=O)n1[C@H]2C[C@@H]([C@H](O2)CO)O)I BTBS00065 c1ccc(cc1)c2cc(oc(=O)c2)c3ccccc3 CD06494 c1ccc(cc1)C(=O)CC(=O)N CD06497 c1cc(oc1CSC#N)[N+](=O)[O-] BTB13657 c1ccc(c(c1)C(=O)NCc2cccnc2)NC(=O)c3c(cccc3F)F CD04338 CC1=C(/C(=N\O)/CC1)c2ccc(cc2)N(C)C BTBG00242 CCOCCOc1cccc2c1c(=O)cc(o2)C(=O)OCC BTB10168 CCOC(=O)c1ccc2c(c1)c(=O)c3cc(ccc3o2)O BTB10185 c1cc(cnc1)CNc2ccc(cc2)Cl CD06422 c1cc(cnc1)/N=C/c2ccc(cc2Cl)Cl CD06425 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2cccnc2)C)C CD06480 CCCCCc1ccc(cc1)/C=N/O BTB12955 Cn1c2c(cc3ccccc3n2)c(=O)n(c1=O)C BTB12961 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2c(cccc2Cl)Cl)C)C CD06488 Cc1ccc(cc1)S(=O)(=O)OCC2CC3CC2C(C3)OS(=O)(=O)c4ccc(cc4)C BTBG00236 CCOC(=O)c1cc(=O)c2c(o1)ccc(c2O)CC=C BTB10025 c1ccc(cc1)/C(=N/O)/C(=O)c2ccccc2 BTBG00156 c1ccc(cc1)C[C@H](C(=O)OCc2ccccc2)NC(=O)[C@H](CCCCNC(=O)OCc3ccccc3)NC(=O)OCc4ccccc4 BTBS00001 CC1Cc2cc(ccc2O1)/C(=N/O)/C BTB12952 CN(C)/C=C/C=C/1\CCCC1=O BTB11050 Cc1c(c(no1)c2ccccc2)NC(=O)O/N=C(/c3ccc(cc3)Cl)\N CD04548 CC(=O)Nc1ccc(cc1C(=O)OC)C(=O)OC BTBG00123 CC(=O)N[C@H](CCc1ccccc1)C(=O)O BTB13547 C=C1CC2CC(C1)CC(=O)C2 BTBG00128 COC(=O)C12CC3CC(C1)CC(C3)(C2)C(=O)OC BTBG00226 c1cc(ccc1/C(=N/O)/CN2CCCCC2)[N+](=O)[O-] BTBG00227 c1ccc(cc1)C(=O)c2cc3c(cc2Br)OCCO3 BTB12840 CC(=O)N[C@@H](Cc1ccccc1)C(=O)O BTB13557 CN(C=C1C=C(C(=C1)/C=C/2\C(=C(c3c2cccc3)c4ccccc4)c5ccccc5)/C=C/6\C(=C(c7c6cccc7)c8ccccc8)c9ccccc9)C BTB11055 c1cc(c(c(c1)I)C(=O)O)C(=O)O BTB12976 c1cc(ccc1C(=O)/C=C/Sc2cc(ccc2Cl)Cl)F BTB11234 C(CC(CCC#N)(CCC#N)[N+](=O)[O-])C#N BTB10274 Cc1c(c(c(c(c1C)C)CN2CCC(CC2)C)C)C CD00073 Cc1c(c(c(c(c1C)C)CN2CCCCC2C)C)C CD00075 c1ccc(cc1)c2ccc(cc2)C(=O)/C=C\3/c4cc(ccc4NC3=O)Br BTBT00025 CC(=O)NCCCCC(C(=O)O)N BTB13551 CCOC(=O)c1ccc(cc1)n2nc(nn2)/C=C/C=C/N3CCCC3 BTB12774 CCOC(=O)c1ccc(cc1)n2nc(nn2)/C=C/C=C/N3CCN(CC3)C BTB12775 CC(=O)N[C@@H](Cc1ccccc1)C(=O)NN BTB13560 Cc1c(nc(s1)c2ccccc2)CC(=O)OC BTB12780 CS(=O)(=O)Cc1c(cccc1Cl)Cl CD04482 CSc1ccc(cc1[N+](=O)[O-])C(F)(F)F CD04457 c1cc(ccc1C(=O)/C=C/Sc2cc(ccc2Cl)Cl)Cl BTB11235 c1cc(cc(c1)Cl)N/C=C/C(=O)c2ccc(cc2)Cl BTB11237 Cc1ccc(cc1)S(=O)(=O)O.CC(C)N/C(=N\C(C)C)/SC BTB10192 CN(C)CC1(CCCCC1)CC(=O)O.Cl BTBG00231 C1CC(C(C1)C(=O)O)C(=O)O BTBG00237 c1ccc(cc1)COc2ccccc2C(=O)CC(c3ccccc3)Sc4ccccc4N BTB13684 c1cc(oc1CO)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04026 CSC1=C(C(=O)NC(S1)c2ccccc2O)C#N CD04067 CCOC(=O)c1cc(=O)c2cc(ccc2o1)I BTB10203 c1cnccc1CN(CCC#N)C(=S)NC2CC3CC2C=C3 CD01843 CCCc1c(ccc(c1O)C(=O)C)SC(=O)N(C)C BTB10118 c1cc(c(c(c1)F)CN2CCCCC2)F.Cl CD04364 CC(C)(C)C(=O)/C(=C/c1cccs1)/C#N CD06675 COc1cccc(c1C(=O)NCCc2ccc(c(c2)OC)OC)OC CD01868 C1C2CC3(CC1CC(C2)(C3)Br)CO BTBG00232 c1cc(ccc1S(=O)(=O)OC2CN3CCC2CC3)Br.Cl BTBG00234 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=O)c2c(onc2c3ccccc3Cl)C CD01985 c1ccc(cc1)C2CC(=NN2c3ccccc3)c4cccc5c4cccc5 BTB13678 CC(CC(=O)c1cccs1)C(=O)c2ccccc2 BTB12889 CS/C(=N\S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/N2CCOCC2 CD04386 c1cc(ccc1NCN2C(=O)CCC2=O)Cl CD04397 CC(C)(C)C1=C(C(C(=C(O1)N)C#N)c2c(cccc2Cl)Cl)C#N CD06681 CC(C)(C)C(=O)/C(=C/c1ccc(s1)[N+](=O)[O-])/C#N CD06682 Cc1cccc(n1)NCN2C(=O)CCC2=O CD04573 c1ccn(c1)c2cc(cc(c2)Cl)Cl CD06290 c1ccc(cc1)Cc2c(c3cccc4c3n(c2=O)CCC4)O BTB10986 Cc1ccc(cc1)n2c(nc3ccccc3c2=O)C BTB10991 CC1(CC(=CC(=O)C1)N2CCOCC2)C BTB10129 c1ccc(cc1)C(=O)NC2CC3CCC2CC3 BTBG00132 CCCCCCCCCCCCCCCCCC1(CC1)O BTB12891 CCOC(=O)/C(=C/c1cccn1c2ccc(cc2)Cl)/C#N CD04375 c1ccn(c1)c2ccc(cc2)I CD04547 CC1([C@@H](NC(S1)c2cc(ccc2OC)OC)C(=O)O)C BTB11155 c1ccc2c(c1)cccc2/C=N/c3c(nc4n3CCS4)c5cccc6c5cccc6 BTB11160 c1cc(cc(c1)Cl)N/C=C/C(=O)c2ccc(cc2)Br BTB11238 Cc1ccc2cccc(c2n1)I BTB12804 CN1CCc2cc(c(cc2C1Cc3ccc(c(c3)OC)OC)O)O BTB12808 CN(C)c1ccc(cc1)C(=O)N/N=C/c2cc(cc(c2O)Br)Br CD01836 COCCCNC(=O)c1nc2ccccc2c(=O)n1NC(=O)c3c(cccc3F)F CD04325 C1C2CC3(CC1CC(C2)(C3)O)C(=O)O BTB12757 c1cc(cnc1)OS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04191 COc1ccc(cc1)N/N=C(\C#N)/C(=O)NCCc2ccc(c(c2)OC)OC CD01855 Cc1cc(c(c(c1)C)CO/N=C/c2ccc(o2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)C CD04339 COc1ccc2c3c1ccc(c3C=CC2=O)OC BTB11147 COc1ccc(cc1)C(=O)CCC(=O)O BTB10244 CCOC(=O)O/N=C(/c1ccc(cc1)Cl)\N CD04463 CCc1c(cnc(n1)N)c2nnnn2c3ccccc3 BTB11241 CCc1c(cnc(n1)N)c2nnnn2c3ccc(cc3)C BTB11245 c1cc(c(c(c1)Cl)CSCC(=O)NNC(=S)Nc2ccc(c(c2)Cl)Cl)Cl CD01994 c1ccc(cc1)CCn2c(=O)c3ccccc3nc2Sc4c(cc(cc4[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD04237 c1ccc(cc1)S/C(=C/C(=O)O)/C(=O)O BTB10031 c1ccc\2c(c1)CSC/C2=N\NC(=S)NCc3ccco3 CD04239 CCCc1cc(=O)c2c(cccc2o1)O BTB10035 CCCc1cc(=O)c2ccc(cc2o1)O BTB10040 COc1cc2c(cc1OC)COC(=O)C2 CD01869 CCOC(=O)COc1ccccc1C(C#N)O BTB11118 CCCCCCOc1ccc(cc1)C(=O)CCC(=O)O BTB10249 c1cc-2c(cc1S(=O)(=O)[O-])C(=O)c3c2ccc(c3)S(=O)(=O)[O-].[K+].[K+] BTB10198 CSCCNc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD06915 c1ccc(cc1)C(=C2c3ccccc3-c4c2cccc4)/C=C/C=C(\c5ccccc5)/C6c7ccccc7-c8c6cccc8 BTB11140 CN(c1ccc(cn1)[N+](=O)[O-])/N=C/c2cc(cc(c2O)Cl)Cl CD06931 c1ccc(c(c1)C2NC(=NO2)CC(=O)N3CCCC3)O CD04515 CC(C)(C)Sc1ccccc1/C=N/O CD07391 c1cc(ccc1C(F)(F)F)NCN2C(=O)CCC2=O CD04435 CCN1C(C(CCC1=O)C(=O)O)c2ccc(cc2)OC CD01972 CCCOc1ccc(cc1)SCC(=O)O BTB12877 COc1ccc(cc1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccccc4 BTB13672 Cc1ccc(cc1)NS(=O)(=O)c2ccc-3c(c2)C(=O)c4c3ccc(c4)S(=O)(=O)Nc5ccc(cc5)C BTB13630 c1cc(c(c(c1)Cl)CSCC(=O)NNC(=S)NC2CC3CC2C=C3)Cl CD01986 CN(C)CCCNC(=O)Nc1ccc(cc1)Cl CD06533 COc1ccc(cc1)C2=NN(C(C2)c3c(cccc3Cl)Cl)c4ccccc4 BTB13673 c1cc(sc1)CNc2ccc(c(c2C#N)NCc3cccs3)[N+](=O)[O-] CD07392 c1ccc(cc1)c2c(nnn2c3ccc(cc3)[N+](=O)[O-])NC(=O)N4CCOCC4 CD04677 CC\1=NNC(=O)/C1=N\Nc2ccc(cc2)OC BTB13755 CN(C)C(c1ccccc1)c2ccccc2 BTB10217 CCOC(=O)COc1ccccc1C#N BTB12990 c1ccc2c(c1)C(=O)NC(=O)CO2 BTB12993 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NN=C2C(=O)NC(=O)NC2=O CD04263 CCN(CC)S(=O)(=O)c1ccc(cc1)C BTB10213 c1ccc2c(c1)c(=O)c3cc(ccc3o2)N BTB10215 Cc1cccc(c1)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccccc4 BTB13674 CC(CC(=O)c1ccccc1)C(=O)c2ccc(cc2)OC BTB12886 Cc1cccc(c1)C2=NN(C(C2)c3c(cccc3Cl)Cl)c4ccccc4 BTB13675 c1ccc(cc1)C(=O)c2cccnc2 BTBS00073 CC(C)(C)CCCCCCCCCCCC(=O)O BTBS00075 c1cc2c(c(c1)Cl)C(=O)c3cccc(c3C2=O)Cl BTB10218 c1ccc2c(c1)C(c3ccccc3O2)C(C(=O)O)C(=O)O BTB10221 CC(C)c1ccc(cc1)/C=C(\C)/C2NCC(O2)c3ccc(cc3)[N+](=O)[O-] BTB12939 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])Sc2cc(c(cc2Cl)Cl)Cl BTB10281 c1cc(cc(c1)[N+](=O)[O-])C(=O)CC2(c3cc(ccc3NC2=O)Br)O BTBT00009 c1ccc2c(c1)c(ccc2Br)Br BTB10259 c1cc(c(c(c1)Cl)C(=O)O)C(=O)O BTB10219 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2ccccc2N)C)C CD06514 c1cc2cccc(c2c(c1)C(=O)O)C(=O)O BTB12931 Cc1c(c(c(c(c1C)C)CN2C(=O)c3ccccc3C2=O)C)C CD00066 COc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD04503 CC1CN=C(S1)Nc2cccc(c2)C(F)(F)F BTB13011 CC1CN=C(S1)NC2CCCCC2 BTB13014 c1ccc2c(c1)C(c3ccccc3O2)CO BTB10230 Cc1c(c(c(c(c1C)C)Br)C)C CD00055 CCOC(=O)c1c(n(c2c1cc(cc2)O)c3ccccc3)C BTB12991 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)/C=N/O BTB12992 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD06528 c1ccc(cc1)NC(=O)NCCc2c[nH]c3c2cccc3 CD06529 c1ccc2c(c1)ccc\3c2-c4ccccc4/C3=C\c5cc6cccc-7c6c(c5)-c8c7cccc8 BTB11079 c1cc(c(c(c1)F)NCN2C(=O)CCC2=O)F CD04505 c1cc(ccc1c2nc(on2)CSc3[nH]c4ccc(cc4n3)C(F)(F)F)Cl CD04510 CCCCCCCCCCCC(=O)N1CC(=O)NC(=O)C1 BTB13000 CC(=O)C(=NNc1c(cccc1F)F)C(=O)C CD04607 CC1(CC(=O)C(=NNc2c(cccc2F)F)C(=O)C1)C CD04610 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)Nc2cccc(c2)OC)C CD04574 CCC(=O)NNc1ccccc1 BTB10204 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc3c(c2)OCO3 CD02021 Cc1c(c(no1)c2ccccc2)C(=O)N3CCCN4C3c5ccccc5C4=O CD02032 CC(C)c1ccc(cc1)NN=C2C(=O)NC(=S)NC2=O CD01922 c1ccc2c(c1)c(c(c(c2Cl)Cl)Cl)O BTB12851 c1cc(c(c(c1)F)C(=O)N2CCN(CC2)C(=O)c3c(cccc3F)F)F CD04652 c1cc(c(c(c1)Cl)C(=O)Oc2ccc(cc2)C#N)Cl CD07382 c1ccc(cc1)C2C(=C(SC(=C2C#N)N)N)C#N BTB13751 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N2CCC3c4ccccc4C(=O)N3C2 CD02031 Cc1c(c(=O)n(n1C)c2ccccc2)NN=C(C(=O)C)C(=O)C BTB13734 CC1CN(CC(O1)C)c2c(cccn2)[N+](=O)[O-] CD07289 c1ccnc(c1)CCNc2c(cccn2)[N+](=O)[O-] CD07290 c1ccc(cc1)N2C(=O)C(C(=O)N(C2=O)c3ccccc3)C(=O)c4ccc(cc4)[N+](=O)[O-] BTB12959 Cc1ccccc1NC2=NCC(S2)(C)C BTB13022 Cc1c(c(no1)c2ccccc2Cl)NC(=O)O/N=C(/c3ccc(cc3)Cl)\N CD04558 Cc1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)O CD04561 COc1ccc(cc1)C(=O)CC2(c3cc(ccc3NC2=O)Br)O BTBT00020 CN(C)/C=C/C=C/C=C1C(=C(C(=C1c2ccccc2)c3ccccc3)c4ccccc4)c5ccccc5 BTB11103 c1cc(c(cc1Cl)Cl)C=C2C(=O)NC(=O)NC2=O CD00164 c1cc(c(cc1C=C2C(=O)NC(=O)NC2=O)Cl)Cl CD00166 CC1CN=C(S1)Nc2ccccc2 BTB13006 CC1CN=C(S1)Nc2ccc(cc2)Cl BTB13008 c1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)Cl CD00170 c1ccc2c(c1)cccc2C=C3C(=O)NC(=O)NC3=O CD00171 c1ccc(cc1)/N=C/2\NC(=O)C(S2)CC(=O)Nc3cc(ccc3Cl)Cl CD00203 c1cc(ccc1C(C(CO)O)O)[N+](=O)[O-] BTB12954 c1cc(ccc1C(=O)c2cc3c(cc2Br)OCCO3)[N+](=O)[O-] BTB12956 CC1(CN=C(S1)Nc2ccc(c(c2)Cl)F)C BTB13019 CC12CCC3C1(COC2(C3)C#N)C BTB11192 c1ccc(cc1)C(=O)OC2=CC(=O)c3cccc4c3c2ccc4 BTB11194 CC1CN=C(S1)Nc2ccc(c(c2)Cl)F BTB13010 c1cc(cnc1)NCN2C(=O)CCC2=O CD04544 CC(=O)Nc1cc(c(cc1OC)Cl)C(F)(F)F CD04545 c1ccc(cc1)c2c(nnn2c3ccc(cc3)[N+](=O)[O-])C(=O)Nc4ccc(cc4)[N+](=O)[O-] CD04660 Cc1ccc(cc1)C(=O)C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 BTB12957 Cc1ccc(cc1)NC2=NCC(S2)(C)C BTB13016 CC1(CN=C(S1)Nc2ccc(cc2)F)C BTB13018 Cc1c(nnn1c2cccc(c2)C(F)(F)F)C(=O)O CD04550 COc1cc(c(cc1C(F)(F)F)NCN2C(=O)CCC2=O)OC CD04554 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3c(cccc3F)F CD04557 c1cc(ccc1CC#N)NC(=O)N CD02039 c1ccc(cc1)CNC(=O)CC2C(=O)N/C(=N\c3ccccc3)/S2 CD00205 c1ccc(cc1)/N=C/2\NC(=O)C(S2)CC(=O)Nc3cccc(c3)Cl CD00206 COc1ccc(cc1OC)C=C2C(=O)NC(=O)NC2=O CD00208 Cc1cccc(c1NC=C2C(=O)NC(=O)NC2=O)C BTB12958 CN(C)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2Cl)N(C)C CD01802 CN(C)c1ccc(cc1)C(=O)NNC(=O)c2cc(c(c(c2)OC)OC)OC CD01814 Cc1ccc(cc1)S(=O)(=O)N2CCC(=N2)N BTB10106 Cc1ccc(cc1)S(=O)(=O)C[C@@H]2[C@H](C[C@@H](O2)n3cc(c(=O)[nH]c3=O)I)O BTBS00069 Cc1c(c(no1)c2ccccc2Cl)NC(=O)OCC#Cc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04567 c1cc(c(cc1CNc2ccc(cn2)[N+](=O)[O-])Cl)Cl CD06608 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc(cc2)CC#N CD02033 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)C CD06530 c1c(c(cc(c1Cl)Cl)Cl)NCN2C(=O)CCC2=O CD04584 CCOC(=O)C(c1ccc(cc1)NC)(C(F)(F)F)O BTB13025 c1ccc2c(c1)c(c[nH]2)CCNC(=O)Nc3ccc(cc3)Cl CD06545 Cc1ccc(cc1)NC(=O)N(c2ccc(cc2)C)C3=NCC(S3)C BTB13596 C(CC(F)(F)F)C(C(=O)O)N BTB12855 c1ccc(cc1)c2cnc(nc2)c3ccccc3 BTB11048 c1ccc2c(c1)c(c(s2)C(=O)N3CCCN4C3c5ccccc5C4=O)Cl CD02034 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)CC#N CD02035 C=CCCCCCCCCC(=O)CCCCCCCC(=O)O BTBS00058 CC12CC3CC(C1)(CC(C3)(C2)Br)C(=O)O BTB12983 c1cc(c(nc1)NCCc2ccncc2)[N+](=O)[O-] CD07287 Cc1c(c(c(c(c1C)C)S(=O)(=O)NC(=N)N)C)C CD06499 Cc1c(c(c(c(c1C)C)S(=O)(=O)N2CCCC2)C)C CD06500 CC12CC3CC(C1)(CC(C3)(C2)C(=O)O)C BTB12972 CC12CC3(CC(C1)(CC(C2)(C3)C(=O)O)C)C BTB12973 COc1ccc(c(c1)C(=O)CCC(=O)OC)OC BTB12894 C1CCC(=NNC(=S)NC2CC3CCC2C3)C1 CD02045 CCOc1ccc(cc1)/C=N/NC(=S)NC2CC3CCC2C3 CD02046 C1CC2CC1CC2NC(=S)NNC(=S)NC3CC4CC3C=C4 CD02048 c1ccc2c(c1)c(=O)cc(o2)c3ccc(cc3)F BTB13705 c1ccc(cc1)C(=O)CC(c2ccccc2Cl)Sc3ccccc3N BTB13690 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NCN3C(=O)CCC3=O CD04583 c1cc(ccc1/C(=C\C=N\c2ccc(cc2)C(F)(F)F)/Nc3ccc(cc3)C(F)(F)F)Br BTB11228 c1ccc(cc1)CC(c2ccccc2)(c3ccccc3/N=C/c4ccc5c(c4)OCO5)O CD01976 CC(=O)Nc1ccc(c(c1)O)CC=C BTB10181 COc1ccc(cc1)OCCN.Cl BTB10107 c1ccc2c(c1)c(=O)cc(o2)c3ccc(c(c3)Cl)Cl BTB13707 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3ccc(c(c3)Cl)Cl CD06531 c1ccc2c(c1)c(=O)n(c(n2)S)c3ccc(c(c3)Cl)F CD06635 COc1ccc(cc1)Oc2cccc(c2C#N)F CD06811 CC1(CC(=O)C(=NNc2ccccc2C#N)C(=O)C1)C BTB13733 c1cc(ccc1C#N)C(=S)N2CCOCC2 BTB10175 c1c(cc(c(c1)Cl)Cl)/C=C\2/C(=O)/C(=C/c3cc(c(cc3)Cl)Cl)/CCC2 BTBT00042 COc1cc(ccc1O)/C=N/NC(=O)CSCc2c(cccc2Cl)Cl CD01981 c1ccc(cc1)C[C@@H](C(=O)OCc2ccccc2)NC(=O)[C@H](CCCCNC(=O)OCc3ccccc3)NC(=O)OCc4ccccc4 BTBS00005 CC(=O)OC(c1ccnc2c1cc(cc2)OC)C3CC4CCN3CC4C=C BW00083 COC(=O)CC1(N(C(=O)c2ccccc2O1)c3cc(cc(c3)Cl)Cl)C(=O)OC CD06850 c1ccc(c(c1)C(=O)N2CCOCC2)F CD06870 c1ccc(c(c1)C(=O)Nc2cc(ccc2Cl)Cl)F CD06906 CN(C)/C=C/C=C/1\c2ccccc2-c3c1cc(cc3)[N+](=O)[O-] BTB11135 c1ccc2c(c1)-c3ccccc3C2C=C4c5ccccc5-c6c4cccc6 BTB11093 CN(C)c1ccc(cc1)Cc2ccc(cc2)N(C)C BTB11222 c1ccc(cc1)C[C@H](C(=O)OCc2ccccc2)NC(=O)[C@@H](CCCCNC(=O)OCc3ccccc3)NC(=O)OCc4ccccc4 BTBS00003 CC(C)(C)C(=O)/C(=C/c1ccc(cc1Cl)Cl)/C#N CD06688 Cc1c(c(no1)c2c(cccc2Cl)Cl)C3=NN(C(O3)c4c(cccc4Cl)Cl)C(=O)C CD06690 c1ccc(cc1)C[C@@H](C(=O)OCc2ccccc2)NC(=O)[C@@H](CCCCNC(=O)OCc3ccccc3)NC(=O)OCc4ccccc4 BTBS00006 c1ccc(cc1)c2cc(c3cc(ccc3n2)Br)C#N BW00130 CS(=O)(=O)NC(=N)c1ccncc1 CD06748 Cc1cc(nn1c2ccccc2)C(=O)n3c(c(c(n3)C)Br)C CD07256 CC(C12CC3CC(C1)CC(C3)C2)N.Cl BTB12981 c1cc(c(cc1NC(=O)N)F)F CD02041 COc1cccc(c1)NC(=S)NNC(=S)NC2CC3CCC2C3 CD02049 C1CC2CC1CC2NC(=S)NNC(=S)NC3CC4CCC3C4 CD02050 COc1ccc(cc1)CC2CCC(=NOC(=O)c3cccc(c3)C(F)(F)F)CC2 BTB13762 CC(=O)c1cc(c(cc1NC(=O)C)OCC=C)C(=O)C BTB10182 c1cc(c(cc1Cl)NC(=S)Nc2ccc(nc2)N3CCOCC3)Cl CD04412 c1cc(c(c(c1)F)C(=O)Nc2ccc(nc2)N3CCOCC3)F CD04415 c1ccc(c(c1)C(=O)Nc2ccc(nc2)N3CCOCC3)Cl CD04416 CC(C)N/C(=N\C(C)C)/SC.I BTB10189 CCC(=O)c1ccc(cc1O)SC(=O)N(C)C BTB10190 C1CN(CCC1CCCC2CCN(CC2)C(=S)NC3CC4CC3C=C4)C(=S)NC5CC6CC5C=C6 CD02084 Cc1c(c(c(c(c1C)C)C(=O)c2cccs2)C)C CD06645 c1ccc(cc1)c2cc(c(c(c2C#N)N)C#N)c3ccco3 BTB13727 Cc1c(c(c(c(c1C)C)CO/N=C(\c2ccccc2)/c3ccc(cc3)Cl)C)C CD02103 c1cc(ccc1CNc2ccc(cn2)[N+](=O)[O-])Cl CD06609 Cc1c(c(c(c(c1C)C)S(=O)(=O)NC(C)(C)C)C)C CD06611 CS/C(=N/c1ccccc1)/Nc2ccccc2.I BTB10187 CCOCCOC(=O)c1cccc2c1-c3ccccc3C2=O BTB13625 C/C(=N/OC(=O)C(C)(C)C)/c1cc(cc2c1CCC2(C)C)C(C)(C)C BTB10231 CCCCCCc1ccc(cc1)c2ccccc2 BTB10235 CC(C)(C)NS(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)NC(C)(C)C BTB13626 c1cc(ccc1NC(=O)N2CCN(CC2)c3ncc(cn3)Br)OC(F)(F)F BTB13730 c1ccnc(c1)/C=N/NC(=S)N BTB13732 c1cc2cccc3c2c(c1)C(=O)NC3=O BTB12933 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCC=C)C)C CD06612 c1ccc(cc1)CC(c2ccccc2)(c3ccccc3/N=C/c4ccc(c(c4)Cl)Cl)O CD01975 CCc1cc(ccc1N2Cc3ccccc3C2)/N=N/c4ccc(cc4)[N+](=O)[O-] BTB11016 Cc1c(c(n(n1)C(=O)c2cccs2)C)Cc3c(cccc3Cl)F CD07535 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Cc3c(cccc3Cl)F CD07536 COC(=C(C#N)C#N)c1ccccc1 BTB13797 c1ccc(cc1)c2c(nnn2c3cccc(c3)C(F)(F)F)C(=O)N CD04622 Cc1c(c(c(c(c1C)C)COc2c(cccc2Cl)Cl)C)C CD02192 c1ccc(c(c1)[N+](=O)[O-])OCCOC2C(OCCO2)OCCOc3ccccc3[N+](=O)[O-] BTB13772 COC(=O)CC1(N(C(=O)c2cc(ccc2O1)Br)c3ccc(cc3F)F)C(=O)OC CD06895 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Br)F CD06900 CN(C)/C=C/C=C/C=C/1\c2ccccc2-c3c1cc(cc3)[N+](=O)[O-] BTB11133 C/C(=N\O)/C12CC3CC(C1)CC(C3)C2 BTB12978 CCC12CC3CC(C1)CC(C3)(C2)C(=O)O BTB12979 CC(=O)c1ccccc1OC(=O)c2c(cccc2F)F CD04634 c1cc(c(c(c1)F)C(=O)Oc2cccnc2)F CD04640 Cc1ccc(c(c1)C)C2=NN(C(C2)c3ccc(cc3)OC)c4ccccc4 BTB13676 Cc1ccc(c(c1)C)C2=NN(C(C2)c3ccc(cc3)Cl)c4ccccc4 BTB13677 CCN(CC)CC(=O)Nc1c(cccc1C)C BTB13834 C1CCN(CC1)S(=O)C23CC4CC(C2)CC(C4)C3 BTB13837 c1cc(ccc1c2nc3c(cc(cn3n2)C(F)(F)F)Cl)Cl BTB10254 COc1ccc(cc1)C(=O)NC23CC4CC(C2)CC(C4)C3 BTB12980 Cc1ccc2c(c1)N(C(CC2C)(C)C)CCO BTB13839 c1ccc(cc1)c2cc(=O)[nH]c(=O)o2 CD06686 c1ccc(cc1)CSc2nc3ccccc3c(=O)n2c4ccc(cc4F)F CD06731 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)NN)C)C CD02129 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccc(cc2)F CD02162 COc1ccc(c(c1)C(=O)c2ccc(cc2)[N+](=O)[O-])OC CD02040 COc1cc(c(cc1NC(=O)CC2C(=O)NC(=N)S2)Cl)OC CD00008 c1cc(ccc1C(=O)CC2(c3cc(ccc3NC2=O)Br)O)F BTBT00019 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCC(C)(C)C CD06860 c1ccc(c(c1)C(=O)Nc2ccccc2F)F CD06866 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)NNC(=O)c3c(c4ccccc4s3)Cl)C)C CD02122 CC(C)(C)C(=O)ON=C(c1cccs1)c2cccs2 BTB11165 C1C2C3C4CC3\5C2/C(=N\O)/C1C4/C5=N\O BTB11169 CCOC(=O)CSC(=S)SCc1c(c(c(c(c1C)C)C)C)C CD02139 Cc1c(c(c(c(c1C)C)CSc2ccc(cc2)Cl)C)C CD02146 c1cc(ccc1C(=O)ON=C2CCCCC2)[N+](=O)[O-] CD02158 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N/N=C/C=C/c2ccccc2 CD02011 Cc1c(c(c(c(c1C)C)CSC(=N)Nc2ccccc2)C)C.Cl CD00214 CSc1cccc(c1)NCN2C(=O)CCC2=O CD04491 c1cc(c(cc1Cl)NCN2C(=O)CCC2=O)Cl CD04492 CCC1C(=O)NC(=O)c2ccccc2O1 BTB12995 CCOC(=S)SCc1c(c(c(c(c1C)C)C)C)C CD02134 CN(C)CCCNc1ccc(c(c1C#N)NCCCN(C)C)[N+](=O)[O-] CD07354 c1cc(c(nc1)NCCCn2ccnc2)[N+](=O)[O-] CD07440 Cc1c(c(n(n1)C(C)(C)C)C)/C=N/OC(=O)Nc2ccc(cc2)Cl CD07443 c1cc(oc1c2nnc(s2)S)[N+](=O)[O-] BTB13666 c1ccc(cc1)N2C(CC(=N2)c3ccc4ccccc4c3)c5ccc(cc5)Cl BTB13681 c1cc(c(c(c1)F)C#N)Oc2c(cccc2Cl)Cl CD06812 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(CCCOC)CCC#N CD06813 c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3cccc(c3C#N)Cl CD07097 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)N3CCOCC3 CD07098 CC(=O)C1=C(c2cccc3c2c(ccc3)C1=O)O BTB11217 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CC(=O)NC(=O)C2 BTB12996 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CC(=O)NC(=O)C2 BTB12999 CCOC(=O)C(c1ccc(c(c1)C)N)(C(F)(F)F)O BTB13026 CC1(CN=C(S1)Nc2cccc(c2)C(F)(F)F)C BTB13020 CC1(CN=C(S1)NC2CCCCC2)C BTB13023 c1ccc(cc1)c2c(nnn2c3ccccc3Oc4ccc(cc4Cl)Cl)C(=O)O CD08446 c1c(cc(c2c1COCO2)CSc3nnc(s3)N)F CD08458 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc3c(c2)OCO3 CD02000 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCCN(C)C CD06799 CN(C)C(=O)Oc1ccc(cc1C(=O)Nc2ccc(c(c2)Cl)F)Br CD07054 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)Nc3ccc(c(c3)Cl)Br)C)C CD02095 c1cc(ccc1NC(=O)N2CCN(CC2)c3ncc(cn3)Br)Br BTB13715 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)NCc3cccnc3)C)C CD02101 CCOC(=O)C(c1ccc(cc1)N)(C(F)(F)F)O BTB13024 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)CSCc2c(cccc2Cl)Cl CD02017 c1cc(ccc1/C=C\2/C(=O)NC(=O)N2)O BTBS00036 c1cc(ccc1C(=O)N2CCN(CC2)c3ncc(cn3)Br)[N+](=O)[O-] BTB13706 c1cc(c(c(c1)F)C(=O)N2CCN(CC2)c3ncc(cn3)Br)F BTB13708 c1ccc(cc1)c2cc(=O)c3cc(ccc3o2)Cl BTB13712 C/C(=N\OC(=O)c1cc(c(c(c1)OC)OC)OC)/c2ccc(cc2)F CD02161 c1cc(cc(c1)Cl)N/C=C/C(=O)c2ccc(cc2)F BTB11236 COc1cccc(c1)NC(=S)NNC(=O)CSCc2c(cccc2Cl)Cl CD01982 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=O)c2cc(c(c(c2)OC)OC)OC CD01983 CC(C)(C)c1ccc(cc1)C(=O)ON=C2CCC(CC2)Cc3ccc(cc3)OC BTB13763 COc1ccc(cc1)CC2CCC(=NOC(=O)c3ccc(cc3)[N+](=O)[O-])CC2 BTB13764 c1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccc5ccccc5c4 BTB13680 c1c(cc(c(c1/C=N/NC(=S)NC2CC3CCC2C3)O)Cl)Cl CD02042 c1ccc(cc1)/C=C/C=N/NC(=S)NC2CC3CCC2C3 CD02043 c1cc(sc1)/C=N/NC(=S)NC2CC3CCC2C3 CD02044 C1C2CC3CC1CC(C2)(C3)Br BTB13004 Cc1ccc(cc1)C(=O)/C=C/Sc2cc(ccc2Cl)Cl BTB11232 COc1ccc(cc1)C(=O)/C=C/Sc2cc(ccc2Cl)Cl BTB11233 COc1cc(c(cc1Cl)OC)N2C(=O)C=CC2=O CD02201 c1cc2c(cc1/C=N/NC(=S)NC3CC4CCC3C4)OCO2 CD02064 COc1ccc(cc1)CC2CCC(=NOC(=O)c3c(cccc3Cl)Cl)CC2 BTB13765 COc1ccc(cc1)CC2CCC(=NOC(=O)C3CCCCC3)CC2 BTB13766 CC(=NNC(=S)NC1CC2CCC1C2)C CD02052 c1ccc(cc1)CC(=NOC(=O)c2c(c3ccccc3s2)Cl)Cc4ccccc4 CD02174 C1CCC(=NNC(=S)NC2C3CCC2CC3)CC1 CD02055 C/C(=N\NC(=O)N)/c1ccc(cc1)F CD02248 c1ccc(cc1)S(=O)(=O)N2CC(=O)NC(=O)C2 BTB13003 C1C2CC3CC1CC(C2)(C3)CC(=O)O BTB13005 c1ccc2c(c1)cc3c(n2)-c4cccc5c4c(ccc5)C3=O BTB12965 CC12CC3CC(C1)CC(C3)(C2)C(=O)O BTB12971 C1C2CC3CC1CC(C2)(C3)CCC(=O)O BTB12974 CCOC(=O)C(c1ccc(c(c1)OC)N)(C(F)(F)F)O BTB13027 c1cc(ccc1C(=O)NNC(=S)NC2CC3CCC2C3)Cl CD02070 Cc1ccc(c(c1)C)NC(=S)NNC(=S)NC2CC3CCC2C3 CD02071 Cc1cc(c(c(c1)C)NC(=O)CSCc2c(cccc2Cl)Cl)C CD02074 CCN(CC)Cc1c(c(c(c(c1C)C)C)C)C CD00241 CC(=O)NN1C(=O)CSC1=S BTB13863 CN(C)/C=C(\C#N)/C(=O)c1cccs1 CD07542 CN(C)/C=C(\C#N)/C(=O)c1ccccc1 CD07544 COc1ccc(cc1)/C(=N/C#N)/N BTB13804 c1ccc(cc1)c2c(cnc(n2)N)c3nnnn3c4ccc(cc4)Br BTB11412 CCN(CCC#N)C(=O)c1c(onc1c2c(cccc2Cl)Cl)C CD06802 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)Oc3c(cccc3Cl)Cl CD07107 COc1cccc(c1C(=O)Nc2cc(c(cc2OC)Cl)C(F)(F)F)OC CD04562 COc1cc(c(cc1NC(=O)c2ccccc2Cl)C(F)(F)F)Cl CD04563 COc1cccc(c1C(=O)Nc2cc(c(cc2OC)OC)C(F)(F)F)OC CD04565 c1ccc(cc1)c2c(nnn2c3ccc(cc3)[N+](=O)[O-])C(=O)N CD04651 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NCCc2ccc(c(c2)OC)OC CD02023 c1cc(cnc1)CNc2ccc(c(c2C#N)NCc3cccnc3)[N+](=O)[O-] CD07424 c1c(cc(cc1Cl)Cl)NC(=S)NC(CO)(CO)CO CD07019 c1c(cc(cc1Cl)Cl)/N=C\2/NC(CS2)(CO)CO CD07027 c1ccc(c(c1)C(=O)Nc2cccc(c2)Cl)F CD06891 COc1ccc(cc1)NC(=O)c2ccccc2F CD06894 c1cc(c(cc1F)F)NC(=O)CCN2CCOCC2 CD07185 c1ccc(c(c1)C(=O)NCc2c(cccc2Cl)F)NC(=O)c3ccccc3Cl CD07240 CC(=O)Nc1cccc(c1Cl)C(=O)O BTB10212 COc1cc(ccc1O)/C=N/NC(=S)NC2CC3CCC2C3 CD02054 C/C(=N\NC(=S)N)/c1cccnc1 BTB13748 c1cc(c(c(c1)Cl)CSCC(=O)Nc2ccc(cc2)Cl)Cl CD02073 COc1ccc(cc1)c2cc(=O)c3cc(ccc3o2)Cl BTB13714 COC(=O)CC1(N(C(=O)c2cc(ccc2O1)Br)c3cc(cc(c3)Cl)Cl)C(=O)OC CD06881 Cc1cccc(c1NC(=O)C2C3CC(C2C(=O)O)C=C3)Cl CD02214 COc1cccc(c1)NC(=S)N(CCC#N)CCC#N CD02223 CCCCOc1ccc(cc1)C(=O)CCC(=O)O BTB10247 CCCCCOc1ccc(cc1)C(=O)CCC(=O)O BTB10248 c1cc(ccc1/C(=C/c2ccc(c(c2)Cl)Cl)/C#N)NC(=O)N CD02284 COc1ccc(cc1OC)CCNC(=O)c2ccccc2c3ccccc3C(=O)O CD02258 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc(cc2)F CD01942 CCCc1c(cnc(n1)N)c2nnnn2c3ccc(cc3)C BTB11246 CC1(COC(OC1)c2ccccc2)[N+](=O)[O-] BTB12905 C[C@@]12[C@@](CC(=O)C1)(CC(=O)C2)C BTB13696 COc1cc(c(cc1I)OC)I BTB13697 c1cc(c(c(c1)Cl)CSCC(=O)Nc2ccc(cc2)F)Cl CD01951 CCOc1ccc(cc1)/C=N/NC(=S)NC2CC3CC2C=C3 CD02117 C/C(=C\C(=O)[O-])/C=C/c1c[nH]c2c1cccc2.[Na+] BTB12909 Cc1c(c(c(c(c1C)C)C(=O)CCCC(=O)O)C)C CD02278 Cc1c(c(c(c(c1C)C)CSCc2c(c(c(c(c2C)C)C)C)C)C)C CD02243 c1cc2c(cc1/C=N/NC(=O)N)OCO2 CD02254 c1ccc2c(c1)[nH]c(n2)SCc3c(c(c(c(c3F)F)F)F)F BTB13794 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(\C)/c3ccc(cc3)F CD02151 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)ON=C2CCCCC2 CD02152 COc1ccc(cc1)/C(=N/OCc2c(cccc2Cl)Cl)/N CD02154 c1ccc2c(c1)[nH]c(n2)SCc3cc(cc4c3OCOC4)F CD08461 C/C(=C\C(=O)O)/C=C/c1c[nH]c2c1cccc2 BTB12908 c1ccc(c(c1)C(=O)Nc2ccc(c(c2)Cl)F)O CD06828 c1cc(c(cc1Br)C(=O)Nc2cc(cc(c2)Cl)Cl)O CD06834 CC(=CCC(CC=C(C)C)(C#N)C(=O)O)C BTB13703 Cc1c(c(c(c(c1C)C)S(=O)(=O)N2CC(OC(C2)C)C)C)C CD06590 Cc1cc(c(c(c1C)C)C)C(=O)c2ccccc2C(=O)O CD02133 c1cc(c(c(c1)Cl)CO/N=C(/c2ccc(cc2)Cl)\N)Cl CD02142 CCCCCCCCc1ccc(cc1)c2ccccc2 BTB10298 c1cc(c(c(c1)Cl)C(=O)Oc2ccc(cc2Cl)Cl)Cl CD07402 c1ccc(cc1)Oc2ccc(c(c2C#N)Oc3ccccc3)[N+](=O)[O-] CD07403 c1cc(c(c(c1)Cl)C(=O)Oc2c(cccc2Cl)Cl)Cl CD07410 c1cc(c(cc1F)F)NC(=O)c2cc(ccc2O)Cl CD06919 C/C(=N\O)/c1c(c2ccccc2n(c1=O)C)O BTB11099 CN(C)/C=C/C=C/C(=O)c1cccs1 BTB11102 CCOC(=O)/C(=N\Nc1ccc(cc1)Br)/C(=O)CSC#N BTB13803 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCc2ccncc2)C)C CD06601 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3c(cccc3Cl)Cl CD06842 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NCCSC CD06844 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCc3ccccc3 CD06897 c1ccc(cc1)S(=O)(=O)c2ccc(cc2)[N+](=O)[O-] BTB10288 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)c2ccc(cc2)[N+](=O)[O-] BTB10289 c1c(cc(cc1Cl)Cl)NC(=O)CN2CCCCC2 CD07184 COc1ccc(cc1)C(=O)/C=C/Sc2nc3ccccc3o2 BTB11323 CCCc1c(ccc2c1oc(cc2=O)C(=O)O)O BTB10150 CCCc1c(ccc(c1O)C(=O)C)OCc2ccccc2 BTB10154 c1cc(sc1)C(=O)N2CCN(CC2)c3ncc(cn3)Br BTB13719 Cc1c(c(=O)n(nc1C(=O)NN)c2ccccc2)C#N BTB13723 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccccc3C(=O)NCc4c(cccc4Cl)F CD07243 c1ccc(c(c1)C(=O)Nc2cc(cc(c2)Cl)Cl)F CD06885 COc1ccc(cc1)C(=O)/C=C/Sc2c(cccc2Cl)Cl BTB11320 c1cc(ccc1/C(=C/c2ccncc2)/C#N)NC(=O)N CD02280 CCCCCCCCOc1ccc(cc1)C(=O)CCC(=O)O BTB10251 CSc1nc2ccccc2c(=O)n1c3ccc(c(c3)Cl)F CD06737 Cc1csc(n1)NS(=O)(=O)c2ccccc2 BTB13828 CCCCCCCNS(=O)(=O)c1c(c(c(c(c1C)C)C)C)C CD06613 Cc1c(c(c(c(c1C)C)CO/N=C(/c2ccc3c(c2)OCO3)\C(=O)C)C)C CD02104 c1ccc(cc1)C2CC(=O)c3ccccc3O2 BTB13717 CCOC(=O)c1cc2cc(ccc2[nH]1)OCc3ccccc3 BTB10162 Cc1cc2c(cc1[N+](=O)[O-])OCCO2 BTB10214 Cc1c(c(sc1C#N)C#N)C CD06621 CCOc1ccc(cc1)C(=O)CCC(=O)O BTB10245 c1cc2c(cc1C=C3C(=O)NC(=O)NC3=O)OCO2 CD00209 COc1cc(cc(c1OC)OC)C=C2C(=O)NC(=O)NC2=O CD00211 c1ccnc(c1)NC2CCCCC2 BTB13829 C1COCCN1S(=O)C23CC4CC(C2)CC(C4)C3 BTB13832 Cc1cccc(c1)NC2=NCC(S2)C BTB13012 Cc1ccccc1NC2=NCC(S2)C BTB13013 CC1(CN=C(S1)Nc2ccccc2)C BTB13015 CC1(CN=C(S1)Nc2ccc(cc2)Cl)C BTB13017 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)c4ncc(cn4)Br BTB13720 Cc1c(c(sc1C(=O)N)C(=O)N)C CD06616 COc1ccc(cc1)Oc2cccc(c2C#N)Oc3ccc(cc3)OC CD06887 c1cc(cnc1)C(=N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD06625 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl)C)C CD06630 c1cc(ccc1NC(=O)N2CCN(CC2)c3ncc(cn3)Br)Cl BTB13721 COc1cc(c2ccc3ccccc3c2c1)C#N BTB11122 c1ccc(cc1)c2cc(c3c(c2)-c4ccccc4CC3)C#N BTB11126 c1ccc(cc1)S(=O)(=O)C2CS(=O)(=O)CC2S(=O)(=O)[O-].[Na+] BTB13822 CS(=O)(=O)C1CS(=O)(=O)CC1O BTB13825 Cc1ccc(cc1)NC2=NCC(S2)C BTB13007 Cc1c(c(c(c(c1C)C)COc2ccc(cc2)[N+](=O)[O-])C)C CD02187 CCOC(=O)CCc1ccc(cc1)OCc2c(c(c(c(c2C)C)C)C)C CD02189 c1cc(cc(c1)NC(=O)CC(=O)Nc2cccc(c2)C(F)(F)F)C(F)(F)F CD02366 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N3CCCN4C3c5ccccc5C4=O CD02379 c1cc(c(c(c1)NC(=O)N2CCOCC2)F)NC(=O)N3CCOCC3 CD10568 c1cc(c(c(c1)Cl)C#N)NC(=O)c2cccs2 CD07315 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=S)NC2CC3CC2C=C3 CD01989 c1cc(ccc1CSC(=N)N)F.Cl CD00226 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)Nc3cc(c(cc3Cl)Cl)Cl CD00237 Cc1c(c(n[nH]1)C)Cc2c(cccc2Cl)F CD07521 Cc1c(c(n(n1)S(=O)(=O)c2ccc(c(c2)Cl)Cl)C)Cc3c(cccc3Cl)F CD07528 COc1cc(c(cc1NC(=O)/C=C/C(=O)O)Cl)OC CD02263 c1cc(ccc1N2C3(CCCC3N=N2)N4CCOCC4)[N+](=O)[O-] CD04611 c1ccc(c(c1)/C=N/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O CD04715 CC(C)(C)SCCNS(=O)(=O)c1ccc(cc1)C#N CD10695 c1ccc(cc1)/C=C/C(=O)O/N=C(/C=C/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N CD04797 c1ccc(c(c1)[N+](=O)[O-])S(=O)c2ccccc2[N+](=O)[O-] BTB10285 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=C/c2nc(on2)C(F)(F)F CD04753 c1ccc2c(c1)nc(s2)SCc3cc(cc4c3OCOC4)F CD08462 Cc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)I)c4ccccc4 BTB11334 CCCCCCCCCc1ccc(cc1)c2ccccc2 BTB10233 C1Cc2c(non2)/C(=N\O)/C1 BTB13034 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(c(c2)Cl)Cl CD01998 c1ccc(cc1)NC(=O)CC2C(=O)N/C(=N\c3ccccc3)/S2 CD00249 COc1ccc(cc1)C(=O)/C=C(/CC(=O)c2ccc(cc2)I)\c3ccccc3 BTB11343 C#Cc1cccc(c1)NS(=O)(=O)c2ccc(cc2)C#N CD10700 c1cc(ccc1C#N)S(=O)(=O)Oc2ccc(cc2Cl)Cl CD10701 c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)C#N CD10702 c1cc2c(cc1Cl)nnc3n2c(nn3)SCC(=O)N4CCOCC4 BTB11459 c1ccc(c(c1)Oc2ccc(cc2Cl)Cl)S(=O)(=O)N3CCOCC3 CD08398 CCOC(=O)c1cnc(nc1C(F)(F)F)N2CCN(CC2)c3ncc(c(n3)C(F)(F)F)C(=O)OCC GK02922 c1cc(ccc1/C=N/Nc2c3ccsc3ncn2)Cl GK02929 Cc1ccc2c(c1)cc(cc2C#N)C BTB11148 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(c3ccc(c(c3)Cl)Cl)O CD06795 Cc1c(c(no1)c2ccccc2)C(=O)ON=C(Cc3ccccc3)Cc4ccccc4 CD02175 CN(C)c1c(nc2cc(ccc2n1)Cl)N(C)C BTB13043 CC(C)(C)C(=O)/C(=C/c1c(cccc1Cl)Cl)/C#N CD06678 CCOC(=O)/C(=C/N1CCCC1c2cccs2)/C#N CD10541 CN(Cc1ccccc1)S(=O)(=O)c2ccc(cc2)Oc3cccc(c3C#N)Cl CD07115 CC(=O)C(=NNc1ccccc1Oc2ccc(cc2Cl)Cl)C(=O)C CD08427 Cc1cc(cc(n1)NNS(=O)(=O)c2ccc(cc2Cl)Cl)C(F)(F)F CD10563 c1c(cc(cc1Cl)Cl)NC(=O)CCN2CCOCC2 CD07168 c1c(cc(cc1Cl)Cl)NC(=O)CN2CCOCC2 CD07180 Cn1c(cc(n1)C(F)(F)F)OS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl CD10512 c1ccc(cc1)NC(=O)Nc2cccc(c2F)NC(=O)Nc3ccccc3 CD10571 CSC(=C(C#N)c1ccc(cc1)[N+](=O)[O-])SC EN00078 C1CS(=O)(=O)CC1SCC(=O)[O-].[Na+] BTB13826 COc1ccc(cc1)c2c(nc(nc2SC)c3ccc(cc3)Cl)N EN00081 Cc1csc(n1)NC(=O)C BTB13830 CSC(=C(C#N)c1ccc(cc1Cl)Cl)SC EN00082 Cc1c(c(n(n1)C(=O)c2c(onc2c3c(cccc3Cl)Cl)C)C)Br CD07238 c1cc(c(c(c1)C(=O)Oc2ccc(cc2)Cl)F)C(=O)Oc3ccc(cc3)Cl CD10542 Cc1cc(cc(n1)NNC(=O)c2ccc(cc2)Cl)C(F)(F)F CD10560 COC(=O)c1ccsc1NC(=O)c2ccc(cc2)C(F)(F)F GK02868 CN1C(=O)c2ccc(cc2C1=O)N BTB13891 c1ccc2c(c1)cccc2NC(=O)C3C4CC(C3C(=O)O)C=C4 CD02219 C1C2CC(C1C=C2)NC(=S)N(CCC#N)CCC#N CD02222 c1cc(c(cc1NC(=S)N(CCC#N)CCC#N)Cl)Cl CD02229 c1ccc2c(c1)CCCN2C(=O)CCC(=O)O CD02235 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=S)Nc2ccc(c(c2)Cl)Cl CD01991 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=S)NCC=C CD01992 COc1cc(cc(c1OC)OC)C(CC(=O)c2ccccc2)Sc3ccccc3N BTB13695 c1ccc(cc1)C(CC(=O)c2cccc3c2cccc3)Sc4ccccc4N BTB13699 CCOC(=O)NC(=O)/C(=C/c1ccc(cc1)N(C)C)/C#N CD02205 c1csc2c1c(ncn2)NCCO GK02882 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccc(cc2)Cl CD08652 CS/C(=N\C(=O)c1c(cccc1Cl)Cl)/NCc2cccs2 EN00057 Cc1cc(c(c2c1C(=O)C(C2)(C)C)C(=O)N)C CD07337 COc1ccc(cc1CSc2ccc(cc2)Cl)C(=O)C[n+]3ccccc3.[I-] CD02455 c1ccc2c(c1)-c3ccccc3C2CC(CN4CCN(CC4)CC(CC5c6ccc(cc6-c7c5c(cc(c7)Br)Br)Br)O)O BTB13902 c1ccc2cc(ccc2c1)OC3=C(C(=O)c4ccccc4C3=O)Cl BTB13037 c1ccc(c(c1)C(=O)Nc2cc(cc(c2)Cl)Cl)O CD06831 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)ON3C(=O)CCC3=O CD06849 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCSC CD06854 CC(C)c1ccc(cc1)NC(=S)NNC(=S)NC2CC3CCC2C3 CD02058 CS/C(=N/S(=O)(=O)c1ccccc1)/NCCc2ccc(cc2)Cl CD08657 c1cc(c(c(c1)COC(=O)c2ccc(cc2)Cl)F)COC(=O)c3ccc(cc3)Cl CD10694 Cc1c(c(n(n1)C(C)(C)C)C)/C=N/OC(=O)c2cccs2 CD07490 c1ccn(c1)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl CD07652 c1ccn(c1)c2ccc(cc2)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD07653 Cc1ccc(cc1)C(=O)/C=C(/CC(=O)c2ccc(cc2)Br)\c3ccccc3 BTB11341 c1ccc(cc1)c2nc(nn2c3ccccc3)S BTB13896 CC1c2cc(c(cc2CCN1)O)O.Br BTB13882 CCCCCCCCCCCC(=O)ON1C(=O)CCC1=O BTB13883 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)Nc3ccc(c(c3)Cl)Cl)C)C CD02061 c1ccc(cc1)NC(=O)C2C3CC(C2C(=O)O)C=C3 CD02186 COc1ccccc1NC(=O)C2C3CC(C2C(=O)O)C=C3 CD02191 c1cc(cc(c1)NC(=S)N(CCC#N)CCC#N)C(F)(F)F CD02226 c1ccc(cc1)NC(=N)SCc2ccc(cc2)[N+](=O)[O-].Br CD00229 CN(c1ccc(cn1)[N+](=O)[O-])NC(=O)c2cccs2 CD07294 CCc1cc2c(cc1C(=O)CSc3ccc(cc3)Cl)C(CCC2(C)C)(C)C CD02423 c1cc(ccc1n2c(=S)sc(n2)S)Cl BTB13892 CN(C)c1ccc(c(c1C#N)N(C)C)[N+](=O)[O-] CD07400 c1ccc(c(c1)C(F)(F)F)NCN2C(=O)CCC2=O CD04692 c1cc(ccc1Oc2ccc(c(c2C#N)Oc3ccc(cc3)Cl)[N+](=O)[O-])Cl CD07405 CC1CCN(CC1)C(=O)CC#N CD00230 Cc1cc(c(cc1CSC(=N)Nc2ccccc2)C)CSC(=N)Nc3ccccc3.Cl.Cl CD00240 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)/N=C/c2cc(cc(c2O)Cl)Cl CD07005 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(\C)/c3ccc(c(c3)CSc4ccccn4)OC CD02465 Cc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)Br)c4ccccc4 BTB11333 c1ccc(cc1)c2cc(nc(c2)c3ccc(cc3)Cl)c4ccccc4 BTB11335 c1ccc(cc1)c2cc(nc(c2)c3ccc(cc3)Br)c4ccccc4 BTB11336 c1ccc(cc1)/C(=C\C(=O)c2ccc(cc2)F)/CC(=O)c3ccccc3 BTB11337 c1ccc(cc1)/C(=C\C(=O)c2ccccc2)/CC(=O)c3ccc(cc3)[N+](=O)[O-] BTB11339 CCN(CC)S(=O)(=O)C1CCS(=O)(=O)C1 BTB13815 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)N3CCOCC3)C)C CD02281 CC(=O)c1ccccc1N/C=C/c2nnnn2c3ccccc3 BTB11259 Cc1c2ccccc2ncc1c3nnnn3c4ccccc4 BTB11260 CS/C(=N/C(=O)c1c(cccc1Cl)Cl)/NNc2c(cc(cc2Cl)Cl)Cl EN00068 c1cc(c(cc1NC(=S)NC(CO)(CO)CO)Cl)F CD07010 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC3CCN(CC3)Cc4ccccc4 CD06873 c1ccc(c(c1)C(=O)Nc2cccc(c2Cl)Cl)F CD06878 c1cc(ccc1c2nc(c(c(n2)N3CCCCC3)Cl)N4CCCCC4)Cl CD07162 Cc1ccc(cc1)n2c(nnn2)c3cnc4ccccc4c3C BTB11258 Cc1c(noc1NC(=O)Nc2c(onc2c3ccccc3Cl)C)C CD02304 Cc1cc(nc(n1)S/C=C/C(=O)c2ccc(cc2)F)C BTB11390 CS/C(=N/C(=O)c1c(cccc1Cl)Cl)/NCCc2ccc(cc2)Cl EN00058 c1ccc(cc1)c2cnnn2c3ccccc3Oc4ccc(cc4Cl)Cl CD08455 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3ccccc3F)Cl CD06925 c1ccc(cc1)CN/C=C/c2nnnn2c3ccc(cc3)Br BTB11261 CN(/C=C/c1n(nnn1)c2ccc(cc2)Cl)CCN(/C=C/c3n(nnn3)c4ccc(cc4)Cl)C BTB11264 Cc1ccc(cc1)NC(=O)C2C3CC(C2C(=O)O)C=C3 CD02228 Cc1cc(nc(n1)S/C=C/C(=O)c2ccc(cc2)Cl)C BTB11391 CSc1cc(n[nH]1)c2ccc(cc2)Cl EN00100 Cc1cc(nc(n1)S/C=C/C(=O)c2cccc(c2)Br)C BTB11392 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3cc(nn3C)C(F)(F)F EN00092 CCOC(=S)SCc1cc(cc2c1OCOC2)F CD08456 Cc1c(c(n[nH]1)C)/N=N/c2ccccc2Oc3ccc(cc3Cl)Cl CD08457 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CC(C3)Oc4ccc(cc4)Cl BTB13757 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=S)NC2CC3CCC2C3 CD02110 COc1cc(cc(c1OC)OC)C(=O)N(CCC#N)CCC#N CD02224 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3ccc(cc3)F CD02301 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=O)c2ccccc2C(=O)c3c(c(c(c(c3C)C)C)C)C)C)C CD02116 Cc1c(c(c(c(c1C)C)C(=O)c2ccccc2C(=O)NNC(=O)c3cccnc3)C)C CD02123 Cc1c(c(c(c(c1C)C)C(=O)c2c(c(c(c(c2Cl)Cl)Cl)Cl)C(=O)O)C)C CD02126 c1ccc(cc1)/C=C/C=C2C(=O)NC(=O)NC2=O CD00168 COc1ccc(cc1)OC(=O)c2c(cccc2Cl)Cl CD07412 c1cc(c(c(c1)Cl)Oc2ccc(c(c2C#N)Oc3c(cccc3Cl)Cl)[N+](=O)[O-])Cl CD07414 Cc1ccc(cc1)/C(=C\C(=O)c2ccccc2)/CC(=O)c3ccccc3 BTB11346 COc1ccc(cc1)CCNC(=O)c2ccc(cc2)[N+](=O)[O-] BTB13756 Cc1ccc(cc1)C(=O)C/C(=C(\C)/C(=O)c2ccccc2)/c3ccccc3 BTB11349 CCN(CC)/C=C/c1nnnn1c2ccc(cc2)Br BTB11351 c1ccc(cc1)c2ncc(c(n2)c3cccc(c3)Cl)c4nnnn4c5ccccc5 BTB11353 c1cc(ccc1C(=O)N2CC(C2)Oc3ccc(cc3)Cl)[N+](=O)[O-] BTB13758 c1cc(ccc1/C(=C/C=C(C#N)C#N)/Nc2ccc(cc2)Cl)Cl BTB11379 C1COCCN1C(=O)COCC(=O)N2CCOCC2 BTB13799 CCCCNC(=O)N1CCN(CC1)c2ncc(cn2)Br BTB13740 c1cc(c(c(c1)F)C(=O)O/N=C(/C=C/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N)F CD04782 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl BTB10286 CSc1c(c(nc(n1)c2ccc(cc2)Cl)SC)Cl CD07165 c1ccc(c(c1)C(=O)NCc2c(cccc2Cl)F)N CD07046 Cc1ccc(cc1)/C(=C/C=C(C#N)C#N)/Nc2ccc(cc2)OC BTB11377 CC1CN(CC(O1)C)c2ccc(cc2[N+](=O)[O-])C(=O)C CD07053 C#CC1(CCCCC1)NC(=O)N CD02314 c1ccc(cc1)c2c(cnn2c3ccc(cc3)[N+](=O)[O-])c4nnnn4c5ccccc5 BTB11256 C(CC(CCC(=O)O)(CCC(=O)O)[N+](=O)[O-])C(=O)O BTB10275 c1ccc(cc1)c2csc(n2)NC(=O)C34CC5CC(C3)CC(C5)C4 BTB13841 CCc1[nH]c2c(n1)c(=O)n(c(=O)n2C)C BTB13805 CC1(CC(=O)C(=NNc2cccc(c2)Br)C(=O)C1)C BTB13739 Cc1ccc(cc1)S(=O)(=O)N2CC(=O)NC(=O)C2 BTB12998 c1ccc(c(c1)C(=O)Nc2ccc(cc2F)F)F CD06884 COC(=O)CC1(N(C(=O)c2cc(ccc2O1)Br)c3ccc(c(c3)Cl)F)C(=O)OC CD06879 C1CN(CCC1CCCC2CCN(CC2)CN3C(=O)CCC3=O)CN4C(=O)CCC4=O CD04593 CC(C1CC1)N(c2ccccc2)C(=O)CCC(=O)O BTB13842 C/C(=N\NC(=O)c1ccc(cc1)Cl)/C2CC2 BTB13846 COC(=O)c1ccccc1N/C=C/c2nnnn2c3ccccc3 BTB11397 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCO CD06927 COc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)Br)c4ccccc4 BTB11330 COc1ccc(cc1)c2cc(cc(n2)c3ccc(cc3)I)c4ccccc4 BTB11331 Cc1ccc(cc1)N/C(=C/C=N/c2ccc(cc2)C)/c3ccc(cc3)Cl BTB11227 c1cc(sc1)/C=N/NC(=O)N CD02265 COc1ccc(cc1)C(=O)/C=C(/CC(=O)c2ccc(cc2)Br)\c3ccccc3 BTB11342 c1cc(sc1)CNC(=O)CCCC(=O)NCc2cccs2 CD07608 Cc1c(nnn1c2ccc(cc2Cl)Cl)C(=O)/C=C/N(C)C CD10519 c1ccc(cc1)OC(=O)c2cccc(c2F)C(=O)Oc3ccccc3 CD10533 c1cc(sc1)C2CCCN2c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD10537 C1CCN(C1)C(=O)CCCC(=O)N2CCCC2 CD07614 Cc1ncc(c(n1)c2ccccc2)c3nnnn3c4ccc(cc4)Cl BTB11400 CSC(=CC(=O)c1ccc(cc1)Cl)SC EN00099 CSC(=CC(=O)c1ccco1)SC EN00101 C/C(=N\OC(=O)c1ccc(cc1)[N+](=O)[O-])/c2ccc(cc2)F CD02159 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3ccccc3OC CD02308 c1ccc(cc1)C=C2C(=O)NC(=O)NC2=O CD00165 C1CC(CC=C1)C=C2C(=O)NC(=O)NC2=O CD00167 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3c(onc3c4ccccc4Cl)C CD04729 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3cccc(c3Cl)Cl CD02313 COc1cccc(c1OC)C=C2C(=O)NC(=O)NC2=O CD00169 c1ccc(cc1)/N=C/2\NC(=O)C(S2)CC(=O)Nc3ccccc3Cl CD00202 COc1ccc(cc1)N/C(=C\C=C(C#N)C#N)/c2ccc(cc2)Cl BTB11380 c1cc(ccc1/C(=C\C=N\c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl BTB11382 Cc1ccc(cc1)C(=O)/C=C/Sc2nc(cc(n2)C)C BTB11386 CCc1ccc(cc1)C(=O)/C=C/Sc2nc(cc(n2)C)C BTB11387 Cc1cc(nc(n1)S/C=C/C(=O)c2ccc(cc2)Br)C BTB11393 c1cc(ccc1C(=O)ON=C2CCCCC2)Cl CD02160 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C(\C)/c3ccc(cc3)F CD02380 c1cc(cc(c1)Oc2ccc(cc2)N)Oc3ccc(cc3)N BTB13887 Cc1ccc(c(c1)Cl)NC(=O)CSC2CC(=O)N(C2=O)c3ccccc3 CD02237 Cc1c(c(c(c(c1C)C)CSC2CC(=O)N(C2=O)c3ccccc3)C)C CD02240 CCOC(=O)C(=CNc1ccc(o1)C(=O)OC)C(=O)OCC EN00164 Cc1c(nnn1c2cc(cc(c2)Cl)Cl)C(=O)C CD09955 COC(CNc1cccc(c1C#N)Cl)OC CD09963 Cc1c(c(on1)C)S(=O)(=O)N2CCOCC2 CD10612 Cc1c(c(on1)C)S(=O)(=O)N2CCCC2 CD10613 c1cc(cc(c1)S(=O)(=O)NCc2ccc(cc2F)F)C(F)(F)F CD10758 Cc1c(c(no1)c2ccccc2)C(=O)NCc3ccc(cc3F)F CD10767 COc1cc(nc(n1)N)c2ccc(cc2)Cl EN00150 COC(=O)CCNc1ccc(cc1)Cl EN00152 COC(=O)c1ccsc1NC(=O)c2ccccc2 GK02860 Cn1c2c(c(=O)n(c1=O)C)[nH]c(n2)NCCO BTB13948 c1cc-2c(cc1S(=O)(=O)NCCO)Cc3c2ccc(c3)S(=O)(=O)NCCO BTB13868 c1cc-2c(cc1S(=O)(=O)NCCO)C(=O)c3c2ccc(c3)S(=O)(=O)NCCO BTB13869 Cc1ccc(cc1)C(=O)Nc2c(ccs2)C(=O)OC GK02867 Cc1c(nnn1c2ccccc2Oc3ccc(cc3Cl)Cl)c4ccccc4 CD08445 Cc1c(c(on1)C)S(=O)(=O)Oc2ccc(cc2)OC CD10615 Cc1c(c(on1)C)S(=O)(=O)Oc2ccccc2 CD10616 c1ccc(c(c1)C(=O)NN)NC(=O)c2ccccc2Cl EN00186 Cc1c(c(on1)C)S(=O)(=O)Oc2ccc(cc2)Cl CD10617 COc1ccc(cc1)NC(CC(=O)C2CC2)c3ccccc3 BTB13844 Cc1c(c(c(c(c1C)C)C(=O)/C(=N\OC(=O)c2ccc(c(c2)Cl)Cl)/c3ccccc3)C)C CD02417 c1ccc(c(c1)C(=O)NN)NC(=O)c2c(cccc2F)F EN00187 Cc1ccc(n1N(C)c2ccc(cn2)[N+](=O)[O-])C CD08598 CCc1cc2c(cc1C(=O)CSc3ccccn3)C(CCC2(C)C)(C)C CD02424 Cn1c(cc(n1)C(F)(F)F)OC(=O)c2ccccc2Cl EN00087 Cn1c2c(c(=O)n(c1=O)C)[nH]c(n2)N(C)Cc3ccccc3 BTB13949 Cc1c(c(n(n1)c2ccccc2)C)/N=N/c3ccccc3Oc4ccc(cc4Cl)Cl CD08443 Cc1c(c(n(n1)C)C)/N=N/c2ccccc2Oc3ccc(cc3Cl)Cl CD08449 Cc1cc(c(cc1Cl)Cl)C(=O)N(c2ccccc2)C(C)C3CC3 BTB13845 c1ccnc(c1)SCc2cc(cc(c2)Br)Br CD08478 CS(=O)(=O)Cc1cc(cc2c1OCOC2)F CD08494 CC(C)(C)c1csc(n1)Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] CD08497 COc1ccc(cc1)N(C(=C)C2CC2)C(=O)c3ccc(cc3)F BTB13849 CC(C1CC1)N(c2ccccc2)C(=O)C BTB13850 Cc1c(nnn1c2cc(ccc2Cl)Cl)c3ccn[nH]3 CD10580 CCOC(=O)/C(=N/Nc1ccccc1C)/C(=O)C BTB13857 CCOC(=O)/C(=N/Nc1ccccc1)/C(=O)C BTB13858 COC(=O)Nc1cccc(c1F)NC(=O)OC CD10583 CN(C)Nc1ccc(c(c1C#N)NN(C)C)[N+](=O)[O-] CD07449 Cc1cc(ccc1O)C2(c3ccccc3N(C2=O)Cc4ccccc4)c5ccc(c(c5)C)O BTB13809 Cc1c(nnn1c2ccc(c(c2)Cl)Cl)C(=O)/C=C/N(C)C CD10518 c1ccn(c1)c2cccc(c2)C(F)(F)F CD02363 c1cc(c(c(c1)CC#N)F)CC#N CD10597 CN(c1c(cccn1)[N+](=O)[O-])NC(=O)c2ccccc2F CD07442 CN(c1c(cccn1)[N+](=O)[O-])NC(=O)c2ccccc2Cl CD07448 c1ccc(cc1)CN2CCC(CC2)Nc3c4ccsc4ncn3 GK02887 c1c(c(cc(c1[N+](=O)[O-])N2CCCC2)N3CCCC3)C#N CD07462 c1cc(c(c(c1)Cl)SCc2c(cccc2Cl)F)[N+](=O)[O-] CD07467 c1csc2c1c(ncn2)N3CCN(CC3)C(=S)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F GK02901 Cn1c(cc(n1)C(F)(F)F)OS(=O)(=O)c2ccc(cc2Cl)Cl CD10535 c1cc(c(c(c1)C(=O)Oc2ccc(cc2Cl)Cl)F)C(=O)Oc3ccc(cc3Cl)Cl CD10540 CC(C)(NC(=S)Nc1ccccc1)/N=N/c2ccccc2 CD10628 COCCCNC1=C(C(=O)NC(S1)c2cccc(c2)[N+](=O)[O-])C#N CD02617 COc1cc(cc(c1OC)OC)C(=O)O/N=C(/c2ccc3c(c2)OCO3)\N CD02625 c1c(cc(c(c1[N+](=O)[O-])Sc2nc[nH]n2)[N+](=O)[O-])C(F)(F)F CD08589 Cc1c(c(on1)C)S(=O)(=O)NNC(=O)Nc2ccc(cc2)Cl CD10633 COCCCNC(=S)NNC(=O)CC#N CD02628 CC(C)(C)n1cnnc1Sc2ccc(cn2)[N+](=O)[O-] CD07587 CC(C)(C)n1cnnc1SCc2c(cccc2Cl)F CD07589 C1CCN(C1)C(=O)CC(=O)N2CCCC2 CD02343 CCOC(=O)C(=CNc1c(ccs1)C(=O)OC)C(=O)OCC GK02872 c1cc(c(c(c1)Cl)/C=C/c2cc[nH]n2)Cl CD09853 C1CSCCN1C(=O)C(Cl)(Cl)Cl CD07926 c1cc(c(cc1Cl)Cl)C(=O)N2CCSCC2 CD07928 c1cc(c(c(c1)F)C(=O)N2CCSCC2)F CD07929 CN(C)/C=C(\C#N)/C(=O)N1CCCC1 CD07554 CSC1=C(C(=O)NC(S1)c2ccc(cc2Cl)Cl)C#N CD07555 CC(C)(C)n1cnnc1S CD07576 c1ccc(c(c1)NC2=C(C(=O)NC(S2)c3c(cccc3Cl)Cl)C#N)Cl CD07581 Cc1c(c(c(c(c1C)C)C(=O)c2ccc(cc2)NC(=O)c3ccccc3C(=O)O)C)C CD02330 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)/C(=C/c4ccccn4)/C#N CD02335 COC(=O)C1=C(CCCC1)N BTB13933 Cc1c(c(c(cn1)CSc2nc(cs2)C(C)(C)C)CO)O CD08419 Cc1cccc(c1)N(C)C(=S)Oc2ccc3ccccc3c2 BTB13928 CN(C)/C=C(\C#N)/C(=O)Nc1cc(cc(c1)Cl)Cl CD08649 c1c(cc(cc1C(F)(F)F)NC(=O)CCCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD07600 COc1ccc2c(c1)nnc3n2c(nn3)SCC(=O)NN BTB11367 CCN(CC)C(=O)CSc1nnc2n1c3ccc(cc3nn2)OC BTB11368 c1ccc2c(c1)nnc3n2c(nn3)SCC(=O)NN BTB11370 CN(C)/C=N/N(C)c1ccc(cn1)[N+](=O)[O-] CD07562 CCN(CC)C(=O)CSc1nnc2n1c3ccc(cc3nn2)C BTB11468 CNC(=O)c1ccccc1Sc2cccc3c2c(ccc3)C(=O)O BTB11475 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccc(c(c2)CSc3ccccn3)OC CD02470 CC(=O)c1ccc(c(c1)CSCC(=O)Nc2ccc(cc2)Cl)OC CD02478 CC(C)(c1ccc(cc1)Oc2ccc3c(c2)C(=O)N(C3=O)C)c4ccc(cc4)Oc5ccc6c(c5)C(=O)N(C6=O)C BTB13885 Cc1ccc(cc1C)Oc2ccc(cc2)[N+](=O)[O-] BTB13886 COc1ccccc1Oc2ccc(c(c2C#N)Oc3ccccc3OC)[N+](=O)[O-] CD07415 CCN(CC)/C=C/c1nnnn1c2ccc(cc2)C BTB11350 Cc1ncc(c(n1)c2cccc(c2)Cl)c3nnnn3c4ccccc4 BTB11352 CSC(=CC(=O)c1cccs1)SC EN00102 c1ccc(c(c1)NC2=C(C(=O)NC(S2)c3ccncc3)C#N)Cl CD07582 c1cc(ccc1Oc2ccc(c(c2C#N)Oc3ccc(cc3)F)[N+](=O)[O-])F CD07408 c1cc(c(cc1Cl)Cl)Oc2ccc(c(c2C#N)Oc3ccc(cc3Cl)Cl)[N+](=O)[O-] CD07409 c1cc(c(c(c1)Cl)C(=O)Oc2ccc(cc2)[N+](=O)[O-])Cl CD07411 c1ccc2c(c1)c(c[nH]2)C(=O)C(F)(F)F BTB13881 CC(C)(C)c1csc(=S)n1CCc2ccc(cc2)Cl CD08400 CC(C)(c1ccc(cc1)Oc2ccc(c(c2)C(=O)O)C(=O)O)c3ccc(cc3)Oc4ccc(c(c4)C(=O)O)C(=O)O BTB13888 C/C(=N\OC(=O)c1c(c2ccccc2s1)Cl)/c3ccc(c(c3)CN4CCOCC4)OC CD02482 CN1C(=O)c2ccc(cc2C1=O)[N+](=O)[O-] BTB13889 c1cc(c(c(c1)Cl)CSCc2ccc(cc2)Cl)F CD07472 CC(C)C1CCC(C(C1C#N)CCC(=O)C)(C)OC(=O)C BTB13925 CC(=O)c1ccc(c(c1)OC)CN2CCOCC2 CD02459 Cc1ccc2c(c1)nc([nH]2)S/C=C/C(=O)c3ccc(cc3)Cl BTB11321 CCc1ccc(cc1)C(=O)/C=C/Sc2nc3ccccc3o2 BTB11322 c1cc(c(c(c1)[N+](=O)[O-])C(=O)Nc2ccc(cc2)F)C(=O)O CD02460 CC(=O)N(c1ccc(cc1)C(F)(F)F)S(=O)(=O)c2ccc(cc2)N3C(=O)CCC3=O GK02873 c1ccc(cc1)Oc2cccc(c2)COC(=O)NC(=O)c3ccccc3Cl CD08383 c1ccc(c(c1)C(=O)NNC(=O)/C=C/C(=O)O)n2cccc2 CD02605 c1ccc(c(c1)C(=O)NN)NC(=O)c2cccs2 EN00194 Cc1c(nnn1c2c(cc(cc2Cl)Cl)Cl)C(=O)C CD09968 COC(=O)c1ccccc1NC(=S)OC EN00195 Cc1ccc(n1N(C)c2cccc(c2C#N)F)C CD08594 Cc1c(c(n(n1)C)N)[N+](=O)[O-] EN00107 C1CCN(C1)C(=O)/C=C/2\NC(=O)CS2 CD07667 C=CCNc1c2ccsc2ncn1 GK02879 Cc1cc(n(n1)C2=NCCN2S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C CD08571 Cc1c(c(c(c(c1C)C)C(=O)Cc2ccccc2)C)C CD02388 Cc1c(c(c(c(c1C)C)C(=O)/C(=N/N=C/c2cc(cc(c2O)Cl)Cl)/c3ccccc3)C)C CD02398 c1cc(c(cc1Cl)Cl)C(=O)Sc2nc(sn2)SC(=O)c3ccc(cc3Cl)Cl CD08536 C1CS(=O)(=O)CC1NCC(=O)O BTB13823 C1C=C(CS1(=O)=O)Cl BTB13824 CS/C(=N/C(=O)c1c(cccc1Cl)Cl)/NNc2ccccc2C(F)(F)F EN00072 CN(c1c(cccn1)[N+](=O)[O-])NC(=O)c2ccc(cc2)Cl CD07445 c1cc(ccc1C(=O)/C=C/S(=O)(=O)c2ccc(cc2)Br)F BTB11383 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c4ccsc4ncn3 GK02909 Cc1ccc(cc1)/C(=C/C=C(C#N)C#N)/Nc2ccc(cc2)Cl BTB11271 c1c(c(sc1S(=O)(=O)N)Br)Br CD08511 Cc1cc(cc(n1)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD10562 c1cc(ccc1C#N)S(=O)(=O)NC2CCCCNC2=O CD10691 c1cc(c(c(c1)C(=O)N)F)C(=O)N CD10573 c1cc(ccc1CCNc2c3ccsc3ncn2)Cl GK02915 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccc(cc2)OC(F)(F)F GK02917 c1ccc(c(c1)C2=NCCCN2)Sc3c(cccn3)[N+](=O)[O-].Cl CD07453 c1cc(c(c(c1)Cl)CSc2c(cccn2)[N+](=O)[O-])F CD07466 c1ccc2c(c1)c\3c([nH]2)CCC/C3=N\OC(=O)c4ccc(cc4Cl)Cl BTB13761 Cc1ccc(cc1)C(=O)/C=C(/CC(=O)c2ccc(cc2)I)\c3ccccc3 BTB11358 c1cc(c(c(c1)Cl)CSc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F CD07468 c1cc(c(c(c1)Cl)CSc2ccc(cc2[N+](=O)[O-])Cl)F CD07469 c1cc(c(c(c1)Cl)CSc2ccc(cn2)[N+](=O)[O-])F CD07471 Cc1ccc(cc1)/C(=C\C=C(C#N)C#N)/Sc2nc3ccccc3s2 BTB11276 COC(=O)CC1(N(C(=O)c2cc(ccc2O1)Cl)c3ccc(cc3F)F)C(=O)OC CD06963 C#CCNS(=O)(=O)c1ccc(cc1)C#N CD10693 c1ccc(c(c1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)n3cccc3 CD02572 CCN(CC)c1c2ccsc2ncn1 GK02877 Cc1c(c(c(c(c1C)C)C(=O)CCc2cccc(c2)NC(=O)C3CCC3)C)C CD02588 c1cc(c(c(c1)Cl)C(=O)N=C2NCCN2)Cl EN00051 Cc1c(c(c(c(c1C)C)CS/C(=C(/C#N)\C(=O)NCCCOC)/Nc2ccc(cc2)F)C)C CD02589 Cc1ccc(cc1)C(=O)/C=C(/CC(=O)c2ccc(cc2)[N+](=O)[O-])\c3ccccc3 BTB11359 CC(C)(CO)NC(=S)Nc1ccc(cc1F)F CD07008 COc1ccc(cc1)C(=O)/C=C(/CC(=O)c2ccc(cc2)F)\c3ccccc3 BTB11360 CC(C)(CO)NC(=S)Nc1ccc(c(c1)Cl)F CD07007 c1ccc2c(c1)nnc3n2c(nn3)SCC(=O)N4CCOCC4 BTB11369 CCN(CC)C(=O)CSc1nnc2n1c3ccccc3nn2 BTB11372 CC(C(=O)NN)Oc1ccc(cc1Cl)Cl BTB11375 CCCC(=O)/C(=C/Nc1c(ccs1)C(=O)OC)/C(=O)OCC GK02875 Cc1c(c(c(c(c1C)C)C(=O)CCc2cccc(c2)/N=C/c3cc(cc(c3O)Cl)Cl)C)C CD02584 c1ccc(c(c1)C(=O)N2CCSCC2)Cl CD07931 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(/c3ccc4c(c3)OCO4)\N CD02621 c1cc2c(cc1/C(=N/OC(=O)c3ccc(c(c3)Cl)Cl)/N)OCO2 CD02622 c1cc(ccc1C(=O)N2CCSCC2)Cl CD07932 c1ccc(cc1)CN/C=C/c2nnnn2c3ccccc3 BTB11262 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] BTB10282 c1cc(ccc1Sc2ccc(cc2Cl)[N+](=O)[O-])Cl BTB10283 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3c(cccc3Cl)Cl CD02345 c1cc-2c(cc1S(=O)(=O)N(CCO)CCO)C(=O)c3c2ccc(c3)S(=O)(=O)N(CCO)CCO BTB13866 c1cc(ccc1CNC(=O)c2ccc(cc2)F)C(F)(F)F CD10747 c1cc(ccc1CNC(=O)c2cc(cc(c2)Cl)Cl)C(F)(F)F CD10749 COc1cc(nc(n1)N)c2ccccc2 EN00147 CN(C)/C=C(\C#N)/C(=O)/N=C/N(C)C CD07546 c1ccc(cc1)c2c(cnc(n2)c3ccccc3)c4nnnn4c5ccc(cc5)F BTB11408 Cc1c(nnn1c2ccc(cc2C#N)Cl)C(=O)C CD10643 Cc1c(c(on1)C)S(=O)(=O)Nc2ccccc2 CD10647 c1ccc(cc1)Oc2c(c(c(c(c2F)F)Oc3ccccc3)F)F BTB13848 Cc1c(c(c(c(c1C)C)CN2CCCC2)C)C CD00220 c1ccc(c(c1)Oc2ccc(cc2Cl)Cl)S(=O)(=O)N CD08381 c1cc(ccc1C(=O)OC2C(OCCO2)OC(=O)c3ccc(cc3)[N+](=O)[O-])[N+](=O)[O-] BTB13776 c1ccc(c(c1)NN=C(C#N)C#N)Oc2ccc(cc2Cl)Cl CD08429 CC(C)(C)c1c(sc(n1)NC(=N)N)Br.Br CD08433 Cc1c(nnn1c2ccc(cc2Cl)Cl)C(=O)C CD10513 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)N[C@@H](CCC(=O)N)C(=O)O BTB13779 Cc1c(c(c(c(c1C)C)S(=O)(=O)/N=C/N(C)C)C)C CD07547 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])Sc2nc[nH]n2 CD08587 Cc1c(nnn1c2ccc(cc2Cl)Cl)c3ccnc(n3)N CD10636 Cc1ccc(c(c1)Cl)NC(=O)c2c(cccc2[N+](=O)[O-])C(=O)O CD02461 C/C(=N\OC(=O)c1cc(c(c(c1)OC)OC)OC)/c2ccc(c(c2)CSc3ccccn3)OC CD02468 CC(=O)Nc1ccc2c(c1)C(=O)N(C2=O)C BTB13890 Cc1cc(c(c(c1C)I)C)C CD07686 COc1ccc(cc1)c2[nH]c(nn2)S BTB13897 CCOC(=O)/C(=N\Nc1ccccc1)/C(=O)CSC#N BTB13778 c1ccc(c(c1)Oc2ccc(cc2Cl)Cl)S(=O)(=O)Nc3cc(cc(c3)Cl)Cl CD08390 c1ccc(c(c1)Oc2ccc(cc2Cl)Cl)S(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD08391 c1ccc(c(c1)Oc2ccc(cc2Cl)Cl)S(=O)(=O)N3CCCCC3 CD08393 Cc1c(c(c(c(c1C)C)CSc2ccccn2)C)C CD02166 Cc1c(c(c(c(c1C)C)CSc2nc3ccccc3o2)C)C CD02172 CCOC(=O)c1nn(c(=N)s1)c2ccc(cc2)C BTB13780 CO[C@@H]1[C@@H]([C@H]([C@@H](O1)COC(=O)c2ccccc2)OC(=O)c3ccccc3)OC(=O)c4ccccc4 BTB13781 CC(C)(C)c1csc(n1)NC(=O)Nc2ccc(cc2)Cl CD08396 c1ccc(c(c1)Oc2ccc(cc2Cl)Cl)S(=O)(=O)Nc3ccc(c(c3)Cl)F CD08397 Cc1cc(cc(c1Cl)C)OCc2c(c(c(c(c2C)C)C)C)C CD02179 Cc1c(c(c(c(c1C)C)I)C)C CD07684 c1cc2c(cc1Br)C(C(=O)N2)O CD07798 c1cc(c(nc1)Sc2nnc(s2)N)[N+](=O)[O-] CD07800 CNC(=O)c1cccc2c1c(ccc2)Sc3ccccc3CO BTB11482 c1ccc(cc1)C=CC=Cc2cc[nH]n2 CD09846 CC(C)(C)n1cnnc1SCc2c(cccc2Cl)Cl CD07585 CC(C)(C)n1cnnc1Sc2c(cccn2)[N+](=O)[O-] CD07586 COc1ccc(cc1)C(=O)/C=C/Nc2cccc(c2)Cl BTB11395 Cc1c(c(c(c(c1C)C)CSC2=NCCS2)C)C CD02177 Cc1c(c(c(c(c1C)C)COc2ccc(cc2Cl)Cl)C)C CD02181 c1ccc(cc1)c2c(cnc(n2)c3ccccc3)c4nnnn4c5ccccc5 BTB11404 Cc1ccc(cc1)n2c(nnn2)c3cnc(nc3c4ccccc4)c5ccccc5 BTB11405 c1ccc(c(c1)CO)Sc2cccc3c2c(ccc3)C(=O)O BTB11481 CN(C)/C=N/S(=O)(=O)c1ccc(c(c1)Cl)Cl CD07557 CN(C)/C=N/S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F CD07558 CNC(=O)c1ccccc1Sc2ccccc2 BTB11485 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCSCc3c(cccc3Cl)F CD07842 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)O/N=C(\C)/c2ccccc2O CD02524 c1c(cc(cc1C(F)(F)F)S(=O)(=O)N2CCSCC2)C(F)(F)F CD07852 Cc1ccc(n1c2c(ccs2)C(=O)OC)C GK02930 Cc1ccc(n1c2c(ccs2)C(=O)O)C GK02934 CC(=O)c1ccc(c(c1)CSc2ccccn2)OC CD02433 c1ccn(c1)CC2CCCN(C2)c3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD09945 Cc1cc(cc(c1F)C)S(=O)(=O)N2CCCC(C2)Cn3cccc3 CD09946 COC(CNC(=S)Nc1ccccc1Cl)OC CD09947 CCOC(=O)c1cnn(c1N)c2c3ccsc3ncn2 GK02918 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccccc2 GK02921 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)C(F)(F)F GK02924 c1c(cc(c(c1[N+](=O)[O-])N2CCSCC2)[N+](=O)[O-])C(F)(F)F CD07853 c1cc(sc1)C(=O)NCCc2ccc(cc2)Cl CD08669 c1ccc(c(c1)C(=O)NCCc2ccc(cc2)Cl)Cl CD08671 CS/C(=N/S(=O)(=O)c1ccccc1)/NNC(=O)c2ccc(cc2)Cl CD08675 c1cc(c(cc1c2ccn[nH]2)Cl)Cl CD08608 c1c(c(sc1S(=O)(=O)N2CCOCC2)Br)Br CD08623 COC(=O)c1c(ccs1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD08632 C/C(=N\O)/c1ccc(c(c1)CSc2ccccn2)OC CD02446 c1cc(ccc1c2cncnc2N)Cl HAN00088 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN/C(=N/S(=O)(=O)c3ccccc3)/SC CD08680 c1ccc(cc1)n2c(nnn2)Sc3c4ccsc4ncn3 GK02926 c1cc(ccc1C(=O)NNc2c3ccsc3ncn2)Cl GK02928 Cc1c(c(no1)c2ccccc2Cl)C(=O)c3ccc(cc3)F CD08716 COC(=O)/C=C(/C(=O)OC)\Nc1ccsc1C(=O)OC CD08720 Cc1c(c(no1)c2ccccc2)C(=O)c3ccc(cc3)F CD08724 c1cc(c(c(c1NCCO)C#N)NCCO)[N+](=O)[O-] CD07420 c1cc(c(c(c1)NC(=O)NCc2cccnc2)F)NC(=O)NCc3cccnc3 CD10587 Cc1c(c(no1)c2ccccc2Cl)C(c3ccc(cc3)F)O CD08747 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3ccccc3 CD08647 c1cc(c(c(c1)[N+](=O)[O-])C(=O)Nc2ccc(c(c2)Cl)Cl)C(=O)O CD02456 c1ccc(c(c1)C(=O)NN)n2cccc2 CD02571 c1ccc(c(c1)C(=O)N/N=C/c2cccnc2)n3cccc3 CD02573 c1ccc(cc1)/C=C/C=N/NC(=O)c2ccccc2n3cccc3 CD02574 c1cn[nH]c1c2cc(cc(c2O)F)F CD07636 CN(C)/C=C/C(=O)c1cc(cc(c1O)Cl)F CD07634 Cc1c(c(n(n1)C)C)NS(=O)(=O)c2cc(sc2Cl)Cl CD09895 CSCC(CSC)OC(=O)NC(=O)c1c(cccc1Cl)Cl CD09894 Cn1c2c(c(=O)n(c1=O)C)[nH]c(n2)[N+](=O)[O-] BTB13947 c1ccc(cc1)CN2c3ccccc3CCC2=S FM00075 C1CC(CCC1C(=O)O)C(=O)O FM00078 c1ccc2c(c1)C(OC2=O)Nc3ccc(cc3F)F CD07937 CN(C)/C=c\1/c(=O)[nH]/c(=C\C(=O)c2cccs2)/s1 CD07669 CCOc1ccc(cc1)/C=N/NC(=S)NC2CC3CC2C4C3CC=C4 CD02544 Cc1c(sc(=S)n1CCc2ccc(cc2)Cl)C(=O)C CD09857 c1cc2c(cc1/C(=N/O)/N)OCO2 CD02598 c1cc(ccc1C(=O)CCCC(=O)c2ccc(cc2)F)F CD08760 c1ccc2c(c1)/C(=C\C3CC4CC3C=C4)/C(=O)N2 CD02656 COCCCNC1=C(C(=O)NC(S1)c2cccs2)C#N CD02657 COCCCNC1=C(C(=O)NC(S1)C2CCC=CC2)C#N CD02658 CCOC(=O)c1nc2ccccc2c(=O)n1/N=C/c3cc(cc(c3O)Cl)Cl CD02660 c1cc(c(cc1Cl)NC(=O)N)Cl CD02675 CN(c1ccccc1[N+](=O)[O-])NC2c3ccccc3C(=O)O2 CD07915 Cc1ccc(cc1)C(=O)c2c(cc(c3c2C(=O)CCC3)c4ccccc4)c5ccccc5 BTB11354 COc1ccc2c(c1)nnc3n2c(nn3)SCC(=O)O BTB11365 COc1ccc2c(c1)nnc3n2c(nn3)SCC(=O)N4CCOCC4 BTB11366 CC(C)(C)n1cnnc1Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F CD07590 c1cc(c(cc1F)F)NC(=O)CCCC(=O)Nc2ccc(cc2F)F CD07596 Cc1cc(c(c(c1)C)I)C CD07694 c1cc(c(c(c1)Cl)Cl)NC(=O)/C=C/C(=O)Nc2cccc(c2Cl)Cl CD07697 c1cc(c(c(c1)Cl)CSCCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)F CD07908 Cn1c2c(cc(s2)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)c(n1)C(F)(F)F GK02698 Cc1ccsc1/C=C/NC(=O)Nc2ccc(cc2)C(C)C GK02703 c1cc(c(cc1Cl)Cl)OC(=O)/C=C/C(=O)Oc2ccc(cc2Cl)Cl CD07710 Cc1c(c(c(c(c1C)C)CSC(=S)SC(C)(C)C)C)C CD07736 COc1cccc(c1O)/C=N/NC(=S)N CD02769 Cc1c(c(c(c(c1C)C)CO)C)C CD02784 c1c(cc(cc1Cl)Cl)NC(=O)CCCC(=O)Nc2cc(cc(c2)Cl)Cl CD07597 c1cc(c(c(c1)Cl)Cl)NC(=O)CCCC(=O)Nc2cccc(c2Cl)Cl CD07598 Cc1c(c(no1)c2ccccc2)NC(=O)N(CCC#N)Cc3ccccc3 CD02346 CC(=O)c1ccc(o1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10821 c1cc(c(cc1F)F)S(=O)(=O)NCc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10810 Cc1cc(c-2c(c1)CC(c3c2[nH]c(n3)c4ccccc4)(C)C)C CD02715 c1c(c(c(cc1Cl)Cl)O)/C=N/C(=C(\N=C\c2c(c(cc(c2)Cl)Cl)O)/C#N)/C#N CD02717 c1ccc2c(c1)CCN(C2)C(=O)C(Cl)(Cl)Cl DSHS01061 c1ccc(cc1)CN2c3ccccc3CCC2=O FM00070 CN(C1CC2CC1C=C2)S(=O)(=O)c3cc(sc3Cl)Cl CD09902 c1cc(c(c(c1)Cl)C(=O)NC(=O)ON(Cc2ccc(cc2)Cl)Cc3ccc(cc3)Cl)Cl CD09914 c1ccc(cc1)C(=O)OCc2cccc(c2F)COC(=O)c3ccccc3 CD10696 CCN(Cc1ccccc1)c2[nH]c3c(n2)n(c(=O)n(c3=O)C)C BTB13950 CC(=O)N(Cc1ccccc1)c2[nH]c3c(n2)n(c(=O)n(c3=O)C)C BTB13951 c1ccc(cc1)c2c(c2=O)c3ccccc3 BTB10303 c1ccc(cc1)C2=C(C(=O)C(=C2c3ccccc3)c4ccccc4)c5ccccc5 BTB10304 Cc1c(c(c(c(c1C)C)C(=O)CCc2cccc(c2)NC(=O)C(Cl)Cl)C)C CD02596 Cc1cc(cc(c1F)C)S(=O)(=O)Nc2ccsc2C(=O)OC CD08631 CC(C)(C)C(=O)c1c(c2c(c(sc2s1)C(=O)C(C)(C)C)N)N CD08635 CN(C)/C=C(\C#N)/C(=O)Nc1cc(ccc1Cl)C(F)(F)F CD08645 CCOC(=O)CSc1ccc(cc1[N+](=O)[O-])C(=O)N(Cc2ccc3c(c2)OCO3)c4ccc(cc4)F DSHS00951 c1cc(ccc1c2nc(on2)CSC(=N)N)Cl.Cl CD02761 CN(C)/C=C(\C#N)/C(=O)NCCCOC CD08655 c1cc(ncc1[N+](=O)[O-])Sc2nnc(s2)N CD07802 CN(c1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])NC2c3ccccc3C(=O)O2 CD07918 Cc1ccc2c(c1)nnc3n2c(nn3)SCC(=O)O BTB11465 CCOC(=O)C(Cc1c(c(c(c(c1C)C)C)C)C)C#N CD02600 c1ccc(cc1)NC(=O)OC2CCSC2 CD10730 Cc1c(c(c(c(c1C)C)C(=O)C2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C)C CD10724 c1ccc2c(c1)c(=O)[nH]c(n2)c3ccccc3O DSHS00977 Cc1c(c(n(n1)C)NNC(=O)c2c(cccc2F)F)[N+](=O)[O-] EN00278 CCOC(=O)c1cnn(c1N)c2c(c(nn2C)C)[N+](=O)[O-] EN00281 c1cc(ccc1Sc2ccc(cc2C(=O)Nc3ccncc3)[N+](=O)[O-])Cl DSHS00978 c1ccc(cc1)Sc2ccc(cc2C(=O)Nc3ccncc3)[N+](=O)[O-] DSHS00980 C1CSCCN1C(=O)C(Cl)Cl CD07925 Cc1c(c(c(c(c1C)C)C(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3F)F)C)C CD10732 c1csc2c1c(ncn2)NNC=C(C#N)C#N GK02937 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)C#N)Oc3ccc(cc3Cl)Cl CD10699 c1cc(cnc1)OS(=O)(=O)c2ccc(cc2)C#N CD10704 c1cc(c(cc1Cl)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl HAN00072 CCN(CC)C(=O)CSc1nnc2n1c3ccc(cc3nn2)Cl BTB11460 c1cc-2c(cc1Cl)NNc3n2c(nn3)SCC(=O)O BTB11461 C/C(=N\OC(=O)c1ccccc1Cl)/C=C/c2ccccc2 EN00220 c1cc(c(cc1S(=O)(=O)NCc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl)Cl CD10814 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)c3ccc(cc3)F CD08705 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(\C)/C=C/c3ccccc3 EN00223 c1ccc(c(c1)SC(=O)Nc2ccc(cc2)Cl)Cl EN00231 CNC(=O)Sc1ccccc1Cl EN00233 c1ccc2c(c1)-c3c(cccc3C(=O)OCCO)C2=O BTB13867 COC(=O)c1ccsc1NC(=O)c2cccs2 GK02863 Cc1ccc2c(c1)nnc3n2c(nn3)SCC(=O)N4CCOCC4 BTB11467 COc1ccc(cc1)C(=O)Nc2c(ccs2)C(=O)OC GK02869 COC(=O)c1ccsc1NC(=O)c2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-] GK02870 c1cc(c(cc1F)F)C(=O)NCc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10823 CC(=O)OCc1cccc2c1c(ccc2)Sc3ccccc3C(=O)O BTB11478 Cc1c(c(c(c(c1C)C)CO/N=C(\c2ccccc2)/C(=O)c3c(c(c(c(c3C)C)C)C)C)C)C CD02472 Cc1c(c(n(n1)C)O)C(=O)c2c(onc2c3c(cccc3Cl)Cl)C CD08707 c1ccc\2c(c1)CC/C2=N\OC(=O)c3cccc(c3)F FM00064 COC(=O)c1ccsc1NC(=O)c2ccco2 GK02866 CC(=O)Nc1ccc(cc1)S(=O)(=O)NNc2c3ccsc3ncn2 GK02919 c1cc(cnc1)/C=N/NC(=S)NC2CC3CC2C4C3CC=C4 CD02542 COc1cc(cc(c1OC)OC)C(=O)Nc2c(ccs2)C(=O)OC GK02871 COc1cc(ccc1O)/C=N/NC(=S)NC2CC3CC2C4C3CC=C4 CD02543 CC1CC(CC(C1)(C)C)NC(=S)NC2CC3CC2C4C3CC=C4 CD02554 COC(=O)c1c(ccs1)NC(=O)C(Cl)Cl CD08691 c1cc(ccc1S(=O)(=O)NNc2c3ccsc3ncn2)Cl GK02931 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)O/N=C(\C)/c2ccc(c(c2)CSc3ccccn3)OC CD02474 c1cc(sc1)C(=O)N2CCN(CC2)c3c4ccsc4ncn3 GK02938 Cc1cc(c(cc1Cl)C)S(=O)(=O)N2CCN(CC2)c3c4ccsc4ncn3 GK02939 c1c(cc(cc1C(F)(F)F)NS(=O)(=O)c2cc(c(cc2F)Br)F)C(F)(F)F HAN00018 Cc1ccc(cc1)NS(=O)(=O)c2cc(c(cc2F)Br)F HAN00020 Cc1cc(c(c(c1)S(=O)(=O)c2ccccc2)[N+](=O)[O-])C HAN00080 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c4ccsc4ncn3 GK02942 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C(\C)/c3ccc(c(c3)CN4CCOCC4)OC CD02483 Cc1c(c(on1)C)S(=O)(=O)/N=C/N(C)C CD10624 CC(=O)Nc1ccc(cc1)C(=O)CCC#N EN00063 c1ccc(cc1)C2CC(=O)c3cc(ccc3O2)O BTB13942 COc1ccc(cc1)C(=C(SC)SC)C#N EN00074 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)c3ccc(cc3)F CD08697 c1cc(cc(c1)S(=O)(=O)NCc2ccc(cc2)C(F)(F)F)C(F)(F)F CD10742 Cc1ccc(cc1)C(=O)N2CCN(CC2)Sc3c4ccsc4ncn3 GK02898 CSc1cc(nc(c1)c2ccncc2)c3ccc(cc3)Cl EN00244 CCC(COC(=O)C)Nc1[nH]c2c(n1)n(c(=O)n(c2=O)C)C BTB13976 c1ccc(cc1)Sc2nc3cc(ccc3s2)Cl EN00198 c1ccc2c(c1)cccc2Sc3c4ccsc4ncn3 GK02907 CCC(C)Nc1c2ccsc2ncn1 GK02908 COCCCNC(=O)CC#N CD02532 Cc1c(c(n(n1)C)C)Cc2c(cccc2Cl)F CD07524 Cc1c(c(n(n1)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)Cc3c(cccc3Cl)F CD07529 CC(=O)c1ccccc1OCc2cccc(c2)C#N CD02531 Cc1c(c(n(n1)S(=O)(=O)c2ccccc2)C)Cc3c(cccc3Cl)F CD07532 Cc1c(c(n(n1)C(=O)c2c(cccc2Cl)Cl)C)Cc3c(cccc3Cl)F CD07537 c1cc(c(cc1/C=N/NC(=S)NC2CC3CC2C4C3CC=C4)Cl)Cl CD02541 CSc1cc(nc(n1)c2ccc(cc2)Cl)c3cccs3 EN00124 CCOc1cc(nc(n1)S)c2ccccc2 EN00127 Cc1c(c(no1)c2ccccc2Cl)C(=O)c3ccccc3 CD08660 Cc1c(nnn1c2ccc(c(c2)Cl)F)C(=O)/C=C/N(C)C CD09941 Cc1c(c(no1)c2ccccc2)C(=O)c3ccccc3 CD08663 c1cc(ccc1SCc2cc(cc(c2)Br)Br)Cl CD08519 CC(C)(C)c1cc(n(n1)C(=O)c2ccc(cc2)Cl)SC CD10659 c1ccc(cc1)NC(=O)OCc2cccc(c2F)COC(=O)Nc3ccccc3 CD10668 c1cc(c(c(c1)N2CCOCC2)C#N)C#N CD10671 CC(=O)NCCSCc1c(cccc1Cl)F CD07753 c1cc(ccc1S(=O)(=O)NC(=N)N2CCOCC2)Cl CD07763 CCOC(=O)C(=C1C2CC3CC(C2)CC1C3)C#N DSHS01035 CCC1(C(=C)S/C(=N\c2ccc(cc2)C(=O)OCC)/N1)CC DSHS01044 c1cc(ccc1C(=O)C2CCNCC2)F.Cl CD09967 c1ccc(cc1)NC(=O)NCCc2ccc(cc2)Cl CD08665 CNC(=O)NCCc1ccc(cc1)Cl CD08666 c1cc(oc1)C(=O)NCCc2ccc(cc2)Cl CD08668 c1c(cc(cc1C(F)(F)F)S(=O)(=O)Nc2cc(c(cc2Cl)Cl)Cl)C(F)(F)F HAN00069 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCSCC3 CD07733 Cc1c(c([nH]n1)N/N=C/c2ccccc2)C(=O)O BTB13900 c1cc2cccc(c2c(c1)CO)Sc3cccc4c3c(ccc4)C(=O)O BTB11483 c1cc(ccc1C(=O)CN)[N+](=O)[O-].Cl BTB13907 c1ccc(cc1)C(=O)N2CCC(=O)CC2 BTB13913 c1cc(c(c(c1)Cl)CN(Cc2c(cccc2Cl)F)O)F CD07550 c1ccn(c1)CC2CCCN(C2)C(=O)Nc3ccc(cc3)Cl CD09943 CCC(CO)Nc1[nH]c2c(n1)n(c(=O)n(c2=O)C)C BTB13975 c1cc(ccc1NC(=S)NNC(=O)CC#N)F CD02494 c1cc(c(cc1NC(=S)NNC(=S)NC2CC3CC2C=C3)Cl)Br CD02506 CSc1cccc(c1)NC(=S)NNC(=S)NC2CC3CC2C=C3 CD02507 Cc1c(c(c(c(c1C)C)COc2ccccc2C(=O)C)C)C CD02516 CC1CN(CC(O1)C)C(=N)NS(=O)(=O)c2ccc(c(c2)Cl)Cl CD07817 CC(CNc1[nH]c2c(n1)n(c(=O)n(c2=O)C)C)O BTB13978 Cc1c(c(c(c(c1C)C)C(=O)CCc2cccc(c2)NC(=O)CCC(=O)O)C)C CD02517 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccccc2O CD02522 CNC(=O)c1ccccc1Sc2cccc3c2c(ccc3)C(=O)NC BTB11484 CNC(=O)c1ccccc1Sc2cccc3c2cccc3 BTB11486 Cc1c(nnn1c2ccc(c(c2)Cl)F)C(=O)C CD09931 c1c(cc(cc1Cl)Cl)CNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10788 c1cc(c(cc1S(=O)(=O)NCc2cc(cc(c2)Cl)Cl)Cl)Cl CD10792 c1cc(ccc1S(=O)(=O)CC(Cn2ccc(n2)C(F)(F)F)O)Cl HAN00292 CCCCNC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl CD02860 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10809 Cc1cccc(c1)NC(=S)N2CC(OC(C2)C)C DSHS01248 c1cc(c(c(c1)Cl)CO/N=C/c2cccs2)Cl CD02525 c1cc-2c(cc1Cl)C(=O)c3c2ccc(c3)Cl BTB13916 c1cc(ccc1NC(=S)NC2CC3CC2C4C3CC=C4)F CD02547 COCCCn1cnn2c(c1=O)nc3ccccc3c2=O CD07615 CS/C(=N/C#N)/NCC#C CD10661 C#Cc1cccc(c1)NC(=O)C(Cl)Cl CD07875 CN(C1CC2CC1C=C2)C(=O)C(Cl)Cl CD09869 c1cc2c(cc1Cl)-c3c(c(nc4c3c(nc(c4C#N)N)O2)N)C#N FM00104 CCOC(=O)c1cnn(c1c2ccccc2)c3c(cc(cc3Cl)Cl)Cl CD10186 c1cc(c(c(c1)Cl)CSC[C@@H](C(=O)O)N)F CD08351 CSCC(CSC)OC(=O)Nc1ccc(cc1)Cl CD08861 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC3=C(CCC3=O)C CD10187 CS/C(=N\C#N)/N1CCN(CC1)c2ccc(cn2)[N+](=O)[O-] CD10028 CS/C(=N\C#N)/N1CCN(CC1)c2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD10029 Cc1c(c(n(n1)C)C)NN=C(C(=O)C)C(=O)C CD10037 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cccc(c3)C#C CD07863 C#Cc1cccc(c1)NS(=O)(=O)c2ccc(c(c2)Cl)Cl CD07869 CN(C)/C=N/n1c(=O)c2ccccc2nc1C(=O)NCCCOC CD07616 c1cc(c(c(c1)COC(=O)Nc2ccc(cc2)Cl)F)COC(=O)Nc3ccc(cc3)Cl CD10679 Cc1c(c(n(n1)C)NNC(=O)c2ccccc2Cl)[N+](=O)[O-] EN00283 Cc1c(c(n(n1)C)NNC(=O)C(C)(C)C)[N+](=O)[O-] EN00288 Cc1ccc(n1c2ccsc2COC(=O)c3c(onc3c4c(cccc4Cl)Cl)C)C CD08866 CC(=O)OCCNc1[nH]c2c(n1)n(c(=O)n(c2=O)C)C BTB13980 CN(C)c1cccc(c1C#N)N(C)C CD08880 c1ccc(cc1)C(c2ccc(cc2)F)/C(=N/O)/NCCc3ccncc3 CD08896 c1ccnc(c1)SCc2nc(no2)c3ccc(cc3)Cl CD02835 c1cc(c(cc1NC(=S)NNC(=O)CC#N)Cl)Cl CD02841 CC(=O)Nc1ccsc1C(=O)OC CD08704 Cc1c(c(no1)c2ccccc2)C(=O)NCc3ccc(cc3)C(F)(F)F CD10741 CSc1nc(n(n1)C(=N)SC)N CD09978 CC(=O)Nc1ccc-2c(c1)Cc3c2nc(c(c3c4ccco4)C#N)OC FM00038 c1cc(ccc1C(=O)CC(=O)CCCO)F CD10820 c1cc(oc1)C(=O)NOC(=O)c2ccc(cc2)Cl CD02797 c1cc(ccc1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl CD02807 c1cc(ccc1c2nc(on2)CSC3=NCCN3)Cl.Cl CD02830 Cc1cc(c2c(c1C#N)CC(C2=O)(C)C)C CD08699 COC(=O)c1c(ccs1)NC(=O)C(Cl)(Cl)Cl CD08700 c1cc(c(cc1Cl)Cl)C(=O)NCc2cc(cc(c2)Cl)Cl CD10793 Cc1cc(=O)oc2c1ccc(c2)Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD08032 c1cc(ccc1C(=N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl CD07987 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NS(=O)(=O)C CD10066 CCOC(=O)c1cnc(nc1C)N CD10070 c1ccc(cc1)NC(=O)NCCC2CC2(Cl)Cl CD10779 c1cc(c(cc1NS(=O)(=O)c2cc(c(s2)Br)Br)Cl)F CD08622 COC(=O)c1c(ccs1)NC(=O)c2ccccc2F CD08630 C/C(=N\OC(=O)c1c(c2ccccc2s1)Cl)/c3ccc(c(c3)CN4CCCC4)OC CD02706 Cn1c(nnc1S)CC#N CD02565 Cc1c(c(c(c(c1C)C)C(=O)c2c(onc2c3c(cccc3Cl)F)C)C)C CD08686 CC(C)(C)C(=O)CSc1nc(c(s1)C(=O)C(C)(C)C)N CD08696 c1ccnc(c1)CCNc2ccc(cc2[N+](=O)[O-])C#N CD08013 c1cc(c(cc1F)F)CNS(=O)(=O)c2ccc(c(c2)Cl)Cl CD10760 c1cc(c(cc1F)F)CNC(=O)c2ccc(cc2Cl)Cl CD10770 c1ccc(c(c1)NC(=S)NCc2ccncc2)Cl DSHS01213 c1cc(cc(c1)NC(=S)NCc2ccncc2)C(F)(F)F DSHS01214 CSc1cc(nc(c1)c2ccc(cc2)Cl)c3ccc(cc3)Cl EN00242 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NS(=O)(=O)c3cc(sc3Cl)Cl CD10054 CN(/C=C(/S(=O)(=O)/C(=C/N(C)C)/C#N)\C#N)C CD09924 CCOC(=O)Cn1c2c(nc1NCc3ccccc3)n(c(=O)n(c2=O)C)C BTB13958 CCOC(=O)CCCn1c2c(nc1NCc3ccccc3)n(c(=O)n(c2=O)C)C BTB13959 c1cc(ccc1C(=O)NCc2ccc(cc2F)F)F CD10762 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C#N CD08015 c1cc(c(nc1)N2CCC(CC2)C(=O)N)[N+](=O)[O-] CD10246 Cc1ccc(cc1)NC(=S)NCc2ccncc2 DSHS01216 Cc1ccc(c(n1)O)C(=S)N FM00043 Cc1ccccc1NC(=S)N2CC(OC(C2)C)C DSHS01247 c1cc(c(c(c1)Cl)/C=N/NC(=O)C(=O)Nc2ccc(cc2)F)Cl CD02664 C1CCNC(=O)C(C1)N/C=N/O CD10120 Cc1cc(c(c(c1)Br)NC(=O)c2ccccc2Cl)Br CD07900 Cc1cc(c(c(c1)Br)NC(=O)c2ccc(cc2)Cl)Br CD07901 CN(c1ccc(cc1[N+](=O)[O-])Cl)NC2c3ccccc3C(=O)O2 CD07916 CC(=O)c1ccc(c(c1)COc2ccc(cc2Cl)Cl)OC CD02689 C/C(=N\O)/c1ccc(c(c1)CN2CCCC2)OC CD02703 COCCCNC(=S)NNC(=S)Nc1ccc(cc1)OC CD02869 COCCCNC(=S)NNC(=S)Nc1cccc(c1)Cl CD02870 c1c(cc(c(c1[N+](=O)[O-])N2CCC(CC2)C(=O)N)[N+](=O)[O-])C(F)(F)F CD10247 CC(=O)c1ccc(c(c1)CSc2nc(sn2)SCc3cc(ccc3OC)C(=O)C)OC CD08345 COC(CNc1ccc(c(c1C#N)NCC(OC)OC)[N+](=O)[O-])OC CD10009 c1c(cc(c(c1[N+](=O)[O-])N2CCNCC2)[N+](=O)[O-])C(F)(F)F CD10027 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N3CCSCC3 CD07848 CCc1c(c(sc1C#N)C(=O)N)CC CD09928 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)OCc3c(cccc3Cl)F CD07955 COCCCNC1=C(C(=O)NC(S1)c2ccc(c(c2)OC)O)C#N CD02632 CN(C)/C=C/C(=O)c1ccc(o1)c2ccc(cc2F)F CD10815 CN(C)/C=N/C(=O)c1ccc(cc1)S(=O)(=O)N2CCOCC2 CD10819 CC(C)(NC(=S)NN)/N=N/c1ccccc1 CD10782 CNC(=O)c1cccc2c1c(ccc2)Sc3ccccc3C(=O)O BTB11473 CNC(=O)c1cccc2c1c(ccc2)Sc3ccccc3C(=O)OC BTB11474 c1cc(c(c(c1)C#N)Sc2ccc(cc2)Cl)C#N CD10727 COc1c(c(c2c(n1)-c3ccccc3C2)c4cccs4)C#N FM00011 CN(C1CC2CC1C=C2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD09908 c1cc(c(c(c1)Cl)CSc2c(c(sn2)SCc3c(cccc3Cl)Cl)C#N)Cl CD02652 c1ccn(c1)c2ccsc2C(=O)NNC(=O)C(Cl)Cl CD08795 c1ccc(cc1)OC(=O)c2c(cccc2Cl)Cl CD08804 c1ccc(cc1)C(=O)NCc2ccc(o2)c3ccc(cc3F)F CD10776 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)c3ccccc3 CD08659 CC(C)(C)SCCN/C(=N\S(=O)(=O)c1ccccc1)/SC CD08662 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)OCc3c(ccs3)n4cccc4 CD08824 c1cc(ccc1NC(=O)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)F CD02662 c1cc(ccc1CNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD10737 Cc1c(c(c(c(c1C)C)C(=O)C2CCN(CC2)C(=O)c3ccc(o3)[N+](=O)[O-])C)C CD10740 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])C(=O)N(Cc3ccc4c(c3)OCO4)c5ccc(cc5)F DSHS00942 Cc1cc(cc(n1)NNC(=O)NC(=O)c2ccccc2Cl)C(F)(F)F CD10714 Cc1cc(cc(c1Cl)C)OCc2cc(ccc2OC)C(=O)C CD02692 CN(C)/C=N/c1ccccc1C2C=NNC2=O CD10082 Cc1cc(c(c(c1)Br)NC(=O)C(Cl)(Cl)Cl)Br CD07894 Cc1c(cnc(n1)N)C(=O)C CD10099 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F)C)C DSHS01002 CC(=O)C(=NNc1cc(c(cc1F)Br)F)C(=O)C HAN00112 Cc1c(cnn1c2ccc(cc2)C#N)C(=O)C CD10715 c1c(c(cc(c1Br)F)Br)F HAN00002 CC(C)c1ccc(cc1)NC(=S)Nc2cccc(c2)C(F)(F)F DSHS01210 CC(C)c1ccc(cc1)NC(=S)Nc2ccccc2Cl DSHS01212 Cc1c(c(no1)c2ccccc2Cl)C(=O)Oc3ccccc3 CD08780 CC1=C(C(=O)CC1)OC(=O)c2cccs2 CD10189 c1cc(c(cc1C(F)(F)F)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)F HAN00101 C1C2CC3CC1CC4(C2)C3NC(=O)O4 FM00024 CN(C)C(=O)Oc1ccc2c(c1)n3c(ccn3)nn2 EN00263 CCOc1c2c(csc2[nH]c(=O)c1C(=O)C)C GK02943 CCOC(=O)/C(=C/Nc1ccsc1C(=O)OC)/C#N CD08718 COC(=O)c1c(ccs1)NC=C(C#N)C#N CD08719 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCC(=O)O HAN00008 c1c(cc(cc1Cl)Cl)CNC(=O)c2cc(cc(c2)Cl)Cl CD10789 CC1(OC(=O)C(=Cc2ccc(cc2)C#N)C(=O)O1)C CD08787 c1ccn(c1)c2ccsc2C(=O)NNS(=O)(=O)c3ccc(c(c3)Cl)Cl CD08799 c1ccc2c(c1)C/C(=C\O)/C2=O FM00016 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)/C=C/2\Cc3ccccc3C2=O FM00017 C1C2CC3CC1CC(C2)(C3)OC(=O)NN FM00019 c1cc(ccc1S(=O)(=O)N2CCSCC2)Cl CD07851 c1ccc2c(c1)C/C(=C\c3cc(cs3)Br)/C2=O FM00031 C#Cc1cccc(c1)NC(=O)c2c(cccc2Cl)Cl CD07866 COC(=O)c1c(ccs1)n2cccc2 CD08721 c1cc(ccc1C2CC(=O)CC(=O)C2)Cl CD09847 Cc1c(c(no1)c2c(cccc2Cl)F)C(c3ccc(cc3)F)O CD08736 C/C(=N\NC(=S)N)/c1ccccc1O CD02640 c1cc(ccc1NC(=O)OC2CCSC2)Cl CD10640 Cc1c(c(no1)c2ccccc2)C(=O)NCc3cc(cc(c3)Cl)Cl CD10795 CN(c1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])/N=C/c2cccc(c2O)OC CD07904 Cc1c(nnn1c2ccc(cc2C#N)Cl)C(=O)/C=C/N(C)C CD10658 c1c(cc(cc1C(F)(F)F)S(=O)(=O)Oc2cc(cc(c2)Cl)Cl)C(F)(F)F CD08079 c1cc(ccc1S(=O)(=O)Oc2ccc(c(c2)Cl)Cl)Cl CD08084 Cc1c(c(c(c(c1C)C)CSCc2n[nH]c(=S)n2c3ccc(cc3)F)C)C DSHS00983 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)Nc2cccc(c2)SC)C)C DSHS00984 c1cc(cc(c1)Br)OS(=O)(=O)CS(=O)(=O)Oc2cccc(c2)Br CD10872 c1cc(ccc1OS(=O)(=O)CS(=O)(=O)Oc2ccc(cc2)I)I CD10882 CS(=O)(=O)CS(=O)(=O)Oc1ccc(cc1)Cl CD10896 CC(C)(C)c1cc([nH]n1)SC CD10657 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCCO)Cc3ccccc3 BTB13966 c1ccc(cc1)C(=O)c2ccccc2NC(=O)c3ccc(cc3)Cl CD02490 COCC(=O)Nc1c(ccs1)C(=O)OC GK02888 CN(CC(OC)OC)c1c2ccsc2ncn1 GK02892 CS(=O)(=O)CS(=O)(=O)Oc1cccc(c1)C(F)(F)F CD10860 CC(=O)c1ccc(o1)c2cc(cc(c2)Cl)Cl CD10867 COc1ccc(cc1)OS(=O)(=O)CS(=O)(=O)Oc2ccc(cc2)OC CD10016 c1ccnc(c1)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl CD02854 CC(C)(C)c1csc(n1)NS(=O)(=O)c2ccc(cc2)Cl CD08354 CC(C)(C)c1csc(n1)NC(=O)c2ccc(cc2Cl)Cl CD08368 c1csc2c1c(ncn2)NCCCN3CCOCC3 GK02884 c1cc(c(cc1F)F)NC(=S)N2CCN(CC2)c3c4ccsc4ncn3 GK02947 CC(CNc1[nH]c2c(n1)n(c(=O)n(c2=O)C)C)OC(=O)C BTB13979 C/C(=N\O)/C=C/c1ccccc1 EN00218 c1cc(c(c(c1)Cl)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl EN00228 c1ccc(cc1)NC(=O)Sc2ccccc2Cl EN00232 Cc1c2cc(sc2n(n1)C)C(=O)OC EN00097 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)OCc3c(cccc3Cl)F CD07967 c1ccc(cc1)C(=O)NC(=S)N2CCSCC2 CD07976 c1ccc2c(c1)cccc2NC(=S)N3CCOCC3 DSHS01237 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCOCC3 DSHS01238 CS/C(=N\C#N)/N1CCC(CC1)C(=O)N CD10252 c1cc(c(c(c1)Cl)CSc2nnc(s2)N)Cl CD10265 CC(=O)c1ccc(cc1)OC(=O)c2c(cccc2Cl)Cl CD08803 c1ccc(cc1)NC(=O)NC2CCCCNC2=O CD10134 CC(C)NC(=O)NC1CCCCNC1=O CD10135 Cn1c(cc(n1)C(F)(F)F)OC(=O)c2cccs2 EN00093 COc1ccc(cc1OC)Cc2n[nH]c(=O)o2 EN00096 C/C(=N\OC(=O)c1cccs1)/C=C/c2ccccc2 EN00222 c1cc(c(c(c1)Cl)/C=C/c2ccnc(n2)N)Cl CD09854 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCC(F)(F)F CD08535 CCOc1cc(nc(n1)N)c2ccccc2 EN00120 c1ccc(cc1)NC(=O)Sc2cc(cc(c2)C(F)(F)F)C(F)(F)F EN00236 CCOC(=O)c1ccc(cc1)NC(=S)NNC(=O)CSCc2c(c(c(c(c2C)C)C)C)C DSHS01003 CN(c1ccc(cn1)[N+](=O)[O-])NC2c3ccccc3C(=O)O2 CD07917 CC1CN(CC(O1)C)C(=S)Nc2cccc(c2)C(F)(F)F DSHS01245 Cc1cccc(c1NC(=S)N2CC(OC(C2)C)C)C DSHS01246 c1cc(c(cc1OS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl)Cl CD08088 CC(C)Cn1c(=O)c2ccccc2nc1SCC(=O)c3ccc(cc3)Br BTB13995 c1ccc(cc1)C(=O)Nc2cc(cc(c2)NC(=O)c3ccccc3)C(F)(F)F CD10953 Cc1cc(n(n1)C2=NCCN2)C.Br CD08547 c1cc(c(cc1Cl)Cl)/C=N/OCc2cc(cc3c2OCOC3)F CD08552 CN(C1CC2CC1C=C2)C(=O)c3cccs3 CD09866 Cc1c2cc(sc2n(n1)C)C(=O)O CC22901 c1cc(cc(c1)NS(=O)(=O)c2c(c(cc(c2Br)F)Br)F)C(F)(F)F HAN00028 c1ccc(cc1)OC(=O)NN DSHS01027 c1ccc(cc1)OC(=O)NNC(=O)c2ccc(cc2)Cl DSHS01032 c1ccc(cc1)CC(C(=O)O)NC(=O)c2ccc(cc2)C(=O)NC(Cc3ccccc3)C(=O)O HAN00044 c1c(cc(cc1Cl)Cl)CNC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10785 c1cc(ccc1C(=O)NCc2ccc(o2)c3ccc(cc3F)F)Cl CD10935 c1cc(c(c(c1)C#N)Oc2ccc(cc2)NC(=O)c3ccc(cc3Cl)Cl)C#N CD10973 c1cc(ccc1c2nc(on2)CSC3=NCC4CCCC4N3)Cl.Cl CD02833 CCOC(=O)c1ccc(cc1)OS(=O)(=O)CS(=O)(=O)Oc2ccc(cc2)C(=O)OCC CD10020 c1ccc(cc1)/C=C/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl CD02855 CC(C)(C)C(=O)NNC(=O)C(C)(C)C CD07623 CN(C)/C=C/C(=O)c1cc(ccc1O)F CD07629 CN(C)/C=C/C(=O)c1cc(cc(c1O)F)F CD07630 c1c(cc(cc1C(F)(F)F)NC(=O)C(F)(F)F)C(F)(F)F CD02821 CS(=O)(=O)n1c(ccn1)c2ccc(o2)c3ccc(cc3F)F CD10941 c1cc(c(c(c1)Cl)OS(=O)(=O)c2cc(c(s2)Br)Br)Cl CD10332 c1cc(c(c(c1)Cl)C#N)NC2CCCCNC2=O CD10132 c1cc(ccc1NC(=O)NC2CCCCNC2=O)Cl CD10133 COc1ccc(cc1)C2c3ccc4ccccc4c3OC(=C2C#N)N FM00120 CC1=C(C(=O)CC1)OS(=O)(=O)c2cc(sc2Cl)Cl CD10169 CC1=C(C(=O)CC1)OS(=O)(=O)c2ccc(cc2F)F CD10173 c1cc(c(cc1F)F)c2ccc(o2)c3ccnn3C(=O)c4ccc(cc4Cl)Cl CD10928 COC(=O)c1ccsc1N GK02784 c1cc2c(cc1Br)C(C(=C(O2)N)C#N)C(C#N)C#N FM00096 CC(=O)c1ccccc1OC(=O)c2ccc(o2)[N+](=O)[O-] CD08758 CCOC(=O)CCSC1=NC(C(=C(N1)C)C(=O)OCC)c2cccs2 FM00079 CCOC(=O)C1=C(N=C2N(C1c3cccs3)C(=O)C(S2)C)C FM00081 COc1ccc2c(c1)C(C(=C(O2)N)C#N)C(C#N)C#N FM00097 Cc1csc(c1N(S(=O)(=O)c2ccc(cc2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)C(F)(F)F)C(=O)OC GK02782 CN(C)/C=C/C(=O)c1ccc(o1)c2cc(cc(c2)Cl)Cl CD10906 CN(C)/C=C/C(=O)c1ccc(o1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10907 c1cc(c(nc1)NCCNc2nccc(n2)C(F)(F)F)C(F)(F)F HAN00250 c1cnc(nc1C(F)(F)F)NCCNc2c(cc(cn2)C(F)(F)F)Cl HAN00252 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NC(=N)N2CCSCC2)C(F)(F)F CD07957 Cc1c(c(n(n1)C)C)/N=N/c2c(nn(c2C)C)C CD10038 Cc1cc(c2c(c1)CC(/C(=N/NC(=O)CC#N)/C2=O)(C)C)C CD02788 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccccc3 CD08774 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CNC(=O)c2cc(cc(c2)Cl)Cl CD10781 Cc1c(c(on1)C)C(=O)Sc2nccc(n2)C(F)(F)F HAN00415 c1ccc(c(c1)NC(=O)C(=O)NCc2cccnc2)Oc3ccc(cc3Cl)Cl CD10335 C1CN=C(N1)SCC2CC2(Cl)Cl.Br CD10343 c1cc(sc1)C(=O)O/N=C(/CN2CCSCC2)\N CD08365 c1ccc(c(c1)C(=O)O/N=C(/CN2CCSCC2)\N)F CD08371 c1ccc(cc1)NC(=O)NC(=O)C2CCN(CC2)c3c(cccn3)[N+](=O)[O-] CD10286 c1cc(c(nc1)N2CCC(CC2)C(=O)NC(=O)Nc3ccc(c(c3Cl)Cl)Cl)[N+](=O)[O-] CD10288 c1cc(ccc1NC(=O)NCc2ccc(o2)c3ccc(cc3F)F)Cl CD10919 c1cc(c(cc1C#N)[N+](=O)[O-])N2CCOCC2 CD08007 c1cc(ccc1CNC(=O)c2ccc(cc2Cl)Cl)C(F)(F)F CD10748 Cc1c(c(n(n1)C)C)NC(=O)/C(=C\N(C)C)/C#N CD10005 c1ccc(cc1)S(=O)(=O)Nc2cc(cc(c2)NS(=O)(=O)c3ccccc3)C(F)(F)F CD10921 COc1ccc(cc1OC)CCNC(=O)CCC(=O)O CD02793 Cc1c(c(no1)c2ccccc2)C(=O)OC CD02796 c1cc(ccc1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F CD02809 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)Sc3nccc(n3)C(F)(F)F HAN00280 CSCC(CSC)OC(=O)Nc1ccccc1 CD08859 c1cc2c(cc1Cl)C(C(=C(O2)N)C#N)C(C#N)C#N FM00094 Cc1c(c(n(n1)C)NNC(=O)c2ccccc2C(=O)O)[N+](=O)[O-] GK02699 c1ccc(cc1)C2(C(C3c4cc(ccc4Oc5c3c(c(c(n5)N)C#N)N2)Cl)C#N)O FM00099 CC(=O)c1ccc(cc1)OS(=O)(=O)CS(=O)(=O)Oc2ccc(cc2)C(=O)C CD10370 c1cc(c(c(c1)Cl)CSc2nc(sn2)SCc3c(cccc3Cl)F)F CD08313 c1ccc2c(c1)c(n[nH]2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl CD08164 c1cc(ccc1C(=O)O/N=C/c2ccc(o2)c3ccc(cc3F)F)Cl CD10913 CCOC(=O)c1ccc(cc1)NC(=S)N2CCN3C2(c4ccccc4C3=O)c5ccccc5 DSHS01084 c1ccc-2c(c1)CCc3c2nc(s3)N.Br FM00124 Cc1ccc(n1c2ccsc2C(=O)NNC(=O)C(Cl)Cl)C CD08906 c1cc(c(cc1F)F)c2ccc(o2)C#N CD10918 c1cnccc1N2C(=O)C3C4CC(C3C2=O)C=C4 DSHS01091 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCC3CC3(Cl)Cl CD10993 Cc1c(sc(n1)NC(=N)N)Br CD10996 CCOC(=O)c1cnn(c1C)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10236 c1cc(ccc1S(=O)(=O)NC(=N)N2CCSCC2)Cl CD07958 c1ccc2c(c1)C(=O)N(C2=O)N3C(=O)C4C5CC(C4C3=O)C=C5 DSHS01087 CC1=C(C(=O)OC1c2c(cccc2Cl)F)O CD08996 c1ccc(c(c1)C(=O)Oc2ccc(c(c2)Cl)Cl)F CD08111 CC(C)(C)C(=O)NCCC1CC1(Cl)Cl CD10987 c1ccn(c1)c2c(cccc2C#N)C#N CD10988 c1cc(ccc1S(=O)(=O)NCCC2CC2(Cl)Cl)Cl CD10990 CC(C)N(CCC#N)C(=S)Nc1ccc(cc1)S(=O)(=O)N2CCCCC2 DSHS01280 c1ccc(cc1)CN(CCC#N)C(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 DSHS01285 CC1(C(=C)S/C(=N\c2cc(c(cc2Cl)Cl)Cl)/N1)C DSHS01074 Cc1ccc(cc1)NC(=S)N(CCC#N)C2CCCCC2 DSHS01205 c1cc(ccc1CCNC(=O)Nc2ccc(cc2)Cl)Cl CD08664 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)C CD10055 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD10056 Cc1c(cnn1c2cccc(c2)Cl)C(=O)C CD10063 c1ccc(c(c1)C(=O)NCCc2ccc(cc2)Cl)F CD08670 c1cc(c(cc1OC(=O)c2ccc(cc2Cl)Cl)Cl)Cl CD08114 Cc1c(nnn1c2ccc(c(c2)Cl)F)c3ccccc3 CD08117 c1cnc(nc1C(F)(F)F)S HAN00409 Cc1cc(n(n1)C2=NCCN2S(=O)(=O)C)C CD10329 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3nc(ns3)c4ccccc4 HAN00380 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)C(=O)CSCC(=O)O HAN00384 CC(C)(C)c1c(sc(n1)N)Br.Br CD08357 Cc1ccc(n1c2ccsc2C(=O)NNC(=O)/C=C/c3ccccc3)C CD08915 c1cc(c(cc1F)F)c2ccc(o2)c3ccnn3S(=O)(=O)c4ccc(cc4F)F CD10929 COc1ccc(cc1)NC(=S)N(CCC#N)C2CCCCC2 DSHS01200 CCOC(=O)c1ccc(cc1)NC(=S)N(CCC#N)C2CCCCC2 DSHS01202 COc1cc(cc(c1OC)OC)/C=N/NC(=O)C(=O)Nc2ccc(cc2)F CD02665 CC(C)(C)c1cc2n(n1)C3=NCCN3C=N2 CD10071 Cc1ccnn1c2ccc(cc2)Cl CD10904 c1cc(cnc1)OS(=O)(=O)c2cc(c(s2)Br)Br CD10333 c1ccc(cc1)OS(=O)(=O)c2cc(c(s2)Br)Br CD10334 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/CN3CCSCC3)\N CD08304 COCCCNC(=S)NNC(=S)NCCCOC CD02867 COCCCNC(=S)NNC(=S)Nc1ccccc1 CD02868 Cc1csc2c1ncnc2N3CCN(CC3)C(=S)NCC4CC4 GK02691 Cc1csc2c1c(ncn2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl GK02709 c1cc(nc(c1)N2C(=O)C3CC=CCC3C2=O)N4C(=O)C5CC=CCC5C4=O DSHS01099 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C#N)Cl CD08017 Cc1csc2c1c(ncn2)N3CCN(CC3)S(=O)(=O)c4cccc(c4)C(F)(F)F GK02711 Cc1csc2c1c(ncn2)N3CCN(CC3)C(=O)Nc4ccc(cc4)OC(F)(F)F GK02713 COc1ccc(cc1)NC(=S)NCc2ccncc2 DSHS01217 C/C(=N\OC(=O)c1ccc(cc1)[N+](=O)[O-])/c2ccc(c(c2)CN3CCOCC3)OC CD02686 CCOC(=O)/C(=C/Nc1ccn[nH]1)/C#N GK02747 Cc1csc(c1NC(=O)/C=C\C(=O)O)C(=O)OC GK02749 COc1c(c(c2c(n1)-c3ccccc3C2)c4cc(cs4)Br)C#N FM00030 c1ccc(cc1)/C=C/C(=O)NNC(=O)c2c(ccs2)n3cccc3 CD08777 c1c(c(cc(c1F)Br)F)N2C(=O)C=CC2=O HAN00116 c1cc(ccc1SC2CC(=O)N(C2=O)c3cc(c(cc3F)Br)F)Cl HAN00117 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl GK02799 Cc1c(noc1N2C(=O)C3C4CC(C3C2=O)C=C4)C DSHS01088 c1cc(ccc1Cc2ccc(cc2)N3C(=O)C4C5CC(C4C3=O)C=C5)N6C(=O)C7C8CC(C7C6=O)C=C8 DSHS01096 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F GK02800 CS/C(=N\C#N)/NC1CCCCNC1=O CD10113 C1CCNC(=O)C(C1)Nc2[nH]nc(n2)N CD10114 c1cc(ccc1SCC(=N)NS(=O)(=O)c2ccc(cc2)Cl)Cl CD08123 C=CCNC(=S)N(CCC#N)C1CCCCC1 DSHS01204 c1ccnc(c1)Sc2ccc(cc2C(=O)Nc3ccncc3)[N+](=O)[O-] DSHS00991 c1cc(ccc1c2cc(c(s2)C(=O)N)NC(=O)/C=C\C(=O)O)Cl GK02752 CCC(CO)N1CCCn2c1nc3c2c(=O)n(c(=O)n3C)C BTB13984 CC(C)(CO)N1CCCn2c1nc3c2c(=O)n(c(=O)n3C)C BTB13985 c1ccc2c(c1)C/C(=C\c3cccs3)/C2=O FM00009 COc1c(c(c2c(n1)-c3ccccc3C2)c4ccco4)C#N FM00010 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])OCCOC(=O)c2ccc(cc2Cl)Cl CD08119 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2cc(c(cc2F)Br)F)Cl HAN00125 Cc1c(c(no1)c2ccccc2)C(=O)OCCOc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] CD08120 Cc1c(c(no1)c2ccccc2)C(=O)OCCOc3ccc(cc3[N+](=O)[O-])C(F)(F)F CD08121 c1cc(sc1)C(=O)Nc2ccsc2C(=O)NN GK02722 CCCCNC(=O)N(C)C1CC2CC1C=C2 CD09877 c1ccc2c(c1)CCC2=C(C#N)C#N FM00032 c1ccc-2c(c1)Cc3c2c(c(c(c3c4ccco4)C#N)N)C#N FM00033 c1ccc(cc1)OC(=O)c2cccs2 CD08775 c1cc(oc1)C(=O)Nc2ccc(c(c2Cl)Cl)Cl CD08070 Cc1c(nnn1c2ccc(cc2F)F)c3ccccc3 CD08073 Cc1c(c(n(n1)C)C)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD09897 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Nc2c(nn(c2C)C)C CD09901 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Oc3ccccc3 CD08776 Cc1csc2c1c(ncn2)N3CCN(CC3)C(=O)Nc4ccc(cc4)SC(F)(F)F GK02714 CC(C)(COC(=O)Nc1ccc(cc1)Cl)n2cccc2 CD09068 CC(C)CC1C(=O)NC(=O)N1 FM00152 Cc1cc(=O)oc2c1ccc(c2)OCC#C CD08041 Cn1cccc1C(=O)/C(=C/c2cccs2)/C#N CD10897 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCSCC3 CD07930 c1cc(oc1)C(=O)N2CCSCC2 CD07933 c1ccc2c(c1)C(OC2=O)Nc3ccc(c(c3)Cl)Cl CD07936 Cc1c(c(no1)c2ccccc2)C(=O)Oc3ccccc3 CD08781 c1cc(c(c(c1)I)C#N)F CD07951 c1ccc(c(c1)C(=O)OCc2c(cccc2Cl)F)Cl CD07953 c1cc(c(c(c1)Cl)COC(=O)c2ccc(cc2)Cl)F CD07954 Cn1cccc1C2=C(C(C(=C(O2)N)C#N)c3c(cccc3Cl)Cl)C#N CD10905 CS(=O)(=O)Nc1cc(cc(c1)NS(=O)(=O)C)C(F)(F)F CD10909 Cc1c2c(n(n1)C)SC(=NS2(=O)=O)N3CCOCC3 CD10431 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2cc(c(cc2F)Br)F)F HAN00123 Cc1ccc(nc1)N2C(=O)C3C4CC(C3C2=O)C=C4 DSHS01092 c1cc(nc(c1)N2C(=O)C3C4CC(C3C2=O)C=C4)N5C(=O)C6C7CC(C6C5=O)C=C7 DSHS01093 c1ccc(c(c1)NC(=S)N(CCC#N)C2CCCCC2)Cl DSHS01201 Cc1c(nnn1c2cccc(c2)C#C)c3ccccc3 CD08057 c1cc(cc(c1)NC(=S)N(CCC#N)C2CCCCC2)C(F)(F)F DSHS01203 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(c(c3Cl)Cl)Cl CD08068 Cn1cccc1C(=O)/C(=C/c2ccc(cc2)C#N)/C#N CD10899 c1cc(c(cc1NC(=O)n2ccc(n2)C(F)(F)F)Cl)Cl HAN00212 CS/C(=N\C#N)/N1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F CD10021 c1cc(oc1c2ccn[nH]2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD10910 Cc1cccc(c1)NC(=S)N2CCOCC2 DSHS01232 CC(=N)NCCc1ccncc1.I CD08170 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCCOc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] CD08093 c1cc(c(c(c1)Cl)C#N)N2CCC(CC2)C(=O)N CD10245 c1cn[nH]c1c2ccsc2 CD10255 c1cc(c(c(c1)Cl)C#N)N2CCC(CC2)C(=O)N/C=N/O CD10257 CCCCNC(=O)NS(=O)(=O)c1cc(sc1Cl)Cl CD10339 COc1c(c(c2c(n1)-c3ccccc3C2)c4ccc[nH]4)C#N FM00013 c1ccc(c(c1)C(=O)Nc2ccc(c(c2Cl)Cl)Cl)Cl CD08066 COCCCNC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl CD02744 COCCCNC(=S)N/N=C/c1cc(ccc1O)Br CD02745 c1cc(sc1)C(=O)n2ccc(n2)C(F)(F)F HAN00209 c1cc(ncc1[N+](=O)[O-])OCCO CD08075 c1cc(c(cc1S(=O)(=O)Oc2cc(cc(c2)Cl)Cl)Cl)Cl CD08078 COCCCNC(=S)N/N=C/C=C/c1ccccc1 CD02746 COCCCNC(=S)N/N=C/c1cccs1 CD02747 COCCCNC(=S)N/N=C/c1ccccn1 CD02750 Cc1cc(no1)NC(=O)C(=O)NC2CCCCNC2=O CD10321 Cc1ccc(cc1[N+](=O)[O-])NC(=S)N2CCN(CC2)c3c4c(csc4ncn3)C GK02717 Cc1csc2c1c(ncn2)N3CCN(CC3)C(=S)NCC4CC4 GK02721 c1ccc2c(c1)C/C(=C\c3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)/C2=O FM00002 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCNCC3 GK02727 Cc1csc(c1NC(=O)/C=C/c2ccccc2)C(=O)OC GK02783 Cc1c(c(no1)c2ccccc2)C(c3ccc(cc3)F)O CD08748 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NC(=O)c3cccs3 CD10143 c1cc(ccc1NC(=O)O/N=C/2\CCSC2)Cl CD10146 CC1=C(C(=O)CC1)OS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10175 Cc1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C(=O)N(Cc3ccc4c(c3)OCO4)c5ccc(cc5)F)C(C)(C)C DSHS00943 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)N(Cc3ccc4c(c3)OCO4)c5ccc(cc5)F DSHS00944 CCOC(=O)c1cnc(nc1C)Nc2nc(cs2)C(C)(C)C CD10188 CCCc1c(cnn1c2c(cc(cc2Cl)Cl)Cl)C(=O)OCC CD10191 Cc1csc(c1NS(=O)(=O)c2ccc(cc2)F)C(=O)OC GK02779 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)C(=O)Nc4ccc(cc4)OC(F)(F)F HAN00373 c1cc(c(c(c1)Cl)C#N)N2CCC(CC2)C(=O)NC(=O)Nc3c(cccc3Cl)Cl CD10347 c1csc2c1c(=O)[nH]cn2 GK02796 CC(C)(C)SCCNS(=O)(=O)c1ccc(cc1)Cl CD08210 c1c[nH]c(=O)nc1C(F)(F)F HAN00230 Cc1c(c(c(c(c1C)C)COC(=O)C)C)C CD02844 CSc1cccc(c1)NC(=S)NNC(=O)CC#N CD02846 c1c(cc(cc1C(F)(F)F)NC(=O)/C=C/C(=O)O)C(F)(F)F CD02850 c1cnc(nc1C(F)(F)F)N2CCOCC2 HAN00251 c1cc(ccc1C(=N)NS(=O)(=O)c2ccc(c(c2)Cl)Cl)Cl CD07986 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])OCCO CD08003 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])C#N CD08016 CC(C)(C)NC(=O)N1CCN(CC1)c2nc(ns2)c3ccccc3 HAN00374 CC(=N)NN(C)c1cccc(c1C#N)F.I CD08178 CC(=O)c1ccc(c(c1)CSC(=S)N2CCSCC2)OC CD08192 c1ccc(cc1)C23c4ccccc4C(=O)N2CCN3S(=O)(=O)c5cccc(c5)C(F)(F)F DSHS01055 CN(C)CCCNC(=O)C(=O)Nc1ccccc1Oc2ccc(cc2Cl)Cl CD10322 c1cc(sc1I)I CD08226 Cc1ccc(c(c1F)C)S(=O)(=O)Oc2ccc(cc2)SC CD08229 c1cc(c(c(c1NC(=O)C(Cl)(Cl)Cl)Cl)Cl)Cl CD08072 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCc3c(ccs3)n4cccc4 CD08864 c1ccc(c(c1)C#N)Oc2ccc(cc2Cl)Cl CD08873 C1CSCC1NC=C(C#N)C#N CD10356 c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3c(cccc3C#N)C#N CD11001 CC(C)(CO)NC(=O)c1cccc(c1F)C(=O)NC(C)(C)CO CD11018 c1ccc(c(c1)N)Sc2nccc(n2)C(F)(F)F HAN00278 c1ccc2c(c1)ncc(n2)/C=C/c3ccc(cc3)Cl CD11255 c1ccc2c(c1)ncc(n2)/C=C/c3c(cccc3Cl)Cl CD11256 CCNS(=O)(=O)c1cc(sc1Cl)Cl CD11257 c1cc(ccc1c2nc(on2)CSC(=S)N3CCSCC3)Cl CD08191 c1ccc2c(c1)CC(=NNc3nc(cs3)c4ccc(cc4)Br)C2 FM00236 COc1ccc(cc1/C=N/Nc2nccc(n2)C(F)(F)F)Br HAN00394 c1cc(c(cc1Cl)Cl)/C=N/Nc2nccc(n2)C(F)(F)F HAN00395 c1ccc2c(c1)ccc3c2OC(=C(C3c4cccs4)C#N)N FM00125 CCOC(=O)C(C(F)(F)F)(NCc1ccccn1)NC(=O)c2cccnc2 JFD02226 c1ccc2c(c1)/C(=C\c3ccc(cc3)C(F)(F)F)/C(=O)N2 CD10828 c1cc(cnc1)/C=C/2\C(=O)C3CCN2CC3 FM00111 c1ccc2c(c1)CC(=NNc3nc(cs3)c4ccc(cc4)[N+](=O)[O-])C2 FM00237 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)NCc2ccco2 JFD02229 c1ccc\2c(c1)CCC/C2=N\NC(=S)N FM00217 c1cc(ccc1C(=O)NC2=CC3C(COC3=O)OC2=O)Cl FM00219 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)n2ccc(n2)c3cc(sc3Cl)Cl CD09209 c1ccc(cc1)S(=O)(=O)NCc2ccc(o2)c3ccc(cc3F)F CD10936 c1cc(ccc1CCNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl CD08318 c1cnc(nc1C(F)(F)F)NNC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F HAN00396 c1ccc2c(c1)ccc3c2OC(=C(C3c4ccc(cc4)F)C#N)N FM00127 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)C(=O)Nc4ccc(cc4)SC(F)(F)F HAN00372 Cc1ccc(c(c1F)C)S(=O)(=O)NCCCN(C)C CD08324 Cc1cc(cc(c1F)C)S(=O)(=O)NC(=N)c2cccnc2 CD08328 COc1c(c(c(c(n1)N)C#N)c2ccc3c(c2)OCO3)C#N FM00239 Cc1cc(cc(n1)n2c(nc(n2)SC)N)C(F)(F)F CD10488 COc1ccc(c2c1cccc2)OC CD10471 c1ccc(cc1)NC(=O)c2cccc(c2F)C(=O)Nc3ccccc3 CD10497 c1cc(sc1)C2CCCN2C(=S)Nc3ccc(cc3Cl)Cl CD10485 c1cc(c(c(c1)C(=O)Nc2ccc(cc2)Cl)F)C(=O)Nc3ccc(cc3)Cl CD10494 c1cc(cnc1)CNC(=S)Nc2ccc(c(c2)Cl)Cl DSHS01228 CC(C)(C)SCCNc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD08251 CC(C)(C)SCCNC(=O)c1cccs1 CD08267 c1cc(c(cc1C(F)(F)F)NS(=O)(=O)c2cc(ccc2Cl)C(F)(F)F)F HAN00102 c1cc(cc(c1)NC(=S)NNc2nccc(n2)C(F)(F)F)C(F)(F)F HAN00403 Cc1cccc(c1NC(=S)Nc2ccc(cc2)C(C)C)C DSHS01211 CC1=CC(=O)N(C1=O)c2c(ccs2)C(=O)OC GK02839 c1cc(cc(c1)NC(=S)NCc2cccnc2)C(F)(F)F DSHS01226 CCCCNC(=S)N(CCC#N)C1CCCCC1 DSHS01261 CCCCNC(=O)Nc1ccccc1SCC(Cn2ccc(n2)C(F)(F)F)O HAN00304 COc1cccc(c1)NC(=S)N2CCOCC2 DSHS01230 CC(C)(C)SCCNC(=O)/C=C/c1ccccc1 CD08260 CC(C)(C)SCCNS(=O)(=O)c1ccc(c(c1)Cl)Cl CD08214 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC(CSC)CSC CD08883 CCOC(=O)c1ccc(cc1)NC(=S)NCc2ccncc2 DSHS01220 c1cc(c(c(c1)Cl)CSC(=S)N2CCSCC2)Cl CD08187 c1ccc2c(c1)c3c(c4c2C(C(=C(O4)N)C#N)c5ccc(cc5)C(F)(F)F)OC(=C(C3c6ccc(cc6)C(F)(F)F)C#N)N FM00138 Cc1c(c(n(n1)C)Cl)S(=O)(=O)N CD10384 CCOC(=O)C1=C(Oc2ccccc2C1C(C#N)C#N)N FM00190 CCOC(=O)c1c(c2c(s1)cccc2Cl)N CD09089 Cc1c(c(n(n1)C(=O)c2c(cccc2Cl)Cl)C)Cc3c(cccc3Cl)Cl CD09078 c1cc(c(c(c1)Cl)C#N)N2CCC(CC2)C(=O)NC(=O)Nc3ccc(cc3)Cl CD10348 c1cc(ccc1S(=O)(=O)NC2CCSC2)Cl CD10351 c1cc(c(c(c1)C(=O)Nc2ccc(cc2)F)F)C(=O)Nc3ccc(cc3)F CD10495 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc(cc2F)F)Oc3ccc(cc3Cl)Cl CD08947 c1ccc(c(c1)C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)Oc3ccc(cc3Cl)Cl CD08948 Cc1ccc(c(c1)C)NC(=S)NCc2ccncc2 DSHS01263 c1ccc(cc1)C(CC(=O)c2ccccc2)C(C#N)C#N FM00136 c1ccc2c(c1)ccc3c2OC(=C(C3c4ccc(cc4)C(F)(F)F)C#N)N FM00137 c1cc(c(c(c1)CSC2=[NH+]CCN2)F)CSC3=[NH+]CCN3.[Br-].[Br-] CD09097 Cc1cc(no1)n2nc(nn2)C/C(=N/OC(=O)NC)/C CD09289 Cc1c(c(n(n1)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)Cc3c(cccc3Cl)Cl CD09094 c1ccc(c(c1)/C=N/NC(=O)c2c(nccn2)N)F HAN00439 c1cc(ccc1/C=N/NC(=O)c2c(nccn2)N)C(F)(F)F HAN00441 c1cc(cnc1)CNC(=O)C(=O)NC2CCCCNC2=O CD10481 CC(C)CC1C(=O)N(C(=O)N1)C FM00182 CC(C)(C)C(=O)NCCSC(C)(C)C CD08272 CC(=O)/C(=C/1\NC(=CS1)C(C)(C)C)/C#N CD09172 CC(C)(C)NC(=O)NNc1nccc(n1)C(F)(F)F HAN00400 c1cc(cc(c1)Cl)NC(=O)NNc2nccc(n2)C(F)(F)F HAN00402 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCSC(C)(C)C CD08232 Cc1ccc(c(c1F)C)S(=O)(=O)Oc2cccnc2 CD08234 COC(=O)C1=C(Oc2ccccc2C1C(C#N)C#N)N FM00181 Cc1csc2c1c(ncn2)N3CCN(CC3)C(=S)Nc4ccc(cc4F)F GK02718 Cc1csc2c1c(ncn2)N3CCN(CC3)C(=S)Nc4ccc(cc4)C(F)(F)F GK02719 c1ccc(cc1)NC(=O)c2c3ccccc3c(=O)n(n2)c4ccc(cc4)Cl CD11089 CN(C)/C=C/C(=O)c1ccc(cc1)Cl CD11104 Cc1cc(cc(c1F)C)S(=O)(=O)Nc2ccc(c(c2)Cl)F CD08239 Cc1cc(cc(c1F)C)S(=O)(=O)NN(C)c2cccc(c2C#N)Cl CD08245 Cc1c(c(n(n1)CCC#N)C)Cc2c(cccc2Cl)Cl CD09006 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(ccc3Cl)/C(=N/O)/C DSHS01069 Cc1c(cccc1Cl)/N=C\2/NC(C(=C)S2)(C)C DSHS01073 CSc1cccc(c1)NC(=S)N2CCN3C2(c4ccccc4C3=O)c5ccccc5 DSHS01083 c1csc(n1)N2C(=O)C3C4CC(C3C2=O)C=C4 DSHS01089 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)N CD11078 CN(C)c1cc(oc(=O)c1Cl)c2cccs2 CD11081 c1cc(c(c(c1)Cl)Cl)S(=O)(=O)O/N=C(/Cn2ccc(n2)C(F)(F)F)\N HAN00332 Cc1ccc(cc1C)NC(=S)N(CCC#N)C2CCCCC2 DSHS01257 c1ccc2c(c1)CC3=C2NC(=C(C#N)C#N)C(=C3c4cccs4)C#N FM00172 c1ccc\2c(c1)CC/C2=N\NC(=O)N FM00215 COc1ccc(cc1)NC(=S)N2CCOCC2 DSHS01235 c1ccc2c(c1)ccn2CC(CSc3ccccc3N)O HAN00317 CC(C)(C)SCCNC(=O)c1cccnc1Oc2ccccc2 CD08268 CC(C)(C)C(=O)/C(=C/c1ccc(cc1)C(F)(F)F)/C#N CD10827 Cc1cc(cc(c1Cl)C)OS(=O)(=O)CS(=O)(=O)Oc2cc(c(c(c2)C)Cl)C CD10434 Cc1cc(c(c(c1Cl)C)Cl)OS(=O)(=O)CS(=O)(=O)Oc2cc(c(c(c2Cl)C)Cl)C CD10438 COc1cc(cc(c1NC(=S)N2CCN3C2(c4ccccc4C3=O)c5ccccc5)OC)Cl DSHS01081 COC(=O)c1c(n(nn1)c2cccc(c2)C#C)c3ccccc3 CD08059 c1ccc\2c(c1)CCC/C2=N\NC(=O)N FM00213 CC(C)(C)c1csc(n1)N CD08308 c1ccc(cc1)NC(=O)Nc2ccc(c(c2F)C#N)F CD09117 CS(=O)(=O)c1cc(cc(c1S(=O)(=O)C)S(=O)(=O)C)C(F)(F)F CD09133 Cc1ccc(cc1)S(=O)(=O)CCC(=O)C FM00331 c1cc(ccc1SCc2c(cc(cn2)C(F)(F)F)Cl)Cl HC00023 c1ccc(cc1)NC(=O)N2CCCC2c3cccs3 CD10407 c1ccc(cc1)S(=O)(=O)N2CCCC2c3cccs3 CD10413 Cn1cccc1C(=O)NNC(=N)CSc2ccc(cc2)Cl CD11171 Cc1c(c(c(c(c1C)C)S(=O)(=O)NN(C)c2ccc(cc2[N+](=O)[O-])C#N)C)C CD08107 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCCOc3ccc(cc3[N+](=O)[O-])C(F)(F)F CD08110 c1ccc2c(c1)cccc2NC(=S)NCc3ccncc3 DSHS01265 COc1cccc(c1)NC(=S)N(CCC#N)C2CCCCC2 DSHS01266 c1cc(ccc1NC(=O)Nc2ccc(c(c2F)C#N)F)Cl CD09120 c1cc(ccc1CSc2nc(sn2)SCc3ccc(cc3)Cl)Cl CD08305 c1cc(cnc1)C2CCCN2C(=O)Nc3ccc(cc3Cl)Cl CD10379 Cc1cc(no1)NC(=O)/C(=C/N(C)C)/C#N CD09208 CCOC(=O)CN(C(=O)c1ccccc1[N+](=O)[O-])C(C)(C)C FM00329 CCOC(=O)Cc1cnc(s1)N/N=C/2\CCCc3c2ccc(c3)OC FM00246 Cc1ccc(c(c1)[N+](=O)[O-])OCC2NCCS2 FM00248 COC(=O)c1c(ccs1)NC(=O)c2ccc(cc2)F GK02790 CSCC(=N)NS(=O)(=O)c1ccc(cc1)Cl CD08133 Cc1c(c(n(n1)C)Sc2ccccc2N)[N+](=O)[O-] EN00010 Cn1c2c(cc(s2)c3nc(no3)c4ccc(cc4)C(F)(F)F)c(n1)C(F)(F)F GK02733 Cc1c(c(no1)c2ccccc2)C(=O)NC(C)(C)CCO DSHS01023 Cc1cc(cc(c1F)C)S(=O)(=O)NC(=N)c2ccc(cc2)C(=O)N CD09014 CCOC(=O)CNC(=O)Nc1ccc(cc1)Cl CD09016 CC1(OC(=O)C(=Cc2cc(cs2)Br)C(=O)O1)C CD09034 Cc1csc(c1NC(=O)c2cccc(c2)C(F)(F)F)C(=O)OC GK02773 Cc1csc(c1NC(=O)c2ccc(cc2)F)C(=O)OC GK02792 Cc1ccccc1NC(=S)N2CCOCC2 DSHS01234 c1cc(ccc1NC(=O)Nc2ccc(cc2)SC(F)(F)F)n3ccc(n3)C(F)(F)F HAN00352 c1cc(cc(c1)Cl)NC(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F HAN00354 c1ccc(cc1)c2csc(n2)N/N=C/3\CCCc4c3cccc4 FM00218 COc1cccc(c1)NC(=S)NCc2ccncc2 DSHS01219 COc1cccc(c1)NC(=S)NCc2cccnc2 DSHS01222 Cc1ccc(cc1F)NC(=O)c2c(onc2c3ccccc3Cl)C DSHS01255 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc(c3)SC DSHS01256 Cc1cc(ccc1Cl)c2csc(n2)C(C#N)C(=O)C CD09158 c1cc(c(c(c1)C(=O)O)F)C(=O)O CD10414 COc1ccc(cc1)NC(=S)NCc2cccnc2 DSHS01224 COc1ccccc1NC(=S)N2CCOCC2 DSHS01231 c1ccc(cc1)C23c4ccccc4C(=O)N2CCN3 DSHS01050 Cc1csc(c1NC(=O)c2ccco2)C(=O)OC GK02786 c1cc(ccc1C(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F)Cl HAN00344 COc1ccc-2c(c1)CCc3c2nc(s3)N.Br FM00121 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)ON=C3C4CC5CC(C4)CC3C5 FM00211 c1cc(c(cc1OC(=O)C23CC4CC(C2)CC(C4)C3)Cl)Cl CD08962 COc1ccc\2c(c1)CCC/C2=N\NC(=S)N FM00220 CS/C(=N\C#N)/NCCC1CC1(Cl)Cl CD10991 c1c(cc(c(c1[N+](=O)[O-])NCCC2CC2(Cl)Cl)[N+](=O)[O-])C(F)(F)F CD10986 CC(=O)/C(=C(\N)/SCc1c(cccc1Cl)Cl)/C#N CD09167 CC(C)(C)c1cc(n(n1)S(=O)(=O)c2ccc(cc2F)F)SC CD11021 c1cc(c(cc1OCC(F)(F)F)c2ccn[nH]2)OCC(F)(F)F CD11164 Cc1cc(=O)oc2c1ccc(c2)OCc3c(cccc3Cl)Cl CD08054 c1cc(c(cc1Cl)Cl)C(=O)Oc2cc(cc(c2)Cl)Cl CD08113 c1ccc(c(c1)C(=O)Oc2cc(cc(c2)Cl)Cl)F CD08115 Cc1c(nnn1c2cc(cc(c2)Cl)Cl)c3ccccc3 CD08116 c1cc(ccc1S(=O)(=O)Oc2cc(cc(c2)Cl)Cl)Cl CD08080 CCOC(=O)C1=C(NC(=S)N(C1c2cccs2)C(=O)C)C FM00083 c1ccc(cc1)C2=NOC(=O)C2C=C3CCCC3 FM00085 c1cc(sc1c2cc[nH]n2)Br CD08137 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)N3CCOCC3)C#N CD10983 Cc1cc(no1)NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N CD09204 CCOC(=O)NNC1(CCSC1)C#N CD11152 c1cc(c(cc1NC(=S)N(CCC#N)C2CCCCC2)Cl)Cl DSHS01267 Cc1c(c(n(n1)C)N2CCOCC2)[N+](=O)[O-] EN00006 CC(C)(C)Sc1ccc(cc1C(=O)Nc2ccncc2)[N+](=O)[O-] DSHS01007 c1cc(c(cc1[N+](=O)[O-])C(=O)Nc2ccncc2)SCCO DSHS01012 CN(C)/C=N/c1nnc(s1)SCc2c(cccc2Cl)F CD10269 CN(C)/C=N/c1nnc(s1)SCc2c(cccc2Cl)Cl CD10270 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)OC2=C(CCC2=O)C CD10174 C1CN(CCC1C(=O)N)C(=S)NC2CC3CC2C=C3 CD10315 CCC1(C(=C)S/C(=N\c2cccc(c2)Cl)/N1)CC DSHS01039 c1cc(c(nc1)N2CCC(CC2)C(=O)NC(=O)Nc3ccc(cc3)Cl)[N+](=O)[O-] CD10282 Cc1ccc(cc1NC(=S)NCc2ccncc2)Cl DSHS01262 Cc1cccc(c1NC(=S)NCc2ccncc2)C DSHS01264 c1cc(ccc1NS(=O)(=O)CC(=O)CS(=O)(=O)Nc2ccc(cc2)Cl)Cl CD11153 CC1=C(Sc2ccccc2N1)C(=O)C CD11239 CCOC(=O)C(C(F)(F)F)(NCCc1ccccc1)NC(=O)c2ccccc2Cl JFD02216 c1ccc(cc1)C2=C(c3ccccc3C2=O)N/C=N/O CD09364 COc1c(c(c2c(n1)-c3ccccc3C2)c4ccc(cc4Cl)Cl)C#N FM00027 CC1/C(=C\c2ccc(cc2)C(F)(F)F)/C(=O)c3cc(ccc3S1)Cl FM00029 c1ccc\2c(c1)CC/C2=C(/C#N)\C(=O)N FM00035 CN(C)/C=C/C(=N)SCc1cc(cc2c1OCOC2)F.Cl CD11192 c1cc(cc(c1)Cl)NC(=O)C(C#N)C(=O)c2cccs2 CD11208 CS(=O)(=O)CS(=O)(=O)Oc1ccc(cc1)Br CD10854 Cc1csc(c1NC(=O)C2CC2)C(=O)OC GK02775 Cc1c2c(n(n1)C)SC(=NS2(=O)=O)SC CD10429 CN(C)c1cc(oc(=O)c1Cl)c2ccc(cc2)Cl CD11120 CCOc1c(c(c(c(n1)N)C#N)c2ccc(cc2)C(F)(F)F)C#N FM00212 COc1ccc\2c(c1)CCC/C2=N\NC(=O)N FM00214 c1ccc2c(c1)ccc3c2OC(=C(C3c4ccc(cc4)Cl)C#N)N FM00122 Cc1csc(n1)NN=C2CCCCC2 FM00242 Cc1c(c(sc1C#N)C(=O)NC(=O)OC(CSC)CSC)C CD10491 Cc1c(c(n(n1)C)NCCCN(C)C)[N+](=O)[O-] EN00016 Cc1ccc(c(c1)C)NC(=S)N(CCC#N)C2CCCCC2 DSHS01258 Cc1cccc(c1NC(=S)N(CCC#N)C2CCCCC2)C DSHS01259 CCOC(=O)C1=C(NC(=NC1c2cccs2)SC)C FM00071 Cc1ccc2c(c1C)NC(=O)CC(=N2)c3ccccc3O FM00074 CC1=C(C(=O)CC1)OC(=O)/C=C/c2ccccc2 CD10221 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F HAN00366 CC(=O)C(=NNc1ccc(cc1)n2ccc(n2)C(F)(F)F)C(=O)C HAN00367 Cc1cc(cc(c1F)C)S(=O)(=O)Nc2ccc(cc2F)F CD08238 CC(C)Oc1c(c(c(c(n1)N)C#N)c2ccc3c(c2)OCO3)C#N FM00234 c1c(cc(cc1Br)Br)C(=O)O CD11016 CS(=O)(=O)CS(=O)(=O)Oc1ccc(cc1)C(F)(F)F CD11214 Cc1cccc(c1)n2c(c(cn2)C(=O)C)C CD11216 c1cc(ccc1NC(=O)Nc2nccc(n2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F)Cl CD11217 CCOC(=O)c1ccc(cc1)NC(=S)NCc2cccnc2 DSHS01227 Cc1cc(cc(c1F)C)S(=O)(=O)Oc2c(cccc2Cl)Cl CD08230 c1cc(c(c(c1NC(=O)C(Cl)Cl)Cl)Cl)Cl CD08083 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2ccc(c(c2)Cl)Cl)C)C CD08089 c1cc(c(c(c1)Cl)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl)Cl CD02856 Cc1cc(no1)NC(=O)C(=O)NCc2cccc(c2)Cl CD10320 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(c(c3)Cl)Cl CD08091 Cc1cc(no1)n2nc(nn2)C/C(=N/O)/C CD09269 Cc1cccc(c1)NC(=S)NCc2cccnc2 DSHS01221 COc1ccccc1NC(=S)NCc2cccnc2 DSHS01223 CC(=O)CC(=O)Nc1ccccc1C(=O)OC CD11243 c1ccc(cc1)C(=O)NC(=S)Nc2nc[nH]n2 DP00864 c1ccc(cc1)c2csc(=N)n2c3cccc(c3Cl)Cl.Cl DP00882 CCOC(=O)c1c(csc1N)c2ccccc2 HAN00457 CC1(OC(=O)C(=CNNc2c(cc(cc2Cl)Cl)Cl)C(=O)O1)C CD11236 c1cc(c(c(c1)Cl)CSC(=S)N2CCSCC2)F CD08185 CCOC(=O)c1c(nc(s1)NN=C2Cc3ccccc3C2)C FM00229 Cc1ccc(cc1)C(=O)NNc2c3ccsc3ncn2 GK02856 c1cc(ccc1NC(=O)O/N=C(/Cn2ccc(n2)C(F)(F)F)\N)Cl HAN00348 c1cc2c(cc1Cl)c3c(c([nH]c(=O)c3c(=N)o2)O)C#N FM00194 c1cc(ccc1NC(=O)O/N=C(/Cn2ccc(n2)C(F)(F)F)\N)SC(F)(F)F HAN00349 COC(=O)c1ccsc1NC(=O)C2CCCCC2 GK02857 Cc1c(c(n(n1)C)Oc2c(cccc2Cl)Cl)[N+](=O)[O-] EN00021 c1cc(ccc1NC(=O)O/N=C(/Cn2ccc(n2)C(F)(F)F)\N)OC(F)(F)F HAN00350 c1cc(ccc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)n3ccc(n3)C(F)(F)F HAN00353 CC(=O)Nc1ccc(cc1)S(=O)(=O)N(c2ccc(cc2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)NC(=O)C GK02833 CCOC(=O)c1c(nc(s1)N/N=C/2\CCCc3c2cccc3)C.Cl FM00233 c1ccc(c(c1)C(=O)O)SC/C(=N\O)/c2ccc(cc2)[N+](=O)[O-] FM00290 CCOC(=O)c1c(nc(s1)N/N=C/2\CCCc3c2ccc(c3)OC)C FM00231 Cc1c(c(on1)C)S(=O)(=O)Nc2cc(cc(c2)Cl)Cl CD10456 c1cc(ccc1C(=O)ON=C2C3CC4CC(C3)CC2C4)Cl FM00196 c1cc(ccc1C(=O)ON=C2C3CC4CC(C3)CC2C4)F FM00197 c1cc(c(c(c1)Cl)C(=O)N=C2NCCCN2)Cl EN00041 Cc1csc(c1NC(=O)CSc2ccc(cc2)Cl)C(=O)OC GK01328 c1cc(cc(c1)C(F)(F)F)C(=O)ON=C2C3CC4CC(C3)CC2C4 FM00198 Cc1cc(no1)NC(=O)CN2CCOCC2 CD09224 Cc1cc(no1)NC(=O)CN2CCSCC2 CD09225 CC(=N)NCCCn1ccnc1.I CD08171 Cc1c2c(n(n1)C)SC(=NS2(=O)=O)SCc3c(cccc3Cl)F CD10467 Cc1cc(no1)NC(=O)CN2CCCC2 CD09226 Cc1cc(no1)n2cnc(n2)c3c[nH]nc3C CD09247 c1ccnc(c1)CCNC(=S)NC2CC3CCC2C3 HR00046 COc1ccccc1NC(=S)NC2CC3CCC2C3 HR00052 CN(C)NC(=S)NC1CC2CCC1C2 HR00053 c1cc(c(cc1Cl)Cl)C2CC(=CC(=O)C2)Cl CD11474 COc1cc(c(cc1OC)c2c[nH][nH]c2=O)CO CD11482 Cc1ccc(cc1)C(=O)CSC#N DP00874 C=CCN1C2CS(=O)(=O)CC2SC1=N.Br JFD02308 c1ccc(cc1)N2C3CS(=O)(=O)CC3SC2=N.Br JFD02309 CCCCN(CCCC)c1ccc(cc1)S(=O)(=O)c2ccccc2 JFD02310 c1ccc(cc1)Oc2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl HC00043 c1ccc2c(c1)c3c(c4c2C(C(=C(O4)N)C#N)c5ccc(cc5)Cl)OC(=C(C3c6ccc(cc6)Cl)C#N)N FM00128 c1ccc2c(c1)c3c(c4c2C(C(=C(O4)N)C#N)c5ccc(cc5)F)OC(=C(C3c6ccc(cc6)F)C#N)N FM00129 CCOC(=O)c1ccc(cc1)NC(=S)NCCc2ccc(c(c2)OC)OC HR00008 Cc1ccc(c(c1)[N+](=O)[O-])OCC2N(CCS2)C(=O)c3ccc(cc3)C(F)(F)F FM00281 Cc1cc(no1)n2cnc(n2)c3cn(nc3C)C CD09260 CC(=O)C(Cc1ccc(cc1)F)(Cc2ccc(cc2)F)C(=O)OC GK02763 Cc1ccc(c(c1)C)NC(=S)Nc2ccc(cc2)C(C)C DSHS01209 Cn1cccc1C(=O)NNC(=N)CN2CCCCC2 CD11169 c1ccc(cc1)C2=C(c3ccccc3C2=O)N CD09182 c1cc(c(cc1[N+](=O)[O-])C(=O)N)C(=O)N CD09423 CN(C)c1cc(oc(=O)c1Cl)c2ccc(cc2)F CD11187 C1CC/C(=N\O)/N(CC1)C(=O)N CD11196 Cc1csc2c1c(ncn2)N3CCN(CC3)C(=O)Nc4ccc(c(c4)Cl)Cl GK02715 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(cc(c3)OC)C(F)(F)F CD11051 CN(C)/C=C/C(=O)c1ccc(cc1)C#N CD11172 CN(C)c1cc(oc(=O)c1Cl)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F CD11174 c1cc(c(cc1C(=O)O)S(=O)(=O)N)Cl JFD00629 c1ccc(c(c1)C(=O)NC(=O)NNc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl CD11304 CC(=O)C(/C=N/c1ccc(cc1Cl)Cl)C(=O)C CD11307 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)C(=O)Nc4ccccc4 HAN00375 CN(C)/C=C/C(=N)SCc1c(cccc1Cl)Cl.Cl CD11182 CSCCC1C(=O)NC(=O)N1 FM00156 CCOC(=O)CNC(=O)Nc1ccccc1 CD09015 c1ccc(c(c1)C(=O)NC2CCSC2)NC(=O)Nc3ccc(cc3)Cl CD10361 Cc1ccc(cc1)S(=O)(=O)O.c1ccc(cc1)COC(=O)C[C@@H](C(=O)OCc2ccccc2)N GK02767 CC(=O)Nc1ccc(cc1)S(=O)(=O)N(c2ccc(cc2F)F)S(=O)(=O)c3ccc(cc3)NC(=O)C GK02830 c1cc(c(cc1Cl)Cl)C2CC(=O)CC(=O)C2 CD11309 c1ccc(cc1)C(c2ccccc2)c3ccnn3C(=O)c4ccccc4 CD11444 CCS(=O)(=O)N1CCN(CC1)c2nc(ns2)c3ccccc3 HAN00382 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)C(=O)/C=C\C(=O)O HAN00385 Cc1ccc(cc1C)NC(=O)c2cc(ccc2[N+](=O)[O-])N DP00911 c1cc(ccc1c2csc(=N)n2c3cc(c(cc3Cl)Cl)Cl)Cl.Cl DP00886 CC(C)c1ccc(cc1)NC(=O)c2ccccc2N DP00887 Cc1cc(no1)NC(=O)/C(=C/c2cc(cs2)Br)/C#N CD09201 Cc1cc(no1)NC(=O)/C(=C/c2ccc(cc2Cl)Cl)/C#N CD09205 c1ccc2c(c1)cc(o2)c3cc[nH]n3 CD09206 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCCC3 DSHS01240 CC(C)(C)SCCNC(=O)c1ccccc1F CD08278 COc1ccc(cc1)/C=C(\C#N)/c2[nH]c3ccccc3n2 FM00191 c1cc(c(c(c1)CSC(=N)N)F)CSC(=N)N CD09096 COc1ccc(cc1)C2CC(=CC(=O)C2)Cl CD11468 CC(C)/N=C/c1ccc(cc1)c2ccccc2 FM00344 c1ccc2c(c1)C(CCO2)O JFD00618 CC1(c2cc(ccc2N(C13C=Nc4c5ccccc5ccc4O3)C)Cl)C JFD00622 CC(=O)c1c(ccs1)N2C(=O)c3ccccc3C2=O GK01413 CCOC(=O)C(C(F)(F)F)(NCCc1ccc(c(c1)OC)OC)NC(=O)c2ccco2 JFD02264 COC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1Cl)O JFD02266 Cc1cc(no1)n2cnc(n2)C/C(=N/O)/C CD09242 c1cc2c(cc1C3CC(=O)CC(=O)C3)OCO2 CD11317 CC(=O)/C=C/c1ccc(c(c1)Cl)Cl CD11322 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)C(=O)c4ccccc4C(=O)O HAN00386 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)CC(CSc4ccccc4)O.Cl HAN00388 Cc1ccc(cc1)S(=O)(=O)ON2C(=O)CNC2=O CD08296 c1ccc(cc1)c2ccc(cc2)/C=N/C3CC3 FM00345 CNn1cnc2ccccc2c1=O CD09515 CC(C)(C)C(=O)C(C#N)C(=O)Nc1ccc(cc1)Cl CD11234 CC(=O)/C(=C(\N)/SCc1csc(n1)c2ccc(cc2)Cl)/C#N CD09243 Cc1cc(no1)n2cnc(n2)c3cnoc3C CD09266 Cc1c(c(n(n1)S(=O)(=O)c2ccc(cc2)Cl)C)Cc3c(cccc3Cl)Cl CD09088 CN(C(=O)Nc1ccc(cc1)Cl)n2cnc3ccccc3c2=O CD09522 CC(=O)/C(=C(\N)/SC)/C#N CD09271 Cc1cc(no1)n2cnc(n2)C/C(=N/OC(=O)Nc3ccc(cc3)Cl)/C CD09278 CSc1ccccc1NC(=O)c2cc(sc2Cl)Cl CD09471 c1cc(c(cc1Cl)Cl)/C=N/OC(=O)c2cc(sc2Cl)Cl CD09473 CN(C)c1cccc(c1CNC(=O)Nc2ccccc2)N(C)C CD09475 c1ccc2c(c1)NC(=O)CC(=N2)C(F)(F)F HAN00425 COC(=O)c1c(ccs1)NC(=S)Nc2ccsc2C(=O)OC GK02769 CC1(OC(=O)C(=CNNc2ccc(cc2)C(F)(F)F)C(=O)O1)C CD11248 CN(C(=O)Nc1ccccc1)n2cnc3ccccc3c2=O CD09519 Cc1ccc(cc1)S(=O)(=O)NNc2nccc(n2)C(F)(F)F HAN00410 Cc1cc(cc(n1)NNC(=O)NC(=O)c2c(cccc2OC)OC)C(F)(F)F CD11353 c1ccc2c(c1)ncc(n2)/C=C/c3c(cccc3Cl)F CD11251 c1cc(sc1)C(=O)Nc2nccc(n2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F CD11254 CN(C)c1cc(oc(=O)c1Cl)c2ccc(cc2)Br CD11144 c1cc(oc1)/C=C/2\C(=O)C3CCN2CC3 FM00113 c1cc(ccc1n2ccc(n2)C(F)(F)F)[N+](=O)[O-] HAN00339 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCCCC3 DSHS01241 CC1CN(CC(O1)C)C(=S)Nc2cccc3c2cccc3 DSHS01244 CC1CN(CC(O1)C)C(=S)Nc2cccc(c2)OC DSHS01249 c1cc(ccc1C(=O)Sc2nccc(n2)C(F)(F)F)Cl HAN00413 c1cc(ccc1C(=O)CSc2nccc(n2)C(F)(F)F)Br HAN00416 Cc1csc(c1Cl)NC(=O)Nc2ccc(cc2F)F GK01363 c1cc(ccc1/C=N/C(=C(/C#N)\N)/C#N)Cl FM00256 c1cc(ccc1/C=N/C(=C(/C#N)\N)/C#N)C(F)(F)F FM00257 CCOC(=O)c1ccc(cc1)NC(=S)N2CCOCC2 DSHS01236 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CC(OC(C3)C)C DSHS01239 c1cc(ccc1NC(=O)/C=C/C(=O)O)n2ccc(n2)C(F)(F)F HAN00356 Cc1cc(no1)N/N=N/c2cc(on2)C CD09180 c1ccc(cc1)NC(=O)Nc2ccccc2C(=O)NCCC3CC3(Cl)Cl CD11000 c1cc(c(nc1)SCCCC#N)C(=O)O FM00193 CCOC(=O)C(/C=N/c1ccc(cc1Cl)Cl)C(=O)C CD11308 Cc1csc(c1Cl)C(=O)O/N=C(/c2ccc(cc2)Cl)\N GK01368 c1cc(c(cc1Cl)Cl)OCc2c(cc(cn2)C(F)(F)F)Cl HC00040 c1cc(ccc1C#N)OCc2c(cc(cn2)C(F)(F)F)Cl HC00041 Cc1c(cnn1c2ccc(c(c2Cl)Cl)Cl)C(=O)C CD11003 Cc1c(cnn1c2ccc(cc2)C(F)(F)F)C(=O)C CD11014 CN(C)/C=N/C1=C(C(=O)c2c1cccc2)c3ccccc3 CD09185 CN(C)c1cc(oc(=O)c1Cl)c2ccc(cc2)C#N CD11173 CN(C)/C=C/C(=O)c1ccc2ccccc2c1 CD11176 Cc1ccc(cc1)C(=O)Nc2nccc(n2)c3ccc4c(c3)OCCO4 FM00204 c1cc(c(c(c1)CN2CCOCC2)F)CN3CCOCC3 CD09081 Cc1ccc(c(c1)[N+](=O)[O-])OCC2N(CCS2)S(=O)(=O)c3cc(cc(c3)Cl)Cl FM00301 Cc1c(sc(n1)NC(=N)NC(=O)Nc2ccc(cc2)Cl)Br CD11055 Cc1ccc(c(c1)[N+](=O)[O-])OCC2N(CCS2)C(=O)c3c(cccc3Cl)Cl FM00282 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)Oc3ccc(cc3)Cl)C#N CD11029 c1cc(ccc1/C=N\C(=C(\C#N)/NC(=O)Nc2ccc(cc2)OC(F)(F)F)\C#N)Cl FM00312 c1ccc(cc1)NC(=O)C(C#N)C(=O)c2cccs2 CD09339 Cc1ccc(cc1)Sc2c(c(nn2C)C)[N+](=O)[O-] EN00009 Cc1c(c(n(n1)C)NCCSCc2c(cccc2Cl)Cl)[N+](=O)[O-] EN00012 Cc1c(c(n(n1)C)Sc2ccc(cc2)Cl)[N+](=O)[O-] EN00013 c1ccc(cc1)CN(S(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl CD11328 CN(C)c1cc(oc(=O)c1Cl)c2ccccc2 CD11145 CCOC(=O)C(C(F)(F)F)(NCc1ccccn1)NC(=O)c2ccccc2Cl JFD02214 CCOC(=O)C(C(F)(F)F)(NCCc1ccc(c(c1)OC)OC)NC(=O)c2ccccc2Cl JFD02215 c1ccc(cc1)c2csc3c2c(=O)[nH]cn3 HAN00459 CC(C)(C)c1cc(c(s1)C#N)N(S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK02815 Cn1cccc1C(=O)N/N=C/c2c(cccc2Cl)Cl CD11061 Cn1cccc1C(=O)N/N=C/c2ccccn2 CD11062 c1cc2c(cc1Br)cc(o2)c3cc[nH]n3 CD09330 c1ccc(cc1)NC(=O)OC(CSc2ccccn2)CSc3ccccn3 CD09337 Cc1c(c(on1)C)C(=O)O/N=C(/Cn2ccc(n2)C(F)(F)F)\N HAN00327 CC(=NNC(=O)c1cccn1C)C CD11063 c1cc(sc1)C(=O)C(C#N)C(=O)Nc2ccc(cc2)Cl CD09340 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCC#C CD11106 c1cc(sc1)/C=C/c2ccnn2S(=O)(=O)c3ccc(cc3)Cl CD11275 Cc1ccc(cc1)SCc2cc(cc3c2OCOC3)F CD08373 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)CC(COc4ccc(cc4)Br)O HAN00387 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)CC(COc4cccc(c4)C(F)(F)F)O HAN00389 c1ccc2c(c1)CC(=NNC(=S)N)C2 FM00222 c1ccc2c(c1)C(=O)N(C2=O)c3ccc(cc3)n4ccc(n4)C(F)(F)F HAN00362 c1ccc(cc1)c2c([nH]nc2O)O CD08938 c1cc(ccc1SCc2cc(cc3c2OCOC3)F)Cl CD08378 c1ccc(cc1)c2csc(n2)NN=C3Cc4ccccc4C3 FM00230 Cc1c(c(no1)c2ccccc2)C(=O)ON=C3C4CC5CC(C4)CC3C5 FM00209 Cc1ccc(n1c2ccsc2COC(=O)Nc3c(onc3c4c(cccc4Cl)F)C)C CD08955 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(/Cn2ccc(n2)C(F)(F)F)\N HAN00328 c1ccc(c(c1)C(=O)NC2CCCCC2)N DP00908 c1cc(sc1)CN(S(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl CD11279 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC(=O)c3ccccc3Oc4ccc(cc4Cl)Cl CD08921 CC(=O)Nc1ccc(cc1)S(=O)(=O)N(c2ccccc2C(F)(F)F)S(=O)(=O)c3ccc(cc3)NC(=O)C GK02832 c1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)Sc3nccc(n3)C(F)(F)F HAN00289 c1cc(c(cc1Cl)Cl)CS(=O)(=O)CC(Cn2ccc(n2)C(F)(F)F)O HAN00290 Cc1ccc(cc1C)n2c(=O)c3ccccc3nn2 DP00909 Cc1ccc(cc1C)NC(=O)c2cc(ccc2N)Cl DP00910 CCOC(=O)C(=CNc1cscc1C)C(=O)OCC GK01407 Cc1csc(c1Cl)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N GK01369 CN(C)c1ccc(cc1)C2CC(=O)CC(=O)C2 CD11315 c1ccc(c(c1)C(=O)NC(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl CD11316 Cc1ccc(cc1[N+](=O)[O-])OCC2NCCS2 FM00313 c1cn(nc1C(F)(F)F)CC(CN2CCCC2)O HAN00287 CCO/C=N\C1=C(C(c2ccc3ccccc3c2O1)c4ccc(cc4)OC)C#N FM00126 c1cc(cnc1)NS(=O)(=O)c2cc(sc2Cl)Cl CD09550 c1cnccc1C(=N)NS(=O)(=O)c2cc(sc2Cl)Cl CD09605 Cc1cc(cc(n1)n2c(c(cn2)C(=O)C)C)C(F)(F)F CD11385 C#CCNC(=O)/C=C/C(=O)O CD11389 c1ccn(c1)S(=O)(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F CD11386 c1ccc(cc1)Oc2ccccc2NC(=O)c3ccccc3Cl CD09559 C1CCN(C1)S(=O)(=O)c2c(c(sc2Cl)Cl)Br CD09560 CC(c1[nH]c2ccccc2n1)O CD09564 c1cc(ccc1OS(=O)(=O)c2c(c(sc2Cl)Cl)Br)Cl CD09627 Cc1c(c(n(n1)C)C)[N+](=O)[O-] CD09637 Cc1ccc(cc1)C(=O)/C=C/N(C)C CD11137 CN(C)/C=C/C(=O)c1ccc(cc1F)F CD11140 CN(C)/C=C/C(=O)c1ccccc1 CD11141 c1cc(c(c(c1)Cl)CC(Cc2c(cccc2Cl)Cl)(C#N)C#N)Cl CD09403 c1cc(sc1)C(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F HAN00341 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F HAN00342 c1cc(ccc1C(=N)NS(=O)(=O)c2cc(sc2Cl)Cl)Cl CD09608 c1cc(ccc1CSC2=NCCN2)Cl.Cl DP01048 c1ccc(c(c1)CSC2=NCCCN2)Cl.Cl DP01052 c1ccc(cc1)CN2CC(CN(C2)Cc3ccccc3)C#N CD11395 CC(C(C)(C)C)N/C=C(\C#N)/c1[nH]nnn1 CD11595 C(c1[nH]nnn1)SCc2[nH]nnn2 CD11605 Cc1c(c(n(n1)C)Oc2ccc(cc2)C(C)(C)C)[N+](=O)[O-] EN00024 CS/C(=N\C(=O)c1c(cccc1Cl)Cl)/N2CCOCC2 EN00029 c1ccc(c(c1)C(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F)C(=O)O HAN00358 c1cc(ccc1n2ccc(n2)C(F)(F)F)N3C(=O)C=CC3=O HAN00359 CS/C(=N\C(=O)c1c(cccc1Cl)Cl)/N2CCSCC2 EN00033 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Cl)n3ccc(n3)C(F)(F)F HAN00364 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)OC(C)c2[nH]c3ccccc3n2 CD09592 c1cc(cnc1)OS(=O)(=O)c2c(c(sc2Cl)Cl)Br CD09626 CN(C(=O)Nc1ccc(cc1)OC(F)(F)F)/N=C/c2c(cc(cn2)C(F)(F)F)Cl HC00080 CNc1ccc(cc1C(=O)NCCc2ccccc2)Cl DP01028 CNc1ccc(cc1C(=O)NCc2ccco2)Cl DP01031 CN1C/C(=C\c2sccc2)/C(=O)/C(=C/c3sccc3)/C1 DP01040 c1ccc(cc1)NC2=CC(=O)CC(C2)c3ccc(cc3)Cl CD11604 c1cc(ccc1S(=O)(=O)Cc2c(cc(cn2)C(F)(F)F)Cl)Cl HC00116 CC(=O)Nc1ccsc1C(=O)O GK00015 c1c(c(sc1Cl)Cl)c2csc(n2)NC(=N)N CD11359 c1cc(ccc1C2CC(=O)CC(=O)C2)F CD11363 CCOC(=O)CC1C(=O)NCCN1 CD11371 COc1ccc(cc1)C2CC(=O)CC(=O)C2 CD11372 Cc1cc(cc(n1)NNC(=O)NC(=O)c2ccc(cc2)Cl)C(F)(F)F CD11377 c1ccc(cc1)C(=O)c2cccc(c2)NC=C3C(=O)NC(=O)NC3=O JFD02302 c1ccc(c(c1)S(=O)(=O)/C(=C/c2c(cc(cn2)C(F)(F)F)Cl)/C#N)Cl HC00084 CSC(=NS(=O)(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F)SC CD11401 c1ccnc(c1)CNS(=O)(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F CD11405 CCOC(=O)C(=CNc1ccsc1C(=O)OC)C(=O)OCC GK00018 c1ccc(c(c1)C(=O)O)SC/C(=N\O)/c2cccc(c2)[N+](=O)[O-] FM00293 C#CCNS(=O)(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F CD11409 Cc1cc(no1)NC(=O)c2ccccc2 CD09215 Cc1cc(no1)NC(=O)CSc2ccc(cc2)Cl CD09229 Cc1cc(cc(c1F)C)S(=O)(=O)n2ccc(n2)c3cc(sc3Cl)Cl CD09218 c1cc(sc1)c2c(c(c(o2)N)c3ccc(cc3Cl)Cl)C#N CD09230 c1ccc\2c(c1)-c3c(cc(nn3)c4cccc(c4)OC(F)(F)F)/C2=N\O FM00341 c1cc(oc1)/C=N/NC(=O)c2c(nccn2)N HAN00440 CN(C)CCCNS(=O)(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F CD11398 c1cc(c(cc1OCC(F)(F)F)S(=O)(=O)N)OCC(F)(F)F CD11399 c1cc(ccc1/C=N/NC(=O)c2c(nccn2)N)Cl HAN00436 CN(C)/C=C/C(=O)c1nccs1 CD11400 COc1ccc(c(c1OC)OC)/C=N/NC(=O)c2c(nccn2)N HAN00442 c1ccc(c(c1)C(=O)O)SCC(=O)c2cccc(c2)[N+](=O)[O-] FM00291 c1ccc(cc1)c2c(nnc(n2)c3ccnc(c3)c4nc(c(nn4)c5ccccc5)c6ccccc6)c7ccccc7 JFD00630 c1c(cc(cc1Cl)Cl)NC(=O)c2cc(sc2Cl)Cl CD09460 c1ccc(c(c1)NC(=O)c2cc(sc2Cl)Cl)Oc3ccc(cc3Cl)Cl CD09462 c1ccc(c(c1)NC(=O)c2cc(sc2Cl)Cl)F CD09463 c1ccc(cc1)C2=C(c3ccccc3C2=O)N/C=N/OC(=O)Nc4ccccc4 CD09396 c1cc(ccc1C(=O)Nc2ccsc2C(=O)O)Cl GK00040 Cc1ccc(cc1C)NC(=O)c2ccccc2N DP00904 CC(C)c1ccc(cc1)n2c(=O)c3ccccc3nn2 DP00905 CN(C)c1cc(oc(=O)c1Cl)c2ccc(cc2)[N+](=O)[O-] CD11156 c1cc(ccc1NS(=O)(=O)CC(=O)CS(=O)(=O)Nc2ccc(cc2)Br)Br CD11162 c1cc2c(cc1Cl)CC(=O)N2 JFD00620 COc1cc(c(cc1I)OC)Cl DP00952 CC1CCN(CC1)C(=S)NC2CC3CCC2C3 HR00044 CNC(=S)NC1CC2CCC1C2 HR00048 Cc1cccn(c1=O)Cc2c(cccc2Cl)F CD09414 c1cc(c(cc1Cl)Cl)OS(=O)(=O)CS(=O)(=O)Oc2ccc(cc2Cl)Cl CD09438 Cc1cc(=O)oc2c1ccc(c2)OCC(=O)O JFD00632 c1c(ccc(c1)Cl)/C=C\2/C(=O)/C(=C/c3ccc(cc3)Cl)/CCC2 DP00954 Cc1cc(no1)NC(=O)CSCC(=O)O CD11549 c1ccc(c(c1)C(=O)NC(=O)NNc2ccccc2C(F)(F)F)Cl CD11294 Cc1ccc(cc1)C2=NC(N=C(O2)N(C)C)(C(F)(F)F)C(F)(F)F JFD02222 CC(C)(C)C(Cc1ccccc1)C(=O)O JFD00644 c1cc(ccc1NN=C(C#N)C#N)n2ccc(n2)C(F)(F)F HAN00369 CCOC(=O)/C(=N/Nc1ccc(cc1)n2ccc(n2)C(F)(F)F)/C(=O)C(F)(F)F HAN00370 C#Cc1cccc(c1)NC(=O)c2cc(sc2Cl)Cl CD09465 CC(C)c1ccc(cc1)NC(=S)NC2CC3CCC2C3 HR00049 c1cc(c(c(c1)Cl)Cl)n2c(csc2=N)c3ccc(cc3)Cl.Cl DP01084 CCOC(=O)c1c(csc1N)C GK00116 c1ccc(cc1)C2=CSC3=NCCCCN23.Br DP01093 COc1ccc(cc1)NC(=O)c2cc(ccc2OCC(F)(F)F)OC CD11286 Cc1ccc(c(c1F)C)S(=O)(=O)N(CCc2ccccc2)S(=O)(=O)c3ccc(cc3)Cl CD11289 c1cc(ccc1CCNS(=O)(=O)c2cc(sc2Cl)Cl)Cl CD09558 c1cc2c(c(c1)Cl)c(n[nH]2)NS(=O)(=O)c3ccc(cc3)Cl CD11431 c1ccc\2c(c1)CC/C2=N\NC(=S)N FM00310 CSCC(=O)Nc1ccc(c(c1)Cl)F CD11422 CC(=O)c1ccc(cc1)Oc2cccc(c2C#N)Cl CD11427 CCCN(CCC)C(=S)Nc1cccc(c1)OC HR00012 CN(C)/C=N/C(=N\OCc1c(cccc1Cl)F)/c2ccc(cc2)Cl CD09663 Cc1c(c(c(c(c1C)C)CSC2=NCCN2Cc3ccccc3)C)C.Cl DP01102 CS(=O)(=O)n1c(ccn1)/C=C/c2cccs2 CD11277 c1ccn(c1)S(=O)(=O)c2cc(sc2Cl)Cl CD09547 Cc1cc(no1)NS(=O)(=O)c2cc(sc2Cl)Cl CD09549 CN(C)CCCNS(=O)(=O)c1cc(sc1Cl)Cl CD09561 c1ccc(cc1)/C=C/C=C\2/C(=O)/C(=C/C=C/c3ccccc3)/CCC2 DP00956 COc1cc(c(cc1Cl)OC)C#N DP00960 CCOC(=O)C(C(F)(F)F)(NCCOC)NC(=O)c1ccccc1Cl JFD02218 CCOC(=O)C(C(F)(F)F)(NCc1ccco1)NC(=O)c2ccccc2Cl JFD02219 CN(C)c1ccsc1C(=O)NN GK00043 CCOC(=O)CC(=O)Nc1ccsc1C(=O)OC GK00044 CN(C)CCCN(S(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD11261 c1cc(sc1)C2CC(=O)CC(=O)C2 CD11291 CCOC(=O)C(C)N(Cc1ccccc1)C(=O)Nc2ccc(cc2)Cl CD09023 CCOC(=O)C(C)N(Cc1ccccc1)C(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C CD09024 c1c(csc1/C=C(\C#N)/C(=O)N)Br CD09036 CN(C)/C=N/C(=S)NC1CC2CC1C=C2 CD09052 c1ccc(cc1)Oc2ccccc2NC(=O)Nc3ccc(cc3)Cl CD09553 Cc1csc(c1NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N)C(=O)OC GK01339 CCOC(=O)C(C(F)(F)F)(NCCc1ccc(cc1)OC)NC(=O)c2ccccc2Cl JFD02217 Cc1nnc(s1)NC(=S)NC(=O)c2ccc(cc2)Cl DP00863 Cc1ccc(cc1)c2csc(=N)n2c3ccccc3.Cl DP00875 c1ccnc(c1)CNC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2 JFD02227 c1ccc(cc1)C(=O)CSC#N DP00881 Cc1ccc(cc1)c2csc(=N)n2c3ccc(cc3)OC.Cl DP00879 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3c(cccc3N(C)C)N(C)C CD09482 c1ccc(cc1)NC(=O)Nc2nccc(n2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F CD11215 c1c(c(sc1Cl)Cl)S(=O)(=O)N2CCCC2 CD09498 c1c(cc2c(c1)OCO2)/C=C\3/C(=O)/C(=C/c4cc5c(cc4)OCO5)/CCC3 DP00953 c1ccc(cc1)CSC[C@H](CO)N JFD00658 CC(C)(C)C(=O)Nc1ccccc1Cc2ccccc2 JFD00662 Cc1ccc(cc1)c2csc(=N)n2c3ccc(cc3)Cl.Cl DP00877 Cc1ccc(cc1)CSC2=NCCCN2.Cl DP01053 Cc1ccc(cc1C)CSC2=NCCCN2.Cl DP01055 c1ccc(cc1)CN2CCNC2=S DP01057 c1cc(ccc1c2cc([nH]n2)CCCO)Cl CD09641 CS(=O)(=O)CS(=O)(=O)Oc1ccc(cc1F)F CD11034 CC(=O)C(C)(CCC#N)CCC#N CD11345 c1cc(ccc1/C=N/Nc2nccc(n2)C(F)(F)F)C(F)(F)F HAN00392 CCN(S(=O)(=O)c1ccc(cc1)F)S(=O)(=O)c2c(c(c(c(c2C)C)C)C)C CD11340 COc1ccc(cc1)S(=O)(=O)N(c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3F)F CD11341 c1cc(ccc1NS(=O)(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)Cl CD11343 Cc1cc(no1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccc(cc2)OC JFD02237 C/C(=N\OC(=O)C)/c1nccs1 CD11516 Cc1ccccc1C2=NC(N=C(O2)N3CCOCC3)(C(F)(F)F)C(F)(F)F JFD02255 Cc1cccc(c1Oc2c(c(nn2C)C)[N+](=O)[O-])Cl EN00026 Cc1c(c(n(n1)C)Oc2ccc(cc2)OC)[N+](=O)[O-] EN00027 CCOC(=O)c1cc(c(nc1/C=C/N(C)C)C(F)(F)F)C(=O)OCC HC00056 CN(C(=O)Nc1ccc(cc1)Cl)/N=C/c2c(cc(cn2)C(F)(F)F)Cl HC00081 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(=O)N/N=C/c3ccc(cc3Cl)Cl HC00113 c1cc(c(cc1F)F)NC(=O)c2cc(sc2Cl)Cl CD09464 CN(C)/C=C(\C#N)/C(=O)NOCc1c(cccc1Cl)F CD11299 CSC(=NC(=O)c1c(cccc1Cl)Cl)SC EN00023 CS/C(=N\C(=O)c1c(cccc1Cl)Cl)/N2CCCC2 EN00032 c1cc(c(c(c1)Cl)/C=N/OC(=O)c2cc(sc2Cl)Cl)Cl CD09467 Cc1cc(no1)NC(=O)c2cc(sc2Cl)Cl CD09468 c1cc(c(c(c1)CSC(=S)N2CCOCC2)F)CSC(=S)N3CCOCC3 CD09100 c1cc(c(c(c1)Cl)C#N)NCCCN2CCCCC2 CD09104 CSc1cc(cc(c1SC)SC)C(F)(F)F CD09130 Cc1ccc(c(c1)[N+](=O)[O-])OCC2N(CCS2)C(=O)c3c(onc3c4c(cccc4Cl)Cl)C FM00297 CN(C)/C=C\1/C(=NOC1=O)c2ccccc2 CD09140 COC(=O)c1ccccc1SCC(=O)c2cccc(c2)[N+](=O)[O-] FM00299 c1cc(ccc1C(=O)N(C2C3CC4CC(C3)CC2C4)OC(=O)c5ccc(cc5)F)F FM00300 COc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C(F)(F)F JFD02235 Cc1c(c(n(n1)C)Oc2ccc(cc2)F)[N+](=O)[O-] EN00025 Cc1ccccc1C2=NC(N=C(O2)N3CCCCC3)(C(F)(F)F)C(F)(F)F JFD02254 c1ccnc(c1)c2c(nccn2)c3ccccn3 JFD00670 CS(=O)(=O)N(CCc1ccc(cc1)Cl)S(=O)(=O)C CD11342 c1ccc(cc1)C(c2ccccc2)c3ccn[nH]3 CD11348 c1cc(c(c(c1)C#N)Oc2ccc(cc2)NC(=O)c3ccc(cc3)Cl)C#N CD11037 Cc1cc(no1)n2nc(nn2)C/C(=N/OC(=O)Nc3ccc(cc3)Cl)/C CD09291 COc1cc(cc(c1)NC(=O)c2ccc(cc2)Cl)C(F)(F)F CD11050 Cc1cc(no1)n2nc(nn2)C/C(=N/OS(=O)(=O)c3ccc(cc3)Cl)/C CD09308 c1ccnc(c1)SCC(CSc2ccccn2)OC(=O)Nc3ccc(cc3)Cl CD09319 CN1C/C(=C\c2ccc(cc2)OC)/C(=O)/C(=C/c3ccc(cc3)OC)/C1 DP00999 CSC(=NS(=O)(=O)c1cc(sc1Cl)Cl)SC CD09539 c1cc(oc1)C2CC(=O)CC(=O)C2 CD11333 CC(=O)C(C)(CCC(=O)O)CCC(=O)O CD11355 c1cc(ccc1c2cc(c(s2)C(=O)N)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl GK01450 Cc1c(c(c(c(c1C)C)CSc2[nH]c3ccccc3n2)C)C.Cl DP01103 Cc1c(c(nn1C)C/C=N/O)[N+](=O)[O-] CD09681 Cc1cn(nc1c2ccccc2)C(=O)NC CD09692 C1COCCN1S(=O)(=O)CS(=O)(=O)N2CCOCC2 CD09392 c1ccc2c(c1)ccn2CC(CNCc3ccc(c(c3)Cl)Cl)O HAN00316 c1cn(nc1C(F)(F)F)C/C(=N\O)/N HAN00323 CCN(S(=O)(=O)c1cc(sc1Cl)Cl)S(=O)(=O)c2cc(sc2Cl)Cl CD11258 c1cc(sc1)/C=C/c2ccnn2C(=O)Nc3ccc(cc3)Cl CD11268 CC(C)(C)c1[nH]c2ccccc2n1 DP01005 CC1CC(CC(C1)(C)C)NC(=O)c2cc(ccc2NC)Cl DP01007 CC(C(C)(C)C)NS(=O)(=O)c1ccc(cc1)Oc2cccc(c2C#N)Cl CD11574 c1ccc(cc1)CN2CC(CN(C2)Cc3ccccc3)CNS(=O)(=O)c4ccc(cc4)Cl CD11575 CN(C)c1ccc(cc1)C2NC(=NN2)c3ccc(cc3)Cl DP01118 c1cc(ccc1C2=NNC(N2)c3ccc(c(c3)Cl)Cl)Cl DP01120 CC1(COCCN1C(=O)c2ccc(cc2)Cl)C HAN00478 c1c(cn2cc(nc2c1Cl)c3nnc(o3)S)C(F)(F)F HAN00486 c1cc(sc1)CN(S(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD11280 COc1ccc(c(c1)C(=O)Nc2cccnc2)OCC(F)(F)F CD11287 c1ccc2c(c1)[nH]c(n2)/C(=C/c3cccs3)/C#N FM00160 Cc1ccc(cc1)c2csc(=N)n2c3ccc(cc3)[N+](=O)[O-].Cl DP00880 c1ccc(cc1)c2csc(=N)n2c3ccc(cc3Cl)Cl.Cl DP00883 Cc1csc(c1NC(=O)c2c(cccc2F)F)C(=O)OC GK01397 Cc1csc(c1NC(=O)c2ccc(cc2)C(C)(C)C)C(=O)OC GK01398 c1cc(ccc1CSc2c(c(sn2)Nc3ccc(cc3)Cl)C#N)Cl DP00892 c1ccc(c(c1)C2=NCCCN2)SCc3cc(sc3Cl)Cl.Cl CD11594 CC(C)(C)c1ccc(cc1)c2nc(c(s2)CC(=O)O)O HAN00458 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H](C(O1)Nc2ccccc2[N+](=O)[O-])OC(=O)C)OC(=O)C)OC(=O)C JFD02281 c1cc2c(c(ccc2)/C=C\3/C(=O)/C(=C/c4c5c(ccc4)cccc5)/CC3)cc1 DP00967 c1ccc(cc1)Oc2ccccc2NC(=O)c3cccs3 CD09557 COc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)F JFD02234 CN(C)/C=N/NC(=O)CC#N CD09173 c1cc2c(cc1S(=O)(=O)[O-])C(=O)C(CC2)S(=O)(=O)[O-].[Na+].[Na+] FM00335 COc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)Cl)F JFD02236 c1ccc(cc1)c2ccc(cc2)/C=C/3\C(=O)Nc4ccccc4S3 FM00343 CCc1cc2c(cc1O)oc(c(c2=O)c3nc4ccccc4n3C)C(F)(F)F JFD02282 COC(=O)c1c(ccs1)NC(=O)/C(=C/c2ccc[nH]2)/C#N GK00049 Cc1c(c(c(c(c1C)C)CNS(=O)(=O)c2ccc(cc2)F)C)C DP01225 Cc1ccc(cc1NC(=O)NN(C)C)NC(=O)NN(C)C DP01235 c1cc(ccc1c2nc(on2)CCCC(=O)O)Cl DP01236 c1ccc(cc1)n2c(c(cn2)C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N)C(F)(F)F GK01509 c1ccc2c(c1)c3ccccc3nn2 JFD00663 CS/C(=N/C#N)/NCc1c(cccc1Cl)Oc2ccccc2 CD11606 c1ccc(cc1)CNC2=CC(=O)CC(C2)c3ccc(cc3)Cl CD11611 CCOC(=O)CN1c2ccc(cc2C3(C1=O)OCCO3)Br JFD00788 Cc1ccc2c(c1)C(=O)C(=O)N2CC=C JFD00790 C1CSCCN1S(=O)(=O)c2c(c(sc2Cl)Cl)Br CD09580 c1cc(cnc1)CNc2c(cccn2)[N+](=O)[O-] CD09585 CN1C/C(=C\c2occc2)/C(=O)/C(=C/c3occc3)/C1 DP01041 CCOC(=O)n1cc(nc1SC(=O)OCC)c2cccc(c2)[N+](=O)[O-] FM00333 c1ccc2c(c1)-c3c(cc(nn3)c4cccc(c4)OC(F)(F)F)C2=O FM00338 CN1C/C(=C\c2ccccc2)/C(=O)/C(=C/c3ccccc3)/C1 DP00995 CCN(CC)c1ccc(c(c1)C)NC(=S)Nc2ccc(cc2)OC HR00187 c1ccc2c(c1)ncc3n2ccc3 HR00214 Cc1csc(c1Cl)C(=O)O/N=C(/c2ccc(cc2)C(C)(C)C)\N GK01380 Cc1csc(c1Cl)c2nc(no2)c3ccc(cc3)Cl GK01381 CC(=O)CSc1ccc(cc1[N+](=O)[O-])C(F)(F)F GK00132 Cc1csc(c1Cl)c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01382 Cc1csc(c1Cl)c2nc(on2)c3ccc(cc3)C(C)(C)C GK01383 c1ccc(c(c1)NC(=O)c2ccc(c(c2)Cl)Cl)n3cccc3 HR00211 COc1cccc(c1)NC(=S)Nc2ccccc2n3cccc3 HR00235 c1cc(ccc1/C(=N/OC(=O)c2c(ccs2)Cl)/N)C(F)(F)F GK01388 CN1C/C(=C\c2cc(c(cc2)OC)OC)/C(=O)/C(=C/c3cc(c(cc3)OC)OC)/C1 DP01044 CN1C/C(=C\c2c(cccc2)Cl)/C(=O)/C(=C/c3c(cccc3)Cl)/C1 DP01045 CCOC(=O)N[C@@H](Cc1ccccc1)C(=O)O JFD02322 c1ccc(cc1)CN2CCC(CC2)O JFD00694 CCCCNC(=N)N[N+](=O)[O-] JFD00695 Cc1cc2c(cc1Cl)c(=O)cc(o2)c3ccccc3 JFD02313 COC(=O)c1c(ccs1)NC(=S)Nc2cccc(c2)F GK00072 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3ccc(cc3)Cl)Cl CD11382 COC(=O)c1c(ccs1)NC(=S)Nc2ccccc2Cl GK00075 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccc(cc1)C)O JFD02269 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1Cl)O JFD02270 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccncc1)O JFD02271 CCOCCOC(=O)C(C)Oc1ccc(cc1)Oc2c(cc(cn2)Cl)Cl JFD02293 CCOC(=O)c1c(csc1NC(=O)CSc2ccc(cc2)Cl)C GK00144 CC1(CN=C(S1)N(C2CCCCC2)C(=O)Nc3cccc(c3)Cl)C JFD02273 CC1CN=C(S1)N(c2ccc(c(c2)Cl)F)C(=O)Nc3cccc(c3)Cl JFD02274 CC(c1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccc(cc3)C(C)C)/CC2)C DP01013 CN1c2ccccc2C(=O)N(CC1=O)C3CCCCC3 DP01016 c1c(cnc(c1Cl)/C=N/NC(=S)N)C(F)(F)F HC00071 CN(C(=S)N)/N=C/c1c(cc(cn1)C(F)(F)F)Cl HC00073 CC1(CC(C(N1)(C)C)C(=O)N)C JFD02327 c1ccc2c(c1)-c3ccccc3C2COC(=O)Nc4ccccc4C(=O)O JFD02331 CC/C(=C\N(C)C)/C(=O)c1c(cccc1F)F CD09732 Cn1c(nc(n1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)SC CD09733 Cc1c(sc(n1)C)c2ccn(n2)C(=O)NC(C)C CD09743 c1coc(c1)/C=C\2/C(=O)/C(=C/c3occc3)/CC2 DP00966 c1cc(ccc1/C=C/2\CCCC3C2=NNC3c4ccc(cc4)Cl)Cl DP00972 CN(c1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccc(cc3)N(C)C)/CCC2)C DP00976 CN(C)c1ccc(cc1)C2NC(=NN2)SC DP00986 Cc1c(sc(n1)C)c2ccn(n2)C(=O)Nc3c(onc3c4c(cccc4Cl)Cl)C CD09744 CCc1cnc(nc1c2c(cccc2F)F)/N=C/N(C)C CD09750 c1c(cc(c(c1/C=N\N=C(N)N)O)Cl)[N+](=O)[O-].Cl JFD00714 CC(=O)N1[C@@H]2C(OC(=O)C1C(S2)(C)C)[C@@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C JFD00716 c1cc(oc1C(=O)Nc2ccsc2C(=O)O)[N+](=O)[O-] GK00023 Cc1ccc(c(c1)[N+](=O)[O-])OCC2N(CCS2)S(=O)(=O)c3ccc(cc3)F FM00303 Cc1ccc(cc1)NC(=S)Nc2ccsc2C(=O)OC GK00076 CNc1ccccc1C(=O)NCCc2ccc(c(c2)OC)OC DP01017 COc1ccc(cc1OC)n2c(csc2=N)c3ccc(cc3)Cl.Cl DP01021 CN1C/C(=C\c2c3c(ccc2)cccc3)/C(=O)/C(=C/c4c5c(ccc4)cccc5)/C1 DP01026 CN(C(=O)c1ccc(cc1)Cl)/N=C/c2c(cc(cn2)C(F)(F)F)Cl HC00078 CSCCN/C(=N\C#N)/SC CD09825 CS/C(=N/C#N)/NCCSCc1c(cccc1Cl)Cl CD09826 CCOC(=O)C(C)Oc1ccc2c(cc(=O)oc2c1)c3ccccc3 JFD02371 CCOC(=O)COc1ccc2c(cc(=O)oc2c1)C JFD02376 COc1cc(c2c(=O)cc(oc2c1)c3ccccc3)O JFD02379 CCOc1cc(c2c(=O)cc(oc2c1)c3ccccc3)O JFD02380 c1ccc(cc1)c2ccc(cc2)/C=C(\C#N)/C(=O)N JA00025 CCOC(=O)c1c(csc1NS(=O)(=O)c2ccc(cc2)C)C GK00162 c1cnn2c1ncc(c2N)C#N GK00176 Cc1csc(c1Cl)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F GK01456 Cc1ccc(c(c1)C)NC(=S)NCCc2ccc(c(c2)OC)OC HR00016 CC(C)(C)N(CC(=O)OC)C(=O)c1ccccc1[N+](=O)[O-] FM00319 CC1(C(CCC1(C)C(=O)O)C(=O)OC)C JFD02357 C1CC2CC1CC2NC(=S)NN HR00050 COc1ccc(cc1OC)CCNC(=S)NC(=O)c2cccc(c2)[N+](=O)[O-] HR00061 CC(=O)C(=CNc1ccsc1C(=O)OC)C(=O)C GK00027 c1cc(c(cc1/C=C(\C#N)/C(=O)N)O)O JA00015 c1cc(ccc1/C=C(\C#N)/C(=O)N)O JA00019 c1ccc2c(c1)ccc(c2/C=C(\C#N)/C(=O)N)O JA00022 CNc1ccccc1C(=O)NCCc2ccccc2 DP01029 c1ccc(cc1)n2c(c(cn2)NC(=O)Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F GK01511 COC(=O)c1c(ccs1)NC(=O)CSCc2ccc(cc2)Cl GK00103 C#CCNS(=O)(=O)c1ccc(cc1)Cl CD11262 COc1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)OCC(F)(F)F CD11264 Cc1csc(c1C(=O)N)NC(=O)C(F)(F)F GK00205 CCc1cnc(nc1c2c(cccc2F)F)N/C=N/O CD09755 Cc1cn(nc1c2cccs2)C(=O)Nc3ccccc3 CD09757 c1cc(ccc1O)Oc2c(cc(cn2)Cl)Cl JFD02296 CCCCCOc1ccc2c(cc(=O)oc2c1)C JFD02301 C[C@]12CCC(=O)C=C1CCC2=O JFD02349 Cc1ccc(cc1)/C=N/N2C(=O)c3ccccc3C2=O JA00046 c1ccc2c(c1)C(=O)N(C2=O)/N=C/c3ccc(cc3)Cl JA00051 CCOC(=O)/C(=C/c1ccc(c(c1)OC)OC)/C#N JA00062 COC(=O)c1c(ccs1)NC(=O)CC(=O)C(F)(F)F GK00047 c1c(c(sc1Cl)Cl)S(=O)(=O)NCCCNS(=O)(=O)c2cc(sc2Cl)Cl CD09544 CC(c1[nH]c2ccccc2n1)OS(=O)(=O)c3ccc(cc3)Cl CD09583 CCCc1c(cnn1c2ccccc2)C(=O)O GK01501 c1cc(cc(c1)n2c(csc2=N)c3ccc(cc3)Cl)C(F)(F)F.Cl DP01011 CN1C/C(=C\c2cc3c(cc2)OCO3)/C(=O)/C(=C/c4cc5c(cc4)OCO5)/C1 DP01012 c1ccc(cc1)n2c(c(cn2)C(=O)O/N=C(/c3ccc(cc3)Cl)\N)C(F)(F)F GK01506 c1ccc(cc1)n2c(c(cn2)c3nc(no3)c4ccc(cc4)Cl)C(F)(F)F GK01507 CN1C/C(=C\C=C\c2ccccc2)/C(=O)/C(=C/C=C/c3ccccc3)/C1 DP01025 CNc1ccc(cc1C(=O)NCCc2ccc(c(c2)OC)OC)Cl DP01027 Cc1csc(c1Cl)C(=O)NNC(=O)c2cccs2 GK01457 CC(=O)Oc1ccc2c3ccccc3c(=O)oc2c1 JFD02304 c1cc(cc(c1)OCc2c(cccc2Cl)Cl)N3CCOCC3 CD09588 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)SCC(CSc3cccs3)O HAN00431 c1cc(c(cc1S(=O)(=O)NCCC#N)N)Cl JFD00649 Cn1cc(c(=O)n(c1=O)C)Br JFD00650 Cc1c(cnn1c2ccccc2)c3ccnn3C(=O)Nc4ccc(cc4)Cl CD09815 Cc1c(c(=O)c2ccc(cc2o1)O)c3ccc4c(c3)OCCO4 JFD02366 C/C(=N/NC(=O)c1ccccc1)/C(=O)O JFD02369 CC(=O)Oc1ccc2c(cc(=O)oc2c1)c3ccccc3 JFD02370 c1cc(c(cc1OS(=O)(=O)CS(=O)(=O)Oc2ccc(c(c2)Cl)Cl)Cl)Cl CD09821 c1ccc(cc1)n2c(c(cn2)C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N)C(F)(F)F GK01508 c1cc(ccc1c2cc(c(s2)C(=O)N)NC(=O)CSc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl GK01513 CC(CNC(=S)NC1CC2CCC1C2)O HR00057 CCC(CO)NC(=S)NC1CC2CCC1C2 HR00058 c1cc(cc(c1)[N+](=O)[O-])C(=O)NC(=S)Nc2c(cccc2Cl)Cl HR00062 c1cc(ccc1c2cc(=O)[nH]c(=O)o2)Cl CD11494 COc1ccc(cc1Br)C#N JFD00651 c1cc(cnc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)NCc2ccco2 JFD02228 CC(C)(C)c1cc2c(c(c1)Cc3cc(cc(c3O)Cc4cc(cc(c4O)Cc5cc(cc(c5O)Cc6cc(cc(c6O)Cc7cc(cc(c7O)C2)C(C)(C)C)C(C)(C)C)C(C)(C)C)C(C)(C)C)C(C)(C)C)O JFD00655 c1ccc(c(c1)C(=O)NCc2ccncc2)N DP00912 c1cc(c(c(c1)Cl)CO/N=C(/c2ccc(cc2)Cl)\N)F CD09661 c1ccc(c(c1)C(=O)NNC(=O)c2ccco2)N DP01072 CN(C)c1ccc(cc1)C(=O)NNC(=O)c2cc(ccc2N)[N+](=O)[O-] DP01073 c1ccc(cc1)CN2CC[NH+]=C2SCc3ccc(cc3)Cl.[Cl-] DP01078 c1cc(c(c(c1)Cl)CO/N=C(/c2ccc(cc2)Cl)\N/C=N/O)F CD09664 c1ccc(cc1)C(c2ccccc2)c3ccnn3C(=O)Nc4ccccc4 CD11433 CS/C(=N\N)/NC12CC3CC(C1)CC(C3)C2.I JFD00721 c1ccc(cc1)C(c2ccccc2)c3ccnn3C(=O)Nc4ccc(cc4)Cl CD11435 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)c4ccc(cc4)S(=O)(=O)Nc5ccc(cc5)C(F)(F)F)[N+](=O)[O-] GK01385 c1cc(ccc1/C(=N/OC(=O)c2c(ccs2)Cl)/N)Cl GK01387 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)F JFD02240 CC1CC(CC(C1)(C)C)NC(=O)c2ccccc2N DP00920 Cc1c(c(c(c(c1C)C)CS/C(=N/N)/N)C)C.Cl DP00921 c1ccc(cc1)C2CC(=CC(=O)C2)SCc3c(cccc3Cl)F CD11505 CSc1nnc(s1)SC2=CC(=O)CC(C2)c3ccccc3 CD11507 COc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)F JFD02246 CC1(OC(=O)C(C(=O)O1)(CC#C)CC#C)C CD11461 CC(C)(C)C(=O)CSC(=S)NCc1cccc(c1)OC CD11465 COc1cc(c(cc1OC)OC)/C=N/N=C(N)N JFD00740 c1cc(ccc1C2CC(=CC(=O)C2)Cl)C(F)(F)F CD11479 c1ccc(cc1)/C=N/N=C(N)N.[N+](=O)(O)[O-] JFD00743 Cc1cccc(c1)NC(=S)NC2CC3CC2C=C3 HR00070 c1ccc(cc1)CN(S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD11325 Cc1cc(cc(n1)NNC(=O)NC(=O)c2c(cccc2F)F)C(F)(F)F CD11327 Cc1ccc(cc1)Sc2c3ccsc3ncn2 GK02851 COc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccc2 JFD02243 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(=O)C)NC(=O)c2ccco2 JFD02259 COc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)Cl)F JFD02247 Cc1ccc(cc1)/C=N/Nc2c3ccsc3ncn2 GK02854 Cc1ccnc(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2OC JFD02248 Cc1csc(c1NC(=O)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)OC GK01330 CCCc1c(cnn1c2ccccc2)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01530 CC1CC(CC(C1)(C)C)NC(=S)NC2CC3CC2C=C3 HR00090 c1ccc(cc1)CC(c2ccccc2)NC(=S)NC3CC4CC3C=C4 HR00091 CC(C)(CCO)NC(=S)NC1CC2CC1C=C2 HR00095 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3)F GK01533 Cc1cc2c(cc(=O)oc2cc1C)O JFD02339 Cc1ccc(cc1)C(=O)C#Cc2ccccc2 JFD02342 CC(C)c1ccc(cc1)NC(=S)NC2CC3CC2C4C3CC=C4 HR00109 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C(=O)C)NC(=O)c2ccccc2OC JFD02262 CCN(CC)/C(=N/C(=O)c1c(cccc1Cl)Cl)/SC EN00034 CC1CCCN(C1)/C(=N/C(=O)c2c(cccc2Cl)Cl)/SC EN00040 c1cc(cnc1)NC(=O)c2cc(sc2Cl)Cl CD09470 CN(C)c1cccc(c1CNC(=O)Nc2ccc(cc2)Cl)N(C)C CD09477 Cc1ccc(cc1)CS/C(=N/N)/N.Cl DP00932 CC(C)(C)c1ccc(cc1)c2nnnn2Cc3c(cccc3Cl)Cl GK02991 C1COCCN1C(=N)N.Br DP00942 COc1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccc(cc3)OC)/CCC2 DP00949 Cc1c(c(n(n1)C)Sc2ncccn2)[N+](=O)[O-] CD11599 Cc1c(c(n(n1)C)Sc2ccc(cn2)C(F)(F)F)[N+](=O)[O-] CD11600 Cc1ccc(cc1)NC(=O)N2c3ccccc3C4(C2=O)OCCO4 JFD00781 c1ccc(cc1)CCNC(=S)NC2CC3CC2C=C3 HR00087 c1ccc2c(c1)C(=O)N(C2=O)/N=C/c3ccc4c(c3)OCO4 JA00044 c1ccc2c(c1)C(=O)N(C2=O)/N=C/c3cc(ccc3O)Br JA00045 CNC(=O)NCc1c(cccc1N(C)C)N(C)C CD09478 c1cc2cccc3c2c(c1)NC(=N3)N.Cl JFD00690 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NCc3c(cccc3N(C)C)N(C)C CD09479 Cc1ccsc1/C=C/c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01453 c1c(c(sc1Cl)Cl)S(=O)(=O)N2CCOCC2 CD09483 c1ccc(cc1)CC2(CCNCC2)O JFD00691 c1ccc(cc1)c2ccc(cc2)c3cnc(o3)c4ccc(cc4)c5ccccc5 JFD00693 CN(C)/C=N/S(=O)(=O)c1cc(sc1Cl)Cl CD09538 c1csc(c1)/C=C\2/C(=O)/C(=C/c3sccc3)/CC2 DP00989 Cc1[nH]c(=O)c2c3c(sc2n1)CCC3 GK00066 Cc1c(sc(c1C(=O)c2cccs2)N)C GK00067 Cc1ccc(c(c1)C)NC(=S)NC2CC3CC2C=C3 HR00088 C1C2CC(C1C=C2)NC(=S)NNCCO HR00096 CN(C)CC[C@H](c1ccc(cc1)Cl)c2ccccn2.C(=C/C(=O)O)\C(=O)O JFD02347 COC(=O)c1c(ccs1)NC(=S)Nc2cccc(c2)C(F)(F)F GK00074 C1C=CC2C1C3CC2C(C3)NC(=S)NN HR00102 Cc1cc(cc(n1)NNC(=O)NC(=O)c2c(cccc2Cl)F)C(F)(F)F CD11352 CC12CCC(=O)C=C1NC(=O)CC2 CD11356 Cc1csc(c1Cl)C(=O)NNC(=O)c2ccco2 GK01458 Cc1csc(c1Cl)C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01461 c1ccc(cc1)C(c2ccc(cc2)Cl)N3CCNCC3 JFD00624 c1cc(c(cc1C2CC(=O)CC(=O)C2)Cl)Cl CD11332 CC1CC(CC(C1)(C)C)NC(=O)c2ccccc2NC DP01001 CC(C)c1[nH]c2ccccc2n1 DP01004 Cc1c(c(sc1C#N)c2nc[nH]n2)C CD11566 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(C)C(C)(C)C CD11571 c1cc(ccc1S(=O)(=O)NNC(=O)c2c(nccn2)N)Cl HAN00445 Cc1csc(c1Cl)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01356 COC(=O)CSCC(=O)Nc1ccsc1C(=O)OC GK00100 Cn1ccc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl GK01366 CCOC(=O)c1c(csc1N)c2cccs2 HAN00443 CC1CN=C(S1)N(C2CCCCC2)C(=O)Nc3cccc(c3)Cl JFD02275 c1cc(c(c(c1)Cl)SCc2c(cc(cn2)C(F)(F)F)Cl)Cl HC00024 CCOC(=O)c1c(csc1N)c2ccco2 HAN00451 CCc1cc2c(cc1O)occ(c2=O)c3[nH]c4ccccc4n3 JFD02276 c1ccc(cc1)C(=O)OCC2C(C(C(O2)n3c(=O)nc(cn3)N)O)O JFD02279 CC(=O)CCS(=O)(=O)c1ccccc1 FM00330 Cc1ccc(cc1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2OC JFD02244 Cc1cccc(n1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2OC JFD02245 COc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccn2 JFD02249 Cc1c(nc(nn1)SCc2cc(cc(c2)Br)Br)O CD09698 Cc1ccccc1C2=NC(N=C(O2)N(C)C)(C(F)(F)F)C(F)(F)F JFD02253 Cc1ccccc1C2=NC(N=C(O2)N=C(SC)SC)(C(F)(F)F)C(F)(F)F JFD02256 Cc1c(=O)nc([nH]n1)SCc2c(cccc2Cl)F CD09699 CCOC(=O)C(C(F)(F)F)(Nc1cc(ccn1)C)NC(=O)c2ccco2 JFD02258 c1cc(c(cc1)Cl)/C=C\2/C(=O)/C(=C/c3c(cccc3)Cl)/CC2 DP00973 CN(c1cc(c(cc1)/C=C\2/C(=O)/C(=C/c3c(cc(cc3)N(C)C)Cl)/CCC2)Cl)C DP00975 CN1C/C(=C\c2ccc(cc2)Cl)/C(=O)/C(=C/c3ccc(cc3)Cl)/C1 DP00990 c1ccc(cc1)C2Nc3ccccc3-c4n2c5ccccc5n4 DP01269 c1ccc(c(c1)C2Nc3cc(ccc3O2)Cl)Cl DP01279 c1ccc2c(c1)cccc2C3Nc4ccccc4O3 DP01282 c1cc(cc(c1)C(F)(F)F)C(=O)ON=C2CCCCCCCCCCC2 JFD00758 Cc1ccc2c(c1)cc3c(n2)c4c(n(c3=O)C)n(c(=O)n(c4=O)C)C JFD00845 c1ccc(c(c1)C(=O)O)Sc2cccc(c2)C(F)(F)F JFD00824 c1ccc(cc1)SCCC(=O)O JFD00825 CNC(=O)c1ccccc1SCCC(=O)O JFD00831 c1ccc(cc1)Oc2cccc(c2CNC(=O)Nc3ccc(cc3)Cl)Cl CD11609 c1ccc(cc1)Oc2cccc(c2CNc3[nH]nc(n3)N)Cl CD11612 CNC(=S)Nc1ccccc1n2cccc2 HR00237 COc1ccc(c(c1)OC)/C=C(\C#N)/C(=O)N JA00014 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O GK01547 c1cc(ccc1n2c(c(cn2)C(=O)O)C(F)(F)F)Cl GK01550 CCCc1c(cnn1c2ccccc2)C(=O)O/N=C/c3ccc(cc3)C#N GK01553 CCOC(=O)c1c[nH]c(=S)nc1C(F)(F)F GK01626 CCCc1c(cnn1c2ccc(cc2)Cl)NC(=O)Nc3ccc(cc3)F GK01561 Cc1c(cnn1c2ccccc2)c3ccnc(n3)N CD09797 c1csc(c1Cl)C(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N GK01389 c1ccc(c(c1)NC(=S)Nc2ccccc2Cl)n3cccc3 HR00236 c1cc(ccc1C(F)(F)F)NS(=O)(=O)c2ccc(cc2)N3C(=O)C=CC3=O GK01394 CCOC(=O)/C(=C/Nc1cscc1C)/C#N GK01410 CC(=O)c1c(ccs1)N2C(=O)CCC2=O GK01414 Cc1ccccc1C(=O)NC(C(=O)OC)(C(F)(F)F)O JFD02265 Cc1c(sc(n1)C)c2cnc(nc2)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD09803 Cc1c(cnn1c2ccccc2)c3ccnn3C(=O)Nc4ccccc4 CD09804 COc1ccccc1NC(=O)N JA00157 c1cc(ccc1/C(=N/N)/N)Cl.I DP01096 CCOC(=O)/C(=N/Nc1ccsc1C(=O)OC)/C#N GK00211 Cc1ccc(cc1)/C(=C/2\C=C/C(=N\O)/C(=C2Cl)Cl)/C#N JA00111 Cc1ccc(cc1)/C(=C/2\C=C/C(=N\O)/C(=C2)Cl)/C#N JA00113 COc1ccc(cc1)/C(=C/2\C=C(/C(=N/O)/C=C2Cl)Br)/C#N JA00115 CCCc1c(cnn1c2ccccc2)C(=O)Sc3ccc(cc3)Br GK01610 CSc1cc(nn1S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3ccc(cc3)F GK01618 c1cc(cc(c1)[N+](=O)[O-])C2NC(=NN2)c3ccc(cc3)Cl DP01119 Cc1csc(c1NC(=O)c2ccc(cc2)Cl)C(=O)OC GK01395 Cn1cnc(c1C#N)n2oo2 JFD02280 Cc1csc(c1C#N)NC(=O)C(F)(F)F GK00149 c1ccc(cc1)c2c3ccccn3c(n2)c4ccc(cc4)I JFD02285 CN(C)c1cccc(c1CNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)N(C)C CD09729 Cn1c(nc(n1)NS(=O)(=O)c2cc(sc2Cl)Cl)SC CD09730 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Nc2nc(n(n2)C)SC CD09731 CCCc1c(cnn1c2ccccc2)c3nc(no3)c4ccc(cc4)Cl GK01540 Cc1csc(c1C(=O)N)NC(=O)CSc2ccc(cc2)Cl GK00215 c1ccc(cc1)c2c(nnc(n2)c3ccc(cc3)Cl)c4ccccc4 DP01101 c1ccc2c(c1)c(=O)n(c(n2)S)NC(=O)c3ccco3 DP01109 CCOC(=O)c1c(csc1NC(=O)C(Cl)(Cl)Cl)C GK00125 COC(=O)c1c(ccs1)NC(=O)c2ccccc2Cl GK00219 COC(=O)c1c(ccs1)NC(=O)c2cccs2 GK00224 COC(=O)c1c(ccs1)NC(=O)c2c(cccc2F)F GK00226 c1cc(ccc1C2=NNC(N2)c3ccc4c(c3)OCO4)Cl DP01121 CC\1(c2ccccc2N(/C1=C\C(=O)c3ccccc3)C)C JFD02286 CCCc1c(cnn1c2ccccc2)C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N GK01537 c1ccc(cc1)c2c(nc(s2)c3ccccc3)n4ccc(=S)[nH]c4=O JFD02423 c1ccc(cc1)c2c(nc(s2)c3ccccc3)n4ccc(nc4=O)N5CCCCC5 JFD02426 CCCc1c(cnn1c2ccccc2)C(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N GK01539 c1c(c(=O)[nH]c(=O)[nH]1)NCCO JFD02430 Cc1ccc2c(c1)c(cc(=O)o2)O JFD02341 CCOC(=O)c1c(csc1NC=C(C#N)C#N)C GK00129 CC(C(=O)O)Oc1ccc2c(cc(=O)oc2c1)c3ccccc3 JFD02372 CN(C)c1cccc(c1CNC(=O)c2ccccc2Cl)N(C)C CD09735 CN(C)c1cccc(c1CNC(=O)c2ccccc2F)N(C)C CD09736 CCc1c[nH]nc1c2c(cccc2F)F CD09751 CC(C(C)(C)C)NS(=O)(=O)c1cccc(c1)C(F)(F)F CD11570 Cc1c(c(nc(n1)OC)OC)[N+](=O)[O-] JFD02428 CC(=O)Nc1ccccc1C(=O)NN DP01060 CC1CNC(=N1)SCc2ccc(cc2)Cl.Cl DP01061 CC1CNC(=N1)SCc2ccccc2.Cl DP01064 c1ccnc(c1)SC/C(=N/OCc2c(cccc2Cl)Cl)/N CD09649 c1cc(ccc1NC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)Cl GK01566 CN(C)c1cccc(c1CNS(=O)(=O)c2cc(sc2Cl)Cl)N(C)C CD09726 CN(C)c1cccc(c1CNC(=O)C(Cl)(Cl)Cl)N(C)C CD09737 CC(C)(C)C(=O)NCc1c(cccc1N(C)C)N(C)C CD09738 c1ccc(cc1)C(=O)N2c3ccccc3OC2c4ccc5c(c4)OCO5 DP01170 Cn1c2c(c(cc(=O)n2c3ccccc3)NCc4ccccc4)c(=O)n(c1=O)C JFD02456 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)c3ccn(n3)c4ccc(cc4)Cl CD11548 c1cc(ccc1c2nc(cs2)c3ccc(cc3)Br)Cl.Br HR00111 CN(C)/C=C(\C#N)/c1nc(cs1)c2ccc(cc2)Cl CD09652 Cn1c(c(cn1)c2nc(cs2)c3ccc(cc3)Cl)N CD09658 c1ccc2c(c1)C(=O)N(C2=O)c3ccc4c(cc(=O)oc4c3)C(F)(F)F GK01459 Cc1c(c(no1)c2ccccc2)C(=O)SCC(=O)C GK00192 c1cc(nn2c1nnc2)N3CCSCC3 GK00201 Cn1c(nc(n1)NS(=O)(=O)c2ccc(cc2F)F)SC CD09734 COc1cc(ccc1O)/C=N/NC(=O)c2ccccc2N DP01156 c1cc(ccc1c2ncon2)Cl DP01166 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=O)c2ccccc2N DP01163 c1c2c(c(n[nH]2)N)c(nc1O)O JA00082 CN(C)c1ccc(cc1)C2Nc3ccccc3O2 DP01231 CN(C)c1ccc(cc1)C2Nc3cc(ccc3O2)Cl DP01232 CCC(C)(C)NC(=O)Nc1ccc(c(c1)NC(=O)NC(C)(C)CC)C DP01234 Cc1csc(c1C#N)N GK00146 c1cc2c(cc1c3coc4cc(ccc4c3=O)O[C@H]5[C@H]([C@@H]([C@H]([C@@H](O5)CO)O)O)O)OCCO2 JFD02375 CCOC(=O)C(C)Oc1ccc2c(cc(=O)oc2c1)C JFD02377 Cc1c(sc(n1)C)c2ccn(n2)C(=O)Nc3ccc(cc3)Cl CD09741 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(c(cs2)C)Cl GK01462 Cc1nc2cc(c(cc2s1)O)O JFD02289 c1ccc(c(c1)n2c(csc2=N)c3ccc(cc3)Cl)F.Cl DP01008 CSc1cccc(c1)n2c(csc2=N)c3ccc(cc3)Cl.Cl DP01009 Cc1ccc2c(c1)/C(=N/N)/C(=O)N2 JA00084 c1ccc(cc1)N\2C(=O)CS/C2=C\C(=O)c3ccc(cc3)Cl JFD00755 c1cc(ccc1C(=O)CC(=O)N)F CD11531 c1ccc2c(c1)ccc(n2)/N=N/c3ccc4ccccc4n3 JFD02394 CN(C)c1cccc(c1CNC(=O)NC(=O)c2c(cccc2Cl)Cl)N(C)C CD09712 c1ccc(cc1)/C(=C\2/C(=O)C(=O)N(C2=S)c3ccc(cc3)Cl)/Nc4ccc(cc4)Cl JFD00749 c1ccc(cc1)n2c(c(cn2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F GK01495 c1ccc2c(c1)ncn2CN3CCCCC3 JFD02364 Cc1c(sc(n1)C)c2cnc(nc2)NS(=O)(=O)c3ccc(cc3)Cl CD09802 CCCc1c(cnn1c2ccc(cc2)Cl)NC(=O)Nc3ccc(cc3)OC(F)(F)F GK01562 CN(C)c1cccc(c1CN/C(=N\C#N)/SC)N(C)C CD09807 C/C(=N/OS(=O)(=O)c1ccccc1)/c2nccs2 CD11518 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)c3ccnc(n3)N CD11521 CC(C)(C)c1cc(nc(n1)N)C(F)(F)F JFD02396 Cc1csc(c1C(=O)N)N GK00199 C#CCC1(C(=O)c2ccccc2C1=O)c3ccccc3 JFD02399 c1ccc(cc1)C2(C(=O)c3ccccc3C2=O)[N+](=O)[O-] JFD02401 Cc1ccc(cc1)S(=O)(=O)NC(=S)NNC(C)(C)C JFD00713 c1ccc(cc1)C2C(=O)c3cc4ccccc4cc3C2=O JFD02402 c1cc(cc(c1)Cl)NN=C(C#N)C#N JFD00702 CCC(=O)C1C(=O)c2ccccc2C1=O JFD02403 C1CCCC23CC(=O)CC2(CC1)CC(=O)C3 JFD02406 COC(=O)c1c(ccs1)NC(=O)/C(=C/c2ccc(s2)[N+](=O)[O-])/C#N GK00050 CCOc1ccccc1NC(=S)NC2CC3CCC2C3 HR00082 c1ccc(cc1)C2(CC(=O)c3c2cccc3)c4ccccc4 JFD02390 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)SC/C(=N/O)/C GK00188 Cc1csc(c1C#N)/N=C/N(C)C GK00197 c1c2c(cc(c1Cl)S(=O)(=O)N)S(=O)(=O)NCN2 JFD00715 c1ccc2c(c1)N(C(O2)c3ccc(c(c3)Cl)Cl)S(=O)(=O)c4ccc(cc4)Cl DP01193 c1cc(cc(c1)[N+](=O)[O-])n2c(csc2=N)c3ccc(cc3)Cl.Cl DP01197 COc1ccc(cc1)C2Nc3ccccc3O2 DP01198 C1COCCN1C(=S)NC2CC3CC2C=C3 HR00072 C1CCC(CC1)NC(=S)NC2CC3CC2C=C3 HR00073 c1ccc(cc1)C(c2ccccc2)c3ccnn3S(=O)(=O)c4ccccc4 CD11437 c1ccc2c(c1)C=Cc3ccccc3N2 JFD00728 CC(C)c1ccc(cc1)NC(=S)NC2CC3CC2C=C3 HR00085 CN(C)/C=C/C(=O)c1ccc(cc1)Oc2cccc(c2C#N)Cl CD11445 c1ccc(cc1)C(c2ccccc2)c3ccnn3S(=O)(=O)C(F)(F)F CD11449 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)c3ccn[nH]3 CD11451 Cc1ccc(cc1)N(C(CC(=O)C2CC2)c3ccccc3)C(=O)Nc4ccccc4Cl JFD02413 c1cc(c(cc1C2Nc3cc(ccc3O2)Cl)Cl)Cl DP01188 c1ccc2c(c1)N(C(O2)c3ccc(c(c3)Cl)Cl)S(=O)(=O)c4ccccc4[N+](=O)[O-] DP01192 c1ccc2c(c1)[nH]c(n2)c3cc(ccc3N)Cl DP01275 c1ccc(c(c1)C2Nc3ccccc3O2)Cl DP01278 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C(=N/OC(=O)/C=C/c2cc(sc2)[N+](=O)[O-])/N GK01668 Cc1ccc(cc1)S(=O)(=O)NNc2c3c(c(cs3)C)ncn2 GK01671 CC(=O)OCC1=C(N2C(C(C2=O)NC(=O)[C@H]([C@@H]([C@@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)SC1)C(=O)O JFD00725 COc1ccc(cc1OC)CCNC(=S)NC2CC3CC2C=C3 HR00068 C1CCCCCC(CCCCC1)NC(=S)NC2CC3CC2C=C3 HR00069 c1ccc(cc1)n2c(c(cn2)C(=O)Sc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F GK01518 CCOc1ccc(cc1)NC(=S)NC2CC3CC2C=C3 HR00081 CC1CCCN(C1)C(=S)NC2CC3CCC2C3 HR00083 COc1ccc(cc1)C2Nc3cc(ccc3O2)Cl DP01199 Cc1c(c(c(c(c1C)C)CCN)C)C.Cl DP01200 Cc1cc(c(cc1CO)CO)C JFD02450 c1cc(ccc1/C(=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)/N)Cl GK01573 Cc1ccc2c(c1)c3c([nH]2)nc4ccccc4n3 JA00031 COC(=O)c1ccccc1NC(=O)CC#N GK00171 c1ccc2c(c1)C(=O)N(C2=O)/N=C/c3ccc(cc3)[N+](=O)[O-] JA00035 CN(C)c1ccc(cc1)/C=N/N2C(=O)c3ccccc3C2=O JA00036 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N GK01583 c1ccc(cc1)C2=C(C(=O)C(=O)N2)C(=O)Nc3ccc(cc3)Br JFD00731 c1ccc(cc1)n2c(c(cn2)C(=O)O/N=C/c3c(cccc3Cl)F)C(F)(F)F GK01520 COc1c(=O)c2ccccc2oc1c3ccccc3 JFD02348 CCCCCCCCCCCOS(=O)(=O)C JFD02354 CCc1cc(c(s1)NC=C(C(=O)OCC)C(=O)OCC)C(=O)OCC GK00092 Cc1ccc(cc1)SCC(=O)Nc2ccsc2C(=O)OC GK00101 CCCc1c(cnn1c2ccccc2)NC(=O)Nc3ccc(cc3)OC(F)(F)F GK01528 Cc1cc(nc(n1)N)OC(F)F JFD00775 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3ccc(cc3Cl)Cl JFD00778 c1ccc(cc1)NC(=O)Nn2cnnc2 JFD00779 CC(=O)CC1(c2ccccc2N(C1=O)Cc3ccccc3)O JFD00780 c1cc(ccc1/C=C(\C#N)/C(=O)N)[N+](=O)[O-] JA00016 Cc1ccc(cc1)/C=C(\C#N)/C(=O)N JA00017 c1cc(ccc1/C(=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)/N)C(F)(F)F GK01575 c1cc(ccc1c2csc(=N)n2c3cc(ccc3Cl)Cl)Cl.Cl DP01083 COc1cc(cc(c1OC)OC)C(=O)NN JFD00733 c1ccc2c(c1)C(=O)N(C2=O)/N=C/c3cc(cc(c3O)Cl)Cl JA00041 COc1cc(ccc1O)/C=N/N2C(=O)c3ccccc3C2=O JA00042 COc1ccc(cc1OC)CS(=O)(=O)c2ccccc2C(=O)OC JFD00817 COc1ccc(cc1OC)C(=O)CC(=O)Nc2ccccc2 JFD00818 c1ccc(cc1)n2c(c(cn2)C(=O)Sc3ccccn3)C(F)(F)F GK01524 c1cc2c(cc1[N+](=O)[O-])OCCOCCOc3ccc(cc3OCCOCCO2)[N+](=O)[O-] JFD02355 c1csc(c1)/C=C\2/C(=O)/C(=C/c3sccc3)/CCC2 DP00958 CCc1cc2c(cc1c3cc(c4cc(ccc4n3)Cl)c5ccccc5)C(CCC2(C)C)(C)C HR00145 c1ccc(cc1)c2c3cc(ccc3nc4c2CCCCCCCCCC4)Cl HR00146 CCOC(=O)C(/C=N/Nc1ccccc1)C(=O)OCC JFD00727 c1cc(cnc1)C(=O)NNC(=S)Nc2c(cc(cc2Cl)Cl)Cl JFD00730 CC1=C(S(=O)(=O)C(C(C1)c2ccc(cc2)OC)C#N)C#N CD11649 c1cc(c(c(c1)Cl)/C=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)F GK01602 CCCc1c(cnn1c2ccccc2)C(=O)Sc3ccc(cc3)Cl GK01608 Cc1ccc(cc1)S(=O)(=O)n2c(cc(n2)c3ccc(cc3)F)SC GK01614 CCCc1c(cnn1c2ccccc2)NC(=O)Nc3ccc(cc3Cl)Cl GK01529 Cc1ccc2c(c1)/C(=N\N=C\c3ccc(cc3)[N+](=O)[O-])/C(=O)N2 JA00091 c1ccc(cc1)c2cc(nc3c2cc(cc3)Cl)c4ccc5c(c4)OCO5 HR00139 c1ccc2c(c1)C(=O)N(C2=O)c3c(c4c(s3)CCCC4)C#N GK01344 CCc1cc(c(s1)NC(=O)CC#N)C(=O)OCC GK00091 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C/c3ccc(cc3)C#N GK01604 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C/c3c(cccc3Cl)F GK01606 c1ccc(cc1)n2c(c(cn2)C(=O)O/N=C/c3ccc(cc3)C#N)C(F)(F)F GK01521 c1ccc(cc1)n2c(c(cn2)C(=O)O/N=C/c3ccc(cc3Cl)Cl)C(F)(F)F GK01522 Cc1ccc2c(cc(nc2c1)c3ccc4c(c3)OCO4)C(=O)O JA00106 Cc1ccc2c(c1)/C(=N\N=C\c3ccc(cc3)Cl)/C(=O)N2 JA00092 c1ccc2c(c1)/C(=N\N=C\c3cc(ccc3O)Br)/C(=O)N2 JA00094 Cn1ccc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01371 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cc(on2)C JFD02241 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C(F)(F)F JFD02242 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C/c3ccc(cc3)OC GK01603 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C/c3ccc(cc3)F GK01605 CSc1cc(n[nH]1)c2ccc(cc2)F GK01607 Cc1c(cnn1c2ccccc2)C(=O)C CD09766 C1C2CC3CC(C2)(CC1C3=O)O JFD02336 Cc1ccc(cc1)CSC2=NCCN2.Cl DP01046 c1ccc(cc1)CSC2=NCCN2.Cl DP01047 CCOC(=O)C(C(F)(F)F)(NCc1ccco1)NC(=O)c2ccco2 JFD02260 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)Cl)NC(=O)c2ccco2 JFD02263 CN(C)c1cccc(c1CNC(=O)NC(=O)c2c(cccc2F)F)N(C)C CD09713 c1cc(sc1)CN2CC(CN(C2)Cc3cccs3)C#N CD11500 COc1ccc(c(c1)/C(=N/O)/N)OC DP01210 CSc1[nH]c2ccccc2n1.I DP01217 c1ccc(cc1)n2c(c(cn2)C(=O)O)C(F)(F)F GK01493 Cc1c(sc(n1)C)c2ccnc(n2)N/C=N/O CD09767 Cc1ccc2c(c1)c(=O)cc(o2)c3ccccc3 JFD02329 CCOC(=O)NNC(=O)NC JFD02334 Cc1c(sc(n1)C)c2ccnc(n2)c3ccc(cc3)Cl CD09768 c1ccc(cc1)N2C(=O)C(=O)/C(=C(\c3ccc(cc3)Cl)/O)/C2=S JFD00752 CCCc1c(cnn1c2ccc(cc2)Cl)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F GK01586 c1ccc(cc1)Cn2cc[nH]c2=O JFD01640 c1cc(c(c(c1)Cl)C(=O)N2CCC(CC2)NC(=O)C3CCCCC3)Cl JFD02515 CN(/C=C/C=C/C=C(C#N)C#N)c1ccccc1 JFD00044 CCOC(=O)C(c1c2ccccc2n(c(=O)c1[N+](=O)[O-])c3ccccc3)C(=O)OCC JFD00854 c1ccc(c(c1)c2ccccc2Sc3ccccc3C(=O)O)[N+](=O)[O-] JFD00834 CCCc1c(cnn1c2ccccc2)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F GK01541 CC(=O)c1ccccc1Sc2ccccc2C(=O)O JFD00837 c1ccc(c(c1)S(=O)(=O)NCC(=O)O)I JFD00838 c1cc(c(cc1[N+](=O)[O-])I)S(=O)(=O)NCC(=O)O JFD00839 Cc1ccc(cc1)CSC2=NC(CN2)C.Cl DP01056 Cc1ccc(cc1)CSc2[nH]c3ccccc3n2.Cl DP01066 c1ccc2c(c1)[nH]c(n2)SCc3ccc(cc3)Cl.Cl DP01076 CC1=C(S(=O)(=O)C(C(C1)c2ccccc2)C#N)C#N CD11635 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)C3CCCCC3 JFD02518 Cc1ccc(cc1)S(=O)(=O)N2CCN=C2SC DP01315 Cc1c(cnn1c2c(cc(cc2Cl)Cl)Cl)C(=O)C CD09772 CSC1=NCCN1S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DP01319 COCCCN1CNC(=NC1)SCc2cccc(c2)C#N.Br DP01320 CSC1=NCCCN1S(=O)(=O)c2ccc(cc2)Cl DP01325 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccsc2C(=O)OC GK00225 CCOC(=O)c1cn(nc1N)c2ccc(nn2)N3CCC(CC3)C GK00228 c1cc(ccc1/C(=C/2\C=C/C(=N\O)/C(=C2)Br)/C#N)Cl JA00136 c1cc(ccc1/C(=C/2\C=C/C(=N\O)/C(=C2)Cl)/C#N)Cl JA00138 Cc1ccc2c(c1)cc3c(n2)n(c(=O)n(c3=O)C)C JFD00841 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)c4ccccc4 GK01544 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)OCC GK01545 Cc1ccc(cc1)S(=O)(=O)Oc2cc(=O)n(c3c2c(=O)n(c(=O)n3C)C)C JFD00843 Cn1c2c(c3c(c1=O)cc4ccccc4n3)c(=O)n(c(=O)n2C)C JFD00844 CCC(C)Nc1c(c(ncn1)N)[N+](=O)[O-] JFD02418 Cn1c2c(c3c(c1=O)cc4cc(ccc4n3)[N+](=O)[O-])c(=O)n(c(=O)n2C)C JFD00860 c1cc(ccc1C2CC(=CC(=O)C2)OC(=O)c3ccc(cc3)Cl)Cl CD11632 CC(=O)C1C(=O)CC(CC1=O)c2ccc(cc2)Cl CD11633 CN(c1cccc(c1C#N)F)NC2c3ccc(c(c3C(=O)O2)OC)OC CD11642 c1cc2c(cc1[N+](=O)[O-])OCCOCCOc3cc(ccc3OCCOCCO2)[N+](=O)[O-] JFD02356 CC1(C(CCC1(C)C(=O)OC)C(=O)O)C JFD02358 CC(/C=N/N1C(=O)c2ccccc2C1=O)c3ccccc3 JA00054 COc1ccc(c(c1)OC)/C=C(\C#N)/c2cccc(c2)Cl JA00141 c1cc(cc(c1)Cl)/C(=C/c2ccc(cc2Cl)Cl)/C#N JA00142 CCc1cc2c(ncnc2s1)OC(=O)N(C)C GK00232 CCOC(=O)c1c(csc1NC(=O)c2cccs2)C GK00237 COc1ccc(cc1)/N=c\2/c(c(ss2)SC)c3ccccc3 JA00146 Cc1ccc(cc1)NC(=O)N JA00151 c1ccc(cc1)C(C(=O)O)Sc2ccccc2C(=O)O JFD00813 COc1ccc(cc1OC)c2ccc3ccccc3n2 JFD00820 Cc1nc2ccccc2n1C3CC(=O)N(C3=O)c4ccccc4 DP01255 c1ccc(cc1)NC(=S)Nc2ccccc2c3[nH]c4ccccc4n3 DP01260 c1ccc(cc1)Oc2ccc(cc2)c3ccn[nH]3 CD11757 c1cc(c(c(c1)Cl)CSC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)F GK01593 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)Sc3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01596 C/C(=N\NC(=S)NC)/c1ccccc1 DP01126 CCOC(=O)c1c(csc1NC(=O)c2ccc(cc2)C(C)(C)C)C GK00236 C/C(=N\NC(=S)NC)/c1ccc(cc1)OC DP01128 C/C(=N\NC(=S)NC)/c1ccc(cc1)F DP01129 CCOC(=O)/C(=C/c1ccc(c(c1)Cl)Cl)/C#N JA00065 CCOC(=O)/C(=C/c1cccc(c1OC)OC)/C#N JA00063 CCOC(=O)/C(=N\Nc1ccsc1C(=O)OC)/C(=O)C GK00209 CSC(=N)c1ccc(cc1)Cl.I DP01090 c1ccc(c(c1)c2[nH]c3ccccc3n2)N DP01095 c1ccc(c(c1)F)S(=O)(=O)CCC#N CD11744 c1ccc(cc1)c2c(cn(n2)c3ccccc3)CC#N JFD00043 c1ccc(cc1)COCC(CN2CCOCC2)O.Cl JFD02490 COc1cc(cc(c1OC)OC)C2N=C(SC(=N2)c3ccc(cc3)Cl)c4ccc(cc4)Cl DP01506 c1cc(ccc1CC2=NC(=O)C(S2)CC(=O)O)Cl DP01529 Cc1c(c(nc(n1)O)O)[N+](=O)[O-] JFD02429 Cn1ccc(n1)NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N GK00344 Cn1ccc(n1)NC(=O)/C(=C/c2ccc(cc2)Cl)/C#N GK00345 Cn1cc(c(n1)NC(=O)c2ccc(c(c2)Cl)Cl)Br GK00350 c1ccc2c(c1)ccc(n2)C(=O)c3ccccn3 JFD02387 CC1CN(CC(O1)C)C(=N)c2ccc(cc2)Cl.I DP01145 C/C(=N\NC(=S)NC)/c1cccc(c1)[N+](=O)[O-] DP01130 Cc1c(c(c(c(c1C)C)CSC2=NC(CN2)C)C)C.Cl DP01136 Cc1nc2ccccc2n1C3CC(=O)N(C3=O)c4ccc(cc4)F DP01256 COc1ccc(cc1Br)Br DP01258 c1ccc(cc1)/C(=C/2\C(=O)C(=O)N(C2=S)c3ccc(cc3)Cl)/O JFD00751 Cn1cc(c(n1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br GK00328 CCOC(=O)/C(=C/Nc1ccn(n1)C)/C#N GK00332 Cn1ccc(n1)NC(=O)/C(=C/c2cc(cs2)Br)/C#N GK00343 CSc1ccn(c(=O)n1)c2c(sc(n2)c3ccccc3)c4ccccc4 JFD02424 c1cc(cnc1)c2nc(cs2)c3ccc(cc3)Cl.Br DP01358 Cc1ccc(cc1Cl)NC(=O)N JA00158 Cc1ccc(cc1)n2c(c(cn2)c3n[nH]nn3)N CD11812 CSc1[nH]c(=O)n2c(n1)ccn2 GK00213 CCOC(=O)/C(=C/c1ccc(c(c1)Br)OC)/C#N JA00078 CCOC(=O)/C(=C/c1cccc2c1cccc2)/C#N JA00079 Cc1ccc(cc1Cl)NC(=O)/C=N/O JA00080 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCCc3ccc(cc3)OC JFD01669 c1cc(cc(c1)SCCC(=O)O)C(F)(F)F JFD00830 c1ccnc(c1)c2nc(on2)CCCC(=O)O DP01247 CCOC(=O)c1c(csc1NC(=O)CC(=O)Nc2c(c(cs2)C)C(=O)OCC)C GK01598 c1cc(ccc1C#N)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCCC3 JFD02527 c1ccc(cc1)C2=C(C(=O)C(=O)O2)C(=S)Nc3ccc(cc3)Cl JFD00750 c1ccc(cc1)/C(=C/2\C(=O)C(=O)N(C2=S)c3ccc(cc3)Br)/O JFD00753 c1c(cc(c(c1[N+](=O)[O-])N2CCC(CC2)C#N)[N+](=O)[O-])C(F)(F)F CD11789 c1cc(c(nc1)N2CCC(CC2)C#N)[N+](=O)[O-] CD11792 CC(C)(C)c1ccc(cc1)c2cc(=O)[nH]c(=O)o2 CD11793 c1ccc(cc1)C(=C2C=CC(=NO)C=C2)C#N JA00056 CCOC(=O)/C(=C/c1ccc(cc1OC)OC)/C#N JA00061 CN(n1cnc2ccsc2c1=O)S(=O)(=O)c3ccc(cc3)Cl CD11795 CCN1CNC(=NC1)SCc2ccc(cc2)Br.Br DP01335 CCOC(=O)/C(=C/c1cc(ccc1OC)OC)/C#N JA00064 CN(n1cnc2ccsc2c1=O)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD11797 CCOC(=O)/C(=C/c1ccc(cc1)c2ccccc2)/C#N JA00066 c1ccc(cc1)n2c3c(c(cc(n3)N4CCCCC4)N5CCCCC5)c(=O)n(c2=O)c6ccccc6 JFD02475 CN(C)c1ccc(c(c1)Cl)C2Nc3ccccc3O2 DP01270 Cc1ccc(cc1)C2CN=NC23C(Oc4ccccc4C3=O)c5ccccc5 JFD01657 c1cc(ccc1c2csc(n2)c3ccc(cc3)Cl)[N+](=O)[O-].Br HR00113 Cc1cccc(c1NC(=S)Nc2c(cccc2Cl)C)Cl HR00159 CCCc1c(cnn1c2ccccc2)C(=O)O/N=C/c3ccc(cc3Cl)Cl GK01554 CCCc1c(cn(n1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)Cl GK01556 C1NC(=S)NCN1CCO DP01350 c1cc(ccc1c2cc(nc(n2)N)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)F GK01712 c1cc(sc1)C(=O)N2CCN(CC2)C(=O)C3CCCCC3 JFD02526 c1ccc(cc1)C2C3(C(CN=N3)c4ccc(cc4)Cl)C(=O)c5ccccc5O2 JFD01654 c1ccc(cc1)C2C3(C(CN=N3)c4ccc(cc4Cl)Cl)C(=O)c5ccccc5O2 JFD01655 c1ccc(c(c1)F)SCCCNC(=O)c2ccc(cc2Cl)Cl CD11815 CCOC(=O)COc1cc(c2c(=O)cc(oc2c1)c3ccccc3)O JFD02381 CCOC(=O)C(C)Oc1cc(c2c(=O)cc(oc2c1)c3ccccc3)O JFD02382 CC1(C2CCC13CS[N@@]4C3(C2)O4)C JFD00704 CC1(C2CCC13CS[N@]4C3(C2)O4)C JFD00705 c1c(c(=O)[nH]c(=O)[n@@]1C2[C@@H]([C@@H]([C@H](O2)CO)O)O)Br JFD00706 Cc1cc(c(cc1CN)CN)C.Cl.Cl JFD02408 C1CCC2(CC1)C(=O)NC(=O)N2 JFD02410 c1ccc(cc1)c2cc(c3ccccc3n2)O JFD00822 c1c(cc(c(c1I)C#N)I)C#N JFD00823 Cc1ccc(cc1)SCCC(=O)O JFD00826 c1ccc2c(c1)cccc2SCCC(=O)O JFD00832 CNS(=O)(=O)c1ccccc1Sc2cccc3c2c(ccc3)C(=O)O JFD00835 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3ccccc3[N+](=O)[O-])/C(=O)N2C JFD02464 Cn1c2c(cc3cc(ccc3n2)OC)c(=O)n(c1=O)C JFD02473 COc1ccc(cc1OC)/C=N/NC(=O)c2ccccc2N DP01155 COc1ccc(cc1)C2N(c3cc(ccc3O2)Cl)S(=O)(=O)c4cc(c(cc4Cl)Cl)Cl DP01204 c1ccc(cc1)NC(=O)c2ccc3ccccc3c2O JFD00720 Cc1ccc(cc1)S(=O)(=O)N2c3ccccc3OC2c4ccc(c(c4)Cl)Cl DP01191 Cc1c(c(=O)c2ccc(cc2o1)O)c3nc4ccccc4n3C JFD02483 COc1ccc2c3ccccc3c(=O)oc2c1 JFD02484 Cn1c2c(cn1)c(=O)[nH]cn2 GK01643 CN1CNC(=NC1)SCc2ccc(c(c2)Cl)Cl.Cl DP01341 c1c(cc(cc1Cl)Cl)OS(=O)(=O)CS(=O)(=O)Oc2cc(cc(c2)Cl)Cl CD09808 CCc1cn(nc1c2c(cccc2F)F)C(=O)c3ccccc3F CD09813 c1cc(ccc1OS(=O)(=O)CS(=O)(=O)Oc2ccc(cc2)Cl)Cl CD09819 Cc1c(c(c2cc(ccc2n1)Cl)c3ccccc3)c4ccc(c(c4)OC)OC HR00134 Cc1ccc(cc1)NC(=O)/C=N/O JA00001 Cc1ccc2c(c1)C(=O)C(=O)N2 JA00002 c1c(cc(c(c1/C=C(\C#N)/C(=O)N)O)Cl)Cl JA00004 COc1cc(ccc1O)/C=C(\C#N)/C(=O)N JA00005 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)Nc3cccc(c3)C(F)(F)F GK01572 Cn1c(nc(n1)NC(=O)C(=O)NCC(OC)OC)SC CD11696 Cc1cc(cc(n1)n2cc(c(n2)N)C#N)C(F)(F)F CD11700 COC(=O)c1c(ccs1)NC(=O)NC(=O)c2c(cccc2Cl)F GK00381 CC1=C(S(=O)(=O)C(C(C1)c2cccc(c2)C(F)(F)F)C#N)C#N CD11710 CCOC(=O)c1cnn(c1/N=C\N(C)C)c2c(c(nn2C)C)[N+](=O)[O-] GK00408 CCOC(=O)/C(=C/c1ccc(cc1)N(C)C)/C#N JA00073 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N GK01584 c1ccc2c(c1)ccc(c2/C=N/N3C(=O)c4ccccc4C3=O)O JA00038 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)SCC(=O)C GK00173 c1ccnc(c1)SC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl GK01590 COC(=O)c1ccccc1NC(=O)/C(=C\c2cc(cc(c2)Cl)Cl)/C#N GK00178 COC(=O)c1ccccc1NC(=O)/C(=C\c2c(cccc2Cl)F)/C#N GK00179 COC(=O)c1ccccc1NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N GK00180 c1cc(ccc1n2c(c(cn2)C(=O)Sc3ccc(cc3)Cl)C(F)(F)F)Cl GK01591 CN(C)/C=C(\C#N)/c1nc2ccccc2s1 GK00397 CC(=O)c1ccc(cc1)Sc2ccccc2 CD11947 CCOC(=O)C(c1c2ccccc2n(c(=O)c1[N+](=O)[O-])C)C(=O)OCC JFD00846 CCOC(=O)C(C#N)c1c2ccccc2n(c(=O)c1[N+](=O)[O-])c3ccccc3 JFD00847 c1cc(c(cc1Cl)S(=O)(=O)N2CCC(CC2)NC(=O)C3CCCCC3)Cl JFD02522 c1ccc(cc1)CN2CNC(=S)NC2 DP01356 c1cc(ccc1CN(c2ccc(cc2)F)C(=O)c3ccc(cc3)[N+](=O)[O-])Br JFD02559 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)Nc4ccc(cc4F)F JFD02564 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccccc3)/N GK01514 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)Sc3ccc(cc3)Cl GK01595 c1ccc(cc1)n2c(c(cn2)c3nc(no3)c4ccc(cc4)C(F)(F)F)C(F)(F)F GK01516 CC(C)(C)c1ccc(cc1)c2nc(on2)c3cnn(c3C(F)(F)F)c4ccccc4 GK01517 c1ccc(cc1)n2c(c(cn2)C(=O)O/N=C/c3ccccc3Cl)C(F)(F)F GK01519 Cc1ccc2cc3c(nc2c1)n(c(=O)n(c3=O)C)C JFD00850 CNC(=S)NN=C1CCCCC1 DP01142 CNC(=S)NN=C1CCCCCC1 DP01143 Cc1cc(cc(n1)N(C)NC2c3ccccc3C(=O)O2)C(F)(F)F CD11699 CCOC(=O)/C(=C/c1cccc(c1)[N+](=O)[O-])/C#N JA00069 CCOC(=O)/C(=C/c1ccc(cc1)C)/C#N JA00070 c1ccc(cc1)/C=C/C=N/NC(=O)c2ccccc2N DP01164 c1cc2c(cc1C3Nc4cc(ccc4O3)Cl)OCO2 DP01169 CCCc1c(cnn1c2ccccc2)C(=O)O/N=C(/c3ccc(cc3)Cl)\N GK01536 Cc1ccc2c(cc(nc2c1)c3ccc(cc3)Cl)C(=O)O JA00102 COc1ccc(cc1)/C=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl GK01599 c1cc(ccc1/C=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)C#N GK01600 c1cc(ccc1/C=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)F GK01601 Cc1ccc2c(cc(nc2c1)c3ccc(cc3)OC)C(=O)O JA00104 CCOC(=O)NC(=S)Nc1ccsc1C(=O)OC GK00272 c1ccc2c(c1)-c3nc4ccccc4n3C(N2)c5ccc(c(c5)Cl)Cl DP01321 c1ccc(cc1)/N=N/c2ccc(cc2O)O JFD00807 c1c2c(cc(c1Cl)Cl)C(=O)NC2=O JFD02318 Cc1ccc2c(c1)c(=O)cc(o2)C(=O)O JFD02319 CCOC(=O)Nc1c(n(c(=O)n(c1=O)C)C)N JFD02321 CC(=O)Oc1c2ccccc2sc1c3ccccc3 JFD00814 Cc1cn(nc1c2cccs2)C(=O)Nc3ccc(cc3)Cl CD09759 Cc1cn(nc1c2cccs2)C(=O)NC CD09761 COc1ccc2c(c1)C(=O)CC(O2)c3ccccc3 JFD02323 COc1ccc2c(c1)c(=O)cc(o2)c3ccccc3 JFD02324 c1ccc2c(c1)C(=O)N(C2=O)Cc3cccc(c3)I JFD02326 c1c(c(cc(c1Cl)Cl)C(=O)N)C(=O)N JFD02328 c1ccc(cc1)c2cc(=O)c3ccccc3s2 JFD00859 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N GK01582 Cc1csc2c1ncnc2N3CC(OC(C3)C)C GK01640 Cc1csc2c1ncnc2N3CCSCC3 GK01646 Cc1ccc(c2c1cccc2)C(c3ccccc3)(c4ccccc4)O JFD02393 Cc1csc2c1ncnc2N3CCCCC3 GK01647 Cc1csc2c1ncnc2NCCc3ccccn3 GK01649 Cc1csc2c1ncnc2N(C)C GK01650 CS/C(=N/S(=O)(=O)c1ccccc1)/NCc2c(cccc2Cl)Oc3ccccc3 CD11620 c1ccc(c(c1)CSC2=NCCN2)Cl.Cl DP01049 c1cc(ccc1CSC2=NCCCN2)Cl.Cl DP01051 c1ccc(cc1)CSC2=NCCCN2.Cl DP01054 c1ccc(cc1)CC(=O)N2CCC(CC2)NC(=O)C3CCCCC3 JFD02507 C1CCC(CC1)C(=O)NC2CCN(CC2)C(=O)C3CCCCC3 JFD02508 c1cc(ccc1CSC2=NCCCN2C3CCCCC3)Cl.Cl DP01442 c1ccc(cc1)CC(=O)NC2CCN(CC2)S(=O)(=O)c3cccc(c3)C(F)(F)F JFD02541 CC(=O)c1ccc(o1)c2ccc(cc2Cl)Cl CD11806 c1cc(cc(c1)S(=O)(=O)N2CCC(CC2)NC(=O)C3CCCCC3)C(F)(F)F JFD02513 COc1ccc(cc1)Cc2nc(cs2)c3ccccc3.Br DP01391 Cc1c(c(c(c(c1C)C)CSC2=NCCCN2C3CCCCC3)C)C.Cl DP01443 c1ccc(cc1)CSC2=NCCCN2C3CCCCC3.Cl DP01446 COc1ccc(cc1)/C(=C/2\C=C/C(=N\O)/C(=C2)Cl)/C#N JA00123 Cc1ccc(cc1)S(=O)(=O)NNc2ccsc2C(=O)OC GK01761 COc1ccc(cc1)N(C(CC(=O)C2CC2)c3ccccc3)C(=O)Nc4ccccc4Cl JFD02414 Cn1ccc(n1)NC(=O)NC(=O)c2c(cccc2Cl)Cl GK00383 Cn1c2c(c(c(c1=O)Cc3ccccc3)O)c(=O)n(c(=O)n2C)C JFD02468 c1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)C(=O)O)I JFD01698 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3cccc(c3)[N+](=O)[O-])/C(=O)N2C JFD02471 Cn1c2c(c3c(cc4cc(c(cc4n3)Cl)Cl)c(=O)n2c5ccccc5)c(=O)n(c1=O)C JFD02474 Cc1ccc2c(cc(nc2c1)c3ccccc3)C(=O)O JA00129 Cn1c(=O)cc(c2c1n(c(=O)n(c2=O)C)C)O JFD00852 Cc1c(nnn1c2ccccc2)C(=O)/C=C/N(C)C CD09794 c1ccc(cc1)Oc2cccc(c2CNc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl CD11614 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3cccs3)Cl CD11615 Cc1ccc2c(cc(nc2c1)c3ccc(c(c3)OC)OC)C(=O)N/N=C/c4ccc(cc4)[N+](=O)[O-] JA00128 Cn1c2c(c3c(c1=O)nc(o3)c4ccc(cc4)[N+](=O)[O-])c(=O)n(c(=O)n2C)C JFD02469 CCOC(=O)c1c(c2ccccc2oc1=O)Cl JFD02470 c1ccc(cc1)Cc2n[nH]c(=S)n2c3ccccc3 JFD00890 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Nc3ccc(cc3)O JFD00893 Cc1ccc(cc1)C(=O)N2CCN(CC2)Cc3ccccc3 JFD02546 c1cc(oc1)C(=O)NNC(=S)Nc2ccc(cc2)Cl JFD00894 Cc1ccc(cc1)C(=O)N2CCC(CC2)NC(=O)Cc3ccccc3 JFD02533 Cc1csc2c1nc(n(c2=O)C)SC GK01829 c1ccc(cc1)Oc2cccc(c2CNS(=O)(=O)c3ccc(cc3)F)Cl CD11616 Cc1csc2c1c(=O)[nH]cn2 GK01657 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)CCC(=O)CCN3C(=O)c4ccccc4C3=O JFD00806 COc1c(cc(cc1)/c/2c\3/nc(/c(c/4\[nH]/c(c(\c5n/c(c(\c6[nH]c2cc6)/c7cc(c(cc7)OC)OC)/C=C5)/c8cc(c(cc8)OC)OC)/cc4)/c9cc(c(cc9)OC)OC)C=C3)OC JFD01715 c1cc(c(cc1)Cl)/c/2c\3/nc(/c(c/4\[nH]/c(c(\c5n/c(c(\c6[nH]c2cc6)/c7c(cccc7)Cl)/C=C5)/c8c(cccc8)Cl)/cc4)/c9c(cccc9)Cl)C=C3 JFD01717 c1ccc(cc1)CC(=O)NC2CCN(CC2)C(=O)Cc3ccccc3 JFD02548 c1ccc(cc1)CC(=O)NC2CCN(CC2)C(=O)c3ccc(cc3)[N+](=O)[O-] JFD02534 Cc1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccccc3 JFD02535 CCOc1cc(ccc1O)/C=N/N2C(=O)c3ccccc3C2=O JA00134 CCOc1cc(ccc1O)/C=C(\C#N)/C(=O)N JA00135 c1cc(sc1)C(=O)N(Cc2ccc(cc2)Br)c3ccc(cc3)F JFD02552 C/C(=N\OC(=O)c1ccc(cc1)[N+](=O)[O-])/CCc2ccc(c(c2)OC)OCc3ccc(c(c3)Cl)Cl JFD02551 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3c(cccc3Cl)Cl JFD02553 COc1cc(c(cc1OC)Br)C(=O)O JFD00811 CCOC(=O)c1cc(c2ccccn2c1=O)C#N CD11728 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 JFD02554 c1ccc(cc1)CC(=O)NC2CCN(CC2)C(=O)c3cccs3 JFD02555 c1cc(ccc1C#N)OS(=O)(=O)c2ccc(s2)c3ccno3 SEW02313 Cc1ccc(c(c1)S(=O)(=O)N)Sc2ccccc2C(=O)O JFD01680 c1ccc(cc1)CC(=S)N DP01377 CC(=O)N[C@@H]1[C@H]([C@@H]([C@H](O[C@H]1O[C@H]2CC[C@]3(C(C2(C)C)CC[C@@]4(C3CC=C5[C@]4(C[C@H](C6C5CC(C[C@H]6C(=O)O)(C)C)O)C)C)C)CO)O)O JFD02451 c1cc(oc1)C(=O)NNC(=S)Nc2cc(ccc2Cl)Cl JFD00877 c1c(cc(cc1Cl)Cl)n2c(c(cn2)c3n[nH]nn3)N CD11921 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)C(F)(F)F CD11927 COCCCN1CNC(=NC1)SCc2ccc(cc2)Cl.Cl DP01331 CCN1CNC(=NC1)SCc2ccc(cc2)[N+](=O)[O-].Br DP01333 COc1cc(cc(c1OC)OC)C2Nc3cc(ccc3O2)Cl DP01284 c1ccc2c(c1)NC(O2)c3cccs3 DP01287 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)c4c(cccc4F)F JFD02557 CSC1=NCCN1C(=O)c2ccc(cc2)Cl DP01338 Cc1nc(cs1)c2ccc(cc2)Cl.Br DP01357 c1cc(ccc1CC(=S)N)Cl DP01382 CC(=O)c1ccc(c(c1)CSC2=NCN(CN2)C)OC.Cl DP01387 CC(=O)c1ccc(cc1)Oc2ccc(cc2)OC CD11916 CC(=O)c1ccc(o1)c2c(cc(cc2Cl)Cl)Cl CD11824 Cc1c(c(n(n1)C)NN2C(=O)c3cccc4c3c(cc(c4)[N+](=O)[O-])C2=O)[N+](=O)[O-] GK01676 c1cc(ccc1c2cc(nc(n2)N)N)F GK01678 CN(C1CC2CC1C=C2)C(=O)Nc3ccc(cc3)Cl CD09837 COc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccccc3C#N JFD01642 C[n+]1ccc(cc1)C(=O)c2c(cccc2OC)OC.[I-] CD11910 COc1ccc(cc1)Oc2ccc(cc2)c3ccn[nH]3 CD11920 c1cc(oc1c2nnc(o2)SCCC(=O)O)[N+](=O)[O-] JFD00895 CN1CNC(=NC1)SCc2c(cccc2Cl)Cl.Cl DP01300 c1cc(cc(c1)[N+](=O)[O-])/C=C(\C#N)/c2cccc(c2)Cl JA00140 c1csc(c1N)C(=O)N GK00439 Cc1ccc(cc1)S(=O)(=O)Oc2ccccc2C(=O)C JFD00874 c1ccc(cc1)C(c2cc3ccccc3cn2)N.Cl JFD02454 CCCC(CCC)(C(=O)O)C(=O)O JFD01643 Cn1c2c(c3c(cc4cc(ccc4n3)OC)c(=O)n2c5ccccc5)c(=O)n(c1=O)C JFD02477 CN(n1cnc2ccsc2c1=O)S(=O)(=O)C CD11780 c1cc(c(c(c1)Sc2ccc(cc2)Cl)C#N)Sc3ccc(cc3)Cl CD11786 c1ccc2c(c1)-c3nc4ccccc4n3C(N2)c5ccc(cc5)Cl DP01272 COc1ccc(cc1)CNc2ccccc2c3[nH]c4ccccc4n3 DP01273 c1ccc(c(c1)/C=N/NC(=O)c2ccc(o2)[N+](=O)[O-])O JFD00888 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)Nc3ccccc3Cl JFD00886 c1ccc(cc1)n2c(n[nH]c2=S)c3ccco3 JFD00887 COC(=O)c1cnc(nc1C(F)(F)F)N2CCN(CC2)c3ncc(c(n3)C(F)(F)F)C(=O)OC GK01865 CC12CCC3[C@H]([C@@H]1CCC2=O)CC=C4C3(CC[C@H](C4)O)C JFD01755 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@H](O1)O[C@H]2[C@H]([C@@H]([C@H]([C@@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD01756 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)Cl CD11928 CCN1CNC(=NC1)SCc2ccc(cc2)Cl.Cl DP01307 COc1ccc(cc1/C=N/N=C/2\c3ccccc3NC2=O)Br JA00097 Cc1ccc(n1N2C(=O)c3ccccc3C2=O)C JA00055 CCC1(CCCCN(C1=O)C)c2cccc(c2)OS(=O)(=O)c3ccc(c(c3)OC)OC JFD02593 COc1ccccc1NC2=C(C(=O)c3ccccc3C2=O)Cl JFD00957 c1ccc(c(c1)C(=O)NNC(=O)/C=C/C(=O)O)[N+](=O)[O-] JFD00030 C1C2C=CC1C(C2(C#N)C#N)(C#N)C#N JFD00035 c1ccc2c(c1)nc(s2)CC(=S)N GK00318 CC(=O)c1cc(ccc1OC)NC(=O)C JFD00872 Cc1cc(cc(n1)n2c(c(cn2)/C(=N/OC(=O)NC(C)(C)C)/C)C)C(F)(F)F CD11723 CC(=O)N[C@@H]1[C@H]([C@@H]([C@H](O[C@H]1O[C@H]2CC[C@]3(C(C2(C)C)CC[C@@]4(C3CC=C5[C@]4(CCC6C5CC(C[C@H]6C(=O)O)(C)C)C)C)C)CO)O)O JFD02452 Cc1ccc2c(cc(nc2c1)c3ccc(c(c3)OC)OC)C(=O)NN JA00127 CS/C(=N/S(=O)(=O)c1ccccc1)/N2CCN(CC2)c3c(cccc3C#N)C#N CD11929 Cc1c(c(n(n1)C)O)/N=N/c2ccccc2 CD11930 CCOC(=O)C(C)Oc1cc2c(c(=O)cc(o2)c3ccccc3)c(c1)OC(C)C(=O)OCC JFD02383 Cc1c(c(n(n1)C)C)NC(=O)C(=O)NCC(OC)OC CD11698 CNS(=O)(=O)c1cc(ccc1Sc2ccccc2C(=O)O)Cl JFD01679 c1ccc2c(c1)nc(s2)CC#N GK00309 c1ccc2c(c1)nc(s2)/C(=C/c3cc(cs3)Br)/C#N GK00310 c1ccc(cc1)Cc2nc(cs2)c3ccc(cc3)Cl.Br DP01381 c1ccc(c(c1)CC(=S)N)Cl DP01383 COc1ccc(cc1)CC(=S)N DP01386 CC1([C@@H](NC(S1)c2ccc(cc2)F)C(=O)O)C JFD00915 c1cc(c(c(c1)Cl)CSc2nnc(o2)c3ccc(o3)[N+](=O)[O-])Cl JFD00907 CCN1CNC(=NC1)SCc2ccc(cc2)C.Cl DP01304 CNn1cnc2ccsc2c1=O CD11674 CC1/C(=N\OC(=O)Nc2c(cccc2Cl)Cl)/CCO1 CD11682 Cc1ccc(cc1I)S(=O)(=O)NC JFD00840 CNC(=S)NN=C1CCCC1 DP01141 Cc1ccc(cc1)/C(=C/2\C=C(/C(=N/O)/C=C2Cl)Cl)/C#N JA00112 c1ccc2c(c1)cccc2C3Nc4cc(ccc4O3)Cl DP01291 CN1CNC(=NC1)SCc2ccccc2Cl.Cl DP01296 CC(C)(C)c1cc(nc(n1)N)N GK01685 CCN1CNC(=NC1)SCc2ccccc2Cl.Cl DP01306 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3cccc(c3Cl)Cl)/C(=O)N2C JFD02476 c1ccc2c(c1)N(C(O2)c3ccc4c(c3)OCO4)C(=O)c5ccc(cc5)Cl DP01171 Cc1ccc(cc1NC(=O)N)Cl JA00159 COc1cccc(c1)NC(=O)N JA00160 CC(C)(C)SCCN/C(=N\C#N)/SC CD09824 c1cc(ccc1/C=C/c2ccnc(n2)N)Cl CD09833 COc1ccc(cc1/C=C(\C#N)/C(=O)N)Br JA00165 c1ccc2c(c1)/C(=N\N=C\c3cc(cc(c3O)Br)Br)/C(=O)N2 JA00093 c1cc2c(cc1O)n3c(c(cn3)Br)nn2 GK00373 COC(=O)c1ccccc1N/C=N/O CD11684 CN1CNC(=NC1)SCc2ccccc2.Cl DP01297 Cn1ccc(n1)NC=C(C#N)C#N GK00333 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2ccccc2 JFD01748 c1c(ccc(c1)Cl)/c/2c\3/nc(/c(c/4\[nH]/c(c(\c5n/c(c(\c6[nH]c2cc6)/c7ccc(cc7)Cl)/C=C5)/c8ccc(cc8)Cl)/cc4)/c9ccc(cc9)Cl)C=C3 JFD01718 CC(CN1CCN(CC1)Cc2ccccc2)N(c3ccccn3)C(=O)c4ccc(cc4)C(C)(C)C.Cl.Cl.Cl JFD01719 c1cc2c(cc[nH]2)c(c1)NC(=O)C3CCCCC3 JFD01722 CC(=O)c1ccc(cc1)Oc2ccc(cc2)[N+](=O)[O-] CD11905 c1ccc2c(c1)nc(s2)/C(=C/c3cccc(c3Cl)Cl)/C#N GK00319 Cc1cc(cc(n1)n2c(c(cn2)/C(=N/OC(=O)Nc3ccccc3)/C)C)C(F)(F)F CD11714 c1cc(c(c(c1)Cl)CSc2[nH]c(=O)n3c(n2)ccn3)Cl GK00379 Cc1csc2c1ncnc2Sc3ccccc3NS(=O)(=O)c4ccc(cc4)Cl GK01696 CSC1=NCCN1S(=O)(=O)c2ccc(cc2)Cl DP01316 c1ccc2c(c1)-c3nc4ccccc4n3C(N2)c5cccc(c5)[N+](=O)[O-] DP01323 Cc1cccc(c1)NC2=C(C(=O)c3ccccc3C2=O)Cl JFD00959 COc1ccc(c(c1)NC(=O)Nc2ccc(cc2Cl)Cl)OC GK01818 COc1ccc(c(c1)/C=C(\C#N)/C(=O)N)OC JA00167 Cc1ccc2c(cc(nc2c1)c3ccc(cc3Cl)Cl)C(=O)O JA00170 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nc(on2)/C=C/c3cc(sc3)[N+](=O)[O-] GK01669 CC1([C@@H](NC(S1)c2cccc(c2)[N+](=O)[O-])C(=O)O)C JFD00913 Cn1c(=O)cc(c2c1n(c(=O)n(c2=O)C)C)NCc3ccccc3 JFD02458 Cc1ccc(cc1)c2nc3c(o2)c4c(n(c(=O)n(c4=O)C)C)n(c3=O)c5ccccc5 JFD02459 COCCCN1CNC(=NC1)SCc2ccc(cc2Cl)Cl.Cl DP01329 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2Sc3c4c(c(cs4)C)ncn3 GK01698 CSC(=CC(=O)c1ccccc1F)SC GK01705 CN1CNC(=NC1)SCc2ccc(cc2)Cl.Cl DP01298 c1cc(c(c(c1)C#N)NC(=O)NC(=O)c2c(cccc2F)F)C#N CD11896 Cc1csc2c1ncnc2SCC(=O)NN GK01659 c1cc(oc1)C(=O)N2CCC(CC2)NC(=O)C3CCCCC3 JFD02503 COc1ccc(cc1)NC(=S)NNC(=O)c2ccc(o2)[N+](=O)[O-] JFD00903 CC(=O)OC[C@@H]1[C@H]([C@@H](C=CO1)OC(=O)C)OC(=O)C JFD00929 CSC1=NCCN1Cc2ccccc2.I DP01289 CCOC(=O)/C(=C/c1ccc(cc1)OC)/C#N JA00076 c1ccc2c(c1)/C(=N\CCC/N=C\3/c4ccccc4NC3=O)/C(=O)N2 JA00085 c1ccc2c(c1)NC(O2)c3ccc(cc3)Cl DP01172 COc1ccc(cc1)c2nc(on2)CCC(=O)O DP01177 c1ccc(cc1)C(=O)N2c3cc(ccc3OC2c4ccc(cc4)Cl)Cl DP01183 CN1CNC(=NC1)SCc2ccc(cc2Cl)Cl.Cl DP01299 c1ccc2c(c1)/C(=N\N=C\c3cc(cc(c3O)Cl)Cl)/C(=O)N2 JA00095 C1CCCCCC(=NN=C(N)N)CCCCC1 JFD00904 c1cc(sc1S(=O)(=O)Nc2c(cn[nH]2)Br)Cl GK00364 c1ccc2c(c1)c(nc(n2)C(=O)NCCc3ccccn3)O DP01491 CC(CN1CNC(=NC1)SCc2ccc(cc2)Cl)O.Cl DP01492 Cn1cc(c(n1)NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br GK00349 COC(=O)c1c(ccs1)N/N=C/c2ccc(cc2)C#N GK01770 Cn1c2c(c3c(c1=O)cc4cc(ccc4n3)Cl)c(=O)n(c(=O)n2c5ccccc5)c6ccccc6 JFD00848 CCOC(=O)C(=CNc1ccn(n1)C)C(=O)OCC GK00322 c1cc(ccc1n2c(c(cn2)C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N)C(F)(F)F)Cl GK01574 COc1ccc(cc1OC)CC(=O)n2c(cc(n2)c3ccc(cc3)F)SC GK01628 Cc1cc(nc(n1)N)C(F)(F)F JFD00777 Cn1c2c(c3c(c1=O)cc4cc(ccc4n3)Cl)c(=O)n(c(=O)n2C)C JFD00855 c1cc(ccc1n2c(c(cn2)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(F)(F)F)Cl GK01578 CC(=O)C(=CNc1ccn(n1)C)C(=O)C GK00338 c1ccc(cc1)CC(=O)NC2CCN(CC2)Cc3ccccc3 JFD02509 Cc1csc2c1ncnc2N(C)CCO GK01656 C=CCN1C(=O)C2(CCCCC2)NC1=O JFD02405 CC1(C(=O)N(C(=O)N1)CC=C)C JFD02409 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)O/N=C(/c3ccc(cc3)Cl)\N GK01581 c1cc(c(c(c1)Cl)/C=C/c2ccnc(n2)N)F CD09836 CC(C)(C)C(=O)N(C)C1CC2CC1C=C2 CD09838 Cc1csc2c1ncnc2OC GK01824 CCc1c(cc(s1)C(C)(C)C)NC(=O)C(Cl)Cl GK01826 c1cc(ccc1S(=O)(=O)N2CCC(CC2)NC(=O)C3CCCCC3)Cl JFD02523 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)C3CCCCC3 JFD02529 c1ccc(cc1)CC(=O)NC2CCN(CC2)C(=O)C3CCCCC3 JFD02532 COc1c(c(cc(c1)/c/2c\3/nc(/c(c/4\[nH]/c(c(\c5n/c(c(\c6[nH]c2cc6)/c7cc(c(c(c7)OC)OC)OC)/C=C5)/c8cc(c(c(c8)OC)OC)OC)/cc4)/c9cc(c(c(c9)OC)OC)OC)C=C3)OC)OC JFD01714 Cn1c2c(c(c(c(=O)n2c3ccccc3)[N+](=O)[O-])O)c(=O)n(c1=O)C JFD00982 c1cc(ccc1C(=O)CSC#N)Br DP01545 c1ccc(c(c1)C2N=C(SC(=N2)c3ccc(cc3)Cl)c4ccc(cc4)Cl)Cl DP01548 c1ccc(cc1)C2CC(=O)c3ccc(cc3O2)Cl JFD00168 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)Cc4ccc(cc4)c5[nH]nnn5 JFD00162 CC(C)CNC1=C(C(=O)c2ccccc2C1=O)Cl JFD00879 c1ccc2c(c1)C(=O)[N-]S(=O)(=O)c3ccccc3S2.[Na+] JFD01700 c1ccc(cc1)CC(=O)NC2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl JFD02539 Cc1ccc2c(cc(nc2c1)c3ccc(c(c3)OC)OC)C(=O)O JA00105 CCOC(=O)c1c(csc1NC(=O)Nc2ccc(cc2)Cl)C GK00541 c1ccc2c(c1)cc(cc2C#N)CCCCc3cc4ccccc4c(c3)C#N JFD00070 c1ccc(cc1)c2csc(n2)Cc3ccc(cc3)Cl.Br DP01388 CCS(=O)CC(=O)Nc1c(=O)c2ccccc2oc1c3ccccc3 JFD00164 Cn1c2c(c(c(c(=O)n2c3ccccc3)[N+](=O)[O-])N)c(=O)n(c1=O)C JFD00988 c1cc(ccc1SCC(=O)Nc2ccsc2C(=O)N)Cl GK00480 Cc1ccc(cc1)Cc2nc(cs2)c3ccccc3 DP01392 Cn1c2c(c3c(c1=O)cc4c(n3)cc(cc4Cl)Cl)c(=O)n(c(=O)n2C)C JFD02479 Cc1ccc(cc1Cl)/N=c\2/c(c(ss2)SC)c3ccccc3 JA00150 CCOC(=O)c1[nH]c(=O)c2c3c(sc2n1)CCCC3 DP01475 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3ccc(c(c3)Cl)Cl)/C(=O)N2C JFD02465 Cc1ccc(cc1)CC(=S)N DP01389 c1ccc(cc1)c2csc(n2)Cc3ccccc3Cl.Br DP01390 C1NC(=S)NCN1CCCO DP01439 CC(CN1CNC(=S)NC1)O DP01414 c1cc(ccc1Cc2nc(cs2)c3ccc(cc3)Cl)Cl.Br DP01393 Cc1ccc(cc1)Cc2nc(cs2)c3ccc(cc3)Cl.Br DP01396 CCOC(=O)CSc1nnc(o1)c2ccc(o2)[N+](=O)[O-] JFD00897 COC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccc(cc3Cl)Cl GK00546 CC(C(=O)N1CCN(CC1)Cc2ccccc2)N3CCN(CC3)Cc4ccccc4 JFD02536 Cc1ccc(cc1)C(=O)C2=NNCC2c3ccccc3 JFD01667 Cc1csc(c1NNS(=O)(=O)c2ccc(cc2)Cl)C(=O)OC GK01789 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCC(CC2)NC(=O)Cc3ccccc3 JFD02543 c1cc(ccc1C2N=C(SC(=N2)c3ccc(cc3)Cl)c4ccc(cc4)Cl)Cl DP01549 c1cc(ccc1C2=NC(N=C(S2)c3ccc(cc3)Cl)c4ccc(c(c4)Cl)Cl)Cl DP01550 CCOC(=O)c1c(n2c(c3c(c(nnc3n2)c4ccccc4)c5ccccc5)nn1)C JFD00961 c1cc2c(nc1)Nc3c(nc4ccc(cc4n3)Cl)O2 JFD00917 c1ccc2c(c1)nc3c(n2)Oc4ccccc4N3 JFD00900 c1ccc2c(c1)[nH]c(n2)C(F)(F)F DP01555 c1cc(cc(c1)n2c(csc2=N)c3ccc(cc3)Br)C(F)(F)F.Cl DP01553 Cc1cc(c(cc1Cl)C)Sc2c3c(cc(s3)c4ccc(cc4)F)ncn2 GK01722 Cc1ccc(cc1)/N=c\2/c(c(ss2)SC)c3ccccc3 JA00147 COc1ccc(cc1)NC(=S)NNC(=O)c2[nH]c(=O)c3ccccc3n2 DP01473 Cc1ccc(cc1)CSc2c(c(=S)ss2)c3ccccc3 JA00148 c1ccc(cc1)CC(=O)NC2CCN(CC2)C(=O)c3ccco3 JFD02544 CC(CN1CCN(CC1)Cc2ccccc2)N(c3ccccn3)C(=O)C4CCC4.Cl.Cl.Cl JFD01697 c1ccc(cc1)NC(=O)N2CCN(CC2)c3c(cccc3C#N)C#N CD11782 c1cc(c(c(c1)Cl)C#N)N2CCC(CC2)C#N CD11790 c1ccc(cc1)CC(=O)NC2CCN(CC2)C(=O)C3CCC3 JFD02540 COC(=O)c1cnc(nc1C(F)(F)F)Sc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01874 c1ccc(cc1)C(=O)OC[C@@H]2[C@H]([C@@H]([C@@H](O2)c3nnc(o3)C(F)(F)F)OC(=O)c4ccccc4)OC(=O)c5ccccc5 JFD01741 c1ccc2c(c1)c(=O)cc(o2)c3ccc(cc3)C(=O)OCC#N JFD01049 CCOC(=O)C1=C(NC(=O)NC1c2ccccc2OC)C JFD01802 CCOC(=O)C(=CNc1ccsc1C(=O)N)C(=O)OCC GK00450 CCCCc1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl JFD00880 c1ccc(cc1)C(=O)CNC(=S)Nc2ccccc2 JFD00881 CC(CN1CCN(CC1)Cc2ccccc2)N(c3ccccn3)C(=O)c4ccoc4.Cl.Cl.Cl JFD01674 Cc1cc(ccc1NC(=O)N)Cl JA00161 c1ccc(c(c1)NC(=O)/C=N/O)Cl JA00163 CCOC(=O)C1=C(NC(=O)NC1c2ccc(c(c2)OC)OC)C JFD01801 Cc1cc(c(c(c1)C)CSC2=NCCCN2C3CCCCC3)C.Cl DP01454 COc1ccc(cc1OC)S(=O)(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 JFD02583 Cn1c2c(c3c(cc4cc(ccc4n3)Cl)c(=O)n2c5ccccc5)c(=O)n(c1=O)C JFD00985 COC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)F GK01857 Cc1csc(c1NN2C(=O)c3c(c(c(c(c3Cl)Cl)Cl)Cl)C2=O)C(=O)OC GK01784 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccc(cc2F)F GK00549 COC(=O)c1cnc(nc1C(F)(F)F)N2CCSCC2 GK01863 c1ccc(c(c1)C(=O)O)Sc2ccccc2S(=O)(=O)NC34CC5CC(C3)CC(C5)C4 JFD01694 CN(C)/C=C/C(=O)c1ccc(cc1)Oc2ccc(cc2)[N+](=O)[O-] CD11907 c1ccc2c(c1)nc(s2)/C(=C/O)/C#N GK00468 CC(C)(C)CC(C)(C)N1CNC(=S)NC1 DP01598 Cc1ccc2c(c1)NC(O2)c3ccc(cc3)NC(=O)C DP01600 Cc1ccc(cc1)CSC2=NCN(CN2)C(C)(C)CC(C)(C)C.Cl DP01604 CCC(CO)N1CNC(=S)NC1 DP01456 Cc1ccc(cc1)/N=N/c2c(nn(c2O)C(C)(C)C)C CD11948 CNC(=S)NNC(=O)c1cccnc1 JFD00934 CC1([C@@H](NCS1)C(=O)[O-])C.[K+] JFD00937 COc1ccc(cc1)C/N=C/c2cc(cc(c2O)Cl)Cl DP01608 c1ccc(cc1)OCC(=O)Nc2ccccc2C(=O)O DP01612 c1cc(ccc1/C(=C\C=C(C#N)C#N)/Sc2c(cc(cn2)C(F)(F)F)Cl)Cl JFD00973 COc1ccccc1N2CCN(CC2)C(=O)Nc3ccc(cc3F)F JFD01736 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Oc3cc(c(cc3Cl)Cl)Cl JFD00950 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl JFD01737 CCOC(=O)/C(=C/NNc1ccsc1C(=O)OC)/C#N GK01777 CC1([C@@H](NCS1)C(=O)[O-])C.[Na+] JFD00938 COC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)C(F)(F)F GK01838 Cc1csc(c1NN2C(=O)c3ccccc3C2=O)C(=O)OC GK01780 CSc1ccccc1NC(=O)c2cnc(nc2C(F)(F)F)N GK01781 Cc1cc(c(c(c1CSC(=N)N)C)CSC(=N)N)C.Cl.Cl DP01469 c1ccc2c(c1)nc3c(n2)Oc4cccnc4N3 JFD00943 Cc1c2ccccc2ncc1c3nnnn3c4ccc(cc4)Cl JFD00980 c1cc(c(cc1S(=O)(=O)Nc2ccsc2C(=O)N)Cl)Cl GK00454 CCOC(=O)/C(=C/Nc1ccsc1C(=O)N)/C#N GK00455 Cc1ccc(cc1)S(=O)(=O)NNc2ncc(c(n2)C(F)(F)F)C(=O)OC GK01836 Cn1c(c(cn1)NC(=O)O/N=C/c2ccccc2)n3cccc3 GK00642 COc1ccc(cc1)N2C(=O)Cc3ccc(cc3C2=O)OC JFD01787 C/C(=C\C(=O)C)/NCCN/C(=C/C(=O)C)/C JFD01792 c1cc(cc(c1)Cl)NC(=O)NCc2c(ccs2)Cl GK01843 CCOC(=O)c1c(csc1NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N)C GK00565 CCOC(=O)CC(=O)Nc1c(c(cs1)C)C(=O)OCC GK00567 CC1(CN=C(S1)Nc2ccccc2F)C JFD00990 Cc1csc(c1NNC(=O)C(F)(F)F)C(=O)OC GK01786 CC(=O)c1ccc(cc1)Oc2ccc(cc2Cl)Cl CD11911 CC(=O)N1CCC(CC1)NC(=O)Oc2ccc(cc2)Cl CD11901 Cn1c2c(c3c(c(=O)n2c4ccccc4)nc(o3)c5ccc(cc5)[N+](=O)[O-])c(=O)n(c1=O)C JFD02460 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3c(cccc3Cl)Cl)/C(=O)N2C JFD02461 C(C(=O)NN)S(=O)(=O)CS(=O)(=O)CC(=O)NN JFD01797 CSC(=CC(=O)c1ccc(cc1)Oc2ccc(cc2Cl)Cl)SC CD12042 COc1ccccc1N2CCN(CC2)C(=O)c3ccc(cc3)Cl JFD01727 COc1ccccc1N2CCN(CC2)C(=O)C3CCCCC3.Cl JFD01729 c1cc(c(cc1F)F)NC(=O)N2CCN(CC2)c3ncc(cn3)Br JFD01732 c1cc(ccc1CN(c2ccc(cc2)F)C(=O)C3CCCCC3)Br JFD02563 CCOC(=O)C(=CN(c1ccc(c(c1)Cl)F)C2=NCC(S2)C)C(=O)OCC JFD00991 Cc1cccc(c1)NC(=O)N2CCN(CC2)c3ccccc3OC JFD01735 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccc3OC JFD01733 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccccc3C(=O)OC JFD01734 CSc1cc(n[nH]1)c2ccc(cc2)Oc3ccccc3 CD11949 Cc1ccc2c(cc(nc2c1)c3ccc(cc3)[N+](=O)[O-])C(=O)O JA00131 c1ccc(cc1)/C(=C/2\C=C/C(=N\O)/C(=C2)Br)/C#N JA00132 CCN1CNC(=NC1)SCc2c(cccc2Cl)Cl.Cl DP01311 CCN1CNC(=NC1)SCc2c(c(c(c(c2C)C)C)C)C.Cl DP01312 c1csc(c1Cl)C(=O)N GK01727 Cc1ccc(c(c1)NS(=O)(=O)c2ccc(s2)c3ccno3)n4cccc4 SEW06408 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Oc3ccc(cc3)N JFD00954 CC(C)OC1=C(C(=O)c2ccccc2C1=O)Cl JFD00958 CCOC(=O)/C(=C(\C)/c1ccc(cc1)NC(=O)C)/C#N DP01502 c1ccc(cc1)C(=O)/C=C(/C(=O)Nc2ccccn2)\O JFD00020 Cc1ccc(cc1)C(=O)/C=C(/C(=O)Nc2ccccc2)\O JFD00021 COc1ccc(cc1OC)C2N=C(SC(=N2)c3ccc(cc3)Cl)c4ccc(cc4)Cl DP01503 c1cc(ccc1C2=NC(N=C(S2)c3ccc(cc3)Cl)c4ccc5c(c4)OCO5)Cl DP01504 c1ccc(cc1)S(=O)(=O)c2ccc(cc2)c3ccn[nH]3 CD11981 CN(C)/C=C/C(=O)c1cccc(c1)Br CD11982 Cn1cc(c(n1)NC(=O)c2cc(cc(c2)Cl)Cl)Br GK00351 CC(=O)c1ccc(o1)c2ccc(c(c2)Cl)F CD11840 CCN1c2ccc(c3c2c(ccc3)C1=O)NC(=O)c4ccccc4C JFD02492 c1ccc(cc1)NC(=S)NNC(=O)c2ccco2 JFD00865 CC(=O)c1cc(ccc1O)OC JFD00869 c1ccc(cc1)NC(=O)/C(=C/C(=O)c2ccc(cc2)Br)/O JFD00022 CN(C)/C=C/C(=O)c1ccc(cc1)S(=O)(=O)c2ccccc2 CD11974 c1ccc(cc1)/C=C/C=C/C=C/C=C/c2ccccc2 JFD00033 COc1ccc(cc1OC)C(=O)Cc2ccccc2 JFD00038 c1cc(ccc1/C=C(\C#N)/C(=O)Nc2ccsc2C(=O)N)C#N GK00531 c1cc(ccc1c2csc(n2)N)Cl.Br DP01364 Cc1csc2c1ncnc2N3CCOCC3 GK01645 Cc1csc2c1ncnc2SCC(=O)OC GK01655 C1CCN(C1)C(=O)C23CC4CCC(C2)CC(C4)C3 JFD02497 c1cc(ccc1C2=CSC3=NCCN23)Cl.Br DP01365 c1ccc(cc1)Nc2nc(cs2)c3ccc(cc3)Cl.Br DP01367 CN1CNC(=NC1)SCc2ccc(cc2)C#N.Br DP01376 COC(=O)/C(=C\1/CCSC1)/C#N GK00474 CC(=O)N1CCC(CC1)C2=NNC(=O)C2/N=N/c3ccc(cc3)Cl CD12046 c1ccc2c(c1)c(=O)cc(o2)c3ccc(cc3)[N+](=O)[O-] JFD00154 COc1ccc(cc1)c2cc(=O)c3cc(ccc3o2)F JFD00155 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)Cl JFD00156 c1ccc(c(c1)C(=O)O)Sc2cc(ccc2S(=O)(=O)N)Cl JFD01687 c1ccc(c(c1)Cc2nc(cs2)c3ccc(cc3)Cl)Cl.Br DP01394 c1ccc(cc1)/N=c/2\nc([nH]c(=N)n2c3ccccc3)N JFD00933 c1ccc(c(c1)n2cc(c(n2)N)c3[nH]nnn3)Cl CD11764 c1ccc(c(c1)c2csc(n2)N)Cl.Br DP01422 Cn1cc(c(n1)NS(=O)(=O)c2ccccc2C(F)(F)F)Br GK00331 CCCCc1ccc(cc1)/N=N/c2c3ccccc3ccc2O JFD00939 Cc1ccc(cc1)/N=N/c2c(nn(c2O)C)c3ccccc3 CD11939 CSC(=CC(=O)c1ccc(cc1)Oc2ccccc2)SC CD11942 CC(C)(C)C(=O)O/N=C/c1ccc2c(c1)OCO2 JFD02721 COc1ccccc1CC(=O)O/N=C/c2ccc3c(c2)OCO3 JFD02722 Cc1ccc(cc1)/N=N/c2c(n[nH]c2O)C CD11944 CCC(=O)Nc1cccc2c1cccc2NC(=O)CC JFD00041 CCOC(=O)C1=C(NCC1=O)C JFD00049 c1csc2c1[nH]cnc2=O GK00357 COc1ccc(cc1)c2cc(nc(n2)N)N GK01808 COc1ccc(c(c1)NC(=O)Nc2ccc(cc2)F)OC GK01816 c1cc(oc1)C(=O)N2CCC(CC2)NC(=O)C3CCC3 JFD02519 c1cc2c(cc1/C=N/OC(=O)C3CCCCC3)OCO2 JFD02723 c1csc(c1NC(=O)C(F)(F)F)C(=O)N GK00487 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)Cl JFD01001 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(c2)Cl JFD01002 CSC1=NCN(CN1)CCCO.Br DP01622 Cc1c(cccc1Cl)NC(=S)N(CCO)N DP01638 CN(C)c1cc(cc(c1)C(F)(F)F)C(F)(F)F DP01640 CCOC(=O)c1c(c2ccccc2s1)N DP01647 Cc1c(c(n(n1)C)N/N=C/c2ccc(cc2)C#N)[N+](=O)[O-] GK00492 Cc1c(c(n(n1)C)N/N=C/c2ccc(cc2)OC)[N+](=O)[O-] GK00493 COC(=O)c1c(ccs1)NNC(=O)C(Cl)Cl GK01758 c1ccc(cc1)CC(=O)NC2CCN(CC2)C(=O)c3c(cccc3Cl)Cl JFD02545 CCN1c2ccc(c3c2c(ccc3)C1=O)NC(=O)c4cccc(c4)[N+](=O)[O-] JFD02493 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCC(CC2)NC(=O)C3CCCCC3 JFD02528 c1cc(ccc1C(=O)N2CCN(CC2)C(=O)C3CCCCC3)[N+](=O)[O-] JFD02530 c1cc(c(cc1Cl)Cl)C(=O)N2CCC(CC2)NC(=O)C3CCCCC3 JFD02521 COC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)C(F)(F)F GK01858 c1cc(sc1)C(=O)N2CCC(CC2)NC(=O)C3CCCCC3 JFD02502 c1ccc(cc1)CC(=O)NC2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F JFD02538 Cc1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)OC GK01869 CCOC(=O)c1c(csc1NC(=O)CC(=O)C(F)(F)F)C GK00557 Cc1c(c(n(n1)C)N/N=C/c2cc(cs2)Br)[N+](=O)[O-] GK00494 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccc(c(c1)C)C JFD01016 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)OC GK01872 c1ccc2c(c1)CCC(O2)C(=O)Nc3ccc(cc3)C(F)(F)F GK01878 COc1ccc(cc1)Cc2nc(cs2)c3ccc(cc3)Cl DP01395 CN(C)/C=C/C(=O)c1ccc(cc1)Oc2ccccc2 CD11750 COC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)Cl GK01837 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)C(Cl)Cl GK00602 CC(=O)c1c(cc(s1)c2ccc(cc2)Cl)N GK00604 Cc1ccc(cc1)/c/2c\3/nc(/c(c/4\[nH]/c(c(\c5n/c(c(\c6[nH]c2cc6)/c7ccc(cc7)C)/C=C5)/c8ccc(cc8)C)/cc4)/c9ccc(cc9)C)C=C3 JFD01716 CCOC(=O)/C(=N/Nc1ccc(cc1C)C)/C(=O)C JFD01764 c1ccc2c(c1)CCC(O2)C(=O)Nc3ccc(cc3Cl)Cl GK01881 c1ccc2c(c1)CCC(O2)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F GK01892 c1ccc(cc1)n2c(csc2=N)c3ccc(cc3)Br.Cl DP01552 CSC1=NCN(CN1)Cc2ccccc2.I DP01558 c1ccc(cc1)CC(=O)NC2CCN(CC2)S(=O)(=O)c3cccc(c3Cl)Cl JFD02537 COC(=O)c1c(ccs1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl GK00550 CCOC(=O)c1c(csc1NC(=O)Nc2c(cccc2Cl)Cl)C GK00551 c1cnc(nc1)S/C(=C/C=C(C#N)C#N)/c2ccc(cc2)Cl JFD00978 c1cc(sc1)C(=O)O/N=C/c2ccc3c(c2)OCO3 JFD02720 CN(CCO)c1ccc(cc1)C(=O)c2ccc(cc2)N(C)CCO JFD02724 CCCCCCCCCCCCN1CNC(=S)NC1 DP01620 c1ccc(c(c1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)NC(=S)N/N=C/c3cc(cc(c3O)Cl)Cl DP01732 COCCCNC(=S)NNC(=O)c1ccncc1 DP01754 CCN(CC)CCN1CNC(=S)NC1 DP01621 CN(C(=S)Nc1cc(ccc1Cl)Cl)N DP01631 CN(C(=S)Nc1ccccc1C(=O)OC)N DP01635 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)NC(=O)Cc3ccccc3 JFD02542 c1ccc(c(c1)CSC2=NCCCN2C3CCCCC3)Cl.Cl DP01441 Cc1c(c(n(n1)C)N/N=C/c2c(cccc2Cl)Cl)[N+](=O)[O-] GK00491 c1cc(c(c(c1)Cl)CSC2=NCCCN2C3CCCCC3)Cl.Cl DP01444 CC(CCc1ccc(c(c1)OC)OC(=O)C2CCCCC2)NC(=O)C3CCCCC3 JFD02575 c1cc(ccc1c2cn3c(n2)sc(n3)C(F)(F)F)F DP01670 Cn\1c2ccccc2s/c1=N\N JFD02742 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)C(F)(F)F GK00607 c1cc(ccc1SCCS(=O)(=O)CCSc2ccc(cc2)Cl)Cl DFP00062 Cc1cc(c(cc1Cl)C)SCCS(=O)(=O)CCSc2cc(c(cc2C)Cl)C DFP00064 CCOc1cc(nc(n1)SCc2c(cccc2Cl)F)c3ccccc3 GK00495 CCOc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)c3ccccc3 GK00496 c1ccc(c(c1)c2csc(n2)c3cccnc3)Cl.Br DP01415 Cc1nc(cs1)c2ccccc2Cl.Br DP01418 Cc1ccc(cc1)CSC2=NCN(CN2)Cc3ccccc3.Cl DP01557 COC(=O)c1c(cc(s1)c2ccccc2)N GK00498 C1CCC(CC1)N2CCCNC2=S DP01428 c1ccnc(c1)NC(=O)c2cc(ccc2N)[N+](=O)[O-] DP01429 CC(C)N(C(C)C)C(=O)NCc1ccccc1 JFD01114 c1ccc(cc1)NC(=O)N2CCCCC2 JFD01117 COc1ccc(cc1)c2cc(=O)c3ccc(cc3o2)O JFD00149 CC(C)c1ccc(cc1)C2CN=NC23CSc4ccccc4C3=O JFD01079 COc1ccc(cc1)C2CN=NC23CSc4ccccc4C3=O JFD01080 c1ccc(cc1)NC(=O)NO JFD01119 c1cc(oc1)c2n[nH]c(=S)n2c3ccc(cc3)Cl JFD00905 CC(=O)N[C@@H]1[C@H]([C@@H]([C@H](O[C@@H]1OC(=O)C)COC(c2ccccc2)(c3ccccc3)c4ccccc4)OC(=O)C)OC(=O)C JFD00908 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Nc3ccc(cc3)N JFD00951 Cc1cccc(c1)OC2=C(C(=O)c3ccccc3C2=O)Cl JFD00953 Cc1csc(c1Cl)C(=O)N GK01748 c1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl JFD00955 c1ccc(cc1)OC2=C(C(=O)c3ccccc3C2=O)Cl JFD00912 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)NCCO JFD00956 Cc1ccc(cc1)S(=O)(=O)Oc2ccsc2C(=O)OC GK01919 COC(=O)c1cnc(nc1C(F)(F)F)Sc2ccc(cc2)Cl GK01933 CC1CN(CC(O1)C)c2ncc(c(n2)C(F)(F)F)C(=O)OCc3ccccc3 GK01936 COC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)[N+](=O)[O-] GK01856 COC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)Cc2ccccc2 GK01859 c1ccc2c(c1)CCC(O2)C(=O)O/N=C(\c3ccc(cc3)Cl)/N GK01888 c1csc(c1Cl)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01974 CCOC(=O)C1=C(NC(=O)NC1c2ccc(c(c2)[N+](=O)[O-])N(C)C)C JFD01807 CCCC1C(=C(NC(=O)N1)C)C(=O)OCC JFD01808 c1ccc2c(c1)CCC(O2)c3nc(no3)c4ccc(cc4)Cl GK01891 Cc1cc(=O)oc2c1cc(cc2)O JFD00974 CCCc1c(cnc(n1)N)C(=O)OCC GK01750 COC(=O)c1c(ccs1)NNS(=O)(=O)c2ccc(cc2)Cl GK01760 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc3c2cc[nH]3 JFD01723 CCCCNC(=O)Nc1ccn(n1)C GK00539 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)Cl JFD01032 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cccc(c1)Cl JFD01033 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(c(c1)F)F JFD01035 Cn1ccc(n1)NC(=O)Nc2ccccc2 GK00538 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccccc1F JFD01019 COC(=O)c1cnc(nc1C(F)(F)F)N/N=C\c2cccc(c2)Cl GK01882 c1ccc2c(c1)CCC(O2)C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N GK01883 COC(=O)c1cnc(nc1C(F)(F)F)N/N=C\c2ccc(cc2)C(F)(F)F GK01885 CCOC(=O)C1=C(NC(=O)NC1c2ccc(c(c2)Br)OC)C JFD01803 c1ccc(cc1)C2N(C(=NN2C(=O)c3ccccc3)NC(=O)c4ccccc4)C(=O)c5ccccc5 JFD01743 CCSC([C@H]([C@@H]([C@@H]([C@H](COC(=O)c1ccccc1)OC(=O)c2ccccc2)OC(=O)c3ccccc3)O)O)SCC JFD01745 c1ccc(c(c1)C(=O)N(Cc2ccc(cc2)Br)c3ccc(cc3)F)Br JFD02556 Cc1ccccc1C(=O)N(Cc2ccc(cc2)Br)c3ccc(cc3)F JFD02560 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)NC(=O)Cc3ccccc3 JFD02562 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2cccc3c2cc[nH]3 JFD01724 c1ccc2c(c1)c(=O)[nH]c(n2)C(=O)NN DP01471 CC(C)(C)c1ccc(cc1)C(=O)Oc2c(csc2C(=O)OC)Br GK01949 c1ccc(cc1)CN2CC(CN(C2)Cc3ccccc3)c4n[nH]nn4 CD12037 c1ccc2c(c1)CCC(O2)C(=O)Nc3ccc(cc3)OC(F)(F)F GK01877 c1cc(oc1)CN2CCS(=O)(=O)CC2 DFP00060 Cc1cc(c(cc1OC)CCCCCc2cc(c(cc2OC)C)OC)OC JFD02750 c1cc(c(cc1Cl)C(=O)NCc2ccncc2)N DP01704 CCC1(CCCCN(C1=O)C)c2cccc(c2)OS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F JFD02597 COC(=O)c1c(c(cs1)Br)OC(=O)c2ccc(cc2Cl)Cl GK01948 c1c2c(nc3c1sc(n3)N)nc(s2)N JFD00922 Cc1ccc2c(c1)NC(O2)c3ccc(cc3)N(C)C DP01586 COC(=O)c1ccccc1NC(=S)Nc2ccccc2 DP01595 CO[C@@H]1[C@@H]([C@H]([C@@H]([C@H](O1)COC(=O)c2ccccc2)O)O)OC(=O)c3ccccc3 JFD00927 C#CCN1CCS(=O)(=O)CC1 DFP00032 CS(=O)(=O)CS(=O)(=O)C JFD02736 c1ccc(cc1)n2c3ccccc3sc2=N JFD02741 c1ccc(cc1)CN2CCNC(C2=O)CC(=O)Nc3ccccc3 DP01683 Cc1ccc2c(c1)OC(N2)c3ccc(cc3)N(C)C DP01585 CC1c2ccsc2CCN1C(=O)Nc3ccccc3 DFP00160 c1ccc(c(c1)NC(=O)Nc2cc(sc2)[N+](=O)[O-])Cl DFP00170 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)S(=O)(=O)N JFD01036 CC(=O)NC(C(F)(F)F)(C(F)(F)F)NCc1ccc(cc1)F JFD01038 C[n+]1ccc(cc1)CCc2cc[n+](cc2)C.[I-].[I-] JFD02751 c1ccc(cc1)Oc2cccc3c2C(=O)c4c(cccc4Oc5ccccc5)C3=O JFD02753 CCOC(=O)c1c2c(sc1NC(=O)Cc3ccccc3)CCCC2 DP01676 CC(C)(C)SCCSCCS(=O)(=O)CCSCCSC(C)(C)C DFP00065 c1ccc(c(c1)c2[nH]c(c(n2)c3ccc(cc3)Cl)c4ccc(cc4)Cl)Cl DP01610 COC(=O)c1c(ccs1)N/N=C/c2ccc(cc2)O GK01771 COC(=O)c1c(ccs1)N/N=C/c2ccc(cc2)F GK01772 COC(=O)c1c(ccs1)N/N=C/c2c(cccc2Cl)F GK01773 C/C(=N\NC(=S)Nc1cccc(c1)F)/c2ccco2 DFP00074 c1cc(sc1)CNC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00085 CC(=O)Nc1ccc2c(c1)c(=O)cc(o2)c3ccc(cc3)C#N JFD01054 c1ccc(c(c1)C(=O)Nc2nnc(s2)C(F)(F)F)NC(=O)c3ccccc3Cl DP01782 Cc1nc(cs1)CSc2ccc(cc2)Cl CD12003 Cc1nc(cs1)CSCc2ccc(cc2Cl)Cl CD12004 CCOC(=O)COc1ccc2c(=O)cc(oc2c1)c3ccccc3 JFD01059 CC(=O)Nc1c(=O)c2ccccc2oc1c3ccccc3 JFD01060 CC(C)(C)n1ccc(n1)c2cc(cc(c2O)F)F CD12010 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccccc1C JFD01014 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccccc1OC JFD01015 Cn1c(c(cn1)NC(=O)O/N=C/c2ccccc2Cl)n3cccc3 GK00641 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1cccc(c1)F JFD01018 CN1c2ccc(cc2C(=O)N3C1=NCC3)Cl DP01777 c1ccc(c(c1)c2ncc3n2cccc3)[N+](=O)[O-] DP01778 Cc1c(nccn1)c2ccnn2S(=O)(=O)c3ccccc3 CD11992 Cc1c(nccn1)c2ccnn2C(=O)C CD11995 c1ccc2c(c1)c(=O)oc(n2)c3ccccc3Cl DP01780 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3cccc(c3)C(F)(F)F JFD02581 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 JFD02582 CC1CCC(C(C1)N(Cc2ccccc2)C(=O)c3ccccc3)C(C)C JFD02584 C1=C(C(=O)C=C(C1=O)Br)Cl JFD02745 Cc1cc(c(cc1OC)C(=O)CCC(=O)O)OC JFD02747 Cc1cc(c(c(c1)C)CSc2ccccn2)C.Cl DP01507 Cc1cc(c(c(c1)C)CSc2nccn2C)C.Cl DP01508 Cc1ccc(cc1)/N=N/c2c(nn(c2O)C)COC CD11954 c1ccc(cc1)CC(=O)O/N=C/c2ccc3c(c2)OCO3 JFD02710 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)OC CD11931 c1cc(oc1)C(=O)O/N=C/c2ccc3c(c2)OCO3 JFD02714 c1ccc(c(c1)C(=O)O/N=C/c2ccc3c(c2)OCO3)Br JFD02716 c1cc(cc(c1)[N+](=O)[O-])C(=O)O/N=C/c2ccc3c(c2)OCO3 JFD02718 c1ccc(cc1)C2=CC(=O)C(=CC2=O)Cl JFD02731 CC(CCc1ccc(c(c1)OC)OC(=O)c2ccco2)NC(=O)c3ccco3 JFD02573 CC(CCc1ccc(c(c1)OC)OC(=O)Cc2ccccc2)NC(=O)Cc3ccccc3 JFD02576 c1ccc(cc1)S(=O)(=O)CS(=O)(=O)c2ccccc2 JFD02737 CCS(=O)(=O)Cc1ccccc1 JFD02738 CC(=O)Nc1ccc(cc1)/C=N/Cc2ccc(cc2)OC DP01609 c1ccc(cc1)CSC(=O)NC2CCCCC2 JFD00113 c1ccc(cc1)SC(=O)OCNC2CCCCC2 JFD00112 CN1CCN(CC1)C(=O)Oc2ccccc2 JFD00116 COc1cc(cc(c1OC)OC)C(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O DP01716 CSc1cc(nn1C(=O)Nc2ccccc2)c3ccc(cc3)Oc4ccccc4 CD11956 CC(C)(C)N1CNC(=S)NC1 DP01531 COc1ccc(cc1Br)/C=C(\C#N)/C(=O)N JA00166 c1cc(c(c(c1)Cl)F)c2ccnc(n2)N CD11958 COc1ccc(cc1/C=N/N2C(=O)c3ccccc3C2=O)Br JA00169 Cc1ccc(c(c1)NS(=O)(=O)c2ccccc2)NS(=O)(=O)c3ccccc3 JFD02739 Cc1ccc2c(c1)NC(O2)c3ccc(c(c3)OC)OC DP01588 c1ccc(cc1)c2csc(=N)n2c3cc(cc(c3)C(F)(F)F)C(F)(F)F DP01594 Cc1ccc2c(c1)OC(N2)c3ccc(cc3)NC(=O)C DP01599 COCOc1ccc(cc1OC)C(=O)O JFD01122 CC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)C(Cl)Cl GK00608 c1ccc(cc1)COc2ccccc2c3cc(no3)c4ccc(cc4)[N+](=O)[O-] JFD01065 CCOC(=O)c1c(csc1NC(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C)C GK00545 c1ccc2c(c1)c(c3ccccc3c2CC#N)CC#N JFD00079 Cc1csc(c1C(=O)N)NC(=O)C GK00519 c1csc(c1NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)C(=O)N GK00452 c1ccc(cc1)/C=C/c2ccncc2 JFD00085 c1ccc-2c(c1)Cc3c2ccc(c3)C#N JFD00086 COc1cccc(c1)n2c(c(c3ccc(cc3c2=O)[N+](=O)[O-])C#N)N JFD01860 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccccc1F JFD01026 Cc1csc(c1N/N=C/c2cccc(c2)OC)C(=O)OC GK01797 Cc1csc(c1N/N=C/c2ccc(cc2)F)C(=O)OC GK01798 COC(=O)c1c(ccs1)NNC(=O)CC#N GK01800 CCOC(=O)C(=CNNc1c(csc1C(=O)OC)C)C(=O)OCC GK01801 c1ccc(c(c1)C(=O)O)Sc2ccccc2S(=O)(=O)NC3CCCCC3 JFD01693 c1cc(ccc1CS(=O)(=O)CCS(=O)(=O)CCS(=O)(=O)Cc2ccc(cc2)Cl)Cl DFP00066 CCCCCCCCCCCCNc1ccc(c2c1C(=O)c3ccccc3C2=O)NCCCCCCCCCCCC JFD00152 CCOC(=O)c1c2c(sc1NC(=O)COc3ccc(cc3Cl)Cl)CCCC2 DP01677 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)C(F)(F)F JFD01028 C/C(=N\Nc1ccsc1C(=O)OC)/c2ccc(cc2)NC(=O)C(Cl)Cl GK01795 Cc1csc(c1N/N=C/c2c(cccc2Cl)F)C(=O)OC GK01796 Cc1nc(cs1)COc2ccc(cc2)C#N CD12030 CN(C)/C=C/C(=O)c1cccc(c1)C#N CD11983 c1c(csc1[N+](=O)[O-])/C(=N/O)/N DFP00021 Cc1c(ccc2c1OC(CNC2=O)(C)C)OC JFD00047 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)NC(=O)C3CCCCC3 JFD02501 c1cc(ccc1C(=O)N2CCC(CC2)NC(=O)C3CCCCC3)[N+](=O)[O-] JFD02505 C1CCC(CC1)C(=O)NC2CCN(CC2)C(=O)C3CCC3 JFD02506 c1ccc(cc1)CC(=O)N2CCN(CC2)Cc3ccccc3 JFD02510 c1c(cc(cc1C(F)(F)F)S(=O)(=O)N2CCC(CC2)NC(=O)C3CCCCC3)C(F)(F)F JFD02511 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCC(CC2)NC(=O)C3CCCCC3 JFD02512 c1ccc-2c(c1)CCc3c2c-4c(c(c3)C#N)CCc5c4cccc5 JFD00068 CSc1cc(nn1C(=O)c2ccc(cc2)Cl)c3ccc(cc3)Oc4ccccc4 CD11960 COc1ccc(cc1)NC(=S)NNC(=NS(=O)(=O)c2ccccc2)NNC(=S)Nc3ccc(cc3)OC CD03272 CC(C)(c1cc(cc(c1)C(F)(F)F)C(F)(F)F)O DP01726 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)OC(F)(F)F JFD01027 c1ccc(cc1)c2cc(=O)c3ccc(cc3o2)OCCCCC#N JFD00150 COc1cc(c(cc1Cl)OC)NC(=S)N(CCO)N DP01662 CC(C)(C)NC(=O)c1ccccc1NC DP01665 c1ccc(cc1)c2cn3c(n2)sc(n3)C(F)(F)F DP01669 CCOc1cc(nc(n1)SCc2ccc(cc2)[N+](=O)[O-])c3ccccc3 GK00497 c1ccc2c(c1)ccc3c2ccc(c3C#N)Cc4cc(c5ccc6ccccc6c5c4)C#N JFD00064 c1ccc2c(c1)ccc3c2cc(cc3C#N)CCCCc4cc(c5ccc6ccccc6c5c4)C#N JFD00065 CCOC(=O)c1cc(cc(c1)C(=O)OCC)CCCCc2cc(cc(c2)C(=O)OCC)C(=O)OCC JFD00066 CCOC(=O)c1c2c(sc1NC(=O)COc3ccccc3)CCCC2 DP01675 Cc1ccccc1NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2 JFD01000 c1c(c(c(c(c1Cl)Cl)I)Cl)Cl DP01708 COc1ccc(cc1OC)C(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O DP01709 C/C(=N\NC(=S)Nc1ccc(cc1)F)/c2ccco2 DFP00091 CC(C)c1ccc(cc1)NC(=S)N/N=C(\C)/c2ccco2 DFP00097 Cn1c2ccccc2n3c1c(c(=O)c4c3nccc4)C#N JFD01861 COC(=O)c1c(cc(s1)c2ccccc2)NC(=O)C(Cl)(Cl)Cl GK00502 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccc(cc1)F JFD01017 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)NCc1ccccc1 JFD01020 c1cc(ccc1CSCC(=O)Nc2ccsc2C(=O)N)Cl GK00513 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccccc1 JFD01022 Cc1ccc(cc1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)C JFD01023 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)F JFD01024 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(c(c1F)F)F JFD01034 c1ccc(cc1)N2C(=Nc3ccccc3C(=O)N2)SCc4ccccc4Cl DP01855 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)O DP01857 c1cc(ccc1NC(=O)c2cc(sc2)[N+](=O)[O-])Cl DFP00056 C1CS(=O)(=O)CCN1CC(=O)O DFP00008 c1cc(ccc1CC(C(=O)O)N2CCS(=O)(=O)CC2)O DFP00009 CC(=O)Oc1coc2c1cccc2OC JFD02803 c1ccc(cc1)C2CNN=C2C(=O)c3ccc4ccccc4c3 JFD01094 COC(=O)NCc1ccccc1 JFD01099 CCN(CC)CCNC(=O)c1ccc(cc1)N JFD01780 CCOC(=O)/C(=C/c1cc(sc1)[N+](=O)[O-])/C#N DFP00018 c1c(csc1[N+](=O)[O-])C=C(C#N)C#N DFP00019 c1ccc(cc1)c2csc(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F DP01684 COc1ccccc1N2CCN(CC2)C(=O)c3ccc(cc3Cl)Cl JFD01730 CC(C)(C)NCC(c1ccc(cc1)[N+](=O)[O-])O JFD01784 c1cc(oc1)C(=O)OCCCCCOc2ccc(cc2)Cl JFD01731 CC(C)(C)n1c(n[nH]c1=S)c2ccncc2 DP01756 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)N GK00598 COC(=O)c1cnc(nc1C(F)(F)F)N2CCOCC2 GK01835 CN(C)/C=C/C(=O)c1ccc(cc1)Sc2ccccc2 CD11950 Cc1c(nccn1)c2ccn[nH]2 CD11962 c1ccc(cc1)n2c(c(cn2)C(=O)NN)C(F)(F)F GK02031 COC(=O)c1cccc(c1)NC(=O)c2ccccc2Cl DFP00255 COC(=O)c1cccc(c1)NC(=O)c2ccc(cc2)Cl DFP00256 CCOC(=O)c1ccc(cc1)NC(=O)c2ccccc2NC(=O)c3ccccc3Cl DP01795 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)c2ccc(cc2)[N+](=O)[O-] JP00177 c1ccc(cc1)n2c(c(cn2)C(=O)NNC(=O)C(Cl)Cl)C(F)(F)F GK02070 c1ccc(cc1)CCn2c(n[nH]c2=S)c3ccncc3 DP01759 c1ccc(c(c1)C(=O)NCc2ccccn2)Cl DP01764 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] DP01639 c1cc(c(cc1Cl)NC(=S)N(CCO)N)Cl DP01643 c1ccnc(c1)CNC(=O)c2cccc(c2)Cl DP01766 CC(=O)N1CCC(CC1)C2=NNC(=O)C2/N=N/c3ccc(cc3F)F CD12048 CC(=O)N1CCC(CC1)C2=NNC(=O)C2/N=N/c3ccccc3SC CD12053 COc1ccc(cc1)C2CNN=C2C(=O)c3ccc4ccccc4c3 JFD01098 CCSC(=O)NCc1ccccc1 JFD01101 Cc1cc(sc1)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK02002 Cc1cc(sc1)NC(=O)Nc2ccc(cc2)C(F)(F)F GK02006 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1cccc(c1)C JFD01013 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccc3OC JFD01738 c1(nnc(s1)N)C(F)(F)F DP01661 Cc1nn(c(=N)s1)Cc2ccccc2Cl.Cl DP01663 c1ccc(cc1)CNC(=O)NCc2ccccc2 JFD01107 CCC(=O)c1c[nH]c2c1cccc2 JFD02818 Cc1cc(sc1)NC(=O)Nc2ccc(cc2Cl)Cl GK02007 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)N3CCOCC3 GK01934 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)Sc3ccccn3 GK01985 CCNCC(c1ccc(cc1)[N+](=O)[O-])O JFD01782 CCOC(=O)C1=C(N(C(=O)N(C1c2ccccc2)C)C)C JFD02827 COc1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3OC JFD01739 COC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01839 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)Sc3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01906 Cc1ccc(cc1)S(=O)(=O)OCC(C)(C)[N+](=O)[O-] JFD02758 c1cc(sc1)CN2CCS(=O)(=O)CC2 DFP00070 CC(C)(C)c1ccc(cc1)C(=O)Oc2ccsc2C(=O)OC GK01916 COc1cccc2c1OCC2=O JFD02807 c1ccc(c(c1)C(=O)N/N=C/c2cc(ccc2O)Br)NC(=S)N/N=C/c3cc(ccc3O)Br DP01736 CN(c1ccccc1[N+](=O)[O-])/N=C/c2cc(cc(c2O)Cl)Cl DP01904 CC1CC(CC(C1)(C)C)NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F DP01905 CC(c1ccccc1)NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F DP01907 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)N2CCC=CC2 DP01909 CC1(CC1(C)C(=O)[O-])C(=O)[O-].[K+].[K+] JFD02761 CCC1(CCCCN(C1=O)C)c2cccc(c2)OS(=O)(=O)c3ccc(cc3)C#N JFD02600 c1cc2c(cc1/C=N/OC(=O)c3ccc(cc3Cl)Cl)OCO2 JFD02712 COC(=O)c1cnc(nc1C(F)(F)F)N/N=C/C=C/c2ccccc2 GK01894 CCc1c(cc(s1)C(C)(C)C)NC(=O)C GK01851 COC(=O)c1c(ccs1)OC(=O)c2ccc(cc2Cl)Cl GK01917 c1ccc(cc1)N/C=C/C=C/C=N/c2ccccc2.Cl JFD02765 c1ccc(cc1)c2c3ccccc3c(o2)c4ccccc4 JFD02768 c1cc(cc(c1)C#N)CSc2ncnc(n2)N JM00335 c1cc(c(c(c1)Cl)CSc2ncnc(n2)N)F JM00336 c1ccc(c(c1)CSc2nccc(n2)O)Cl JM00408 CCCc1cc(nc(n1)SCc2ccccc2Cl)O JM00418 CC(C)c1ccc(cc1)Nc2ncc(c(n2)C(F)(F)F)C(=O)OCc3ccc(cc3)Cl GK02055 CCN(CC)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 JFD02774 c1nnc(s1)NC(=S)N DP01875 c1ccc(cc1)CN2CCS(=O)(=O)CC2 DFP00030 c1ccc(cc1)c2ncc3n2cccc3 DP01774 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3nnc(s3)C(F)(F)F DP01781 Cc1cc(c(cc1OC)CCc2cc(c(cc2OC)C)OC)OC JFD02771 c1cc(c(c(c1)Cl)C(=O)O/N=C/c2ccc3c(c2)OCO3)Cl JFD02713 c1cc(ccc1C(=O)O/N=C/c2ccc3c(c2)OCO3)Cl JFD02715 c1cc(ccc1C(=O)O/N=C/c2ccc3c(c2)OCO3)[N+](=O)[O-] JFD02719 CC(C)NS(=O)(=O)NC(C)C JFD02763 c1ccc(cc1)CS(=O)(=O)c2ccccc2 JFD02766 COC(=O)c1cnc(nc1C(F)(F)F)NN2C(=O)CCC2=O GK01927 Cc1cc(sc1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01999 Cn1c(c(cn1)NC(=O)Nc2cc(ccc2Cl)Cl)n3cccc3 GK00623 CCCCNC(=O)NNc1cc(c(c(n1)N(C)C)C#N)N(C)C GK00627 CN(C)c1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 JFD02773 CC(=O)Oc1c2ccccc2n(c(=O)c1I)C JFD02846 Cc1ccc(cc1)S(=O)(=O)NCc2ccccn2 DP01796 c1cc(c(cc1[N+](=O)[O-])Cl)N2CCOCC2 DP01803 c1cc(c(cc1N)Cl)N2CCOCC2 DP01809 c1cc(ccc1NC(=O)O/N=C(\c2cc(sc2)[N+](=O)[O-])/N)Cl DFP00026 CCN(CC)CCSCC(=O)Nc1c(=O)c2ccccc2oc1c3ccccc3.C(=O)(C(=O)O)O JFD00166 CCOC(=O)C1=C(NC(=O)NC1c2cccc(c2)OC)C JFD01805 C=C(c1ccc(cc1)Cl)NCc2cccnc2.I DP01771 Cc1ccc(cc1)N2C(=O)Cc3ccc(cc3C2=O)OC JFD01789 COc1ccc(cc1)C=C2C(=O)N(C(=O)N(C2=O)c3ccccc3)c4ccccc4 JFD02772 C1C2N(C(S1)CS2)NC(=S)N JM00037 CC(C)(C)c1cc(c(s1)C(=O)OC)NC(=O)Nc2ccc(cc2)Cl GK00700 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)N3CCSCC3 GK01935 CC(C)NC(=O)NNc1cc(c(c(n1)N(C)C)C#N)N(C)C GK00630 C=C(c1ccc(cc1)Cl)NCc2ccco2.I DP01773 c1ccc(cc1)CNS(=O)(=O)c2cc(c(cc2N)Cl)S(=O)(=O)N JFD01751 CN1c2ccccc2C(=O)N3C1=NCC3 DP01776 c1ccc2c(c1)c(=O)c(c(o2)c3ccc(cc3)Cl)N JFD01063 c1c(csc1[N+](=O)[O-])C(=O)O DFP00046 c1cc(ccc1CSc2ncnc(n2)N)Cl JM00334 CNc1ccccc1C(=O)NN DP01747 c1c(csc1[N+](=O)[O-])C#N DFP00020 CC(=O)O/N=C(\c1cc(sc1)[N+](=O)[O-])/N DFP00022 c1ccc(c(c1)C(=O)NCCCNC(=O)c2ccccc2N)N DP01957 c1c(cc(cc1C(F)(F)F)NC(=O)c2cc(sc2)[N+](=O)[O-])C(F)(F)F DFP00054 c1ccc(cc1)CCNC(=S)NNC(=O)c2ccncc2 DP01755 Cc1ccc2c(c1)CCCN2C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F DP01910 c1ccc(cc1)CNC(=O)NC2CCCCC2 JFD00125 c1ccc(cc1)CN2CCN=C2NNC(=O)c3cccc(c3)Cl DP01964 CCCCCn1c(n[nH]c1=S)c2ccncc2 DP01757 Cc1cc(c(c(c1Cl)C)Cl)OCc2csc(n2)C CD12016 c1ccc(c(c1)C(=O)NNC(=O)c2ccccc2Cl)Cl JP00137 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)N3CCSCC3)Cl GK02037 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)Nc3ccc(cc3)F)Cl GK02043 Cc1cc(sc1)C(=O)Nc2cccc(c2)C(F)(F)F GK01995 c1ccc(cc1)n2c(c(cn2)C(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F GK02082 CC1CN(CC(O1)C)c2ncc(c(n2)C(F)(F)F)C(=O)OCc3ccc(cc3)Cl GK02038 Cc1cc(c(cc1OC)c2cc(c(cc2OC)C)OC)OC JFD02749 CCC1(CCCCN(C1=O)C)c2cccc(c2)OS(=O)(=O)c3cc(c(cc3Cl)Cl)C JFD02591 Cc1cc(c(c(c1)C)N=C=Nc2c(cc(cc2C)C)C)C JFD02752 c1ccc(cc1)[C@H]2[C@H](N=C(N2)c3ccccc3)c4ccccc4 JFD02754 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)c4cccc(c4)C(F)(F)F DP01564 CCOC(=O)c1c2c(sc1NC(=O)C)CCCC2 DP01565 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=S)N DP01682 COc1ccc(cc1)C2CC(=O)c3cc(ccc3O2)Cl JFD00171 COC(=O)c1c(c(c(s1)Br)Br)OC(=O)c2ccc(cc2Cl)Cl GK01959 COC(=O)c1cnc(nc1C(F)(F)F)Nc2ccccc2 GK01961 COC(=O)c1cnc(nc1C(F)(F)F)Sc2ccccn2 GK01964 CC12CC3(CC(C1)(CC(C2)(C3)Br)C)C JFD02928 c1c(c(nc(n1)N2CCOCC2)C(F)(F)F)C(=O)OCC3CC3 GK02052 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01966 c1cc(ccc1C(F)(F)F)NC(=O)Nc2c(ccs2)Cl GK01970 c1cc(ccc1NC(=O)Nc2c(ccs2)Cl)F GK01971 c1ccc2c(c1)c(=O)oc(n2)COc3ccc(cc3Cl)Cl DP01614 c1cc(c(cc1CSC2=NCN(CN2)CCO)Cl)Cl.Cl DP01615 c1ccc(c(c1)C(=O)C(C#N)c2[nH]c3ccccc3n2)Cl JFD01854 c1ccc(c(c1)C(=O)NCc2ccccn2)N DP01707 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cccc(c1)F JFD01025 Cc1csc(c1NNS(=O)(=O)c2ccc(cc2)C(F)(F)F)C(=O)OC GK01791 Cc1cccc2c1oc(=O)c(c2O)NC(=O)c3c(onc3c4ccccc4)C JFD00200 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3cccnc3 JFD02788 CC(C)c1ccc(cc1)NC(=O)C DP01941 COC(=O)c1ccc(o1)Oc2cc(cc(c2)Cl)Cl JM00046 c1ccc(cc1)Oc2ccc(cc2)c3cc([nH]n3)N4CCOCC4 CD12001 Cc1nc(cs1)CO/N=C(\c2ccc(cc2)C(F)(F)F)/N CD12023 Cc1csc2c1[nH]c(=S)n(c2=O)C GK01823 c1ccn2c(c1)cnc2c3ccc(cc3)[N+](=O)[O-] DP01793 CCOC(=O)c1c[nH]nc1C(F)(F)F GK00722 C1[C@H]([C@@H](CSS1)O)O JFD01841 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)c2cc(c(c(c2)OC)OC)OC JP00139 CNc1ccccc1C(=O)NNC(=O)c2ccccc2 DP01962 c1ccc(cc1)CN2CCN=C2NNC(=O)c3ccccc3 DP01963 c1cc(c(cc1F)F)CN2CCS(=O)(=O)CC2 DFP00061 c1cc(ccc1CSCCS(=O)(=O)CCSCc2ccc(cc2)Cl)Cl DFP00063 Cc1c(=O)c2ccccc2oc1c3ccccc3 JFD00157 COc1ccc(c(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)OC GK01815 COc1ccc(c(c1)NC(=O)Nc2cccc(c2)C(F)(F)F)OC GK01817 COC(=O)c1c(ccs1)OC(=O)c2ccc(cc2)Cl GK01893 C/C(=N\OC(=O)c1ccc(cc1)C(C)(C)C)/CCc2ccc(c(c2)OC)OCc3ccc(c(c3)Cl)Cl JFD02571 CCC1=CC(=O)C=C(C1=O)CC JFD02728 c1cc2cccc3c2c(c1)CC3=O JFD00083 COc1ccc2c(c1)cccc2OC JFD00084 Cc1ccc(cc1)C(=O)C2=NNCC2c3ccc(cc3Cl)Cl JFD01092 CC(C)c1ccc(cc1)[C@H]2[C@@H](C(=O)c3ccccc3O2)OS(=O)(=O)C JFD00183 c1ccc2c(c1)c3c(c4c2nc5ccccc5s4)oc6cc7c(cc6n3)nc8c9ccccc9c1c(c8o7)sc2ccccc2n1 JFD00243 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)N3CCCCC3)Cl GK02039 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1cccc(c1)C(F)(F)F JFD01029 c1ccc(cc1)C2=C(C(=O)c3ccccc3S2(=O)=O)Cc4ccc(cc4)c5[nH]nnn5 JFD00136 Cc1cc(=O)c2ccc(cc2o1)O JFD00137 CNc1ccc(cc1C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)Cl DP01826 CNc1ccc(cc1C(=O)N/N=C/c2ccc(cc2)N(C)C)Cl DP01827 Cn1c(c(cn1)NC(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N)n3cccc3 GK00653 CC(C)(C)OC(=O)N/C(=N/C(=O)OC(C)(C)C)/SC JFD02790 c1[nH]c2c(n1)c(ncn2)N3CCOCC3 JFD02793 Cc1ccccc1/C=C/2\C(=O)c3ccccc3S2 JFD00186 Cc1cccc(c1)/C=C/2\C(=O)c3ccccc3S2 JFD00187 CSc1cc(nc(c1)c2cccs2)c3ccncc3 GK00584 CC(C)(C)c1cc(c(s1)C(=O)OC)NC(=O)C(Cl)(Cl)Cl GK00675 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccccc1C(F)(F)F JFD01030 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(c(c1)Cl)F JFD01031 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccccc1 JFD01011 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccc(cc1)C JFD01012 CN1c2ccc(cc2C(=O)NNC1=S)Cl DP01830 c1ccc2c(c1)C(=O)NNC(=N2)SCc3ccc(cc3)Br DP01840 COCOc1ccc(cc1)C(=O)CC(=O)c2ccccc2O JFD00128 CSc1cc(nc(c1)c2ccco2)c3ccc(cc3)Cl GK00594 CC(C)C(=O)Nc1[nH]c(=O)c2c(n1)n(cn2)[C@H]3CC([C@H](O3)COC(c4ccccc4)(c5ccc(cc5)OC)c6ccc(cc6)OC)O JFD01821 Cc1cn(c(=O)[nH]c1=O)[C@H]2CC([C@H](O2)COS(=O)(=O)c3c(cc(cc3C(C)C)C(C)C)C(C)C)O JFD01836 c1[nH]c2c(n1)c(ncn2)NCC(=O)O JFD02795 CC(C)(C)OC(=O)N1CCN(CC1)Cc2ccccc2 JFD02796 COc1ccc(cc1)c2cc(=O)c3c(o2)cc(cc3OC)OC JFD02797 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)NNS(=O)(=O)c3ccc(cc3)Cl GK01975 c1cc(ccc1CN)C(=O)NN JFD01774 CCOC(=O)c1c(csc1NC(=O)/C(=C/c2ccc(cc2)O)/C#N)C GK00573 CC1CN=C(S1)N(c2ccc(cc2)Cl)C(=O)NC JFD00993 COc1ccccc1N2CCN(CC2)C(=O)c3cccs3 JFD01728 c1ccc(cc1)n2c(=S)n(nn2)CO JFD01888 c1cc(ccc1/C=N/N2CCOCC2)Cl DFP00218 c1cc(ccc1c2cncn2N3CCCCC3)Cl DFP00220 c1ccc(cc1)/C(=N/O)/c2ccccc2/N=C/c3cc(ccc3O)Br JP00303 CCc1c(cc(s1)C(C)(C)C)NC(=O)c2ccccc2 GK02015 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2NS(=O)(=O)c3ccc(cc3)C JFD01184 CC(C)NC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] JFD01188 COC(=O)c1cccc(c1)NC(=O)Nc2ccc(cc2Cl)Cl DFP00272 CC1c2ccsc2CCN1C(=S)NC(=O)c3ccccc3Cl DFP00274 Cc1cc(c(c(c1)Br)N2C(=O)C=CC2=O)Br GK02019 CNCC(c1ccc(cc1)[N+](=O)[O-])O JFD01783 CC(=O)N1CCC(CC1)C2=NNC(=O)C2/N=N/c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD12047 Cc1cc(nc(n1)NNC(=O)CC(=O)NNc2nc(cc(n2)C)C)C JFD01845 Cn1c2ccccc2nc1c3c4ccc(cc4c(=O)n(c3N)Cc5ccccc5)[N+](=O)[O-] JFD01849 c1ccc(cc1)CN2CC(CN(C2)Cc3ccccc3)c4nnn(n4)C(=O)Nc5ccccc5 CD12049 c1c(csc1[N+](=O)[O-])/C=N/N2CCOCC2 DFP00002 CC(=O)N1CCC(CC1)C2=NNC(=O)C2/N=N/c3ccc(cc3)OC CD12050 C/C(=C\C(=O)O)/C=C/c1cccnc1 JFD01146 c1c(cc(cc1C(F)(F)F)Sc2ncc(c(n2)C(F)(F)F)C(=O)OCC3CC3)C(F)(F)F GK02017 c1ccc(cc1)n2c(nnn2)S/C(=C/C=C(C#N)C#N)/c3ccc(cc3)Cl JFD00261 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ncccn2 JFD02937 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2cn(nc2C(F)(F)F)C)/N GK00806 CC(=O)Nc1ccc(cc1)F DP01919 COC(=O)c1ccccc1NC(=S)N(CCO)N DP01685 Cc1ccc(cc1)NC(=O)CC2C(=O)N(CCN2)Cc3ccccc3 DP01689 c1cc(ccc1NC(=O)C2C3CC(C2C(=O)O)C=C3)Cl DP01691 c1ccc(cc1)C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3 DP01812 CC1=CC(=O)N(C1=O)Nc2ncc(c(n2)C(F)(F)F)C(=O)OC GK01905 CN(C)C(=O)Nc1ccc(cc1)Cl JFD01116 c1cc(cc(c1)[N+](=O)[O-])c2nnc(o2)c3cccc(c3)Cl DFP00241 CCOC(=O)c1cnc2ccc(cc2c1O)Cl DFP00243 CC(=O)NNC(=O)c1cccc(c1)[N+](=O)[O-] DFP00246 COC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)C(Cl)Cl GK01913 c1ccc(cc1)C2CS(=O)(=O)C(=CNc3ccccn3)S(=O)(=O)C2 JFD01895 c1ccc(c(c1)CSc2nc(nc(n2)O)c3ccc(cc3)Cl)Cl JM00125 Cc1cccc2c1N(CCC2)C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F DP01911 CSc1nnnn1c2ccccc2 JFD01899 c1ccc(c(c1)C(=O)c2cc3cc(ccc3o2)Cl)Cl DP02006 c1ccc(cc1)NC(=O)/C=N/O JFD01130 c1ccc(cc1)Sc2ccc(cc2Cl)[N+](=O)[O-] DP01922 CC(=O)Nc1ccc(cc1[N+](=O)[O-])F DP01929 C1CCC(CC1)C(C(=O)O)N.Cl JFD01160 c1ccc(c(c1)C(=O)NNc2cc(cc(c2)Cl)Cl)N DP01932 CCC(C)C(C(=O)NCC(=O)O)NC(=O)OCc1ccccc1 JFD01126 CC(C)(C)CC(=O)NC(C)(C)C JFD01770 c1ccc(cc1)C2C(=O)NC(=O)N2 JFD01132 c1cc(oc1)COC(=O)c2cnc(nc2C(F)(F)F)Nc3ccc(cc3)OC(F)(F)F GK02096 CC(C)c1ccc(cc1)Nc2ncc(c(n2)C(F)(F)F)C(=O)OCc3ccco3 GK02097 Cc1c(c(c(c(c1C)C)CSc2ccccc2N)C)C JP00411 C/C(=C\C(=O)O)/C=C/c1cccnc1.Cl JFD01148 Cc1ccc(cc1[N+](=O)[O-])NC(=O)/C=C/c2ccc(cc2)Cl JP00318 Cc1ccc(cc1)Sc2ncc(c(n2)C(F)(F)F)C(=O)OCc3ccc(cc3)Cl GK02008 COC(=O)c1c(c(cs1)Br)OC(=O)c2ccc(cc2)Cl GK01946 c1cc2c(cc(c3c2c4c1c(cc(c4cc3)S(=O)(=O)[O-])O)S(=O)(=O)[O-])S(=O)(=O)[O-].[Na+].[Na+].[Na+] JFD02789 Cc1cc(c(c(c1)Br)N2C(=O)CCC2=O)Br GK02018 COC(=O)c1cscc1NC=C(C#N)C#N GK02025 C=CCN1Cc2ccc3ccccc3c2-c4c(ccc5c4cccc5)C1 JFD02817 CC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2N JP00415 c1ccc2c(c1)C(OC2=O)Nc3ccccc3Sc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-] JP00440 c1cc(cc(c1)C(F)(F)F)c2nnc(o2)c3ccncc3 DP01994 CC(C)c1cccc(c1N=C=Nc2c(cccc2C(C)C)C(C)C)C(C)C JFD02966 CCCc1c(cnn1C)C(=O)Nc2ccc(cc2)Cl GK00818 Cn1c(cc(n1)O)Nc2ccccc2 JM00017 CCCc1c(cnn1C)C(=O)Nc2cc(ccc2F)F GK00822 CC(C)(C)c1cc(c(s1)C(=O)OC)NC(=O)NC(=O)c2c(cccc2Cl)Cl GK00725 Cc1nnc(s1)NC(=S)N DP01877 c1ccc(c(c1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)N DP01887 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)Cl)N3CCOCC3 DP01822 c1ccnc(c1)CNC(=O)c2cc(ccc2N)Cl DP01705 c1ccc2c(c1)ccc3c2/C(=N/NC(=S)N)/CCO3 DP01891 c1ccc2c(c1)ccc3c2/C(=N/O)/CCO3 DP01895 c1ccc2c(c1)ccc3c2/C(=N/NC(=O)N)/CCO3 DP01896 c1cc2c(cc1C(=O)O)OCCCO2 CC13201 c1cc(ccc1C(=O)O/C=C/C(=O)c2ccc(cc2)F)C(F)(F)F JFD00266 CCCc1c(cn(n1)C(=O)c2ccco2)C(=O)OCC GK00797 c1cc(ccc1S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl DP02035 CC(c1ccccc1)NC(=O)c2cc(cc\3c2-c4ccc(cc4/C3=N\O)[N+](=O)[O-])[N+](=O)[O-] JFD01195 Cc1csc2c1c(ncn2)NCCc3ccc(cc3)Cl GK02176 CC(=O)C1=CN(C=C(C1c2ccccc2)C(=O)C)c3ccccc3 JFD00211 c1ccc(cc1)Cn2cncc2c3ccccc3O DFP00126 c1ccc2c(c1)C(=O)[C@H]([C@@H](O2)c3ccc(cc3)Cl)O JFD00177 c1ccc(cc1)/C=C/2\C(=O)c3ccccc3S2 JFD00185 Cc1n(c2c([n+]1C)C(=O)c3ccccc3C2=O)c4ccccc4.[I-] JFD01855 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)OCC(C(F)F)(F)F JFD01196 CCCCNS(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)NCCCC)C2=O JFD01199 CC(C)CCNS(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)NCCC(C)C)C2=O JFD01200 c1cc(c(c(c1)Cl)NC(=O)Nc2cc(sc2)[N+](=O)[O-])Cl DFP00173 c1cc(ccc1c2cnco2)NC(=O)NC(=O)c3ccc(cc3)Cl DFP00212 COc1cc(cc(c1OC)OC)/C=C/C(=O)Nc2ccc(c(c2)Cl)Cl JP00323 COc1cc(cc(c1OC)OC)/C=C/C(=O)Nc2cccc(c2)Cl JP00327 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2ccc(cc2)[N+](=O)[O-] DFP00235 CCOC(=O)C(=CNc1ccc(cc1)Cl)C(=O)OCC DFP00237 COC(=O)c1c(c(c(s1)Br)Br)OC(=O)c2ccc(cc2)Cl GK01957 COC(=O)c1c(c(c(s1)Br)Br)O GK01947 c1c(c(nc(n1)N2CCCCC2)C(F)(F)F)C(=O)OCC3CC3 GK02058 CC1c2ccsc2CCN1C(=O)NC(C)C DFP00157 c1ccc(c(c1)COC(=O)c2cc(cc\3c2-c4ccc(cc4/C3=N\O)[N+](=O)[O-])[N+](=O)[O-])Br JFD01191 Cc1csc2c1c(ncn2)N3CC(OC(C3)C)C GK02162 COC(=O)c1c(c(cs1)Br)OS(=O)(=O)c2ccc(cc2)F GK02171 C[C@H](CCC(=O)O)C1CC[C@@H]2C1([C@H](CC3C2CCC4C3(CC[C@H](C4)O)C)O)C JFD01229 CCCCCCCCCCNS(=O)(=O)c1ccc-2c(c1)C(=O)c3c2ccc(c3)S(=O)(=O)NCCCCCCCCCC JFD01203 C#CCNC(=O)Nc1cc(sc1)[N+](=O)[O-] DFP00176 c1ccc(cc1)C2CC2(C(=O)c3ccccc3)C(=O)c4ccccc4 JFD00206 CCO/C=C\1/c2ccc(cc2C(=O)N(C1=O)c3ccc(cc3)OC)OC JFD01785 c1ccc(c(c1)c2ccc(o2)C=C3C(=O)NC(=O)NC3=O)[N+](=O)[O-] JFD02778 c1ccc(c(c1)C(=O)N/N=C/c2cccnc2)N DP01889 c1ccc(cc1)c2[nH]c(=S)[nH]c(=O)n2 JM00119 CSc1nc(nc(n1)O)c2ccccc2 JM00121 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)Nc3ccc(cc3)F GK02149 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)CC(=O)Nc3ccc(cc3)OC(F)(F)F GK02150 Cc1csc2c1ncnc2SCC(=O)NNC(=O)C(Cl)Cl GK02153 c1ccc(cc1)C(=O)NC(=O)Nc2ccc(cc2)c3cnco3 DFP00210 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc(cc2)c3cnco3)Cl DFP00211 c1ccc(c(c1)/N=C/c2cc(ccc2O)Cl)F DP02032 c1cc(cc(c1)Cl)NC(=O)N/C=C/c2ccco2 GK00877 c1cc(oc1)/C=C/NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00878 c1ccc(cc1)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F DP02036 c1cc(c(cc1Cl)Cl)CSc2nccc(n2)O JM00421 CCCCCCCCCCCCSCc1csc(n1)Cc2ccc(cc2)OC JM00468 Cc1c2ccccc2nc(c1Cl)O JM00483 c1cc(ccc1NC(=O)Nc2cc(sc2)[N+](=O)[O-])Cl DFP00172 c1cc(ccc1c2[nH]nc(n2)CSc3ccc(cc3)Cl)Cl DP01920 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)Br)C JFD01800 CCCNC(=O)O/N=C(\c1cc(sc1)[N+](=O)[O-])/N DFP00028 CS/C(=N/C(=N)Nc1ccc(cc1)Cl)/N.Cl JM00281 CCCNC(=O)Nc1cccc(c1)C(=O)OC DFP00267 CC(C)NC(=O)Nc1cccc(c1)C(=O)OC DFP00268 COC(=O)c1cccc(c1)NC(=O)Nc2ccccc2 DFP00270 COC(=O)c1cccc(c1)NC(=O)Nc2ccc(cc2)Cl DFP00271 c1ccc(c(c1)/C=N/Nc2cccc(c2)C(F)(F)F)O DP02039 c1cc(cc(c1)N/N=C/c2cc(ccc2O)Cl)C(F)(F)F DP02040 CCOC(=O)c1c(c2cc(ccc2s1)NC(=O)c3ccccc3Cl)C DP02042 Cc1cc(=O)oc2c1ccc(c2)OC JFD01814 c1ccc(cc1)N2C(=O)C(=Cc3ccc(cc3)Cl)C(=O)N(C2=S)c4ccccc4 JFD01811 CCOC(=O)c1cn(nc1C(F)(F)F)S(=O)(=O)c2ccc(cc2F)F GK00749 c1cc(ccc1C#N)c2cnco2 DFP00102 COc1ccc(c(c1)[N+](=O)[O-])NC(=S)Nc2ccc(cc2F)F DFP00136 CCCC(=O)O[C@H]1[C@@H](Oc2ccccc2C1=O)c3ccccc3 JFD00180 c1ccc(cc1)C/N=C/c2cc(ccc2O)Cl DP02026 c1cc(ccc1/N=C/c2cc(ccc2O)Cl)F DP02033 COC(=O)c1c(cc(s1)c2ccccc2)NC(=O)CC(=O)C(F)(F)F GK00718 CC(=O)c1c(ccs1)NC(=O)CSCc2ccc(cc2)Cl GK00680 CC(C)(C)c1cc(c(s1)C(=O)OC)NS(=O)(=O)c2ccc(cc2)OC GK00683 CC(C)(C)NC(=O)Oc1ccccc1 JFD00114 CC(C)CNC(=O)Oc1ccccc1 JFD00115 CC1CN(CC(O1)C)c2ncc(c(n2)C(F)(F)F)C(=O)OCC3CC3 GK02057 Cc1ccc(cc1)/C=C/2\C(=O)c3ccccc3S2 JFD00188 c1cc(sc1)CC(=O)Nc2ccc(cc2)OC(F)(F)F GK01980 CC(C)NC(=O)Oc1ccc(cc1)[N+](=O)[O-] JFD00117 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)NNc3ncc(c(n3)C(F)(F)F)C(=O)OCc4ccc(cc4)Cl)Cl GK02059 CCCC(=O)/C(=C/Nc1ccsc1C(=O)OC)/C(=O)OCC GK00747 CCCC(=O)/C(=C\Nc1ccc(o1)C(=O)OC)/C(=O)OCC GK00748 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(CO)CO JFD01833 C=C(C1CC1)N(Cc2ccccc2)C(=O)c3cccc(c3)F JFD01877 CC(=O)N1C(C(=O)NC1=S)c2ccccc2 JFD01131 c1ccc(cc1)/C=N/NC(=N)N JFD01134 COC(=O)CSc1[nH]c(nn1)c2ccc(cc2)Cl DP01847 c1ccc(cc1)N2C(=S)Nc3ccccc3C(=O)N2 DP01852 CC1=CC(=O)OC(C1)c2ccccc2 JFD01159 Cc1c(c(c(c(c1C)C)CSc2ccccc2NC3c4ccccc4C(=O)O3)C)C JP00441 COC(=O)c1c(ccs1)NC(=O)Cc2cccs2 GK01981 CCOC(=O)C(=NNc1cccc(c1)[N+](=O)[O-])C(=O)OCC JFD01796 CCOC(=O)C(=CNc1cc(sc1C(=O)OC)C(C)(C)C)C(=O)OCC GK00698 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)Sc3ccc(cc3)Cl GK01983 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)NNS(=O)(=O)c3ccc(cc3)F GK01986 CCOC(=O)C1=C(NC(=O)NC1c2cc(ccc2OC)Br)C JFD01806 COc1cccc(c1OCC(=O)O)C(=O)O JFD02804 c1ccc(cc1)CN2CCn3c2nc4ccccc4c3=O DP01801 c1ccc(c(c1)C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3)Cl DP01813 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nc(on2)CCC(=O)O DP01820 c1ccc(c(c1)N)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F JP00450 c1ccc2c(c1)C(OC2=O)Nc3ccccc3Sc4ccc(cc4[N+](=O)[O-])Cl JP00444 c1ccc(cc1)C(=O)CCC(=O)c2ccccc2 JFD00234 CC(C)(C)c1cc(c(s1)C(=O)OC)NC(=O)Nc2cc(cc(c2)Cl)Cl GK00702 COCCCn1c(n[nH]c1=S)c2ccncc2 DP01758 c1cc(ccc1C(=N)NCc2ccncc2)Cl.I DP01770 Cc1ccc(cc1)c2c(c(=O)c3ccccc3o2)O JFD00159 COc1ccc(c(c1)OCC(=O)O)C(=O)O JFD02805 Cc1nc(cs1)COc2ccc(cc2)/C(=N/OC(=O)N(C)C)/N JM00492 c1cc(ccc1NC(=O)N/C=C/c2ccsc2)F GK00859 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OCc2ccccc2)OC(=O)C)OC(=O)C)O[C@H]3[C@@H]([C@H]([C@H]([C@H](O3)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD01225 CCOC(=O)/C(=C/Nc1cc(sc1C(=O)OC)C(C)(C)C)/C#N GK00686 Cc1ccc(c(c1)C)C(=O)NNC(=O)c2ccncc2.Cl DP01990 COc1ccc(cc1)c2c(c(=O)c3cc(ccc3o2)Cl)O JFD00161 c1ccc(cc1)C2CC(=O)c3cc(ccc3O2)Cl JFD00169 c1ccc(cc1)C2/C(=C\c3ccc(cc3)c4[nH]nnn4)/C(=O)c5ccccc5O2 JFD00174 c1ccc(cc1)COC(=O)c2cnc(nc2C(F)(F)F)Nc3ccc(cc3)F GK02013 COC(=O)c1cc(ccc1Sc2ccccc2)[N+](=O)[O-] DP01998 COC(=O)c1cc(ccc1Sc2ccc(cc2)Cl)[N+](=O)[O-] DP01999 Cc1ccc(cc1)S(=O)(=O)OC(C)C(C(=O)OC)NC(=O)OCc2ccccc2 JFD02831 c1ccc2c(c1)C(=O)/C(=C\c3ccc(cc3)F)/S2 JFD00191 c1ccc2c(c1)[nH]c(n2)NC(=N)N JFD01760 CCOC(=O)/C(=N/Nc1ccc(cc1)OC)/C(=O)C JFD01762 CC(C)(C)NC(=O)NCc1ccccc1 JFD00123 c1ccc2cc(ccc2c1)C(=O)C3=NNCC3c4ccc(cc4)Cl JFD01095 c1ccc2cc(ccc2c1)C(=O)C3=NNCC3c4ccc(cc4Cl)Cl JFD01096 CCOC(=O)CSc1ccc(cc1Cl)[N+](=O)[O-] DP01987 c1ccc(cc1)C(=O)NNC(=O)c2ccncc2.Cl DP01988 CCOC(=O)C1=C(NC(=NC1c2ccccc2)SC)C JFD02823 C/C(=N\NC(=O)c1ccccc1N)/c2ccccc2O DP01885 COc1ccc(cc1OC)CCNC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F DP01906 c1cc(ccc1/C=N/N2CCCCC2)Cl DFP00219 c1cc(ccc1c2cnco2)NC(=O)C3CC3 DFP00222 c1ccnc(c1)CNC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F DP01908 c1ccc2c(c1)cc3ccccc3c2/C=N/NC(=O)c4ccc(cc4)Br JFD01183 c1ccc(cc1)S(=O)(=O)CCCCCS(=O)(=O)c2ccccc2 JFD01765 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCCCCCCN.Cl JFD02800 CC(=C)c1cccc(c1)C(C)(C)NC(=O)CC(=O)C JFD02802 Cc1cn(c(=O)[nH]c1=O)[C@H]2CC([C@H](O2)COC(c3ccccc3)(c4ccc(cc4)OC)c5ccc(cc5)OC)O JFD01818 CCOC(=O)CSc1nc2ccccc2s1 JFD01768 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OC[C@@H]4C(C[C@@H](O4)n5ccc(nc5=O)NC(=O)c6ccccc6)O JFD01819 CC(=O)Oc1coc2c1ccc(c2)OC JFD02808 COc1ccc(cc1)NC(=O)c2ccccc2NC(=O)c3ccccc3Cl DP01783 c1ccc(c(c1)C(=O)N/N=C/c2cc(ccc2O)Br)N DP01888 COc1ccc2c(c1)sc(n2)NC(=O)CCCCC(=O)Nc3nc4ccc(cc4s3)OC JFD01885 c1ccc(cc1)/C(=N\O)/c2ccccc2NC(=O)c3cccc(c3)[N+](=O)[O-] JP00297 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=O)c3c(onc3c4ccccc4Cl)C JP00138 Cc1cc2ccccc2c(c1C#N)/N=C/c3cccs3 DSHS00335 Cc1c(c(sc1c2ccc(c(c2)OC)OC)/N=C/c3ccc(cc3)c4ccccc4)C#N DSHS00323 Cc1c(c(sc1c2ccc(c(c2)OC)OC)/N=C/c3ccc(cc3)N(C)CCC#N)C#N DSHS00333 CCC(c1ccccc1)C(=O)NNC(=O)c2cc(c(c(c2)OC)OC)OC JP00186 Cc1c(c(sc1c2ccc(c(c2)OC)OC)/N=C/c3cccs3)C#N DSHS00334 CCC(CC)(C#C)NC(=O)c1cc(c(c(c1)OC)OC)OC DSHS00339 CCC(CC)(C#C)NC(=O)COc1cc(c(cc1Cl)Cl)Cl DSHS00341 CCOC(=O)C1=C(NC(=C(C1c2ccccc2OC)C(=O)OCC)C)C JFD01211 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)Sc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl GK02004 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)Sc3ccc(cc3)Cl)Cl GK02005 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)Nc3ccc(cc3)OC(F)(F)F)Cl GK02042 c1ccc2c(c1)C(=O)N(C2=O)c3nc(cs3)c4ccc(cc4)Cl GK02045 Cc1ccc(cc1)C(=O)NNc2c3c(csc3ncn2)C GK02233 c1ccc(cc1)Cn2c(c(c3ccc(cc3c2=O)[N+](=O)[O-])C#N)N JFD01875 Cc1ccc(cc1C)NC(=O)Nc2ccc(cc2)Cc3ccc(cc3)NC(=O)Nc4ccc(c(c4)C)C JFD01881 CC(C)C(=O)Nc1c2c([nH]cn2)ncn1 JFD00287 COc1ccc(cc1OC)CCNC2(CCCCC2)C#N DSHS00036 CC1(O[C@H]2CO[C@H]3[C@@H]([C@H]2O1)OC(O3)(C)C)C JFD00290 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC(=O)C)OC(=O)C)OC(=O)C)O[C@@H]2[C@@H]([C@H]([C@@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00291 CCCCN(CCCC)S(=O)(=O)c1ccc-2c(c1)C(=NO)c3c2ccc(c3)S(=O)(=O)N(CCCC)CCCC JFD01207 CC(C)CCNC(=O)c1cccc-2c1C(=O)c3c2cccc3 JFD01212 Cc1ccc2c(c1)NC(=O)CC(O2)C JFD00293 c1ccc(cc1)C[C@H]2COC(=N2)C3=N[C@@H](CO3)Cc4ccccc4 JFD02812 c1cc(cc(c1)C(F)(F)F)c2ccc(o2)C(=O)O JFD02813 CC(C)(C)NC(=S)NN1C2CSC1CS2 JM00038 CN(C)C(=O)c1ccc(o1)Oc2cc(cc(c2)Cl)Cl JM00090 c1ccnc(c1)Sc2ncc(c(n2)C(F)(F)F)C(=O)OCc3ccc(cc3)Cl GK02009 COC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])Cl GK02093 CC(C)(C)c1ccc(cc1)C(=O)c2[nH]ccn2 JM00132 Cc1cc(=O)[nH]c(n1)N/N=C/c2ccc(cc2)[N+](=O)[O-] JFD01245 c1ccc(cc1)C[C@H](C(=O)O)NC(=O)C(Cl)(Cl)Cl JFD01248 c1ccc(c(c1)C(CO)O)[N+](=O)[O-] JFD01250 c1cc(cc(c1)S(=O)(=O)N2CCCC2)C(F)(F)F JP00278 c1ccc2c(c1)[nH]c(n2)CSCSCc3[nH]c4ccccc4n3 JFD01354 CCOC(=O)C(=CNc1ccccc1Cl)C(=O)OCC JFD01357 CNc1ccccc1C(=O)NNc2ccc(cc2)Cl DP01933 c1ccn(c1)c2ccc(cc2[N+](=O)[O-])F DP01952 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(C4CCCCC4)C(=O)O JFD01161 c1ccc2c(c1)ccc3c2-c4c(ccc5c4cccc5)CNC3 JFD02816 CCOC(=O)c1c(c2cc(ccc2s1)NS(=O)(=O)c3ccc(cc3)C)C DP02043 Cc1c(c(c(c(c1C)C)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)C DP02047 COC(=O)c1c(ccs1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F GK02072 c1ccc(cc1)CNC(=O)CSc2ccc(cc2Cl)[N+](=O)[O-] DP02049 C/C(=N\NC1=NCCN1)/c2ccccc2 DP02064 c1ccc(cc1)n2c(c(cn2)C(=O)NNC(=O)C(F)(F)F)C(F)(F)F GK02073 C/C(=N\NC1=NCCN1)/c2ccc(cc2)Cl DP02065 c1cc(c(c(c1)Cl)CSc2nc(nc(n2)O)c3ccc(cc3)Cl)Cl JM00126 CC(/C=C\c1cc[n+](cc1)C)O.[I-] JFD01153 c1cc(ccc1c2cnco2)N DFP00120 c1cc(ccc1n2c(c(cn2)C(=O)NNS(=O)(=O)c3ccc(cc3)F)C(F)(F)F)Cl GK02106 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)NNC(=O)C(Cl)Cl)Cl GK02109 c1ccc(cc1)CN2CCN=C2NNC(=O)c3ccccc3Cl DP01965 COCc1c[nH]c2c1cccc2 JFD01168 c1ccc2c(c1)c3cc(ccc3[nH]2)Cl JFD01172 COc1ccc(cc1OC)/C(=C/N2CCOCC2)/C#N JFD01179 CCOC(=O)OC(c1ccnc2c1cc(cc2)OC)C3CC4CCN3CC4C=C DSHS00055 CCc1cc2c(cc1C(=O)CCN3CCOCC3)C(CCC2(C)C)(C)C.Cl DSHS00075 c1cc(ccc1C(=O)CCN2CCOCC2)F.Cl DSHS00079 c1c(cc(c(c1/C=N/n2cnnc2)O)Br)Br JFD01208 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl GK02094 COC(=O)c1c(ccs1)Oc2ccc(cc2N)C(F)(F)F GK02095 CC(=O)c1c(cc(s1)C(C)(C)C)NC(=O)CCC(=O)O GK02214 CN(C)c1ccsc1C(=O)NNS(=O)(=O)c2ccc(cc2)Cl GK00705 CN(C)c1ccsc1C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00708 c1ccc2c(c1)cccc2/C=C/C(=O)N(C3CCCCC3)C4CCCCC4 JP00387 CC1CN(CC(O1)C)C(=O)/C=C/c2cccc3c2cccc3 JP00388 c1cc(ccc1S(=O)(=O)c2ccc(cc2Cl)[N+](=O)[O-])Cl DP01985 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2ccncc2.Cl DP01991 Cc1nnc(o1)[C@H]2C(C(C(CO2)OC(=O)c3ccccc3)OC(=O)c4ccccc4)OC(=O)c5ccccc5 JFD01231 CCOc1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl JFD00253 c1ccc(cc1)/C(=N\O)/c2cc(ccc2N)Cl DSHS00142 C[C@H](CCC(=O)O)C1CC[C@@H]2C1(C(=O)C[C@H]3C2C(=O)CC4C3(CCC(=O)C4)C)C JFD01238 Cn1cc(c(n1)C(F)(F)F)NC(=O)Nc2ccc(cc2)Cl GK00837 Cn1cc(c(n1)C(F)(F)F)NC(=O)Nc2ccc(cc2)C(F)(F)F GK00838 c1ccc(cc1)C(=O)O[C@@H]2CSSC[C@H]2OC(=O)c3ccccc3 JFD01840 CCn1c([n+](c2c1cccc2)CC)C.[I-] JFD01846 c1cc(cc(c1)Nc2ncc(c(n2)C(F)(F)F)C(=O)OCc3ccc(cc3)Cl)C(F)(F)F GK02054 c1ccc(cc1)n2c(c(cn2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F)C(F)(F)F GK02062 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(ccs2)N(C)C GK00709 Cc1c(c(n(n1)C)Sc2ccccc2NC(=O)C(Cl)Cl)[N+](=O)[O-] GK00715 CC(=C(C#N)C#N)Cc1ccc(c(c1)OC)OC DSHS00303 CC(C)(C)C(=O)Nc1ccc(cc1C(=O)c2ccccc2)Cl DSHS00309 c1cc(sc1)/C=C/2\C(=O)C3CCN2CC3 DSHS00364 CC(C)(CCO)NC(=O)c1cc(c(c(c1)OC)OC)OC DSHS00383 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)Br)C(=O)OCC)C)C JFD01209 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)OC)C(=O)OCC)C)C JFD01210 c1cc(ccc1c2[nH]c(=S)[nH]c(=O)n2)Cl JM00152 COc1ccc(cc1OC)CCNC(=O)c2ccc(cc2Cl)Cl JFD01864 CCCCCCCCCCNS(=O)(=O)c1ccc-2c(c1)Cc3c2ccc(c3)S(=O)(=O)NCCCCCCCCCC JFD01204 CCC(C)(C)OC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] JFD01205 Cc1csc2c1ncnc2SCC(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F GK02144 CC1c2ccsc2CCN1C(=O)c3ccc(cc3)C(F)(F)F DFP00182 c1ccc(c(c1)c2[nH]c(=S)[nH]c(=O)n2)Cl JM00122 c1ccc2c(c1)[nH]c(n2)Sc3ccc(cc3Cl)[N+](=O)[O-] DP01917 c1ccc2cc(ccc2c1)NC(=O)c3ccco3 JFD01850 c1ccc2c(c1)C(=O)c3c(ccc(c3C2=O)NC4CCCCC4)NC5CCCCC5 JFD00242 c1cc(ccc1C(=O)CCN2CCOCC2)O.Cl DSHS00086 CCc1cc2c(cc1C(=O)CCN3CCCC3)C(CCC2(C)C)(C)C.Cl DSHS00095 c1cc(c(c(c1Cl)Cl)Cl)Cl JFD01285 CCCCCCS(=O)(=O)CC#N JFD01280 CC(C)c1ccc(cc1)S(=O)(=O)CC#N JFD01281 CC1c2ccsc2CCN1C(=O)NC(=O)c3ccc(cc3)Cl DFP00205 c1ccc(cc1)c2nc(cs2)c3cc4cc(ccc4o3)Cl DP02024 CC(c1ccccc1)/N=C/c2cc(ccc2O)Cl DP02027 CC(C)(C)C(=O)Nc1cccc(c1)C(=O)OC DFP00259 COC(=O)c1cccc(c1)NC(=O)C2CC2 DFP00260 CCc1nnc(o1)c2cccc(c2)[N+](=O)[O-] DFP00264 Cc1nnc(o1)c2cccc(c2)[N+](=O)[O-] DFP00265 c1ccc(cc1)/C=C/2\CCc3ccccc3\C2=N\Nc4ccc(cc4[N+](=O)[O-])[N+](=O)[O-] DSHS00178 CC1(C2CCC1(/C(=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])/C2)C)C DSHS00180 Cn1cc(c(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl GK00785 c1c(cc(cc1C(F)(F)F)F)C(=O)O JFD01237 CCCc1c(cn(n1)S(=O)(=O)c2ccc(cc2F)F)C(=O)OCC GK00787 C[C@]1([C@@H](CC2CC1C2(C)C)O)O JFD01247 CCOC(=O)c1cn(nc1C(F)(F)F)C(=O)c2ccco2 GK00798 c1ccc(cc1)/N=c/2\nc(nc(n2c3ccccc3)N)N JFD01239 Cc1cc(=O)[nH]c(n1)N/N=C/c2ccc(cc2OC)OC JFD01244 CCCc1c(cn(n1)C(=O)c2ccc(cc2)Cl)C(=O)OCC GK00802 Cn1cc(c(n1)C(F)(F)F)C(=O)O/N=C(\c2ccc(cc2)Cl)/N GK00805 COc1ccc(cc1OC)CC/N=C/c2cc(ccc2O)Cl DP02028 c1cc(ccc1S(=O)(=O)c2ccc(cc2Cl)/N=C/c3cc(cc(c3O)Cl)Cl)Cl DP02016 CC(C)c1ccc(c(c1)Br)/N=C/c2cc(ccc2O)Br DP02021 c1cc(ccc1c2nc(cs2)c3cc4cc(ccc4o3)Cl)Cl DP02025 COC(=O)c1c(cc(s1)c2ccccc2)NC(=O)CC#N GK00714 Cn1cc(c(n1)NC(=O)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br GK02240 c1ccc(cc1)c2nc(nc(n2)SCc3c(cccc3Cl)F)O JM00210 Cc1cc(sc1)C(=O)NCC(=O)NNS(=O)(=O)c2ccc(cc2)F GK02247 CN(C)c1nc(nc(n1)O)c2ccc(cc2)Cl JM00217 CN(C)c1nc(nc(n1)O)c2ccccc2 JM00221 CC(C)(C)c1ccc(cc1)c2nc(n(n2)C)O JM00243 CC(=O)O[C@@H]1CSSC[C@H]1OC(=O)C JFD01839 CCC(C)C1=CC(=Nc2c(n(n(c2=O)c3ccccc3)C)C)C=C(C1=O)C(C)CC JFD01186 CCCCCCCNC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] JFD01187 c1ccc(c(c1)COC(=O)c2cc(cc3c2-c4ccc(cc4C3=O)[N+](=O)[O-])[N+](=O)[O-])Br JFD01189 CCOC(=O)c1ccc(c(c1)NC(=O)c2c(onc2c3ccccc3Cl)C)N4CCCCC4 JP00645 CCOC(=O)c1ccc(c(c1)NC(=O)c2c(onc2c3ccccc3)C)N4CCCCC4 JP00648 CCOC(=O)c1ccc(c(c1)NC(=O)c2cc(c(c(c2)OC)OC)OC)N3CCCCC3 JP00649 c1ccc2c(c1)C(OC2=O)Nc3ccc(cn3)[N+](=O)[O-] JP00566 Cc1cc(sc1)C(=O)NNC(=O)C(Cl)Cl GK02254 c1ccc2c(c1)c(ccc2F)C(=O)O JFD01253 c1ccc(cc1)c2nnc(o2)c3cccc4c3cccc4 JFD01255 C1CCNC(=O)C(C1)N2CCS(=O)(=O)CC2 DFP00072 C/C(=N\NC(=S)NCC1CCCO1)/c2cccs2 DFP00094 CCOC(=O)c1c(nc(s1)SC)NC(=O)C(Cl)Cl GK00780 CCN(CC)c1ccc(cc1)/C=N/NC(=O)c2ccccc2O JFD01862 c1ccc2c(c1)c3cc(ccc3[nH]2)Br JFD01173 CC(=O)Cc1c[nH]c2c1cccc2 JFD01174 c1cc(c(cc1S(=O)(=O)N2CCOCC2)[N+](=O)[O-])N3CCOCC3 JP00498 c1ccc(cc1)CC(c2ccccc2)NC3(CCCCCC3)C#N DSHS00187 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)CCC(=O)O)[N+](=O)[O-] DSHS00198 COc1cc(c(cc1OC)[N+](=O)[O-])CC#N JFD01178 Cc1ccc(c(c1)C)C(C)NC(=O)C(C)(C)C DSHS00245 Cc1ccc(c(c1)C)C(C)NC(=O)c2ccc(c(c2)Cl)Cl DSHS00250 COc1ccc(cc1)/C=N/NC(=N)N JFD01135 c1cc(c(cc1Cl)Cl)/C=N/NC(=N)N JFD01136 c1ccnc(c1)CNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DP01798 c1cc(ccc1c2cnco2)NC(=O)NC(=O)c3ccc(cc3)C(F)(F)F DFP00213 CC(=C)c1ccccc(=O)c1O GK02122 Cc1cc(sc1)C(=O)O/N=C/c2ccc(cc2Cl)Cl GK02273 COC(=O)c1c(ccs1)Oc2ccc(cc2)[N+](=O)[O-] GK02136 Cc1cc(sc1)C(=O)NCC(=O)NNC(=O)C GK02287 CSc1cc(nn1S(=O)(=O)c2cccc(c2)C(F)(F)F)c3ccc(cc3)F GK02139 CC(C)Cc1ccc(cc1)c2cc(c(s2)C(=O)OC)N GK02141 Cc1cc(sc1)c2nc(no2)c3ccc(cc3)C(F)(F)F GK02280 Cc1nc(cs1)COc2ccc(cc2)/C(=N/O)/N JM00487 c1cc(ccc1c2cc(c(s2)C(=O)N)NC(=O)CCC(=O)O)Cl GK02084 c1cc(ccc1c2cnco2)NC(=O)Nc3ccc(cc3)Cl DFP00215 c1cc(ccc1Sc2ncc(c(n2)C(F)(F)F)C(=O)OCC3CC3)Cl GK02089 Cc1cc(sc1)C(=O)NCC(=O)NNC(=O)c2cccc(c2)Cl GK02244 CCCc1cc(nc(n1)SCc2ccc(cc2Cl)Cl)O JM00428 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=O)CSc3cc(c(cc3OC)[N+](=O)[O-])OC JP00518 CCOC(=O)c1ccc(cc1)N=C(N2CCOCC2)SCc3c(c(c(c(c3C)C)C)C)C JP00551 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCOCC2 JP00568 CCOC(=O)c1ccc(c(c1)N)N2CCOCC2 JP00572 c1ccc(c(c1)/C=N/c2ccc(c(c2)Cl)S(=O)(=O)c3ccc(cc3)Cl)O DP02017 c1cc(c(cc1Cl)c2cc[nH]n2)O JFD01904 Cn1cc2cc(ccc2n1)[N+](=O)[O-] JFD01269 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OC[C@@H]4C(C[C@@H](O4)n5cnc6c5ncnc6NC(=O)c7ccccc7)O JFD01820 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)NC JM00239 Cn1c(nc(n1)c2ccc(cc2)Cl)O JM00242 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OC[C@@H]4C(C[C@@H](O4)n5ccc(nc5=O)N)O JFD01824 CC(=O)c1cc(ccc1Sc2ccccn2)[N+](=O)[O-] DP01970 c1cc(ccc1c2cnco2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl DFP00294 CC1c2ccsc2CCN1C(=S)NC(=O)c3cccs3 DFP00297 Cn1c2c(c3c(cc4cc(ccc4n3)[N+](=O)[O-])c(=O)n2c5ccccc5)c(=O)n(c1=O)C JFD01337 c1cc(ccc1C2CS(=O)(=O)CS(=O)(=O)C2)Cl JFD01340 c1cc(sc1)CCCCC(=O)O JFD01271 Cc1ccc(c(c1)c2cc(ccc2C)C)C JFD01273 Cc1ccc(cc1)NC(=O)Cn2nc(nn2)c3cccc(c3)C(F)(F)F GK02157 c1ccc2c(c1)cc(o2)C(=O)c3ccc(cc3)Cl DP02001 Cc1c2ccccc2oc1C(=O)c3ccc(cc3)Cl DP02002 CC(=O)c1cc2cc(cc(c2o1)Cl)Cl DP02003 CCN(CC)c1cccc(c1)NC(=O)C JFD02921 CNC(=S)N/N=C/1\CCOc2c1c3ccccc3cc2 DP01876 Cc1cccc(c1)OC(=O)Nc2ccc(cc2)Cc3ccc(cc3)NC(=O)Oc4cccc(c4)C JFD01879 c1ccc(cc1)Sc2c(c(c(c(c2Sc3ccccc3)Sc4ccccc4)Sc5ccccc5)Sc6ccccc6)Sc7ccccc7 JFD01880 Cc1ccc(cc1C)Oc2c(c(c(c(c2F)F)Oc3ccc(c(c3)C)C)F)F JFD01882 c1ccc(c(c1)/C=N/NC(=O)c2ccccc2N)O DP01884 Cc1ccc(cc1)S(=O)(=O)NNC(=O)CSc2c3c(csc3ncn2)C GK02146 c1cc(ccc1C(=O)O/N=C(/C2CSCCS2)\N)Cl GK02155 c1ccc(cc1)COC(=O)C(C(C(=O)OCc2ccccc2)O)O JFD00284 CCOC(=O)c1ccc(c(c1)/N=C/c2cc(cc(c2O)Br)Br)N3CCOCC3 JP00574 CN(c1ccccc1C(=O)OC)C(=O)c2cc(c(c(c2)OC)OC)OC JP00030 CCOC(=O)c1ccc(c(c1)/N=C/c2cccc(c2O)OC)N3CCOCC3 JP00575 CCOC(=O)c1c2c(sc1N)CCCC2 DSHS00273 CCOC(=O)c1ccc(c(c1)/N=C/c2cc(ccc2O)Cl)N3CCOCC3 JP00576 c1cc(ccc1C(=O)NNC(=O)C(=O)NNC(=O)c2ccc(cc2)Cl)Cl JP00163 CCSC(=O)NC1CCCCC1 JFD01103 c1ccc(cc1)c2nnc(o2)c3cccc(c3)[N+](=O)[O-] DFP00239 c1cc(ccc1NC(=O)NC2CCCCC2)Cl JFD01113 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)O JFD01115 c1ccc(cc1)Oc2ccc(cc2)OC(=O)c3cccs3 JFD01374 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)Oc3ccccc3 JFD01375 COC(=O)c1cccc(c1)NC(=S)NCC=C DFP00329 Cc1cc(sc1)C(=O)NNC(=O)c2cc(cc(c2)Cl)Cl GK02263 c1ccc(cc1)CNC(=O)CNC(=O)CSc2nc3ccccc3s2 JFD02016 CC1c2ccsc2CCN1S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F DFP00363 CC1c2ccsc2CCN1S(=O)(=O)C DFP00364 c1ccc(cc1)C2=C(c3ccccc3C2=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F DMP00010 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)c2ccc(c(c2)Cl)Cl JP00187 COc1ccc(cc1OC)CCNC(=O)CSc2ccc(cc2Cl)[N+](=O)[O-] DP02050 c1cc(c(c(c1)Cl)CSc2nccc(n2)O)F JM00416 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(C)(C)CCO DSHS00348 Cc1cc(ccc1Nc2c(c(c(s2)C(=O)c3cc4cc(ccc4o3)Cl)N)C#N)Cl DP02063 c1ccc\2c(c1)CCC/C2=N\NC3=NCCN3 DP02066 Cc1cc(sc1)C(=O)NNC(=O)Cc2ccccc2 GK02265 Cc1cc(sc1)C(=O)O/N=C(/c2ccc(cc2)C(C)(C)C)\N GK02269 CCOC(=O)c1c(c(sc1NCc2ccccc2)C(=O)c3ccc(cc3)Br)N DP00026 c1ccc2c(c1)cccc2/C=C/C(=O)N3CCOCC3 JP00386 COc1ccc(cc1)/C=C/C(=O)N2CCOCC2 JP00398 CC1c2ccsc2CCN1C(=O)c3ccco3 DFP00311 COC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(cc2)Cl DFP00314 CCC(CC)(C#C)NC(=O)/C=C/c1ccccc1 DSHS00346 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC(=O)C)OC(=O)C)OC(=O)C)O[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00292 CCCc1c(cn(n1)C)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N GK00844 c1cc2c(cc1/C=N/NCCC#N)OCO2 DSHS00013 C([C@@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)NN=C(N)N)O)O)O)O.N(=O)(=O)O JFD01241 C1[C@H](NC(S1)[C@@H]([C@@H]([C@H]([C@H](CO)O)O)O)O)C(=O)O JFD01243 c1ccc(cc1)Nc2nn(c(=S)n2c3ccccc3)CN4CCCCC4 JFD01893 CCOC(=O)CSc1nnnn1c2ccccc2 JFD01897 CCOC(=O)c1c(c(sc1Nc2ccccc2OC)C(=O)c3ccccc3)N DP00028 COC(=O)c1cccc(c1)NS(=O)(=O)c2cc(cc(c2)Cl)Cl DFP00316 COC(=O)c1cccc(c1)NC(=S)Nc2ccccc2Cl DFP00317 c1ccc2c(c1)cccc2/C=C/C(=O)N3CCCCC3 JP00399 CCN(CC)c1ccc(c(c1)O)/N=N/c2ccc(cn2)Br JFD01902 COc1cc(cc(c1OC)OC)/C=C/C(=O)Nc2ccc(cc2)F JP00328 c1cc(cc(c1)Cl)NC(=O)/C=C/c2ccc3c(c2)OCO3 JP00340 c1ccc(cc1)NC(=O)/C=C/c2ccccc2Cl JP00366 COc1cc(cc(c1OC)OC)NC(=O)/C=C/c2ccccc2Cl JP00368 c1cc(cc(c1)[N+](=O)[O-])c2nnc(o2)c3ccc(cc3)Cl DFP00240 CC(C)NC(=O)NNC(=O)c1cccc(c1)[N+](=O)[O-] DFP00251 c1cc(cnc1)CNC(=O)/C=C/c2ccc(c(c2)Cl)Cl JP00369 c1cc2c(cc1C(=O)CCN3CCOCC3)OCCO2.Cl DSHS00083 Cc1ccc(c(c1)C)C(=O)CCN2CCOCC2.Cl DSHS00085 CC(C)(C)c1nnc(o1)c2cccc(c2)[N+](=O)[O-] DFP00263 CC(C)(C)NC(=O)Nc1cccc(c1)C(=O)OC DFP00269 CC1c2ccsc2CCN1C(=S)NC(=O)c3ccc(cc3)C(C)(C)C DFP00276 CCOC(=O)c1c(c(sc1Nc2ccccc2OC)C(=O)c3ccc(cc3)Br)N DP00029 CCOC(=O)c1cc2cc(ccc2[nH]1)[N+](=O)[O-] JFD01905 CCCCCCCCCCOc1ccccc1OCCCCCCCCCC JFD01906 CC(C)(C)c1cc(cc(n1)c2ccccn2)SC GK00864 CCc1cccc(c1NC(=O)COc2cc3c(cc2OC)C=CC(O3)(C)C)C JFD00345 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3cccc(c3)[N+](=O)[O-] DFP00242 c1ccc\2c(c1)CC/C2=N\NC3=NCCN3 DP02067 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2cc(cc(c2)C(F)(F)F)C(F)(F)F DP02069 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cnn(c2C(F)(F)F)c3ccccc3 GK02080 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=O)Nc2ccc(cc2)Cl DFP00253 COC(=O)c1cccc(c1)NC(=O)c2ccccc2 DFP00254 c1ccc(cc1)n2c(c(cn2)C(=O)NNS(=O)(=O)c3ccc(cc3)C(F)(F)F)C(F)(F)F GK02083 CCOC(=O)c1ccc(c(c1)/N=C/c2cc(ccc2O)Br)N3CCOCC3 JP00577 CCOC(=O)c1ccc(c(c1)/N=C/c2c3ccccc3ccc2O)N4CCOCC4 JP00578 Cc1ccsc1/C=C/C(=O)Nc2ccccc2C(F)(F)F GK00971 Cc1ccsc1/C=C/C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N GK00976 Cc1ccc(cc1)S(=O)(=O)NC2CC3CCC2(C3(C)C)C JFD01382 c1cc(cc(c1)Cl)NC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK02434 CCC(=O)NC(=S)NNC(=O)c1cccc(c1)[N+](=O)[O-] DFP00336 Cc1c(c(cs1)NC(=O)c2ccc(cc2)Cl)C(=O)OC GK02317 Cc1c(c(cs1)NC(=O)c2ccccc2Cl)C(=O)OC GK02320 Cc1c(c(cs1)NS(=O)(=O)c2ccccc2)C(=O)OC GK02327 C1CCC(CC1)NC2(CCCCC2)C#N DSHS00023 CSc1nc(nc(n1)O)c2ccc(cc2)Cl JM00155 c1cc(c(c(c1)Cl)CSc2nc(nc(n2)O)c3ccc(cc3)Cl)F JM00158 c1ccc(cc1)c2nc(nc(n2)SCc3ccc(cc3)Cl)O JM00159 c1ccnc(c1)Sc2ncc(c(n2)C(F)(F)F)C(=O)OCC3CC3 GK02088 c1cc(ccc1n2c(c(cn2)C(=O)NN)C(F)(F)F)Cl GK02092 COC(=O)c1c(csc1C(=O)OC)NS(=O)(=O)c2ccccc2 GK02312 Cc1csc(c1N2C(=O)C=CC2=O)C(=O)OC GK02295 Cc1c(c(cs1)NC(=O)c2ccccc2)C(=O)OC GK02315 Cc1nc(cs1)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl JP00723 COc1cc2c(cc1OC)C(=NCC2)c3ccccc3N JP00735 Cc1ccc(cc1)NC2=C(C(=O)c3ccccc3C2=O)Cl JFD01935 Cc1ccccc1OC2=C(C(=O)c3ccccc3C2=O)Cl JFD01936 CC(=O)OC[C@H]1[C@@H]([C@H]([C@@H]([C@H](O1)Oc2ccc(cc2)c3coc4cc(cc(c4c3=O)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD01219 Cn1c2ccccc2n3c1c(c(=S)c4c3cccc4)C#N JFD01872 c1cc(oc1C(=O)NNC(=S)N)[N+](=O)[O-] JFD01228 c1cc(cc(c1)Nc2cc(ncn2)O)C(F)(F)F JM00204 CC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccccn2 JP00671 c1cscc1/C=C/NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00860 COC(=O)c1cccc(c1)NC(=S)NC(=O)c2ccc(cc2)Cl DFP00277 c1ccc(c(c1)NC(=O)C(Cl)Cl)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F JP00512 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])Cl JP00516 c1ccc(cc1)Oc2ccc(cc2)OC(=O)c3c(cccc3F)F JFD01376 CC1(C2CCC1(C(C2)NS(=O)(=O)c3ccc(cc3)Cl)C)C JFD01381 CC(=O)c1c(cc(s1)C(C)(C)C)NC(=O)c2ccccc2C(=O)O GK02215 Cc1csc2c1c(ncn2)NNC(=O)c3ccc(cc3)Cl GK02225 c1ccc(c(c1)CSc2ccccc2NC3c4ccccc4C(=O)O3)Cl JP00451 CCCC(CC(=O)O)CC(=O)O JFD01264 c1cc(sc1C(=O)O)C(=O)O JFD01268 CC(=O)O[C@@H]1CO[C@H]([C@@H]([C@H]1OC(=O)C)OC(=O)C)OC(=O)C JFD00286 Cc1csc(c1NC(=O)c2cccc(c2)C#N)C(=O)OC GK02380 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)Cl)Oc3ccc(cc3)F GK02387 COc1ccc(cc1)c2nc3cc4c(cc3o2)Oc5ccccc5N4 JFD01932 CC1(C(=C)S/C(=N\c2cccc(c2)OC)/N1)C DSHS00444 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3/C(=N/c4ccccc4OC)/SC(=C)C35CCCCC5 DSHS00445 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3/C(=N/c4ccccc4Cl)/SC(=C)C3(C)C DSHS00452 COC(=O)c1c(csc1C(=O)OC)NS(=O)(=O)c2cccc(c2)C(F)(F)F GK02308 c1cc(cc(c1)Cl)NC(=O)N/C=C/c2ccsc2 GK00866 c1ccc(cc1)Sc2cc(c(cc2[N+](=O)[O-])Cl)Sc3ccccc3 JP00492 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCOC(C3C)c4ccccc4 DSHS00160 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N/N=C/2\CCCCC2CCC#N DSHS00163 c1cc(ccc1/C(=C\C=C(C#N)C#N)/Sc2ccc(cc2)Br)Cl JFD00256 COC(=O)c1c(ccs1)NC(=O)C2CC2 GK02395 CC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccc(cc2)Cl JP00670 COc1ccccc1/N=C/2\NC3(CCCCC3)C(=C)S2 DSHS00429 C=C1C2(CCCCC2)N/C(=N\c3ccccc3Cl)/S1 DSHS00431 Cc1ccc(c(c1)C)/N=C\2/NC3(CCCCC3)C(=C)S2 DSHS00432 Cc1c(c2c(s1)c(cc(=O)[nH]2)C(F)(F)F)C(=O)OC GK02383 COC(=O)c1c(ccs1)NC(=O)c2ccc(cc2)C#N GK02384 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)F GK02386 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3/C(=N/c4cccc(c4)OC)/SC(=C)C3(C)C DSHS00456 CC1(CC(=CC(=O)C1)Sc2nc3cc(ccc3s2)Cl)C JFD00263 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(=O)NN DSHS00173 CCOC([C@H]([C@@H]([C@@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)SCC JFD01222 c1ccc(cc1)c2c3ccccc3[nH]c2c4ccccc4 JFD01251 Cn1cc(c(n1)C(F)(F)F)C(=O)O/N=C/c2c(cccc2Cl)Cl GK00819 CS(=O)(=O)c1ccccc1C(=O)O JFD01922 COC(=O)c1cccc(c1)NC(=S)NC(=O)c2ccccc2 DFP00279 COC(=O)c1cccc(c1)NC(=O)NC(=O)c2ccccc2 DFP00283 c1cc(ccc1N2CCCC2=O)S(=O)(=O)CO JFD01320 CCOC(=O)C(c1c2cccc3c2n(c(=O)c1[N+](=O)[O-])CCC3)C(=O)OCC JFD01327 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc(cs2)C GK02259 c1ccc(cc1)CN2CCN=C2NNC(=O)c3cccc(c3)C(F)(F)F DP01967 c1ccc(cc1)S(=O)(=O)c2ccc(cc2Cl)[N+](=O)[O-] DP01984 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2ccccc2[N+](=O)[O-])N3CCCCC3 JP00622 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)N3CCCCC3 JP00624 c1cc(sc1)C(=O)c2ccc(cc2)F JFD01296 COC(=O)c1cccc(c1)NC(=O)NC(=O)c2cccs2 DFP00305 c1cc(ccc1NC(=O)/C=C/c2ccc3c(c2)OCO3)Br JP00336 c1cc2c(cc1/C=C/C(=O)Nc3ccc(cc3Cl)Cl)OCO2 JP00341 c1ccc2c(c1)-c3ccccc3C2=Cc4ccc(cc4)Cl JP00352 c1ccc(c(c1)COC(=O)c2cc(cc3c2-c4ccc(cc4C3=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-])Br JFD01190 CCCCN(C)C(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] JFD01192 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)Nc4ccc(cc4Cl)Cl JFD01193 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])SCC(=O)Nc2c(cc(cc2C)C)C JP00547 Cc1ccc(cc1)S(=O)(=O)Nc2c(cc(cc2C)NC(=O)C)C JFD01197 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)NCCCO JFD01202 CCn1cc(c(=O)c2c1ccc(c2)Cl)C(=O)O DFP00296 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCC(CC3)CCCC4CCN(CC4)C(=O)c5c(onc5c6ccccc6Cl)C DSHS00151 Cc1cc(cc2c1C(CC(O2)(C)C)O)OCc3ccc(cc3)Cl JFD00315 c1cscc1/C=C/NC(=O)Sc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00890 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)C(Cl)Cl)C(F)(F)F GK02101 c1cc(ccc1n2c(c(cn2)C(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F)Cl GK02107 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccccc3C(=O)OC DSHS00254 CC1CC(=O)Nc2ccccc2O1 JFD00283 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)[N+](=O)[O-] GK02108 COc1ccc(c(c1)S(=O)(=O)Nc2ccc(cc2)OC(F)(F)F)OC GK02112 COc1ccc(c(c1)S(=O)(=O)Nc2ccsc2C(=O)OC)OC GK02113 CCOC(=O)NCc1ccccc1 DSHS00133 CCOC(=O)c1ccc(c(c1)NC(=S)Nc2cccc(c2)SC)N3CCOCC3 JP00586 CCOC(=O)c1ccc(c(c1)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C)N4CCOCC4 JP00582 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)F)N3CCOCC3 JP00593 Cn1c(=O)[nH]c(n1)c2cccnc2 JM00244 Cc1csc(c1NC(=O)c2ccc(cc2)C(F)(F)F)C(=O)OC GK02291 Cc1csc(c1NS(=O)(=O)c2ccc(cc2)NC(=O)C)C(=O)OC GK02292 Cc1cc(cc(c1)c2cc(cc(c2)C)C)C JFD01279 c1cc(ccc1CSc2nccc(n2)O)Cl JM00409 c1cc(cc(c1)NC(=O)O/N=C(/C2CSCCS2)\N)C(F)(F)F GK02372 c1cc(ccc1[N+](=O)[O-])Oc2ccc(cc2)F GK02378 Cc1csc2c1c(ncn2)N/N=C/c3ccccc3Cl GK02221 Cc1csc2c1c(ncn2)N/N=C/c3ccc(cc3)OC GK02222 CC(C)(C)OC(=O)N1CCC(CC1)(c2ccccc2)C(=O)O JFD01929 c1cc(c(cc1F)Br)/N=C/c2cc(ccc2O)Cl DP02019 CC(C)c1ccc(c(c1)Br)/N=C/c2ccccc2O DP02020 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc(c2)C(=O)OC DFP00257 CC(=O)Nc1cccc(c1)C(=O)OC DFP00258 c1cc2c(cc1Cl)cc(o2)c3csc(n3)N.Br DP02022 C=CCNc1nc(cs1)c2cc3cc(ccc3o2)Cl.Br DP02023 COc1cc(c(cc1SCC(=O)NN)OC)[N+](=O)[O-] JP00515 c1cc(ccc1CSc2nccc(n2)O)[N+](=O)[O-] JM00410 COC(=O)c1cccc(c1)NC(=O)NC(=O)c2ccc(cc2)C(F)(F)F DFP00286 COC(=O)c1cccc(c1)NC(=S)NC(=O)c2ccco2 DFP00287 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3cnco3 DFP00291 Cc1csc2c1c(ncn2)Sc3ccccc3NC(=O)c4ccc(cc4)[N+](=O)[O-] GK02208 CC12[C@H](C=C[C@@]3([C@@H]1[C@@H]([C@]45[C@H]3CC[C@](C4)(C(=C)C5)O)C(=O)O)OC2=O)O JFD01925 Cc1csc2c1c(ncn2)N/N=C/c3ccc(cc3)C(F)(F)F GK02220 c1ccc2c(c1)cccc2/C=C/3\CCc4ccccc4\C3=N\Nc5ccc(cc5[N+](=O)[O-])[N+](=O)[O-] DSHS00186 CCCCCCCCNC1=C(C(=O)c2ccccc2C1=O)Cl JFD00241 CCCC(=O)/C(=C\Nc1ccccc1C(=O)OC)/C(=O)OCC GK00736 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)COc2ccc(cc2Cl)Cl JP00182 c1ccc2c(c1)C3N(C2=O)CCCN3S(=O)(=O)c4cccc(c4)C(F)(F)F JP00274 Cc1c2c(n(c(=O)c1c3ccccc3)C)n(c(=O)n(c2=O)c4ccccc4)c5ccccc5 JFD01334 CCc1c(c2ccccc2n(c1=O)C)OS(=O)(=O)c3ccc(cc3)C JFD01336 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3cccc(c3)C(F)(F)F JP00275 c1ccc2c(c1)cccc2/C=C/3\CCc4ccccc4C3=O DSHS00182 CC(=O)NC(=S)NNC(=O)c1cccc(c1)[N+](=O)[O-] DFP00335 CC(c1ccc2c(c1)OCCO2)NC(=O)c3ccccc3C(=O)NC(C)c4ccc5c(c4)OCCO5 DSHS00248 c1cc(ccc1S(=O)(=O)NNC(=O)c2c(ccs2)I)Cl GK00931 Cc1c(c(no1)c2ccccc2Cl)C(=O)N(C3CCCCC3)C4CCCCC4 DSHS00284 C1CCc2c(c(c(s2)N)C(=O)N)C1 DSHS00288 c1cc(c(cc1Cl)Cl)CS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00757 CC1CN(CC(O1)C)S(=O)(=O)c2cccc(c2)C(F)(F)F JP00277 Cc1c(c(sc1c2ccccc2)N)C#N DSHS00315 Cc1ccc(c(c1)C)C(C)NC(=O)/C=C/c2ccccc2 DSHS00246 Cc1ccc(c(c1)C)C(C)NC(=O)c2ccccc2C(=O)NC(C)c3ccc(cc3C)C DSHS00247 CC1CCC(C(C1)NC(=O)c2c(cccc2Cl)Cl)C(C)C JFD01371 COc1ccc(cc1)C(=O)/C=C\2/N(C(=O)C(=O)S2)c3ccccc3 JFD00369 c1ccc(cc1)/C(=C/2\C(=O)C(=O)N(C2=O)c3ccc(cc3)Cl)/Nc4ccccc4 JFD00364 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(c2)F JFD01389 CC(=O)c1c(ccs1)NC(=O)c2ccccc2C(=O)O GK02425 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c(ccs2)I GK00934 CCOC1=C(C(=O)c2ccccc2C1=O)Cl JFD01941 Cc1ccc(cc1)S(=O)(=O)NNC(=O)CNC(=O)c2cc(cs2)C GK02246 Cc1c(c(no1)c2ccccc2Cl)C(=O)N(CCC#N)C3CCCCC3 DSHS00241 Cc1c(c(no1)c2ccccc2Cl)C(=O)N(CCC#N)C(C)C DSHS00242 Cc1ccc(c(c1)C)C(C)NC(=O)c2c(onc2c3ccccc3Cl)C DSHS00243 Cc1ccc(c(c1)C)C(C)NC(=O)c2cc(c(c(c2)OC)OC)OC DSHS00244 COC(=O)c1cccc(c1)NS(=O)(=O)c2ccc(c(c2)Cl)Cl DFP00315 c1ccc(cc1)c2c3cc(ccc3no2)Cl JFD01363 c1cc(c(cc1F)F)NC(=O)c2cnc(nc2C(F)(F)F)N GK02462 c1cc(ccc1SC(=O)N/C=C/c2ccsc2)Cl GK00886 COC(=O)c1c(ccs1)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00898 CSc1cccc(c1)NC2c3ccccc3C(=O)O2 JP00781 c1ccc(c(c1)N)Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] JP00413 c1ccc(c(c1)N)SCc2c(cccc2Cl)Cl JP00414 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=S)Nc2ccc(c(c2)Cl)Cl DFP00322 Cc1cccc(c1)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] DFP00323 COC(=O)c1cccc(c1)NC(=S)NCc2ccccc2 DFP00326 CN(CCC#N)C(=S)Nc1ccc(cc1)F JP00956 CCOC(=O)C(C#N)c1c2cccc3c2n(c(=O)c1[N+](=O)[O-])CCC3 JFD01326 C[C@]12CC[C@H](CC1CCC3C2CC[C@](C3/C=C/4\C(=O)c5ccccc5N4)(C)C(=O)O)O DSHS00507 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N(c2cccc(c2)SC)C3c4ccccc4C(=O)O3 JP00789 Cc1ccc(cc1)Nc2cc(=O)n(c3c2c(=O)n(c(=O)n3C)C)c4ccccc4 JFD01331 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cccc(c4)[N+](=O)[O-] DSHS00522 COC(=O)c1cccc(c1)NC(=S)Nc2ccc(c(c2)Cl)Cl DFP00318 COC(=O)c1cccc(c1)NS(=O)(=O)C DFP00321 c1ccc(c(c1)CSc2ccccc2N)Cl JP00446 c1ccnc(c1)SCc2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-] JFD01977 c1cc(ccc1C(=O)NCC(=O)O)Br JFD01985 Cc1cc(sc1)C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK02257 Cc1cc(sc1)C(=O)NNS(=O)(=O)c2ccc(cc2)C(F)(F)F GK02258 Cc1cc(sc1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F GK02262 c1(c([nH]c(=O)[nH]c1=O)N)Br JFD01950 CCN(CC)CCC1S(=O)(=O)C(C(C(S1(=O)=O)C(=O)OCC)c2ccccc2)C(=O)OCC JFD01350 COc1ccsc1C(=O)OC GK02497 COc1ccccc1N2CCN(CC2)CN3c4ccc(cc4C(=O)C3=O)Br DSHS00619 c1cc(ccc1S(=O)(=O)N(CCC#N)C2CCCCC2)Br DSHS00623 CCN(CC)CCC1S(=O)(=O)CC(CS1(=O)=O)c2ccccc2 JFD01351 CCOC(=O)C1=C(NC2=C(C1c3ccc(cc3)[N+](=O)[O-])C(=O)c4c2cccc4)C JFD00435 CC1=C(C(C2=C(N1)c3ccccc3C2=O)c4ccccc4)C(=O)C JFD00440 c1ccc(c(c1)CS(=O)(=O)c2nc3ccccc3s2)[N+](=O)[O-] JFD01986 Cc1c([nH]c2c1cccc2[N+](=O)[O-])C JFD01907 c1ccc(cc1)c2ccc(o2)c3ccccc3 JFD01909 CCOC(=O)c1cc2cccc(c2[nH]1)[N+](=O)[O-] JFD01911 CCc1cccc(c1NC(=O)COc2cc3c(cc2OC)C=CC(O3)(C)C)CC JFD00346 c1ccc2c(c1)C(OC2=O)Nc3ccccc3SCc4ccc(cc4)C#N JP00455 CNC(=S)Nc1cccc(c1)C(=O)OC DFP00327 CCOC(=O)C(=CNc1ccc(cc1)C(F)(F)F)C(=O)OCC DFP00334 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC(=O)C)OC(=O)C)OC(=O)C)O[C@H]2[C@@H]([C@H]([C@@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00294 CC(=O)OC[C@@H]([C@@H]([C@H]([C@@H](C(=O)N)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00297 CC1CC(=O)Nc2cc(ccc2O1)Cl JFD00298 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-])/N GK02444 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccsc2C(=O)OC GK00899 c1ccnc(c1)CCc2cccc(c2)NS(=O)(=O)c3ccc(cc3)Cl DSHS00541 Cc1ccc(cc1)S(=O)(=O)NNC(=O)CSc2cc(c(cc2OC)[N+](=O)[O-])OC JP00535 Cc1cc(sc1)c2nc(no2)c3ccc(cc3)C(C)(C)C GK02281 CC1c2ccsc2CCN1S(=O)(=O)c3cccs3 DFP00365 CCC12CCCN3C1c4c(c5ccccc5n4C(=O)C2)CC3 JFD01913 CCC(=O)Nc1cccc(c1)C(=O)OC DFP00261 c1cc(cc(c1)[N+](=O)[O-])c2nnc(o2)C3CC3 DFP00262 CCCCc1c(nc(nc1O)N)COC GK02331 Cc1ccc(cc1)SC(=O)N/C=C/c2ccsc2 GK00889 Cc1c(c(c(c(c1C)C)C(=O)/C(=C/c2cccs2)/C)C)C JP00818 c1cc(ccc1n2c(c(cn2)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] GK02438 c1cc(ccc1/C(=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-])/N)Cl GK02445 c1cc(ccc1c2cc(c(s2)C(=O)N)NC(=O)C(Cl)Cl)F GK01107 Cc1cc(sc1)c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK02282 Cc1c(c(cs1)NS(=O)(=O)c2cccc(c2)Cl)C(=O)OC GK02330 CCOC(=O)C(=CNc1csc(c1C(=O)OC)C)C(=O)OCC GK02332 Cc1c(c(cs1)NS(=O)(=O)c2ccccc2Cl)C(=O)OC GK02334 c1ccc(c(c1)N/N=C(/N=N/c2ccccc2O)\[N+](=O)[O-])O JFD01297 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cc(c(c(c4)OC)OC)OC DSHS00516 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccccc4Cl DSHS00520 Cc1ccc(cc1)C(=O)Nc2csc(c2C(=O)OC)C GK02319 Cc1c(c(cs1)NC(=O)C)C(=O)OC GK02321 Cc1c(c(cs1)NC(=O)C(C)(C)C)C(=O)OC GK02322 c1cc2c(cc1Br)C(=O)C(=O)N2CN(CCC#N)C3CCCCC3 DSHS00622 c1ccnc(c1)SC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK02449 c1cc(ccc1c2nc(on2)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-])C(F)(F)F GK02451 c1ccc2c(c1)CCN(C2)c3ccc(cc3[N+](=O)[O-])S(=O)(=O)N4CCc5ccccc5C4 JP00501 CC(C)c1ccc(cc1)S(=O)(=O)NNC(=O)CSc2ccccc2[N+](=O)[O-] JP00502 CCOC(=O)c1ccc(cc1)N/N=C/c2ccccc2O JP00739 COC(=O)c1c(csc1C(=O)OC)N.Cl GK02289 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4cc(c(cc4Cl)Cl)Cl DSHS00580 COC(=O)c1c(cc(s1)c2ccc(cc2)F)NC(=O)C(F)(F)F GK01139 COC(=O)c1c(cc(s1)c2ccc(cc2)F)NC(=O)C(Cl)Cl GK01142 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)C(C)(C)C DSHS00524 c1ccc(cc1)C2=C(C(=O)C(=O)N2)C(=O)Nc3ccccc3 JFD00353 CS(=O)(=O)N1CCCN2C1c3ccccc3C2=O DSHS00421 CCOC(=O)c1ccc(cc1)/N=C\2/NC3(CCCCC3)C(=C)S2 DSHS00427 C=C1C2(CCCCC2)N/C(=N\c3cccc(c3)C(F)(F)F)/S1 DSHS00428 C1CSSC1CCCCC(=O)N JFD01918 c1ccc(cc1)c2cc(c(s2)C(=O)N)NS(=O)(=O)c3ccc(cc3)F GK01017 COC(=O)c1c(ccs1)NC(=S)OC GK02355 CCOC(=O)c1ccc(c(c1)NC(=O)c2c(onc2c3ccccc3)C)N4CCOCC4 JP00581 Cn1cc(c(n1)C(F)(F)F)C(=O)O/N=C/c2ccc(cc2)Cl GK00843 c1ccc(cc1)n2c(=S)n(nn2)CN3CCOCC3 JFD01889 CCc1cccc(c1NC(=O)COc2ccc3c(c2)OC(C=C3)(C)C)C JFD00330 CCc1cccc(c1NC(=O)COc2cc(c3c(c2)OC(C=C3)(C)C)C)CC JFD00334 CN(C)c1ccc(cc1)C(c2ccc(cc2)N(C)C)c3ccc(cc3)[N+](=O)[O-] JFD01996 COC(=O)C(c1ccccc1)C(=O)O JFD01998 CCc1cccc(c1NC(=O)COc2ccc3c(c2C)OC(C=C3)(C)C)CC JFD00338 c1cn[nH]c1NC(=O)CC#N GK00927 c1ccc(cc1)c2ccc(cc2)/C=C\3/C(=O)C4CCN3CC4 DSHS00358 CCOC(=O)c1c[nH]c2ccc(cc2c1=O)C(F)(F)F DFP00346 c1cc(sc1)CN2CC(CC2=O)C(=O)O DFP00358 c1cc(oc1)CN2CC(CC2=O)C(=O)O DFP00359 c1ccc(cc1)c2cc(c(s2)C(=O)N)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01018 COc1ccc(cc1)C(CCC#N)(CCC#N)C#N DSHS00340 CC1=CCCC(C1/C=C(\C)/C(=O)/C=C/c2cccs2)(C)C JP00816 c1ccc(cc1)/C=N/NC(=O)CC#N DP00066 c1c(cc(cc1C(F)(F)F)NC(=S)N(CCC#N)CC2CCCO2)C(F)(F)F JP00914 CC(C)c1ccc(cc1)/C=N/NC(=O)CC#N DP00085 Cc1ccccc1C(=O)NNC(=O)c2ccccc2C3=NCCCN3 DSHS00409 CN(C)c1ccc(cc1)/C=C/2\C(=O)C3CCN2CC3 DSHS00398 c1ccc(c(c1)C2=NCCCN2)C(=O)NNC(=O)c3ccc(cc3)Cl DSHS00406 COC(=O)c1cccc(c1)NC(=O)NC(=O)c2ccccc2Cl DFP00284 c1cc2c(cc1/C=C/3\C(=O)C4CCN3CC4)OCO2 DSHS00408 c1cc(c(cc1C2C3C(=NN2)C4CCN3CC4)Cl)Cl DSHS00412 CN(C)/C=C(\c1nnnn1c2ccccc2)/C(=O)c3ccc(cc3)C(F)(F)F JFD00271 Cc1ccc(cc1)/C(=C\2/C(=O)C(=O)N(C2=S)c3ccccc3)/O JFD00374 Cc1ccc(cc1)S(=O)(=O)N(CCC#N)CC2CCCO2 DSHS00632 c1ccc2c(c1)nc(s2)SCCCCSc3nc4ccccc4s3 JFD01984 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)OC([C@@H](COC(=O)C)OC(=O)C)[C@@H]([C@H](C(=O)N)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00296 c1ccc2cc(ccc2c1)C(=O)CCN3CCOCC3.Cl DSHS00080 c1ccc2c(c1)CC(=C2)N3CCOCC3 JFD00276 CCSC([C@@H]([C@H]([C@@H](CO)O)O)O)SCC JFD00281 CCSC([C@@H]([C@H]([C@H](CO)O)O)O)SCC JFD00282 c1ccc2cc(ccc2c1)C(=O)CCN3CCCC3.Cl DSHS00100 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NC(=S)NN)OC(=O)C)OC(=O)C)OC(=O)C JFD00301 CCOC(=O)/C(=C\1/N(C(=CS1)c2ccccc2)c3c(cccc3C)C)/C#N DP00107 CC1=C(C(NC(=O)N1)c2ccccc2)C(=O)OC JFD00469 CC1=C(C(C2=C(N1)c3ccccc3C2=O)c4ccccc4)C#N JFD00441 c1cc(ccc1C(F)(F)F)NC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK02435 COc1ccc(cc1[N+](=O)[O-])C(=O)CCN2CCOCC2.Cl DSHS00087 c1ccc(cc1)COc2ccc(cc2)C(=O)CCN3CCOCC3.Cl DSHS00098 c1ccc(cc1)C(=O)OC[C@@H]2[C@@H]([C@@H]([C@H]([C@H](O2)OC(=O)c3ccccc3)OC(=O)c4ccccc4)OC(=O)c5ccccc5)OC(=O)c6ccccc6 JFD01240 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(/C2CSCCS2)\N GK02368 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)C)N3CCCCC3 JP00621 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2cccc(c2)C(F)(F)F)N3CCCCC3 JP00623 COc1cc(c(cc1Cl)OC)NC(=S)Nc2ccc(c(c2)Cl)Cl JP00626 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2ccc(cc2)Cc3ccc(cc3)NC(=O)c4cccc(c4)[N+](=O)[O-] JP00639 CCOC(=O)c1ccc(c(c1)NC(=O)c2c(c3ccccc3s2)Cl)N4CCCCC4 JP00646 CCOC(=O)c1ccc(c(c1)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C)N4CCCCC4 JP00647 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)F JFD01388 COC(=O)CSC(=O)N/C=C/c1ccsc1 GK00891 Cc1cc(c(cc1Cl)C)SC(=O)N/C=C/c2ccco2 GK00893 COC(=O)c1c(ccs1)NC(=O)c2ccccc2C(=O)O GK02188 c1cc(ccc1NC(=O)/C=C/c2ccsc2)F GK00882 CC1CCCCN1S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DP00321 c1ccc(cc1)c2c(c3nnnn3nc2c4ccccc4)c5nn(c(=S)o5)CN6CCOCC6 JFD00401 c1ccc(cc1)c2c(c3n[nH]c(=O)n3nc2c4ccccc4)c5ccccc5 JFD00404 Cc1csc2c1c(ncn2)Sc3ccccc3NS(=O)(=O)c4ccc(cc4)F GK02206 COc1ccc(cc1Br)/C=C/2\C(=O)C3CCN2CC3 DSHS00401 CCOc1cc(ccc1O)/C=N/NC(=O)CC#N DP00070 Cc1ccsc1/C=C/C(=O)O/N=C/c2c(cccc2Cl)F GK00985 CC(C)OC(C(F)(F)F)(C(F)(F)F)NC(=O)c1ccccc1 JFD01405 CNC(=O)c1ccc(cc1)/C=C\2/C(=O)C3CCN2CC3 DSHS00411 CCOC(=O)c1c(c(sc1Nc2c(cccc2C)C)C(=O)c3ccc(cc3)Br)N DP00108 CC(C)(C)c1cc(c(s1)C(=O)N)N GK00992 c1cscc1/C=C/C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00883 Cc1csc2c1c(ncn2)Sc3ccccc3NC(=O)c4ccc(cc4)C(F)(F)F GK02202 CS(=O)(=O)c1ccc(cc1)C#N JFD01921 Cc1csc2c1c(ncn2)Sc3ccccc3NC(=O)c4cc(cc(c4)Cl)Cl GK02207 c1cc(cc(c1)Cl)NC(=O)/C=C/c2ccc(cc2)Cl JP00319 Cn1c2c(c(c(c1=O)[N+](=O)[O-])N)c(=O)n(c(=O)n2C)C JFD01324 c1cc2cccc3c2c(c1)C(=C(C3=O)[N+](=O)[O-])O JFD01325 COc1cccc(c1OC)/C=N/NC(=O)CC#N DP00128 COC(=O)c1cccc(c1)NC(=S)NC(=O)c2cccs2 DFP00288 CCc1cccc(c1NC(=O)COc2ccc3c(c2)OC(C=C3)(C)C)CC JFD00331 c1cc(cc(c1)NC2(CCCCCC2)C#N)C(F)(F)F DSHS00208 COC(=O)c1cccc(c1)NC(=S)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00289 c1ccc(cc1)C2CS(=O)(=O)C(S(=O)(=O)C2)CCN3CCOCC3 JFD01348 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl GK02432 CCOC(=O)C/C(=N/Nc1ccsc1C(=O)OC)/C(F)(F)F GK02512 COC(=O)c1c(c(sc1NCC=C)C(=O)OC)N DP00123 Cc1ccc(c(c1)C)C(C)NC2(C3CC4CC(C3)CC2C4)C#N DSHS00235 Cc1c(c(no1)c2ccccc2Cl)C(=O)N(CCC#N)Cc3ccccc3 DSHS00240 c1csc(c1I)C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00932 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3nc4ccc(cc4s3)C DSHS00525 CC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccccc1Cl JFD01416 CCOC(=O)/C(=N/Nc1ccccc1)/C JFD01359 c1ccc(cc1)CN2CCC(=NO)CC2 JFD01360 CC1(CN=C(S1)N(c2ccc(cc2)Cl)C(=O)NC)C JFD01421 c1ccc(c(c1)CC(=O)NCCc2c[nH]c3c2cccc3)F JFD01361 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)N4CCN(CC4)c5ncc(cn5)Br JFD01365 COC(=O)c1c(ccs1)N/N=C/c2ccc(cc2)C(F)(F)F GK02415 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK02431 CCCc1c(cnn1c2ccc(cc2)[N+](=O)[O-])C(=O)OCC GK02420 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)NC2CCCCC2 JFD01401 Cc1ccsc1/C=C/C(=O)O/N=C(/c2ccc(cc2)Cl)\N GK00974 CC1(CC(c2ccc(cc2O1)OCc3ccc(cc3)Cl)O)C JFD00314 COc1ccc(cc1)c2cc(c(s2)C(=O)N)NS(=O)(=O)c3ccc(cc3)Cl GK01173 COc1ccc(cc1)c2cc(c(s2)C(=O)N)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01174 CC1CCN(CC1)S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DP00325 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3cc(ccc3Cl)Cl DP00330 c1ccc(c(c1)CO)C(=O)N/N=C/c2cccs2 JPV00053 COc1c(csc1c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Br GK02600 CCOC(=O)c1ccc(cc1)N/N=C/c2ccc3c(c2)OCO3 JP00740 Cc1cscc1NC(=O)/C=C/C(=O)O GK02478 CCOC(=O)CC(=O)Nc1ccn[nH]1 GK00920 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2SCCC#N JP00793 Cc1cccc(c1/N=C\2/NC(C(=C)S2)(C)C)C DSHS00483 c1cc(ccc1c2cc(c(s2)C#N)N)F GK02483 CCOc1ccsc1C(=O)OC GK02484 c1ccc(cc1)CN(CCC#N)C(=S)Nc2ccc(cc2)F JP00952 CC(C)c1ccc(cc1)/C=N/c2ccc(cc2)C(=O)O DSHS00500 c1ccc2c(c1)Nc3ccccc3S2 JFD01943 c1cc(c(cc1NC(=O)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)Cl)Cl JPV00015 COC(=O)c1c(ccs1)NNC(=O)c2ccc(cc2)C(F)(F)F GK02413 c1ccnc(c1)/C=N/NC(=O)C(=O)Nc2ccc(cc2Cl)Cl JPV00021 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)N GK02419 CCOC(=O)c1c2ccc(cn2c3c1C(=O)c4ccccc4C3=O)C JP00797 c1cc(cc(c1)NC(=O)COc2cc(c(cc2Cl)Cl)Cl)C(F)(F)F DSHS00486 Cc1ccc(cc1)C(=O)CN2C(=O)CCC2=O DP00268 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCCC2 DP00317 c1ccc2c(c1)c(=O)c(c-3sc4ccccc4nc23)Oc5ccc(cc5)Cl JFD01949 CCOC(=O)C1=C(NC2=C(C1c3ccccc3)C(=O)c4c2cccc4)C JFD00429 CN(C)c1ccc(cc1)C2C(S(=O)(=O)CS(=O)(=O)C2C(=O)OC)C(=O)OC JFD01346 CC1(CN=C(S1)N(c2ccccc2F)C(=O)Nc3ccccc3)C JFD01432 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCC=CC2 DSHS00685 COc1cc(c(cc1Cl)OC)NS(=O)(=O)c2ccc(cc2)Cl DSHS00687 c1cc(ccc1NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)F DSHS00690 CCOc1ccc(cc1)/C=C(\C#N)/C(=O)N2CCCC2 DP00498 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)N)C(C)(C)C GK01000 c1cc(ccc1CC#N)NC2(CCCC2)C#N DSHS00692 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(c(cc3OC)Cl)OC DSHS00694 CCOC(=O)CNC(=O)c1ccc(cc1)Br JFD02015 C1[C@@H]2C=C[C@H]1C3C2C(=O)C4[C@H]5C[C@@H](C4C3=O)C=C5 JFD02026 CC(CCC(=O)NCC(=O)[O-])C1CCC2C1(CCC3C2C(CC4C3(CCC(C4)O)C)O)C.[Na+] DSHS00533 c1cc(ccc1n2c(c(cn2)C(=O)NN)C(F)(F)F)[N+](=O)[O-] GK02440 Cc1ccc(cc1F)NC(=O)Nc2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK02441 COc1cccc(c1CCOC(=O)c2c(cccc2F)F)OC JFD01377 c1cc(ccc1/C(=N/OC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-])/N)C(F)(F)F GK02443 CCOC(=O)C(C(F)(F)F)(Nc1nc2ccccc2s1)NC(=O)OCC JFD01440 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)S(=O)(=O)N)NC(=O)OCC JFD01441 c1ccc(cc1)C(=O)NCC(=O)NN JFD02006 CC(=O)c1c(ccs1)NC(=O)/C=C/C(=O)O GK02525 CC1=CC(=O)N(C1=O)c2ccsc2C(=O)OC GK01180 CC(C)(C)c1ccc(cc1)c2nc(on2)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-] GK02452 c1ccc(cc1)SCC(=O)Nc2nc(cs2)CC(=O)O JFD01990 COc1cc2c(cc1OC)C(=NCC2)c3ccccc3NC(=O)c4ccc(cc4)F JP00751 CCOC(=O)[C@@H]1CSC2N1CCN3C2SC[C@H]3C(=O)OCC JFD00427 c1ccc(cc1)CC(=O)NNC(=S)Nc2ccccc2 JFD00428 Cc1cc(=O)[nH]c(n1)N/N=C/c2ccncc2 JFD00430 CCOC(=O)Cc1csc(n1)NC(=O)CSc2ccccn2 JFD02017 c1ccc2c(c1)nc(s2)SCC(=O)Nc3nc(cs3)CC(=O)O JFD02019 c1cc(c(cc1/C=C(\C#N)/C(=O)N2CCOCC2)Cl)Cl DP00517 c1cc(ccc1/C=C(\C#N)/C(=O)N)Cl DP00522 c1ccc(c(c1)/C=C(\C#N)/C(=O)N)Cl DP00523 C=C1C2(CCCCC2)NC(=Nc3ccc(cc3)S(=O)(=O)N4CCCCC4)S1 DSHS00434 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)Cl)c4cccs4 JP00805 c1ccc(cc1)/C(=N\Nc2ccccc2O)/C(=O)O JFD01301 COc1ccc(cc1OC)C(=C)c2c3cc(c(cc3ccn2)OC)OC JFD01955 c1cc(ccc1C(=O)O)/N=C/c2ccc3c(c2)OCO3 DSHS00502 COC(=O)c1c(csc1C(=O)OC)NS(=O)(=O)c2ccc(cc2Cl)Cl GK02309 c1ccc(cc1)OCC(=O)NCC(=O)N JFD02072 CCOC(=O)CNC(=O)COc1ccccc1 JFD02007 CCOC(=O)CNC(=O)CSc1nc2ccccc2s1 JFD02011 c1ccc2c(c1)nc(s2)SCC(=O)NCC(=O)NN JFD02012 c1ccnc(c1)CCc2cccc(c2)NS(=O)(=O)c3cc(ccc3Cl)Cl DSHS00552 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)CCc3ccccn3 DSHS00536 COC(=O)c1cccc(c1)NS(=O)(=O)c2ccccc2 DFP00313 CCOc1ccsc1C(=O)NNC(=O)C2CC2 GK02533 c1ccc2c(c1)CCN(C2)CN3c4ccc(cc4C(=O)C3=O)Br DSHS00617 Cc1ccc(cc1)S(=O)(=O)NC2CC3CC[C@@]2(C3(C)C)C JFD01378 C[C@@]12CCC(C1(C)C)CC2NS(=O)(=O)c3ccc(cc3)Cl JFD01379 COc1c(csc1c2nc(no2)c3ccc(cc3)C(F)(F)F)Br GK02556 COc1cc(cc(c1OC)OC)/C=C(\C#N)/C(=O)N2CCOCC2 DP00503 COc1cc(cc(c1OC)OC)/C=C(\C#N)/C(=O)N DP00504 c1ccc(cc1)S(=O)(=O)N2CCCN3C2c4ccccc4C3=O DSHS00425 CN1C(C2C(=N1)C3CCN2CC3)c4ccc(c(c4)Cl)Cl DSHS00426 CS(=O)(=O)Nc1cc(sc1C(=O)N)c2ccccc2 GK01020 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)N)c3ccccc3 GK01019 CCOc1ccc(cc1)/C=N/NC(=O)CC#N DP00083 C1CCC(=NNC(=O)CC#N)CC1 DP00092 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)N3CCOCC3 JP00595 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2ccccc2[N+](=O)[O-])N3CCOCC3 JP00596 CCOC(=O)c1ccc(c(c1)NC(=O)c2ccc(c(c2)Cl)Cl)N3CCOCC3 JP00603 c1cc2c(cc1/C=C(\C#N)/C(=O)N3CCOCC3)OCO2 DP00494 c1cc2c(cc1/C=C(\C#N)/C(=O)N3CCCC3)OCO2 DP00496 CC1(CC1C(=O)Nc2ccc(cc2)Oc3ccc(cc3)C(C)(C)c4ccc(cc4)Oc5ccc(cc5)NC(=O)C6CC6(C)C)C JFD00453 Cc1cc(c(c(c1)C)NC(=O)CC#N)C DP00152 c1ccc(cc1)Oc2ccc(cc2S(=O)(=O)O)N3C(=O)CC(=N3)N JFD00458 Cc1ccc(c(c1)C)NC(=O)CC#N DP00164 COc1cc2c(c(c1)[N+](=O)[O-])NC(CC2c3ccccc3)c4ccccc4 DP00188 c1cc\2c(cc1)NC(=O)/C2=N\c3ccc(cc3)Cc4ccc(cc4)/N=C/5\C(=O)Nc6c5cccc6 JFD00459 c1cc(ccc1NC(=S)N(CCC#N)CC2CCCO2)F JP00951 c1ccnc(c1)CCc2cccc(c2)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl DSHS00540 CCOC(=O)c1ccc(c(c1)N)N2CCCCC2 JP00617 COc1ccc(cc1)C2=NN(C(C2)c3cccs3)c4ccccc4 JP00806 CCOC(=O)c1ccc(cc1)N/N=C/c2cc(cc(c2O)Cl)Cl JP00738 COc1ccc(cc1OC)/C=C(\C#N)/C(=O)N DP00534 c1ccc(cc1)S(=O)(=O)CCN2CCSCC2 KM00011 CC1CCCN(C1)CCS(=O)(=O)c2ccccc2 KM00014 Cc1c(c(=O)n(n1C)c2ccccc2)CN3CCSCC3.Cl KM00015 Cc1ccc(cc1)S(=O)(=O)N(Cc2ccccc2)C(C#N)c3ccc4c(c3)OCO4 DSHS00548 Cc1ccsc1/C=C/NC(=O)Nc2ccc(cc2F)F GK00961 CCOC(=O)/C(=C/1\N(C(=CS1)c2ccc(cc2)Br)Cc3ccccc3)/C#N DP00110 c1cc2c(cc1C3C4C(=NN3)C5CCN4CC5)OCO2 DSHS00416 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)N4C(=O)CSC4=O JFD02009 c1cc2c(cc1Br)C(=O)C(=O)N2CN3CCOCC3 DSHS00611 CCNc1c(c(c(s1)C(=O)OC)N)C#N DP00125 COc1c(csc1C(=O)O/N=C(/c2ccc(cc2)Cl)\N)Br GK02596 c1ccn2cc(nc2c1)C34CC5CC(C3)CC(C5)C4 JFD00395 CC(C)S(=O)(=O)CC(=O)Nc1ccc(cc1)C(=O)O JFD02075 CCOC(=O)c1ccc(cc1)NC(=O)CS(=O)(=O)C(C)C JFD02077 CC(C)SCC(=O)Nc1ccc(cc1)C(=O)O JFD02078 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCOCC2 JP00679 c1ccc(cc1)C2=NCCNC3=C2C(=O)N(C3=O)c4ccc(cc4)Br JFD00358 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=S)NC(=O)C2CC2 DFP00338 c1ccc(cc1)C(=O)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] DFP00342 c1ccc(c(c1)C(=O)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-])Cl DFP00343 CCOC(=O)C1=C(NC2(C1(C(=O)c3c2cccc3)O)O)C JFD00467 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc4c(c3)OCO4)C(=O)OC JFD00468 COc1c(csc1C(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N)Br GK02598 c1ccc(cc1)c2c3c([nH][nH]c3=O)nnc2c4ccccc4 JFD00398 c1ccc(cc1)OCC(=O)NCC(=O)NN JFD02070 Cc1ccc(cc1)S(=O)(=O)Nc2c(c3c(s2)CCCC3)C(=O)N JP00673 c1ccnc(c1)Sc2cc(c(cc2Sc3ccccn3)C#N)C#N JFD02051 CCOC(=O)CNC(=O)c1ccccc1C(=O)NCC(=O)OCC JFD02054 COc1cc(cc(c1OC)OC)c2[nH]c(=O)c3ccccc3n2 DSHS00654 COc1cccc(c1O)/C=N/c2ccccc2SCCC#N JP00782 c1ccc(cc1)SCc2ccc(cc2)[N+](=O)[O-] JFD02021 c1ccnc(c1)NC(=O)CCCCC(=O)Nc2ccccn2 JFD02028 COc1ccc(cc1)NC(=O)C2=C(NC(=O)C2=O)c3ccccc3 JFD00354 CCCc1cc(nc(n1)SC/C=C/c2ccccc2)O JFD02042 c1cc(ccc1CSc2ccc(cc2)Cl)[N+](=O)[O-] JFD02043 c1cc(ccc1CS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] JFD02048 c1ccc(c(c1)NC(=S)C(C#N)C(=O)N2CCCC2)Cl DP00456 c1ccc(c(c1)NC(=S)C(C#N)C(=O)N2CCOCC2)Cl DP00457 COc1ccccc1NC(=S)C(C#N)C(=O)N2CCOCC2 DP00461 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3ccc(cc3)Cl)/C(=O)N2C JFD01335 CCOC(=O)C1C(C(S(=O)(=O)CS1(=O)=O)C(=O)OCC)c2ccccc2 JFD01338 COC(=O)C1C(C(S(=O)(=O)CS1(=O)=O)C(=O)OC)c2ccc(cc2)Cl JFD01339 COc1ccc(c(c1OC)OC)/C=C/2\C(=O)C3CCN2CC3 DSHS00366 c1ccnc(c1)SCC(=O)NCC(=O)N JFD02003 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccc2F JFD01390 CCOC(=O)c1ccc(cc1)NC(=O)CSc2nncn2C JFD02010 CC1(C(=C)S/C(=N\c2ccccc2Cl)/N1C(=O)COc3cc(c(cc3Cl)Cl)Cl)C DSHS00462 CC1(C(=C)S/C(=N\c2ccccc2Cl)/N1C(=O)c3ccc(cc3)OC)C DSHS00463 Cc1ccc(c(c1)C)/N=C\2/NC(C(=C)S2)(C)C DSHS00479 Cc1ccc(c(c1)C)NC(=S)C(C#N)C(=O)Nc2c(cccc2Cl)C DP00455 CN(C)c1ccc(cc1)C(=O)NNS(=O)(=O)c2ccc(cc2)Cl DSHS00720 c1cc(ccc1/N=C/c2cc(cc(c2O)Br)Br)F DSHS00722 COc1cc(cc(c1OC)OC)/C=N/c2ccc(cc2)F DSHS00724 c1ccc2c(c1)c(=O)nc([nH]2)c3cccs3 DSHS00731 CCOC(=O)C1=C(NC2=C(C1c3ccc(cc3)OC)C(=O)c4c2cccc4)C JFD00439 Cc1ccc(cc1)S(=O)(=O)Nc2ccsc2C#N GK02472 c1cc(c(c(c1)F)NC(=O)c2cnc(nc2C(F)(F)F)N)F GK02476 c1ccc2cc(ccc2c1)C(=O)Cn3ccsc3=N JFD01979 Cc1c2c([nH]n1)NC(C3=C2CC(CC3=O)(C)C)c4ccc(cc4)N(C)C JFD01321 Cn1c2c(c(c(c1=O)[N+](=O)[O-])O)c(=O)n(c(=O)n2c3ccccc3)c4ccccc4 JFD01322 Cc1cc(n(n1)C)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C KM00008 Cc1cc(n(n1)C)NC(=O)c2ccc(cc2)[N+](=O)[O-] KM00009 CC(=O)c1c(cc(s1)c2ccccc2)N GK01045 Cc1ccc(cc1)C(=O)NNc2ccsc2C(=O)OC GK02414 COC(=O)c1c(ccs1)NNS(=O)(=O)c2ccccc2 GK02418 c1cc(sc1)/C=N/NC(=O)C(=O)Nc2ccc(c(c2)Cl)Cl JPV00019 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] DFP00345 COc1cc(cc(c1OC)OC)C(C#N)NCc2ccccc2 DSHS00560 COC(=O)C1C(C(S(=O)(=O)CS1(=O)=O)C(=O)OC)c2ccc(cc2)[N+](=O)[O-] JFD01345 CC1CC(CC(C1)(C)C)NC(=O)CC#N DP00481 CCOC(=O)C(=CNc1cc(sc1C(=O)C)C(C)(C)C)C(=O)OCC GK01041 COC(=O)c1c(ccs1)NNC(=O)c2ccc(cc2)[N+](=O)[O-] GK02412 CC(=O)c1c(ccs1)NC(=O)CCC(=O)O GK02426 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccccc3SCCC#N)Cl JP00790 COc1cc(cc(c1OC)OC)NC(=O)COc2cc(c(cc2Cl)Cl)Cl DSHS00484 COc1cc(cc(c1OC)OC)c2[nH]c3ccccc3c(=O)n2 DSHS00662 c1ccc(c(c1)C2Nc3ccccc3C(=O)N2)Cl DSHS00663 c1cc(cnc1)CN(CCC#N)C(=S)Nc2ccc(cc2)F JP00950 CC(C)(C)c1cc(c(s1)C(=O)N)NC(=O)C(Cl)Cl GK00993 COC(=O)c1cccc(c1)NC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00306 COC(=O)c1cccc(c1)NC(=O)NC(=O)c2ccco2 DFP00307 COC(=O)c1c(ccs1)NNC(=O)c2ccc(cc2)Cl GK02411 c1ccc(c(c1)CNC(=S)NC23CC4CC(C2)CC(C4)C3)Cl JFD00425 COC(=O)c1c(ccs1)N/N=C/c2cccc(c2)Cl GK02416 CC1c2ccsc2CCN1C(=O)c3cccs3 DFP00309 CC1c2ccsc2CCN1C(=O)c3cc(sc3)[N+](=O)[O-] DFP00310 CN(CCC#N)C(=S)Nc1cc(c(cc1OC)Cl)OC JP00762 COc1cccc2c1nc(cc2C(=O)O)c3ccccc3 DSHS00647 c1ccc(cc1)C2(c3cc(ccc3N=C2N)Cl)O DSHS00649 C/C(=N/NC(=O)N)/c1ccc(c(c1)[N+](=O)[O-])Sc2ccc(cc2)Cl JP00939 Cc1cc(n(n1)C(C)(C)C)NC(=O)Nc2ccc(cc2)Cl KM00050 Cc1cc(n(n1)C(C)(C)C)NC(=O)NC KM00051 CC1CC(CC1(C#N)Nc2ccc(cc2)CC#N)(C)C DSHS00679 c1cc(ccc1NCc2cc(ccc2O)Br)F DSHS00681 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCOCC2 DSHS00682 c1ccc(cc1)c2cc(n[nH]2)N KM00060 c1cc(ccc1S(=O)(=O)CCN2CCSCC2)Cl KM00061 c1cc(ccc1S(=O)(=O)CCN2CCOCC2)Cl KM00062 Cc1ccc(cc1)SCCS(=O)(=O)c2ccc(cc2)Cl KM00067 COc1cc(c(cc1Cl)OC)NS(=O)(=O)c2cccc(c2)C(F)(F)F DSHS00689 COc1cc(c(cc1Cl)OC)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DSHS00691 CC1(CN=C(S1)N(c2ccccc2)C(=O)Nc3ccc(c(c3)Cl)Cl)C JFD01426 COc1ccc(cc1)CC2CCC(=O)CC2 JFD01369 COC(=O)/C(=C/c1ccccc1)/c2ccccc2 JFD01370 c1cc2c(cc1F)c3c([nH]2)CCN(C3)Cc4ccc(cc4Cl)Cl JFD01372 CN1CCCCC(C1=O)C2=C(C(=O)CCC2)Cl JFD01358 Cc1ccccc1NC(C(F)(F)F)(C(F)(F)F)NC(=O)C JFD01414 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4c(onc4c5ccccc5Cl)C DSHS00515 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccccc4C DSHS00523 CC1CCCCN1S(=O)(=O)c2cc(ccc2Cl)Cl DP00320 Cc1cc(=O)n2c([nH]1)cc(n2)C KM00085 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(c(c3)F)F DSHS00810 c1ccc(c(c1)C(=O)Nc2ccccc2SCc3ccc(cc3)C#N)I DSHS00821 c1ccn(c1)c2ccsc2C(=O)O CC22101 c1cc(cnc1)CNC(=O)C(=O)Nc2ccc(cc2Cl)Cl JPV00031 CC1CCCN(C1)S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DP00323 CC1CCN(CC1)S(=O)(=O)c2cc(ccc2Cl)Cl DP00324 c1cc(ccc1NC(=S)N(CCC#N)C2CCCCC2)F JP00957 Cc1csc(c1NC(=S)OC)C(=O)OC GK02408 CCCCCCCCCCCCOc1ccc(cc1)C(=O)C JFD01510 CCOc1ccsc1C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N GK02545 CCOc1ccsc1c2nnc(o2)c3ccc(cc3)[N+](=O)[O-] GK02549 CC1=NN(C(=O)C1)c2ccc(cc2)C(=O)O JFD01519 COc1c(csc1C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N)Br GK02555 c1ccc(cc1)n2c(c(cn2)c3nnc(o3)c4cc(cc(c4)Cl)Cl)C(F)(F)F GK02559 Cc1ccc(cc1)S(=O)(=O)N(CCC#N)Cc2cccnc2 DSHS00634 CCOC(=O)c1ccc(cc1)N/N=C/c2cc(c(c(c2)OC)OC)OC JP00741 CSc1cccc(c1)NC(=O)C(=O)N/N=C/c2ccc(cc2)Cl JPV00082 c1cc(ccc1c2nc(on2)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-])Cl GK02453 c1cc(c(cc1Cl)Cl)NC(=O)C(=O)NCc2ccncc2 JPV00034 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3C(=O)c4ccccc4)Cl DSHS00641 CCOC(=O)/C(=C/c1ccc(cc1Cl)N(C)C)/C#N DP00692 CN(c1cc(c(cc1)/C=N/NC(=O)N/N=C/c2c(cc(cc2)N(C)C)Cl)Cl)C DP00695 c1ccc2c(c1)/C(=N/c3ccc(cc3)O)/C(=O)N2 JFD00460 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3ccccn3 DP00697 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3cccnc3 DP00698 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)F)Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00762 CSc1c(c(c(s1)NC(=O)N2CCOCC2)c3ccc(cc3)Cl)C#N KM01265 Cc1ccc(cc1)S(=O)(=O)CCSc2ccccc2 KM00156 c1ccc(cc1)S(=O)(=O)Cc2ccccc2[N+](=O)[O-] JFD01989 c1cc(ccc1CC#N)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DSHS00699 c1cc(sc1)/C=C(\C#N)/C(=O)N2CCCC2 DP00526 COc1cc(cc(c1OC)OC)C(=O)Nc2ccc(cc2C(=O)c3ccccc3)Cl DSHS00642 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3ccc(cc3Cl)Cl)Cl DSHS00646 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)Cl)NC(=O)OCC JFD01437 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(c2)C(F)(F)F JFD01393 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)NC JFD02099 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2F)F JFD01394 COc1ccc(cc1)/N=C/2\c3cc(ccc3N=C2O)Br DP00571 C/C(=N\NC(=O)CC#N)/c1ccccc1 DP00065 COc1ccc(cc1OC)/C=N/NC(=O)CC#N DP00067 COc1cc(ccc1O)/C=N/NC(=O)CC#N DP00069 CN(C)c1ccc(cc1)/C=N/NC(=O)CC#N DP00071 CCOc1ccsc1C(=O)NNC(=O)c2ccc(cc2)Cl GK02531 c1cc2c(cc1Cl)nco2 JFD01498 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C)NC(=O)c2cccc(c2)Cl JFD01438 Cn1cnnc1S(=O)(=O)Cc2ccccc2[N+](=O)[O-] JFD01994 c1ccc2c(c1)c(=O)n(c(=O)[nH]2)CCSc3ccccn3 JFD02000 Cc1ccc(c(c1)C)NC(=S)C(C#N)C(=O)N2CCCC2 DP00470 c1ccc(c(c1)NC(=O)c2cnc(nc2C(F)(F)F)N)F GK02464 c1cc(cc(c1)F)NC(=O)c2cnc(nc2C(F)(F)F)N GK02467 Cc1ccc(cc1)c2c(nc3ccccc3n2)c4ccc(cc4)Cl DP00568 c1cc(ccc1N2CCCC2=O)S(=O)(=O)Oc3ccc(cc3)Cl JFD00481 c1cc(ccc1n2c(c(cn2)C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N)C(F)(F)F)[N+](=O)[O-] GK02446 Cc1ccc(cc1)SC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK02448 c1cnccc1CNC(=O)CC#N DP00472 Cc1cc(n(n1)C)NC(=O)c2ccc(cc2Cl)Cl KM00006 CC1CC(CC(C1)(C)C)NC(=O)C(=O)Nc2ccc(cc2Cl)Cl JPV00037 CCCCCCCC(=O)c1ccc(cc1O)OCC JFD00497 c1cc(cc(c1)NC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)Nc4cccc(c4)C(F)(F)F)C(F)(F)F JP00964 c1ccc(cc1)Nc2c3c4c(sc3ncn2)CCCC4 JFD00496 c1ccc(cc1)CNC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2 JFD01398 c1cc(cnc1)C2SCCCS2 JFD02112 CCOc1ccccc1/C=C(\C#N)/C(=O)N DP00537 c1ccc(cc1)CC(=O)c2ccc(cc2)Cl DP00540 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)Cl)F JFD01402 CC1CN(CC(O1)C)CCC(=O)Nc2ccc(cc2C(=O)c3ccccc3)Cl DSHS00667 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2C#N DSHS00671 c1cc(ccc1/N=C/c2cc(ccc2O)Br)F DSHS00672 c1ccc2cc(c(cc2c1)C(=O)O)OC(=O)c3cccc(c3)Cl JP00902 c1cc(ccc1n2c(c(cn2)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] GK02454 CCCCCCCNC(=O)CCCCSc1[nH]c(c(n1)c2ccccc2)c3ccccc3 JFD02064 c1cc(ccc1CC#N)NC2(CCCCC2)C#N DSHS00675 CCCCCC/C=N/Nc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-] JFD00513 Cc1c(c(c(c(c1C)C)C(=O)CCC(=O)O)C)C DP00853 Cn1c(=O)c2ccccc2cn1 DP00854 CCc1ccc(cc1)C(=O)/C=C/Sc2nc3ccc(cc3s2)OCC JFD00592 CC(=O)OC[C@H]([C@H]([C@@H]([C@H](c1[nH]nnn1)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00519 c1cc(c(cc1NC(=O)C(=O)NN)Cl)Cl JPV00003 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCC(CC3)CCCC4CCN(CC4)C(=O)c5c(onc5c6c(cccc6Cl)Cl)C JP00999 c1ccc(cc1)n2c(=S)n(nn2)CN3CCCCC3 JFD02029 COC(=O)Nc1ccc(cc1)S(=O)(=O)C(F)(F)F JFD02031 c1cc(sc1)/C=C(\C#N)/C(=O)N2CCOCC2 DP00527 c1cc(sc1)/C=C(\C#N)/C(=O)N DP00529 c1cc2c(cc1/C=C(\C#N)/C(=O)N)OCO2 DP00533 c1ccc(cc1)C(=O)Nc2ccccc2 DP00449 c1cc(ccc1CC#N)NC2(C3CC4CC(C3)CC2C4)C#N DSHS00676 Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2OC)Cl)OC DSHS00677 COc1ccc(cc1)/C=C(\C#N)/C(=O)N2CCCC2 DP00491 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(cc3)F DP00602 C1[C@H](N[C@H](S1)[C@@H]([C@H]([C@@H](CO)O)O)O)C(=O)O JFD00420 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=S)Nc3ccccc3 JFD00423 Cc1c(c(=O)c2ccc(cc2o1)OC(=O)C)Oc3ccc(cc3)Cl JFD02125 CC(C)(C)c1cc(n[nH]1)C(F)(F)F JFD02132 c1ccc(cc1)C(=O)NC(=O)NC(C(C(F)(F)F)(F)F)(F)F JFD02134 CCOC(=O)/C(=C/Nc1cc(sc1C(=O)C)C(C)(C)C)/C#N GK01038 CNC(=O)Nc1ccc(cc1)C(C(=O)OC)(C(F)(F)F)O JFD02135 CCOC(=O)C(c1ccc(cc1)NC(=O)NC)(C(F)(F)F)O JFD02136 Cc1ccc(n1c2ccsc2C(=O)O)C GK02514 CCC(=O)Nc1ccsc1C(=O)OC GK02516 CS(=O)(=O)c1ccc(c(c1)Cl)C(=O)O JFD01500 c1ccc2c(c1)NC(N2)c3cccs3 DP00612 Cc1ccc(cc1)c2cn3c(n2)scn3 DP00620 c1cc(ccc1C(=O)CCCC(=O)O)F JFD02063 c1cc(ccc1c2cc(c(s2)C(=O)N)NC=C(C#N)C#N)Cl GK01071 CCc1nnc(s1)N DP00628 COc1ccc(cc1)C2C(=O)NC(=O)N2 JFD00506 c1ccc(cc1)C(=O)N[C@@H]2[C@H]([C@@H]([C@H](O[C@@H]2OC(=O)c3ccccc3)COC(=O)c4ccccc4)OC(=O)c5ccccc5)OC(=O)c6ccccc6 JFD00415 c1cc(ccc1C(=O)NCC(=O)NN)Br JFD02079 c1ccc(cc1)C(=O)N[C@@H]2[C@H]([C@@H]([C@H](O[C@H]2OC(=O)c3ccccc3)COC(=O)c4ccccc4)OC(=O)c5ccccc5)OC(=O)c6ccccc6 JFD00417 CC(=O)OC[C@@H]([C@@H]([C@H]([C@@H](C(=O)Nc1ccccc1)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00521 CC(=O)Oc1ccc(cc1OC(=O)C)c2c(c(=O)c3c(o2)cc(cc3OC(=O)C)OC(=O)C)OC(=O)C JFD00524 Cc1cccc(c1)NC(=O)c2ccccc2 DP00450 Cc1ccccc1NC(=O)c2ccccc2 DP00451 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)Oc2ccc3c(c2)OC(CC3=O)c4ccccc4)OC(=O)C)OC(=O)C)OC(=O)C JFD00526 Cc1ccc(c(c1)C)NC(=S)C(C#N)C(=O)N2CCOCC2 DP00453 c1ccc2c(c1)C(=O)C(C2=O)C#N JFD02082 CC(=O)C1C(=O)c2cccc(c2C1=O)[N+](=O)[O-] JFD02083 CC(=O)c1c(cc(s1)c2ccccc2)NC(=O)C(Cl)Cl GK01047 COc1ccccc1/N=C\2/N(C3(CCCCC3)C(=C)S2)C(=O)c4ccccc4Cl DSHS00446 c1c2c(cc(c1Cl)Cl)C(=O)CC2=O JFD02085 CC(=O)c1ccc(c(c1)[N+](=O)[O-])Sc2ccccc2 JP00697 CC1(C(=C)S/C(=N\c2cccc(c2)OC)/N1C(=O)c3ccc(cc3)Cl)C DSHS00449 CC(C)c1ccc(cc1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00840 c1cc(oc1/C=C/C(=O)N2CCCCC2)[N+](=O)[O-] JFD00509 Cc1cccnc1n2c(=O)c3ccccc3nc2c4ccccc4 DP00700 Cc1ccnc(c1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00701 CCOC(=O)c1c2c(sc1NC(=O)C(F)(F)F)CCCC2 JFD00466 Cc1cccc(n1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00702 COc1ccccc1/N=C\2/N(C3(CCCCC3)C(=C)S2)C(=O)c4cccc(c4)Cl DSHS00447 c1ccc2c(c1)C(=O)NC(N2)c3ccc(cc3)Cl DSHS00664 CC1CCN(CC1)C(=O)C(C#N)C(=S)Nc2cccc(c2)OC DP00464 CC1(C(=C)S/C(=N\c2cccc(c2)OC)/N1C(=O)c3ccc(cc3)[N+](=O)[O-])C DSHS00454 CC1(C(=C)S/C(=N\c2ccccc2Cl)/N1C(=O)c3cc(c(c(c3)OC)OC)OC)C DSHS00455 Cc1ccc(c(c1)C)NC(=S)C(C#N)C(=O)Nc2ccccc2C DP00452 Cc1ccc(c(c1)C)NC(=S)C(C#N)C(=O)N2CCC(CC2)C DP00454 Cc1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=S)N2 JFD00448 c1c(nc(nc1O)S)C(F)(F)F GK02562 c1cc(c(cc1Cl)Cl)NC(=O)C(=O)NN JPV00016 Cc1ccc(cc1)C(=O)NNC(=O)CSc2c3c(c(cs3)C)ncn2 GK02563 Cc1csc2c1ncnc2SCC(=O)NNS(=O)(=O)c3ccc(cc3)NC(=O)C GK02568 Cc1c(c(n(n1)C)NC(=O)c2ccccc2)Br KM00016 Cc1csc2c1ncnc2SCC(=O)NNS(=O)(=O)c3ccc(cc3)C(F)(F)F GK02570 c1ccc(c(c1)NC(=S)C(C#N)C(=O)Nc2cccc(c2)C(F)(F)F)Cl DP00477 COC(=O)C1C(C(S(=O)(=O)CS1(=O)=O)C(=O)OC)c2ccc(cc2)O JFD01343 c1cc(c(c(c1)Cl)/C=N/NC(=O)C2CC2)F JW00043 c1ccc(c(c1)c2nc(no2)c3ccc(cc3F)F)Cl GK02641 Cn1c2c(cc(s2)C(=O)OC)c(n1)C(F)(F)F GK02644 c1cc(c(cc1Cl)S(=O)(=O)N2CCCCC2)Cl DP00318 c1ccc(cc1)C(=O)N(C(=O)c2ccccc2)C(=O)c3ccccc3 JFD00418 c1ccc(c(c1)/C=N/C(=C(/C#N)\N)/C#N)[N+](=O)[O-] KM00024 CCOC(=O)c1c2c(sc1NS(=O)(=O)c3ccc(cc3)C)CCCC2 DSHS00656 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)CCN3CCCc4c3cccc4)Cl DSHS00657 CCOC(=O)c1c2c(sc1NS(=O)(=O)c3ccc(cc3)Br)CCCC2 DSHS00660 Cc1c(c(n(n1)C)NC(=O)c2ccccc2Cl)Br KM00031 Cc1c(c(n(n1)C)NC(=O)c2ccc(cc2)[N+](=O)[O-])Cl KM00037 c1ccc2c(c1)C(=O)NC(N2)c3ccc(c(c3)Cl)Cl DSHS00665 c1ccc(cc1)COC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2 JFD01409 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccc(cc1)Cl JFD01412 Cc1c(c(=O)n(n1C)c2ccccc2)CN3CCCC(C3)C.Cl KM00039 COc1ccccc1N2CCN(CC2)Cc3ccc(cc3)F JFD01356 CCN(CC)CCC1S(=O)(=O)C(C(C(S1(=O)=O)C(=O)OC)c2ccc(cc2)OC)C(=O)OC JFD01353 c1ccc(cc1)C2C3=C(c4ccccc4C3=O)NC(=S)N2 JFD00447 CC(C)(C)c1cc(c(s1)C(=O)N)NC(=O)CC#N GK01052 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N/N=C/c2cc(cc(c2O)Cl)Cl JP00662 CC1CC(CC(C1)(C)C)N(CCC#N)C(=O)c2cc(c(c(c2)OC)OC)OC DSHS00772 COc1cc(cc(c1OC)OC)C(=O)N(CCC#N)Cc2ccncc2 DSHS00776 COc1cc(cc(c1OC)OC)C(=O)N(CCC#N)Cc2cccnc2 DSHS00777 Cc1ccc(n1c2ccsc2C(=O)OC)C GK02496 COc1c(csc1C(=O)OC)Br GK02499 CCOC(=O)c1ccc(cc1)S(=O)(=O)NC2(CCCCC2)C#C DSHS00780 COc1c(c(sc1C(=O)OC)Br)Br GK02500 CCOc1ccsc1C(=O)Nc2ccc(cc2)Cl GK02507 c1ccc(cc1)C(=O)c2cc3c4ccccc4ccc3oc2=O JFD01483 C/C(=N\OCc1ccc(cc1)[N+](=O)[O-])/c2ccc(c(c2)[N+](=O)[O-])Sc3ccccn3 JP00692 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C GK02430 c1cc(c(cc1Cl)Cl)NC(=O)C(=O)NC2CCCCC2 JPV00030 COc1cc2c(cc1OC)C(=NCC2)c3ccccc3NC(=O)c4cccc(c4)Cl JP00750 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1nc2ccccc2s1 JFD01413 c1ccc(c(c1)NC(=O)c2ccc(cc2)[N+](=O)[O-])Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00747 Cc1csc2c1ncnc2N3CCN(CC3)C(=O)Nc4ccc(cc4)OC(F)(F)F GK02681 Cc1ccc(cc1[N+](=O)[O-])NC(=S)N2CCN(CC2)c3c4c(c(cs4)C)ncn3 GK02685 c1ccc(c(c1)NC(=O)C(Cl)Cl)Sc2ccc(cc2[N+](=O)[O-])Cl DSHS00753 Cc1cc2c(cc1C)/N=C(\c3ccccc3C(=O)N2)/c4ccccc4 DP00764 c1ccc(c(c1)OS(=O)(=O)c2ccc(cc2)N3CCCC3=O)Cl JFD00480 c1ccnc(c1)/C=C/c2cccc(c2)[N+](=O)[O-] DSHS00492 CN(CCC#N)c1ccc(cc1)/C=N/c2ccc(cc2)C(=O)O DSHS00503 C[C@@]1(CCC2C(C1/C=C/3\C(=O)c4ccccc4N3)CCC5[C@@]2(CC=CC5)C)C(=O)O DSHS00509 COc1cc(cc(c1OC)OC)C(=O)Nc2cc(c(cc2OC)Cl)OC DSHS00696 COc1ccc(c(c1)NC(=O)c2ccccc2NC(=O)c3ccccc3)OC DP00708 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)OC)NC(=O)c2ccccc2Cl JFD02204 Cc1ccc(cc1C)c2c3ccccc3c(=O)n(n2)c4ccccc4 DP00594 Cc1csc(c1NC(=O)C(Cl)Cl)C(=O)OC GK01263 CCOC(=O)C(c1ccc(cc1)N(C)C(=O)Nc2ccc(cc2)Cl)(C(F)(F)F)O JFD02190 CCOC(=O)C(c1ccc(cc1)N(C)C(=O)Nc2cccc(c2)Cl)(C(F)(F)F)O JFD02191 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3ccc(cc3)Cl DP00714 c1cc(ccc1SCCS(=O)(=O)c2ccc(cc2)Cl)Cl KM00070 c1ccc(cc1)c2cc(=O)n3c([nH]2)cc(n3)c4ccccc4 KM00073 COc1ccc(cc1OC)CCNC(=O)CC#N KM00078 c1cc(ccc1CC#N)NC2(CCCCCCCCCCC2)C#N DSHS00695 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccccc2C(F)(F)F JFD01392 CCN(CCS(=O)(=O)c1ccccc1)S(=O)(=O)c2ccc(cc2)Cl KM00076 CCN(CCS(=O)(=O)c1ccccc1)S(=O)(=O)c2ccc(cc2)C KM00077 c1ccc(cc1)S(=O)(=O)CCS(=O)(=O)c2ccc(cc2)Cl KM00080 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C)NC(=O)OCC JFD01435 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)F)NC(=O)OCC JFD01436 Cc1ccc(cc1C)c2c3ccccc3c(=O)n(n2)CCO DP00595 c1ccc2c(c1)c(nn(c2=O)CCO)c3ccc(cc3)F DP00597 c1ccc(cc1)n2c(cc(n2)C3CC3)NC(=O)Nc4ccc(cc4)Cl KM00207 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNC(=O)Sc3ccccc3[N+](=O)[O-] DSHS00865 Cc1c(csc1C(=O)N/N=C/c2cccs2)S(=O)(=O)c3ccc(cc3)Cl KM01382 CCOC(=O)C(C(F)(F)F)(Nc1ccccn1)NC(=O)c2ccccc2Cl JFD02207 CCOC(=O)C(C(F)(F)F)(Nc1cc(ccn1)C)NC(=O)c2ccccc2Cl JFD02210 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(=O)C)NC(=O)c2ccccc2Cl JFD02212 Cc1ccc(cc1)c2c3ccccc3c(=O)[nH]n2 DP00604 Cc1ccc(cc1C)c2c3ccccc3c(=O)[nH]n2 DP00605 Cc1ccccc1N(C2=NCC(S2)(C)C)C(=O)Nc3ccccc3 JFD01433 CCOc1ccsc1C(=O)NNC(=O)c2ccc(cc2)[N+](=O)[O-] GK02532 CCOc1ccsc1C(=O)NNC(=O)c2ccco2 GK02535 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1F)F)NC(=O)OCC JFD01439 CCOc1ccsc1NC(=O)Nc2ccc(cc2)OC(F)(F)F GK02541 CCOc1ccsc1NC(=O)Nc2cccc(c2)C(F)(F)F GK02542 COc1ccccc1NC(=S)NNC(=O)CSc2ccccc2[N+](=O)[O-] DSHS00871 c1ccc(c(c1)[N+](=O)[O-])SCC(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F DSHS00872 CCCSc1ccc(c(c1)/N=C(/NC(=O)OC)\SC)[N+](=O)[O-] JFD00573 CCSc1c(c(c(s1)C(=O)O)c2cccs2)C#N KM01657 CCCSc1c(c(c(s1)C(=O)O)c2cccs2)C#N KM01658 CCOC(=O)c1cnc2cc(nn2c1C)c3ccc(cc3)Cl KM01666 CCCCCCCCOc1ccc(cc1)C(=O)C JFD01529 COc1ccc(c(c1)NC(=O)C(=O)NN)OC JPV00086 CCOc1ccsc1c2nnc(o2)c3ccc(cc3)Cl GK02544 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)N)Cl DP00525 c1ccc2c(c1)c(c[nH]2)/C=C(\C#N)/C(=O)N DP00532 CC(=O)Nc1ccc(cc1)NC(=O)C2CC2(C)C JFD00451 c1ccc(cc1)c2c3ccccc3c(=O)on2 DP00671 COC(=O)c1c(cc(s1)c2ccc(cc2)F)N GK01138 c1cc(sc1)C(=O)Nc2cc(sc2C(=O)N)c3ccsc3 GK01161 c1cc(cc(c1)F)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2 JFD02193 c1ccc(cc1)c2c(c3n[nH]c(=S)n3nc2c4ccccc4)c5ccccc5 JFD00403 CCOC(=O)c1c(c2c(c(nnc2s1)c3ccccc3)c4ccccc4)N JFD00406 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)NN)N JFD00407 CN(C)c1ccc(c(c1)Cl)/C=C(\C#N)/C(=O)N DP00691 Cc1c(c(=O)c2ccc(cc2o1)O)Oc3ccc(cc3)Cl JFD02121 Cc1c(c(n(n1)c2ccccc2)NC(=O)C(Cl)(Cl)Cl)Br KM00144 c1ccc(cc1)c2c3ccccc3c(nn2)O DP00601 Cc1c(c(n(n1)C)NC(=O)c2ccc(cc2)Cl)Br KM00032 CCOC(=O)c1c(nc(s1)N)C(F)(F)F JFD01572 Cc1c(c(=O)n(n1C)c2ccccc2)CN3CCCCC3C.Cl KM00040 Cc1csc2c1ncnc2N3CCN(CC3)C(=O)c4ccc(cc4)Cl GK02667 Cc1csc2c1ncnc2N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl GK02675 c1ccc(cc1)c2cc3nnc(c(n3n2)c4ccccc4Cl)C(=O)N KM00219 c1cc(ccc1F)SCC#N KM01391 COC(C(F)(F)F)(C(F)(F)F)NC(=O)c1ccccc1 JFD01403 c1ccc(cc1)c2c(nc(s2)N)c3ccc(cc3)Cl.Br DP00543 Cc1nc(c(s1)c2ccccc2)c3ccc(cc3)Cl.Br DP00547 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)F)F JFD01407 Cc1c(c(n(n1)C)NC(=O)c2ccccc2Cl)Cl KM00034 COc1ccc(cc1)c2cc(c(s2)C(=O)N)NS(=O)(=O)c3ccc(cc3)C(F)(F)F GK01172 Cc1ccc(cc1)SCCS(=O)(=O)c2ccc(cc2)C KM00155 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2F)F)F JFD01406 CCOc1ccsc1C(=O)O GK02486 COC(=O)c1c(ccs1)NC(=O)c2ccc(cc2Cl)Cl GK02488 CCNc1nc(c(s1)c2ccc(cc2)C)c3ccc(cc3)Cl.Br DP00557 c1cc(ccc1NC(=S)N(CCC#N)Cc2ccncc2)F JP00958 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)N(C5=O)c6ccc(c(c6)Cl)Cl JFD00491 Cc1csc(c1Cl)C(=O)OC GK01297 c1csc(c1Cl)C(=O)O GK01306 c1cc(ccc1NC(=O)c2c(ccs2)Cl)Cl GK01308 CCOc1ccc2c(c1)sc(n2)S/C=C/C(=O)c3ccc(cc3)C JFD00591 c1cc(sc1)c2cc(c(s2)C(=O)N)N GK01164 c1cc(cnc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)N2CCCC2=O JFD02194 Cc1ccc(cc1)C(=O)Nc2cc(sc2C#N)c3ccc(cc3)F GK02581 COc1ccc(cc1)C(=O)c2ccccc2C(=O)O DP00607 Cc1c(c(n(n1)C)NC(=O)c2ccc(cc2)Cl)Cl KM00036 c1cc(ccc1C(F)(F)F)S(=O)(=O)Nc2cc(sc2C(=O)N)c3ccsc3 GK01157 c1cc(c(cc1Cl)S(=O)(=O)N2CCOCC2)Cl DP00314 c1cc(ccc1c2nnc3n2nc(s3)c4ccc(cc4)Cl)Cl DP00725 CN\1C(=O)C(S/C1=N/N=C/c2cc(c(c(c2)OC)OC)OC)CC(=O)O DP00734 Cc1ccc(cc1)c2c(nc(s2)N)c3ccc(cc3)Cl.Br DP00554 c1ccc(cc1)c2c(nc3ccccc3n2)c4ccc(cc4)Cl DP00564 Cc1ccc(cc1)S(=O)(=O)C=C KM00150 Cc1c(c(c2ccccc2n1)C(=O)O)C(=O)O KM00251 c1ccc(c(c1)NC(=S)NNC(=O)CSc2ccccc2[N+](=O)[O-])Cl DSHS00873 COc1ccccc1n2c(nnc2S)CSc3ccccc3[N+](=O)[O-] DSHS00875 C=CCn1c(nnc1S)CSc2ccccc2[N+](=O)[O-] DSHS00884 Cc1csc(c1N2C(=O)c3ccccc3C2=O)C(=O)OC GK01271 c1cc(c(cc1Cl)S(=O)(=O)N2CCCC2)Cl DP00316 CC(=O)NC(CC#N)[C@H]([C@@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00442 Cc1ccc(cc1C)C(=O)Nc2ccccc2Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00743 CC1=C(C(C2=C(N1)c3ccccc3C2=O)c4ccccc4)C(=O)Nc5ccccc5 JFD00444 Cc1cc(=O)n2c([nH]1)cc(n2)c3cccs3 KM00124 c1ccc(cc1)c2cc(=O)n3c([nH]2)cc(n3)c4cccs4 KM00126 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N)Cl DSHS00892 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N DSHS00893 CSC(=CC(=O)c1ccc(cc1)F)SC GK01204 CC(C)(C)c1ccc(cc1)C(CCCN2CCC(CC2)C(c3ccccc3)(c4ccccc4)O)O JFD01583 COc1cccc(c1)C2C(=O)c3ccccc3C2=O JFD02086 COc1cc(ccc1NC(=O)Nc2ccc3ccccc3c2)C(C(=O)OC)(C(F)(F)F)O JFD02161 c1ccc2c(c1)nc-3c(n2)-c4cccc5c4c3ccc5 JFD01477 CC(=O)c1c(cc(s1)c2ccccc2)NC(=O)C(F)(F)F GK01049 Cc1ccc(cc1C)C(=O)c2ccccc2C(=O)O DP00590 c1ccc(c(c1)C(=O)c2ccc(cc2)F)C(=O)O DP00596 CCOC(=O)C(c1ccc(cc1)NC(=O)Oc2ccccc2)(C(F)(F)F)O JFD02145 CCOC(=O)C(c1ccc(cc1)N(C)C(=O)c2ccc(c(c2)Cl)Cl)(C(F)(F)F)O JFD02147 CCOC(=O)Cc1csc(n1)NC(=O)CSc2nnc(s2)C JFD02081 c1ccnc(c1)CCNC(=O)CC#N DP00485 C1CC(OC1)CNC(=O)CC#N DP00489 Cc1cc(ccc1NC(=O)Nc2ccc3ccccc3c2)C(C(=O)OC)(C(F)(F)F)O JFD02160 CC(C)SCC(=O)Nc1nc(cs1)CC(=O)O JFD02047 CCNC(=O)SCC(C(=O)O)N JFD00511 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4ccc(cc4)F DP00598 CC(=O)O[C@@H]1[C@H]2CO[C@H](O2)[C@@H]([C@H]1OC(=O)C)OC(=O)C JFD00517 c1c(c(cc(c1Cl)Cl)C(=O)O)C(=O)O JFD02055 c1ccc(c(c1)C(=O)Nc2c(csc2Br)S(=O)(=O)c3ccc(cc3)Cl)Cl KM01650 Cc1c(c(c(c(c1C)C)CSCC(=O)NNS(=O)(=O)c2ccc(cc2)F)C)C DSHS00853 C#CC1(CCCCC1)NS(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccccc3N DSHS00855 Cc1c(nnc2n1nc(c2)c3ccccc3)C(=O)N KM00216 c1ccc2c(c1)CCc3ccccc3NC2.Cl JFD01542 Cc1ccc(c(c1)C)NC(=O)C(C#N)C(=S)Nc2ccccc2Cl DP00458 COc1ccccc1NC(=S)C(C#N)C(=O)N2CCCC2 DP00460 CC(C)(C)/C=N/NC(=O)C1CC1 JW00044 Cc1cc([nH]n1)NS(=O)(=O)c2cccs2 JW00053 COc1cccc(c1)NC(=S)C(C#N)C(=O)N2CCCC2 DP00463 C1CCc2c(sc(c2C#N)N)CC1 DP00789 c1ccc(cc1)/C/2=N/CCCOC(=O)c3c2cccc3 DP00809 c1ccc2c(c1)c(ncn2)Nc3cccc(c3)Cl.Cl DP00818 c1ccc2c(c1)c(ncn2)Nc3ccc(cc3)Br.Cl DP00820 CC(=O)c1ccccc1N/C=C/c2nnnn2c3ccc(cc3)I JFD00608 Cc1ccc(cc1)n2c(nnn2)/C=C/Nc3ccccc3C#N JFD00610 c1ccc(cc1)n2c(nnn2)C/C=N/Nc3cc(cc(c3)Cl)Cl JFD00612 CCN(CCS(=O)(=O)c1ccc(cc1)Cl)C(=O)Nc2ccc(cc2)Cl KM00107 CCN(CCS(=O)(=O)c1ccc(cc1)Cl)C(=S)Nc2ccccc2Cl KM00108 CCN(CCS(=O)(=O)c1ccc(cc1)Cl)C(=S)Nc2ccc(c(c2)Cl)Cl KM00112 CCOC(=O)c1cnn(c1NC(=O)c2ccc(cc2Cl)Cl)C GK01091 c1csc(c1C#N)NC(=O)C(Cl)Cl GK01097 c1cc(oc1)CNC(=O)CC#N DP00466 c1ccc(c(c1)CO)C(=O)NNC(=O)c2ccc(c(c2)Cl)Cl JPV00059 c1ccc(c(c1)CO)C(=O)N/N=C/c2ccccc2Cl JPV00062 c1cc(ccc1Sc2ncc(c(n2)C(F)(F)F)C(=O)Sc3ccc(cc3)Cl)Cl GK02605 CCc1nn2cc(nc2s1)c3ccc(cc3)F DP00639 C1CCc2c(c(c(s2)NC(=O)/C=C/C(=O)O)C#N)C1 GK02610 c1ccc(c(c1)CO)C(=O)N/N=C/c2ccc(cc2)O JPV00065 CC1(c2ccccc2N(C13C=Cc4cccc(c4O3)[N+](=O)[O-])C)C JFD01538 CC(C)(C)c1cc(c(s1)C(=O)N)NC(=O)/C(=C/c2cccc(c2Cl)Cl)/C#N GK01083 Cn1cc(c(n1)C(F)(F)F)COC(=O)Nc2c(cccc2Cl)Cl GK01084 c1cc(ccc1c2cc(nc(n2)N)N)Cl GK01237 Cn1cc(c(n1)N2C(=O)C=CC2=O)Br GK01249 c1ccc(c(c1)C2C(=O)c3ccccc3C2=O)[N+](=O)[O-] JFD02090 CCOc1ccc(cc1)/C=C(\C#N)/C(=O)N2CCOCC2 DP00500 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C(C(=O)OCC)(C(F)(F)F)O JFD02184 COc1c(csc1c2nnc(o2)c3cccc(c3)[N+](=O)[O-])Br GK02588 c1cc(ccc1S(=O)(=O)N(CCC#N)CC2CCCO2)Br DSHS00633 COc1cc(cc(c1OC)OC)C(=O)N/N=C/c2ccc3c(c2)OCO3 DSHS00638 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)C(Cl)Cl)Cl DSHS00639 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3ccc(cc3)Cl)Cl DSHS00640 Cc1cc(n(n1)C)NC(=O)NC KM00018 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3ccccc3Cl)Cl DSHS00644 c1ccc2c(c1)C(=NC(N2)c3cccc(c3)[N+](=O)[O-])O DSHS00650 c1ccc2c(c1)c(nc(n2)c3cccc(c3)[N+](=O)[O-])O DSHS00651 Cc1cc(n(n1)C)NC(=O)Nc2ccccc2 KM00019 Cc1cc(n(n1)C)NC(=O)Nc2ccc(cc2)Cl KM00020 CCOC(=O)c1cnc(nc1C(F)(F)F)N GK01243 CCOC(=O)C(c1ccc(cc1)N2C(=O)c3ccccc3C2=O)(C(F)(F)F)O JFD02151 COc1cc(ccc1NC(=O)Nc2cccc(c2)Cl)C(C(=O)OC)(C(F)(F)F)O JFD02176 CCOC(=O)C(c1ccc(c(c1)C)NC(=O)Nc2ccc(cc2)Cl)(C(F)(F)F)O JFD02179 c1ccc2c(c1)cccc2/C=C(\C#N)/C(=O)N DP00538 CSc1cccc(c1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00710 c1ccc(cc1)c2c(nc(s2)Nc3ccccc3)c4ccc(cc4)Cl.Br DP00544 CC(C)(C)C(=O)Nc1cc(nn1c2ccccc2)C3CC3 KM00258 Cc1cc(n(n1)C)NC(=O)C(C)(C)C KM00043 Cc1cc(n(n1)C)NC(=O)Nc2cccc(c2)C(F)(F)F KM00021 c1ccc(c(c1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00770 CC1(C(CCC1(C)C(=O)N2CCOCC2)C(=O)N3CCOCC3)C JFD02113 CCOc1ccc(cc1)/C=C(\C#N)/C(=O)N DP00536 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccccc2SCc3ccc(cc3)C#N DSHS00826 CCOC(=O)/C(=N/Nc1cc(n[nH]1)c2ccccc2)/C#N KM00204 Cc1csc2c1n3c(c(nn3)C#N)[nH]c2=O GK01317 Cc1c(c(no1)c2ccccc2)C(=O)NNC(=O)CSc3ccccc3[N+](=O)[O-] DSHS00863 c1ccc(c(c1)C(=O)Nc2ccccc2Sc3ccc(cc3[N+](=O)[O-])Cl)Cl DSHS00748 c1ccc(cc1)CN2CCCC2C(=O)Nc3ccccc3C(=O)c4ccccc4 JFD01484 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C#N)C(C)(C)C GK02510 CCOc1ccsc1C(=O)Nc2ccc(cc2)OC(F)(F)F GK02492 Cc1cc(n(n1)C(C)(C)C)N KM00047 Cc1cc(n(n1)C(C)(C)C)NC(=O)Nc2ccccc2 KM00049 Cc1csc2c1ncnc2N3CCN(CC3)S(=O)(=O)c4ccsc4C(=O)OC GK02678 c1cc(ccc1/N=C/c2cc(cc(c2O)Cl)Cl)F DSHS00723 CN(C)c1ccc(cc1)C(=O)NNS(=O)(=O)c2cccc(c2)C(F)(F)F DSHS00727 CN(C)c1ccc(cc1)C(=O)NNS(=O)(=O)c2ccc(cc2)F DSHS00728 CN(C)c1ccc(cc1)C(=O)NNS(=O)(=O)c2ccc(c(c2)OC)OC DSHS00729 c1ccc2c(c1)C(=O)NC(N2)c3cccs3 DSHS00730 c1ccc(c(c1)N)Sc2ccccc2[N+](=O)[O-] DSHS00737 CCOC(=O)c1cnn(c1NS(=O)(=O)c2ccc(cc2)Cl)C GK01133 CCN(CC)c1ccc2cc(c(=O)oc2c1)C(=O)c3cc4ccc(cc4oc3=O)N(CC)CC JFD01496 CC1CC(CC(C1)(C)C)N(CCC#N)S(=O)(=O)c2ccc(cc2)Br DSHS00624 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N(CCC#N)C2CCCCC2 DSHS00625 CCOC(=O)C(c1ccc(cc1)N(C)C(=O)OCC)(C(F)(F)F)O JFD02089 CC(=O)C1C(=O)c2c(c(c(c(c2Cl)Cl)Cl)Cl)C1=O JFD02091 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccccc3Sc4ccc(cc4[N+](=O)[O-])Cl)Cl DSHS00745 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC2CC3CCC2(C3(C)C)C JFD01383 c1ccc(cc1)Oc2cc(c3c(c2N)C(=O)c4ccccc4C3=O)O JFD02095 Cc1cccc(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccccc2 JFD01387 c1cc(ccc1c2cc(c(s2)C(=O)N)NS(=O)(=O)c3ccc(cc3)C(F)(F)F)F GK01149 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)N)c3ccsc3 GK01154 c1ccc(cc1)n2c(=O)c3ccccc3cn2 DP00855 c1ccc(cc1)Cn2c(=O)c3ccccc3cn2 DP00856 c1ccc(cc1)C(=O)NC(=S)Nc2c(c(n[nH]2)C3CC3)/N=N/c4ccc(cc4)Br KM00434 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(=O)N(CCC#N)C3CCCCC3 DSHS00897 CC(C)(C)OC(=O)NCC(=O)OCc1ccc(cc1)CC(=O)O JFD01594 c1cc(oc1)c2c(c(nc(c2C#N)Sc3ccc(cc3)Cl)N)C#N KM00563 c1ccc(c(c1)c2c(c(nc(c2C#N)Sc3ccc(cc3)Cl)N)C#N)Cl KM00564 Cc1ccc(cc1)CC(=O)c2ccc(cc2)Cl DP00550 CC(C)(C#C)NC(=O)NCCCCCCNC(=O)NC(C)(C)C#C DP00784 CC(C)(C)c1cc(c(s1)C(=O)N)NC(=O)/C(=C/c2ccc(cc2)C(F)(F)F)/C#N GK01080 CC1=CC(=O)N(C1=O)c2ccn(n2)C GK01232 CC(c1ccccc1)(C(=O)O)O JFD02109 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1F)NC(=O)c2ccccc2Cl JFD02200 CC(=O)OI(c1cccc(c1)OC)OC(=O)C JFD01485 Cc1c(c(n(n1)Cc2nnc(o2)SCC(=O)Nc3ccc(cc3Cl)Cl)C)Br KM04747 CCO/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl KM00449 C#CC1(CCCCC1)NS(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccc(cc3)Cl DSHS00901 CC1(C2CCC13CS(=O)(=O)[N@]4C3(C2)O4)C JFD01493 CCOC(=O)CSc1ccc(cc1[N+](=O)[O-])S(=O)(=O)NC2(CCCCC2)C#C DSHS00911 C#CC1(CCCCC1)NC(=O)NCCCCCCNC(=O)NC2(CCCCC2)C#C DP00786 Cc1cc2c(cc1C)nc(c(n2)c3ccccc3)c4ccc(cc4)Cl DP00618 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3ccc(cc3)F DP00707 Cc1c(c(=O)n(n1C)c2ccccc2)N3C(=O)c4ccc(cc4C3=O)Br JFD00474 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)C(F)(F)F)NC(=O)c2ccccc2Cl JFD02201 CCC(=O)NC(C(=O)OCC)(C(F)(F)F)Nc1ccc(cc1OC)C(C(=O)OCC)(C(F)(F)F)O JFD02138 Cc1ccc(cc1)C(=O)c2ccccc2C(=O)O DP00589 CN1c2ccccc2C(=O)/C(=C\Nc3ccc(cc3)F)/S1(=O)=O KM01336 COc1ccc(cc1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00715 c1cc(ccc1C(=O)CSC2=NCCCCC2)[N+](=O)[O-].Br DP00716 CCOC(=O)C(c1ccc(c(c1)C)NC(=O)Nc2cccc(c2)Cl)(C(F)(F)F)O JFD02181 COc1c(csc1C(=O)O/N=C(/c2ccc(cc2F)F)\N)Br GK02599 CCc1ccccc1NC(=O)c2c(c(cs2)Br)OC GK02603 CN(C)CCS(=O)(=O)C JFD00577 Cc1cc(=O)[nH]n(c1=O)C(=O)Cc2ccc(c(c2)OC)OC GK01226 c1cscc1c2cc(c(s2)C(=O)N)N GK01140 Cc1c(c(c(c(c1C)C)CSCC(=O)NNS(=O)(=O)c2cccc(c2)C(F)(F)F)C)C DSHS00858 c1ccc(c(c1)[N+](=O)[O-])SCC(=O)NN DSHS00862 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=O)CSc3ccccc3[N+](=O)[O-] DSHS00864 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3ccc(cc3)Br DP00717 Cc1cc(n(n1)C)NC(=S)Nc2ccccc2F KM00063 c1ccc(cc1)c2cc(n(n2)c3ccccc3)N KM00154 CN(C)/C=N/c1c(csc1C(=O)OC)C#N KM01705 COc1c(ccc(c1)/C=N/NC(=S)N/N=C/c2cc(c(cc2)O)OC)O DP00721 COc1cc(cc(c1OC)OC)/C=N/NC(=S)N DP00728 C(C1C(=O)NC(=N)S1)C(=O)O DP00739 Cc1cc2nnc(c(n2n1)C)C(=O)C KM01302 c1cscc1/C=C/C(=O)Nc2cc(sc2C(=O)N)c3ccsc3 GK01176 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1)NC(=O)c2ccccc2Cl JFD02197 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4ccc(cc4)Cl DP00586 Cc1ccc(cc1)C(=O)/C=C/S(=O)(=O)c2cc(ccc2Cl)Cl JFD00589 c1cscc1c2cc(c(s2)C(=O)N)NC(=O)C(F)(F)F GK01147 c1ccc(cc1)S(=O)(=O)CCSCC(=O)O KM01716 CC(=N)Nc1cc(n[nH]1)c2ccccc2.I KM00554 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])S(=O)(=O)Nc3ccc(c(c3)C(F)(F)F)Cl)Cl DSHS00918 Cn1c(cc(n1)C2CC2)NC(=O)Nc3ccc(cc3)OC(F)(F)F KM04533 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCc4cccc(c4)Cl KM04542 CSc1c2c([nH]cn2)ncn1 JFD01558 c1cc2ccc3ccc(c4c3c2c(c1)cc4)CCCC(=O)O JFD01560 c1ccc(cc1)c2cnc(o2)c3cccc4c3cccc4 JFD01563 Cc1nn2cc(nc2s1)c3cccc(c3)[N+](=O)[O-] DP00633 CC(C)(C)c1cc2[nH]c(cc(=O)n2n1)C(F)(F)F KM00318 CC(C)(C)c1cc2[nH]c(cc(=O)n2n1)c3ccccc3 KM00321 CCOC(=O)N/N=C/c1ccc(cc1)N(C)CCC#N DP00688 c1cc(ccc1c2cc(c(s2)C(=O)N)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)F GK01148 Cn1ccc(n1)N2C(=O)c3ccccc3C2=O GK01235 CCOC(=O)C(C(F)(F)F)(Nc1ccc(c(c1)Cl)F)NC(=O)c2ccccc2Cl JFD02203 CS(=O)(=O)c1ccc(cc1)CC(=O)O JFD01525 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OC(=O)c3cccc(c3)C(F)(F)F KM04529 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OC(=O)c3ccccc3Cl KM04530 CC(C)(C)OC(=O)N[C@@H](CCC(=O)N)C(=O)OCc1ccc(cc1)CC(=O)O JFD01584 c1ccnc(c1)S(=O)(=O)CCS(=O)(=O)c2ccc(cc2)Cl KM00081 Cc1cc(n(n1)C(C)(C)C)NC(=O)c2ccccc2Cl KM00083 CN1c2ccccc2C(=O)/C(=C\Nc3ccc(cc3F)F)/S1(=O)=O KM01341 CN1c2ccccc2C(=O)/C(=C\Nc3ccccn3)/S1(=O)=O KM01344 CCOC(=O)N/N=C/c1ccc(cc1Cl)N(C)C DP00693 Cc1cc(n2c(n1)cc(n2)C(C)(C)C)C KM00322 c1cc(sc1)/C=C(\C#N)/C(=O)C2CC2 KM00326 CC1(CC(N(C(=O)N1C)c2ccc(cc2)Cl)(C)O)C JFD00495 Cc1ccc(cc1)S(=O)(=O)N(c2cc(nn2C)C)S(=O)(=O)c3ccc(cc3)C KM00017 Cc1c(c(n(n1)C)NC(=O)c2ccc(cc2Cl)Cl)Br KM00022 Cc1c(c(=O)n(n1C)c2ccccc2)CN3CCOCC3.Cl KM00023 Cc1c(csc1C(=O)Nc2ccc(cc2F)F)S(=O)(=O)c3ccc(cc3)Cl KM01366 CC(=O)Nc1nc(nc(n1)N2CCCCC2)N GK02639 C[C@@]12CCC(C1)C(C2NC(=O)c3ccc(cc3)C(C)(C)C)(C)C JFD01613 CC1(CC(=CC(=O)C1)Sc2nc3ccccc3o2)C JFD00597 c1cc(=O)n(c2c1CCCC2)CCC#N JFD00498 CC(=O)c1ccc(cc1)O[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00528 CCOC(=O)C(=CNc1c(csc1C(=O)OC)C)C(=O)OCC GK01281 Cc1csc(c1NC(=O)CC#N)C(=O)OC GK01283 CCC(C)NCCS(=O)(=O)c1ccc(cc1)Cl.Cl KM00329 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3ccccc3 DP00696 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3nccs3 DP00703 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3nncs3 DP00704 c1cc(oc1)/C=C(\C#N)/C(=O)C2CC2 KM00332 c1ccc(cc1)c2csc(n2)S/C(=C/C=C(C#N)C#N)/c3ccc(cc3)Cl JFD00586 c1cc(sc1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM01298 CN1c2ccccc2C(=O)/C(=C\Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)/S1(=O)=O KM01339 CN1c2ccccc2C(=O)/C(=C\Nc3ccc(c(c3)Cl)F)/S1(=O)=O KM01340 Cc1cc(c(cc1Cl)C)Sc2ncc(c(n2)C(F)(F)F)C(=O)Sc3cc(c(cc3C)Cl)C GK02607 CC(C)(C)c1ccc(cc1)C(=O)O/N=C/2\CCCc3c2c4ccccc4n3C JFD01617 COc1ccc(cc1)C(=O)NNC(=O)c2c(c(cs2)Br)OC GK02587 CCOc1ccc2c(c1)sc(n2)S/C=C/C(=O)c3ccccc3 JFD00590 Cc1ccc(cc1)n2c(nnn2)c3c[nH]c4ccccc4c3=O JFD00601 COc1c(csc1Cl)C(=O)O/N=C/c2c(cccc2Cl)F KM00602 COc1c(csc1Cl)C(=O)O/N=C/c2ccc(cc2Cl)Cl KM00603 CN(C)C(=O)Nc1csc(c1OC)Cl KM00612 Cc1ccc(cc1)S(=O)(=O)CC#N KM00613 c1cc(ccc1NC(=O)Nc2ccc(cc2)Br)Br JFD01635 Cc1c(csc1C(=O)O)S(=O)(=O)c2ccc(cc2)Cl KM01338 c1ccc(cc1)c2c(c(nc(c2C#N)Sc3ccc(cc3)Cl)N)C#N KM00566 CC(C)(C)OC(=O)N[C@@H](CCCCNC(=O)OCc1ccccc1)C(=O)OCc2ccc(cc2)CC(=O)O JFD01597 CC(C)(C)OC(=O)N[C@@H](CCSC)C(=O)OCc1ccc(cc1)CC(=O)O JFD01598 CCOC(=O)C(c1ccc(cc1)N(C)C(=O)c2ccc(cc2)C)(C(F)(F)F)O JFD02142 c1ccc(c(c1)C(=O)ON2C(=O)CCC2=O)Cl JFD02065 Cc1nnc(s1)SCc2ccccc2[N+](=O)[O-] JFD02066 c1ccc(cc1)OCC(=O)ON2C(=O)CCC2=O JFD02068 c1cc(c(c(c1)Cl)CN/C(=C(/C#N)\N)/C#N)F KM00327 c1cc(ncc1C(F)(F)F)N2CCC(CC2)C(=O)O KM07694 CCOC(=O)CC(=O)Nc1c(csc1C(=O)OC)C GK01285 Cc1csc2c1ncnc2SCC(=O)NNC(=O)c3cccc(c3)[N+](=O)[O-] GK02566 CC(C)(C)OC(=O)N[C@@H](CC(=O)N)C(=O)OCc1ccc(cc1)CC(=O)O JFD01556 C[C@@]12CCC(C1)C(C2NC(=O)C3CCCCC3)(C)C JFD01611 CC1=CCC23CC1C(=O)C=C2CC(CC3=O)(C)C JFD01539 c1cc(ccc1C(F)(F)F)N2CCCCC2=O JFD01541 C[C@@]12CCC(C1)C(C2NC(=O)c3c(cccc3Cl)Cl)(C)C JFD01614 CCOc1ccccc1/C=C(\C#N)/C(=O)N2CCOCC2 DP00501 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)N2CCCC2)Cl DP00518 c1cc(c(c(c1)Cl)/C=C(\C#N)/C(=O)N2CCOCC2)Cl DP00519 COC(=O)C(c1ccc(cc1)/N=C/c2ccccc2O)(C(F)(F)F)O JFD02163 Cc1csc(n1)[C@@H]([C@H]([C@@H]([C@@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00522 CO[C@H]1[C@H]2[C@@H](COC(O2)c3ccccc3)O[C@@H]([C@@H]1OC)OC JFD00525 c1ccc(c(c1)n2cc(c(=O)[nH]c2=O)C#N)Cl KM07699 c1ccc(cc1)NC(=O)Nc2cscc2S(=O)(=O)c3ccc(cc3)Cl KM01645 C[C@@]12CCC(C1)C(C2NC(=O)c3ccc(cc3Cl)Cl)(C)C JFD01612 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OS(=O)(=O)c3ccc(cc3F)F KM04579 c1cc(cc(c1)Cl)C(=O)CC#N KM01406 Cn1c(cc(n1)C(F)(F)F)OS(=O)(=O)c2ccc(cc2)C(F)(F)F GK01215 Cc1cc(nc(n1)C)N/C=C/2\C(=O)c3ccccc3N(S2(=O)=O)C KM01409 CCN(CCS(=O)(=O)c1ccc(cc1)Cl)C(=O)Nc2ccccc2 KM00106 CCOc1ccc2c(c1)sc(n2)S/C=C/C(=O)c3ccc(cc3)OC JFD00593 CCOc1ccc2c(c1)sc(n2)S/C=C/C(=O)c3ccc(cc3)Cl JFD00594 CCOc1ccc2c(c1)sc(n2)S/C=C/C(=O)c3ccc(cc3)Br JFD00595 c1cc(sc1)c2cc(n[nH]2)N KM00087 c1ccc2c(c1)nc(c(n2)S)S JFD01548 Cc1c2ccccc2ncc1c3nnnn3c4ccc(cc4)Br JFD00599 Cc1cc2[nH]c(cc(=O)n2n1)c3ccccc3 KM00095 Cc1c(c(n(n1)C(C)(C)C)NC(=O)c2ccccc2)C#N KM00098 Cc1c(c(n(n1)C)NC(=O)C(Cl)Cl)Br KM00100 c1cc(ccc1OC2CN(C2)C(=O)N3CC(C3)Oc4ccc(cc4)Cl)Cl JFD01634 Cc1cc(ccc1N2C(=O)c3ccccc3C2=O)C(C(=O)OC)(C(F)(F)F)O JFD02150 CCOC(=O)C(c1ccc(cc1)NC(=O)Nc2ccccc2)(C(F)(F)F)O JFD02152 CC(C)(C)c1cc2ncc(c(n2n1)N)S(=O)(=O)c3ccc(cc3)Cl KM00588 CCN(CCS(=O)(=O)c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)Cl KM00113 Cc1cc(nc(n1)C)N/C=C(\C(=O)C)/S(=O)(=O)c2ccc(cc2)Cl KM01435 CSc1c(c(n(n1)c2ccccc2)N)S(=O)(=O)c3ccc(cc3)Cl KM01440 CC(C)(C)n1c(c(c(n1)C2CC2)Br)NC(=O)c3ccccc3 KM00309 c1ccc(c(c1)N)Sc2ccc(cc2[N+](=O)[O-])Cl DSHS00740 c1ccc(c(c1)[N+](=O)[O-])SCc2nnc(n2c3cccc(c3)C(F)(F)F)S DSHS00876 Cn1c(cc(n1)C(F)(F)F)OS(=O)(=O)c2ccc(cc2)Cl GK01217 Cc1csc2c1ncnc2SCC(=O)NNC(=O)c3ccc(cc3)Cl GK02564 Cc1csc2c1ncnc2SCC(=O)NNC(=O)c3ccc(cc3)C(C)(C)C GK02565 c1ccc(c(c1)n2c(nnc2S)CSc3ccccc3[N+](=O)[O-])Cl DSHS00879 c1ccc2c(c1)nc(s2)SCC(=O)NCC(=O)N JFD02074 COc1c(csc1Br)C(=O)O KM00596 Cn1c2ccccc2c\3c1CCC/C3=N\OC(=O)c4cccc5c4cccc5 JFD01625 c1ccc2c(c1)cccc2CNCc3cccc4c3cccc4.Cl JFD01628 c1ccc2cc(ccc2c1)CNCc3cccc4c3cccc4 JFD01630 c1ccc2c(c1)c(ncn2)Nc3ccc(cc3)Cl.Cl DP00817 c1ccc(c(c1)C(F)(F)F)n2ccnc2 JFD01564 c1cc(ccc1S(=O)(=O)c2cscc2NC(=O)C(Cl)(Cl)Cl)Cl KM01752 c1c(c(=O)[nH]c(=O)[nH]1)C(F)(F)F JFD01566 C=C1[C@H]([C@@H]([C@H]([C@@H](O1)OC(=O)c2ccccc2)OC(=O)c3ccccc3)OC(=O)c4ccccc4)OC(=O)c5ccccc5 JFD02101 CCOC(=O)/C(=C/c1ccc(cc1)N(C)CCC#N)/C#N DP00647 CCOC(=O)c1ccc(cc1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00718 CC1(C(NC(S1)(C)C)C(=O)O)C.Cl JFD02104 CCOC(=O)C(c1ccc(cc1)NC(=O)Nc2cccc(c2)Cl)(C(F)(F)F)O JFD02172 c1cc2c(cc[nH]2)cc1Cl JFD02106 c1ccc(cc1)C(=O)NC(=S)Nc2cc(n[nH]2)c3cccs3 KM00432 COc1ccc(cc1OC)CC(=O)n2c(=O)ccc(=O)[nH]2 GK01228 CC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)CSc3ccc(cc3)Cl GK01233 Cc1csc(n1)c2c(c(c(s2)SC)C(=O)C)C KM04592 c1ccc(cc1)C(=O)NC(=S)Nc2c(c(n[nH]2)C3CC3)/N=N/c4ccc(cc4)F KM00446 CC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)CSCc3c(cccc3Cl)F GK01239 c1csc(c1)/C=N/NC(=S)N/N=C/c2sccc2 DP00720 C=CCNc1nc(c(s1)c2ccccc2)c3ccc(cc3)Cl.Br DP00545 COc1ccc(cc1)c2nc(c(s2)c3ccccc3)c4ccc(cc4)Cl DP00548 c1ccc(cc1)c2c(nc(s2)c3ccc(cc3)Cl)c4ccc(cc4)Cl DP00549 Cc1cc(n(n1)C(C)(C)C)NC(=O)c2ccc(cc2)Cl KM00090 Cc1c(c(n(n1)C(C)(C)C)NC(=O)c2ccc(cc2Cl)Cl)Br KM00092 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(c(c3)F)F)Cl DSHS00816 Cc1c(cnc(n1)N2CCCCC2)S(=O)(=O)c3ccc(cc3)Cl KM01330 CCOC(=O)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Cl DSHS00713 CO/N=C/1\CCCc2c1c(sc2C(=O)NNC(=O)c3ccc(cc3)Cl)SC KM04742 CN(c1ccc(cc1)C(C(=O)OC)(C(F)(F)F)O)C(=O)Nc2ccc(cc2)Cl JFD02175 COc1cc(ccc1NC(=O)Nc2ccc(cc2)Cl)C(C(=O)OC)(C(F)(F)F)O JFD02177 CCOC(=O)C(C(=O)OCC)NC(=O)C KM04753 Cc1csc2c1c(c(s2)/C=N/Cc3cccs3)C KM04756 CN(c1ccc(cc1)C(C(=O)OC)(C(F)(F)F)O)C(=O)Nc2cccc(c2)Cl JFD02178 CCOC(=O)C(c1ccc(c(c1)OC)NC(=O)Nc2ccc(cc2)Cl)(C(F)(F)F)O JFD02180 CCOC(=O)c1ccc(cc1)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C DSHS00702 CCOC(=O)/C=C(\C)/NC(=O)c1c(onc1c2c(cccc2Cl)Cl)C DSHS00703 Cc1nnc(s1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00705 c1ccc(c(c1)[N+](=O)[O-])SCC(=O)NNC(=S)NC2CC3CC2C=C3 DSHS00878 c1ccc(c(c1)/C=N/c2ccc(cc2)F)O DSHS00721 COc1cc2c(cc1OC)/C(=C\C#N)/NCC2 KM00101 CCCC(=O)c1ccc(cc1)O[C@H]2[C@@H]([C@H]([C@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00529 c1ccc2c(c1)C3=C(C2=O)C(SC(=O)N3)c4ccc(cc4)[N+](=O)[O-] JFD00450 Cc1cc(nc(n1)N/C=C(\C(=O)C)/S(=O)(=O)c2ccc(cc2)Cl)C KM01432 CCOC(=O)NC(=O)/C(=C/Nc1ccc(cc1)OC(F)(F)F)/C#N KM07679 Cc1c2c(=O)[nH]c(cn2cn1)c3ccc(cc3Cl)Cl KM07686 COC(=O)C(c1ccc(cc1)NC(=O)Nc2ccc3ccccc3c2)(C(F)(F)F)O JFD02156 CCOC(=O)NC(=O)/C(=C/Nc1ccc(cc1F)F)/C#N KM07689 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00742 Cn1c(cc(n1)C(F)(F)F)OS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01220 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2OC)C(C(=O)OC)(C(F)(F)F)O JFD02168 CCOC(=O)C(c1ccc(cc1)NC(=O)Nc2ccc3ccccc3c2)(C(F)(F)F)O JFD02131 Cc1c(c(n(n1)c2ccccc2)NC(=O)C(Cl)Cl)Cl KM00167 c1cc(cc(c1)Oc2c(c(ncn2)Oc3cccc(c3)C(F)(F)F)[N+](=O)[O-])C(F)(F)F KM07742 CSc1c(cn(n1)c2ccccc2)/C(=N/O)/N KM07757 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCC(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F KM07759 c1cc(ccc1S(=O)(=O)CCSCCO)Cl KM01782 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(on3)c4cccs4 KM07774 CCOC(=O)C1CN(C(=O)C1=O)C2CCCCC2 KM00129 c1cc(oc1)/C=C\2/C(=O)N3C(S2)C(=C(C(=C3N)C#N)c4ccco4)C#N KM00535 C#CC1(CCCCC1)NS(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccccn3 DSHS00903 Cc1c(c(c(c(c1C)C)CSCC(=O)NNS(=O)(=O)c2ccc(cc2)Cl)C)C DSHS00857 CCC(C)COC(=O)/C=C/c1ccc(cc1)/N=C/c2ccc(cc2)OC JFD01516 CC(=O)c1ccc(cc1)S(=O)(=O)C JFD01520 CCN(CCS(=O)(=O)c1ccc(cc1)C)C(=O)Nc2ccc(cc2)Cl KM00248 CCOC(=O)CSc1ccc(cc1[N+](=O)[O-])S(=O)(=O)N DSHS00900 C#CC1(CCCCC1)NS(=O)(=O)c2ccc(c(c2)[N+](=O)[O-])Sc3ccccc3 DSHS00902 c1ccc(cc1)S(=O)(=O)c2cscc2NC(=O)c3ccccc3Cl KM01791 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])C(=O)N3CCC=CC3.Cl DSHS00931 CSc1c(cn(n1)c2ccccc2)/C(=N/OC(=O)c3ccc(cc3Cl)Cl)/N KM07799 Cc1ccc(cc1)S(=O)(=O)OC2=C(CSC2)C(=O)OC KM04813 CSc1c(cn(n1)c2ccccc2)/C(=N/OC(=O)c3ccc(cc3)C(F)(F)F)/N KM07800 CC1(C2CCC13CS(=O)(=O)[N@@]4C3(C2)O4)C JFD01494 COc1ccc2cc(c(=O)oc2c1)C(=O)c3cc4ccc(cc4oc3=O)OC JFD01497 c1cc(ccc1C2(CCCCC2)C#N)Cl JFD01501 CC(C)(C)Sc1ccc(cc1[N+](=O)[O-])S(=O)(=O)NC2(CCCCC2)C#C DSHS00925 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C(C(=O)OC)(C(F)(F)F)O JFD02183 COC(=O)C(c1ccc(cc1)NC(=O)Nc2ccc(cc2)Cl)(C(F)(F)F)O JFD02171 CC1(Cc2c(cnc(n2)SCC(=O)Nc3ccc(cc3F)F)C(=O)C1)C KM04731 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl KM04517 CCCCCCCCCCOc1ccc(cc1)C(=O)C JFD01506 c1ccc(cc1)C(=O)c2ccccc2C(=O)c3ccccc3 JFD01507 Cc1ccc(cc1)NC(=O)c2ccccc2NC(=O)c3ccccc3 DP00713 CC1(CC(=O)C(=CNc2ccc(c(c2)Cl)F)C(=O)C1)C KM01520 Cc1ccc(cc1)c2c(c(n[nH]2)S(=O)(=O)C)C#N KM01525 c1ccnc(c1)SCc2cccc(c2)/C(=N/OC(=O)c3ccc(cc3)Cl)/N KM01526 CNC(=S)NNC(=O)c1c2c(c(s1)SC)C=CCC2 KM04762 CCOC(=O)c1c(c(sc1NC(=O)c2cc(c(s2)SC)S(=O)(=O)C(C)C)C)C KM04807 COC(=O)c1csc2c1[nH]c(=O)cc2C(F)(F)F GK02676 Cc1csc2c1ncnc2N3CCN(CC3)S(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F GK02679 Cc1csc2c1ncnc2N3CCN(CC3)C(=S)Nc4ccc(cc4)C(F)(F)F GK02688 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2C)C(C(=O)OCC)(C(F)(F)F)O JFD02185 c1cc(cc(c1)n2cc(c(=O)[nH]c2=O)C#N)C(F)(F)F KM07693 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2C)C(C(=O)OC)(C(F)(F)F)O JFD02187 c1c(c(=O)[nH]c(=O)n1C2CC2)C#N KM07678 Cc1ccc(cc1)S(=O)(=O)NC2[C@@]3(CCC(C3)C2(C)C)C JFD01608 COC(=O)Cn1nc(nn1)N2CCOCC2 GK02621 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3c4c(c(cs4)C)ncn3 GK02671 c1cc(sc1)/C=c\2/c(=O)n3c(=C(C(C(=C3N)C#N)c4cccs4)C#N)s2 KM00532 C[C@@]12CCC(C1)C(C2NC(=O)c3cccc(c3)C(F)(F)F)(C)C JFD01605 c1ccc(c(c1)c2nc(no2)CS(=O)(=O)c3ccccn3)Cl KM01283 c1ccc(cc1)c2cc3nnc(c(n3n2)N)C(=O)N KM00230 c1cc(sc1)/C=N/C(=C(\C#N)/N)/C#N KM00235 CN(C)n1cccc1/C=N/C(=C(/C#N)\N)/C#N KM04619 c1c(ccc(c1)Cl)/C=N/NC(=S)N/N=C/c2ccc(cc2)Cl DP00750 c1ccc(cc1)/C/2=N/c3ccccc3NC(=O)c4c2cccc4 DP00759 c1cc(sc1)S(=O)(=O)/C(=C/Nc2ccc(cc2F)F)/C#N KM01307 CC(C)(C)CN/C(=C(/C#N)\N=C\c1ccccc1Cl)/C#N KM00231 CSc1c(c(c(s1)C(=O)N2CCCCC2)c3cccs3)C#N KM01702 CSc1c(c(c(s1)C(=O)N2CCOCC2)c3cccs3)C#N KM01703 CC(C)(C)CN/C(=C(/C#N)\N)/C#N KM00227 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Oc3ccc(cc3)Cl KM04566 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl KM04569 c1ccc(c(c1)C(=O)OCCSCCS(=O)(=O)c2ccc(cc2)Cl)Cl KM01819 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCc4c(cccc4Cl)Cl KM04547 CC1(Cc2c(c(sc2C(=O)OC)Sc3ccc(cn3)C(F)(F)F)C(=O)C1)C KM04768 c1cc(oc1)C2C(=C(OC(=C2C#N)N)C3CC3)C#N KM00374 c1cc(ccc1S(=O)(=O)CCSCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl KM01527 c1ccc(cc1)/C=N/C(=C(/C#N)\NCc2c(cccc2Cl)F)/C#N KM00378 CCN(CCS(=O)(=O)c1ccc(cc1)C)S(=O)(=O)c2ccccc2 KM00241 c1ccc2c(c1)nc(s2)Sc3ccc(cc3[N+](=O)[O-])S(=O)(=O)N DSHS00895 c1cc(ccc1N(Cc2ccc3c(c2)OCO3)C(=O)c4ccc(c(c4)[N+](=O)[O-])Sc5ccc(cc5)Cl)F DSHS00941 c1cc(cc(c1)Cl)CN/C(=C(/C#N)\N=C\c2ccco2)/C#N KM00282 Cc1cc(nc2c1c(nn2C)C)O KM00293 COc1c(csc1C(=O)Nc2cccc(c2)C(F)(F)F)Br GK02592 c1cc(ccc1S(=O)(=O)CCSCCOC(=O)C(Cl)(Cl)Cl)Cl KM01820 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCc4ccc(cc4)Cl KM04541 c1ccc(c(c1)CSc2ccc(cc2)Cl)OCC(=O)N/N=C/c3ccc(cc3)C(F)(F)F KM04786 Cc1c2c(c3ccccc3n1)C(=O)NC2=O KM00253 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl KM04573 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCC(=O)Nc4cccc(c4)C(F)(F)F KM04574 CC1C(C1C(=O)NN)C(=O)NN JFD01639 CCOC(=O)C(C(F)(F)F)(Nc1cc(on1)C)NC(=O)c2ccccc2Cl JFD02211 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl)C(F)(F)F KM04543 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)OCc2ccc(cc2)CC(=O)O JFD01599 C[C@@]12CCC(C1)C(C2NS(=O)(=O)c3ccc(cc3)Cl)(C)C JFD01610 CSc1nc2cc(nn2c(n1)N)c3ccc(cc3)Cl KM01572 c1ccc(c(c1)CSc2ccc(cc2)Cl)OCC(=O)N/N=C\c3ccc(cc3)Cl KM04787 CCOC(=O)C(=CNc1cccc(c1)c2c(cn(n2)C)Br)C(=O)OCC KM04788 CSc1nc2cc(nn2c(n1)N)c3cccs3 KM01577 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC2[C@@]3(CCC(C3)C2(C)C)C JFD01606 CNC(=O)Oc1ccc(cc1)NC2=C(CSC2)C(=O)OC KM04571 c1ccc(cc1)NC(=O)OCCSCCS(=O)(=O)c2ccc(cc2)Cl KM01830 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)Oc3cccc(c3)[N+](=O)[O-])C(F)(F)F KM04544 CC(C)(C)OC(=O)N[C@@H](COCc1ccccc1)C(=O)OCc2ccc(cc2)CC(=O)O.C1CCC(CC1)NC2CCCCC2 JFD01601 Cn1c2ccccc2c\3c1CCC/C3=N\OC(=O)C4CCCCC4 JFD01621 c1ccc2c(c1)c\3c([nH]2)CCC/C3=N\OC(=O)c4cccc(c4)C(F)(F)F JFD01624 CCc1cc(c(s1)NC(=O)c2ccccc2C(=O)O)C(=O)OCC GK02660 CSc1c(c(nn1C(=O)c2ccccc2Cl)c3ccc(cc3)Cl)C#N KM01284 CSc1c(c(nn1C(=O)c2cccs2)c3ccc(cc3)Cl)C#N KM01285 c1ccc2c(c1)cccc2CNCc3cccc4c3cccc4 JFD01629 Cn1c(nnc1SCC(=O)c2ccccc2)CSc3cccs3 KM04848 C[C@@]12CCC(C1)C(C2NS(=O)(=O)c3ccc(cc3)F)(C)C JFD01607 CN(C)n1cccc1/C=C(\C#N)/C(=O)c2ccccc2Cl KM04614 CN(C)n1cccc1/C=C(\C#N)/C(=O)c2ccco2 KM04615 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)CSc3cccs3 KM04849 CCOC(=O)/C(=C\Nc1cc(cc(c1)Cl)Cl)/S(=O)(=O)c2ccc(cc2)Cl KM01312 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cc(c(cc3Cl)Cl)Cl DSHS00811 c1cc(cc(c1)C#N)CS(=O)(=O)c2ccc(cc2)Cl KM00589 c1ccc(cc1)c2cc3ncc(c(n3n2)N)S(=O)(=O)c4ccc(cc4)Cl KM00583 CN(C)n1cccc1/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM04525 Cn1c2ccccc2c\3c1CCC/C3=N\OC(=O)c4ccc(cc4)Cl JFD01623 CN(C)n1cccc1/C=C(\C#N)/S(=O)(=O)c2cccc(c2)Cl KM04610 c1ccc(c(c1)OCC(=O)NNC(=O)c2cccc(c2)C(F)(F)F)SCc3ccc(cc3)Cl KM04794 CCOC(=O)C(C(F)(F)F)(Nc1ncccn1)NC(=O)c2ccccc2Cl JFD02206 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)CC3C(=O)Nc4ccccc4S3 KM07501 Cn1c(nnc1SCC(=O)c2ccccc2)CC3C(=O)Nc4ccccc4S3 KM07502 c1cc(c(cc1n2c(=O)ccs2)Cl)F KM04549 c1cc(c(c(c1)Cl)F)n2c(=O)ccs2 KM04550 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC)CC3C(=O)Nc4ccccc4S3 KM07503 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)CC3C(=O)Nc4ccccc4S3 KM07504 CS(=O)(=O)c1cccs1 KM01427 COc1ccc(cc1OC)CC(=O)n2c(=O)c3ccccc3c(=O)[nH]2 GK01222 CS/C(=C(/C#N)\C(=O)C1CC1)/NCc2cccnc2 KM01630 CN(C)n1cccc1/C=C(\C#N)/S(=O)(=O)c2ccccn2 KM04611 CCOC(=O)c1c2c(c(s1)N/N=C/c3ccccc3Cl)C(=O)CC(C2)(C)C KM04791 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C)NC(=O)c2ccccc2Cl JFD02198 Cn1c(nnc1SCc2ccc(cc2)Cl)CC3C(=O)Nc4ccccc4S3 KM07499 c1ccnc(c1)S(=O)(=O)/C(=N\O)/C#N KM01405 CN1c2ccccc2C(=O)/C(=C\Nc3ncccn3)/S1(=O)=O KM01410 COc1ccc(cc1)C(=O)C(=C(SC)SC)C#N KM01418 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(C)(C)C KM07847 CS(=NS(=O)(=O)c1cc(cs1)S(=O)(=O)c2ccccc2)(=O)c3ccccc3 KM04839 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OC(=O)Nc3ccc(cc3)OC(F)(F)F KM04560 c1cc(c(c(c1)F)/C(=N/OC(=O)/C=C/c2cc(sc2)[N+](=O)[O-])/N)F GK01191 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl KM04556 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OC(=O)Nc3cccc(c3)Cl KM04570 Cc1cc(n(n1)C(C)(C)C)NC(=O)c2ccc(cc2Cl)Cl KM00086 c1cc(sc1)C(=O)Nc2ccc(cc2)Cl KM04585 Cc1c(c(sc1c2nc(cs2)C(C)(C)C)SC)C(=O)C KM04587 CCOC(=O)c1csc(n1)c2c(c(c(s2)SC)C(=O)C)C KM04588 Cn1c(nnc1SCC(=O)c2ccccc2)CSc3cc(nc4c3cccc4)C(F)(F)F KM07796 c1ccc(c(c1)C(=O)/C(=N/Nc2ccccc2Cl)/C#N)OC(F)(F)F KM04877 Cn1c2ccccc2c\3c1CCC/C3=N\OC(=O)c4ccc(cc4Cl)Cl JFD01619 CCOC(=O)C(c1ccc(cc1)NC(C(=O)OCC)(C(F)(F)F)NC(=O)C)(C(F)(F)F)O JFD02139 CCOC(=O)C(c1ccc(cc1)NC(=O)c2ccc(cc2)C)(C(F)(F)F)O JFD02141 Cc1cc(n(n1)C(C)(C)C)NC(=O)c2ccccc2F KM00088 Cc1ccc(cc1)C(=O)N(C)c2ccc(cc2)C(C(=O)OC)(C(F)(F)F)O JFD02144 COC(=O)C(c1ccc(cc1)NC(=O)Oc2ccccc2)(C(F)(F)F)O JFD02146 c1cc(sc1)c2cc3ncc(c(n3n2)N)S(=O)(=O)c4ccc(cc4)Cl KM00585 CC(=O)CSc1nnc(n1C)CSc2cc(nc3c2cccc3)C(F)(F)F KM07797 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)N3CCCC3 KM04802 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)N3CCCCC3 KM04803 Cc1c(csc1S(=O)(=O)N/N=C/c2c(cccc2Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl KM01381 Cc1csc(c1n2cccc2)C(=O)OC GK01274 CCOC(=O)C(C(F)(F)F)(Nc1cccc(n1)C)NC(=O)c2ccccc2Cl JFD02208 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cn1)C)NC(=O)c2ccccc2Cl JFD02209 c1cc(cc(c1)Nc2c(c(ncn2)Nc3cccc(c3)C(F)(F)F)[N+](=O)[O-])C(F)(F)F KM07743 CCN(CCS(=O)(=O)c1ccc(cc1)Cl)S(=O)(=O)c2ccc(cc2)C KM00114 c1ccc(cc1)SCCS(=O)(=O)c2ccccc2 KM00118 Cc1ccc(cc1)SCCS(=O)(=O)c2ccccc2 KM00119 c1cc(cc(c1)[N+](=O)[O-])C(=O)ON=C2CCC3(CC2)OCCO3 JFD01616 Cn1c2ccccc2c\3c1CCC/C3=N\OC(=O)c4c(cccc4Cl)Cl JFD01620 CC(C)(C)c1ccc(cc1)C(=O)O/N=C/2\CCCc3c2c4ccccc4[nH]3 JFD01622 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)OCCN(C)C KM07508 COc1cscc1C(=O)OC KM00444 CCOC(=O)/C(=C\Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/S(=O)(=O)c2ccc(cc2)Cl KM01388 c1cc(ccc1F)S(=O)(=O)CC#N KM01392 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)F)NC(=O)c2ccccc2Cl JFD02199 c1ccc(cc1)n2c(=O)cc([nH]2)C(F)(F)F KM00122 Cn1cc(c(=O)n(c1=O)Cc2ccccc2)/C(=N/O)/N KM07720 c1ccc(c(c1)n2cc(c(=O)n(c2=O)Cc3ccc(cc3)Cl)C#N)Cl KM07719 Cc1ccc(cc1)NC(=O)c2c(ccs2)Cl GK01325 CS(=O)(=O)c1ccc(cc1)Cl KM00170 c1ccc(c(c1)NS(=O)(=O)c2cccc(c2)C(F)(F)F)Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00769 c1ccc(c(c1)NS(=O)(=O)c2ccccc2[N+](=O)[O-])Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00771 c1ccc(c(c1)C(=O)N(CCC#N)C2CCCCC2)Cl DSHS00779 CC(C)(C#C)NS(=O)(=O)c1ccc(cc1)F DSHS00786 CC(C)(C#C)NS(=O)(=O)c1cc(c(cc1Cl)Cl)Cl DSHS00788 c1ccc(cc1)NC(=O)Nc2cc(nn2c3ccccc3)C4CC4 KM00200 c1ccc(cc1)C(CS(=O)(=O)c2ccc(cc2)Cl)N3CCOCC3 KM00201 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C(F)(F)F)NC(=O)c2ccccc2Cl JFD02202 c1ccc(c(c1)C(=O)NNC(=O)COc2ccccc2SCc3ccc(cc3)Cl)Cl KM04793 Cn1c(nnc1SCc2ccccc2)CSc3cc(nc4c3cccc4)C(F)(F)F KM07730 Cn1c(nnc1SCc2c(cccc2Cl)Cl)CSc3cc(nc4c3cccc4)C(F)(F)F KM07732 c1ccc(cc1)C2=c3c(=C(S2(=O)=O)c4ccccc4)oc(=O)o3 JFD01555 c1cc(c(c(c1)Cl)Cn2c(=O)c(cn(c2=O)c3ccc(cc3)Cl)C#N)Cl KM07723 c1ccc(c(c1)OCC(=O)NNC(=O)c2ccc(cc2)Cl)SCc3ccc(cc3)Cl KM04789 c1cc(oc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4cccs4 KM00402 CCOC(=O)c1c2c(c(s1)N/N=C/c3cccs3)C(=O)CC(C2)(C)C KM04792 COc1ccc(cc1)OS(=O)(=O)c2ccc(s2)c3ccccn3 KM04567 c1cc(ccc1S(=O)(=O)/C(=C/N2CCOCC2)/C#N)Cl KM00450 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C(C(=O)OC)(C(F)(F)F)O JFD02165 CCOC(=O)C(c1ccc(cc1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccc(cc2)C)(C(F)(F)F)O JFD02166 CCOC(=O)c1c(c2cccnc2s1)NC(=O)C(Cl)Cl GK01200 CN(C)/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl KM00459 CCOC(=O)c1c2c(c(s1)N3CCCCC3)C(=O)CC(C2)(C)C KM04736 CC(C)(C)OC(=O)N[C@@H](CC(=O)OC1CCCCC1)C(=O)OCc2ccc(cc2)CC(=O)O JFD01557 c1ccc(cc1)S(=O)(=O)CCSc2ccc(cc2)Cl KM00120 c1cc(sc1)Sc2c(c(ncn2)Sc3cccs3)[N+](=O)[O-] KM07711 CCOC(=O)NC(=O)c1cn(c(=O)n(c1=O)C)Cc2cccs2 KM07716 Cc1ccc(n1c2c(csc2C(=O)OC)C)C GK01278 Cc1csc(c1n2cccc2)C(=O)NN GK01282 c1cc(oc1)c2cc3[nH]c4c(c(=O)n3n2)CSC4 KM00483 Cc1cc2nc3c(c(n2n1)O)CSC3 KM00484 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)C(C(=O)OC)(C(F)(F)F)O JFD02143 CCOC(=O)C(c1ccc(c(c1)OC)NC(=O)Nc2cccc(c2)Cl)(C(F)(F)F)O JFD02182 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Cc2ccco2 KM07672 COc1cc(ccc1NC(=O)c2ccc(c(c2)Cl)Cl)C(C(=O)OC)(C(F)(F)F)O JFD02148 CSC(=C(C#N)C(=O)c1cccc(c1)Cl)SC KM01421 Cc1nc(nc(n1)OC)N/C=C/2\C(=O)c3ccccc3N(S2(=O)=O)C KM01423 c1cc(oc1)Cn2cc(c(=O)[nH]c2=O)C#N KM07677 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2OC)C(C(=O)OC)(C(F)(F)F)O JFD02186 c1ccnc(c1)c2ccc(s2)C#CCOC(=O)Nc3ccc(cc3)Cl KM07842 c1ccnc(c1)c2ccc(s2)C#CCOC(=O)Nc3cccc(c3)Cl KM07843 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)Nc2ccsc2C(=O)OC KM04806 Cc1c(c(n(n1)c2ccccc2)NC(=O)c3ccc(cc3Cl)Cl)Cl KM00175 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)/C(=N/OC(=O)c3ccccc3Cl)/N KM07750 CN(CCC#N)c1ccc(cc1)C=C(C#N)C#N DP00648 CC(C)(C)CN/C(=C(/C#N)\NCc1cccc(c1)Cl)/C#N KM00313 CC(C)(C#C)NC(=O)Nc1ccccc1 DP00745 COc1ccc(cc1)n2cc(c(=O)[nH]c2=O)C#N KM07690 c1cc(c(cc1F)F)n2cc(c(=O)[nH]c2=O)C#N KM07692 CC(=O)/C(=C\Nc1ncccn1)/S(=O)(=O)c2ccc(cc2)Cl KM01434 Cc1ccc(c(c1)C)Nc2c3ccccc3ncn2.Cl DP00802 Cc1cc(n(n1)c2ccccc2)NC(=O)C(Cl)(Cl)Cl KM00141 c1ccc(cc1)S(=O)(=O)CC#N KM00475 Cc1ccc(cc1)S(=O)(=O)Nc2c(c(n[nH]2)c3ccc(cc3)C(C)(C)C)Br KM00525 Cc1ccc(cc1)S(=O)(=O)CCSc2ccc(cc2)Cl KM00157 Cc1c(sc2c1C(=C(S(=O)(=O)N2C)C(=O)Nc3cccc(c3)Cl)O)C KM04705 CC(C)(C)c1nnc(o1)c2cccc(c2)NS(=O)(=O)c3ccc(s3)c4ccno4 SEW06646 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)NC(=S)Nc2ccccc2Cl KM04818 c1ccc(cc1)c2c(c([nH]n2)NC(=O)c3ccc(cc3)Cl)Br KM00364 c1cc(cc(c1)C(F)(F)F)C(=O)OC2=C(C(=O)CCC2)Cl KM05004 CC1(COC(=N1)c2ccc(c(c2)OC)OC)C KM07779 COC(=O)c1c(c(cs1)S(=O)(=O)c2ccccc2)N KM01698 c1ccc(c(c1)C(F)(F)F)NC(=S)N KM00543 CC1(Cc2c(cnc(n2)SC)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/C1)C KM04775 CC(C)(C)C(=O)/C(=C/Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C#N KM01772 CC1(Cc2c(sc(c2C(=O)C1)SCC(=O)OC)C#N)C KM04819 CC(C)(C)S(=O)(=O)/C(=C/N1CCOCC1)/C#N KM01867 CC(C)C[C@@H](C(=O)O)NC(=O)c1cccnc1SC KM01873 c1cc(ccc1S(=O)(=O)c2cnc(nc2N)N3CCOCC3)Cl KM00655 CC1(Cc2c(sc(c2C(=O)C1)SCC(=O)NN)C#N)C KM04826 COC(=O)C1=C(CSC1)Sc2ccc(cc2)Cl KM04829 CSCCC(C(=O)O)NC(=O)c1cccnc1SC KM01874 CCOC(=O)CNC(=O)C(CCSC)NC(=O)c1cccnc1SC KM01878 CC(C)(C)S(=O)(=O)/C(=C/N/N=C/c1c(cccc1Cl)Cl)/C#N KM01888 CC(C)(C)c1ccc(cc1)c2cc([nH]n2)NC(=O)c3ccc(cc3)Cl KM00512 CN1c2ccccc2C(=O)/C(=N\Nc3ccccc3C(F)(F)F)/S1(=O)=O KM00513 CC(=O)c1ccc(s1)C#CC(C)(C)O KM07839 Cn1c(nnc1S)c2c3c(c(s2)SC)C=CCC3 KM04757 CC1(CC(=O)C(=CNc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)C1)C KM01514 c1cc(oc1)CNc2c(c(ncn2)NCc3ccco3)[N+](=O)[O-] KM07745 Cn1c(nnc1SCC(=O)Nc2cccc(c2)Cl)CSc3cc(nc4c3cccc4)C(F)(F)F KM07748 Cc1cc(n2c(n1)c(cn2)C#N)C KM00656 CC(=O)Nc1ccc(cc1)C2SCCS2 KM00658 CSc1c(cn(n1)c2ccccc2)c3nc(on3)c4cccs4 KM07822 c1cc(ccc1S(=O)(=O)c2cnc(nc2N)N3CCCCC3)Cl KM00660 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(on3)c4ccccc4Cl KM07751 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)/C(=N/O)/N KM07752 Cc1nc(nc(n1)N(CCS(=O)(=O)c2ccccc2)CCS(=O)(=O)c3ccccc3)C KM00664 CC(=O)Oc1ccc(cc1C(=O)O)Cl KM04902 c1cc(ccc1Sc2cscc2C(=O)O)Cl KM04905 CC1(Cc2c(sc(c2C(=O)C1)NCc3ccco3)C#N)C KM04824 Cc1csc2c1ncnc2N3CCN(CC3)C(=S)Nc4ccc(cc4F)F GK02690 c1ccc2cc(ccc2c1)S(=O)(=O)/C(=C/Nc3ccccc3Cl)/C#N KM01272 c1cc(c(c(c1)Cl)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)Cl KM00517 Cc1ccc(cc1)S(=O)(=O)NC(=O)NN2CCCCCC2 JFD01580 COc1cscc1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM01769 CSc1c(cn(n1)c2ccccc2)c3nc(on3)c4ccc(cc4Cl)Cl KM07823 c1cc(ccc1S(=O)(=O)/C(=C/N2CCCCC2)/C#N)Cl KM00456 c1ccnc(c1)c2ccc(s2)C#CCOC(=O)c3ccc(cc3)Cl KM07825 CC(C)(C)C(=O)/C(=C/Nc1cc(cc(c1)Cl)Cl)/C#N KM01773 Cc1nc(c(c(n1)SC)C#N)C2CC2 KM01777 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCCNC(=O)Nc3ccc(cc3)Cl KM07826 CC(C)c1ccc(cc1)NC(=O)CSc2ncc3c(n2)CC(CC3=O)(C)C KM04732 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)Oc3ccc(cc3)Cl)C(F)(F)F KM04526 CNC(=S)NNC(=O)c1ccsc1 KM04528 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)C(=S)N KM07783 CN1c2ccccc2C(=O)/C(=N\Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)/S1(=O)=O KM00524 c1ccc(cc1)Sc2ccc(s2)c3ccccn3 KM04831 c1ccnc(c1)S(=O)(=O)C/C(=N/OC(=O)c2cccs2)/N KM01278 CSc1c(cn(n1)c2ccccc2)C#N KM07728 CC(C)(C)n1c(c(c(n1)C2CC2)Br)NC(=O)c3ccccc3Cl KM00303 COC(=O)c1c(ccs1)NS(=O)(=O)C KM03307 Cc1cc(n2c(n1)c(cn2)/C(=N/OC(=O)Nc3ccccc3)/N)C KM00754 Cc1ccc(cc1)C2C(=C(OC(=C2C#N)N)C3CC3)C#N KM00341 c1cc(ccc1N/N=C(\C#N)/C(=O)C2CC2)Cl KM00369 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)Cl KM00370 Cc1csc(c1Cl)C(=O)NN GK01304 Cc1c(c(n(n1)Cc2nnc(o2)S)C)Br KM04636 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCC(=O)Nc4ccc(cc4Cl)Cl KM04575 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)Oc3cccc(c3)C(F)(F)F KM04519 CCCCNC(=O)OCCSCCS(=O)(=O)c1ccc(cc1)Cl KM01839 c1ccnc(c1)N/C=C(\C#N)/C(=O)c2ccc(cc2)OC(F)(F)F KM04859 COc1c(csc1S(=O)(=O)Nc2ccc(cc2)Cl)C(=O)OC KM07784 Cc1c(cnc2n1nc(c2)c3ccccc3)C(=O)C KM01798 Cc1cc(no1)N/C=C(\C#N)/C(=O)c2cccs2 KM01806 COc1ccc(cc1)C2C(=C(OC(=C2C#N)N)C3CC3)C#N KM00344 CC(C)(C)C(=O)Nc1c(c(nn1c2ccccc2)C3CC3)Cl KM00345 CCOC(=O)c1ccccc1N/C=C/c2nnnn2c3ccc(cc3)C JFD00609 c1ccc(cc1)n2c(nnn2)/C=C/Nc3ccccc3[N+](=O)[O-] JFD00611 c1ccc(cc1)c2cc([nH]n2)NC(=S)NC(=O)c3ccccc3 KM00431 CCOC(=O)c1c2c(c(s1)N3CCCC3)C(=O)CC(C2)(C)C KM04737 Cc1ccc(cc1)C(=O)CC#N KM01491 CCOC(=O)c1cnc2cc(nn2c1C)C KM01494 c1cc(ccc1N/C=C(\C#N)/C(=O)C2CC2)F KM01495 c1cc(ccc1S(=O)(=O)CCSCC(=O)N2CCCCC2)Cl KM01552 CSc1nccc(n1)c2ccsc2 KM04554 c1cc(sc1)c2c(c(nc(c2C#N)Sc3ccc(cc3)Cl)N)C#N KM00567 COc1ccc(cc1)c2c(c(nc(c2C#N)Sc3ccc(cc3)Cl)N)C#N KM00571 c1cc(ccc1S(=O)(=O)CCS(=O)(=O)c2c(c(cc(c2F)F)F)F)Cl KM00573 Cc1cc(no1)N/C=C(/C#N)\C(=O)C2CC2 KM01807 c1cc(ccc1OC(F)(F)F)S(=O)(=O)CC#N KM04653 CCOC(=O)C(=CNc1cc(nn1C)C2CC2)C(=O)OCC KM00433 c1cc(ccc1S(=O)(=O)/C(=C/N2CCCC2)/C#N)Cl KM00457 CC(C)S(=O)(=O)c1cc(sc1)NC(=O)Nc2ccc(cc2)C(F)(F)F KM03309 c1ccc(cc1)c2c(c([nH]n2)NC(=O)c3ccccc3Cl)Br KM00363 CC([C@@H](C(=O)OCc1ccc(cc1)CC(=O)O)NC(=O)OC(C)(C)C)OCc2ccccc2.C1CCC(CC1)NC2CCCCC2 JFD01602 CCOC(=O)/C(=C\Nc1ccc(cc1)F)/S(=O)(=O)c2ccc(cc2)Cl KM01309 CCOC(=O)/C(=C\Nc1ccc(c(c1)Cl)F)/S(=O)(=O)c2ccc(cc2)Cl KM01311 c1cc(ccc1C(=O)/C(=C/Nc2ccc(cc2)Cl)/C#N)OC(F)(F)F KM04856 CC1(Cc2c(cnc(n2)SCCS(=O)(=O)c3ccc(cc3)Cl)C(=O)C1)C KM04782 c1ccc(c(c1)CSc2ccc(cc2)Cl)OCC(=O)N/N=C\c3cccs3 KM04785 c1cc(ccc1C(=O)CC#N)OC(F)(F)F KM04838 c1cc(ccc1S(=O)(=O)/C(=N/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl KM01532 Cc1c(c(n(n1)Cc2ccc(o2)C(=O)Sc3ccc(cn3)C(F)(F)F)C)Br KM07522 Cc1c(c(n(n1)Cc2ccc(o2)C(=O)Oc3ccc(cc3)Cl)C)Br KM07523 CC(C)(C)c1ccc(cc1)C(=O)/C(=C/c2ccc3c(c2)OCO3)/C#N KM00437 c1cc(cnc1)N/C=C(\C#N)/C(=O)c2ccc(cc2)OC(F)(F)F KM04857 CC(=O)Nc1c(c(nn1c2ccccc2)C3CC3)Br KM00276 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OS(=O)(=O)c3ccccc3Cl KM04580 c1ccc(c(c1)C(F)(F)F)Oc2cc(nc3c2cccc3Br)C(F)(F)F KM07495 CS(=NS(=O)(=O)c1cc(cs1)S(=O)(=O)c2ccccc2)(=O)c3ccc(cc3)Cl KM04840 Cc1c(cnc(n1)N2CCCC2)S(=O)(=O)c3ccc(cc3)Cl KM01327 c1ccc(cc1)c2cc(n(n2)c3ccccc3)NC(=O)c4ccccc4Cl KM00205 Cn1c(nnc1SCC(=O)Nc2ccc(cc2F)F)CSc3cccs3 KM04672 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C)CSc3cccs3 KM04673 Cc1c(sc2c1C(=C(S(=O)(=O)N2C)C(=O)Nc3ccc(cc3)OC(F)(F)F)O)C KM04706 CC(C)(C)c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4cccs4 KM00395 Cn1c(nnc1SCc2c(cccc2Cl)Cl)CSc3cccs3 KM04623 Cn1c(nnc1SCc2ccc(cc2)OC)CSc3cccs3 KM04624 Cn1c(nnc1SCc2ccccc2)CSc3cccs3 KM04625 Cc1csc(n1)c2c(c(c(s2)SC)c3ccn(n3)S(=O)(=O)C)C KM05007 c1cc(ccc1OC(F)(F)F)S(=O)(=O)CCN2CCOCC2 KM05011 c1ccc(cc1)Nc2c3ccccc3ncn2.Cl DP00797 C[C@@]12CCC(C1)C(C2NC(=O)c3ccco3)(C)C JFD01609 CCOC(=O)c1c(c(c([nH]1)C)C(=O)C)c2ccccc2 KM00582 CSc1c(cn(n1)c2ccccc2)/C(=N/OC(=O)c3cccs3)/N KM07794 CCOC(=O)C(=CNc1cc(nn1C)C(C)(C)C)C(=O)OCC KM00531 Cc1cc(n2c(n1)cc(n2)c3ccccc3)C KM00221 Cc1cc(nc2c1c(nn2C(C)(C)C)C)O KM00300 c1ccc(cc1)S(=O)(=O)c2ccsc2 KM04620 c1ccc(c(c1)C(=O)Nc2cscc2S(=O)(=O)c3ccc(cc3)Cl)Cl KM01648 c1cc(ccc1S(=O)(=O)/C(=N/O)/C#N)Cl KM01346 c1cc(ccc1/C=C(\C#N)/C(=O)c2ccc(cc2)OC(F)(F)F)Cl KM04864 CS(=O)(=O)c1cc2cc(ccc2oc1=O)Cl KM04866 Cc1ccc(cc1)/C=C(\C#N)/C(=O)c2ccc(cc2)OC(F)(F)F KM04865 Cc1c(csc1C(=O)Nc2ccccc2Cl)S(=O)(=O)c3ccc(cc3)Cl KM01363 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)N3CCOCC3 KM04801 Cc1c(csc1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl KM01368 c1ccc(cc1)N/C=C(\C#N)/C(=O)c2ccc(cc2)OC(F)(F)F KM04872 CSc1c(c(c(s1)C(=O)Nc2ccccc2Cl)c3cccs3)C#N KM01689 c1cc(ccc1SC(=O)CSCCS(=O)(=O)c2ccc(cc2)Cl)Cl KM01694 c1cc(ccc1NC(=O)ONC(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl KM07588 c1cc(ccc1S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl KM00462 CCOC(=O)c1cnc2c(c1N3CCOCC3)c(nn2C)C4CC4 KM00476 c1cc(ccc1S(=O)(=O)CCSCC(=O)N2CCOCC2)Cl KM01545 CC(=O)Nc1cc(nn1c2ccccc2)C3CC3 KM00257 CC(C)(C)C(=O)Nc1c(c(nn1c2ccccc2)C3CC3)Br KM00275 CO/N=C/1\CCCc2c1c(sc2C(=O)N/N=C/c3ccccc3Cl)SC KM04598 CC(C)(C)/C=N/NC(=O)c1c2c(c(s1)SC)/C(=N/OC)/CCC2 KM04600 Cc1c(csc1C(=O)N/N=C/C(C)(C)C)S(=O)(=O)c2ccc(cc2)Cl KM01377 Cn1c(nnc1SC)c2cc(sc2)S(=O)(=O)Nc3cccc(c3)Cl KM04605 c1ccc(c(c1)C2CC(=O)C=C(S2)SCC(=O)Nc3ccc(cc3Cl)Cl)Cl KM04607 c1ccc(cc1)c2cc3[nH]c4c(c(=O)n3n2)CSC4 KM00498 c1ccc2c(c1)N=C3C(S2)CC(=O)N3Cc4ccccn4 KM07630 c1cc(sc1)c2cc(n3c(n2)cc(n3)c4cccs4)C(F)(F)F KM00396 CC(C)(C)c1ccc(cc1)c2cc([nH]n2)NS(=O)(=O)c3ccc(cc3)Cl KM00499 CCOC(=O)c1c2c(c(s1)Sc3nnc(n3C)C(F)(F)F)C(=O)CC(C2)(C)C KM04771 Cc1cc2nc(nc(n2n1)/N=C/N(C)C)SC KM01550 CC(C)(C)c1ccc(cc1)c2c(c([nH]n2)NS(=O)(=O)c3ccccc3)Br KM00519 CC1(Cc2c(sc(c2C(=O)C1)SCc3ccc(cc3)Cl)C#N)C KM03311 CCOC(=O)NC(=O)c1cn(c(=O)n(c1=O)Cc2ccccc2)Cc3ccco3 KM07701 c1c(c(=O)[nH]c(=O)n1C2CCCCC2)C#N KM07704 CCC(CC)(C#C)NC(=O)NCCCCCCNC(=O)NC(CC)(CC)C#C DP00785 C#CC1(CCCCC1)NC(=O)Nc2ccccc2 DP00787 c1cc(sc1S(=O)(=O)N/N=C/c2ccsc2)Cl KM01761 CN1CCN(CC1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2 JFD02192 c1cc(ncc1C(F)(F)F)Sc2c(c(ncn2)Sc3ccc(cn3)C(F)(F)F)[N+](=O)[O-] KM07705 CCOC(=O)NC(=O)c1cn(c(=O)n(c1=O)Cc2c(cccc2Cl)Cl)Cc3ccccn3 KM07707 Cn1c(nnc1Sc2c(c(ncn2)Sc3nnc(n3C)C(F)(F)F)[N+](=O)[O-])C(F)(F)F KM07709 CS(=O)(=O)c1c2c(c(s1)NC(=O)Nc3cccc(c3)C(F)(F)F)CCC=C2 KM04665 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)CSc3cccs3 KM04671 Cn1c(nnc1SCCS(=O)(=O)c2ccc(cc2)OC(F)(F)F)C(F)(F)F KM05000 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl KM04701 c1cc(ccc1NC(=O)C2CCN(CC2)c3ccc(cn3)C(F)(F)F)Cl KM07703 c1cc(c(c(c1)Cl)/C=N/C(=C(\C#N)/N)/C#N)F KM00312 Cc1cc(=O)n2c([nH]1)cc(n2)C(C)(C)C KM00319 CC1(Cc2c(c(sc2C(=O)/C=C/N(C)C)SC)C(=O)C1)C KM03313 CS(=NS(=O)(=O)c1ccc(s1)S(=O)(=O)c2ccc(cn2)C(F)(F)F)(=O)c3ccc(cc3)Cl KM04974 CNC(=S)NNC(=O)CSc1cc(nc2c1cccc2)C(F)(F)F KM07712 CSc1c(c(n[nH]1)c2cccc(c2)Cl)C#N KM01429 Cn1c(nnc1SCC(=O)Nc2cccc(c2)C(F)(F)F)CC3C(=O)Nc4ccccc4S3 KM07505 CCOC(=O)C1=C(C(=O)N(C1)C2CCCCC2)Nc3ccc(cc3)F KM00133 CCOC(=O)Cn1c(=O)c(cn(c1=O)Cc2ccco2)C(=O)NC(=O)OCC KM07724 Cc1ccc(cc1C)Nc2c3ccccc3ncn2.Cl DP00801 COc1cscc1C(=O)Nc2ccc(cc2)Cl KM01763 c1ccc(c(c1)/C=c/2\c(=O)n3c(=C(C(C(=C3N)C#N)c4ccccc4Cl)C#N)s2)Cl KM00534 c1ccc(c(c1)C(=O)OCC#Cc2ccc(s2)c3ccccn3)Cl KM07837 c1ccnc(c1)c2ccc(s2)C#CCOC(=O)c3cccs3 KM07838 c1cc(ccc1S(=O)(=O)CC#N)Cl KM00415 Cc1cc(n2c(n1)c(c(n2)c3ccccc3)Br)O KM00421 CCOC(=O)c1c[nH]c2cc(nn2c1=O)c3cccs3 KM00423 CCOC(=O)c1c[nH]c2cc(nn2c1=O)c3ccc(cc3)C(C)(C)C KM00424 CCOC(=O)NC(=O)c1cn(c(=O)n(c1=O)Cc2ccc(cc2)Cl)Cc3cccs3 KM07706 CN1c2ccccc2C(=O)CS1(=O)=O KM00425 CCOC(=O)Cn1c(=O)c(cn(c1=O)Cc2cccs2)C(=O)NC(=O)OCC KM07714 CCOC(=O)c1c[nH]c2cc(nn2c1=O)C(C)(C)C KM00426 c1ccc(cc1)CN/C(=C(/C#N)\NCc2c(cccc2Cl)F)/C#N KM00427 COc1ccc(cc1)n2cc(c(=O)n(c2=O)Cc3ccccc3)C#N KM07715 CCOC(=O)c1cnc2cc(nn2c1C)c3ccccc3 KM01667 CSc1c(c(c(s1)C(=O)Nc2ccc(cc2F)F)c3cccs3)C#N KM01687 Cc1csc(c1NC(=O)C(Cl)(Cl)Cl)C(=O)OC GK01264 CSc1c(c(c(s1)C(=O)Nc2cccc(c2)Cl)c3cccs3)C#N KM01690 CCOC(c1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccccn2)OCC KM01692 CSc1nc(nc(n1)N/C=C(\C#N)/C(=O)C2CC2)C3CC3 KM01707 CNc1ccc(cc1C(F)(F)F)CSc2ccc(cn2)C(F)(F)F KM04726 CN(C)c1nc(nc(n1)SC)N/C=C(/C#N)\C(=O)C2CC2 KM01708 Cc1ccc(cc1)S(=O)(=O)Nc2cc(n[nH]2)c3ccc(cc3)C(C)(C)C KM00511 CSc1c2c(c(s1)C(=O)NN)CCC=C2 KM04727 c1ccc(cc1)S(=O)(=O)c2cccs2 KM04728 c1cc(ccc1S(=O)(=O)CCN2CCC(CC2)C(=O)N)Cl KM07638 Cc1csc(c1N)C(=O)OC.Cl GK01294 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)N(C)c2ccc(cc2)C(C(=O)OC)(C(F)(F)F)O JFD02189 CN1c2ccccc2C(=O)/C(=N\Nc3ccccc3F)/S1(=O)=O KM00501 CC1(Cc2c(c(sc2C(=O)OC)Sc3cccs3)C(=O)C1)C KM04770 CC1(Cc2c(cnc(n2)SC)/C(=N\OC(=O)c3ccc(cc3)Cl)/C1)C KM04772 CC(C)(C)c1ccc(cc1)c2c(c(n[nH]2)NC(=O)c3ccc(cc3Cl)Cl)Br KM00516 CCOC(=O)C(C(F)(F)F)(NCCc1ccccc1)NC(=O)C JFD02195 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C(F)(F)F)NC(=O)c2ccccc2Cl JFD02196 CC1(Cc2c(cnc(n2)SC)/C(=N/OC(=O)c3ccccc3Cl)/C1)C KM04773 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4cccc5c4nsn5 KM07665 CCOC(=O)NC(=O)CC#N KM07667 CC(C)(C)c1ccc(cc1)c2c(c([nH]n2)NC(=O)c3ccccc3F)Br KM00515 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)N=S(=O)(C)c3ccccc3 KM04939 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)Oc3cccc(c3)C(F)(F)F KM04703 CCOC(=O)c1c(c(c([nH]1)C)C(=O)C)C BTB09323 CCCS(=O)(=O)c1cc2ccccc2oc1=O KM04886 c1cc(cc(c1)C(F)(F)F)C(=O)/C(=C/Nc2cnccn2)/C#N KM04888 CSc1c(cn(n1)c2ccccc2)c3nc(on3)c4ccc(cc4)C(F)(F)F KM07824 CCCS(=O)(=O)c1cc2cc(ccc2oc1=O)Cl KM04822 Cn1c(nnc1SCC(=O)Nc2cccc(c2)C(F)(F)F)CSc3cc(nc4c3cccc4)C(F)(F)F KM07747 c1ccc(cc1)c2cc(=O)n3c([nH]2)cc(n3)c4ccco4 KM00181 CCCCc1c([nH]c2cc(nn2c1=O)c3ccco3)C KM00185 CN(C)/C=C/C(=O)c1ccccc1O KM07559 c1ccc(cc1)NC(=O)Nc2ccc(cc2)C3SCCS3 KM00724 CCOC(=O)/C(=C/c1ccccc1Cl)/C#N KM00728 c1c(cnc(c1Cl)C(=O)NO)C(F)(F)F KM07580 Cc1ccc(cc1)S(=O)(=O)CCN(CCS(=O)(=O)c2ccc(cc2)C)c3ncccn3 KM00729 Cc1ccc(cc1)S(=O)(=O)CCN2CCN(CC2)CCS(=O)(=O)c3ccc(cc3)C KM00730 COc1cccc(c1)C(=O)/C=C/2\NC(=O)CS2 KM00372 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)F KM00373 Cc1c(csc1C(=O)N2CC(OC(C2)C)C)S(=O)(=O)c3ccc(cc3)Cl KM01469 CS(=O)(=O)c1c(c(n[nH]1)c2ccccc2Cl)C#N KM01470 c1ccc(cc1)n2c(nnn2)c3c[nH]c4ccccc4c3=O JFD00602 Cc1cc(n2c(n1)cc(n2)C3CC3)C KM00339 CS(=O)(=O)c1c(c(on1)c2cccs2)C#N KM01485 Cc1ccccc1C(=O)/C(=C\N(C)C)/c2nnnn2c3ccccc3 JFD00604 CN(C)/C=C(/c1nnnn1c2ccccc2)\C(=O)c3cccc(c3)C(F)(F)F JFD00605 c1ccc(cc1)C2C(=C(OC(=C2C#N)N)C3CC3)C#N KM00340 c1cc(ccc1Nc2c(c(ncn2)Nc3ccc(cc3)Cl)[N+](=O)[O-])Cl KM07734 CC(C)n1cc(c(=O)[nH]c1=O)C#N KM07737 c1ccc(cc1)S(=O)(=O)CCN(CCS(=O)(=O)c2ccccc2)c3ncccn3 KM00760 CCOC(=O)/C(=C\NCc1ccncc1)/C(=O)NC(=O)OCC KM07820 Cc1ccc(cc1)S(=O)(=O)NCCSc2cc(nc3c2cccc3)C(F)(F)F KM07835 Cc1cc(n2c(n1)c(cn2)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N)C KM00763 CC(=O)c1c2c(c(s1)SC)C(=O)CC(C2)(C)C KM03306 CN1c2cc(ccc2C(=O)/C(=C/Nc3ccc(cc3)OC)/S1(=O)=O)C(=O)OC KM05052 CC(C)(C)S(=O)(=O)c1cnc(nc1N)c2cnccn2 KM05055 Cn1c(nnc1SCc2ccc(cc2)Cl)CSc3cc(nc4c3cccc4)C(F)(F)F KM07731 CC(C)(C)S(=O)(=O)/C(=C/N/N=C/c1ccccc1Cl)/C#N KM01891 CC1CN(CC(O1)C)C(=O)Nc2csc(c2OC)Cl KM00615 COc1c(csc1Cl)NC(=O)N2CCCCC2 KM00616 Cn1c(nnc1SCC(=O)Nc2ccccc2Cl)CSc3cc(nc4c3cccc4)C(F)(F)F KM07735 CC(C(=O)/C=C/N(C)C)SC KM07740 c1ccc(cc1)c2cc3ncc(c(n3n2)N)C#N KM00647 CC(C)(C)/C=N/NS(=O)(=O)c1ccc(s1)Cl KM01760 Cc1c(c(on1)c2ccccc2)NC(=O)NCc3csc(n3)c4ccccc4 HTS13966 c1ccc(c(c1)C2CC(=O)C=C(S2)SCC(=O)c3ccc(cc3)[N+](=O)[O-])Cl KM04603 COc1c(csc1S(=O)(=O)N2CCOCC2)C(=O)OC KM07850 c1cc(ccc1c2cc(n(n2)c3ccc(c(c3)Cl)Cl)N)OC(F)(F)F KM04991 CC1(Cc2c(sc(c2C(=O)C1)SC)C#N)C KM03308 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccc(cc4Cl)Cl KM07862 c1cc(ccc1OC(F)(F)F)S(=O)(=O)CCSc2ccc(cc2)Cl KM04996 c1cc(ncc1C(F)(F)F)S(=O)(=O)c2ccc(s2)S(=O)(=O)N3CCCCC3 KM04909 COc1c(c(ncn1)OC)[N+](=O)[O-] KM07755 CSc1c(c(nc(n1)C2CC2)C3CC3)C#N KM01779 CCOC(c1ccc(cc1)C=C(C#N)C#N)OCC KM01762 CSC(=C(C#N)C(=O)c1ccc(cc1)OC(F)(F)F)SC KM04926 CC1(Cc2c(c(sc2Cl)SC)C(=O)C1)C KM04928 COc1cscc1C(=O)O KM00448 c1cc(cc(c1)/C(=N/O)/N)CS(=O)(=O)c2ccc(cc2)Cl KM00591 c1ccc(c(c1)C(=O)O/N=C(/c2cccc(c2)CS(=O)(=O)c3ccc(cc3)Cl)\N)Cl KM00593 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/C(=C(/C#N)\N)/C#N KM04652 c1cc(ccc1Oc2ccc(cn2)C(F)(F)F)Br KM07899 c1cc(ccc1S(=O)(=O)CCSCC(=O)Nc2ccc(c(c2)Cl)F)Cl KM01534 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)Sc3ccc(cc3)Cl KM07875 c1cc(ccc1Oc2c(nccn2)C#N)Cl KM07878 Cc1c(c(sc1C(=O)OC)SC)C(=O)C KM02005 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCCNS(=O)(=O)c3ccc(cc3)Cl KM07832 Cc1c(cnc2n1nc(c2)c3ccc(cc3)Cl)C(=O)C KM01787 Cc1c(cnc2n1nc(c2)C3CC3)C(=O)C KM01788 CS(=O)(=O)NCCSc1cc(nc2c1cccc2)C(F)(F)F KM07834 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Cc2ccccn2 KM07673 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=O)c2cccs2 KM09030 Cc1ccc(cc1)S(=O)(=O)CCN2CCN(CC2)c3cc(nc4c3cc(cc4)C)C(F)(F)F KM09031 Cc1c2c(=O)[nH]c(cn2cn1)c3ccc(cc3)Cl KM07685 c1ccc(c(c1)NC(=O)CSCCS(=O)(=O)c2ccc(cc2)Cl)Cl KM01537 c1cc(cc(c1)C#N)COc2ccc(cc2)[N+](=O)[O-] KM00762 c1ccnc(c1)SCc2cccc(c2)/C(=N/OC(=O)c3cccs3)/N KM01530 CC(C)(C)c1ccc(cc1)C(=O)/C=C/2\NC(=O)CS2 KM00371 COc1cccc(c1)C(=O)/C=c/2\[nH]c(=O)/c(=C\c3cccs3)/s2 KM00399 CC(C)(C)C(=O)C(=C1SCCCS1)C#N KM00826 c1cc(ccc1/N=N/c2c(n[nH]c2N)C3CC3)Cl KM00407 c1cc(ccc1SCC#N)Cl KM00412 CCOC(=O)c1c[nH]c2cc(nn2c1=O)c3ccccc3 KM00419 Cc1c(sc2c1c(c(s2)C(=O)C)C)C#N KM03449 CNc1c(c(ncn1)Sc2ccc(cc2)Cl)[N+](=O)[O-] KM07909 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCC(=O)NNC(=O)c3ccc(cc3)Cl KM07675 CC(C)(C)c1ccc(cc1)C(=O)/C(=C/c2cccs2)/C#N KM00388 c1ccc(c(c1)/N=N/c2c(n[nH]c2N)C3CC3)Cl KM00390 CC(C)(C)c1ccc(cc1)C(=O)/C(=C/c2ccccc2Cl)/C#N KM00389 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)OC)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01319 c1cc(ccc1n2cc(c(=O)[nH]c2=O)C#N)OC(F)(F)F KM07691 CC(C)(C)c1ccc(cc1)C(=O)/C=c/2\[nH]c(=O)/c(=C\c3cccs3)/s2 KM00391 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4cccs4 KM00392 CN1c2ccccc2C(=C(S1(=O)=O)C(=O)Nc3ccc(cc3)OC(F)(F)F)O KM04647 c1cc(sc1)c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F KM00403 c1ccc(cc1)NC(=O)OCC#Cc2ccc(s2)c3ccccn3 KM07841 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)N=S(=O)(C)c3ccc(cc3)Cl)C)Br KM06367 Cc1csc(n1)c2cn(c(=O)n(c2=O)Cc3ccccc3)C(C)C KM07846 CNc1c(c(ncn1)N2CCCC2)[N+](=O)[O-] KM07925 CNc1c(c(ncn1)Oc2ccc(cc2)Cl)[N+](=O)[O-] KM07926 Cc1cccc(c1)c2c(c(nc(n2)N)SC)C#N KM02054 c1csc(c1Cl)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK01324 CCCS(=O)(=O)C1=C(OC(=C(C1c2ccc(cc2)Cl)C#N)c3ccccc3)N KM01623 CC(C)(C)c1ccc(cc1)C(=O)/C(=C/c2cccc(c2O)OC)/C#N KM00438 CC(C)(C)c1ccc(cc1)c2cc([nH]n2)NC(=S)NC(=O)c3ccccc3 KM00440 CCSc1c(c(c(s1)C(=O)OC)c2cccs2)C#N KM01637 CCCSc1c(c(c(s1)C(=O)OC)c2cccs2)C#N KM01638 COc1c(csc1Cl)C(=O)O KM00452 c1cc(ccc1/C=N/OC(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl KM07568 CC(C)S(=O)(=O)c1cc(sc1)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM03305 c1ccc(cc1)C2CC(=O)C=C(S2)SCC#N KM04658 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)Oc3ccc(cc3)Cl KM04661 c1cc(ccc1OC(F)(F)F)S(=O)(=O)CCSc2ccc(cn2)C(F)(F)F KM04994 Cc1c(cnc2n1nc(c2)C3CC3)S(=O)(=O)c4ccc(cc4)Cl KM02038 Cc1c(c(sc1C(=O)OC)SC)c2cc[nH]n2 KM02052 CSC(=C(C#N)C(=O)c1ccccc1)SC KM00767 c1ccc(cc1)C(=O)NC(=S)Nc2c(c(n[nH]2)C3CC3)/N=N/c4ccc(cc4)Cl KM00439 COc1cc(nc2c1csc2C(=O)OC)C(F)(F)F KM07528 CC(C)(C)c1cc([nH]n1)NC(=S)NC(=O)c2ccccc2 KM00442 c1cc(ncc1C(F)(F)F)SC/C(=N/OC(=O)c2c(cc(cn2)C(F)(F)F)Cl)/N KM07571 c1ccc(cc1)C(=O)NC(=S)Nc2c(c(n[nH]2)C3CC3)/N=N/c4ccccc4Cl KM00454 c1ccc(cc1)c2cc([nH]n2)NC(=O)c3ccccc3F KM00357 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CCCCN4C(=O)c5ccccc5C4=O KM07914 Cn1cc(c(n1)c2cccc(c2)NC(=O)C(Cl)(Cl)Cl)Br KM02046 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3c4c(c(s3)SC)C=CCC4 KM04946 CC(C)NC(=O)CSc1nnc(n1C)c2c3c(c(s2)SC)C=CCC3 KM04948 CC1(Cc2c(c(sc2C(=O)OC)SC)/C(=N\O)/C1)C KM03450 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=O)Nc3cccc(c3)Cl KM07954 Cc1c(c(n(n1)Cc2ccc(o2)C(=O)Nc3cc(cc(c3)Cl)Cl)C)Br KM07518 CCCCOc1cc(nc2c1cc(cc2)CSc3[nH]c4ccccc4n3)C(F)(F)F KM07521 CC(=O)CSc1ccccc1C(=O)OC KM07591 CNc1c(c(ncn1)N2CCCCC2)[N+](=O)[O-] KM07923 c1cc(ccc1S(=O)(=O)CCSCC(=O)O)Cl KM01502 COCCCN/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl KM00752 c1ccc(cc1)c2cc([nH]n2)NC(=O)c3ccc(cc3)Cl KM00360 Cc1cc(n2c(n1)c(cn2)/C(=N/OC(=O)c3ccccc3Cl)/N)C KM00753 c1ccc(c(c1)C(=O)OC2=C(C(=O)CCC2)Cl)Cl KM05003 CSc1c(c(cs1)c2cccs2)C#N KM02035 Cc1cc2ncc(c(n2n1)C)S(=O)(=O)c3ccc(cc3)Cl KM02037 c1cc(ccc1/N=N/c2c(n[nH]c2N)C3CC3)F KM00404 Cc1cc2nc(c(c(n2n1)c3ccccc3)C#N)SC KM00814 c1ccc(c(c1)C(=O)C(=C2SCCCS2)C#N)Cl KM00825 COc1c(cccn1)C(=O)O KM01841 Cc1cccc(c1)C(=O)C(=C(SC)SC)C#N KM01822 CC(C)(C)c1ccc(cc1)c2c(c([nH]n2)S(=O)(=O)C)C#N KM00830 Cc1c2c(cc(nc2n(n1)C)O)COC KM00834 c1cc(cc(c1)C#N)CSc2ccc(cc2)Cl KM00581 c1ccc(cc1)c2c(c([nH]n2)N)Br KM00411 CC(C)(C)c1ccc(cc1)c2cc(n(n2)C)N KM00414 c1cc(ccc1n2cc(c(=O)[nH]c2=O)C#N)Cl KM07700 CCOC(=O)c1cnc2cc(nn2c1C)c3cccs3 KM01668 COc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)CS(=O)(=O)C3 KM07618 CSc1c(cn(n1)c2ccccc2)c3nc(on3)c4ccc(cc4)Cl KM07790 c1cc2c(cc1/C=C(\C#N)/C(=O)C3CC3)OCO2 KM00710 c1cc(ccc1C2SCCS2)NC(=O)CSc3ccc(cc3)F KM00712 Cn1c(c(cn1)C(=O)Nc2ccc(c(c2)Cl)Cl)[N+](=O)[O-] KM00805 c1cc(ccc1S(=O)(=O)CC(=O)NN)Cl KM01605 c1cc(ccc1N2C(=O)CSCC2=O)Cl KM06409 c1cc2c(c(c1)S(=O)(=O)NCC(=O)NN)nsn2 KM06410 CCOC(=O)Cn1c(=O)c(cn(c1=O)C(C)C)C(=S)N KM07876 c1ccc(cc1)COc2ccc(cc2)C(=O)O KM07877 CC(C)C(=O)Nc1cscc1S(=O)(=O)c2ccc(cc2)Cl KM01655 CCOC(=O)CNC(=O)c1c(n2c(cc(n2)C)nn1)C KM01656 Cn1c(nnc1SCC(=O)NCC=C)CSc2cccs2 KM04674 COC(=O)c1c(c(c(s1)S(=O)(=O)C)C#N)c2cccs2 KM01670 c1cc(ccc1S(=O)(=O)/C(=C/Nc2nccs2)/C#N)Cl KM01673 c1cc(ccc1C(=O)Nc2cscc2S(=O)(=O)c3ccc(cc3)Cl)Cl KM01679 Cc1c(c(n(n1)Cc2nnc(o2)SCc3c(cccc3Cl)Cl)C)Br KM04682 c1cc2c(cc1N)CS(=O)(=O)C2 KM07609 c1cc(ccc1NC(=O)OCCSCCS(=O)(=O)c2ccc(cc2)Cl)Cl KM01838 CCOC(=O)c1cnc([nH]1)SCC(=O)c2ccc(cc2Cl)Cl KM06333 CCCS(=O)(=O)c1cscc1NC(=O)CSCCS(=O)(=O)c2ccc(cc2)Cl KM03435 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(=O)NNC(=O)c4ccccc4Cl KM07918 c1cc(ccc1OC/C(=N/OC(=O)c2c(cc(cn2)C(F)(F)F)Cl)/N)Cl KM07589 COc1cccc(c1)C(=O)/C(=C/c2cccs2)/C#N KM00480 CC(C)(C)c1ccc(cc1)c2cc([nH]n2)NC(=O)c3ccccc3F KM00481 c1cc(sc1)c2cc3[nH]c4c(c(=O)n3n2)CSC4 KM00482 Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)CS(=O)(=O)C3 KM07612 CC(C)(C)c1cc(n(n1)C)N KM00494 CCOC(=O)c1cn[nH]c1N KM00785 c1cc(c(cc1N/N=C(\C#N)/C(=O)C2CC2)Cl)Cl KM00386 c1ccc(cc1)OC(=O)c2ccc(o2)CS(=O)(=O)c3ccc(cn3)C(F)(F)F KM06326 CCOC(=O)c1cnc2c(c1Sc3ccc(cn3)C(F)(F)F)c(nn2C)C KM06335 c1cc2c(c(c1)S(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)nsn2 KM06386 CC(C)Sc1c(c(ncn1)NC)[N+](=O)[O-] KM07912 CN1CCN(C(C1)C(=O)NN)C KM07913 c1cc(oc1)CN/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00668 c1cc(ccc1OC(F)(F)F)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM04952 Cc1cccc(c1)C(=O)CC#N KM01815 Cc1cc2ncc(c(n2n1)C)C(=O)/C=C/N(C)C KM01818 c1cc(ccc1S(=O)(=O)CCSCC(=O)N2CCCC2)Cl KM01553 c1cc(cc(c1)C(F)(F)F)C(=O)c2cc3cc(ccc3oc2=O)Cl KM04777 c1cc(ccc1C(=O)CSC#N)Cl KM04778 Cc1cc2ncc(c(n2n1)C)C(=O)O KM01560 c1ccc(c(c1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)Cl KM00523 COc1cccc(c1)C(=O)/C=c/2\[nH]c(=O)/c(=C\c3ccccc3)/s2 KM00387 CSC(=C(C#N)C(=O)c1ccccc1Cl)SC KM00792 c1cc(c(c(c1)Cl)CN/C(=C(/C#N)\NCc2cccs2)/C#N)F KM00420 CCOC(=O)c1c2c(c(s1)N(C(=O)c3ccccc3Cl)NC(=O)c4ccccc4Cl)C(=O)CC(C2)(C)C KM04815 COC(=O)c1c(c(cs1)S(=O)(=O)C)N KM01956 Cc1cc2ncc(c(n2n1)C)C(=O)C KM01797 Cc1cc(no1)N/C=C(\C#N)/C(=O)c2ccc(cc2)Cl KM01804 CCCS(=O)(=O)c1csc(c1N)C(=O)OC KM01968 COCc1cc(=O)n2c([nH]1)cc(n2)c3ccccc3 KM00727 c1cc(sc1)C2C(=C(OC(=C2C#N)N)C3CC3)C#N KM00346 c1ccc(c(c1)C2C(=C(OC(=C2C#N)N)C3CC3)C#N)Cl KM00342 Cc1c(c2ccccc2[nH]1)SCC(=O)NN KM07803 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)/C(=N/OC(=O)c3cccs3)/N KM07811 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=O)c3ccc(cc3)Cl KM07812 CCOC(=O)CC(=O)NC(=O)OCC KM07813 CCOC(=O)c1c2c(c(s1)N(C(=O)c3ccc(cc3)Cl)NC(=O)c4ccc(cc4)Cl)C(=O)CC(C2)(C)C KM04814 CCOC(=O)c1c2c(c(s1)N(C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NC(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(=O)CC(C2)(C)C KM04816 CCOC(=O)/C(=C\NCc1cccs1)/C(=O)NC(=O)OCC KM07817 CCOC(=O)Cn1c(=O)c(cn(c1=O)Cc2ccccn2)C(=O)NC(=O)OCC KM07725 CSc1c(c(n(n1)c2ccccc2)N)C#N KM07726 CCCCOc1cc(nc2c1cc(cc2)C)C(F)(F)F KM07509 c1ccc(cc1)NC(=O)O/N=C(\c2cccc(c2)CS(=O)(=O)c3ccccn3)/N KM01595 c1ccnc(c1)S(=O)(=O)Cc2cccc(c2)/C(=N/OC(=O)c3ccc(c(c3)Cl)Cl)/N KM01601 Cc1csc2c1c(c(s2)/C=C(\C#N)/S(=O)(=O)c3cccs3)C KM03488 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F KM07956 COc1cc(nc2c1cc(cc2)C#CCOC(=O)Nc3cccc(c3)Cl)C(F)(F)F KM08015 c1cc(cc(c1)n2cc(c(=O)n(c2=O)Cc3ccc(cc3)Cl)C#N)C(F)(F)F KM07718 Cc1c(c(c2ccccc2n1)C(=O)O)N KM00428 COc1ccc(cc1)OS(=O)(=O)c2cc(cs2)S(=O)(=O)c3ccccc3 KM04702 c1cc(ccc1Oc2c(c(ncn2)Oc3ccc(cc3)Cl)[N+](=O)[O-])Cl KM07722 CN(C)n1cccc1/C=N/NC(=O)c2ccc(cc2)Cl KM04713 CN(C)n1cccc1/C=N/NC(=O)c2cccc(c2)C(F)(F)F KM04714 CC(C)(C)c1ccc(cc1)c2cc([nH]n2)NS(=O)(=O)c3ccccc3 KM00505 c1cc(ccc1S(=O)(=O)CCN2CCC(CC2)C#N)Cl KM07660 Cc1cc(n2c(n1)c(cn2)/C(=N/O)/N)C KM00721 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2nc(nc(n2)SC)C)/C#N KM00942 COc1c(csc1S(=O)(=O)N2CCCC2)C(=O)OC KM07854 Cc1ccc(cc1)S(=O)(=O)/C(=N/O)/C#N KM01751 c1ccc(cc1)S(=O)(=O)CCN2CCC(CC2)C#N KM07653 c1ccc(cc1)S(=O)(=O)c2csc(c2N)C(=O)O KM01757 COc1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00503 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4ccc(s4)Cl KM07661 c1cc(ncc1C(F)(F)F)N2CCC(CC2)C(=O)N KM07664 CN1c2ccccc2C(=O)/C(=N\Nc3ccc(cc3)F)/S1(=O)=O KM00506 CCOC(=O)c1c[nH]c2cc(nn2c1=O)c3ccco3 KM00422 CSc1c2c(c(s1)Cl)CCCC2=O KM05032 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)NC(=O)Nc3cccc(c3)C(F)(F)F)C)Br KM06388 Cn1ccnc1SCC(=O)N2CCC(CC2)n3cccc3 KM09107 CCOC(=O)/C(=C\NC(C)C)/C(=O)NC(=O)OCC KM07819 Cc1cc(nc2c1ccc(n2)NC(=O)c3ccc(cc3)C(F)(F)F)C KM01958 CN(C)n1cccc1/C=C(\C#N)/C(=O)c2ccc(cc2)Cl KM04613 COC(=O)C1=C(CSC1)Nc2ccc(c(c2)Cl)F KM01972 COC(=O)C1=C(CSC1)Nc2ccc(cc2F)F KM01973 COC(=O)c1c(c(cs1)S(=O)(=O)C)Cl KM01975 CC(C)(C)c1ccc(cc1)c2c(c(n[nH]2)NC(=O)c3ccccc3Cl)Br KM00526 COc1ccc(cc1)/C=C\2/C(=O)N3C(S2)C(=C(C(=C3N)C#N)c4ccc(cc4)OC)C#N KM00527 c1cc(oc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00528 CS(=O)(=O)/C(=C/Nc1cnccn1)/C#N KM04893 c1ccc(cc1)S(=O)(=O)c2cc(sc2)[N+](=O)[O-] KM04899 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)CCSc2cc(nc3c2cccc3)C(F)(F)F KM07828 c1cc(ccc1NC(=O)O/N=C(/c2cnccn2)\N)OC(F)(F)F KM05039 c1ccc(cc1)C(=O)NNC(=O)CSCC(=O)Nc2ccccc2 KM09028 Cc1ccc(cc1)C(=O)/C(=C\N(C)C)/c2nnnn2c3ccccc3 JFD00603 CS(=O)(=O)c1c(c(on1)c2ccc(cc2)Cl)C#N KM01484 CO/N=C/1\CCCc2c1c(sc2C(=O)N/N=C/c3cccs3)SC KM04599 Cc1c(c(n(n1)Cc2ccc(o2)C(=O)O)C)Br KM07512 CCCCOc1cc(nc2c1cc(cc2)CSc3nc4ccccc4s3)C(F)(F)F KM07516 CS(=O)(=O)c1c(c(n[nH]1)c2ccc(cc2)Cl)C#N KM01441 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)SCCS(=O)(=O)c3ccc(cc3)Cl KM02016 CS(=NS(=O)(=O)c1ccc(cc1Cl)Cl)(=O)c2ccc(cc2)Cl KM05078 c1ccnc(c1)c2ccc(s2)S(=O)c3ccc(cc3)Cl KM05079 CSc1c-2c(cs1)CCc3c2nc(nc3)SCc4ccc(cc4)Cl KM05089 c1cc(c(cc1Cl)Cl)NC(=O)N=S2CCN(CC2)c3c(ccs3)[N+](=O)[O-] KM06304 CC(=O)N1CSCC1C(=O)NNS(=O)(=O)c2ccccc2 KM06306 c1cc(c(cc1Cl)Cl)OC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F KM06312 CNC(=S)NNC(=O)CSCC(=O)Nc1ccccc1 KM09040 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)CCS(=O)(=O)c4ccc(cc4)Cl KM09041 c1ccc(cc1)NC(=O)OCC#Cc2ccc(cc2)C#N KM09052 Cc1nc(nc(n1)SC)N/C=C(\C#N)/C(=O)C2CC2 KM01616 c1cc(sc1/C=C(\C#N)/C(=O)C2CC2)[N+](=O)[O-] KM00713 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)S(=O)(=O)c4ccccc4)C(F)(F)F KM09134 CSc1c(cc(s1)C(=O)NC(=O)Nc2cccc(c2)C(F)(F)F)C#N KM03396 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)c3c4c(c(s3)SC)C=CCC4 KM04947 CSc1c(c(n[nH]1)c2ccccc2)C#N KM00774 CC(C)(C)c1cc2nc(cc(n2n1)N/N=C/c3ccc(cc3)C(F)(F)F)C(F)(F)F KM07981 COc1cccc(c1)c2cc(n(n2)c3c(cc(cc3Cl)Cl)Cl)N KM00791 c1cc(sc1)C(=O)OCC#Cc2ccc(cc2)C#N KM09061 CS(=NC(=O)c1ccc(cc1Cl)Cl)(=O)c2ccc(cc2)Cl KM05122 CCOC(=O)c1c(c(c(s1)SCc2cccc(c2)Cl)S(=O)(=O)C(C)C)N KM03336 CCOC(=O)c1c2c(c(s1)SC)C(CCC2)O KM03342 CCN1CC(=C(C1=O)Nc2ccc(cc2)F)C(=O)OCC KM00384 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(/c2cnccn2)\N KM05047 CO/N=C/1\CCCc2c1c(sc2C(=O)NNS(=O)(=O)c3ccccc3Cl)SC KM04631 c1ccc(cc1)NC(=O)OCc2nccn2Cc3ccc(cc3)Cl KM08012 c1ccc(cc1)C(=O)CSC2=CC(=O)CC(S2)c3ccc(cc3)Cl KM04644 Cn1c(cc(n1)c2ccc(s2)Sc3ccc(cc3)Cl)C(F)(F)F KM04989 Cc1cc2ncc(c(n2n1)N)S(=O)(=O)C(C)(C)C KM02026 CC(C)(C)c1cc2nc(cc(n2n1)NNC(=O)Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F KM07970 CCCCNC(=O)NNc1cc(nc2n1nc(c2)C(C)(C)C)C(F)(F)F KM07971 CCOC(=O)Cn1cc(c(=O)[nH]c1=O)C#N KM07975 CC(C)(C)N/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Br KM00756 Cc1csc(n1)c2c(c(c(s2)SC)c3ccnc(n3)SCc4c(cccc4Cl)Cl)C KM05097 CCOC(=O)c1cnc2c(c1Oc3ccc(cc3)Cl)c(nn2C)C KM05102 c1cc(ccc1C#CCOC(=O)Nc2cc(cc(c2)Cl)Cl)C#N KM09053 COc1cscc1C(=O)N KM01620 c1ccc(cc1)S(=O)(=O)c2cc3ccccc3oc2=O KM04868 c1cc(ccc1C(=O)/C(=C/c2ccc(c(c2)Cl)Cl)/C#N)OC(F)(F)F KM04871 Cc1csc(n1)c2c(c(c(s2)SC)c3cc[nH]n3)C KM04949 CSc1c2c(c(s1)C(=O)NNC(=O)c3ccc(cc3)Cl)CCCC2O KM03406 CSc1c2c(c(s1)C(=O)Nc3ccc(cc3F)F)CCC=C2 KM03410 c1cc(ccc1C(=O)OC2=C(C(=O)CCC2)Cl)Cl KM05002 CC(C)NC(=O)c1c(c(cs1)S(=O)(=O)C)Cl KM02101 COC(=O)c1ccc(c(c1)NS(=O)(=O)C)C(=O)OC KM05005 Cc1csc(n1)c2c(c(c(s2)SC)c3ccnc(n3)SCc4ccc(cc4)Cl)C KM05021 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C)CSCC(=O)Nc3ccccc3 KM09157 CCOC(=O)CSc1nnc(n1C)CSc2c([nH]c3c2cccc3)C KM07993 c1cc(ccc1Cn2ccnc2COC(=O)c3ccc(cc3)Cl)Cl KM08002 COc1cc(nc2c1cc(cc2)C#CCOC(=O)c3ccccc3)C(F)(F)F KM08006 CCSc1c\2c(c(s1)C(=O)OC)CC(C/C2=N\O)(C)C KM04982 CN(c1cc(ccc1C(=O)OC)C(=O)OC)S(=O)(=O)C KM05015 CS(=O)(=O)c1c2c(c(s1)C(=O)NC(=O)Nc3ccccc3Cl)CCC=C2 KM05025 Cn1ccnc1Sc2cc(nc3c2csc3C(=O)OC)C(F)(F)F KM07894 c1cc(ccc1C(=O)Nc2ccc3c(c2)CS(=O)(=O)C3)Cl KM07610 CC(=O)Nc1cc(n[nH]1)C2CC2 KM00787 c1ccc2c(c1)c(cc(n2)C(F)(F)F)NN KM07986 COC(=O)CC(=O)NC(CSC(=O)Nc1ccc(cc1)SC(F)(F)F)C(=O)OC KM07987 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(=O)NNS(=O)(=O)c4ccc(s4)Cl KM07989 CCOC(=O)c1c(c(c(s1)SCc2c(cccc2Cl)Cl)S(=O)(=O)C(C)C)N KM03333 CSc1c-2c(cs1)CCc3c2nc(nc3)SCC(=O)NCC=C KM05116 COC(=O)c1c(c2c(s1)nccn2)N/C=C(\C#N)/C(=O)c3ccc(cc3)Cl KM05120 Cc1c(c2ccccc2[nH]1)SCc3nnc(n3C)SCC(=O)Nc4ccc(cc4)Cl KM07995 c1cc(ccc1C(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)OC(F)(F)F KM04874 c1cc(oc1)CS(=O)(=O)c2cnc(nc2N)c3ccncc3 KM03338 CCOC(=O)C(=NNc1ccccc1Cl)C(=O)OCC KM07802 CCOC(=O)c1csc(n1)c2cn(c(=O)n(c2=O)Cc3ccccc3)C(C)C KM07848 CC(C)(C)C(=O)/C(=N/Nc1c(csc1C(=O)OC)S(=O)(=O)Cc2ccco2)/C#N KM03423 CSc1c2c(c(s1)C(=O)NNC(=O)Nc3ccc(cc3)Cl)CCC=C2 KM03476 CNC(=O)NNC(=O)c1c2c(c(s1)SC)C=CCC2 KM03477 Cn1c(nnc1SCC(=O)Nc2cccc(c2)C(F)(F)F)Cc3nc(no3)c4cnccn4 KM09213 c1ccc2c(c1)C(CS2(=O)=O)N3CCOCC3 KM08142 c1cc(c2c(c1)nsn2)N KM06374 c1cc2c(cc1N/C=C(\C#N)/S(=O)(=O)c3ccc(cn3)C(F)(F)F)OCCO2 KM05178 CCCS(=O)(=O)/C(=C/Nc1ccc2c(c1)OCCO2)/C#N KM05179 c1cc(ncc1C(F)(F)F)S(=O)(=O)c2cnc(nc2N)N3CCCC3 KM05182 CCOC(=O)Cn1c(=O)c(cn(c1=O)C(C)C)c2nc(cs2)C(C)(C)C KM07930 CCOC(=O)Cn1c(=O)c(cn(c1=O)C(C)C)c2nc(cs2)c3ccc(cc3)Cl KM07931 Cc1cc(n2c(n1)c(cn2)/C(=N/OC(=O)c3ccccc3F)/N)C KM00793 Cn1c(c(cn1)C(=O)Nc2ccc(cc2F)F)[N+](=O)[O-] KM00797 c1cc(cc(c1)Oc2c(nccn2)/C(=N/O)/N)C(F)(F)F KM07849 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)OCC)C)C KM03416 CSc1c(cc(s1)NC(=O)Nc2cccc(c2)C(F)(F)F)C#N KM03417 CC1(Cc2c(c(sc2c3cc[nH]n3)SC)C(=O)C1)C KM03422 CC(C)S(=O)(=O)c1csc(c1N)C(=O)O KM02125 CC(C)S(=O)(=O)c1csc(c1N)C(=O)OCC(=O)c2ccc(cc2)Cl KM02143 CCOC(=O)c1c(c(c(s1)SCc2ccccc2)S(=O)(=O)C(C)C)n3cccc3 KM03354 c1ccc(cc1)C(=O)OCc2nccn2Cc3ccc(cc3)Cl KM08009 CSc1c(cc(s1)C(=O)Nc2cccc(c2)C(F)(F)F)C#N KM03349 CNC(=O)c1cc(c(s1)SC)C#N KM03350 CCOC(=O)c1c(c(c(s1)SCc2ccc(cc2)Cl)S(=O)(=O)C(C)C)n3cccc3 KM03353 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=O)c3ccccc3Cl KM07816 CCOC(=O)/C(=C\NCc1ccco1)/C(=O)NC(=O)OCC KM07818 Cc1c2c(cc(nc2n(n1)C)OC(=O)N(C)C)COC KM00876 c1ccc(cc1)C#Cc2ccc(cc2)/C=N/O KM08078 CC(C)(C)c1cc2nc(cc(n2n1)Sc3nnc(n3C)C(F)(F)F)C(F)(F)F KM08083 COc1cccc(c1)/C=N/NC(=O)Cc2nc(no2)c3cnccn3 KM09176 c1ccc(cc1)/C=N/CCN2CCN(CC2)C(=O)c3ccc(cc3)Cl KM08147 Cn1c(nnc1SCc2c(cccc2Cl)Cl)Cc3nc(no3)c4cnccn4 KM09214 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(=O)NNC(=O)C(C)(C)C KM07917 CNc1c(c(ncn1)N2CCOCC2)[N+](=O)[O-] KM07924 CSc1c2c(c(s1)C#N)CC(CC2=O)c3ccccc3 KM03569 c1cc(sc1)C(=O)/C(=N/Nc2ccc(cc2)OC(F)(F)F)/C#N KM03570 c1cc(cc(c1)Cl)NC(=O)OCc2nccn2Cc3ccc(cc3)Cl KM08021 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)N/N=C/c3ccccc3 KM02162 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)O)C)Br KM06350 COc1cccc(c1)C(=O)C(=C(SC)SC)C#N KM00799 c1cc(ccc1S(=O)(=O)CCSCCOC(=O)c2cc(cc(c2)Cl)Cl)Cl KM01828 CCSc1c(cccn1)C(=O)NC(CCSC)C(=O)O KM01831 c1cc(ccc1CS(=O)(=O)c2cnc(nc2N)c3cnccn3)Cl KM05048 COc1c(csc1S(=O)(=O)N2CCCCC2)C(=O)OC KM07853 c1cc(cc(c1)Oc2c(nccn2)/C(=N/OC(=O)c3ccc(cc3)Cl)/N)C(F)(F)F KM07859 CSc1c(c(nc(n1)c2cnccn2)c3ccco3)C#N KM05044 Cc1ccc(cc1)C(=O)NNC(=O)CSCC(=O)Nc2ccccc2 KM09029 CS(=NC(=O)Nc1ccc(cc1)SC(F)(F)F)(=O)c2ccccc2 KM05026 CSc1c2c(c(s1)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F)CCCC2O KM03424 COc1ccc(cc1)S(=O)(=O)NNC(=O)c2c3c(c(s2)SC)C=CCC3 KM03479 CSc1cccc(c1)NC(=O)NCc2ccccc2 KM09219 c1ccc(c(c1)C(=O)OCc2nccn2Cc3ccc(cc3)Cl)Cl KM08011 CSc1c(c(nn1CC(=O)N/N=C/c2cccs2)c3cccs3)C#N KM00932 Cn1c(=O)c(cn(c1=O)c2ccsc2C(=O)OC)C#N KM08018 c1cc(c(cc1N2CCSCC2)[N+](=O)[O-])C#N KM06341 CCc1cccc(c1NC(=O)COc2cc3c(cc2OC)OC(C=C3)(C)C)C JFD00341 CCCN(C(=O)CC#N)C(=O)Nc1ccc(cc1)Cl KM09077 CC(=O)c1c2c(c(s1)SCc3c(cccc3Cl)Cl)C(=O)CC(C2)(C)C KM03317 CC(C)S(=O)(=O)c1cc(sc1)NC(=O)Nc2cc(cc(c2)Cl)Cl KM03318 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)Oc3ccc(cc3)Cl KM07936 CC(C)(C)c1cc2nc(cc(n2n1)SCC(=O)OC)C(F)(F)F KM07939 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)Oc3ccccc3C(F)(F)F KM07940 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(=O)NNC(=O)c4cccs4 KM07919 COC(=O)c1c(c(cs1)S(=O)(=O)Cc2ccco2)NN=C(C#N)C#N KM03453 CN(C)/C=N/c1c(csc1C(=O)OC)S(=O)(=O)C KM02036 Cc1c(cnc2n1nc(c2)C(C)(C)C)S(=O)(=O)c3ccc(cc3)Cl KM02039 CCOC(=O)c1c(c(c([nH]1)C)/C(=N/O)/C)C KM00584 c1ccc(c(c1)/C(=C/C#N)/Nc2ccc(cc2F)F)Cl KM00586 CS(=O)(=O)c1c2c(c(s1)C(=O)NC(=O)Nc3cccc(c3)C(F)(F)F)CCC=C2 KM05009 Cc1c(c(n(n1)Cc2nnc(o2)SCc3cccc(c3)C(F)(F)F)C)Br KM04680 CCOC(=O)CSc1c2c(c(s1)C(=O)OCC)-c3ccccc3N(S2(=O)=O)C KM03304 COC(=O)C1=C(CSC1)NNc2ccccc2 KM04986 COC(=N)c1c(nccn1)SCc2ccc(cc2)F KM06397 CSc1nnc(s1)SCCS(=O)(=O)c2ccc(cc2)Cl KM06402 c1cc(cc(c1)C(F)(F)F)C(=O)/C(=C\Nc2cc(cc(n2)C(F)(F)F)C(F)(F)F)/C#N KM05022 CSc1c2c(c(s1)C(=O)/C(=N/Nc3ccc(cc3)Cl)/C#N)CCC=C2 KM05068 c1cc2c(c(c1)S(=O)(=O)NCC(=O)NNC(=O)c3ccc(cc3)Cl)nsn2 KM06430 CC(C)(C)c1cc2nc(cc(n2n1)Oc3ccccc3)C(F)(F)F KM08086 CC1(Cc2c(c(sc2C(=O)OC)SC)/C(=N/OC(=O)c3ccccc3Cl)/C1)C KM03493 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)Nc3ccc(cc3)Cl)C(F)(F)F KM08152 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2ccc(s2)C#CC(C)(C)O KM08026 c1cc(sc1)Sc2c(nccn2)C#N KM06344 CCOC(=O)C(=CNc1cc(nn1C)C)C(=O)OCC KM02169 CCCNC(=O)Nc1ccc(cc1)Cl KM09074 c1cc2c(c(c1)S(=O)(=O)Oc3ccc(cc3)Cl)nsn2 KM06363 c1ccc(cc1)c2c(c3ccccc3nn2)C(=O)O KM09072 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F KM06372 C([C@@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)NNC(=S)N)O)O)O)O JFD02100 COC(=O)[C@H](CCSC)NC(=O)c1cccnc1SC KM01866 CC(C)(C)S(=O)(=O)/C(=C/N1CCCCC1)/C#N KM01880 COc1ccc(cc1)Oc2c(nccn2)C#N KM07880 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)OC KM03328 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=O)Nc3ccc(cc3)Cl KM07953 Cc1ncc(c(n1)N)S(=O)(=O)C(C)(C)C KM02043 c1ccc(cc1)NC(=O)O/N=C(/c2c(nccn2)Sc3ccc(cc3)Cl)\N KM06435 Cc1cc(nc2c1ccc(n2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl)C KM01924 COc1c(cccn1)C(=O)Nc2ccccc2Cl KM01929 CNc1c(c(ncn1)Oc2cccc(c2)C(F)(F)F)[N+](=O)[O-] KM07929 c1ccc2c(c1)c(cc(n2)C(F)(F)F)O KM07594 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(on3)c4ccc(cc4)C(F)(F)F KM07775 CN1c2ccsc2C(=C(S1(=O)=O)C(=O)Nc3cccc(c3)Cl)O KM04688 c1ccc(c(c1)CSc2ccc(cc2)Cl)OCC(=O)NN KM04691 COc1cc(nc2c1csc2C(=O)NNC(=O)c3ccc(cc3)Cl)C(F)(F)F KM07935 c1cc(ccc1S(=O)(=O)c2cnc(nc2N)N3CCCC3)Cl KM00693 CCCn1c(=O)c(cn(c1=O)c2ccc(cc2)Cl)C#N KM09182 CC(C)Sc1c2c(c(s1)C(=O)C)CC(CC2=O)(C)C KM03320 CC(C)S(=O)(=O)c1cc(sc1)NC(=O)Nc2cccc(c2)Cl KM03321 CCOC(=O)c1cn(c2cc(nn2c1=O)C)Cc3cccc(c3)Cl KM07941 CCOC(=O)c1cn(c2cc(nn2c1=O)C)Cc3ccccc3 KM07947 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(c(cc3Cl)Cl)Cl DSHS00819 CCOC(=O)C(C(F)(F)F)(Nc1cccc(c1)Cl)NC(=O)c2ccccc2Cl JFD02205 COc1ccc(cc1OC2CCCC2)C(=O)O KM09079 CC(C)S(=O)(=O)c1cscc1NS(=O)(=O)c2ccc(cc2)Cl KM02172 c1ccc(cc1)c2cc3ccccc3nn2 KM09098 c1ccc(cc1)NC(=O)NNC(=O)CSCC(=O)Nc2ccc(cc2)OC(F)(F)F KM09102 CC(C)(C)S(=O)(=O)c1csc(c1N)C(=O)OC KM01882 c1cc(ccc1C(=O)N2CCSC2C(=O)O)Cl KM06336 CCO/C=C(\C#N)/S(=O)(=O)C(C)C KM01894 Cc1cc(nc2c1ccc(n2)N)C KM01901 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2c(cccc2Cl)Cl)/C#N KM00620 c1cc(ccc1SCC2C(=O)C3CCN2CC3)Cl KM07965 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccc(cc4)Cl KM07863 Cn1cc(c(n1)c2cccc(c2)NS(=O)(=O)c3ccc(cc3)Cl)Br KM02067 c1cc(ccc1C(=O)O/N=C(/c2c(nccn2)Sc3ccc(cc3)Cl)\N)Cl KM06439 c1cc(c(cc1Cl)Cl)SCC#N KM06445 CC(C)(C)c1cc2nc(c(c(n2n1)N)S(=O)(=O)c3ccc(cc3)Cl)SC KM02066 c1cc(ccc1NC(=O)c2cscc2Sc3ccc(cc3)Cl)OC(F)(F)F KM04953 COc1ccc(cc1)OC(=O)c2cscc2Sc3ccc(cc3)Cl KM04956 c1cc(ccc1Sc2cscc2C(=O)Oc3cc(cc(c3)Cl)Cl)Cl KM04957 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)c4ccc(cc4)Cl KM07785 c1ccc(cc1)C(=O)Nc2ccc(cc2)C3SCCS3 KM00706 CCCSc1c(c(c(s1)C(=O)OCC)c2ccc(cc2)OC(F)(F)F)C#N KM04961 c1cc(sc1S(=O)(=O)N)Cl KM01833 CCOC(=O)c1cn(c2cc(nn2c1=O)C)Cc3ccc(cc3Cl)Cl KM07948 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=O)Nc3ccccc3 KM07957 COc1cc(nc2c1csc2C(=O)NNC(=O)c3ccccc3)C(F)(F)F KM07960 Cn1cc(c(n1)c2cccc(c2)NC(=O)c3ccccc3Cl)Br KM02044 c1cc(ccc1NC(=O)O/N=C(/c2c(nccn2)Sc3ccc(cc3)Cl)\N)Cl KM06433 c1cc(cc(c1)Cl)NC(=O)O/N=C(/c2c(nccn2)Sc3ccc(cc3)Cl)\N KM06434 c1cc(ccc1NC(=O)CSCC(=O)NNC(=O)Nc2ccc(cc2)Cl)OC(F)(F)F KM09103 CC1(Cc2c(c(sc2C(=O)c3cccc(c3)[N+](=O)[O-])SC)C(=O)C1)C KM03365 CCOC(=O)c1c2c(c(s1)S(=O)C)C(=O)CCC2 KM03369 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)Nc3ccc(cc3)Cl)C)Br KM06357 c1cnc(c(n1)C#N)S(=O)(=O)CCO KM06360 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)Nc3cccc(c3)C(F)(F)F)C)Br KM06364 CS(=O)(=O)c1csc(c1Cl)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02084 COC(=O)C1=C(CSC1)Nc2ccc(cc2)Cl KM01966 COC(=O)c1c(c(cs1)S(=O)(=O)C)n2cccc2 KM01974 c1cc(sc1)/C=N/NC(=O)Cc2nc(no2)c3cnccn3 KM09180 COC(=O)C1=C(CSC1)Nc2cc(cc(c2)Cl)Cl KM01977 c1cc(ccc1CC2C(=O)NC(=N)S2)OC(F)(F)F KM09026 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=O)c2ccc(cc2)Cl KM09027 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)OC KM01986 COC(=O)c1c(c(cs1)C#N)n2cccc2 KM01988 CCOC(=O)CNS(=O)(=O)c1cccc2c1nsn2 KM06403 CN(C)/C=N/C(=O)c1c2c(c(s1)S(=O)(=O)C)C=CCC2 KM04995 CCOC(=O)NC(=O)/C(=C/Nc1ccsc1C(=O)OC)/C#N KM07961 CS(=O)(=O)c1csc(c1Cl)C(=O)O KM02078 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)Nc4cccc(c4)Cl KM07872 CCOC(=O)Cn1c(=O)ccc2c1nc(cc2C)C KM01961 Cc1c(c(sc1C(=O)OC)SC)c2ccn(n2)C(=O)c3ccc(cc3)Cl KM02062 CS(=O)(=O)c1c(c(cs1)c2ccc(cc2)Cl)C#N KM02064 CC(C)(C)/C=N/NC(=O)CNS(=O)(=O)c1cccc2c1nsn2 KM06447 CSc1c(c(n[nH]1)c2ccco2)C#N KM00801 CCOC(=O)c1c2c(c(s1)S(=O)(=O)Cc3ccccc3)C(=O)CC(C2)(C)C KM03370 c1ccc2c(c1)OCC(O2)C#N KM06484 C/S(=N/S(=O)(=O)c1ccccc1Cl)/c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06487 CS(=N/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl)(=O)c2ccc(cc2)Cl KM03379 c1ccc(cc1)N/N=C/c2ccc(cc2)[N+](=O)[O-] KM09080 CCCn1c(=O)cc(n(c1=O)c2ccc(cc2)Cl)N KM09082 c1ccnc(c1)CN/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00657 Cn1c(cc(n1)c2cccs2)N KM00835 c1ccc(cc1)C(=O)/C(=C/Nc2ccccn2)/C#N KM00838 Cc1ccc(cc1)S(=O)(=O)C(=C(SC)SC)C#N KM00848 c1ccnc(c1)S(=O)(=O)/C(=C/c2ccc(cc2)C=C(C#N)C#N)/C#N KM01994 c1cc(sc1)C(=O)C(=C2SCCCS2)C#N KM00823 C1CSC(=C(C#N)C(=O)C2CC2)SC1 KM00827 c1cc(ccc1NC(=O)NNC(=O)Cc2nc(no2)c3cnccn3)Cl KM09192 CSc1c2c(c(s1)C(=O)NNC(=O)c3ccc(cc3)Cl)CCC=C2 KM03462 c1ccc(cc1)S(=O)(=O)CCN2CCN(CC2)CCS(=O)(=O)c3ccccc3 KM00731 Cc1cc(=O)n2c([nH]1)cc(n2)c3ccc(cc3)C(C)(C)C KM00347 Cc1c(c(c2cc(ccc2n1)Br)C(=O)O)I KM00349 CCCS(=O)(=O)/C(=C/Nc1ncccn1)/C#N KM01942 CC(C)(C)S(=O)(=O)/C(=C/Nc1ncccn1)/C#N KM01950 CSc1c2c(c(s1)C(=O)Sc3ccc(cc3)Cl)CCC=C2 KM03427 CN1c2cc(ccc2C(=O)CS1(=O)=O)C(=O)OC KM05028 CC(C)S(=O)(=O)c1csc(c1N)C(=O)OC KM01952 Cc1ccc(cc1)N/C=C(\C#N)/C(=O)c2ccc(cc2)OC(F)(F)F KM04855 CC(C)(C)S(=O)(=O)C/C(=N/OC(=O)c1ccc(cc1)Cl)/N KM02092 CC(C)SC(=O)c1c(c(cs1)S(=O)(=O)C)Cl KM02094 CC(C)S(=O)(=O)/C(=C/Nc1ncccn1)/C#N KM01980 CC(C)(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)OC KM01983 CSc1c(c(n[nH]1)c2ccccc2Cl)C#N KM00816 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C(F)(F)F KM09165 CC(C)(C)c1cc2nc(nc(n2n1)N)SC KM00818 CC(C)(C)c1ccc(cc1)C(=O)C(=C2SCCCS2)C#N KM00820 CC(C)(C)S(=O)(=O)C/C(=N/OS(=O)(=O)c1ccc(cc1F)F)/N KM09171 CNC(=S)NNC(=O)Cc1nc(no1)c2cnccn2 KM09173 CC(C)(C)S(=O)(=O)/C(=C/N=S(=O)(C)c1ccccc1)/C#N KM03380 COC(=O)c1cccc(c1)NC(=O)NCc2ccccc2 KM09220 CSc1cccc(c1)NC(=O)N(Cc2ccccc2)C(=O)CC#N KM09226 c1ccc2c(c1)c(c(nn2)c3cccs3)C(=O)O KM09101 c1ccc(cc1)Sc2c(cc(s2)c3ccccn3)Br KM04920 CS(=N/C=C(\C#N)/C(=O)c1ccco1)(=O)c2ccc(cc2)Cl KM03368 CC(C)(C)c1ccc(cc1)C(=O)/C(=C/c2ccc(cc2)Cl)/C#N KM00717 c1cc(ccc1S(=O)(=O)/C(=C/N)/C#N)Cl KM00722 c1ccc(c(c1)C(=O)C(=C2SCCS2)C#N)Cl KM00861 c1ccc(cc1)C(=O)C(=C2SCCS2)C#N KM00864 c1cc(sc1)C(=O)C(=C2SCCS2)C#N KM00865 COCc1cc(=O)n2c([nH]1)cc(n2)c3cccc(c3)OC KM00734 CC(C)(C)c1cc2[nH]c(cc(=O)n2n1)COC KM00736 c1cc(ccc1c2nc(no2)c3cnccn3)Cl KM05037 c1cc(ccc1NC(=O)O/N=C(/c2cnccn2)\N)Cl KM05038 CSc1c2c(c(s1)C(=O)NNC(=O)Nc3ccccc3)CCC=C2 KM03478 CC(C)S(=O)(=O)c1cnc(nc1N)c2cnccn2 KM05054 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl KM04845 CN(c1ccsc1C(=O)OC)S(=O)(=O)C KM03314 CC(=O)c1c2c(c(s1)SCc3ccc(cc3)Cl)C(=O)CC(C2)(C)C KM03316 CSc1c(cn(n1)c2ccccc2)/C(=N/OC(=O)Nc3ccccc3)/N KM07782 CSc1c(cn(n1)c2ccccc2)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N KM07787 c1cc(ccc1SC2=C(CSC2)C(=O)O)Cl KM04862 CC(C)S(=O)(=O)c1cc(sc1)NC(=O)Nc2ccccc2Cl KM03324 CC(C)S(=O)(=O)c1cc(sc1)NC(=O)Nc2ccc(cc2)[N+](=O)[O-] KM03325 CSc1c(cn(n1)c2ccccc2)/C(=N/OC(=O)Nc3cccc(c3)Cl)/N KM07788 CSc1c(cn(n1)c2ccccc2)/C(=N/OC(=O)Nc3ccc(cc3)OC(F)(F)F)/N KM07789 CCOC(=O)Cn1c(=O)c(cn(c1=O)C(C)C)C#N KM07867 Cn1c2c(c(cc(n2)O)COC)c(n1)c3cccs3 KM00849 c1ccn2c(c1)ncc(c2=O)C(=O)c3cccs3 KM00851 Cc1cc2nc(c(c(n2n1)c3ccc(cc3)C(C)(C)C)C#N)SC KM00852 CSC(=C(C#N)S(=O)(=O)c1ccc(cc1)Cl)SC KM00853 c1cc(ccc1C2SCCS2)NC(=O)CSc3c(c(c(c(c3F)F)F)F)F KM00714 Cc1ccc2c(c1)c(ns2)C(=O)N KM09184 CC(=O)NC(=O)/C(=C/N1CCOCC1)/C#N KM09187 Cc1cc(nc2c1c(nn2C)C)OC(=O)N(C)C KM00829 c1ccnc(c1)c2ccc(s2)Sc3ccc(cc3)Cl KM05029 Cc1c(ncn1Cc2ccc(cc2)Cl)C(=O)NNC(=O)c3ccc(cc3)Cl KM05033 CC(C)(C)N1CC(OC1=O)CO BTB15174 CCOC(=O)c1cnc2c(c1Sc3cccc(c3)Cl)c(nn2C)C KM02180 Cc1ccc(cc1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM00927 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)Nc3ccc(cc3)OC)C)Br KM06365 CC1(Cc2c(c(sc2C(=O)OC)S(=O)C)C(=O)C1)C KM03375 CCOC(=O)c1c(c2c(s1)nccn2)N KM04925 CCCCOC(=O)c1c(c2c(csc2s1)C)C KM04929 COc1ccc(cc1OC)CCn2c(=O)c3ccccc3nn2 DP00914 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)Nc3ccc(cc3)C(C)C HR00033 CSc1c2c(c(s1)C(=O)/C(=C/Nc3ccc(cc3)Cl)/C#N)CCC=C2 KM05057 Cc1c(cnc(n1)c2cnccn2)S(=O)(=O)c3ccc(cc3)Cl KM05061 c1cc(ncc1C(F)(F)F)S(=O)(=O)c2ccc(s2)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl KM04972 c1cc(ccc1OC(F)(F)F)S(=O)(=O)CCN2CCCCC2 KM05013 CC1(Cc2c(c(sc2C(=O)OC)S(=O)(=O)C)C(=O)C1)C KM03357 CC1(Cc2c(c(sc2C(=O)c3ccc(cc3)Cl)SC)C(=O)C1)C KM03359 CSc1ccc(cc1)Oc2cccc(c2C#N)F KM06531 CC(C)(C)C(=O)CSc1nnc(n1C)CSCCOc2ccccc2 KM06539 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cccs4 KM07864 C/C=C/COc1ccccc1C(=O)N JFD01636 c1cc(cc(c1)Oc2c(nccn2)/C(=N/OC(=O)c3cccs3)/N)C(F)(F)F KM07869 c1cc(c(cc1N/C=C(\C#N)/C(=O)C2CC2)Cl)F KM01497 c1cc(ccc1C2SCCS2)NC(=O)CSc3c(c(cc(c3F)F)F)F KM00715 CCOC(=O)C1C(C(C(S1)c2ccc(cc2)Cl)C#N)(c3ccccc3)O KM00737 Cc1cc2nc(c(c(n2n1)c3ccco3)C#N)SC KM00872 CCC(C)N/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Br KM00755 CSc1c2c(c(s1)C(=O)Sc3ccc(cc3)C(F)(F)F)CCC=C2 KM03468 CSc1c2c(c(s1)C(=O)NNS(=O)(=O)c3ccccc3C(F)(F)F)CCCC2O KM03471 c1cc(oc1)c2c(sc3c2c(c(s3)C#N)N)C#N KM03472 CSc1c(c(nc(n1)c2cnccn2)c3ccccc3Cl)C#N KM05043 CSc1c(c(nc(n1)c2cnccn2)C3CC3)C#N KM05045 CSc1c2c(c(s1)C(=O)NNS(=O)(=O)C)CCC=C2 KM03480 c1ccc(cc1)C(=NOC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F)c4ccccc4 KM06368 c1cc(c(c(c1)Cl)Cl)C(=O)NNC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F KM06369 c1cc(sc1)C(=O)/C(=C/Nc2ncccn2)/C#N KM00935 CSc1nc(nc(n1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)C3CC3 KM00938 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=S)N=S(=O)(C)c3ccc(cc3)Cl KM04938 c1ccc(cc1)NC(=O)O/N=C(/c2c(nccn2)Oc3cccc(c3)C(F)(F)F)\N KM07855 COc1ccc(cc1)S(=O)(=O)NCCSc2cc(nc3c2cccc3)C(F)(F)F KM07833 c1ccc(cc1)C#Cc2cc(sc2)/C=C(\C#N)/C(=O)c3ccco3 KM08111 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)c3ccc(cc3)Cl)C(F)(F)F KM08113 CC(C)(C#Cc1ccc(cc1)/C=N/OC(=O)c2ccc(cc2)Cl)O KM08114 CCOC(=O)c1ccc(cc1)OCC#Cc2ccc(cn2)C(F)(F)F KM08118 c1ccc(cc1)/C=N/NC(=O)Cc2nc(no2)c3cnccn3 KM09179 c1cc(ccc1Cn2ccnc2COC(=O)Nc3ccc(cc3)OC(F)(F)F)Cl KM08024 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=S)NC KM07962 Cc1ccc(cc1)OC2=C(C(=O)c3ccccc3C2=O)Cl JFD00883 CCCS(=O)(=O)c1csc(c1n2cccc2)C(=O)OC KM01982 CSc1c(c(n(n1)c2c(cc(cc2Cl)Cl)Cl)N)S(=O)(=O)c3ccc(cc3)Cl KM01489 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)Nc2ccccc2SCCS(=O)(=O)c3ccc(cc3)Cl KM02010 COCc1cc(=O)n2c([nH]1)cc(n2)c3ccco3 KM00732 Cc1cc2[nH]c(cc(=O)n2n1)COC KM00739 COCc1cc(=O)n2c([nH]1)cc(n2)c3cccs3 KM00733 c1cc(c(cc1F)F)N/C=C(\C#N)/C(=O)C2CC2 KM01498 c1cc(ccc1S(=O)(=O)CCSCC(=O)Nc2cscc2S(=O)(=O)c3ccc(cc3)Cl)Cl KM03434 CCOC(=O)c1c2c(c(s1)S(=O)(=O)C)C(CCC2)O KM03445 Cc1cn(nc1c2ccccc2)C(=O)Nc3ccc(cc3)Cl CD09690 c1ccc(c(c1)/C=C(\C#N)/C(=O)c2ccc(cc2)OC(F)(F)F)Cl KM04979 CS(=O)(=O)c1c2c(c(s1)C(=O)N)CCC=C2 KM04981 c1cc(ccc1C(=O)NNC(=O)Cc2nc(no2)c3cnccn3)Cl KM09162 CSc1c2c(c(s1)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl)CCC=C2 KM03481 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)Oc3ccccc3 KM07943 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(=O)NNS(=O)(=O)c4ccc(cc4)Cl KM07937 COc1cc(nc2c1cc(cc2)C#CCOC(=O)c3cccs3)C(F)(F)F KM08005 CC(=O)c1ccc(s1)C#Cc2ccccc2 KM08029 c1cc(cc(c1)Cl)C(=O)NNC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F KM06377 c1cc2c(c(c1)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl)nsn2 KM06382 c1cc2c(c(c1)S(=O)(=O)Oc3ccc(cc3)[N+](=O)[O-])nsn2 KM06383 Cc1ccc(cc1)NS(=O)(=O)c2c(csc2C(=O)OC)C GK01445 COc1c(cc(cc1)/C=C\2/C(=O)/C(=C/c3cc(c(cc3)OC)OC)/CC2)OC DP00962 CCCS(=O)(=O)/C(=C/Nc1ccccn1)/C#N KM01920 c1cc(ccc1C(=O)NNC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F)Cl KM06373 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(=O)NNC(=O)c4ccc(cc4)Cl KM07882 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)NC(=O)Nc3ccccc3Cl)C)Br KM06411 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)NC(=O)Nc3ccc(cc3)Cl)C)Br KM06412 Cc1cc(=O)n2c([nH]1)cc(n2)C3CC3 KM00747 COc1ccc(cc1)/C=C(\C#N)/C(=O)C2CC2 KM00323 c1ccc(c(c1)/C=C(\C#N)/C(=O)C2CC2)Cl KM00324 c1ccc(cc1)/C=C(\C#N)/C(=O)C2CC2 KM00325 CCOC(=O)c1cn(c2cc(nn2c1=O)C)Cc3ccc(cc3)F KM07949 CCO/C=C(\C#N)/S(=O)(=O)Cc1ccco1 KM03326 CC1(Cc2c(c(sc2C(=O)/C=C/N(C)C)SCc3ccc(cc3)Cl)C(=O)C1)C KM03327 CC(=O)NC(=O)/C(=C/N1CCN(CC1)Cc2ccccc2)/C#N KM09186 CC(=O)NC(=O)/C(=C/Nc1ccc(cc1)OC)/C#N KM09189 CC(C)(C#Cc1ccc(cc1)/C=N/OC(=O)Nc2ccc(cc2)Cl)O KM08124 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)c3ccccc3)C(F)(F)F KM08128 CS(=N/C=C(\C#N)/C(=O)c1ccc(cc1)Cl)(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06547 c1ccc(cc1)C(=N)Nc2ccccc2 KM06550 c1cc2c(c(c1)NC(=O)CSc3ccc(cn3)C(F)(F)F)nsn2 KM06552 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)OC(F)(F)F)/C#N)Cl KM03571 c1cc(cc(c1)C(F)(F)F)C(=O)/C(=C/Nc2ccc3c(c2)OCCO3)/C#N KM05184 c1cc(cc(c1)S(=O)(=O)CCSc2c(cccn2)C(=O)Oc3ccc(cc3Cl)Cl)C(F)(F)F KM06295 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)N)C)Br KM06378 CCOC(=O)c1c(c(c(s1)SC)c2ccccc2)N KM03315 CS(=O)(=O)/C(=C/Nc1ncccn1)/C#N KM01943 CS(=NS(=O)(=O)c1cccc2c1nsn2)(=O)c3ccccc3 KM06395 Cc1ccc(cc1)S(=NS(=O)(=O)c2cccc3c2nsn3)(=O)C KM06396 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)c4ccc(cn4)C(F)(F)F)C(F)(F)F KM09137 CCOC(=O)N1CCC(CC1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM09139 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)CSCC(=O)Nc3ccccc3 KM09141 CCOC(=O)c1c[nH]c2cc(nn2c1=O)C KM02153 COC(=O)c1c(c(c(s1)SC)C#N)c2ccccc2Cl KM00902 c1ccnc(c1)CNC(=O)c2cccnc2SCCS(=O)(=O)c3cccc(c3)C(F)(F)F KM06288 c1cc(ccc1S(=O)(=O)CCNC2CCCCC2)Cl KM00328 c1cc(ccc1C(=O)O/N=C(/c2cnccn2)\N)Cl KM04980 Cc1csc(n1)c2c(c(c(s2)SC)c3ccnc(n3)S)C KM04984 CCOC(=O)c1c2c(c(s1)SC)C3(CCC2)SCCS3 KM04985 c1ccc(c(c1)C(=O)O/N=C(/c2c(nccn2)Oc3cccc(c3)C(F)(F)F)\N)Cl KM07870 c1ccc(cc1)COC(=O)N2CCNC(=O)C2 KM07871 CSc1nc2ccc(cc2s1)NC(=O)NC(=O)c3ccccc3[N+](=O)[O-] KM07549 Cn1c(nnc1SCc2ccccc2)Cc3nc(no3)c4cnccn4 KM09215 COC(=O)CSc1cc(nc2c1csc2C(=O)OC)C(F)(F)F KM07891 Cc1csc(n1)c2cn(c(=O)n(c2=O)CC(=O)NN)C(C)C KM07892 Cc1c(c2ccccc2[nH]1)SCc3nnc(n3C)S KM07963 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)/C=C(/S(=O)(=O)c3ccccc3)\C#N)/C#N KM02070 CSc1c(c(n2c(n1)cc(n2)C3CC3)N)S(=O)(=O)c4ccc(cc4)Cl KM02072 CNc1ccccc1C(=O)NCc2ccncc2 DP01706 COC(=O)c1c(ccs1)NN2C(=O)c3ccccc3C2=O GK01764 CC(C)S(=O)(=O)c1csc(c1N)C(=O)OCC(=O)c2ccccc2 KM02158 c1cc(cc(c1)S(=O)(=O)CCSc2c(cccn2)C(=O)Sc3ccc(cc3Cl)Cl)C(F)(F)F KM06298 c1ccc(cc1)NC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F KM06308 CC(C)(C)SC(=O)c1cccnc1SCCS(=O)(=O)c2cccc(c2)C(F)(F)F KM06317 Cc1cc2c(cc1C)CSC2 KM07654 c1ccc2c(c1)nc(o2)SCC(=O)N3CCC(CC3)n4cccc4 KM09108 Cc1ncc(c(n1)N)S(=O)(=O)c2ccc(cc2)Cl KM00671 c1cc(ccc1S(=O)(=O)c2cnc(nc2N)N)Cl KM00680 c1ccc(c(c1)N/N=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)Cl KM00691 c1ccc(c(c1)NS(=O)(=O)c2ccc(c(c2)Cl)Cl)SCCS(=O)(=O)c3ccc(cc3)Cl KM02007 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)C(=O)Nc4ccccc4)C(F)(F)F KM09152 CS(=O)(=O)CCSc1c(cccn1)C(=O)Sc2ccc(cc2Cl)Cl KM06301 CSc1nc(nc(n1)N)c2cnccn2 KM05093 Cc1csc(n1)c2c(c(c(s2)SC)c3cnc(nc3)SCc4cccc(c4)C(F)(F)F)C KM05095 c1ccc(cc1)C(=O)N2CCN(CC2)c3c(nccn3)C#N KM09033 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)c3nc(cs3)C(=O)NN KM07866 COC(=O)c1c(ccs1)Oc2c(nccn2)C#N KM07879 CCCCOc1cc(nc2c1cc(cc2)CS(=O)(=O)c3[nH]c4ccccc4n3)C(F)(F)F KM07524 CSc1nc2ccc(cc2s1)NC(=O)NC(=O)c3c(cccc3F)F KM07548 Cc1nc(nc(n1)SC)N/C=C(\C#N)/S(=O)(=O)C KM02014 c1cc(cc(c1)Oc2c(nccn2)c3nc(on3)c4cccs4)C(F)(F)F KM07888 CC1(CC(=O)C(=CNc2ccc(cc2F)F)C(=O)C1)C KM01519 c1ccc(c(c1)N)SCCS(=O)(=O)c2ccc(cc2)Cl KM02002 Cn1c(nnc1SCC(=O)c2ccc(c(c2)F)F)CSCC(=O)Nc3ccccc3 KM09143 CCOC(=O)N1CCC(CC1)N/C=C(\C#N)/S(=O)(=O)c2cccnc2 KM09144 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)C(=O)c4ccccc4)C(F)(F)F KM09148 CSc1c(c(cs1)c2ccc(cc2)Cl)C#N KM02006 COC(=O)c1ccc(o1)CS(=O)(=O)c2ccc(cn2)C(F)(F)F KM06279 CSc1nc2cc(nn2c(n1)N)C3CC3 KM00878 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/Nc2cccc(c2)C(F)(F)F KM00887 Cc1ccc(cc1)S(=O)(=O)C(=C2SCCS2)C#N KM00906 CCOC(=O)NC(=O)CC(=O)NC(=O)OCC KM07666 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Cc2cccs2 KM07670 c1ccc(cc1)c2c(c3ccccc3nn2)C(=O)Oc4ccccc4 KM09116 c1cc(ccc1C2SCCS2)NC(=O)c3ccc(cc3Cl)Cl KM00708 c1cc(ccc1/C=C(\C#N)/C(=O)C2CC2)Cl KM00709 c1ccc(cc1)NC(=S)NNC(=O)CSCC(=O)Nc2ccc(cc2)OC(F)(F)F KM09128 c1cc(ccc1S(=O)(=O)/C(=C/NC2CCCCC2)/C#N)Cl KM00758 c1cc(ccc1C#CCOC(=O)Nc2ccc(cc2)Cl)C#N KM09037 c1cc(ccc1C#CCOC(=O)c2ccc(cc2)Cl)C#N KM09039 c1cc(ccc1C#CCOC(=O)Nc2ccc(cc2)OC(F)(F)F)C#N KM09054 c1ccc(cc1)SCC(=O)N2CCC(CC2)n3cccc3 KM09057 c1cc(ccc1C#CCOC(=O)c2ccc(cc2)C(F)(F)F)C#N KM09060 Cc1csc(n1)c2c(c(c(s2)SC)c3ccnc(n3)SCC(=O)Nc4ccccc4Cl)C KM05109 c1ccc(c(c1)C(=O)Nc2ccccc2SCCS(=O)(=O)c3ccc(cc3)Cl)Cl KM02017 CN(C)/C=N/c1nc(nc2n1nc(c2)c3ccccc3)SC KM01559 c1ccnc(c1)S(=O)(=O)Cc2cccc(c2)/C(=N/O)/N KM01565 CSc1c(c(nc(n1)N)c2ccccc2Cl)C#N KM02061 c1cc(ccc1N/N=C(\C#N)/C(=O)C2CC2)F KM00380 c1ccnc(c1)S(=O)(=O)Cc2cccc(c2)/C(=N/OC(=O)c3ccc(cc3)Cl)/N KM01584 CC(C)(C)c1ccc(cc1)C(=O)/C=c\2/[nH]c(=O)/c(=C/c3ccccc3)/s2 KM00398 CC1(Cc2c(c(sc2C(=O)OC)SC)/C(=N/OC(=O)c3ccc(cc3)Cl)/C1)C KM03485 COC(=O)c1c(ccs1)Oc2cc(nc3c2csc3C(=O)OC)C(F)(F)F KM07950 CC(C)c1ncc(c(n1)N)S(=O)(=O)c2ccc(cn2)C(F)(F)F KM05160 CC(C)(C)c1ncc(c(n1)N)S(=O)(=O)c2ccc(cn2)C(F)(F)F KM05161 CC1(CCc2cc(ccc2O1)/C=C(\C#N)/S(=O)(=O)C)C KM05207 c1ccnc(c1)N/C=C(\C#N)/C(=O)c2ccco2 KM00843 Cc1csc2c1c(ncn2)SCC(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK02143 CSc1c-2c(c(s1)C#N)CCc3c2onc3 KM05180 c1ccc(cc1)S(=O)(=O)NNC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09420 c1ccc(cc1)C#Cc2ccc(cc2)/C=N\OC(=O)Nc3ccc(cc3)Cl KM08095 c1ccc(c(c1)C(=O)O/N=C(/c2c(nccn2)Sc3ccc(cc3)Cl)\N)Cl KM06440 CC(=O)O/N=C/1\CCCc2c1c(sc2C#N)SC KM03511 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)NNC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM02347 Cc1csc2c1c(c(s2)C(=O)Nc3ccc(cc3)Cl)C KM03513 C/C(=N\Nc1ccccc1C(F)(F)F)/c2ccc(s2)C#CC(C)(C)O KM08031 c1ccc(cc1)C#Cc2ccc(s2)c3ccn(n3)C(=O)c4ccccc4Cl KM08064 c1ccc(cc1)c2c(c3ccccc3nn2)C(=O)Oc4cccc(c4)C(F)(F)F KM09118 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)OCc2ccc(cc2)F JFD01410 c1ccc(cc1)CSc2nnc(o2)CSCCOc3ccc(cc3Cl)Cl KM06558 c1cc(oc1)CS(=O)(=O)/C(=C/NCc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM03334 c1cc(sc1)C(=O)/C(=C/Nc2cnccn2)/C#N KM04889 CSc1ncc(c(n1)N)S(=O)(=O)Cc2ccco2 KM03339 CCOC(=O)c1c2c(c(s1)SC)C(=O)/C(=C/N(C)C)/CC2 KM03344 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)CNS(=O)(=O)c2cccc3c2nsn3 KM06452 c1cnc(cn1)c2nc(on2)CC(=O)NNC(=O)Nc3cc(cc(c3)Cl)Cl KM09196 c1cc(ccc1NC(=O)NNC(=O)Cc2nc(no2)c3cnccn3)OC(F)(F)F KM09197 CC1(CCc2cc(ccc2O1)/C=N/C(=C(/C#N)\N)/C#N)C KM05242 Cc1cc(nc(n1)N/C=C(\C#N)/C(=O)c2ccoc2C)C KM06525 COC(=O)C1=C(CSC1)Nc2ccc3c(c2)OCCO3 KM05175 CCOC(=O)c1cnc2ccc(cc2c1O)OC(F)(F)F KM09296 CC(C)(C)c1cc2nc(cc(n2n1)Sc3ccc(cc3)Cl)C(F)(F)F KM08080 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/N2CCOCC2 KM01004 c1cc(ccc1C(=O)/C(=C/Nc2ccc3c(c2)OCCO3)/C#N)Cl KM05185 c1cc(ccc1NC(=O)Nc2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-])F GK02439 Cc1ccc(cc1)C(=O)/C=C\2/N(C(=O)C(=O)S2)c3ccccc3 JFD00371 CC(C)(C)C(=O)/C(=C/Nc1cccc2c1nsn2)/C#N KM06489 c1ccc2c(c1)OCC(O2)/C(=N\O)/N KM06490 C/C(=N\OCC(=O)O/N=C(/COc1ccc(cc1)OC)\N)/c2ccc(cc2)Cl KM06419 c1ccc(cc1)S(=O)(=O)NNC(=O)Cc2nc(no2)c3cnccn3 KM09190 Cc1nccc(n1)c2cccc(c2)N/N=C(\C#N)/S(=O)(=O)c3ccccc3 KM02266 CCOC(=O)c1cnc2c(c1Oc3cc(cc(c3)Cl)Cl)c(nn2C)C KM02367 c1ccc(cc1)CNC(=O)Nc2cccc(c2)Cl KM09303 c1ccc(cc1)CNC(=O)Nc2ccc(cc2)F KM09310 CC(C)(C)S(=O)(=O)/C(=C/Nc1ccc(cn1)Cl)/C#N KM02237 CC(=O)/C(=C\N=S(=O)(C)c1ccc(cc1)Cl)/S(=O)(=O)c2ccc(cc2)Cl KM05146 Cc1ccc(cc1)S(=N/C=C(\C(=O)C)/S(=O)(=O)c2ccc(cc2)Cl)(=O)C KM05147 CCCS(=O)(=O)C/C(=N/OC(=O)c1ccc(cc1)Cl)/N KM02252 CC(C)S(=O)(=O)C/C(=N/OC(=O)c1cc(cc(c1)Cl)Cl)/N KM02253 CNc1c(c(ncn1)NNC(=O)Nc2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] KM08041 c1cc(oc1)CS(=O)(=O)C(=C2SCCS2)C#N KM03348 c1ccnc(c1)c2ccc(s2)[N+](=O)[O-] KM04897 CCOC(=O)NC(=O)c1cn(c(=O)n(c1=O)Cc2ccccc2)C(C)C KM07810 CCOC(=O)c1c(c(c(s1)SCc2cccc(c2)Cl)S(=O)(=O)C(C)C)n3cccc3 KM03355 CCOC(=O)c1c(c(c(s1)SC)C#N)N KM03356 c1ccc2c(c1)C(CS2(=O)=O)Sc3ccc(cc3)Cl KM08109 CC(C)S(=O)(=O)c1c(csc1SC)NC(=O)Nc2cc(cc(c2)Cl)Cl KM09172 c1ccc(cc1)C(=O)NNC(=O)Cc2nc(no2)c3cnccn3 KM09175 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)Cc3nc(no3)c4cnccn4 KM09208 c1ccc2c(c1)CCN2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM05391 c1ccc2c(c1)CCN2/C=C(\C#N)/S(=O)(=O)Cc3ccco3 KM05392 c1ccc(cc1)C(=O)O/N=C/c2ccc3c(c2)CCO3 KM06698 c1ccc(c(c1)CS(=O)(=O)c2cccs2)F KM02354 CCOC(=O)c1cnc2c(c1Oc3ccc(cc3)OC)c(nn2C)C KM02360 CCOC(=O)c1cnc2c(c1Oc3ccc(cc3)F)c(nn2C)C KM02366 c1cc(ccc1N/N=C(\C#N)/C(=O)C2CC2)OC(F)(F)F KM03572 c1ccc(cc1)c2c(c3ccccc3nn2)C(=O)Oc4ccc(cc4)Cl KM09112 COC(=O)c1ccccc1SCC#N KM00945 Cn1ccnc1SCc2ccc(cc2)[N+](=O)[O-] JFD02045 c1ccc(cc1)C#Cc2ccc(s2)c3ccn(n3)C(=O)c4ccc(cc4)Cl KM08066 C/C(=N\OCC(=O)O/N=C(/COc1cccc(c1)Cl)\N)/c2ccc(cc2)Cl KM06420 C/C(=N\OCC(=O)O/N=C(/COc1ccc(cc1Cl)Cl)\N)/c2ccc(cc2)Cl KM06421 c1ccc(cc1)C#Cc2ccc(cc2)/C=C(\C#N)/C(=O)c3cccs3 KM08063 Cn1c(nnc1S)CSCCOc2ccccc2 KM06499 CCCn1c(=O)cc(n(c1=O)c2ccc(cc2)OC(F)(F)F)N KM09138 CC(C)(C)S(=O)(=O)C/C(=N/OS(=O)(=O)c1ccc(c(c1)Cl)Cl)/N KM02276 CC(C)S(=O)(=O)C/C(=N/OS(=O)(=O)c1ccc(cc1)Cl)/N KM02283 CN1c2ccccc2C(=O)/C(=C\N(C)C)/S1(=O)=O KM01114 c1cc(sc1)C2CC(CS2)C3SCCS3 KM05278 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2ccc(cn2)Cl)/C#N KM02208 CSc1c2c(c(s1)C(=O)N/N=C/c3cccs3)CCCC2O KM03405 CSc1c2c(c(s1)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)CCC=C2 KM03409 c1cc(ccc1C(F)(F)F)N/N=C(\C#N)/C(=O)C2CC2 KM02190 CC(C)S(=O)(=O)c1cscc1NC(=O)Nc2ccccc2 KM02191 CNC(=S)NCCSc1cc(nc2c1cccc2)C(F)(F)F KM07827 Cn1cc(c(n1)c2cccc(c2)NC3=C(CSC3)C(=O)OC)Br KM05171 c1cc(ncc1C(F)(F)F)S(=O)(=O)c2cnc(nc2N)N3CCOCC3 KM05172 COC(=O)c1cccc(c1)NC(=O)NC(=O)c2ccc(cc2)Cl DFP00285 CS(=O)(=O)c1cccc(c1)C(=O)O JFD01919 c1ccc(cc1)NC(=O)O/N=C(/CSc2cccs2)\N KM02380 c1cc(cc(c1)/C(=N/OC(=O)Nc2ccc(cc2)Cl)/N)CS(=O)(=O)c3cccs3 KM02384 CC(C)S(=O)(=O)c1csc(c1Cl)C(=O)N/N=C\c2ccccc2Cl KM02396 CNC(=S)NNC(=O)CCN(Cc1ccco1)S(=O)(=O)c2ccc(cc2)Cl KM09426 CC(C)(C)c1cc2nc(cc(n2n1)Oc3ccc(cc3)OC)C(F)(F)F KM08098 CCOC(=O)c1c(c(c(s1)SC)C(C)O)C KM03520 CCOC(=O)/C(=N/Nc1ccccc1Cl)/C KM09292 c1ccnc(c1)S(=O)(=O)/C(=C/c2ccc(cc2)C#N)/C#N KM01151 c1cc(ccc1C(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl KM01152 Cc1cc(nc(n1)N/C=C(\C#N)/S(=O)(=O)c2ccccn2)C KM01169 c1ccc(cc1)C#Cc2ccc(s2)c3ccn(n3)C(=O)c4cccs4 KM08067 COc1cccc(c1)/C=N/NC(=O)CSCC(=O)Nc2ccc(cc2)OC(F)(F)F KM09126 CS(=N)(=O)c1ccc(cc1)Oc2cccc(c2C#N)F KM06572 c1cc(ccc1c2cc3nc(cc(n3n2)C(F)(F)F)C(F)(F)F)Cl KM02247 c1ccc(cc1)NC(=O)NNc2cc(nc3c2cccc3)C(F)(F)F KM08025 Cn1c(nnc1SCC(=O)c2ccccc2)CSCC(=O)Nc3ccccc3 KM09140 COC(=O)CC(=O)NC(CSC(=O)Nc1ccc(cc1)OC(F)(F)F)C(=O)OC KM07983 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)C(=O)c4cccs4)C(F)(F)F KM09150 CN(C)c1nc(nc(n1)SC)N/C=C(\C#N)/S(=O)(=O)c2ccccc2Cl KM01071 Cc1cc(no1)NS(=O)(=O)c2ccc(s2)Cl KM01073 c1cc(cc(c1)Cl)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM01133 c1cc(cc(c1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F KM01134 CC(C)S(=O)(=O)c1c(csc1SC)NC(=O)c2ccc(cc2)Cl KM09265 CC(=O)Nc1ccc(cc1O)[N+](=O)[O-] KM09267 Cc1ccc(cc1)S(=O)(=O)NNC2CS(=O)(=O)c3c2cccc3 KM08164 Cc1nccc(n1)c2cccc(c2)NC(=O)c3ccccc3Cl KM02226 COC(=O)c1c(c(c(s1)SC)C#N)N KM02075 Cc1c(c(n(n1)CC(=O)N/N=C/c2c(cccc2Cl)F)C)Br KM01047 Cn1cncc1S(=O)(=O)/C(=C/c2ccccc2Sc3ccc(cc3)Cl)/C#N KM02231 CN(C)/C=C(\C#N)/S/C(=C/N(C)C)/C(=O)OC KM01860 CCO/C=C(\C#N)/S(=O)(=O)C(C)(C)C KM01862 CSc1ccc(cc1)OC(=O)c2ccc(cc2)Cl KM06328 c1cc(c(cc1Cl)Cl)OC(=O)c2ccc(o2)CS(=O)(=O)c3ccc(cn3)C(F)(F)F KM06325 CC(=O)O/N=C(/c1c(nccn1)Sc2ccc(cc2)Cl)\N KM06441 CSc1nnc(s1)Sc2c(nccn2)C#N KM06443 CN(C)c1ccc(cc1)/C=C(\C#N)/S(=O)(=O)c2cccs2 KM02272 c1ccc(c(c1)N/C=C(\C#N)/S(=O)(=O)c2ccccn2)Cl KM01178 Cc1ccc(cc1)SCc2nccn2Cc3ccc(cc3)Cl KM08043 c1cc(c(cc1F)F)N/N=C(\C#N)/C(=O)C2CC2 KM02188 CSc1c2c(c(s1)C(=O)Nc3ccc(cc3)Cl)CCC=C2 KM03398 c1ccc(cc1)C#Cc2ccc(s2)c3cc[nH]n3 KM08047 CCOC(=O)N1CCC(CC1)N/C=C(\C#N)/S(=O)(=O)C(C)C KM09151 CCOC(=O)C(=CNc1cc(cc(c1)Cl)Cl)C(=O)OCC KM09236 Cc1cc(n2c(n1)c(c(n2)SC)C#N)C KM02104 CCOC(=O)c1cnc2cc(cc(c2c1O)Cl)Cl KM09238 C/C(=N\O)/c1cccc(c1)Br KM09160 Cc1c(c2ccccc2[nH]1)SCc3nnc(n3C)SCC(=O)Nc4ccccc4 KM07994 c1ccnc(c1)S(=O)(=O)/C(=C/c2c(cccc2Cl)F)/C#N KM01144 Cc1cc(nc2c1c(nn2C)c3ccccc3)O KM01147 C/C(=N\O)/c1ccc(cc1Cl)Cl KM06478 CC1(Cc2c(c(sc2C(=O)OCc3ccccc3)SC)C(=O)C1)C KM03537 CCOC(=O)/C(=N/Nc1cc(cc(c1)Cl)Cl)/C(=O)C KM00961 Cn1c(=O)c(cn(c1=O)c2ccccc2)c3nc(on3)c4ccc(cc4)Cl KM08174 c1ccc(cc1)CSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-] KM08176 Cn1c(=O)c(cn(c1=O)c2ccccc2)/C(=N/OC(=O)c3ccccc3)/N KM08180 Cn1ccnc1S(=O)(=O)/C(=C/c2ccc(cc2)C(F)(F)F)/C#N KM02173 Cn1c(nnc1SCc2ccccc2)CSCC(=O)Nc3ccccc3 KM09090 Cn1c(nnc1SCc2ccc(cc2)Cl)CSCC(=O)Nc3ccccc3 KM09091 C/C(=N\OCC(=O)O)/c1cccs1 KM06352 CC(C)CC(C(=O)NC(CCSC)C(=O)OC)NC(=O)c1cccnc1SC KM01884 CC(C)(C)/C=N/N/C=C(\C#N)/S(=O)(=O)C(C)(C)C KM01892 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)OC)C)Br KM06349 c1cc(sc1)/C=C(\C#N)/S(=O)(=O)c2cccs2 KM02273 Cc1csc2c1c(c(s2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)C KM03489 C/C(=N/O)/c1c2c(c(s1)SC)/C(=N\O)/CC(C2)(C)C KM03490 CC(C)(C)C(=O)/C(=C/Nc1ccc(cn1)Cl)/C#N KM02215 c1ccc(cc1)NC(=O)C2CCN(CC2)c3ccc(cn3)C(F)(F)F KM08166 c1ccc(cc1)/C=N/CCN2CCN(CC2)C(=O)c3ccc(cc3)[N+](=O)[O-] KM08170 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/NC2CCCCC2 KM01022 Cc1nccc(n1)c2cccc(c2)NS(=O)(=O)c3ccccc3C(F)(F)F KM02220 c1ccc(c(c1)C(=O)ONC(=O)CS(=O)(=O)c2ccc(cc2)Cl)Cl KM02122 Cc1cc2nc(nc(n2n1)N/C=C(\C#N)/C(=O)c3cccs3)SC KM01031 c1cc(ccc1CS(=O)(=O)CC#N)Cl KM01033 COc1cc(nc2c1cc(cc2)C#CCOC(=O)Nc3ccccc3)C(F)(F)F KM08017 c1ccc(cc1)C2CCC(=O)/C(=C/Nc3ccc(cc3)Cl)/C2=O KM05254 CC(=O)c1c2c(c(s1)SCCOS(=O)(=O)c3ccc(cc3)Cl)C(=O)CC(C2)(C)C KM05257 CSc1c(c(nn1CNC(=O)Nc2ccccc2C(F)(F)F)c3cccs3)C#N KM00990 CCOC(=O)Cn1c(c(c(n1)C)Br)C KM00996 c1cc(sc1)SCC(=O)Nc2ccc(cc2)Cl KM02407 c1ccc(cc1)/C=N/NC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F KM09318 c1cc2c(cc1/C=N/O)CCO2 KM06460 c1cc(ccc1NC(=O)CSCC(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F)OC(F)(F)F KM09105 CS(=O)(=O)c1c2c(c(s1)C#N)CCCC2=O KM03363 CSc1c2c(c(s1)C(=O)c3ccc(cc3)Cl)CCCC2=O KM03364 c1cnc(c(n1)C#N)SCCO KM06355 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2ccccc2Cl)/C#N KM00623 CCOC(=O)Cc1c(c(cn1C)C)C(=O)OCC KM09062 c1ccc(cc1)N/N=C/c2cccs2 KM09075 CCOC(=O)CN/C(=C(/C#N)\C(=O)c1cccs1)/SC KM01130 c1cc(ccc1N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)Cl KM00949 Cc1ccc(c(c1)C)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00950 CC1(Cc2c(c(sc2C(=O)OCC=C)SC)C(=O)C1)C KM03542 CSc1nc2cc(nn2c(n1)N)c3ccccc3 KM00983 Cc1c(c(n(n1)CC(=O)N/N=C/c2ccccc2Cl)C)Br KM01048 CS(=O)(=O)c1csc(c1Cl)C(=O)Nc2cccc(c2)Cl KM02091 c1cc(ccc1S(=O)(=O)/C(=C/Nc2ccc(cn2)Cl)/C#N)Cl KM02234 c1ccc(cc1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00952 Cc1cc(nc(n1)C)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM01055 c1ccc(c(c1)C(=O)/C(=C\Nc2ccc3c(c2)OCCO3)/C#N)Cl KM05186 CSc1c2c(c(s1)C(=O)N/N=C/c3ccccc3)CCCC24SCCS4 KM05187 Cn1c(c(c(n1)c2cccs2)C#N)SC KM00885 CSc1c2c(c(s1)C(=O)NNC(=O)c3ccc(cc3)Cl)CCCC24SCCS4 KM05197 c1ccc(cc1)C2CCC(=O)/C(=C/Nc3cccnc3)/C2=O KM05270 Cn1c(nnc1SCC(=O)N=S(=O)(C)c2ccc(cc2)Cl)C(F)(F)F KM05271 c1cc(ccc1F)SCC(=O)O KM09206 Cn1c(nnc1SCc2ccc(cc2)Cl)Cc3nc(no3)c4cnccn4 KM09207 c1ccc(c(c1)NC=C2C(=O)CC(CC2=O)c3cccs3)Cl KM05149 c1cc(cc(c1)NC=C2C(=O)CC(CC2=O)c3cccs3)C(F)(F)F KM05150 COC(=O)c1c(ccs1)NC=C2C(=O)CC(CC2=O)c3cccs3 KM05168 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)c3cccc(c3)[N+](=O)[O-])C)C KM03554 COC(=O)c1cc(c(s1)SC)C(=O)N KM03556 CCOC(=O)c1c2c(c(s1)S(=O)C)C(=O)CC(C2)c3ccccc3 KM03609 c1ccc2c(c1)c(n[nH]c2=O)CSc3ccc(cc3)Cl KM09200 c1ccc(cc1)c2cc([nH]n2)NC(=O)Nc3ccccc3 KM09203 CCOC(=O)CS(=O)c1c2c(c(s1)C(=O)OCC)CCCC2=O KM03373 CS(=O)c1c2c(c(s1)C#N)CCCC2=O KM03374 COC(=O)CSCc1c2ccccc2c(=O)[nH]n1 KM09205 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)c4cc(nc5n4nc(c5)C(C)(C)C)C(F)(F)F)C(F)(F)F KM09073 c1cc(sc1)c2cc3ncc(c(n3n2)N)C#N KM00645 COC(=O)CSCC(=O)Nc1ccc(cc1)OC(F)(F)F KM09083 c1cc(ccc1NC(=O)CSCC(=O)NN)OC(F)(F)F KM09089 c1ccc(c(c1)/C=C(\C#N)/S(=O)(=O)c2ccccn2)Cl KM01142 C/C(=N\O)/c1ccc2c(c1)CCO2 KM06461 CSc1ccc(cc1)OS(=O)(=O)c2cc(cs2)S(=O)(=O)c3ccccc3 KM06465 COc1cc(nc2c1cc(cc2)C#CCOC(=O)c3ccc(cc3)Cl)C(F)(F)F KM08004 c1ccc(cc1)OC(=O)C2CCN(CC2)c3ccc(cn3)C(F)(F)F KM08181 Cn1c(=O)c(cn(c1=O)c2ccccc2)c3nc(on3)c4ccccc4 KM08190 CS(=O)(=O)/C(=N/Nc1ccc(cc1)OC(F)(F)F)/C#N KM03552 c1ccc(cc1)C(=O)c2cnc3ccccn3c2=O KM00845 CCOC(=O)/C(=N/Nc1c(csc1C(=O)OC)S(=O)(=O)Cc2ccco2)/C#N KM03451 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)C)C)C KM03524 CCOC(=O)c1c(c(c(s1)SC)C#N)c2cccs2 KM00897 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)/C=C(\C#N)/S(=O)(=O)c4cccs4)C(F)(F)F KM09164 CC1(Cc2c(c(sc2C(=O)OC)SCCOC(=O)Nc3ccccc3)C(=O)C1)C KM05212 CSC(=C(C#N)C(=O)c1ccc(cc1)Cl)SC KM01156 CC1CN=C(S1)N(c2ccccc2)C(=O)Nc3cccc(c3)Cl JFD02272 CCOC(=O)CN/C(=C(/C#N)\C(=O)c1ccc(cc1)Cl)/SC KM01160 c1cc(cc(c1)Cl)NC(=S)NC2CC3CC2C=C3 HR00097 c1ccc(cc1)OCCSCC(=O)NCc2ccncc2 KM06692 CSc1ccc(cc1)n2c(cc(=O)n(c2=O)Cc3ccccc3)N KM09348 COc1cccc(c1)n2c(cc(=O)n(c2=O)Cc3ccccc3)N KM09356 C/C(=N\OCc1cccc(c1)C(=O)OC)/c2ccc(c(c2)Cl)Cl KM06695 CSc1c(c(c(s1)C(=O)Nc2ccc(c(c2)Cl)F)c3ccc(cc3)Cl)C#N KM01207 CSc1c2c(c(s1)C#N)CCCC2O KM03378 CC(C)S(=O)(=O)c1c(csc1SC)NC(=O)Nc2ccc(cc2)OC(F)(F)F KM09227 CCOC(=O)c1c2c(c(s1)SC)C=CCC2 KM03381 CS(=N/C=C(\C#N)/S(=O)(=O)c1ccccn1)(=O)c2ccc(cc2)Cl KM03383 CC(=O)c1cc(c(s1)NC2CCCCC2)[N+](=O)[O-] KM03388 Cc1ccc(cc1)CSc2nnc(n2C)CSCC(=O)Nc3ccccc3 KM09092 Cc1cc(=O)n2c([nH]1)c(cn2)C#N KM00650 CS(=O)(=O)c1c2c(c(s1)C(=O)NC(=S)Nc3ccc(cc3)OC(F)(F)F)CCC=C2 KM04917 CSc1c2c(c(s1)C#N)CCCC2=O KM03362 COc1cc(nc2c1cc(cc2)C#CCOC(=O)c3ccccc3Cl)C(F)(F)F KM08007 C/S(=N/C(=O)c1ccc(cc1)Cl)/c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06471 CCOC(=O)c1c2c(c(s1)C#N)C(=O)CC(C2)(C)C KM05247 c1c(cc(cc1Cl)Cl)OS(=O)(=O)c2cc(sc2Cl)S(=O)(=O)Oc3cc(cc(c3)Cl)Cl KM05250 CC1(CCc2cc(ccc2O1)/C=N/NC(=O)c3ccc(cc3)Cl)C KM05265 CC1(CCc2cc(ccc2O1)/C=C(\C#N)/C(=O)c3cccc(c3)C(F)(F)F)C KM05194 CCOC(=O)c1c2c(c(s1)SCc3ccccc3)C(CC(C2)c4ccc(cc4)C)O KM03601 CCOC(=O)c1c(c(sc1NC=C2C(=O)CC(CC2=O)c3cccs3)C)C KM05170 Cc1c(c(sc1C(=O)O)SC)C=C KM03564 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)NN KM03565 CS(=O)(=O)Nc1ccc(cc1)Cl KM05166 COc1ccc(cc1)N/C=C(\C#N)/C(=O)c2c3c(c(s2)SC)C=CCC3 KM05059 CSc1c2c(c(s1)C(=O)NN)CCCC23SCCS3 KM05167 c1cc(nc(c1)COC(=O)Nc2ccc(cc2)Cl)COC(=O)Nc3ccc(cc3)Cl CD11603 CCOC(=O)/C(=N\Nc1ccc(cc1F)F)/C(=O)C KM00946 c1cc(sc1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F KM02365 Cc1ccc(cc1)S(=O)(=O)NCc2c(c(c(c(c2C)C)C)C)C DP01224 c1ccnc(c1)c2ccc(s2)Sc3cccc(c3)Cl KM05085 CC(=O)NNC(=O)c1c2c(c(s1)SC)C=CCC2 KM03463 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)c3cccs3)C(F)(F)F KM08129 CC1(Cc2c(c(sc2C(=O)OC)SC)/C(=N/OC(=O)Nc3ccccc3)/C1)C KM03498 C/C(=N\Nc1cc(ccc1Cl)C(F)(F)F)/c2ccc(s2)C#CC(C)(C)O KM08032 c1ccc2c(c1)c(cc(n2)C(F)(F)F)NNC(=O)Nc3ccc(cc3)Cl KM08033 c1cc2c(cc1OC(F)(F)F)cc([nH]2)C(=O)O KM09272 CC(C)S(=O)(=O)c1c(csc1SC)NS(=O)(=O)c2ccc(cc2)Cl KM09279 CNc1c(c(ncn1)NNC(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] KM08039 CC(=O)O/N=C/1\CC(Cc2c1c(sc2C(=O)OC)SC)(C)C KM03491 CSc1c(c(n2c(n1)c(c(n2)SC)C#N)c3ccc(cc3)Cl)C#N KM02182 COC(=O)C12CCCC(C1)(CCC2)C(=O)N BTB14980 c1cc(c(cc1)Cl)/C=C\2/C(=O)/C(=C/c3c(cccc3)Cl)/CCC2 DP00955 COC(=O)c1c(c(c(s1)SC)C#N)c2cccs2 KM00918 CS(=N/C=C(\C#N)/C(=O)c1cccs1)(=O)c2ccc(cc2)Cl KM03367 c1cc(ccc1NC(=O)c2cscc2Sc3ccc(cc3)Cl)Cl KM04919 CC(=O)c1cc(c(s1)SCCO)[N+](=O)[O-] KM03385 CC1(Cc2c(c(sc2Cl)S(=O)(=O)C)C(=O)C1)C KM04931 CC1(CCc2cc(ccc2O1)/C=N\NC(=O)c3cccc(c3Cl)Cl)C KM05266 c1ccc2c(c1)c(n[nH]c2=O)CSc3ccccn3 KM09201 Cc1csc2c1c(c(s2)C(=O)N=S(=O)(C)c3ccc(cc3)Cl)C KM03549 CC(C)OC(=O)c1c2c(c(s1)SC)C(=O)CC(C2)(C)C KM03550 CCOC(=O)c1c2c(c(s1)Sc3ccc(cn3)C(F)(F)F)C(=O)CC(C2)(C)C KM05274 Cc1c2c(c(sc2sc1C(=O)C)C(=O)O)C KM03566 CC1CCCCN1CCCNS(=O)(=O)c2ccc(s2)S(=O)(=O)c3ccc(cn3)C(F)(F)F KM05210 COc1ccc(cc1)NC=C2C(=O)CC(CC2=O)c3ccccc3 KM03614 Cc1ccc(cc1)NC(=O)O/N=C/c2ccc3c(c2)CCO3 KM06700 c1cc2c(c(c1)S(=O)(=O)N(CCC(=O)O)Cc3ccco3)nsn2 KM09364 c1cc(ccc1S(=O)(=O)n2c(c(cn2)C#N)C3CC3)Cl KM09368 Cc1ccc(cc1)OC(=O)c2c3ccccc3nnc2c4ccccc4 KM09117 c1cc(ccc1S(=O)(=O)/C(=C/Nc2ccc3c(c2)OCCO3)/C#N)Cl KM05176 c1cc(sc1)S(=O)(=O)/C(=C/Nc2ccc3c(c2)OCCO3)/C#N KM05177 c1ccc(cc1)C#Cc2ccc(cc2)/C=N/OC(=O)c3ccc(cc3)Cl KM08090 C/S(=N/C(=O)Nc1ccc(cc1)Cl)/c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06500 CC(C)(C)c1cc2nc(cc(n2n1)NNC(=O)c3ccc(cc3)Cl)C(F)(F)F KM07972 CC(C)(C)c1cc2nc(cc(n2n1)NNC(=O)c3ccccc3)C(F)(F)F KM07973 COc1ccc(cc1)S(=O)(=O)NNC(=O)c2c3c(c(s2)SC)C(CCC3)O KM03470 c1cc(sc1)S(=O)(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/C#N KM02309 Cc1csc2c1c(c(s2)/C=C(\C#N)/S(=O)(=O)C)C KM03486 CC(C)S(=O)(=O)c1csc(c1N)C(=O)OCC(=O)c2ccc(c(c2)Cl)Cl KM02159 c1ccc(cc1)CNC(=O)Nc2cccc(c2)F KM09311 CNc1c(c(ncn1)NNC(=O)Nc2cccc(c2)Cl)[N+](=O)[O-] KM08040 COC(=O)c1c(ccs1)n2cc(c(=O)n(c2=O)Cc3ccccc3)C#N KM08042 Cc1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccc(s3)C#Cc4ccccc4 KM08074 COc1cc2c(cc1OC)Cc3cc(c(cc3Cc4cc(c(cc4C2)OC)OC)OC)OC JFD01505 CC#N.Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=S)N=S(=O)(C)c3ccccc3 KM04933 CN(C(=O)c1ccc(cc1Cl)F)/N=C/c2c(cc(cn2)C(F)(F)F)Cl HC00077 c1cc(cc(c1)Oc2c(nccn2)/C(=N/OC(=O)Nc3ccc(cc3)OC(F)(F)F)/N)C(F)(F)F KM07857 CNc1ccccc1C(=O)NC2CCCCC2 DP01000 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC)Cc3nc(no3)c4cnccn4 KM09209 c1ccc(cc1)NC(=O)NNC(=O)Cc2nc(no2)c3cnccn3 KM09211 COc1ccc(cc1)/C=N/N=C(N)N JFD00735 CCOC(=O)NS(=O)(=O)c1ccc(s1)c2cc(n(n2)C)C(F)(F)F KM05155 CCSc1nnc(s1)S JFD02941 Cc1cccc(c1)NC(=O)O/N=C/c2ccc3c(c2)CCO3 KM06704 c1ccc2c(c1)c(cc(n2)C(F)(F)F)NNC(=O)Nc3cccc(c3)Cl KM08034 Cn1ccnc1SCc2nccn2Cc3ccc(cc3)Cl KM08037 c1cc(ccc1NC(=O)CSCC(=O)NNC(=S)Nc2ccc(cc2)Cl)OC(F)(F)F KM09129 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)C(=O)c4ccc(cc4)Cl)C(F)(F)F KM09132 CN(c1ccccc1)S(=O)(=O)C KM05145 c1cc(sc1)C2CC(=O)C(=CNc3ccc(cc3)Cl)C(=O)C2 KM05143 CC(C)(C#Cc1ccc(cc1)/C=N/Nc2ccc(cc2)I)O KM08105 Cc1c(c2ccccc2[nH]1)SCc3nnc(n3C)SCc4ccccc4 KM07990 CS/C(=C(/C#N)\C(=O)c1cccs1)/NCc2cccnc2 KM00909 c1c(ccc(c1)Cl)S(=O)(=O)/C(=C/NCCN/C=C(/S(=O)(=O)c2ccc(cc2)Cl)\C#N)/C#N KM01116 c1cc(ccc1N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)F KM01129 Cn1ccnc1S(=O)(=O)/C(=C/c2ccc3c(c2)OCO3)/C#N KM02176 CCOC(=O)c1cnc2c(c1Sc3ccc(cc3)Cl)c(nn2C)C KM02178 CSc1c(c(nc(n1)N2CCOCC2)c3ccccc3)C#N KM01155 c1cc(cc(c1)Cl)CS(=O)(=O)c2cccs2 KM02249 c1ccc(c(c1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)Sc3ccc(cc3)Cl KM02229 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCCN KM07807 CC(C)(C)c1cc2nc(cc(n2n1)Sc3ccccc3)C(F)(F)F KM08082 CN(C)/C=C/C(=O)c1ccc(cc1)Oc2ccc(cc2)OC CD11917 CS(=O)c1c2c(c(s1)Cl)CCCC2=O KM05073 c1ccc(cc1)S(=O)(=O)CCN2CCC(CC2)C(F)(F)F KM08085 CCN1c2ccc(c3c2c(ccc3)C1=O)NC(=O)c4ccccc4Cl JFD02491 CC(=O)CS(=O)(=O)c1ccc(cc1)Cl KM01166 CCOC(=O)/C(=N/Nc1ccc(cc1)C(F)(F)F)/C KM09294 C/C(=N\O)/c1ccc(s1)C#Cc2ccccc2 KM09300 c1ccc(cc1)CC(=O)NNC(=O)Cc2ccccc2 JFD00898 Cc1nccc(n1)c2cccc(c2)NC(=O)Nc3ccc(cc3)Cl KM02242 CSc1c2c(c(s1)C(=O)N/N=C/c3ccccc3Cl)CCCC2O KM03403 Cn1c(nnc1SCc2nccn2Cc3ccc(cc3)Cl)C(F)(F)F KM08036 c1ccc(cc1)C#Cc2ccc(cc2)/C=C(\C#N)/C(=O)c3ccc(cc3)Cl KM08071 c1ccc(cc1)C#Cc2ccc(s2)c3ccn(n3)S(=O)(=O)c4ccccc4 KM08073 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/CS(=O)(=O)C(C)(C)C)\N KM02274 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/N2CCCCC2 KM01009 CSc1c-2c(cs1)CCc3c2nc(nc3)SCc4cccc(c4)C(F)(F)F KM05106 c1cc2c(cc1/C=C(\C#N)/S(=O)(=O)c3ccc(cc3Cl)Cl)CCO2 KM06458 CCOC(=O)Cn1c(c(c(n1)c2cccs2)C#N)SC KM00915 CCOC(=O)c1cc2cc(ccc2[nH]1)OC(F)(F)F KM09260 Cc1ccc(cc1)C(=O)Nc2csc(c2S(=O)(=O)C(C)C)SC KM09264 CS(=NS(=O)(=O)c1cccc2c1non2)(=O)c3ccc(cc3)Cl KM06585 c1cc(sc1)SCc2ccc(cc2)[N+](=O)[O-] KM02263 c1ccc(cc1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM01007 CSc1c(c(nc(n1)c2cccnc2)c3ccccc3)C#N KM00962 COC(=O)c1c(c(cs1)S(=O)(=O)c2ccc(cc2)Cl)N KM00975 CCOC(=O)c1cnc(nc1C(F)(F)F)O GK01680 Cc1c(c(n(n1)Cc2nnc(o2)SCC(=O)c3ccc(cc3)Cl)C)Br KM04719 Cc1c(c(n(n1)Cc2nnc(o2)SCC(=O)C(C)(C)C)C)Br KM04721 c1cc(c(cc1Cl)Cl)S(=O)(=O)N=S2CCN(CC2)c3c(ccs3)[N+](=O)[O-] KM06290 CS(=O)(=O)CCSc1c(cccn1)C(=O)NCc2cccs2 KM06292 c1cc(ccc1Sc2c(nccn2)C#N)Cl KM06379 CC(C)S(=O)(=O)/C(=C/Nc1cccnc1)/C#N KM01925 CC(C)(C)S(=O)(=O)/C(=C/Nc1ccccn1)/C#N KM01926 COc1c(cccn1)C(=O)Nc2ccc(cc2F)F KM01927 c1cc2c(c(c1)S(=O)(=O)Nc3ccc(cc3)OC(F)(F)F)nsn2 KM06385 CSc1c2c(c(s1)C(=O)NNC(=O)Nc3ccc(cc3)Cl)CCCC2O KM03467 Cc1cc(n2c(n1)cc(n2)c3ccc(cc3)C(C)(C)C)C(F)(F)F KM02307 c1cc(ccc1c2c(sc3c2c(c(s3)C#N)N)C#N)Cl KM03474 c1cc(sc1)S(=O)(=O)/C(=N/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM02308 Cc1c2c(c(sc2sc1Br)Br)C KM03514 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl KM02333 CS(=N/C=C(\C#N)/S(=O)(=O)c1cccs1)(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06560 c1ccc2c(c1)OCC(O2)/C(=N\OC(=O)c3ccc(cc3Cl)Cl)/N KM06563 CS(=O)c1ccc(cc1)Oc2cccc(c2C#N)F KM06567 Cc1nccc(n1)c2cccc(c2)NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM02221 c1ccc(c(c1)/C=C(\C#N)/S(=O)(=O)c2ccccn2)Sc3ccc(cc3)Cl KM02224 Cc1nccc(n1)c2cccc(c2)NC(=O)NC KM02244 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)C(=O)c4ccc(cc4)C(F)(F)F)C(F)(F)F KM09149 Cc1csc(n1)c2c(c(c(s2)SC)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl)C KM05107 CC(C)S(=O)(=O)c1cscc1NC(=O)c2ccc(cc2)Cl KM02133 c1cc(ccc1CS(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl KM01083 C/S(=N/S(=O)(=O)c1ccc(cc1)Cl)/c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06470 c1ccc(c(c1)C(=O)/C(=C/Nc2ncccn2)/C#N)Cl KM00939 Cc1csc2c1c(c(s2)C(=O)N3CCOCC3)C KM03532 c1cc2c(c(c1)S(=O)(=O)N(CC/C(=N/O)/N)Cc3ccco3)nsn2 KM09339 C1CN2CCC1C(C2)(C#N)O KM09340 Cc1c(c(n(n1)S(=O)(=O)c2ccc(s2)Cl)C)[N+](=O)[O-] KM01040 CSC(=C(C#N)C(=O)C1CC1)SC KM01000 c1cc(ccc1/C=N/NC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F)Cl KM09319 CC(=NOC(=O)c1ccc(o1)CSc2ccc(cn2)C(F)(F)F)C KM06314 COC(=O)CSc1cc(nc2c1cccc2)C(F)(F)F KM07633 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCC(=O)NN KM07636 c1ccc(cc1)S(=O)(=O)CCN2CCC(CC2)C(=O)N KM07646 c1cc(ccc1C2SCCS2)N.Cl KM00666 Cn1c(nnc1S)CSC2CN(C2)C(c3ccccc3)c4ccccc4 KM09109 CCCNC(=O)Nc1ccc(cc1)OC(F)(F)F KM09113 c1ccc(cc1)c2c(c3ccccc3nn2)C(=O)Nc4ccc(cc4)OC(F)(F)F KM09111 COc1cc(cc(c1)OC)NC(=O)c2c3ccccc3nnc2c4ccccc4 KM09120 Cc1c(c(n(n1)CC#N)C)Br KM01157 Cn1ccnc1S(=O)(=O)/C(=C/c2ccccc2Cl)/C#N KM02168 c1cc(cc(c1)F)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM01131 CCCS(=O)(=O)C/C(=N/OC(=O)c1ccccc1Cl)/N KM02254 COc1ccc(cc1)NC(=O)O/N=C(\C2COc3ccccc3O2)/N KM06578 c1ccc2c(c1)OCC(O2)/C(=N\OC(=O)Nc3cccc(c3)C(F)(F)F)/N KM06580 Cc1ccc(cc1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00951 c1ccc2c(c1)OCC(O2)/C(=N\OC(=O)Nc3ccc(cc3Cl)Cl)/N KM06591 c1ccc(cc1)CNC(=O)Nc2cccc(c2)Br KM09326 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC(F)(F)F)CSCC(=O)Nc3ccccc3 KM09156 CC(C)S(=O)(=O)C/C(=N/OC(=O)Nc1ccc(cc1)Cl)/N KM02261 Cc1csc2c1c(c(s2)/C=C(\C#N)/C(=O)c3ccc(cc3)Cl)C KM03495 Cn1c(nnc1SCC(=O)Nc2cccc(c2)Cl)CSCC(=O)Nc3ccccc3 KM09158 Cc1ccc(cc1)S(=NS(=O)(=O)c2ccc(cc2Cl)Cl)(=O)C KM05123 c1cc(ccc1S(=O)(=O)C(=C2SCCS2)C#N)Cl KM00889 CC1(CCc2cc(ccc2O1)/C=N/OC(=O)c3cccc(c3)Cl)C KM05220 Cn1c(nnc1S)Cc2nc(no2)c3cnccn3 KM09194 CS(=N/C=C(\C#N)/S(=O)(=O)c1ccc(cn1)C(F)(F)F)(=O)c2ccc(cc2)Cl KM05136 CC(C)/N=N/NC(=O)c1c2c(c(s1)SC)C(CCC2)O KM03543 CC1(Cc2c(c(sc2C(=O)Oc3ccccc3)SC)C(=O)C1)C KM03544 c1cc2c(c(c1)S(=O)(=O)N(CC/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N)Cc4ccco4)nsn2 KM09371 c1ccc(cc1)CSc2c3c(c(s2)C#N)CC(CC3=O)c4ccccc4 KM03584 c1ccc(cc1)C2CC(=O)C(=CNc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)C2 KM03611 c1cc(ncc1C(F)(F)F)S(=O)(=O)Cc2ccc(o2)C(=O)N3CCOCC3 KM06322 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4ccc(c(c4)OC)OC KM07663 CCOC(=O)c1c(n2c(c(c(n2)C)Br)nn1)C KM07668 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3c(nccn3)C#N KM09034 c1cc(ccc1N/N=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)F KM00694 c1ccc(c(c1)C(=O)Nc2ccc(cc2)C3SCCS3)F KM00699 CCOC(=O)C1C(C(C(S1)c2ccccc2)C#N)(c3ccccc3)O KM00702 c1ccc(c(c1)C(=O)Nc2ccc(cc2)C3SCCS3)Cl KM00707 CC(C)c1ccc(cc1)NC(=O)c2c3ccccc3nnc2c4ccccc4 KM09121 COc1ccc(cc1)NC(=S)NNC(=O)CSCC(=O)Nc2ccc(cc2)OC(F)(F)F KM09130 COc1ccc(cc1)N/N=C(\C#N)/C(=O)C2CC2 KM02186 c1cc(cc(c1)F)N/N=C(\C#N)/C(=O)C2CC2 KM02187 CC(=O)NC(=O)c1cnn(c1N)c2ccccc2 KM09240 c1c(cc(c2c1ncc(c2O)C(=O)O)Cl)Cl KM09246 CSc1c(c(nc(n1)N2CCCC2)c3ccco3)C#N KM01143 CN(C)/C=C(\C#N)/C(=O)C1CC1 KM09329 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/NCc2ccco2 KM01012 CS/C(=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl)/NCc2cccs2 KM01015 c1cc(ccc1c2nc3c(c(n2)O)CSC3)Cl KM02403 CC(C)S(=O)(=O)c1csc(c1I)C(=O)OC KM02095 Cc1c2c(c(sc2sc1C(=O)O)C(=O)O)C KM03433 Cc1csc2c1c(c(s2)COC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C KM03505 CSc1c\2c(c(s1)C#N)CCC/C2=N\OC(=O)c3ccc(cc3)Cl KM03509 CSc1c\2c(c(s1)C#N)CCC/C2=N\OC(=O)c3ccccc3Cl KM03510 C#Cc1cccc(c1)NC(=O)c2ccccc2 KM08013 CC1(Cc2c(sc(c2C(=O)C1)C#N)C#N)C KM05233 c1cc(ccc1/C=N/NC(=O)Cc2nc(no2)c3cnccn3)Cl KM09166 C/C(=N\O)/c1ccccc1Cl KM09168 CC(C)(C)OC(=O)C1CNC(=O)N1C(=O)OCc2ccccc2 KM09170 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=O)c2cccc(c2)Cl DFP00234 Cc1c(c(sc1C(=O)OC)SC)c2ccno2 KM05165 CC(=O)c1cc2cc(ccc2o1)Cl DP02005 c1ccc(cc1)C2CC(=O)C(=CNc3ccc(cc3)Cl)C(=O)C2 KM03612 Cn1c(c(c(n1)c2ccc(cc2)Cl)C(=O)NC(=O)OCC#C)SC KM01208 c1cc(ccc1C#CCO)C#N KM09036 c1ccnc(c1)S(=O)(=O)Cc2cccc(c2)/C(=N\OC(=O)Nc3ccc(cc3)Cl)/N KM01602 CS/C(=C(\C#N)/C(=O)C1CC1)/N2CCOCC2 KM01608 c1cc(ccc1N2C(=O)C3N(C2=O)CCS3)OC(F)(F)F KM09043 c1ccc(cc1)CN2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccccn3 KM09049 c1ccc(c(c1)C(F)(F)F)NC(=S)NNC(=O)CSCC(=O)Nc2ccc(cc2)OC(F)(F)F KM09131 CSc1c(c(nc(n1)c2cccnc2)c3ccc(cc3)OC(F)(F)F)C#N KM04942 CSc1c(c(n(n1)c2ccccc2)c3ccc(cc3)OC(F)(F)F)C#N KM04945 c1cc(ccc1N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)OC(F)(F)F)Cl KM04950 CSc1c(c(nn1CC(=O)NN)c2ccccc2)C#N KM00931 CSc1c(c(nn1CC(=O)N/N=C/c2c(cccc2Cl)F)c3cccs3)C#N KM00933 CCOC(=O)CSc1c(c(c(s1)C(=O)OCC)C)C#N KM03531 c1cc2c(c(c1)S(=O)(=O)NCC(=O)NNS(=O)(=O)c3ccc(cc3)Cl)nsn2 KM06481 CSc1ccc(cc1)NC(=O)N(Cc2ccccc2)C(=O)CC#N KM09345 c1ccc(cc1)NC(=O)O/N=C(/CCN(Cc2ccco2)S(=O)(=O)c3cccc4c3nsn4)\N KM09365 CCOC(=O)c1c(c(c(s1)SC)S(=O)(=O)C)N KM09366 CC1(CCc2cc(ccc2O1)/C=N/O)C KM05202 CSc1c2c(c(s1)C(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F)CCCC24SCCS4 KM05203 CC1c2ccsc2CCN1C(=S)NC(=O)c3ccc(cc3)Cl DFP00275 CSc1c2c(c(s1)C(=O)Sc3c(cc(cc3Cl)Cl)Cl)CCC=C2 KM03455 CSc1c2c(c(s1)C(=O)/C(=N/Nc3ccccc3Cl)/C#N)CCC=C2 KM05069 Cn1c(nnc1SCC(=O)Nc2ccccc2)Cc3nc(no3)c4cnccn4 KM09202 c1cc(cc(c1)C#N)CS(=O)(=O)c2cccs2 KM02374 COC(=O)c1cccc(c1)NC(=O)N KM09276 CC(C)S(=O)(=O)c1cscc1N2C(=O)c3ccccc3C2=O KM05378 CC1(Cc2c(sc(c2C(=O)C1)SCCOC(=O)Nc3cccc(c3)Cl)C#N)C KM05382 Cn1c(=O)c(cn(c1=O)c2ccccc2)C(=S)N KM08159 c1cc(ccc1S(=O)(=O)/C(=N/Nc2cc(cc(c2)Cl)Cl)/C#N)Cl KM01217 c1ccnc(c1)c2ccc(s2)C(=O)Oc3cc(cc(c3)Cl)Cl KM02567 CC(C)S(=O)(=O)c1csc(c1N/N=C(\C#N)/C(=O)c2cccs2)C(=O)OC KM02573 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NNC(=O)Nc3ccc(cc3)Cl KM03722 c1ccc(cc1)C#Cc2ccc(cc2)C#N KM08057 CC(C)(C#Cc1ccc(cc1)C#N)O KM08059 c1ccc(cc1)N2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccccn3 KM09050 Cn1c(nnc1S)CSCC(=O)Nc2ccccc2 KM09058 CCOC(=O)c1c(c(c(s1)SCc2ccc(cc2)Cl)S(=O)(=O)C(C)C)N KM03330 CC(=NNC(=O)c1c2c(c(s1)SC)C(CCC2)O)C KM03402 CSc1c2c(c(s1)C(=O)N/N=C/c3ccc(cc3)Cl)CCCC2O KM03404 c1cc(ccc1OC(=O)c2cscc2Sc3ccc(cc3)Cl)Cl KM04955 CN(C)S(=O)(=O)c1cc(sc1Cl)S(=O)(=O)N(C)C KM05230 Cc1cc(cc(c1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)C KM00947 CN1c2ccsc2C(=O)/C(=C\N=S(=O)(C)c3ccc(cc3)Cl)/S1(=O)=O KM05130 CC1(Cc2c(c(sc2C(=O)OC3CCCCC3)SC)C(=O)C1)C KM03541 c1ccc(cc1)C(=O)CSc2nnnn2c3ccccc3 JFD01898 CC(=O)/C(=C\N=S(=O)(C)c1ccccc1)/S(=O)(=O)c2ccc(cc2)Cl KM05148 CCOC(=O)c1cnc(nc1C(F)(F)F)SCc2ccc(cc2)C GK03010 CCOC(=O)c1cnc(nc1C(F)(F)F)SCc2c(cc(cc2C)C)C GK03011 CSc1c-2c(c(s1)C(=O)NC(=O)Nc3ccc(cc3)Cl)CCc4c2onc4 KM05396 Cn1c(cc(n1)c2ccc(s2)/C=C(\C#N)/S(=O)(=O)C)C(F)(F)F KM05314 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)Br GK03006 Cn1c(cc(n1)c2ccc(s2)/C=C(\C#N)/C(=O)c3ccccc3)C(F)(F)F KM05316 c1cc(cnc1)CN/C=C(\C#N)/S(=O)(=O)Cc2ccc(cc2)Cl KM01096 Cn1c(cc(n1)c2ccc(s2)/C=C(\C#N)/C(=O)c3ccco3)C(F)(F)F KM05318 CC(C)S(=O)(=O)c1cscc1NC(=O)c2ccc(s2)c3cc(nn3C)C(F)(F)F KM05325 CSc1c(c(c(s1)C(=O)O)c2cccs2)C#N KM01102 COc1ccc(cc1)C2Cc3c(sc(c3C(=O)C2)SCc4ccccc4)C#N KM03653 Cc1c(sc(c1c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl)SC)C#N KM03666 c1ccc(cc1)NC(=O)CN2c3cc(ccc3SCC2=O)C(F)(F)F KM08274 Cc1c(sc(c1C(=O)C)SC)C#N KM03563 CCOC(=O)c1c2c(c(s1)SCc3ccccc3)C(=O)CC(C2)c4ccccc4 KM03568 CC(C)S(=O)(=O)c1cc(sc1S(=O)C)C(=O)OC KM03573 CC(C)(C)S(=O)(=O)/C(=C/Nc1ccc(cc1)OC(F)(F)F)/C#N KM03575 CN(C)/C=C/C(=O)c1c(c(c(s1)SC)C#N)c2ccccc2 KM05330 CCOC(=O)c1c2c(c(s1)SC)-c3c(cno3)CC2 KM05333 CC(=O)N1CCc2c1cccc2 KM05451 C/C(=N\OCc1nc(no1)c2cccc(c2)Cl)/c3ccc(cc3)Cl KM06423 c1ccc(cc1)C#Cc2ccc(cc2)/C=C(\C#N)/C(=O)c3ccco3 KM08070 Cc1c(cco1)C(=O)C(=C(SC)SC)C#N KM06512 Cn1c(nnc1S)CSCCOc2ccc(cc2Cl)Cl KM06513 Cc1c(c(=O)n(n1C)c2ccccc2)/C=N/C(=C(/C#N)\N)/C#N KM03645 CCOC(=O)c1c2c(c(s1)SCc3ccccc3)C(=O)CC(C2)c4ccc(cc4)OC KM03647 Cc1csc2c1c(c(s2)C(=O)OC)C KM03654 c1cc(sc1)/C=N/NC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F KM09320 COc1cccc(c1)NC(=O)NCc2ccccc2 KM09325 Cc1cc(n(n1)c2ncc(c(n2)N)S(=O)(=O)C(C)(C)C)C KM05400 CC(C)(C)c1ccc(cc1)C(=O)OCc2ccc(s2)C#Cc3ccccc3 KM08266 c1cc(c(c(c1)Cl)CN2c3cc(ccc3SCC2=O)C(F)(F)F)Cl KM08276 Cc1ccc(cc1)S(=NC(=O)CSc2ccc(cc2)Cl)(=O)C KM05321 CC1(Cc2c(sc(c2C(=O)C1)SCCO)C#N)C KM05322 CCCS(=O)(=O)c1cscc1NC(=O)c2ccc(s2)c3cc(nn3C)C(F)(F)F KM05324 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2Cl)Cl GK03023 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)F GK03024 CCOC(=O)c1c2c(c(s1)SCCO)C(=O)CC(C2)(C)C KM05217 c1cc(ccc1Sc2c(ccs2)[N+](=O)[O-])Cl KM05336 c1cc(sc1/C=N/O)Br KM08194 CCCCCCSc1nnc(s1)S JFD02940 CN(C)C=O.c1ccc2c(c1)c(c(s2)C(=O)Nc3nnc(s3)Sc4ccnc5c4ccc(c5)Cl)Cl RH00427 c1cc(ccc1NC(=O)CN2c3cc(ccc3SCC2=O)C(F)(F)F)Cl KM08292 COC(=O)c1c(c(cs1)C#N)NN=C(C#N)C#N KM02513 CS(=O)c1c(c(on1)c2ccc(cc2)Cl)C#N KM02520 c1cc(ccc1C(CC(=O)O)N)Cl KM08205 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)/C=C(\C#N)/S(=O)(=O)c4ccccc4 KM08206 CC(C)(C)c1csc(n1)c2cn(c(=O)n(c2=O)C)c3ccccc3 KM08224 CCOC(=O)N1CCC(CC1)N/C=C(\C(=O)C)/S(=O)(=O)c2ccc(cc2)Cl KM09145 Cc1c(c2ccccc2[nH]1)SCc3nnc(n3C)SCc4ccc(cc4)Cl KM07991 Cn1c(nnc1SCc2ccc(cc2Cl)Cl)CSCCOc3ccc(cc3Cl)Cl KM06521 C/C(=N\OCc1ccc(o1)C(=O)N2CCOCC2)/c3ccc(cc3Cl)Cl KM06522 CC(=O)NC(=O)/C(=C/Nc1ccc(c(c1)Cl)F)/C#N KM09231 Cc1csc(n1)c2cc(sc2SC)C(=O)NN KM03663 COC(=O)c1c(ccs1)N/N=C(\C#N)/C(=O)c2ccco2 KM03675 CC(=O)OCc1ccc(o1)/C=C(\C#N)/S(=O)(=O)C KM03560 CCOC(=O)c1c(c(c(s1)S(=O)(=O)C)C=C)C KM03561 CC(C)S(=O)(=O)c1cc(sc1S(=O)(=O)C)C(=O)OC KM03562 c1cc(sc1)S(=O)(=O)c2cccs2 KM05454 c1ccc(cc1)C#Cc2ccc(s2)/C=C(\C#N)/C(=O)c3ccco3 KM08200 c1cc(sc1)S(=N)(=O)c2ccc(cc2)Cl KM05456 c1cc(sc1)Sc2c(cc(cn2)C(F)(F)F)Cl KM05458 CCOC(=O)c1c2c(c(s1)S(=O)C)-c3c(cno3)CC2 KM05465 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4ccc(s4)Br KM08209 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)/C=C(\C#N)/S(=O)(=O)c4ccc(cc4)Cl KM08208 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4ccc(s4)Cl KM08212 CC(C)(C)OC(=O)N1CCN(CC1)CCNC(=O)Nc2ccc(cc2)Cl KM08230 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4cc(cc(c4)Cl)Cl KM08243 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccc(cc4)OC(F)(F)F KM08244 CC(C)(C)OC(=O)N1CCN(CC1)CCNC(=O)c2ccccc2 KM08250 c1ccc(c(c1)C(=O)NCCCn2ccnc2)NC(=O)c3ccc(o3)[N+](=O)[O-] BTB05615 CCOC(=O)/C(=N/Nc1c(csc1C(=O)OC)C#N)/C#N KM02523 c1ccnc(c1)c2ccc(s2)C(=O)N3CCCCC3 KM02527 c1cc2c(c(c1)S(=O)(=O)Nc3ccc(cc3)Cl)non2 KM06557 Cn1c(=O)c(cn(c1=O)c2ccccc2)c3nc(cs3)c4ccccc4 KM08225 CCOC(=O)c1csc(n1)c2cn(c(=O)n(c2=O)C)c3ccccc3 KM08226 c1cc2c(cc1[N+](=O)[O-])S(=O)(=O)CC2SCCO KM08337 c1cc(sc1)Sc2ccc(cc2)NC(=O)c3ccc(cc3)Cl KM02459 Cn1c(nnc1SCC(=O)Nc2ccccc2)CSCC(=O)Nc3ccccc3 KM09155 Cc1c(c(sc1C(=O)OC)SC)c2ccn(n2)S(=O)(=O)c3ccc(cc3F)F KM02109 Cc1c(c(sc1C(=O)OC)SC)c2ccn(n2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM02110 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/NCc2cccnc2 KM01011 c1ccc(c(c1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl KM01027 Cc1csc2c1c(c(s2)C(=O)Oc3ccc(cc3)Cl)C KM03548 c1ccc(cc1)c2cn(cnc2=O)Cc3cccs3 BTB05538 CC(c1ccccc1)NC(=O)c2cc(cc3c2-c4ccc(cc4C3=O)[N+](=O)[O-])[N+](=O)[O-] RJC00482 c1ccc2c(c1)CCN=C2SCC(=O)c3ccc(c(c3)Cl)Cl.Br KM08234 c1ccc(c(c1)NC(=O)CN2c3cc(ccc3SCC2=O)C(F)(F)F)Cl KM08291 c1cc(ccc1NC(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])OC(F)(F)F AW00590 Cc1ccc2cccc(c2n1)OS(=O)(=O)c3cc(cc(c3)Cl)Cl BTB05592 Cc1nc(cs1)c2ccc(cc2)Br KM02515 COC(=O)C(C#N)c1ccccc1[N+](=O)[O-] KM08213 COC(=O)C(C#N)c1ccc(cc1[N+](=O)[O-])C(F)(F)F KM08218 COC(=O)CSc1c(ccs1)[N+](=O)[O-] KM05477 c1cc(ccc1Oc2c(ccs2)[N+](=O)[O-])Cl KM05478 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)O KM08328 CCOC(=O)C(Cc1cc(c(c(c1)[N+](=O)[O-])Oc2ccc(cc2)OC)[N+](=O)[O-])NC(=O)C KM08336 c1ccc(cc1)C#Cc2ccc(cc2)/C=N\OC(=O)Nc3cccc(c3)Cl KM08108 COc1ccc(cc1)C(=O)/C(=C/c2cc(cs2)C#Cc3ccccc3)/C#N KM08110 Cc1cc(nc2n1nc(c2Br)c3ccc(cc3)Cl)C(F)(F)F KM02449 c1cc2c(c(c1)NS(=O)(=O)c3ccc(s3)Cl)nsn2 KM06528 c1cc2c(c(c1)NS(=O)(=O)c3cc(sc3Cl)Cl)nsn2 KM06529 CC(=O)N1CCc2c1ccc(c2)Br KM08258 c1ccc(cc1)NC(=O)O/N=C(\C2COc3ccccc3O2)/N KM06579 CS(=NS(=O)(=O)c1cccc2c1non2)(=O)c3ccccc3 KM06584 Cc1cc(nc2n1ncc2c3nc(on3)C)C(F)(F)F KM02544 CC1(OC(=O)C(=CNc2ccccn2)C(=O)O1)C KM02546 CC(C)(C)NC(=O)c1c(c(c(s1)SC)C#N)c2ccc(cc2)Cl KM01233 CCO/C=C(\C#N)/S(=O)(=O)c1ccc2ccccc2c1 KM01241 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)N2CCCCC2 KM02461 c1cc(c(nc1)Sc2cccs2)C(=O)Nc3ccc(c(c3)Cl)F KM02462 c1cc2c(cc1C(=O)O)non2 CC09701 CC(=O)n1ccc(n1)c2c3c(c(s2)SC)C(=O)CC(C3)(C)C KM03430 CC1(Cc2c(c(sc2c3c(c[nH]n3)Br)SC)C(=O)C1)C KM03431 Cc1nccc(n1)c2cccc(c2)N CC31614 CC(C)S(=O)(=O)c1csc(c1N)C(=O)OCC(=O)C(C)(C)C KM02157 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccc(cc4)Cl KM08242 Cc1c(cco1)C(=O)/C(=C/Nc2ccsc2C(=O)OC)/C#N KM06526 c1cc2c(c(c1)NS(=O)(=O)c3cccs3)nsn2 KM06530 CC(C)(C)c1ccc(s1)C(=O)OCc2ccc3c(c2)OCO3 MBE00154 c1ccc(cc1)OCCSCc2nnc(o2)S KM06568 c1cc(c(cc1Cl)Cl)CSc2nnc(o2)CSCCOc3ccc(cc3Cl)Cl KM06570 c1ccc(cc1)C(=O)NNC(=O)CN2c3cc(ccc3SCC2=O)C(F)(F)F KM08340 Cc1ccc(cc1)S(=NC(=O)c2cc(on2)C)(=O)C KM08343 c1cc(c(nc1)SCC(=O)O)[N+](=O)[O-] KM08121 CC(C)(C#Cc1ccc(cc1)/C=N/OC(=O)Nc2cccc(c2)Cl)O KM08125 CC(C)C(=O)Nc1ccccc1NC2=C(CSC2)C(=O)OC KM02469 CCSc1c(c(c(s1)C(=O)OC)c2ccc(cc2)Cl)C#N KM02470 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)c3cccs3 KM02471 COc1ccc(cc1)S(=O)(=O)Nc2ccccc2NC3=C(CSC3)C(=O)OC KM02473 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc4c3nsn4 KM06544 CCCS(=O)(=O)c1csc(c1N/N=C/c2cccs2)C(=O)OC KM02497 CCCS(=O)(=O)c1csc(c1N/N=C/c2ccc(cc2)N(C)C)C(=O)OC KM02498 CCCS(=O)(=O)c1csc(c1NNC(=O)c2cc(cc(c2)Cl)Cl)C(=O)OC KM02500 c1ccc(cc1)CNC(=O)Nc2cccc(c2)[N+](=O)[O-] KM09331 c1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3ccc(cc3)F)N KM09332 c1ccc(cc1)CN(C(=O)CC#N)C(=O)Nc2cccc(c2)F KM09334 c1ccc2cc(ccc2c1)S(=O)(=O)/C(=C/Nc3ccc(cc3)F)/C#N KM01257 Cc1cc(n2c(n1)cc(n2)c3ccccc3)C(F)(F)F KM02232 CSc1c(c(n2c(n1)cc(n2)c3ccc(cc3)Cl)N)C#N KM02096 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)c3ccc(cc3)Cl)C)C KM03517 CCOC(=O)c1c(c2c(c(sc2s1)C#N)C)C KM03442 Cc1csc2c1c(cs2)C KM03443 CSc1c2c(c(s1)C(=O)N/N=C/c3ccc(cc3)Cl)CCCC24SCCS4 KM05188 CSc1c2c(c(s1)C(=O)N/N=C/c3cccs3)CCCC24SCCS4 KM05189 Cc1ccc2c(c1[N+](=O)[O-])c(cc(n2)C(F)(F)F)OC KM08256 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cccc4c3nsn4 KM06541 CNC(=O)Nc1ccccc1NC2=C(CSC2)C(=O)OC KM02489 CC1(OC(=O)C(=CNc2cccc(c2)C(F)(F)F)C(=O)O1)C KM02528 CC1(OC(=O)C(=CNc2ccc(c(c2)Cl)F)C(=O)O1)C KM02534 c1cc2c(c(c1)S(=O)(=O)Oc3cccnc3)non2 KM06588 c1ccnc(c1)c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F KM09546 COC(=O)C1=C(CSC1)Nc2ccccc2NS(=O)(=O)c3ccccc3C(F)(F)F KM02472 COC(=O)C1=C(CSC1)Nc2ccccc2NS(=O)(=O)c3ccccc3Cl KM02474 COC(=O)C1=C(CSC1)Nc2ccccc2NS(=O)(=O)c3ccc(cc3)Cl KM02475 c1cc(sc1)S(=O)(=O)C/C(=N/OC(=O)Nc2ccc(cc2)Cl)/N KM02311 c1cc(sc1)S(=O)(=O)/C(=N/Nc2ccc(cc2)F)/C#N KM02314 c1cc(c(cc1Cl)Cl)Oc2c(ccs2)[N+](=O)[O-] KM05346 Cn1c(nnc1SCC(=O)Nc2cccc3c2nsn3)C(F)(F)F KM06553 c1cc(c(cc1Cl)Cl)OCCSCc2nnc(o2)S KM06555 CC(=O)C(=C(SC)SC)S(=O)(=O)c1ccc(cc1)Cl KM01234 c1ccnc(c1)S(=O)(=O)Cc2nc(on2)c3ccc(cc3)Cl KM01250 c1cc(ccc1F)Sc2ccc(c3c2non3)[N+](=O)[O-] KM06837 COc1ccc(cc1)Oc2ccc(c3c2non3)[N+](=O)[O-] KM06839 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)N/N=C/c2c(cccc2Cl)Cl KM03578 Cn1c2c(c(cc(n2)OC(=O)N(C)C)COC)c(n1)c3cccs3 KM00965 CSc1c(c(nn1CNC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3cccs3)C#N KM00989 CSc1c2c(c(s1)C(=O)/C(=C/Nc3ccccc3Cl)/C#N)CCC=C2 KM05058 CC(=O)NNC(=O)c1c2c(c(s1)SC)C3(CCC2)SCCS3 KM05199 CSc1c2c(c(s1)C(=O)NNC(=O)Nc3ccc(cc3)Cl)CCCC24SCCS4 KM05200 Cc1ccc2c(c1)C(=O)C(=O)S2 KM09178 CC1(Cc2c(c(sc2C(=O)OC)SCCOC(=O)c3ccc(cc3)Cl)C(=O)C1)C KM05237 CCCS(=O)(=O)c1csc(c1N/N=C\c2c(cccc2Cl)F)C(=O)OC KM02496 CS(=N/C=C(\C#N)/C(=O)c1ccccc1)(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06548 CS(=N/C=C(\C#N)/C(=O)c1cccs1)(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06549 C(CSCCC(=O)N)C(=O)N KM09274 c1cc2c(cc1OC(F)(F)F)c(ccn2)O KM09327 c1ccnc(c1)S(=O)(=O)C/C(=N/OC(=O)c2ccc(cc2)Cl)/N KM01240 COc1ccc(cc1)/N=C/c2ccccc2O BTB00241 c1cc2c(c(c1)S(=O)(=O)N(CCC#N)CC3CCCO3)nsn2 KM09335 CC(=C(C#N)C#N)c1ccc(cc1)Cl KM03729 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)/C=C(\C#N)/C(=O)c3cccc(c3)C(F)(F)F KM05355 CSc1c2c(c(s1)C(=O)/C(=C/Nc3ccccn3)/C#N)CCC=C2 KM05357 Cc1cc(n2c(n1)cc(n2)c3cccs3)C(F)(F)F KM02329 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)/C=C(\C#N)/C(=O)c3ccccc3 KM05353 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)/C=C(\C#N)/C(=O)c3ccco3 KM05354 CS(=O)(=O)c1c2c(c(s1)C#N)CC(CC2=O)c3ccccc3 KM03583 c1cc2c(cc(nc2c(c1)C(F)(F)F)C(F)(F)F)O KM09512 c1ccc(cc1)NC(=O)NNC(=O)CC2C(=O)Nc3ccccc3S2 KM03725 CNC(=O)NNC(=O)CC1C(=O)Nc2ccccc2S1 KM03726 CSc1c(c(c(s1)c2cc[nH]n2)c3ccccc3)C#N KM05362 CSc1c2c(c(s1)C(=O)/C(=C/Nc3ccc(cn3)Cl)/C#N)CCC=C2 KM05363 C/S(=N/C(=O)c1cccc(c1)Cl)/c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06494 CCCS(=O)(=O)c1csc(c1NNS(=O)(=O)c2ccc(cc2)Cl)C(=O)OC KM02503 CCCS(=O)(=O)c1csc(c1NNS(=O)(=O)c2cccc(c2)Cl)C(=O)OC KM02504 CCCS(=O)(=O)c1csc(c1NNS(=O)(=O)c2ccccc2C(F)(F)F)C(=O)OC KM02505 c1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3cccc(c3)F)N KM09336 c1cc2c(c(c1)S(=O)(=O)N(CCC#N)Cc3cccs3)nsn2 KM09346 Cc1ccc(cc1)SCC(=O)Nc2cc(ccc2Cl)C(F)(F)F NRB00040 CCC(=O)c1cc(c(cc1OC)OC)OC RH00912 CC(C)(C#Cc1ccc(cc1)/C=N/O)O KM08088 c1ccc(cc1)C#Cc2ccc(cc2)/C=N/OC(=O)c3ccccc3Cl KM08091 c1ccc(cc1)C#Cc2ccc(cc2)/C=N/OC(=O)c3ccccc3 KM08092 c1ccc(cc1)C#Cc2ccc(cc2)/C=N/OC(=O)c3cccs3 KM08093 CCCCCCNC(=O)NC(Cc1ccccc1)C(=O)OCC NRB00828 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)NNC(=O)Nc3ccc(cc3)Cl KM02336 Cc1cc2nnc(c(n2n1)C)C(=O)O KM01115 c1cc(oc1)CN(CCC(=O)NNC(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM09404 C/C(=N\O)/c1ccc(c(c1)Cl)Cl KM06672 CN1c2ccccc2C(=O)/C(=C/N=S(=O)(C)C)/S1(=O)=O KM05275 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)NNC(=O)c2ccc(cc2)Cl KM03594 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)NNC(=O)c2ccccc2Cl KM03595 Cc1cccc2c1nc(cc2O)C(F)(F)F KM09513 CCCCC#Cc1ccc(o1)C(=O)N/N=C/c2ccccc2 KM09518 CSc1c(c([nH]n1)NC(=O)Nc2ccccc2)S(=O)(=O)c3ccc(cc3)Cl KM01264 c1ccc(cc1)C2CC(=O)C(=CNc3ccccc3Cl)C(=O)C2 KM03613 Cc1ccc(cc1F)NC(=O)c2c3ccccc3nnc2c4ccccc4 KM09122 CC(C)(C)c1cc2nc(cc(n2n1)NNC(=O)Nc3ccc(cc3)Cl)C(F)(F)F KM07968 CC(C)(C)c1cc2nc(cc(n2n1)NNC(=O)Nc3ccccc3)C(F)(F)F KM07969 C/C(=N\OCc1ccc(o1)C(=O)OC)/c2ccc(cc2Cl)Cl KM06498 c1ccc(cc1)C#Cc2cc(sc2)/C=C(\C#N)/C(=O)c3ccccc3 KM08096 CC(C)(C)c1cc2nc(cc(n2n1)N/N=C/c3ccccc3)C(F)(F)F KM07978 c1ccc2cc(ccc2c1)S(=O)(=O)/C(=C/Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)/C#N KM01256 c1ccnc(c1)S(=O)(=O)/C(=C/Nc2ccc(cc2)Cl)/C#N KM01176 c1ccnc(c1)S(=O)(=O)/C(=C/Nc2ccc(c(c2)Cl)F)/C#N KM01177 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)Nc4ccc(cc4)Cl KM06849 C/C(=N\OCc1cccc(c1)C(=O)O)/c2ccc(c(c2)Cl)Cl KM06720 Cc1c(sc(c1C(=O)/C=C/N(C)C)SC)C#N KM03591 c1ccc(cc1)C(=O)O/N=C(/C2COc3ccccc3O2)\N KM06603 c1cc2c(cccc2S(=O)(=O)N3CCOCC3)c(c1)N NRB00864 Cc1cccc(c1NC(=O)CSC(=O)c2cccs2)C BTB02791 c1cc(sc1)C(=O)/C(=C/Nc2ccc(cc2)OC(F)(F)F)/C#N KM03617 Cn1c(cc(n1)c2ccccc2)N KM01136 c1cc(ccc1S(=O)(=O)/C(=C/Nc2ccc(c(c2)Cl)Cl)/C#N)Cl KM01139 CC1(CCc2cc(ccc2O1)C(=O)/C=C/N(C)C)C KM05282 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCC(CC3)n4cccc4 KM09459 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)SCC(=O)OCC BTB00877 Cc1cccc(c1)NC(=S)NNC(=O)c2cc(c(c(c2)OC)OC)OC ML00355 Cn1c(nnc1SC)C(F)(F)F KM05422 c1cc(ccc1NC(=O)NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)Cl KM05423 c1cc(ccc1C(=O)N2CCSC2=S)Cl KM06398 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)C(=O)Nc4ccc(cc4)Cl)C(F)(F)F KM09133 CC(=O)c1cc(c(s1)NCC#C)[N+](=O)[O-] KM03391 CC(=O)c1cc(c(s1)N2CCOCC2)[N+](=O)[O-] KM03394 c1ccc(cc1)C#Cc2ccc(s2)c3ccn(n3)C(=O)c4ccccc4 KM08065 CC(C)(C)c1cc2nc(cc(n2n1)N/N=C/c3ccc(cc3)Cl)C(F)(F)F KM07980 COC(=O)CC(=O)NC(CSC(=O)Nc1ccc(cc1)Cl)C(=O)OC KM07982 COC(=O)c1c(c(c(s1)SC)C#N)c2ccco2 KM00899 c1cc(c(c(c1)Cl)/C=C(\C#N)/S(=O)(=O)c2cccs2)Cl KM02271 CC(=O)NC(=O)/C(=C/Nc1cc(c(cc1OC)Cl)OC)/C#N KM09234 c1cc(ccc1N/N=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)Cl KM01179 CC(=O)NCCc1ccc(cc1)OC(=O)C KM06677 c1ccc(cc1)OCCSCC(=O)N2CCOCC2 KM06681 CCOC(=O)c1c2c(c(s1)SCCS(=O)(=O)c3ccc(cc3)C)C(=O)CC(C2)(C)C KM05279 CCOC(=O)c1c2c(c(s1)SC)C(=O)CC(C2)c3ccc(cc3)C KM03592 Cc1csc(n1)c2cc(sc2SC)C(=O)OC KM03599 Cc1c(c(sc1C(=O)N)SC)C=C KM03607 CSc1c(c(n[nH]1)c2ccc(cc2)Cl)C#N KM01262 Cc1ccc(cc1)C2Cc3c(sc(c3C(=O)C2)SC)C#N KM03610 C/C(=N\OCc1ccc(o1)C(=O)N2CCCCC2)/c3cccc(c3)C(F)(F)F KM06613 CCOC(=O)CC1C(=O)Nc2ccccc2S1 KM03628 Cc1ccc(cc1)C2Cc3c(sc(c3C(=O)C2)S(=O)C)C#N KM03631 CCOC(=O)c1c2c(c(s1)SCCS(=O)(=O)c3ccc(cc3)Cl)C(=O)CCC2 KM05252 Cc1c(c(sc1C(=O)NNC(=O)C)SC)C=C KM03641 c1cc(oc1)CN(CCC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM09466 c1cc2c(cc(nc2c(c1)F)C(F)(F)F)O KM09485 c1c(c(sc1S(=O)(=O)N2CCOCC2)Cl)S(=O)(=O)N3CCOCC3 KM05299 CC(=O)c1c2c(c(s1)SCCS(=O)(=O)c3ccc(cc3)Cl)C(=O)CCC2 KM05300 Cc1cccc2c1N(CCC2)C(=S)Nc3cccc(c3)Cl BTB01026 Cc1c(cco1)C(=O)C(=C2SCCCCS2)C#N KM06602 COc1ccc(cc1)C(=O)O/N=C(\C2COc3ccccc3O2)/N KM06604 c1ccc(cc1)C#Cc2ccc(cc2)/C=C(\C#N)/C(=O)c3ccccc3 KM08069 c1cc(c(c(c1)Cl)CSc2cccs2)Cl KM02235 CCOC(=O)c1ccc(cc1)OCC#C KM08077 Cc1ccc(cc1)CS(=O)(=O)c2cccs2 KM02236 Cn1c(nnc1SCC(=O)c2ccc(cc2)C(F)(F)F)CSCC(=O)Nc3ccccc3 KM09142 COc1cccc(c1)c2c(c(sc2C(=O)OC)SC)C#N KM00911 Cc1csc(n1)c2c(c(c(s2)SC)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl)C KM05098 CCCS(=O)(=O)C/C(=N/OS(=O)(=O)c1ccc(cc1F)F)/N KM02284 CCOC(=O)c1c2c(c(s1)SCCS(=O)(=O)c3ccccc3)C(=O)CC(C2)(C)C KM05280 c1ccc(cc1)OCCSCC(=O)NCc2ccco2 KM06691 CCCCC#Cc1cc(cnc1)C(=O)N/N=C/c2cccs2 KM09454 CC(C)NC(=O)c1ccccc1[N+](=O)[O-] KM09470 CSc1c(c(c(s1)NC(=O)Nc2ccccc2C(F)(F)F)c3ccc(cc3)Cl)C#N KM01263 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)C#N GK02993 c1cc(ncc1C(F)(F)F)Sc2c(ccs2)[N+](=O)[O-] KM05412 Cc1cc(n(n1)c2ncc(c(n2)N)C#N)C KM05419 c1ccc(c(c1)NC(=O)C(Cl)(Cl)Cl)Oc2ccc(cc2Cl)Cl BTB04866 c1cc(ccc1NC(=O)NNC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F)OC(F)(F)F KM09380 Cn1c(nnc1SCC(=O)c2ccc(cc2Cl)Cl)CSCCOc3ccccc3 KM06506 Cc1c(cco1)C(=O)C(=C(NCc2cccnc2)NCc3cccnc3)C#N KM06514 c1cc(ccc1NC(=O)NNC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F)Cl KM09381 c1cc(cc(c1)C(=O)CC#N)CSc2ccc(cc2)Cl KM05273 Cn1c(=O)c(cn(c1=O)c2ccccc2)C#N KM08136 CCOc1ccc(cc1)/C=N/NC(=S)NC ML00327 Cc1ccc(cc1)SC2CS(=O)(=O)c3c2cccc3 KM08139 c1cc2c(cc1OC(F)(F)F)c(cc(n2)C(F)(F)F)O KM09486 CCOC(=O)c1c(c(c(s1)SCCS(=O)(=O)c2ccc(cc2)Cl)C#N)c3ccccc3 KM05305 COC(=O)CSC1CS(=O)(=O)c2c1ccc(c2)[N+](=O)[O-] KM08161 Cc1ccc2c(c1NC(=O)Nc3ccc(cc3)Cl)c(cc(n2)C(F)(F)F)OC KM08303 c1ccc2c(c1)OCC(O2)C(=S)N KM06624 CCOC(=O)c1cc(cnc1)C#CCOC(=O)Nc2cc(cc(c2)Cl)Cl KM08313 c1cc(sc1)S(=O)(=O)Cc2ccc(c(c2)Cl)Cl KM02250 CC(C)S(=O)(=O)C/C(=N/OC(=O)Nc1ccccc1)/N KM02258 CCCS(=O)(=O)C/C(=N/OC(=O)Nc1ccc(cc1)Cl)/N KM02260 c1cc(sc1)SCc2ccc(cc2)Cl KM02262 Cn1cc(c(n1)c2cccc(c2)NC(=O)Nc3ccccc3)Br KM02088 c1cc(cnc1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM01078 CSc1c-2c(cs1)CCc3c2nc(nc3)SCC(=O)c4ccc(cc4)Cl KM05108 Cc1csc(n1)c2c(c(c(s2)SC)c3cnc(nc3)SCC(=O)Nc4cccc(c4)C(F)(F)F)C KM05110 c1ccc2c(c1)nc(s2)SCC#N KM01080 CC(C)(C)C(=O)CSc1ncc2c(n1)-c3c(csc3SC)CC2 KM05111 Cc1ccc(cc1)S(=O)(=O)CCSc2c3c(c(s2)C#N)CC(CC3=O)(C)C KM05291 c1cc2c(cc1F)c(cc(n2)C(F)(F)F)O KM09478 CCOc1cc(ccc1OC)C(=O)O KM09479 CCOC(=O)c1cnc2c(c1Sc3nnc(s3)SC)c(nn2C)C KM06598 COC(=O)c1cccc(c1)CN2C(=O)CSC2=O KM05425 COc1ccc(cc1)C(=O)NC(=O)N=S(=O)(C)c2ccc(cn2)C(F)(F)F KM05432 Cn1c(cc(n1)c2ccc(s2)/C=N/NC(=O)c3ccc(cc3Cl)Cl)C(F)(F)F KM05440 c1ccc(cc1)S(=O)(=O)N(CCC#N)Cc2ccco2 KM09397 COC(=O)CCN(Cc1ccco1)S(=O)(=O)c2ccc(cc2)Cl KM09400 c1cc(oc1)CN(CCC(=O)NN)S(=O)(=O)c2ccc(cc2)Cl KM09401 CSc1ncc(c(n1)N)C#N KM08141 Cc1ccc(cc1)NC(=O)O/N=C(/C)\c2ccc3c(c2)CCO3 KM06631 Cc1cccc(c1)NC(=O)O/N=C(/C)\c2ccc3c(c2)CCO3 KM06632 CC(C)c1ccc(cc1)N/N=C/c2cc(cs2)C#Cc3ccccc3 KM08146 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F KM08154 c1cc(sc1)SC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-] KM08165 COc1ccc(cc1)NC(=O)C2CCN(CC2)c3ccc(cn3)C(F)(F)F KM08167 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NNS(=O)(=O)c3ccc(cc3)Cl KM03694 COC(=O)c1c(ccs1)N/C=C(\C#N)/C(=O)c2ccco2 KM03697 Cc1ccc(cc1)S(=NS(=O)(=O)c2c(c3cc(ccc3s2)Cl)C)(=O)C KM08175 Cc1ccc2c(c1NC(=O)Nc3ccc(cc3)OC(F)(F)F)c(cc(n2)C(F)(F)F)OC KM08311 c1cc(ccc1Sc2ccc3c(c2[N+](=O)[O-])nsn3)Cl KM06626 c1ccc(cc1)C(=O)NNC(=O)CSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-] KM08318 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)C(=O)Nc4ccc(cc4)OC(F)(F)F)C(F)(F)F KM09153 CC1(Cc2c(c(sc2C(=O)OC)SC)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/C1)C KM03499 Cc1csc2c1c(c(s2)COC(=O)c3ccc(cc3)Cl)C KM03504 Cc1cc(nc(n1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)C KM01054 Cc1c(c([nH]n1)N)Br.Br KM01090 CC1CN(CC(O1)C)/C=C(\C#N)/S(=O)(=O)Cc2ccc(cc2)Cl KM01092 CC1(CCc2cc(ccc2O1)/C=N/OC(=O)Nc3cccc(c3)Cl)C KM05214 c1cc(ccc1S(=O)(=O)C(=C2SCCCS2)C#N)Cl KM00890 CC(=O)c1c2c(c(s1)SCCS(=O)(=O)c3ccccc3)C(=O)CC(C2)(C)C KM05301 Cc1ccc(cc1)S(=O)(=O)CCSc2c3c(c(s2)C(=O)C)CC(CC3=O)(C)C KM05302 Cn1c(nnc1SCc2cccc(c2)C(=O)OC)C(F)(F)F KM05304 c1ccc(c(c1)C(=O)NNC(=O)CC2C(=O)Nc3ccccc3S2)Cl KM03690 c1cc2c(cc1Cl)nsn2 KM06618 CCOC(=O)c1cc(cnc1)C#CCOC(=O)Nc2ccc(cc2)Cl KM08305 c1cc(sc1)S(=O)(=O)/C(=C/c2c[nH]cn2)/C#N KM08307 CC(C)S(=O)(=O)/C(=C/c1c[nH]cn1)/C#N KM08308 C/C(=N\OCc1ccc(o1)C(=O)N2CCOCC2)/c3cccc(c3)C(F)(F)F KM06621 CC(C)(C#Cc1ccc(cc1)/C=N/Nc2ccccc2)O KM08102 CC(C)(C#Cc1ccc(cc1)/C=N/Nc2c(cc(cc2Cl)Cl)Cl)O KM08103 Cc1nccc(n1)c2cccc(c2)N/N=C(\C#N)/S(=O)(=O)c3ccccn3 KM02267 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)N/N=C/C(C)(C)C KM02270 c1ccc(cc1)S(=O)(=O)CCS(=O)(=O)c2cccs2 KM02420 c1cc2c(cc1C(F)(F)F)NC(=O)CS2 KM08155 c1ccc2c(c1)C(CS2(=O)=O)S(=O)(=O)c3cccs3 KM08156 CC(=O)c1ccc(s1)Br KM02339 CC(C)S(=O)(=O)c1csc(c1N/N=C/c2ccccc2Cl)C(=O)OC KM02340 c1ccc(cc1)C#Cc2ccc(s2)/C=C(\C#N)/C(=O)c3ccccc3 KM08179 Cn1c(=O)c(cn(c1=O)c2ccccc2)/C(=N/OC(=O)c3ccccc3Cl)/N KM08182 COc1ccc(cc1)OC(=O)C2CCN(CC2)c3ccc(cn3)C(F)(F)F KM08187 CCCS(=O)(=O)c1csc(c1NNC(=O)C(C)C)C(=O)OC KM02506 c1ccc(c(c1)C(=O)NNC(=O)CSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-])Cl KM08319 Cc1ccc2c(c1NC(=O)c3ccccc3)c(cc(n2)C(F)(F)F)OC KM08323 CCOC(=O)c1ccc(cc1)Oc2c(ccs2)[N+](=O)[O-] KM05483 Cn1c(cc(n1)c2ccc(s2)/C=N/C(=C(/C#N)\N)/C#N)C(F)(F)F KM05484 Cc1c2c(c(cnc2n(n1)C)C(=O)N)Oc3ccc(cc3)Cl KM05485 Cc1cc(nc2c1c(nn2C)c3cccs3)O KM00841 c1ccnc(c1)N/C=C(\C#N)/C(=O)c2cccs2 KM00842 CNC(=O)c1c2c(c(s1)SC)C=CCC2 KM03440 CCOC(=O)c1c(c(c(s1)SC)C(=O)C)C KM03516 CC1(Cc2c(c(sc2C(=O)OC)SCCOC(=O)Nc3ccc(cc3)Cl)C(=O)C1)C KM05227 Cc1ccc(cc1)S(=O)(=O)C2CS(=O)(=O)c3c2cccc3 KM08157 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NNC(=O)c3cccs3 KM03691 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NNC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM03692 c1cc(cc(c1)Cl)NC(=O)C2CCN(CC2)c3ccc(cn3)C(F)(F)F KM08168 Cc1c2cc(ccc2sc1Br)Cl KM08172 COC(=O)c1c(ccs1)N/N=C(\C#N)/S(=O)(=O)c2cccs2 KM03702 Cc1cc(nc2n1nc(c2Br)C(C)(C)C)C(F)(F)F KM02418 Cc1cc(nc2n1nc(c2Br)C)C(F)(F)F KM02428 CCOC(=O)c1cc(cnc1)C#CCOC(=O)Nc2ccc(cc2)OC(F)(F)F KM08315 Cc1ccc2c(c1NC(=O)c3ccc(cc3)Cl)c(cc(n2)C(F)(F)F)OC KM08316 c1cc(ccc1C(=O)NNC(=O)CSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-])Cl KM08317 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02436 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)Nc2ccc(cc2)Cl KM02437 CC(C)S(=O)(=O)C/C(=N/OS(=O)(=O)c1cc(ccc1Cl)Cl)/N KM02282 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)NNS(=O)(=O)c3ccc(cc3F)F KM02348 c1ccc(cc1)OCCSCC(=O)Nc2ccc(cc2Cl)Cl KM06660 c1cc(oc1)CN(CCC(=O)NNC(=O)c2cccs2)S(=O)(=O)c3ccc(cc3)Cl KM09411 Cc1c(c(sc1C(=O)NC)S(=O)(=O)C)C=C KM03705 c1cc(ccc1OC(=O)C2CCN(CC2)c3ccc(cn3)C(F)(F)F)F KM08188 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)C GK03001 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] GK03005 c1cc(cc(c1)Oc2c(ccs2)[N+](=O)[O-])C(F)(F)F KM05490 COC(=O)C1=C(CSC1)Nc2ccc(cc2)OC(F)(F)F KM03838 CSc1c(c(c(s1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3ccc(cc3)Cl)C#N KM01228 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)OCC)N)c3ccc(cc3)Cl KM03461 c1csc(n1)NC(=O)CCCCC(=O)Nc2nccs2 JFD01883 CCOC(=O)c1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)N3CCOCC3 JP00573 CSc1c2c(c(s1)C(=O)NNC(=O)c3ccccc3Cl)CCCC24SCCS4 KM05198 c1cc(ccc1SC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-])Cl KM08160 c1ccc(cc1)OCCSCC(=O)O KM06649 c1cc(sc1)Sc2ccc(cc2[N+](=O)[O-])C#N KM02349 COC(=O)c1c(ccs1)N/N=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM03707 COC(=O)c1c(ccs1)N/N=C(\C#N)/S(=O)(=O)c2ccccn2 KM03708 Cn1c2ccc(cc2c(=O)s1)S(=O)(=O)NCCc3ccncc3 BTB03427 Cn1c(=O)c(cn(c1=O)c2ccccc2)/C(=N/OC(=O)c3cccs3)/N KM08183 Cn1c(=O)c(cn(c1=O)c2ccccc2)c3nc(on3)c4ccccc4Cl KM08189 c1ccnc(c1)c2ccc(s2)C(=O)O CC02201 Cn1c(c(c(n1)c2ccc(cc2)Cl)C(=O)N)SC KM01188 CSc1c(c(nn1C(=O)C(Cl)(Cl)Cl)c2cccs2)C#N KM01189 CCOC(=O)c1cc(cnc1)C#CCOC(=O)c2ccc(cc2)Cl KM08326 CN(C)CC#Cc1ccc(s1)c2cc[nH]n2 KM08327 Cc1ccc(cc1)c2csc(c2C#N)S(=O)C KM02562 CSc1c(c(nn1S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3cccs3)C#N KM01199 Cn1c(c(c(n1)c2ccccc2)C(=O)N)SC KM01200 Cc1cc(nc(n1)N/C=C(\C#N)/S(=O)(=O)c2ccccc2C(=O)OC)C KM01061 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4ccc5c(c4)non5 KM09624 CCCCC#Cc1ccc(o1)c2nnc(n2C)SCc3ccc(cc3)Cl KM09629 c1cc(oc1)CN(CCC(=O)O)S(=O)(=O)c2ccc(cc2)Cl KM09436 CCOC(=O)CCN(Cc1ccco1)S(=O)(=O)c2ccc(cc2)Cl KM09437 c1cc2c(cc1OC(F)(F)F)c(c(cn2)C(=O)O)O KM09299 c1ccc(cc1)CN(C(=O)CC#N)C(=O)Nc2cccc(c2)Cl KM09309 COc1ccc(cc1)NC(=O)N(Cc2ccccc2)C(=O)CC#N KM09313 CSc1ccc(cc1)NC(=O)NCc2ccccc2 KM09314 c1ccc2c(c1)CCN2/C=C(\C#N)/S(=O)(=O)c3ccc(cn3)C(F)(F)F KM05393 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccccc2C GK03002 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)N)Cl GK03009 Cc1ccc(cc1)S(=NC(=O)CSc2ccc(cn2)C(F)(F)F)(=O)C KM05319 c1cc(ccc1S(=O)(=O)/C(=N/[O-])/C#N)Cl.[Na+] KM01218 Cc1cc(nc(n1)C)N/C=C(\C#N)/S(=O)(=O)c2ccccc2Cl KM01063 c1ccc(c(c1)S(=O)(=O)/C(=C/Nc2ncccn2)/C#N)Cl KM01068 c1cc(c(nc1)Sc2cccs2)[N+](=O)[O-] KM02353 c1cc(c(c(c1)Cl)CS(=O)(=O)c2cccs2)F KM02355 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccncc3 KM09413 c1cc(oc1)CN(CCC(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl KM09416 Cn1c(=O)c(cn(c1=O)c2ccccc2)c3nc(on3)c4cccs4 KM08191 COC(=O)c1cc(cc(c1)Cl)Cl KM02512 CC(=O)c1c(c(c(s1)SC)C#N)c2ccc(cc2)Cl KM05373 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)C(F)(F)F GK03007 CSc1c(c([nH]n1)NC(=O)c2ccc(c(c2)Cl)Cl)S(=O)(=O)c3ccc(cc3)Cl KM01222 CC(C)S(=O)(=O)c1cnc(nc1N)c2ccccn2 KM02583 c1ccc2cc(ccc2c1)SCC#N KM01226 CSc1c(c(c(s1)C(=O)Nc2ccc(cc2F)F)c3ccc(cc3)Cl)C#N KM01229 CCOC(=O)/C(=C\1/C(=CC=CN1)OC(=O)C)/C#N KM05308 COC(=O)c1ccccc1S(=O)(=O)/C(=C/Nc2nc(nc(n2)SC)C3CC3)/C#N KM01069 CSc1nc(nc(n1)N/C=C(\C#N)/S(=O)(=O)c2ccccc2Cl)C3CC3 KM01070 c1ccnc(c1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM01077 c1ccnc(c1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM01153 c1ccc\2c(c1)CCC/C2=N\O KM09261 COc1ccc(cc1OC2CCCC2)C(=O)N KM09271 c1ccc(c(c1)CN/C(=C(/C#N)\N=C\c2ccc(cc2)Cl)/C#N)Sc3ccc(cc3)Cl KM03650 CSc1c(c(c(s1)c2ccnc(n2)SCc3ccc(cc3)Cl)c4ccccc4)C#N KM05394 c1ccc(cc1)CN2c3cc(ccc3SCC2=O)C(F)(F)F KM08269 CCOC(=O)c1c2c(c(s1)SC)C(=O)CC(C2)c3ccccc3 KM03557 CCOC(=O)c1c(c2c(c(sc2s1)c3cc[nH]n3)C)C KM03558 CCOC(=O)C1CCN(CC1)/C=C(\C#N)/S(=O)(=O)c2ccccn2 KM08273 Cc1ccccc1C(=O)Oc2cc(sc2C(=O)OC)OC GK03015 COc1cc(c(s1)C(=O)OC)OC(=O)c2ccc(cc2)F GK03016 COc1cc(c(s1)C(=O)OC)OC(=O)c2ccco2 GK03020 CC(=O)OC1=CC=CNC1=C(C#N)C#N KM05329 COc1ccc2c(c1)non2 KM06417 CCCCC#Cc1ccc(o1)c2nnc(n2C)SCc3ccccc3 KM09642 CCCCC#Cc1ccc(o1)c2nnc(n2C)SCc3cc(cc(c3)F)F KM09643 Cc1cc(n(n1)c2nc(c(c(n2)SC)C#N)c3ccco3)C KM05404 Cc1c(nc(n(c1=O)C)N)C KM09442 CCCS(=O)(=O)c1cnc(nc1N)SC KM02619 c1ccc(c(c1)/C=N/C(=C(\C#N)/N)/C#N)Sc2ccc(cc2)Cl KM03627 CC1(CCc2cc(ccc2O1)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl)C KM05599 CCOC(=O)c1cc(cnc1)C#CCOC(=O)c2c(onc2c3c(cccc3Cl)Cl)C KM08353 CCCCCCC#Cc1cc(cnc1)C(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F KM09475 c1ccc(cc1)C#Cc2ccc(s2)COC(=O)c3ccc(cc3)Cl KM08257 COc1ccc(cc1)OC(=O)c2ccc3c(c2)non3 KM09594 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)O KM09477 Cc1cc(nc(n1)NC=C2C(=O)OC(OC2=O)(C)C)C KM02556 CC1(OC(=O)C(=CNc2ncccn2)C(=O)O1)C KM02557 CC(C)(C)C(=O)C=C(SC)SC KM02559 COc1ccc(cc1)C2C3CCc4ccccc4C3=Nc5ccccc5S2 JFD02624 c1cc(ccc1NC(=O)Nc2ccc3c(c2)non3)Cl KM09748 Cc1c(c(n(n1)Cc2nc(cs2)C(C)(C)C)C)Br KM03830 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)/C=N/c3ccc(cc3)Cl KM05611 CC1(CCc2cc(ccc2O1)c3ccn(n3)S(=O)(=O)c4ccccc4Cl)C KM05614 CC1(CCc2cc(ccc2O1)c3ccn(n3)S(=O)(=O)c4ccc(cc4)OC)C KM05617 CCS(=O)c1c(c(cs1)c2ccc(cc2)Cl)C#N KM02495 c1cc(ccc1NC(=O)NNC(=O)c2ccc3c(c2)non3)Cl KM09655 CSc1c-2c(cs1)CCc3c2nn(c3)C(=O)c4ccc(cc4)Cl KM03871 c1ccc(cc1)C#Cc2ccc(s2)/C=C(\C#N)/C(=O)c3cccs3 KM08199 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4cccs4 KM08207 Cc1ccc(cc1)S(=O)(=O)CCN2CCC(CC2)C(F)(F)F KM08106 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)/C=N/c3ccc(cc3)OC KM05433 CC1(CC(=O)CC(=O)C1C(=O)OC)C RJC03508 c1ccc(cc1)N2CCN(CC2)C3CC(=O)C(=C3)Nc4ccc(cc4)Cl NRB00487 CCOC(=O)CC1C(=Nc2ccccc2S1)SCC(=O)Nc3ccc(cc3)Cl KM06807 CC1CCN(CC1)Cc2cc(c(c(c2)Cl)O)Cl.Cl BTB04042 COc1ccc(cc1)Nc2ccc(c3c2non3)[N+](=O)[O-] KM06816 c1cc2cc(ccc2nc1)C(=O)N3CCOCC3 KM10150 Cn1c(nnc1SCc2ccc(cc2)Cl)c3ccc4c(c3)non4 KM09727 CCCC(=O)NNc1ncc(c(n1)C(F)(F)F)C(=O)OCC GK03043 CCOC(=O)c1cc(cnc1)C#CCOC(=O)c2ccc(cn2)Cl KM08362 CCCS(=O)(=O)c1cnc(nc1N)C2COc3ccccc3O2 KM09670 CC(C)S(=O)(=O)c1csc(c1N/N=C(\C#N)/C(=O)c2ccccc2)C(=O)OC KM02589 c1cc(c(cc1N2CCSCC2)O)[N+](=O)[O-] BTB05899 Cc1ccc(cc1)S(=O)(=O)CCSC2=CC(=O)CC(S2)(C)C KM03965 CC1(CC(=O)C=C(S1)SCCS(=O)(=O)c2ccc(cc2)Cl)C KM03967 c1cc(cc(c1)NC(=O)Nc2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)C(F)(F)F KM05710 CSc1c(c(c(s1)c2ccnc(n2)SC)c3ccccc3)C#N KM05771 c1cc(sc1)CN(CCS(=O)(=O)c2ccc(cc2)Cl)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM03875 CC1(Cc2c(c(sc2c3ccnc(n3)S)SC)C(=O)C1)C KM03878 COc1ccc(cc1)CSC2C(C3CCN2CC3)C(=O)NNC(=S)Nc4ccccc4 KM06942 c1ccc2c(c1)CCN=C2SCC(=O)c3ccccc3Cl.Br KM08235 c1cc(c(cc1NC(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl)F BTB06123 CC(C)(C)c1cc2nc(cc(n2n1)SCCO)C(F)(F)F KM08107 Cn1c(=O)c(cn(c1=O)c2ccccc2)c3nc(cs3)c4ccc(cc4)Cl KM08223 CC(C)(C)OC(=O)N1CCN(CC1)CCNC(=O)Nc2ccccc2 KM08228 c1ccc(cc1)C#Cc2cc(sc2)/C=C(\C#N)/C(=O)c3cccs3 KM08112 c1c(csc1C2SCCS2)Br KM02456 CC(C)(C#Cc1ccc(cc1)/C=N/OC(=O)c2ccccc2Cl)O KM08116 c1cc(ccc1C(=O)O/N=C/c2ccc3c(c2)CCO3)Cl KM06697 c1cc(ccc1NC(=O)O/N=C/c2ccc3c(c2)CCO3)Cl KM06699 c1cc(ccc1CO/N=C/c2ccc3c(c2)CCO3)Cl KM06701 CC(C)(C)S(=O)(=O)c1cnc(nc1N)c2ccccn2 KM02695 CC1(OC(=O)C(=CNc2ccc(cn2)Cl)C(=O)O1)C KM02551 CS(=NS(=O)(=O)c1ccccc1Cl)(=O)c2ccc(cn2)C(F)(F)F KM05606 CS(=N/C=C(\C#N)/C(=O)c1ccc(cc1)Cl)(=O)c2ccc(cn2)C(F)(F)F KM05618 c1ccc(cc1)CS(=O)(=O)c2ccc(cn2)C(F)(F)F KM05621 Cc1c(c(n(n1)CC(=S)N)C)Br KM03747 Cc1c(c(on1)NC(=O)c2ccc(cc2)C(F)(F)F)[N+](=O)[O-] KM03750 Cc1nccc(n1)c2cccc(c2)NN=C(C#N)C#N KM02492 CC1(Cc2csc(c2C(=O)C1)S(=O)C)C KM03767 Cc1nccc(n1)c2cccc(c2)N/N=C(\C#N)/C(=O)c3ccccc3 KM02507 C/S(=N\S(=O)(=O)c1ccccc1)/c2c(cc(cn2)Cl)C(F)(F)F KM05705 c1ccc(cc1)NC(=O)OCCSCc2ccc3c(c2)ccc(n3)C(F)(F)F KM08530 c1cc(cc(c1)Oc2c(nccn2)C(=O)Nc3ccc(cc3F)F)C(F)(F)F KM05545 CCOC(=O)c1cnc(nc1C(F)(F)F)O/N=C(/c2ccc(cc2)C(F)(F)F)\N GK02994 CCOC(=O)CN1c2cccc(c2OC(C1=O)C(C)C)C(C)C KM06732 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)SCc4ccco4 KM06860 c1cc(c(cc1Cl)Cl)C(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-] KM06863 CC(C)(C)OC(=O)N1CCN(CC1)CCNC(=O)c2ccc(cc2)Cl KM08238 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccccc4 KM08241 C/C(=N\OCc1cccc(c1)C(=O)O)/c2ccc(cc2)Cl KM06722 C/C(=N\OCc1cccc(c1)C(=O)Oc2ccccc2)/c3ccc(c(c3)OC)OC KM06725 CC(C)(C#Cc1ccc(cc1)CO)O KM08119 C#CCOc1ccc(cc1)C#N KM08122 c1ccc(cc1)C#Cc2ccc(cc2)/C=N\OC(=O)Nc3ccc(cc3)OC(F)(F)F KM08120 COc1ccc(cc1)NC(=O)c2ccc3c(c2)cccn3 KM10123 CC(C(=O)O)Oc1ccc2c(c1)c(=O)c3ccccc3o2 JFD02525 c1ccc(cc1)CNC(=O)c2ccc3c(c2)cccn3 KM10129 CC(C)(C)c1ccc(cc1)c2nc(on2)c3cc(cnc3)C#Cc4ccccc4 KM08384 Cc1ccc(cc1)/C(=N/OC(=O)c2cc(cnc2)C#Cc3ccccc3)/N KM08387 c1cc(ccc1c2ccnc(n2)S)Cl KM05717 c1cc(ccc1c2ccnc(n2)SCCS(=O)(=O)c3ccc(cc3)Cl)Cl KM05729 CC1(Cc2c(sc(c2C(=O)C1)SCCOC(=O)c3ccccc3Cl)C#N)C KM05375 Cc1c(c(on1)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C)[N+](=O)[O-] KM03735 c1cc(ccc1F)S(=O)(=O)C/C(=N/O)/N KM08532 CC1(Cc2c(sc(c2C(=O)C1)SCCOC(=O)Nc3ccc(cc3)OC(F)(F)F)C#N)C KM05383 C1CC(C(=O)NC1)C(=O)NN BTB00340 CN(C)c1ccc(cc1)/C=N/NC(=O)c2ccncc2 BTB00391 Cc1c(c(c2n1CCS2)C(=O)OC)C(=O)OC KM05547 Cc1c2c(=O)c3c([nH]c2n(n1)C)CSC3 KM05405 c1cc(ccc1S(=O)(=O)C(=C2SCCCCS2)C#N)Cl KM05407 c1cc(cc(c1)C(F)(F)F)C(=O)C(=C2SCCCCS2)C#N KM05409 CCCCOc1c(c(=O)c1=O)Nc2cccc(c2)OC KM09701 CCOC(=O)c1cccc(c1)CO/N=C(\C)/c2ccc(c(c2)Cl)Cl KM06748 c1cc(ccc1C(=O)O/N=C(/c2ccc3c(c2)non3)\N)Cl KM06759 c1cc(ccc1C(=O)Nc2ccc3c(c2)C(=O)OC3)Cl KM08468 CSc1c(c(c(s1)Cl)c2ccc(cc2)Cl)C#N KM02713 CC(C)c1cccc2c1OC(C(=O)N2)C(C)C KM06729 c1cc2c(c(c1)S(=O)(=O)N(CC/C(=N/OC(=O)c3ccc(cc3)Cl)/N)Cc4ccco4)nsn2 KM09398 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)c3ccccc3Cl)C(F)(F)F KM08130 c1cc(ccc1c2nc(on2)CCC(=O)NNS(=O)(=O)c3ccc(cc3)Cl)Cl BTB02459 COc1ccc(cc1)NC(=O)Nc2ccc3c(c2)non3 KM09749 c1ccc(cc1)C#Cc2cc(cnc2)c3nc(no3)c4ccccc4 KM08391 c1cc(c(c2c1nsn2)[N+](=O)[O-])N3CCCC3 KM06736 c1ccc(cc1)Nc2ccc3c(c2[N+](=O)[O-])nsn3 KM06738 CCOC(=O)c1csc(n1)C2COc3ccccc3O2 KM06742 C/C(=N\OCc1cccc(c1)C(=O)Oc2ccc(cc2)C(F)(F)F)/c3ccc(c(c3)Cl)Cl KM06747 c1ccc(cc1)C#Cc2ccc(s2)COC(=O)Nc3ccc(cc3)Cl KM08253 c1ccc(cc1)C#Cc2ccc(s2)COC(=O)Nc3cc(cc(c3)Cl)Cl KM08254 c1ccc2c(c1)OCC(=O)O2 RH00750 Cc1cc(n(n1)c2ncc(c(n2)N)S(=O)(=O)c3ccc(cc3)Cl)C KM05399 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)O/N=C(/c3cccc(c3)C(F)(F)F)\N KM08386 CSc1c(cn(n1)c2ccccc2)c3nc(cs3)c4ccc(cc4)Cl KM08393 CCOC(=O)/C(=C/c1ccc(s1)c2cc(n(n2)C)C(F)(F)F)/C#N KM05415 CC(C)(C#Cc1ccc(cc1)/C=N/Nc2c(cc(cn2)C(F)(F)F)Cl)O KM08410 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Nc3ccc(cc3)Cl KM08330 Cc1cc(no1)C(=O)N=S(=O)(C)c2ccccc2 KM08344 c1cc2c(cc1[N+](=O)[O-])S(=O)(=O)CC2SCCOC(=O)Nc3cc(cc(c3)Cl)Cl KM08351 CCOC(=O)c1c2c(c(s1)SCc3ccccc3)C(=O)CCC2 KM03709 COC(=O)c1c(ccs1)N/C=C(\C#N)/S(=O)(=O)c2cccs2 KM03713 CSc1c(cn(n1)c2ccccc2)C(=S)N KM08388 Cc1ccc(cc1)Oc2ccsc2C=C(C#N)C#N KM05347 c1ccc(cc1)NC(=O)N(CCS(=O)(=O)c2ccc(cc2)Cl)Cc3cccs3 KM03768 Cc1cc(nc2c1c(nn2C)C)NNC(=O)c3cccc(c3)C(F)(F)F KM03973 CN1c2cc(ccc2C(=O)/C(=C/N(C)C)/S1(=O)=O)C(=O)OC KM07024 Cc1ccc(cc1)C(=O)NNC(=O)Cn2nc(nn2)c3ccccc3C(F)(F)F GK02995 CCOC(=O)c1cnc(nc1C(F)(F)F)O/N=C/c2ccc(cc2)C#N GK02997 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)Oc4ccc(cc4)Cl KM06864 COc1ccc(cc1)C(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-] KM06867 CSCCC(C(=O)NN)NS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F KM02714 c1ccc(c(c1)C(=O)O/N=C(/c2ccc3c(c2)non3)\N)Cl KM06760 COc1cc(cc(c1OC)OC)/C=N/c2cc(c(cc2OC)Cl)OC BTB00729 c1ccc(cc1)NC(=O)NNC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F KM09379 c1cc(ccc1C(=O)n2c(c(cn2)C#N)C3CC3)Cl KM09388 c1cc(cc(c1)Cl)NC(=O)O/N=C(/c2ccc3c(c2)non3)\N KM06734 CS(=N)(=O)c1ccc(cc1)Oc2ccc(cn2)[N+](=O)[O-] KM06668 c1cnc(cc1C(F)(F)F)N2CCC(CC2)C(=O)N KM08411 CC(C)(C#Cc1ccc(cc1)/C=N/Nc2cccc(n2)C(F)(F)F)O KM08414 Cn1c(cc(n1)c2ccc(s2)/C=N/NC(=O)c3ccc(cc3)Cl)C(F)(F)F KM05439 c1ccc(cc1)CN2CCC(CC2)OCCC(=O)N KM08299 CC(C)S(=O)(=O)c1cscc1N/C=C(/C#N)\C(=O)c2ccccc2 KM02734 COC(=O)c1c(c(c(s1)SC)C#N)c2cccc(c2)C(F)(F)F KM02741 CC(C)S(=O)(=O)c1cnc(nc1N)c2cccnc2 KM02598 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)N KM02600 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Sc3ccc(cc3)Cl KM08483 c1ccc(cc1)C#Cc2cc(cnc2)c3nc(no3)c4cccc(c4)C(F)(F)F KM08389 Cc1ccc(cc1)c2nc(on2)c3cc(cnc3)C#Cc4ccccc4 KM08390 CC1(CCC(N=C(N1)SCC(=O)c2ccc(cc2)Cl)(C)C)C.Br BTB02718 CC1(Cc2c(sc(c2C(=O)C1)SCCOC(=O)c3cccc(c3)C(F)(F)F)C#N)C KM05376 c1ccc2c(c1)C(=O)N(C2=O)c3cscc3S(=O)(=O)c4ccc(cc4)Cl KM05380 c1cc(oc1)CN(CCC(=O)NNC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM09405 CCOC(=O)c1cnc(nc1C(F)(F)F)O/N=C/c2ccc(cc2)F GK02998 Cn1c(nnc1Sc2c(ccs2)[N+](=O)[O-])C(F)(F)F KM05413 c1cc(sc1)Sc2c(ccs2)[N+](=O)[O-] KM05414 CCCCCCC#Cc1cc(cnc1)c2nnc(n2C)SCc3ccc(cc3)Cl KM09556 CS(=O)(=O)c1c(c(c(s1)Cl)c2ccc(cc2)Cl)C#N KM02725 Cc1c(c(sc1C(=O)O)SC)C(=O)C KM02728 COc1ccccc1NC(=O)c2cc(cnc2)C#Cc3ccccc3 KM08357 c1cc(oc1)CN(CCC(=O)N/N=C/c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM09409 c1ccc(cc1)C(=O)NNC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09410 c1cc(cc(c1)Cl)C(=O)O/N=C(/c2ccc3c(c2)non3)\N KM06761 c1cc2c(cc1C(=O)Nc3ccc(cc3F)F)non2 KM09558 COC(=O)c1c(c(c(s1)SC)C#N)c2ccc(cc2)F KM02648 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)N/N=C(\C#N)/S(=O)(=O)c2ccccc2 KM02660 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)N/N=C(\C#N)/S(=O)(=O)c2ccccn2 KM02661 c1ccc(cc1)OCCSCC(=O)N2CCCC2 KM06682 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4cc(ccn4)C(F)(F)F KM08425 c1cc(ccc1C(=O)NNC(=O)CN2c3cc(ccc3SCC2=O)C(F)(F)F)Cl KM08321 c1cc(sc1)SCC(=O)Nc2ccc(c(c2)Cl)F KM02687 c1cc(cc(c1)Cl)NC(=O)CSc2cccs2 KM02688 c1ccc(cc1)CN2CCC(CC2)n3c4c(cccn4)nn3 KM10142 CC(C)Sc1c(cccc1Cl)NC(=O)Nc2ccc(cc2)Cl KM10143 CCCCSc1c(c(c(s1)C(=O)OC)c2ccc(cc2)Cl)C#N KM02614 Cc1c(c(=O)n(n1C)c2ccccc2)/C=N/OC(=O)c3ccc(cc3)Cl KM03744 CS(=O)(=O)c1c2c(c(s1)C(=O)O)CCC=C2 KM03748 Cc1c(cco1)C(=O)C(=C2SCCCS2)C#N KM06595 CC(C)(C)c1cc2nc(cc(n2n1)Oc3ccc(cc3)Cl)C(F)(F)F KM08097 CC(C)(C)c1cc2nc(cc(n2n1)Oc3cccc(c3)C(F)(F)F)C(F)(F)F KM08099 c1ccc2c(c1)OCC(O2)/C(=N\OC(=O)c3cccc(c3)C(F)(F)F)/N KM06605 c1cc(oc1)CN(CCC(=O)NNS(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM09408 CC(C)N/C=C/1\C(=O)c2ccccc2N(S1(=O)=O)C KM01118 Cc1csc2c1c(c(s2)C(=O)C)C KM03621 c1cc(sc1)C2CC(=O)CS2 KM05246 C/S(=N\S(=O)(=O)c1cccc2c1non2)/c3ccc(cn3)C(F)(F)F KM08404 c1c(cnc(c1C(F)(F)F)N2CCC(CC2)C(=O)N)Cl KM08408 COC(=O)CSCCC(=S)N KM05434 CC(=O)N/N=C/c1ccc(s1)c2cc(n(n2)C)C(F)(F)F KM05438 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Oc3cccc(c3)C(F)(F)F KM08365 CC(C)Sc1c(cccc1Cl)NC(=O)Nc2cccc(c2)C(F)(F)F KM10139 Cc1cc(cc(c1)NC(=O)Nc2cccc(c2SC(C)C)Cl)C KM10141 CS(=NC(=O)Nc1ccc(cc1)Cl)(=O)c2ccc(cc2)Cl KM02601 CNC(=S)NNC(=O)c1c2c(c(s1)SC)C(CCC2)O KM03629 COc1ccc(cc1)NC(=O)c2ccc3c(c2)non3 KM09573 CCCCc1ccc(cc1)Nc2ncc(c(n2)C(F)(F)F)C(=O)OCC GK03049 CCCCC#Cc1ccc(o1)C(=O)NNC(=O)c2ccc(cc2)Cl KM09520 CCCCC#Cc1ccc(o1)C(=O)NNC(=O)Nc2ccccc2 KM09530 c1ccn(c1)C2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM09450 c1cc(sc1)c2cc(on2)C(F)(F)F KM09455 COC(=O)c1c(ccs1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM03711 CC(C)(C)S(=O)(=O)/C(=C/Nc1ccsc1C(=O)OC)/C#N KM03712 COC(=O)C(CCSC)NS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F KM02708 CCOC(=O)c1csc(n1)Cn2c(c(c(n2)C)Br)C KM03826 c1ccc(c(c1)CNC(=O)Nc2ccccc2[N+](=O)[O-])F KM09715 c1ccc(c(c1)CNC(=O)Nc2ccccc2C(F)(F)F)F KM09717 c1cc(sc1)CN(CCS(=O)(=O)c2ccc(cc2)Cl)C(=O)c3ccc(cc3)Cl KM03758 Cc1c(c(=O)n(n1C)c2ccccc2)/C=N/OC(=O)c3ccccc3Cl KM03762 Cc1cccc(c1NC(=S)N(Cc2ccccc2)Cc3cc(c(c(c3)OC)OC)OC)C BTB00728 CNC(=S)NNC(=O)CSCCOc1ccccc1 KM06492 CSc1c2c(c(s1)C(=O)NNC(=S)Nc3ccccc3Cl)CCCC2O KM03624 CC1(CCc2cc(ccc2O1)C3SCCS3)C KM05255 CC(=O)c1cc(c(cc1Cl)Cl)F BTB15028 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N=S(=O)(C)c3ccc(cn3)C(F)(F)F KM08418 Cc1ccc2c(c1NC(=O)Nc3cc(cc(c3)Cl)Cl)c(cc(n2)C(F)(F)F)OC KM08310 CCOC(=O)c1cc(cnc1)C#CCOC(=O)Nc2ccccc2 KM08314 CC(C)S(=O)(=O)c1csc(c1N/N=C(\C#N)/C(=O)c2ccc(cc2)Cl)C(=O)OC KM02608 COc1ccc(cc1)c2csc(c2C#N)S(=O)C KM02630 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccccc2F GK03025 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)Cl GK03026 c1ccc(cc1)Oc2ccsc2/C=C(\C#N)/C(=O)c3ccc(cc3)Cl KM05514 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Nc3cccc(c3)C(F)(F)F KM08355 c1cc2c(cc1C(=O)NN)non2 KM09589 c1cc(ccc1Nc2ccc(c3c2non3)[N+](=O)[O-])F KM06820 c1ccc(cc1)NC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09480 COc1ccc(cc1)CSc2ccc(c3c2non3)[N+](=O)[O-] KM06831 c1cc(c2c(c1[N+](=O)[O-])non2)SCCO KM06833 c1cc2c(cc1C(=O)NNC(=O)Nc3cc(cc(c3)Cl)Cl)non2 KM09657 c1cc(sc1)CNCCS(=O)(=O)c2ccc(cc2)Cl KM03720 CCCSc1c2c(c(s1)C(=O)OCC)CCCC2=O KM03728 CCOC(=O)C1CCN(CC1)c2nc3ccc(cc3s2)Cl AW00325 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2cccc(c2)C GK03046 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)C(C)(C)C GK03047 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Oc3ccc(cc3)Cl KM08363 COc1ccc(cc1)OC(=O)c2cc(cnc2)C#Cc3ccccc3 KM08366 c1cc2c(ccc(n2)C(F)(F)F)cc1CSCCOC(=O)Nc3cc(cc(c3)Cl)Cl KM08527 C/S(=N/C(=O)Nc1ccc(cc1)OC(F)(F)F)/c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06501 c1cc(c(cc1Cl)Cl)OCCSCC(=O)NN KM06504 c1cc(sc1)C(=O)n2c(c(cn2)C#N)C3CC3 KM09391 c1ccc(cc1)C2CCC(=O)/C(=C/Nc3ccccc3Cl)/C2=O KM05262 COC(=O)c1c(ccs1)N/C=C/2\C(=O)CCC(C2=O)c3ccccc3 KM05263 CCOC(=O)c1c(c(sc1N/C=C/2\C(=O)CCC(C2=O)c3ccccc3)C)C KM05264 Cc1ccc2c(c1NC(=O)Nc3ccccc3)c(cc(n2)C(F)(F)F)OC KM08312 COC(=O)c1c(c(cs1)C#N)N/N=C(\C#N)/C(=O)c2cccs2 KM02554 CC(C)c1ccc(cc1)NC(=O)CSc2cccs2 KM02699 CC(C)S(=O)(=O)c1cnc(nc1N)N KM02704 COC(=O)c1c(c(cs1)S(=O)(=O)Cc2cccs2)N/N=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM03814 Cc1cc(c(cc1Br)[N+](=O)[O-])NC(=O)C KM10164 c1ccc(cc1)C#Cc2ccc(s2)COC(=O)Nc3ccc(cc3)OC(F)(F)F KM08255 Cc1csc2c1c(c(s2)c3cc[nH]n3)C KM03754 COC(=O)c1c(ccs1)N/N=C(/C#N)\C(=O)c2ccc(cc2)Cl KM03677 COC(=O)c1ccccc1NC(=O)/C=N/O KM10109 c1cc(cc(c1)NC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F KM09509 CSc1c(c(cs1)c2cccc(c2)Cl)C#N KM02580 Cc1ccc(cc1)C2C3CCc4ccccc4C3=Nc5ccccc5S2 JFD02623 Cn1c(nnc1SCc2ccccc2)c3ccc4c(c3)non4 KM09729 c1ccc(cc1)NC(=O)c2ccc3c(c2)CCO3 KM07014 CS(=NC(=O)Nc1ccccc1)(=O)c2ccsc2 KM05774 CSc1nccc(n1)c2ccc(cc2)Cl KM05777 CCOC(=O)C1CN(C(=O)C1=O)Cc2ccco2 KM02778 c1ccc(cc1)NC(=O)NNC(=O)c2ccc3c(c2)non3 KM09654 CSc1c(c(c(s1)c2cc[nH]n2)c3cccs3)C#N KM05495 CC(C)S(=O)(=O)c1c(csc1SC)NC(=O)Nc2cccc(c2)Cl KM09228 CC(=O)NC(=O)/C(=C/Nc1ccccc1OC(F)(F)F)/C#N KM09230 c1cc(cnc1)c2cc(=O)n3c([nH]2)cc(n3)c4ccco4 KM09394 c1ccc(cc1)S(=O)(=O)CCSc2cccs2 KM02409 C1[C@@H]([C@@H]([C@H]([C@@H](O1)NN=C(N)N)O)O)O.N(=O)(=O)O RJC00059 c1cc(ccc1OCOc2ccc(cc2)F)F BTB05116 c1ccc2c(c1)C(CS2(=O)=O)Sc3cccs3 KM08138 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])SCC(=O)O KM08150 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)Nc3cccc(c3)Cl)C(F)(F)F KM08153 CC(=O)OCc1ccc(o1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM03715 CC(=O)OCc1ccc(o1)/C=C(/C#N)\S(=O)(=O)c2ccccn2 KM03716 c1cc(sc1)CN(CCS(=O)(=O)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)Cl KM03733 Cc1c(c(=O)n(n1C)c2ccccc2)/C=N/O KM03736 Cc1c(c(sc1C(=O)Oc2ccccc2)S(=O)(=O)C)C=C KM03738 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2cc(cc(c2)Cl)Cl GK03038 CCOC(=O)c1cc(cnc1)C#CCOC(=O)c2c(onc2c3ccccc3)C KM08361 C/C(=N/OC(=O)c1ccc(cc1)Cl)/c2ccc3c(c2)CCO3 KM06628 Cc1cc(no1)NC(=O)C2COc3ccccc3O2 KM06630 CC(C)S(=O)(=O)C(=C(SC)SC)C#N KM02595 C/C(=N/OC)/c1ccc2c(c1)CCO2 KM06637 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NNC(=O)c3ccc(cc3)Cl KM03689 COC(=O)c1c(ccs1)N/C=C(\C#N)/C(=O)c2ccccc2 KM03695 c1cc(sc1)c2c3c(cc(nc3[nH]n2)C(F)(F)F)O KM06804 Cn1c(nnc1SCc2c(cccc2Cl)Cl)c3ccc4c(c3)non4 KM09728 c1cc(ccc1Cn2cc(c(=O)[nH]c2=O)C#N)F KM09877 Cn1c(nnc1SCc2cc(cc(c2)F)F)c3ccc4c(c3)non4 KM09730 c1ccc(cc1)CN2CCN(CC2)CCS(=O)(=O)c3ccc(cc3)F KM09878 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)c4cc(nc5c4cccc5Cl)C(F)(F)F KM09879 c1ccc(c(c1)NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)Cl KM05634 COc1cc(c(s1)C(=O)OC)OC(=O)c2ccc(cc2Cl)Cl GK03014 c1ccnc(c1)CNS(=O)(=O)c2ccc(s2)S(=O)(=O)c3c(cc(cn3)C(F)(F)F)Cl KM05590 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2cc(ccc2OC)Cl GK03012 c1cc(cc(c1)Oc2c(nccn2)C#N)C(F)(F)F KM05504 Cn1c(cc(n1)c2ccc(s2)c3ccn(n3)C(=O)c4ccc(cc4)Cl)C(F)(F)F KM03848 CC(=O)n1ccc(n1)c2ccc(s2)c3cc(n(n3)C)C(F)(F)F KM03849 CNC(=S)N(CCS(=O)(=O)c1ccc(cc1)Cl)Cc2cccs2 KM03858 c1ccc(c(c1)C(CC(=O)O)N)[N+](=O)[O-] KM08101 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/CSc2cccs2)\N KM02410 Cc1ccc(cc1)S(=O)(=O)CCS(=O)(=O)c2cccs2 KM02415 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)Nc2ccccc2Cl KM02416 C/C(=N\OCc1ccc(cc1)Cl)/c2ccc3c(c2)CCO3 KM06634 c1cc(ccc1C2=C(C(=O)OC2)C#N)Cl KM06635 c1ccc(cc1)NC(=O)O/N=C(/c2ccc3c(c2)non3)\N KM06709 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccc(c(c2)Cl)C GK02957 CC(C)S(=O)(=O)c1c(c(sc1SCC#N)C#N)N KM03831 CCCCS(=O)c1c2c(c(s1)C(=O)OCC)CCCC2=O KM03839 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)/C=N/c3cccc(c3)C(F)(F)F KM05491 COC(=O)c1ccc(cc1)Br KM05492 c1cc(sc1)CNC(=O)c2ccc(cc2)Cl KM03841 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3cccnc3 KM09610 CCCCSc1c(c(c(s1)C(=O)O)c2ccc(cc2)Cl)C#N KM02616 CCCS(=O)(=O)c1cnc(nc1N)C KM02620 CCOC(=O)c1c(c(c(s1)SC(C)C)C#N)c2ccc(cc2)Cl KM02623 CC(C)S(=O)(=O)C/C(=N/OCc1ccc(cc1)Cl)/N KM05622 c1ccc(cc1)C#Cc2ccc(s2)COC(=O)c3cccs3 KM08267 CCOC(=O)C1CCN(CC1)/C=C(\C#N)/S(=O)(=O)c2ccccc2 KM08270 CCOC(=O)C1CCN(CC1)/C=C(\C#N)/S(=O)(=O)C(C)(C)C KM08271 CS(=O)(=O)c1c2c(c(s1)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)CCC=C2 KM03771 CS(=O)(=O)c1c2c(c(s1)C(=O)Sc3ccc(cc3)Cl)CCC=C2 KM03772 COc1cc(c(s1)C(=O)OC)OS(=O)(=O)c2ccc(cc2)Cl GK03019 c1ccc(cc1)Oc2ccsc2/C=N/Nc3ccc(cc3)Cl KM08451 Cc1cc(c(c(c1)C)S(=O)(=O)O)C.c1cc(sc1)S(=N)c2ccc(cc2)Cl KM05453 CN(CCOC(=O)c1ccc(cc1Cl)Cl)c2cc(nc3c2cccc3)C(F)(F)F KM08444 c1cc(ccc1NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)Cl KM05457 c1ccc(cc1)Oc2ccsc2/C=C(\C#N)/S(=O)(=O)c3ccc(cn3)C(F)(F)F KM05512 c1ccc(cc1)Oc2ccsc2/C=C(\C#N)/C(=O)C3CC3 KM05513 Cn1c(nnc1SCc2ccc(cc2)Cl)CN3c4cc(ccc4SCC3=O)C(F)(F)F KM08368 c1ccc(cc1)C(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-] KM06874 Cc1cc(nc2n1nc(c2[N+](=O)[O-])C(C)(C)C)C(F)(F)F KM02430 CC(C)(C)S(=O)(=O)C/C(=N/OS(=O)(=O)c1ccccc1C(F)(F)F)/N KM02279 c1cc(sc1)SC/C(=N/OC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/N KM02439 c1ccc(cc1)CN2CCC(CC2)Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F KM10117 c1cc(sc1)S(=O)(=O)/C(=N/OC(=O)c2ccc(cc2)C(F)(F)F)/C#N KM02561 CSc1c(c(c(s1)C(=O)NCc2cccs2)c3ccc(cc3)Cl)C#N KM01232 CCOC(=O)c1cnc(nc1C(F)(F)F)O/N=C/c2ccc(cc2Cl)Cl GK02999 c1ccc(cc1)N2CCN(CC2)C(=O)c3ccc4c(c3)cccn4 KM10135 Cn1c(cc(n1)c2ccc(s2)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl)C(F)(F)F KM03836 C/C(=N\OCc1cccc(c1)C(=O)N=S(=O)(C)c2ccccc2)/c3ccc(cc3)Cl KM06887 c1ccc2c(c1)/C(=C/C(=O)O)/OC2=O KM06895 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N)C(F)(F)F KM03853 c1cc(cc(c1)Oc2c(nccn2)C(=O)N)C(F)(F)F KM05505 c1ccc2c(c1)cc(o2)C(=O)Nc3ccc(cc3)Cl KM05508 Cn1c(cc(n1)c2ccccc2)NC(=O)C3COc4ccccc4O3 KM06661 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09412 COc1ccc(cc1)/C=N/NC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09419 COC(=O)c1c(cc(s1)c2cccs2)N GK03031 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2c(cccc2OC)OC GK03033 c1cc(ccc1CN2c3cc(ccc3SCC2=O)C(F)(F)F)F KM08280 CCOC(=O)c1cc(cnc1)C#Cc2ccccc2 KM08293 CC1(Cc2c(c(sc2Br)S(=O)(=O)C)C(=O)C1)C KM03791 c1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3ccccc3)N KM09679 c1ccc(cc1)S(=O)(=O)c2cnc(nc2N)C3COc4ccccc4O3 KM09680 Cc1c(cnc(n1)C2COc3ccccc3O2)S(=O)(=O)c4ccc(cc4)Cl KM09686 c1cc(cc(c1)NC(=O)c2ccc3c(c2)non3)C(F)(F)F KM09572 c1cc(ccc1NC(=O)c2ccc3c(c2)non3)Cl KM09574 Cc1c(csc1C(=O)OC)S(=O)(=O)c2ccc(cc2)Cl KM01184 CSc1c(c(c(s1)C(=O)O)c2ccc(cc2)Cl)C#N KM01185 COc1ccc(cc1)c2c(c(sc2C(=O)OC)SC)C#N KM02603 CCOC(=O)c1cnc(nc1C(F)(F)F)O/N=C(/c2ccc(cc2)C(C)(C)C)\N GK03000 Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2NS(=O)(=O)c3ccc(cc3)C)Br)C KM10138 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CCS(=O)(=O)c4ccc(cc4)Cl KM09883 Cc1c(csc1S(=O)(=O)NNC(=O)c2cccc(c2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM03928 CC1(CCc2cc(ccc2O1)c3cc[nH]n3)C KM05595 CN(C)CC#Cc1cc(cnc1)C(=O)NNC(=O)Nc2ccc(cc2)Cl KM08436 CN(CCOC(=O)c1ccccc1)c2cc(nc3c2cccc3)C(F)(F)F KM08441 c1ccc(cc1)Sc2ccc(s2)S(=O)(=O)N KM03857 Cc1cc(ccc1NC(=S)NNC(=O)c2ccccc2Cl)Cl BTB01231 Cn1c(nnc1SCC(=O)c2ccccc2)CN3c4cc(ccc4SCC3=O)C(F)(F)F KM08374 COc1ccc(cc1)S(=O)(=O)NNC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09422 Cc1c(nc(nc1O)N(C)C)C KM09428 CCCCC#Cc1cc(cnc1)C(=O)NN KM09438 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)[N+](=O)[O-] GK03040 Cc1c(c(n(n1)Cc2nnc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C)Br KM03796 c1ccnc(c1)c2ccc(s2)C(=O)N3CCOCC3 KM02526 CC1(OC(=O)C(=CNc2ccccc2OC)C(=O)O1)C KM02530 c1cc(sc1S(=O)(=O)N)Br KM03804 Cn1c(cc(n1)c2ccc(s2)c3cc[nH]n3)C(F)(F)F KM03800 CC(=O)N(CCS(=O)(=O)c1ccc(cc1)Cl)Cc2cccs2 KM03803 c1ccc(cc1)NC(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-] KM06884 c1cc(oc1)CNc2ccc(c3c2non3)[N+](=O)[O-] KM06885 c1cc(ccc1OC(=O)c2ccc3c(c2)non3)Cl KM09588 c1cc(c(c(c1)F)F)OC(=O)c2ccc3c(c2)non3 KM09596 Cc1c(c(on1)NC(=O)c2c(onc2c3c(cccc3Cl)F)C)[N+](=O)[O-] KM03742 CS(=O)(=O)c1c2c(c(s1)C(=O)Nc3ccc(cc3)Cl)CCC=C2 KM03751 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)O)N KM02606 COc1ccc(cc1)c2c(c(sc2C(=O)O)SC)C#N KM02613 c1ccc(cc1)c2cc([nH]n2)NC(=O)C3COc4ccccc4O3 KM06646 CC(C)(C)c1cc([nH]n1)NC(=O)C2COc3ccccc3O2 KM06647 c1cc(ccc1[N+](=O)[O-])Oc2ccc(cc2)Cl KM08443 CC1(Cc2c(sc(c2C(=O)C1)S(=O)(=O)C)C#N)C KM03776 CCOC(=O)C1CCN(CC1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM08272 c1cc2c(cc1C(F)(F)F)N(C(=O)CS2)Cc3ccc(cc3Cl)Cl KM08279 Cc1ccc(cc1)S(=O)(=O)Oc2cc(sc2C(=O)OC)OC GK03022 CN(C)/C=C/C(=O)c1c(c(c(s1)SC)C#N)c2cccs2 KM05460 CN(CCOC(=O)c1cccc(c1)C(F)(F)F)c2cc(nc3c2cccc3)C(F)(F)F KM08456 CNC(=S)NNC(=O)c1cc(cnc1)C#Cc2ccccc2 KM08457 COc1ccc(cc1OC2CCCC2)/C(=N/O)/N KM09557 c1cc(sc1)CNS(=O)(=O)c2ccc(cc2)Cl KM06879 CCOC(=O)c1c2c(c(s1)SC)C(=O)CC(C2)c3ccc(cc3)OC KM03646 CCOC(=O)c1c2c(c(s1)S(=O)(=O)C)-c3c(cno3)CC2 KM05486 CCOC(=O)c1c[nH]c2cc(cc(c2c1=O)Cl)Cl BTB03757 Cc1ccc(cc1)c2c(c(sc2C(=O)OC)SC)C#N KM02542 CS(=O)c1c(c(cs1)c2ccc(cc2)Cl)C#N KM02545 COC(=O)c1c(c(cs1)C#N)N/N=C(\C#N)/S(=O)(=O)c2cccs2 KM02549 CN(C)c1ccc(c2c1non2)[N+](=O)[O-] KM06827 CC(=O)OCc1ccc(o1)/C=C(\C#N)/S(=O)(=O)c2cccs2 KM03714 COC(=O)c1c(c(cs1)S(=O)(=O)Cc2cccs2)N/N=C(\C#N)/S(=O)(=O)c3cccs3 KM03813 CC1(Cc2c(c(sc2C(=O)OC)SC)C(=O)C1)C KM02609 c1cc(c(cc1Cl)Cl)NC(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-] KM06900 Cc1cccc(c1)C(=O)NCCCNC(=O)c2cccc(c2)C JFD02665 CCCCCCC#Cc1cc(cnc1)c2nnc(n2C)SCc3cc(cc(c3)F)F KM09586 Cn1c(cc(n1)c2ccc(s2)/C=C(\C#N)/S(=O)(=O)c3ccc(cn3)C(F)(F)F)C(F)(F)F KM05312 Cn1c(cc(n1)c2ccc(s2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F KM05313 Cc1nc(nc(n1)SC)N/C=C(\C#N)/C(=O)c2ccccc2Cl KM01104 CN1c2ccccc2-c3c(c(sc3C(=O)Nc4ccc(cc4)Cl)SC)S1(=O)=O KM03780 Cn1c(cc(n1)c2ccc(s2)C(=O)/C=C/N(C)C)C(F)(F)F KM03793 c1cc(cc(c1)NC(=O)CN2c3cc(ccc3SCC2=O)C(F)(F)F)C(F)(F)F KM08294 CSc1c(c(c(s1)c2ccno2)c3ccccc3)C#N KM05462 Cc1ccccc1NC(=O)NCc2ccco2 KM09687 Cc1ccccc1NC(=O)N(Cc2ccco2)C(=O)CC#N KM09697 CCOC1O[C@@H]2[C@H](O[C@H]([C@@H]2O1)n3cnc4c3ncnc4N)CO KM09581 Cc1ccc(cc1)/S(=N/C(=O)c2cccc(c2)CO/N=C(\C)/c3ccc(cc3)Cl)/C KM06888 c1cc(ccc1NC(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-])F KM06891 c1cc(cc(c1)S(=O)(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-])C(F)(F)F KM06894 Cc1ccc(cc1)S(=NC(=O)c2cc3ccccc3o2)(=O)C KM05488 COC(=O)c1c(ccs1)N/N=C(/C#N)\C(=O)C2CC2 KM03676 Cn1c(nnc1SCc2ccccc2)CN3c4cc(ccc4SCC3=O)C(F)(F)F KM08367 c1ccc(cc1)OCCSCC(=O)NCc2ccccn2 KM06693 c1ccc(cc1)OCCSCC(=O)NCc2cccnc2 KM06694 CN(C)CC#Cc1ccc(cc1)C=C(C#N)C#N KM08325 c1cc(sc1)C(=O)NNC(=O)CSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-] KM08320 Cc1ccc(cc1)C2C3Cc4ccccc4C3=Nc5ccccc5S2 JFD02637 c1cc(sc1)CN(CCS(=O)(=O)c2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM03730 c1cc(sc1)CS(=O)(=O)CC#N KM03732 c1ccc(c(c1)Cn2c(=O)cc(n(c2=O)c3ccccc3F)N)F KM09713 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Nc3ccccc3 KM08356 c1cc(ccc1NC(=O)NNC(=O)CN2c3cc(ccc3SCC2=O)C(F)(F)F)Cl KM08358 CC(C)S(=O)(=O)c1cnc(nc1N)N2CCOCC2 KM02590 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)C=C(C#N)C#N KM05331 CC1(CCc2cc(ccc2O1)/C=N/OC(=O)Nc3ccc(cc3)Cl)C KM05213 CC1(CCc2cc(ccc2O1)/C=N/OC(=O)Nc3ccc(cc3)OC(F)(F)F)C KM05215 CC1(Cc2c(c(sc2C(=O)OC)SCCOC(=O)c3ccccc3Cl)C(=O)C1)C KM05228 COC(=O)c1c(c(cs1)C#N)N/N=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM02524 CCOC(=O)c1c2c(c(s1)SCC=C)C(=O)CCC2 KM03795 COC(=O)c1c(c(cs1)C#N)N/N=C(\C#N)/C(=O)c2ccccc2 KM02532 c1cc(sc1)S(=O)(=O)/C(=N/OS(=O)(=O)c2ccc(cc2)Cl)/C#N KM02539 CCOC(=O)c1ccc2c(c1)non2 KM09541 COc1ccc(cc1)c2c(c(sc2Br)S(=O)(=O)C)C#N KM02723 c1cc(sc1)CS(=O)(=O)c2cnc(nc2N)N KM03805 Cc1c(c(n(n1)Cc2nnc(o2)c3cccs3)C)Br KM03810 COC(=O)c1c(ccs1)N/C=C(\C#N)/S(=O)(=O)C KM03710 CC(C)Sc1ccc(cc1[N+](=O)[O-])C(F)(F)F KM10169 CCCc1ccc(cc1)NC(=S)OC NH00697 c1cc(ccc1C2CCCCC2)NC(=S)NCCO NH00700 COC(=O)c1cc(cc(c1c2c(cc(cc2Cl)Cl)C(=O)OC)Cl)Cl JFD02706 CCCCCCCOc1ccc(cc1)/C(=N\O)/c2ccccc2 JFD03016 C1CN=C(N1)N2CCOCC2 NH00798 Cn1c(nnc1SCC(=O)Nc2cccc(c2)Cl)c3ccc4c(c3)non4 KM09763 c1ccc(cc1)CN2CCC(CC2)COCCC#N KM09628 c1ccc(cc1)/C=N/NC(=O)c2ccc3c(c2)non3 KM09651 COc1ccc(cc1)NC(=S)NC(=O)c2ccc3c(c2)non3 KM09783 CC1(Cc2c(c(sc2c3ccnc(n3)SCC(=O)C(C)(C)C)SC)C(=O)C1)C KM03983 c1ccc(cc1)C#Cc2cc(cnc2)NC(=O)N3CCCCC3 KM08629 Cc1c(nc(s1)c2ccccc2)CC(=O)NNC(=O)c3cccc(c3)OC(F)(F)F RH01238 Cc1ccc(cc1)SC(=O)c2ccc(o2)C#Cc3ccccc3 KM08669 c1ccc(cc1)C#Cc2ccc(o2)C(=O)Sc3ccccc3 KM08670 CN(C)CC1COc2ccccc2C1=O.Cl KM07079 Cn1c(cnc1SC)c2nnc(n2C)S KM07080 C1C2C(=O)NC(=O)N2CS1 KM08712 Cn1c(nnc1S)C(CCSC)NC(=O)c2ccc(cc2)C(F)(F)F KM07069 CC1(Cc2csc(c2/C(=N/OC(=O)Nc3ccc(cc3)Cl)/C1)SC)C KM03900 c1cc(cc(c1)C(F)(F)F)C(=O)/C(=C/c2ccco2)/C#N KM03904 Cn1c(cnc1SC)C(=O)NN KM07075 c1ccc2c(c1)OCC(O2)C(=O)N3CCNCC3.Cl KM08535 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC3CCSC3=O KM03961 CCOC(=O)c1cc(c(s1)SC)S(=O)(=O)C(C)C KM03963 CC1(CCc2cc(ccc2O1)c3ccn(n3)S(=O)(=O)c4cccc(c4)C(F)(F)F)C KM05616 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)C#N JFD02862 CCOC(=O)C(=CNc1cc(ccc1Oc2cc(c(c(c2)C)Cl)C)C(F)(F)F)C(=O)OCC BTB02802 c1cc(c(cc1S(=O)(=O)NC2CCSC2=O)Cl)Cl KM03863 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NC2CCSC2=O)C(F)(F)F KM03864 c1cc(sc1)/C=N/NC(=O)c2ccc3c(c2)non3 KM09652 CS(=O)(=O)c1c2c(c(s1)C(=O)Nc3ccccc3Cl)CCC=C2 KM03770 CS(=O)(=O)c1c2c(c(s1)C(=O)Sc3ccccc3)CCC=C2 KM03773 CC(=O)c1cc(c(s1)Nc2ccccc2)[N+](=O)[O-] KM08539 CN(C)/C=C(\C#N)/c1csc2c1cc(cc2)Cl MWP00265 Cc1ccccc1NC(=O)NCc2ccccc2[N+](=O)[O-] KM09836 c1ccn(c1)C2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] KM08678 CC1(Cc2c(c(sc2c3ccnc(n3)SCC(=O)Nc4ccccc4Cl)SC)C(=O)C1)C KM03975 Cn1c(nnc1SCC(=O)c2ccccc2)C3COc4ccccc4O3 KM07026 COC(=O)c1c(ccs1)N/C=C(\C#N)/C(=O)c2cccc(c2)CSc3ccccc3 KM05732 CCO/C(=N\OC(=O)c1c(onc1c2c(cccc2Cl)F)C)/C KM05734 CC(C)(C)S(=O)(=O)c1cnc(nc1N)N2CCCC2 KM02634 CCCSc1c(c(cs1)c2ccc(cc2)Cl)C#N KM02639 CC1(CC(=CC(=S)S1)N2CCCCC2)C KM03891 CCOC(=O)c1c2c(c(s1)SCC)C(=O)CC(C2)(C)C KM03785 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)CN3c4cc(ccc4SCC3=O)C(F)(F)F KM08373 Cn1c(nnc1SCC(=O)Nc2ccccc2)CN3c4cc(ccc4SCC3=O)C(F)(F)F KM08376 CCc1cccc(c1NC(=O)NNC(=O)Cc2c(sc(n2)c3ccccc3)C)C RH01256 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)N3CCOCC3 KM03979 c1ccc(cc1)C#Cc2cccc(c2)/C=C\3/C(=O)NC(=O)S3 KM08711 CCOC(=O)NC(=O)/C(=N/Nc1ccccc1)/C#N KM08714 c1cc(sc1)Sc2ccc(s2)S(=O)(=O)N KM05739 Cc1c2c(c(sc2sc1C(=O)C)Br)C KM03880 CN1c2ccccc2C(=O)/C(=N\Nc3ccsc3C(=O)OC)/S1(=O)=O KM03885 CSc1c-2c(cs1)CCc3c2n[nH]c3 KM03777 c1cc(sc1c2cc(on2)C(F)(F)F)S(=O)(=O)N3CCOCC3 KM09812 c1ccc(cc1)C(=O)OCCSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-] KM08437 Cc1ccccc1n2c(cc(=O)n(c2=O)Cc3cccs3)N KM09693 Cc1ccccc1n2c(cc(=O)n(c2=O)Cc3ccco3)N KM09698 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)NCc3cccs3)C(F)(F)F KM03895 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N3CCCCC3 KM03985 C/C(=N\Nc1nc(cs1)C(C)(C)C)/c2ccc(cc2)Br.Br BTB05166 CC(C)N(Cc1ccc(cc1)N(C)C)S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl BTB01296 C/C=C(\C)/C(=O)Nc1ccc(cc1)N2CCOCC2 BTB01789 c1cc(ccc1F)S(=O)(=O)C/C(=N/OC(=O)Nc2cc(cc(c2)Cl)Cl)/N KM08565 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)O)I KM02656 c1cc(sc1)CNC(=S)NN NH00538 CC1(CC(=O)c2ccc(cc2O1)OCc3ccc(cc3)[N+](=O)[O-])C RJC00184 c1cc(cc(c1)NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)C(F)(F)F KM05633 C/C(=N\N=C(\N=C\N(C)C)/SC)/c1ccc(cc1)Br BTB05189 C/C(=C\c1ccccc1)/C(=N/O)/C NRB01487 CSc1c(cn(n1)c2ccccc2)c3nc(cs3)c4ccccc4 KM08395 c1cc(ccc1CSCC(=O)Nc2ccc(cc2)F)Cl NRB00081 CC(C)(C)S(=O)(=O)c1cnc(nc1N)N2CCOCC2 KM02635 CN1c2ccccc2-c3c(sc(c3S1(=O)=O)SC)C#N KM03854 c1cc(cc(c1)F)NC(=S)N(CCS(=O)(=O)c2ccc(cc2)Cl)Cc3cccs3 KM03859 CC(C)N(Cc1ccc(cc1)N(C)C)C(=S)Nc2ccc(cc2)F BTB01070 COC(=O)c1c(ccs1)O SB01952 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)N/N=C(\C#N)/C(=O)c2ccccc2 KM02651 Cc1cc(c(c(n1)O)C#N)C(F)(F)F RF01004 Cc1cc(c2cc(ccc2n1)Br)C(=O)N/N=C(/C)\c3ccccc3O BTB01806 c1cc(oc1)C(=O)N/N=C\2/c3cc(ccc3NC2=O)Br ML00454 C/S(=N\S(=O)(=O)c1cccc2c1nsn2)/c3ccc(cn3)C(F)(F)F KM08402 CC(C)/C(=N/O)/c1ccc(cc1)[N+](=O)[O-] NRB02331 Cc1ccc(cc1)S(=O)(=O)/N=S(\C)/c2ccc(cn2)C(F)(F)F KM05635 CC1(Cc2csc(c2/C(=N/OC(=O)Nc3ccccc3)/C1)SC)C KM03899 CC1(CC(=O)C=C(S1)SCC(=O)Nc2ccc(cc2)Cl)C KM03950 CC1(CC(=O)C=C(S1)SCc2cccc(c2)Cl)C KM03952 Cc1csc2c1c(c(s2)C(=O)C=C(SC)SC)C KM03913 Cc1cc(c2nncn2n1)O KM03809 c1cc(c(cc1F)Cl)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05411 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])OC(=O)c2ccc(cc2Cl)Cl BTB05422 c1cc(sc1)C2=NN(CC2)CCC(=O)c3cccs3 KM06917 c1ccc(cc1)C(=O)N2CCC(CC2)n3cccc3 KM08578 c1ccn(c1)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM08584 CNC(=O)c1cnn2c1nc(cc2C(F)(F)F)C(F)(F)F KM05656 c1cc(ccc1C#N)Oc2c(ccs2)[N+](=O)[O-] KM05662 c1cc2c(cc1Cl)non2 KM06670 C/C(=N\OCc1cccc(c1)C(=O)OC)/c2ccc(c(c2)OC)OC KM06674 c1cc2c(cc1/C(=N/O)/N)non2 KM06678 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)N/N=C(/C#N)\C(=O)c2ccc(cc2)C(C)(C)C KM02657 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccc(c(c2)Cl)OC GK03051 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2c3nnc(o3)c4cc(ccc4Br)OC BTB06960 c1cc(oc1)c2ccnc(n2)SCc3ccc(cc3)[N+](=O)[O-] MWP00520 c1cc(sc1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)F KM08540 c1cc(ccc1CSC2C(C3CCN2CC3)C(=O)NNS(=O)(=O)c4ccc(cc4Cl)Cl)Cl.Cl KM06921 c1cc(cc(c1)OC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)C(F)(F)F KM05642 CCC1=C2CCC3C4CC[C@](C4(CCC3C2(CCC1=O)C)C)(C)O NRB03850 CCOC(=O)c1csc(n1)c2ccc3c(c2)non3 KM06809 CCOC(=O)CC1C(=Nc2ccccc2S1)SCC(=O)Nc3ccc(cc3Cl)Cl KM06811 CSc1c2c(c(s1)Br)CCCC2=O KM03816 Cc1c(c(n(n1)Cc2nc(cs2)c3cccc(c3)[N+](=O)[O-])C)Br KM03819 CN1c2ccccc2SC(CC1=O)c3ccsc3 MWP00645 CCOC(=O)CC(C)Nc1cc(ccc1OC)NC(=O)C NRB02089 CC(=O)c1cc(c(s1)Nc2ccc(cc2)Cl)[N+](=O)[O-] KM08549 c1cc(ccc1NC(=O)Nc2ccc3c(c2)C(=O)OC3)Cl KM08477 c1cc2c(cc1NC(=O)Nc3cc(cc(c3)Cl)Cl)C(=O)OC2 KM08479 c1cc(c(cc1N/N=C(\C#N)/C(=O)C2CC2)Cl)F KM06939 CSCCC(C(=O)NNC(=O)c1ccc(cc1)Cl)NC(=O)c2ccc(cc2)C(F)(F)F KM02870 C/C(=N\OCc1cccc(c1)C(=O)Sc2ccc(cc2)C(F)(F)F)/c3ccc(c(c3)Cl)Cl KM06745 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccncc4 KM09407 c1cc(oc1)C(=O)/C(=C/Nc2ccc(cc2)OC(F)(F)F)/C#N KM03616 CC1(Cc2csc(c2C(=O)C1)SC)C KM03636 CSc1nccc(n1)c2ccc(s2)S(=O)(=O)N(CCC#N)Cc3ccco3 KM09445 c1cc2c(c(c1)S(=O)(=O)N(CCC#N)Cc3ccco3)non2 KM09446 CCCCC#Cc1cc(cnc1)C(=O)N/N=C/c2ccccc2 KM09447 CCCCC#Cc1cc(cnc1)C(=O)NNC(=O)c2ccc(cc2)Cl KM09456 CC(C)S(=O)(=O)C/C(=N/OCc1cccc(c1)Cl)/N KM05631 CC(C)S(=O)(=O)C/C(=N/OCc1c(cccc1Cl)Cl)/N KM05632 c1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccc(s3)Br KM08556 c1cc(c(cc1Cl)S(=O)(=O)n2ccc(n2)c3ccc(s3)Br)Cl KM08557 CC(C)S(=O)(=O)c1csc(c1Cl)C(=O)N KM02856 CC(C)(C)C(=O)/C(=N/Nc1ccc(cc1)F)/C#N KM06940 C/C(=N\OCc1cccc(c1)C(=O)Sc2ccc(cc2)C(F)(F)F)/c3ccc(c(c3)OC)OC KM06943 CCOC(=O)CC1C(=Nc2ccccc2S1)SCC(=O)Nc3cccc(c3)C(F)(F)F KM06812 c1ccc(cc1)C(=O)c2cccc(c2)Cl SB01950 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)F)/C#N)Cl KM06945 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)Cl)/C#N)Cl KM06946 Cc1cccc(c1)Nc2ccc(c3c2non3)[N+](=O)[O-] KM06836 c1cc(cc(c1)Cl)Sc2ccc(c3c2non3)[N+](=O)[O-] KM06838 CCC(C)Sc1c(c(c(s1)C(=O)OCC)c2ccc(cc2)Cl)C#N KM02807 CCC(C)Sc1c(c(c(s1)C(=O)O)c2ccc(cc2)Cl)C#N KM02811 c1ccc(cc1)C(=O)/C(=C/Nc2ccc3c(c2)C(=O)OC3)/C#N KM08491 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Sc3ccc(cn3)C(F)(F)F KM08498 c1cc(ccc1OS(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F)Cl KM09802 c1cc(cc(c1)OS(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F)C(F)(F)F KM09809 CSCCC(C(=O)NNS(=O)(=O)c1ccccc1Cl)NC(=O)c2ccc(cc2)C(F)(F)F KM02888 CSCCC(C(=O)NNS(=O)(=O)c1ccc(cc1)Cl)NC(=O)c2ccc(cc2)C(F)(F)F KM02889 c1cc(ccc1NS(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F)Cl KM09560 CCCCCCC#Cc1cc(cnc1)c2nnc(n2C)SCc3c(cccc3Cl)Cl KM09568 c1cc2c(cc1[N+](=O)[O-])C(=O)OC2 KM08350 c1ccc(c(c1)CN/C(=C(\C#N)/N)/C#N)Sc2ccc(cc2)Cl KM03637 CCCCCCC#Cc1cc(cnc1)NC(=O)N2CCN(CC2)c3ccccc3 KM09587 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCC(CC3)n4cccc4 KM09467 c1cc(c2c(c1N3CCOCC3)non2)[N+](=O)[O-] KM06823 Cc1ccc(cc1)Nc2ccc(c3c2non3)[N+](=O)[O-] KM06826 c1cc(c(cc1Cl)Cl)Sc2ccc(c3c2non3)[N+](=O)[O-] KM06828 c1cc2c(cc1C(=O)O)CCO2 CC00801 c1cc(oc1)c2cc([nH]n2)NC(=O)Nc3cc(cc(c3)Cl)Cl KM08488 c1cc(sc1)c2cc([nH]n2)NC(=O)Nc3ccc(cc3)OC(F)(F)F KM08495 CC(C)S(=O)(=O)c1c(c(sc1SC)Br)Cl KM02812 CC(C)S(=O)(=O)c1c(c(sc1SC)Cl)Cl KM02815 Cc1c2c(c(cnc2n(n1)C)C(=O)Nc3ccc(cc3)Cl)OC KM02882 CC(c1ccccc1)NC(=O)c2cc(c(c(c2)OC)OC)OC JFD02693 c1ccc(cc1)/C(=C/C(=C/2\C(=O)N=C(S2)N3CCCC3)/c4ccc(cc4)Br)/CC(=O)c5ccc(cc5)Br JFD03035 c1cc(sc1c2cc(on2)C(F)(F)F)S(=O)(=O)N3CCCC3 KM09814 c1ccc(cc1)CN2CCC(CC2)N/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM08513 c1cc(ccc1SCc2ccc3c(c2)ccc(n3)C(F)(F)F)Cl KM08517 CCOC(=O)c1c(c(c(s1)SCC(C)C)C#N)c2ccc(cc2)Cl KM02819 Cc1c(c(no1)c2ccccc2)C(=O)N=S(=O)(C)c3ccccc3 KM02826 CC1CN(CC(O1)C)c2ccc(cc2)NC(=S)N3CCSCC3 NH00688 Cc1c(nc(s1)c2ccccc2)CC(=O)NNC(=O)c3cc(c(c(c3)OC)OC)OC RH01236 Cc1ccc(cc1)n2c(nnn2)c3cnoc3c4ccc(cc4)Cl JFD03042 c1ccc(cc1)n2c(nnn2)c3cnoc3c4ccc(c(c4)Cl)Cl JFD03045 Cn1c(nnc1SCC(=O)Nc2ccc(c(c2)Cl)F)c3cc(cnc3)C#Cc4ccccc4 KM08501 Cn1c(nnc1SCc2ccc(cc2Cl)Cl)CN3c4cc(ccc4SCC3=O)C(F)(F)F KM08370 c1cc(ccc1COc2ccc(cc2)S(=O)(=O)c3ccc(cc3)OCc4ccc(cc4)Br)Br BTB05049 c1cc(cc(c1)OC(=O)c2ccc3c(c2)non3)C(F)(F)F KM09595 c1ccc(cc1)CNC(=O)Nc2ccc(cc2)Cl KM09659 c1ccc2c(c1)OCC(O2)C(=N)N.Cl KM09660 CCc1cc2c3ccccc3ccc2c4c1cccc4 KM09662 c1ccc(cc1)OC(=O)c2csc(n2)C3COc4ccccc4O3 KM06865 CCC(C)S(=O)(=O)c1c(c(cs1)c2ccc(cc2)Cl)C#N KM02816 CCOC(=O)C(=CNc1cscc1S(=O)(=O)C(C)C)C(=O)OCC KM02817 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3cc(cnc3)C#Cc4ccccc4 KM08497 CSCCC(C(=O)N/N=C/c1cccs1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02751 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F KM09815 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)S(=O)(=O)c4ccc(s4)c5cc(on5)C(F)(F)F KM09819 c1ccc(cc1)n2c(cc(n2)C3CC3)NC(=O)Nc4ccc(cc4)OC(F)(F)F KM09824 c1cc(cc(c1)Cl)N2CCN(CC2)CCCSc3ccc(cc3)Cl KM08504 CC(C)S(=O)(=O)c1cnc(nc1N)N2CCCCC2 KM02674 CCCCc1ccc(c(c1)C)Nc2ncc(c(n2)C(F)(F)F)C(=O)OCC GK03050 c1ccc2c(c1)c(n[nH]c2=O)CC(=O)O KM06914 CCCCCCC#Cc1cc(cnc1)C(=O)Nc2ccc(cc2)Cl KM09497 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)NCc4cccs4 KM06857 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)NCc4ccco4 KM06859 c1ccc(c(c1)CNC(=O)Nc2ccccc2F)F KM09699 c1ccc(c(c1)CNC(=O)NC2CCCCC2)F KM09704 c1ccc(cc1)Cn2cc(c(=O)[nH]c2=O)C#N KM09852 c1ccc(c(c1)Cn2cc(c(=O)[nH]c2=O)C#N)Cl KM09855 CSCCC(C(=O)NNC(=O)c1cccs1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02757 CCCc1ccc(cc1)NC(=S)NCCO NH00703 C/C=C(\C)/C(=O)Nc1cc(ccc1n2cccc2)C BTB01780 c1ccc(cc1)CSc2[nH]c(=S)c(c(n2)c3ccccc3)C#N JFD03060 c1cc(sc1c2csc(n2)N)Cl RH01263 CCO/C(=N/OC(=O)Nc1ccc(cc1)OC(F)(F)F)/C KM05750 c1ccc(cc1)CN2CCC(CC2)N/C=C(\C#N)/S(=O)(=O)c3ccccn3 KM08516 c1cc(ccc1/C=N/NC(=O)c2ccc3c(c2)non3)Cl KM09633 CCCS(=O)(=O)c1csc(c1NNC(=O)c2ccccc2Cl)C(=O)OC KM02501 CCOC(=O)c1c2c(c(s1)SCc3ccccc3)/C(=N/O)/CC(C2)c4ccc(cc4)OC KM03688 COc1ccc(cc1)CSC2C(C3CCN2CC3)C(=O)NNC(=O)c4ccc(cc4Cl)Cl.Cl KM06977 Cc1ccc(cc1)NC(=O)c2cc(cc3c2OCC3)Br KM06978 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)c4c(nccn4)C#N KM09850 CSc1ccccc1NC(=O)NCc2ccccc2F KM09722 Cc1ccccc1NC(=O)NC(=O)CC#N KM09723 CCOC(=O)c1cnc2c(csc2c1Sc3ccc(cc3)Cl)S(=O)(=O)C(C)C KM02829 COc1ccc(cc1)C(=O)Oc2ccc3c4ccccc4c(=O)oc3c2 JFD02978 CCCCCCCCCCCCNC(=S)NNC(=O)Cc1c(sc(n1)c2ccccc2)C RH01257 Cc1cccc(c1)Nc2c(nc3ccccc3n2)/C=C/c4cccs4 JFD03054 Cn1c(nnc1SCc2ccc3c(c2)ccc(n3)C(F)(F)F)C(F)(F)F KM08520 CCCCCCC#Cc1cc(cnc1)C(=O)Nc2ccc(cc2F)F KM09500 CCOC(=O)Cc1c2ccccc2c(=O)[nH]n1 KM06915 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccccc2Br GK03048 CCCCC#Cc1ccc(o1)C(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F KM09533 c1ccc(cc1)N2CCN(CC2)c3c(nccn3)C#N KM09857 Cc1ccccc1n2c(cc(=O)n(c2=O)Cc3ccccc3)N KM09709 CC1(CC(=C(C(=O)C1)Sc2ccc(cc2)[N+](=O)[O-])OC(=O)c3ccc(cc3)F)C JFD03012 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NC(=O)c3c(cccc3F)F BTB02071 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NC(=O)c3ccco3 BTB02073 c1ccn(c1)C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F KM08690 CCOC(=O)c1cnc2cc(c(cc2c1Sc3ccc(cc3)Cl)F)Cl BTB03787 CCOC(=O)c1cnc2cc(c(cc2c1N3CC(OC(C3)C)C)F)Cl BTB03788 CCOC(=O)c1cnc2cc(c(cc2c1N3CCOCC3)F)Cl BTB03789 COc1ccc2c(c1)cc(o2)C(=O)c3ccc(cc3)Cl BTB02899 COc1ccc2cc(oc2c1)C(=O)c3ccc(cc3)Cl BTB02900 Cc1cc(n2c(n1)cc(n2)C(C)C)C(F)(F)F KM06786 CC(C)(C)c1ccccc1n2c(cc(=O)n(c2=O)Cc3ccccc3F)N KM09806 c1ccc(cc1)/C=N/NC(=O)CSCCc2nc(cs2)c3ccc(cc3)Cl KM05529 c1cc(ccc1S(=O)(=O)CCC2CCCCC2=O)Cl KM05533 COc1ccc(cc1)OS(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F KM09808 COc1ccccc1CCn2cc(c(=O)[nH]c2=O)C#N KM09859 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)CCS(=O)(=O)c4ccc(cc4)F KM09864 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)N3CCOCC3 KM09871 Cc1ccccc1n2c(cc(=O)[nH]c2=O)N KM09724 COc1ccc(cc1)/C(=C\C=C(C#N)C#N)/Sc2nc3ccccc3s2 JFD03032 CSCCC(C(=O)N/N=C/c1ccc(cc1)Cl)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02769 C/C(=N/OCc1cccc(c1)C(=O)Oc2ccc(cc2)C(F)(F)F)/c3ccc(c(c3)OC)OC KM06871 c1ccn(c1)C2CCN(CC2)c3ccc(cc3C#N)[N+](=O)[O-] KM08691 CC(=O)Oc1cccc(c1[N+](=O)[O-])OC(=O)C KM08696 Cc1ccc(cc1)S(=O)(=O)NN2C(Nc3ccccc3C2=O)c4cc(cc(c4O)Cl)Cl BTB02074 CS(=NC(=O)c1ccccc1)(=O)c2ccsc2 KM05753 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2cc(cc(c2)Cl)Cl KM08485 c1ccc(cc1)c2cc([nH]n2)NC(=O)Nc3cc(cc(c3)Cl)Cl KM08486 CC(C)Sc1c(cccc1Cl)[N+](=O)[O-] KM10099 c1cc(sc1c2cc(on2)C(F)(F)F)S(=O)(=O)N3CCCCC3 KM09813 C#Cc1cccc(c1)NC(=S)NNC(=S)Nc2cccc(c2)C#C NH00820 CCCCCCCOc1ccc(cc1)/C(=N\O)/c2ccc(cc2)OC JFD03022 c1ccc(c(c1)C(=O)OCCSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-])Cl KM08438 CCCS(=O)(=O)C1=C(OC(=C(C1c2ccccc2)C#N)c3ccccc3)N KM03942 c1cc(cc(c1)NC(=O)OCCSc2ccc(c3c2non3)[N+](=O)[O-])C(F)(F)F KM06897 CC1(CCc2cc(ccc2O1)c3ccn(n3)C(=O)c4ccc(cc4)Cl)C KM05644 C/C=C(\C)/C(=O)Nc1ccc(cc1C(=O)c2ccccc2)Cl BTB01790 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)Cl KM02649 c1ccc(cc1)c2cc([nH]n2)NC(=O)Nc3ccc(cc3)OC(F)(F)F KM08494 c1cc(oc1)c2cc([nH]n2)NC(=O)Nc3ccc(cc3)OC(F)(F)F KM08496 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)Sc3cccs3 KM08499 CS(=O)(=O)c1c2c(c(s1)C(=O)Sc3cccs3)CCC=C2 KM03774 c1cc(ccc1C(F)(F)F)NS(=O)(=O)c2ccc(s2)S(=O)(=O)c3c(cc(cn3)C(F)(F)F)Cl KM05582 CC(=O)c1c(cc(s1)c2cccs2)N GK03030 CCCSc1c(c(c(s1)C(=O)OC)c2ccc(cc2)Cl)C#N KM02625 COc1ccc(cc1)c2csc(c2C#N)S(=O)(=O)C KM02631 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccccc4 KM07142 Cc1cc(ccc1Cl)C(=O)c2cc3cc(ccc3o2)Cl BTB02949 Cc1cc(ccc1Cl)C(=O)c2cc3ccc(cc3o2)OC BTB02950 COc1ccc(c(c1)C(=O)Nc2ccc(c(c2)Cl)F)OC NH00843 COc1ccc(c(c1)C(=O)Nc2ccc(cc2F)F)OC NH00853 c1ccc(cc1)Oc2ccsc2/C=N/O KM08446 CC(C)N(Cc1ccc(cc1)N(C)C)C(=S)Nc2cccc(c2)C(F)(F)F BTB01071 c1cc(sc1)c2cc([nH]n2)NC(=O)Nc3cc(cc(c3)Cl)Cl KM08487 c1cc(ccc1C(=O)/C(=C/Nc2ccc3c(c2)C(=O)OC3)/C#N)Cl KM08492 c1cc(ccc1NC(=O)NNC(=O)c2ccc3c(c2)non3)OC(F)(F)F KM09656 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)I KM02653 CC(C)S(=O)(=O)c1cscc1N/C=C(/C#N)\C(=O)C2CC2 KM02744 CC(C)(C#Cc1ccc(cc1)/C=N/Nc2c(cc(cn2)Cl)C(F)(F)F)O KM08412 Cc1cc(nc2c1c(nn2C)C)NNS(=O)(=O)c3ccc(cc3)Cl KM03974 Cn1c(cc(n1)c2ccc(s2)c3ccn(n3)S(=O)(=O)C)C(F)(F)F KM03843 Cn1c(nnc1SCC(=O)NCc2ccccc2)c3ccc4c(c3)non4 KM09764 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3ccc4c(c3)non4 KM09767 CSc1c(c(cs1)c2cccc(c2)C(F)(F)F)C#N KM02749 Cc1cscc1S(=O)(=O)c2ccc(cc2)Cl KM02750 CS(=O)(=O)c1c(c(cs1)c2cccc(c2)C(F)(F)F)C#N KM02755 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)OC)N/N=C(\C#N)/S(=O)(=O)C(C)C KM02662 c1ccc(cc1)/C=N/NC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09417 CN(C)c1c(c(ncn1)N(C)C)[N+](=O)[O-] KM09430 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)OC(F)(F)F GK03034 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccco2 GK03036 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2cccs2 GK03037 c1ccc(cc1)N/N=C/c2c(ccs2)Oc3ccccc3 KM08447 c1ccc(cc1)Oc2ccsc2/C=N/Nc3ccc(cc3F)F KM08448 c1cc(ccc1[N+](=O)[O-])Oc2c(cc(cc2Cl)Cl)Cl KM08450 c1ccc(cc1)S(=O)(=O)CCSc2ccc(cn2)C(F)(F)F KM03976 c1cc(ccc1S(=O)(=O)CCSc2ccc(cn2)C(F)(F)F)Cl KM03977 Cn1c(nnc1SCC(=O)Nc2cccc(c2)SC)c3ccc4c(c3)non4 KM09758 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)C(F)(F)F)c3ccc4c(c3)non4 KM09760 Cc1ccccc1NC(=O)NCCc2ccccc2 KM09770 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NC(=O)c3c(c4ccccc4s3)Cl BTB02072 CS(=O)(=O)c1c(c(cs1)c2cccs2)C#N KM02747 CSc1c(c(c(s1)C(=O)O)c2cccc(c2)C(F)(F)F)C#N KM02746 CC1(Cc2c(c(sc2C(=O)OCc3ccccc3)S(=O)(=O)C)C(=O)C1)C KM03787 c1cc(ccc1c2c(c(sc2C(=O)O)SC3CCCCC3)C#N)Cl KM02773 Cc1ccccc1NC(=O)NCc2cccs2 KM09682 c1ccc(c(c1)CNC(=O)Nc2ccc(cc2)Cl)F KM09692 CSc1c(c(cs1)c2cc(cc(c2)Cl)Cl)C#N KM02677 CS(=NS(=O)(=O)c1ccccc1C(F)(F)F)(=O)c2ccc(cc2)Cl KM02790 CSc1c2c(c(s1)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl)CCCC2=O KM03981 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N3CCOCC3 KM03984 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NC(=O)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F BTB02797 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F BTB02798 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NC(=O)c3c(cccc3F)F)C(F)(F)F BTB02799 CCSc1c2c(c(s1)C#N)CC(CC2=O)(C)C KM03865 CSCCC(C(=O)NNC(=O)c1ccc(cc1)Cl)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02760 CC(C)Sc1c(c(cs1)c2ccc(cc2)Cl)C#N KM02762 Cn1cc(nc1)S(=O)(=O)Nc2ccc(cc2)OC KM06774 CCCCC#Cc1cc(cnc1)C(=O)O KM09434 c1ccc(c(c1)CN/C(=C(/C#N)\N=C\c2cccs2)/C#N)Sc3ccc(cc3)Cl KM03651 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)C2CC2 GK03042 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2cc(c(c(c2)OC)OC)OC GK03041 CCOC(=O)c1cnc(nc1C(F)(F)F)SCc2ccc(cc2)Cl GK02963 c1cc(sc1)C(=O)Nc2ccc3c(c2)C(=O)OC3 KM08469 c1ccc(cc1)C(=O)Nc2ccc3c(c2)C(=O)OC3 KM08470 c1cc(ccc1F)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02501 c1cc(ccc1S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br BTB02502 c1ccc(cc1)NC(=S)NC(=O)c2ccc3c(c2)non3 KM09778 Cn1c(cc(n1)c2ccc(s2)c3ccn(n3)C(=O)c4cccc(c4)C(F)(F)F)C(F)(F)F KM03861 c1ccnc(c1)c2ccc(s2)NC(=O)N3CCOCC3 KM02665 CC(C)Sc1c(c(c(s1)C(=O)O)c2ccc(cc2)Cl)C#N KM02756 CS(=O)c1c(c(cs1)c2cccc(c2)C(F)(F)F)C#N KM02758 CC(C)C(=O)NNC(=O)C(CCSC)NS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F KM02759 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4c(cc(cn4)Cl)C(F)(F)F KM08422 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F KM08423 CN(C)/C=C(\C#N)/S(=O)(=O)c1cccs1 KM02804 CC(C)S(=O)(=O)c1c(csc1SC)Cl KM02806 CS(=O)(=O)c1c(c(cs1)c2ccc(cc2Cl)Cl)C#N KM02715 CC(C)S(=O)(=O)c1c(c(sc1SC)C(=O)O)Cl KM02726 CC1(C=Cc2cc(ccc2O1)/C(=N/OC(=O)c3cccs3)/N)C KM06991 Cc1ccc(cc1)c2cc([nH]n2)N KM06993 CSc1c-2c(cs1)CCc3c2nn(c3)C(=O)c4cccc(c4)C(F)(F)F KM03869 CC(=O)n1cc2c(n1)-c3c(csc3SC)CC2 KM03872 CCOC(=O)CSc1c(c(c(s1)C(=O)OCC)c2ccc(cc2)Cl)C#N KM02770 CN1c2ccsc2C(=O)/C(=C/N(C)C)/S1(=O)=O KM06773 Cc1c2c(c(cnc2n(n1)C)C(=O)N)Oc3cccnc3 KM06777 COc1cc(cc(c1OC)OC)C(=O)NCCNC(=O)c2cc(c(c(c2)OC)OC)OC JFD02691 CCOC(=O)c1c2c(c(s1)S(=O)(=O)C)/C(=N\O)/CC(C2)(C)C KM03655 Cc1c(sc(c1c2ccn(n2)C(=O)c3ccc(cc3)Cl)SC)C#N KM03669 Cc1c(sc(c1c2ccn(n2)C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)SC)C#N KM03671 CSc1c(c(c(s1)c2cc[nH]n2)c3ccco3)C#N KM05496 COc1ccc(cc1)N2CC3CCCc4ccccc4C3=N2 KM06984 CC1(C=Cc2cc(ccc2O1)/C(=N/OC(=O)Nc3ccc(cc3)OC)/N)C KM06988 CC1(C=Cc2cc(ccc2O1)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/N)C KM06990 Cc1ccc(cc1)c2c(c(sc2Cl)S(=O)(=O)C)C#N KM02724 c1cc(c(cc1F)Cl)S(=O)(=O)NC2CCSC2=O KM03862 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NS(=O)(=O)C)C(F)(F)F BTB02800 CC1(Cc2csc(c2/C(=N\O)/C1)SC)C KM03881 c1cc(sc1)CN(CCS(=O)(=O)c2ccc(cc2)Cl)/C=C(\C#N)/S(=O)(=O)c3cccs3 KM03877 Cc1c(csc1[N+](=O)[O-])S(=O)(=O)c2ccc(cc2)Cl KM02767 CN(C)c1ccc2c(c1[N+](=O)[O-])nsn2 KM06779 COC(=O)COc1c2ccccc2sc1C(=O)OC KM02684 C1CN(CCN(CCCN(CCN(C1)CCC#N)CCC#N)CCC#N)CCC#N JFD02931 CC1(C=Cc2cc(ccc2O1)c3nc(on3)c4ccc(cc4)Cl)C KM06994 CC(C)S(=O)(=O)c1cscc1N/C=C(/C#N)\C(=O)c2cccs2 KM02743 c1ccc2c(c1)C3=Nc4ccccc4SC(C3CO2)c5ccc(cc5)Cl JFD02631 CC(C)c1ccc(cc1)C2C3CSc4ccccc4C3=Nc5ccccc5S2 JFD02634 c1cc(ccc1C(F)(F)F)NC(=O)c2ccc3c(c2)CCO3 KM07010 CCOC(=O)c1c(c(c(s1)SC)S(=O)(=O)C(C)C)N KM03883 Cc1cc(n(n1)S(=O)(=O)c2ccc(s2)c3ccccn3)C KM04004 CC1(Cc2c(c(sc2Br)SC)/C(=N\O)/C1)C KM04005 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N3CCCCC3)C(F)(F)F KM03894 Cn1cc(nc1)S(=O)(=O)Oc2ccsc2C(=O)OC KM06792 CC(=O)Nc1ccc2c(c1)scn2 KM06799 c1cc(cc(c1)NC(=S)NC(=O)c2ccc3c(c2)non3)C(F)(F)F KM09752 c1ccc(cc1)Oc2ccsc2/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM05511 Cc1nc2ccc(cc2c(=O)n1c3ccccc3N4CCOCC4)Br BTB02228 CC(=O)CSc1nnc(n1C)CN2c3cc(ccc3SCC2=O)C(F)(F)F KM08372 CCCCC#Cc1ccc(o1)C(=O)NNC(=O)Nc2cc(cc(c2)Cl)Cl KM09532 CSC(=C(C#N)C(=O)c1cccc(c1)C(F)(F)F)SC KM02738 c1ccc2c(c1)OCC(O2)C(=O)NN KM07000 Cc1cc(nc2c1c(nn2C)C)NNC(=O)Nc3cccc(c3)Cl KM04001 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)Sc4cccs4 KM06782 CN(C)/C=C(/c1nnnn1c2ccc(cc2)Cl)\C(=O)c3ccc(cc3)Cl JFD02828 Cn1c(nnc1SCC(=O)NCC=C)c2ccc3c(c2)non3 KM09754 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)Sc4ccccn4 KM06803 c1cc2cc(ccc2nc1)C(=O)Nc3ccc(cc3F)F KM10119 c1ccc(cc1)CN2CCC(CC2)Nc3c(cccn3)[N+](=O)[O-] KM10120 CCOC(=O)/C(=N\Nc1cccc(c1)C)/c2csc(n2)N JFD02976 Cc1c(c(sc1C(=O)NC(=O)NC)SC)c2ccno2 KM05666 COc1cccc(c1)n2c(n[nH]c2=S)C3CCCNC3=O BTB00472 Cc1cccc(c1NC(=O)c2ccccc2I)C JFD02670 COC(=O)c1c(ccs1)NC(=O)c2ccc3c(c2)cccn3 KM10156 COc1cccc(c1)NC(=O)c2ccc(c(c2)OC)OC JFD02676 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC)c3ccc4c(c3)non4 KM09756 c1cc2c(cc1NC(=O)N3CCOCC3)non2 KM09757 Cn1c(nnc1SCC(=O)Nc2ccc(cc2Cl)Cl)c3ccc4c(c3)non4 KM09759 c1ccc(cc1)N2CCN(CC2)C(=O)c3ccc4c(c3)non4 KM09616 c1cc(cnc1)c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F KM09619 CCOC(=O)CCN(Cc1ccco1)S(=O)(=O)c2ccc(s2)c3ccnc(n3)SC KM09537 c1ccc(cc1)C#Cc2ccc(s2)COC(=O)c3ccccc3Cl KM08265 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)N3CCC(CC3)n4cccc4 KM09481 c1ccc(cc1)c2coc3cc(ccc3c2=O)OS(=O)(=O)c4ccccc4 JFD02646 Cc1ccc(cc1)S(=O)(=O)Oc2ccc3c(c2)occ(c3=O)c4ccccc4 JFD02647 COc1ccc(cc1)c2coc3cc(ccc3c2=O)OS(=O)(=O)c4ccccc4 JFD02650 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)CCS(=O)(=O)c4ccc(cc4)Cl KM09884 c1ccc(cc1)Cn2c(n[nH]c2=S)C3CCCNC3=O BTB00471 CN1c2ccccc2-c3c(c(sc3C(=O)Nc4ccccc4Cl)SC)S1(=O)=O KM04012 CC(C)c1cccc(c1OC(=O)NC(=O)c2c(cccc2Cl)Cl)C(C)C BTB05066 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C)c3ccc4c(c3)non4 KM09755 Cn1c(nnc1SCC(=O)Nc2ccc(cc2F)F)c3ccc4c(c3)non4 KM09761 c1ccc2c(c1)OCC(O2)c3ncc(c(n3)N)C#N KM09762 Cc1c(c(sc1C(=O)NC(=O)NCc2cccnc2)SC)c3ccno3 KM05669 c1cc2cc(ccc2nc1)C(=O)Nc3ccc(cc3)Cl KM10128 c1ccc2c(c1)CCC3C2=Nc4ccccc4SC3c5ccc(cc5)Br JFD02627 CS(=NC(=O)c1ccc(cc1)Cl)(=O)c2cccs2 KM05683 CCOC(=O)c1c(c(sc1NC(=O)c2ccc3c(c2)cccn3)C)C KM10157 c1cc(ccc1N(Cc2ccc3c(c2)OCO3)S(=O)(=O)c4ccc(cc4)F)F BTB00985 CC(=O)NC1CCN(CC1)C(=S)Nc2ccccc2Cl BTB01006 CC(C)(C)SCCNC(=S)NCCO NH00745 C1CCN(CC1)C2=NCCS2 NH00614 c1ccc2c(c1)C(=O)c3c(ccc(c3C2=O)F)F JFD02848 CC1CCCC(N1c2[nH]c(=O)n(n2)C)C NH00609 Cn1c(nnc1SCC(=O)Nc2cc(cc(c2)Cl)Cl)c3ccc4c(c3)non4 KM09766 c1cc2c(cc1NC(=O)N3CCCCC3)non2 KM09773 c1ccc(c(c1)NC(=S)NC(=O)c2ccc3c(c2)non3)Cl KM09776 CCCCC#Cc1ccc(o1)c2nnc(n2C)SCc3c(cccc3Cl)Cl KM09641 c1ccc2c(c1)CC(C2)C(=O)N3CCOCC3 KM06919 CCCCC#Cc1ccc(o1)C(=O)N/N=C/c2cccs2 KM09519 Cc1ccccc1NC(=O)NCc2ccccc2C(F)(F)F KM09675 c1ccc(cc1)CNc2c(ccs2)[N+](=O)[O-] KM05527 CCCCC#Cc1ccc(o1)C(=O)N/N=C/c2ccc(cc2)C(F)(F)F KM09523 c1ccc(c(c1)C(=O)NC(=S)NC(=O)N)Cl BTB00526 c1ccc2c(c1)c(c(s2)C(=O)NNC(=S)Nc3cc(ccc3Cl)Cl)Cl BTB00809 COc1ccc(cc1OC)C(=O)Nc2cccc3c2cccc3 JFD02684 COc1ccc(cc1)NC(=O)c2cc(c(c(c2)OC)OC)OC JFD02687 c1cc(ccc1C(=O)c2cc3cc(ccc3o2)Cl)Cl BTB02898 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCC(=O)c4ccc(cc4)C(F)(F)F)c5ccco5 SPB07920 Cc1cc(nc(n1)N/C=C(\C#N)/S(=O)(=O)Cc2ccco2)C KM03110 c1cc(oc1)CS(=O)(=O)C/C(=N/OC(=O)c2ccc(cc2)Cl)/N KM03113 CC1(Cc2csc(c2/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/C1)SC)C KM03908 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)NNC(=O)c3cccc(c3)Cl)C(F)(F)F KM03909 CC(=O)NNS(=O)(=O)c1ccc(s1)c2cc(n(n2)C)C(F)(F)F KM03915 Cn1c(cnc1SC)c2nnc(n2C)SCc3ccccc3 KM07081 c1cc(ccc1S(=O)(=O)n2ccc(n2)c3ccc(s3)Br)Cl KM08546 CC(=O)c1cc(c(s1)Nc2ccc(cc2)OC)[N+](=O)[O-] KM08548 CC(C)S(=O)(=O)/C(=C(/N1CCOCC1)\SC)/C#N KM02928 CC1=CS(=O)(=O)c2c1cc(cc2)Cl KM08552 COC(=O)c1cc(ccc1N2CCC(CC2)n3cccc3)[N+](=O)[O-] KM08689 CS(=O)c1ccc(cc1[N+](=O)[O-])C(F)(F)F KM02974 Cc1c2c(c(cnc2n(n1)C)C(=O)Nc3ccc(c(c3)Cl)F)SC(C)C KM02986 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC(=O)C(F)(F)F BTB02839 c1ccc(cc1)C(c2ccccc2)N3CC(C3)O KM08723 CC(=O)NN(C)c1ccc(cc1NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F BTB02853 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC(=O)c2ccncc2 BTB02863 Cc1c(csc1S(=O)(=O)N2CCCC2)S(=O)(=O)c3ccc(cc3)Cl KM03922 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2n3cccc3)C(F)(F)F BTB02835 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC(=S)Nc2cc(ccc2Cl)Cl BTB02837 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC(=O)c2ccc(cc2)[N+](=O)[O-] BTB02838 c1ccn(c1)C2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM08636 Cc1ccc(cc1)S(=O)(=O)CCN2CCC(CC2)n3cccc3 KM08639 CN1c2ccccc2C(=O)C(=C3SCCS3)S1(=O)=O KM08641 c1ccc(cc1)NC(=O)NNC(=O)CSCCCN2CCN(CC2)c3cccc(c3)Cl KM08642 CC(C)(C)c1csc(n1)CS(=O)(=O)c2cccs2 KM03021 Cc1cc(n2c(n1)c(c(n2)C(C)(C)C)Br)C KM07373 c1ccc2c(c1)cc(o2)C(=O)c3ccc(c(c3)Cl)Cl BTB02914 CN(c1ccc(cc1[N+](=O)[O-])C(F)(F)F)NC(=O)C(Cl)(Cl)Cl BTB02840 Cc1c(c(no1)c2ccccc2)NC(=O)NN(C)c3ccc(cc3[N+](=O)[O-])C(F)(F)F BTB02841 CC(=O)NN(C)c1ccc(cc1[N+](=O)[O-])C(F)(F)F BTB02848 CC(=O)NN(C)c1ccc(cc1NC(=O)c2c(c3ccccc3s2)Cl)C(F)(F)F BTB02852 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NC(=O)C(Cl)Cl)C(F)(F)F BTB02828 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NC=C(C#N)C#N)C(F)(F)F BTB02834 Cc1c2c(cc(=O)oc2n(n1)c3ccccc3)C(F)(F)F BTB06792 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N=S(=O)(C)c3ccccc3 KM02827 COC(=O)c1c(c(c(s1)N2CCCC2)C#N)N KM02947 COC(=O)c1c(c(c(s1)N2CCCCC2)C#N)N KM02948 CSc1c(c(c(s1)c2ccnc(n2)SCCS(=O)(=O)c3ccccc3)c4ccccc4)C#N KM05767 CS(=NS(=O)(=O)c1ccc(s1)Cl)(=O)c2ccccc2 KM02988 CS(=NS(=O)(=O)c1ccc(s1)Cl)(=O)c2ccc(cc2)Cl KM02989 CSc1c(c(c(s1)c2ccnc(n2)SCCS(=O)(=O)c3ccc(cn3)C(F)(F)F)c4ccccc4)C#N KM05768 c1cc(c(cc1NC(=O)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4)Cl)Cl SPB07892 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)NCC2CC2 KM04028 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)N(C)C KM04030 CCN(CC)c1ccc(c(c1)C)N=C2C=CC(=O)c3c2cccc3 NRB01462 CC(=O)/C(=N/Nc1ccc(cc1)F)/C#N KM06947 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2Cl)Cl)/C#N)Cl KM06948 CC1(Cc2c(c(sc2c3ccn(n3)C(=O)c4cccc(c4)C(F)(F)F)SC)/C(=N/OC)/C1)C KM04021 CC1(Cc2c(c(sc2Br)SC)/C(=N/OC(=O)c3ccccc3Cl)/C1)C KM04067 c1ccc2c(c1)OCC(O2)c3ncc(c(n3)N)S(=O)(=O)c4ccc(cc4)Cl KM09681 c1ccc(c(c1)NC(=S)Nc2cccc(c2)C(F)(F)F)SCCS(=O)(=O)c3ccc(cc3)Cl KM09847 c1cc(cc(c1)C(F)(F)F)C(=O)/C(=C/c2cccs2)/C#N KM03903 Cc1cc(nc(n1)N/C=C(\C#N)/C(=O)c2cccc(c2)CSc3ccccc3)C KM05759 CCCS(=O)(=O)c1cscc1NC(=O)c2c(onc2c3c(cccc3Cl)F)C KM02981 c1ccc(c(c1)c2csc(n2)CS(=O)(=O)c3cccs3)Cl KM03019 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)C(=O)N(C)C KM03032 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)Sc2ccc(cc2)Cl KM04018 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)Sc2ccccc2 KM04019 CC(=O)NN(C)c1ccc(cc1NC(=S)Nc2cc(ccc2Cl)Cl)C(F)(F)F BTB02850 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)COc3ccc(cc3)Cl BTB02879 Cn1c(c(cn1)C(=O)N=S(=O)(C)c2ccccc2)[N+](=O)[O-] KM02839 Cn1c(c(cn1)C(=O)N=S(=O)(C)c2ccc(cc2)Cl)[N+](=O)[O-] KM02841 COC(=O)C(CCSC)NC(=O)c1ccc(cc1)C(F)(F)F KM02844 c1ccc(cc1)C(=N)NC(=O)c2cnccc2C(F)(F)F SPB07187 CN(c1ccc(cc1)Cl)/N=C(\C#N)/C(=O)C2CC2 KM02845 CSc1c(c(c(s1)c2ccnc(n2)SCC(=O)c3ccc(cc3)Cl)c4ccccc4)C#N KM05779 c1cc(ccc1n2c(nnc2Sc3c(cc(cn3)Br)[N+](=O)[O-])O)Cl SPB07421 c1c(cnc(c1[N+](=O)[O-])Sc2nnc(s2)SCC3CC3)Br SPB07427 CC(C)(C)/C=N/NS(=O)(=O)c1ccc(s1)c2ccccn2 KM04034 CC(C)CC(C(=O)NN)NC(=O)Cc1ccsc1 KM02891 c1cc2c(cc1Cl)sc(n2)N3CCCN(CC3)C(=O)c4cc(cc(c4)Cl)Cl SPB07915 Cc1ccc(cc1)NC(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl SPB07917 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N/N=C/c3ccc(cc3)Cl KM04031 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N/N=C/c3cccs3 KM04033 CC(C)C(=O)/C(=N/Nc1ccc(cc1)F)/C#N KM06963 c1ccc(cc1)N2CC3CCc4ccccc4C3=N2 KM06969 COc1ccc(cc1)N2CC3CCc4ccccc4C3=N2 KM06970 Cn1c(cc(n1)c2ccc(cc2)Cl)N KM04038 CC(=O)O/N=C/1\CC(Cc2c1c(sc2)SC)(C)C KM03907 c1cc(sc1)CN(CCS(=O)(=O)c2ccc(cc2)Cl)C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM03802 CSc1ncc(c(n1)N)S(=O)(=O)Cc2cccs2 KM03807 Cc1ncc(c(n1)N)S(=O)(=O)Cc2cccs2 KM03808 c1cc(ccc1C(=O)NCc2ccc(s2)S(=O)(=O)N3CCOCC3)Cl KM03919 c1c(nc2c(cnn2c1C(F)(F)F)C#N)C(F)(F)F KM02997 Cc1ccc(cc1)N(C(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C)S(=O)C KM03040 CC1(Cc2c(c(sc2c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl)SC)/C(=N/OC)/C1)C KM04047 CC(C)CCCC(C)C1CCC2C1(CCC3C2CC([C@@]4(C3(CCC(C4)O)C)O)O)C NRB03774 CCn1c(cc(n1)C)C(=O)NN SPB02493 CC1(Cc2c(c(sc2c3ccn(n3)C(=O)c4cccs4)SC)/C(=N/OC)/C1)C KM04022 c1cc(ccc1C(=O)/C(=N/Nc2ccc(c(c2)Cl)F)/C#N)Cl KM06955 c1ccc(c(c1)/C=N/NS(=O)(=O)c2ccc(s2)c3ccccn3)Cl KM04032 c1cc(oc1)CNC(=S)NNC(=O)C(F)(F)F SPB07403 c1cc2c(cc1NC(=S)N3CCSCC3)CCC2 NH00712 c1ccc(cc1)C(=O)Oc2ccc3c(c2)oc(=O)c4c3CCC4 JFD02999 Cn1c(nnc1Sc2c(cc(cn2)Br)[N+](=O)[O-])C(F)(F)F SPB07419 c1ccc(c(c1)NC(=S)NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)Cl KM05822 CNC(=O)c1ccc2c(c1)CCO2 KM07016 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)Sc3c(cc(cn3)Br)[N+](=O)[O-] SPB07428 CCCCNC(=O)N1CCC(CC1)n2cccc2 KM08601 c1cc(c(c(c1)Cl)CSc2nnc(s2)Sc3c(cc(cn3)Br)[N+](=O)[O-])Cl SPB07429 COC(=O)c1cc(c(nc1)Sc2nnc(n2C3CCCCC3)O)[N+](=O)[O-] SPB07447 CS(=NS(=O)(=O)c1ccc(s1)c2ccccn2)(=O)c3ccc(cc3)Cl KM04044 CC1(Cc2c(c(sc2c3ccn(n3)S(=O)(=O)c4ccccc4Cl)SC)/C(=N/OC)/C1)C KM04048 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4c(nccn4)C#N KM09849 Cc1c(csc1S(=O)(=O)N2CCCCC2)S(=O)(=O)c3ccc(cc3)Cl KM03921 Cc1c(c(n(n1)Cc2n[nH]nn2)C)Br KM03827 c1ccc(cc1)/C=N/Nc2c(cncc2Cl)Cl RF01359 Cc1ccc(cc1)S(=O)(=O)CCSc2nccn2C KM05784 CC(C)(C)OC(=O)c1cccc(c1)NC(=O)Nc2ccccc2 KM08586 c1ccc(cc1)c2nc(no2)CS(=O)(=O)c3ccc(cc3)F KM08587 C=CCn1c(nnc1Sc2c(cc(cn2)Br)[N+](=O)[O-])O SPB07423 CSc1n[nH]c(=O)n1c2ccc(cc2)OCc3ccccc3 SPB07899 c1cc(ncc1C(F)(F)F)c2nnc(s2)S SPB06944 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)N3CCCCC3 KM04040 CC1(C=Cc2cc(ccc2O1)/C(=N/OC(=O)c3ccccc3)/N)C KM06972 COc1ccc(cc1)CSC2C(C3CCN2CC3)C(=O)NNC(=O)c4ccccc4.Cl KM06976 c1ccc(c(c1)C(F)(F)F)NC(=O)c2ccc3c(c2)CCO3 KM07019 COC(=O)c1cc(c(nc1)Sc2ccccc2NC(=O)Nc3ccc(cc3)Cl)[N+](=O)[O-] SPB07478 COC(=O)c1ccc(o1)Br KM08612 c1ccc(cc1)C#Cc2cc(cnc2)NC(=O)Nc3ccccc3Cl KM08615 COc1ccc(cc1)NC(=O)Nc2cc(cnc2)C#Cc3ccccc3 KM08616 c1cc(ccc1C(=O)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4)F SPB07887 CN(C)C(=O)c1cc(cc2c1OCC2)Br KM07178 CCOC(=O)c1cnc(n1C)S KM06817 c1cc(cc(c1)Cl)N2CCN(CC2)CCCSc3ccc(cn3)C(F)(F)F KM08508 Cn1c(nnc1SCc2ccc(c(c2)Cl)Cl)c3cc(cnc3)C#Cc4ccccc4 KM08506 c1cc(c2c(c1N3CCCCC3)non2)[N+](=O)[O-] KM06818 c1cc(c2c(c1N3CCCC3)non2)[N+](=O)[O-] KM06824 Cc1csc(c1C(=O)C)SC KM02730 Cc1c(sc(n1)C2COc3ccccc3O2)C(=O)O KM06956 Cn1c(nnc1Sc2c(cc(cn2)C(=O)OC)[N+](=O)[O-])C(F)(F)F SPB07441 COC(=O)c1cc(c(nc1)Sc2nnc(n2c3ccc(cc3)Cl)O)[N+](=O)[O-] SPB07445 c1ccn(c1)C2CCN(CC2)C(=O)Nc3ccc(cc3)Cl KM08594 c1cc(sc1)c2nc(no2)CS(=O)(=O)c3ccc(cc3)F KM08600 c1ccn(c1)C2CCN(CC2)c3ccc(cn3)C(F)(F)F KM08603 CC(=O)Nc1ccc(cc1Cl)Cl TL00914 CC(=O)N(C)c1ccc(cc1Cl)Cl TL00916 Cn1c(cnc1SC)c2nnc(n2C)SCC(=O)Nc3ccccc3 KM07083 c1ccc(cc1)CN2CCN(CC2)c3c(nccn3)C#N KM09851 CC1(Cc2c(c(sc2c3ccn(n3)S(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)SC)/C(=N/OC)/C1)C KM04049 c1ccc(cc1)CN2CCC(CC2)n3cc(c(=O)[nH]c3=O)C#N KM09854 CC(C)(C)c1ccc(cc1)CSc2nnc(n2C)C3COc4ccccc4O3 KM07031 c1ccc(cc1)/C=N/NC(=O)CSCCCN2CCN(CC2)c3cccc(c3)Cl KM08660 Cn1c(nnc1S)c2cccs2 KM02901 c1ccc(c(c1)C(F)(F)F)NC(=O)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4 SPB07890 c1cc(cc(c1)NC(=S)Nc2cc(n[nH]2)c3cccs3)C(F)(F)F KM09844 c1cc(sc1)S(=O)(=O)Cc2ccc3c(c2)non3 KM07055 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)CC(=S)N KM07060 Cc1ccc(cc1)CSc2ccc(c3c2non3)[N+](=O)[O-] KM06835 c1cc(sc1)C(=O)NNC(=O)c2ccc3c(c2)non3 KM09663 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N3CCOCC3)C(F)(F)F KM03892 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N3CCCC3)C(F)(F)F KM03893 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2ccc3c(c2)non3 KM09665 CCCCC#Cc1cc(cnc1)C(=O)NNC(=O)Nc2ccccc2 KM09471 CSc1c(c2nc(cc(n2n1)C(F)(F)F)C(F)(F)F)C(=O)N KM06960 c1ccc(cc1)NC(=O)c2csc(n2)C3COc4ccccc4O3 KM06853 CN(C)C(=O)c1csc(n1)C2COc3ccccc3O2 KM06855 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCc4cc(cc(c4)Cl)Cl SPB07878 c1cc(c(cc1C(=O)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4)Cl)Cl SPB07879 Cc1ccc(cc1)C(=O)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4 SPB07885 CN(C)c1c(c(c(s1)C(=O)OC)c2ccccc2)C#N KM02893 CNC(=O)N(c1ccccc1)c2ccccc2 KM07189 c1cc(sc1)c2cc([nH]n2)NC(=S)Nc3ccc(c(c3)Cl)Cl KM09828 CN1c2cc(ccc2-c3c(cnc(n3)SCC(=O)Nc4ccccc4)S1(=O)=O)C(=O)OC KM07052 c1cc(sc1)SCc2ccc3c(c2)non3 KM07053 CCOc1ccc(cc1)NC(=S)Nc2cc(n[nH]2)c3cccs3 KM09838 Cn1c(cnc1S)C(=O)OC KM05812 c1cc(cc(c1)S(=O)(=O)N(Cc2ccc3c(c2)OCO3)c4ccc(cc4)F)C(F)(F)F BTB00984 COc1ccc(cc1OC)CC2c3cc(c(cc3CCN2C(=S)Nc4cc(c(cc4Cl)Cl)Cl)OC)OC BTB00994 CSCCC(C(=O)NNS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)NC(=O)c2ccc(cc2)C(F)(F)F KM02887 c1ccc(cc1)/C(=C/C(=C/2\C(=O)N=C(S2)N3CCCC3)/c4ccc(cc4)F)/CC(=O)c5ccc(cc5)F JFD03037 c1cc(cc(c1)Cl)N2CCN(CC2)CCCSCC(=O)N/N=C\c3cccs3 KM08661 CCOC(=O)c1c(nc(s1)COc2ccc3c(c2)non3)C KM07310 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)NCC(=O)NNS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F KM04131 c1cc2c(cc1CSc3ccc(cn3)C(F)(F)F)non2 KM07054 CN1c2ccccc2-c3c(c(sc3C(=O)N(C)C)SC)S1(=O)=O KM04138 c1cc(ccc1NC(=O)NCCSCc2csc3c2cc(cc3)Cl)OC(F)(F)F KM07369 CCOC(=O)N/N=C(/CN1C(=O)c2ccccc2C1=O)\c3ccccc3 SPB07966 c1ccc(cc1)c2c(snn2)N3C(=O)c4ccccc4C3=O SPB07967 CCCCC#Cc1cc(cnc1)C(=O)NNC(=O)Nc2ccc(cc2)Cl KM09473 CCCCCCC#Cc1cc(cnc1)C(=O)NNC(=O)Nc2cc(cc(c2)Cl)Cl KM09474 CNC(=S)NNC(=O)C1C2CCN(C1SCc3ccc(cc3)Cl)CC2 KM06909 CSCCC(C(=O)N/N=C/c1cccs1)NC(=O)c2ccc(cc2)C(F)(F)F KM02867 CSCCC(C(=O)NNC(=O)c1ccccc1Cl)NC(=O)c2ccc(cc2)C(F)(F)F KM02876 c1ccc(cc1)C#Cc2ccc(o2)C(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F KM08655 Cc1ccc(cc1)C(=O)C/C(=C\C(=C\2/C(=O)N=C(S2)N3CCCC3)\c4ccc(cc4)C)/c5ccc(cc5)Cl JFD03038 CNC(=S)NNC(=O)c1cccs1 KM02894 c1cc(sc1)S(=O)Cc2ccc3c(c2)non3 KM07059 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)NCc3ccco3)C(F)(F)F KM03896 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)NCc3cccnc3)C(F)(F)F KM03897 c1cc2c(cc1CS(=O)(=O)c3ccc(cn3)C(F)(F)F)non2 KM07065 CC1(CC(=O)C=C(S1)SCCS(=O)(=O)c2ccccc2)C KM03966 Cc1cc(nc2c1c(nn2C)C)NNC(=O)c3ccc(cc3)Cl KM03972 c1ccc(cc1)C#Cc2cc(cnc2)NC(=O)N3CCOCC3 KM08628 Cc1ccc(cc1)S(=O)(=O)CCSc2ccc(cn2)C(F)(F)F KM03978 c1ccc(cc1)NC(=O)c2cc(cc3c2OCC3)Br KM07167 CNC(=O)c1cc(cc2c1OCC2)Br KM07175 c1cc(ccc1S(=O)(=O)NCCSCc2csc3c2cc(cc3)Cl)Cl KM07370 c1ccn(c1)C2CCN(CC2)c3ccc(cc3)NC(=O)c4cccs4 KM08699 Cn1c(cc(n1)c2ccc(s2)c3ccnc(n3)S)C(F)(F)F KM05984 c1cc(c(cc1F)F)C(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3F)F SEW05769 Cn1ccnc1SCCS(=O)(=O)c2ccccc2 KM05783 CS(=NC(=O)c1ccc(cc1)Cl)(=O)c2ccc(cc2)Cl KM02786 CS(=NS(=O)(=O)c1cc(ccc1Cl)Cl)(=O)c2ccc(cc2)Cl KM02787 CCCCC#Cc1ccc(o1)C(=O)NNC(=O)c2ccccc2 KM09525 CCCCC#Cc1ccc(o1)C(=O)NNC(=O)c2cccs2 KM09526 CCCCC#Cc1ccc(o1)C(=O)NNC(=O)Nc2ccc(cc2)Cl KM09531 c1cc(ccc1CSC2C(C3CCN2CC3)C(=O)NNC(=O)c4ccc(cc4Cl)Cl)Cl.Cl KM06923 COc1ccc(cc1)C(=O)NNC(=O)CSCCCN2CCN(CC2)c3cccc(c3)Cl KM08663 Cc1c(nc(s1)c2ccccc2)CC(=O)NNC(=O)c3ccc(cc3)C(F)(F)F RH01237 c1ccc(cc1)C2=CC(=NN=C(C2)c3ccccc3)c4ccccc4 JFD03039 c1cc(ccc1C(F)(F)F)NC(=O)c2cc(cc3c2OCC3)Br KM07169 CN(C)/C=C/C(=O)c1ccc(cc1)OC KM04140 c1cc(oc1)CSCc2ccc3c(c2)non3 KM07062 Cn1c(nnc1SCc2ccccc2)C(CCSC)NC(=O)c3ccc(cc3)C(F)(F)F KM07072 CC(C)(C)N(C)C(=O)c1ccc2c(c1)CCO2 KM07074 CNC(=S)NNC(=O)C(CCSC)NC(=O)c1ccc(cc1)C(F)(F)F KM07066 CSCCC(C(=O)NNS(=O)(=O)c1ccc(cc1)Cl)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02775 c1cc(ccc1c2csc(c2C#N)S(=O)(=O)C3CCCCC3)Cl KM02783 CSc1c(c(c(s1)c2ccnc(n2)SCC(=O)c3ccccc3)c4ccccc4)C#N KM05780 CC1(CC(=O)C=C(S1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C KM03949 c1cc(ccc1S(=O)(=O)Cc2ccc(cc2F)Br)Cl KM07110 CN(CCC#N)S(=O)(=O)c1ccc(cc1)Oc2c(cccc2Cl)[N+](=O)[O-] BTB02917 c1cc(c(c(c1)Cl)Oc2ccc(cc2)S(=O)(=O)N3CCOCC3)[N+](=O)[O-] BTB02918 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)OC(=O)c3ccccc3Cl KM05716 Cc1cc(ccc1Cl)c2csc(=N)n2c3cccc(c3)C(F)(F)F.Cl BTB03019 CCO/C(=N\OC(=O)c1c(onc1c2c(cccc2Cl)Cl)C)/C KM05735 c1ccn(c1)C2CCN(CC2)c3ccc(cc3)NC(=O)c4ccc(cc4)Cl KM08702 c1ccc(cc1)C#Cc2ccc(o2)c3nc(no3)c4cccc(c4)C(F)(F)F KM08704 c1ccc(c(c1)NS(=O)(=O)c2ccc(s2)c3ccccn3)Cl KM03998 Cn1c(nnc1SCCS(=O)(=O)c2ccc(cc2)F)C(F)(F)F KM08592 c1ccc(cc1)C#Cc2cc(cnc2)NC(=O)Nc3ccccc3 KM08602 c1ccn(c1)C2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl KM08604 c1cc(ccc1F)S(=O)(=O)CCSc2ccc(cc2)Cl KM08606 c1cc(ccc1C2CCCCC2)NC(=S)N3CCSCC3 NH00682 c1ccc2c(c1)C(=O)N(C2=O)CC3COc4ccccc4O3 KM07106 c1ccnc(c1)S(=O)(=O)Cc2ccc(cc2F)Br KM07109 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)S(=O)(=O)N KM03948 c1c(cc(c2c1CCO2)C(=O)N3CCCCC3)Br KM07177 Cc1ccc(cc1)Sc2cc(c(cc2F)[N+](=O)[O-])NC(=O)C BTB03664 Cc1cc(no1)C(=O)NNC(=O)NC(C)C SPB01197 Cc1cc(no1)C(=O)NNC(=O)Nc2ccccc2 SPB01199 Cc1cc(c(cc1Cl)C)SCc2cc(on2)C SPB01284 Cc1c(c(n(n1)S(=O)(=O)c2ccc(s2)c3ccccn3)C)Br KM04007 Cc1ccc(cc1)S(=NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)(=O)C KM02791 c1cc(sc1)S(=O)(=O)C(=C2SCCCS2)C#N KM02800 c1cc(c(c(c1)Cl)Oc2ccc(cc2)S(=O)(=O)N3CCOCC3)N BTB02924 CC(c1ccccc1)NS(=O)(=O)c2ccc(cc2)Oc3c(cccc3Cl)[N+](=O)[O-] BTB02927 CC(C)(C)c1ccc(cc1)OCc2nc(no2)c3cccc(c3)[N+](=O)[O-] BTB02942 c1ccc(c(c1)c2nc(no2)c3ccc(cc3)Cl)NC(=O)C(F)(F)F BTB03493 CCOC(=O)c1cc(c(c(c1)Cl)NC(=O)C(F)(F)F)Cl BTB03509 CC1(Cc2c(c(sc2Br)SC)/C(=N/OC(=O)c3cccs3)/C1)C KM04081 Cc1c(c(n(n1)S(=O)(=O)c2ccc(s2)c3cc(n(n3)C)C(F)(F)F)C)Br KM04087 c1cc(c(cc1Cl)[N+](=O)[O-])c2ccc(o2)C#N JFD02866 c1ccc2c(c1)C[C@@H]3[C@H]2N=C(O3)CC4=NC5c6ccccc6CC5O4 JFD02877 COC(=O)c1c(c(c(s1)N2CCOCC2)C#N)c3ccc(cc3)Cl KM02892 CC(C(C(=O)O)NC(=O)C(CSC(C)(C)C)NC(=O)C(CCC(=O)OC(C)(C)C)NC(=O)OCC1c2ccccc2-c3c1cccc3)OC(C)(C)C JFD02943 c1c(cncc1Br)C#N KM08398 c1ccc(cc1)Oc2ccsc2CO KM08526 c1cc(ccc1C(=O)NNC(=O)c2ccc3c(c2)non3)Cl KM09666 C/S(=N\S(=O)(=O)c1cccc2c1nsn2)/c3c(cc(cn3)C(F)(F)F)Cl KM08415 Cc1ccc(c(c1)C)n2c(csc2=N)c3ccc(c(c3)C)Cl.Cl BTB03023 c1ccc(cc1)S(=O)(=O)CCSc2nccc(n2)c3ccc(cc3)Cl KM05730 CSc1c(c(c(s1)c2ccnc(n2)SC(=O)CNc3ccccc3)c4ccccc4)C#N KM05746 c1ccc(cc1)CN2C3CCCC2CC(=NOC(=O)Nc4ccccc4)C3 KM08825 CN1c2ccccc2-c3c(c(sc3C(=O)Nc4cccc(c4)C(F)(F)F)SC)S1(=O)=O KM04013 c1ccn(c1)C2CCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl KM08595 c1cc(sc1)SCCS(=O)(=O)c2ccc(cc2)F KM08607 COC(=O)c1ccc(o1)C#Cc2ccccc2 KM08614 c1cc(c(cc1Cl)Cl)/C=C(\C#N)/C(=O)O JFD02888 c1ccc(cc1)CSc2[nH]c3ccccc3n2 JFD02896 CC1(CC(=O)C=C(S1)Sc2ccc(cc2[N+](=O)[O-])C#N)C KM04054 Cc1ccc(cc1)S(=O)(=O)CCN2C(=O)CSC2=O KM04062 c1cc(cc(c1)Cl)N2CCN(CC2)CCCSCC(=O)NN KM08561 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccc(s2)c3ccnc(n3)SC KM08564 Cc1c(c(n(n1)S(=O)(=O)c2ccc(s2)c3nnc(n3C)SC)C)Br KM04091 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)N=S(=O)(C)c3ccc(cc3)Cl KM04099 CC(C)CC(C(=O)NNS(=O)(=O)c1ccc(cc1)Cl)NC(=O)Cc2ccsc2 KM02922 COC(=O)c1c(c(c(s1)N2CCCC2)C#N)c3cccs3 KM02895 CC(=O)n1ccc(n1)c2c3c(c(s2)SC)/C(=N/OC)/CC(C3)(C)C KM04020 CC(C)CC(C(=O)NC(CCCCNC(=O)OC(C)(C)C)C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 JFD02953 CC(C)(C)C1=CC(C=C(C1=O)C(C)(C)C)(c2ccccc2)O JFD02963 CC(C)CC(C(=O)NNC(=O)c1ccccc1Cl)NC(=O)Cc2ccsc2 KM02921 CSCCC(C(=O)NNS(=O)(=O)c1ccccc1C(F)(F)F)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02776 CSCCC(C(=O)NNS(=O)(=O)c1ccc(c(c1)Cl)Cl)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02777 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)c4cccc(n4)C(F)(F)F KM08424 CSc1c(c(c(s1)c2ccnc(n2)SCC(=O)N)c3ccccc3)C#N KM05747 CSc1c(c(c(s1)c2ccnc(n2)SCCS(=O)(=O)c3ccc(cc3)Cl)c4ccccc4)C#N KM05748 Cc1cc(nc2c1c(nn2C)C)NNC(=O)Nc3ccc(cc3)Cl KM04083 Cc1cc(n(n1)S(=O)(=O)c2ccc(s2)c3cc(n(n3)C)C(F)(F)F)C KM04086 c1ccc2c(c1)nc(s2)c3ccc(cc3)Cl JFD02911 Cc1cc(c(c(c1S(=O)(=O)NC(=N)NCCCC(C(=O)NC(COC(C)(C)C)C(=O)N2CCCC2C(=O)NC(CC(C)C)C(=O)O)NC(=O)OCC3c4ccccc4-c5c3cccc5)C)C)OC JFD02946 Cc1cc(nc2c1c(c(s2)C(=O)N)N)C JFD02960 CC1(C=Cc2cc(ccc2O1)c3nc(on3)c4cccc(c4)C(F)(F)F)C KM06995 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)F)/C#N)OC(F)(F)F KM07002 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NNC(=O)Nc3cccc(c3)Cl KM04072 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N=S(=O)(C)c3ccccc3)C(F)(F)F KM04079 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)N=S(=O)(C)c3ccccc3 KM04100 CC(C)S(=O)(=O)c1cscc1Cl KM02847 c1cc(cc(c1)Cl)C(=O)/C(=N/Nc2ccc(cc2)F)/C#N KM07172 CC(=O)C(=NNc1cc(cc(c1)Cl)Cl)C(=O)C BTB03531 CC(=O)Nc1cc(c(cc1[N+](=O)[O-])F)Sc2ccc(cc2)Cl BTB03663 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3cc(ccc3Cl)C(F)(F)F)Oc4ccc(cc4Cl)Cl MBE00149 CS(=NC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F)(=O)c2ccc(cc2)Cl KM02792 CN(CCOC(=O)c1ccc(cc1)Cl)c2cc(nc3c2cccc3)C(F)(F)F KM08435 c1cc(ccc1NC(=O)O/N=C(/CS(=O)(=O)c2ccc(cc2)F)\N)Cl KM08568 c1ccc(cc1)Oc2ccsc2COC(=O)c3ccc(cc3)Cl KM08573 c1cc(ccc1C(=O)O/N=C(/CS(=O)(=O)c2ccc(cc2)F)\N)Cl KM08574 Cc1ccc(cc1)S(=O)(=O)CCN(Cc2cccnc2)C(=O)c3ccccc3 KM04097 c1cc(cc(c1)n2c(nnc2Sc3c(cc(cn3)Br)[N+](=O)[O-])O)C(F)(F)F SPB07422 COC(=O)c1c(ccs1)NS(=O)(=O)c2cccc3c2nsn3 KM07160 c1ccc(cc1)NC(=S)NNC(=O)c2cc(ccc2O)Cl RH01279 c1cc(cc(c1)NC(=O)c2cc(cc3c2OCC3)Br)C(F)(F)F KM07168 CN(C)c1c(c(cs1)c2ccc(cc2)Cl)C#N KM02924 CO/C=N/c1nc-2c(s1)CCc3c2cccc3 RH01285 CCCCCCCCCC(=O)Nc1nc-2c(s1)CCc3c2cccc3 RH01286 CCOC(=O)c1ccc(s1)c2ccc(cc2)Cl MBE00071 c1ccc(c(c1)C(F)(F)F)NC(=S)NNC(=O)c2ccc(s2)c3ccc(cc3)Cl MBE00145 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)CC#N KM07008 c1cc(cc(c1)NC(=O)c2ccc3c(c2)CCO3)C(F)(F)F KM07009 CSCCC(C(=O)NN)NC(=O)c1ccc(cc1)C(F)(F)F KM02850 Cc1c2c(c(cnc2n(n1)C)C(=O)OC)OC KM02864 CC(=O)Nc1cc(c(cc1[N+](=O)[O-])F)N2CCOCC2 BTB03665 Cc1cccc(c1n2c(n[nH]c2=S)c3ccncc3)C ML00380 c1ccc(c(c1)c2nnc(o2)Cc3cc(sc3Br)Br)Cl SPB02950 Cc1c2c(c(cnc2n(n1)C)C(=O)N=S(=O)(C)c3ccccc3)SC(C)C KM05686 CC(=O)Oc1cc(cc(c1OC(=O)C)OC)C=C(C#N)C#N JFD02881 CC(C)(C)S(=O)(=O)c1cnc(nc1N)c2ccncc2 KM02694 CC(C)Sc1c(cccc1Cl)NC(=O)c2ccc(cc2)Cl KM10122 c1ccn(c1)C2CCN(CC2)C(=O)c3cccs3 KM08581 c1ccn(c1)C2CCN(CC2)S(=O)(=O)c3cccs3 KM08583 Cc1c(c(n(n1)Cc2nnn(n2)CC(=O)N/N=C/c3ccc(cc3)Cl)C)Br KM05835 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3ccccc3C(F)(F)F)Oc4ccc(cc4Cl)Cl MBE00147 c1c(cc(c(c1Cl)NC(=O)C(F)(F)F)Cl)C#N BTB03635 CC(C)S(=O)(=O)C/C(=N/OCCS(=O)(=O)c1ccc(cc1)Cl)/N KM05674 CS(=NC(=O)Nc1ccccc1)(=O)c2cccs2 KM05687 COc1ccc(c(c1)OC)NC(=S)NNC(=O)c2ccc(s2)c3ccc(cc3)Cl MBE00152 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)OC(=O)Nc3ccccc3 KM05793 CCOC(=O)COc1ccccc1/C=C(\C#N)/C(=O)c2ccc(cc2)Cl KM05794 CCOC(=O)COc1ccccc1/C=C(\C#N)/C(=O)c2cccc(c2)C(F)(F)F KM05796 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCCc4c3cccc4 BTB00796 Cc1ccc2c(c1)CCCN2C(=O)c3c(onc3c4c(cccc4Cl)Cl)C BTB00797 CSCCC(C(=O)N/N=C\c1c(cccc1Cl)F)NC(=O)c2ccc(cc2)C(F)(F)F KM02865 c1cc(cc(c1)C(=O)CC#N)CSc2cccc(c2)C(F)(F)F KM05854 CC1(CCc2cc(ccc2O1)c3ccnc(n3)SCC(=O)c4ccccc4)C KM05855 CC1(CCc2cc(ccc2O1)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl)C KM05856 c1cc(ccc1COC(=O)c2ccc(c(c2)Cl)F)[N+](=O)[O-] BTB03718 c1cc2c(cc1OS(=O)(=O)c3ccc(s3)Cl)non2 KM07100 c1ccc(cc1)n2c(cc(n2)C3CC3)NC(=O)Nc4cccc(c4)C(F)(F)F KM09825 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)n3ccnc3)C(F)(F)F KM03936 CC(C)CC(C(=O)NCc1ccccc1)NC(=O)OC(C)(C)C JFD02958 c1cc(c(c(c1)Cl)C(=O)N2CCN(CC2)C(=O)C3CCCCC3)Cl JFD02516 CC(C)Sc1c(cccc1Cl)NC(=O)Nc2ccccc2 KM10126 C/S(=N\C(=O)Nc1ccc(cc1)Cl)/c2c3c(c(s2)Cl)CCCC3=O KM05837 CC1(Cc2c(c(sc2Cl)/S(=N\C(=O)Nc3ccc(cc3)Cl)/C)C(=O)C1)C KM05853 CCSC1=NCN(CN1)Cc2cccs2.I BTB03554 c1cc(ccc1c2csc(n2)c3ccc(c(c3)Cl)F)[N+](=O)[O-].Br BTB03708 CCOC(=O)COc1ccccc1/C=C(\C#N)/C(=O)c2cccs2 KM05795 CCOC(=O)COc1ccccc1/C=C(/C#N)\S(=O)(=O)c2ccccc2 KM05797 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)N3CCCCC3 KM09869 c1ccc(cc1)CN2CCN(CC2)c3cc(nc4c3cccc4Cl)C(F)(F)F KM09880 CC1(CC(=O)C=C(S1)SC)C KM03927 Cn1c(cnc1SC)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)Cl KM07084 c1ccc2c(c1)OCC(O2)CNC(=O)Nc3ccc(cc3)Cl KM07122 Cc1ccc(cc1)NC(=O)NCC2COc3ccccc3O2 KM07123 c1ccc2c(c1)OCC(O2)CNC(=S)NC(=O)c3ccc(cc3)Cl KM07127 c1ccc(cc1)OC(=O)c2ccc3c(c2)CCO3 KM07043 CN(C)c1c(c(c(s1)C(=O)OC)c2ccc(cc2)Cl)C#N KM02911 Cc1cc(c2ccccc2n1)O BTB01126 Cn1c(cnc1SCC(=O)Nc2cccc(c2)Cl)C(=O)OC KM05888 c1cc(sc1)C(=O)NCCSCc2ccc3c(c2)non3 KM07101 Cn1c(nnc1SCc2ccc(cc2F)Br)C(F)(F)F KM07107 c1cc(sc1)S(=O)(=O)Cc2ccc(cc2F)Br KM07108 Cc1ccc(cc1)S(=NC(=O)c2ccc(s2)c3cc(nn3C)C(F)(F)F)(=O)C KM03055 c1cc2c(cc1OS(=O)(=O)c3ccc(cc3Cl)Cl)non2 KM07096 CSc1c(cccn1)C(=O)N=S(=O)(C)c2ccccc2 KM02929 c1ccc(cc1)Cn2c(=O)c(nn(c2=O)c3ccccc3)C#N KM08754 c1ccc(cc1)CCNC(=O)c2ccc3c(c2)cccn3 KM10130 Cc1c(c(sc1C(=O)NC(=O)NCc2ccncc2)SC)c3ccno3 KM05670 c1ccc2c(c1)C3=Nc4ccccc4SC(C3CO2)c5ccc(cc5)F JFD02630 COC(=O)c1c(ccs1)N/C=C(\C#N)/C(=O)c2cccc(c2)CSc3cccc(c3)C(F)(F)F KM05863 CN(C)c1c(c(cs1)c2ccccc2)C#N KM02905 CC(C)CC(C(=O)N/N=C/c1c(cccc1Cl)F)NC(=O)Cc2ccsc2 KM02908 c1cc2c(cc1CSCCNC(=O)c3ccc(cc3Cl)Cl)non2 KM07092 CS(=O)(=O)Oc1ccc2c(c1)non2 KM07098 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Oc3ccc4c(c3)non4 KM07099 CC1(CC(=O)C=C(S1)SCc2ccc(cc2)Cl)C KM03941 CC1(Cc2c(c(sc2c3ccn(n3)C(=O)c4ccc(cc4)Cl)SC)/C(=N/OC)/C1)C KM03945 Cc1ccc(cc1)CSc2n[nH]c(=O)n2c3ccc(cc3)OCc4ccccc4 SPB07884 CN1c2ccsc2C(=O)/C(=N\Nc3ccc(cc3)Cl)/S1(=O)=O KM04202 c1cc(ccc1C#N)c2csc(n2)COc3ccc4c(c3)non4 KM07328 c1cc(sc1)S(=O)(=O)Cc2nc(cs2)c3ccc(cc3)Cl KM03015 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)CS(=O)(=O)c3cccs3 KM03018 CS(=NC(=O)NS(=O)(=O)Oc1ccc(cc1Cl)Cl)(=O)c2ccc(cc2)Cl KM03064 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NC(=O)C(F)(F)F)C(F)(F)F BTB02830 CCOC(=O)c1c(c2c(ccc(c2nc1SC)C)Cl)O KM08757 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F BTB02801 COc1cc(ccc1Cc2ccc(cc2)[N+](=O)[O-])CC=C KM03918 Cc1ccc(cc1)S(=NC(=O)c2cnc3c(c2SC(C)C)c(nn3C)C)(=O)C KM05695 Cc1cc(c(c(c1)C)S(=O)(=O)O)C.CS(=N)c1ccsc1 KM05697 c1cc(c(c(c1)Cl)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)F)Cl KM08537 CC(C)N(Cc1ccc(cc1)N(C)C)S(=O)(=O)c2cccc(c2)C(F)(F)F BTB01293 CC(C)N(Cc1ccc(cc1)N(C)C)S(=O)(=O)c2ccc(cc2)F BTB01294 C/C=C(\C)/C(=O)Nc1ccccc1CC2c3ccccc3CCN2C BTB01778 CNC(=S)NNC(=O)CSCc1nc(cs1)c2ccc(cc2)Cl KM05897 Cn1cc(cc1/C=C(\C#N)/C(=O)c2ccc(cc2)Cl)C(=O)c3ccc(cc3)Cl KM07208 CCOC(=O)c1cnc2c(c1N3CCOCC3)cc(cc2F)F BTB03780 CC(C)(C)NC(=S)N(C)/N=C/c1cc(cc(c1O)Cl)Cl BTB03785 c1ccc(cc1)CN2CCN=C2SCc3nc(no3)c4cccc(c4)[N+](=O)[O-].Cl BTB02880 Cc1c2c(cc(=O)oc2n(n1)c3ccccc3)c4ccc(cc4)[N+](=O)[O-] NRB00459 Cc1ccc(c(c1)C)C(C)NC(=S)Nc2ccc(cc2)Cl SW00068 c1cc(ccc1NC(=S)N(CCC#N)C2CCCCC2)Cl SW00109 CC(C)S(=O)(=O)c1c(c(sc1N2CCCC2)C(=O)OC)N KM02935 CCOC(=O)c1c(c(sc1N/C=C(\C#N)/C(=O)NC(=O)OCC)C)C KM08763 COC(=O)C1N(CCS1)S(=O)(=O)c2ccc(cc2)Cl KM05893 c1cc(ccc1c2csc(n2)CSCC(=O)NN)Cl KM05896 CCOC(=O)c1c(c2cccc(c2nc1SC)Cl)Sc3cccs3 KM08779 c1cc(ccc1C2SCCS2)OCC(=O)NN SPB01291 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)NNC(=O)C(C)(C)C SPB01249 CC(C)(C)c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Oc3c(cccc3Cl)[N+](=O)[O-] BTB02919 COc1ccc2c(c1)cc(o2)C(=O)c3ccc(c(c3)Cl)Cl BTB02921 c1cc(c(c(c1)Cl)Oc2ccc(cc2)S(=O)(=O)Nc3ccc(cc3)F)N BTB02925 CCOC(=O)c1cnc2c(csc2c1Sc3cccc(c3)Cl)S(=O)(=O)C(C)C KM02832 CS(=NC(=O)Nc1ccc(cc1)Cl)(=O)c2ccccc2 KM02833 Cc1ccc(cc1)S(=NC(=O)c2cccnc2Oc3ccccc3)(=O)C KM02963 Cc1c(csc1C(=O)N(c2ccccc2)S(=O)C)S(=O)(=O)c3ccc(cc3)Cl KM02966 CCOC(=O)c1cc(n(n1)c2nc3cc(ccc3s2)Cl)N SPB01238 CC(C)(C)C(=O)NNC(=O)COc1ccc(cc1)C2SCCS2 SPB01295 Cn1c(cc(n1)c2ccc(s2)C(=O)N(C)c3ccccc3)C(F)(F)F KM03035 Cc1cc(nn1C)C(=O)O/N=C/c2ccccc2 SPB01252 c1cc(ccc1NC(=S)N(CCCN2CCOCC2)CCC#N)Cl SW00119 C1CC2C3C4C1C5C2(C3C45C(=O)O)C(=O)O RJC03406 c1cc(c(c(c1)Cl)Oc2ccc(cc2)S(=O)(=O)N3CCOCC3)NC(=O)C(F)(F)F BTB02926 Cc1ccc(cc1)S(=NC(=S)NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)(=O)C KM05825 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)C(=O)N=S(=O)(C)c3ccccc3 KM03049 c1ccc(cc1)Oc2c(cccn2)C(=O)NCCSc3ccc(cc3)Cl BTB03480 Cc1ccc(cc1)SCCNC(=O)c2cccnc2Oc3ccccc3 BTB03481 c1ccc(cc1)c2c(nc3cc(c(cc3n2)F)Cl)c4ccccc4 BTB03695 c1c2c(cc(c1Cl)F)nn[nH]2 BTB03699 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)NNC(=O)C(C)C SPB01250 Cc1cc(nc(n1)c2ccc(cc2)C(F)(F)F)O SPB01315 COc1cc(c(cc1N2CCOCC2)Nc3ccccn3)[N+](=O)[O-] NRB03404 COc1cc(c(cc1Cl)Cl)Cl KM07229 Cc1ccc(cc1)C(=O)/C(=C/c2cc(cn2C)C(=O)c3ccc(cc3)Cl)/C#N KM07223 c1cc(cc(c1)[N+](=O)[O-])c2nc(on2)CSC3=NCCN3.Cl BTB02947 Cn1cc(cc1/C=C(\C#N)/S(=O)(=O)c2ccc(cn2)C(F)(F)F)C(=O)c3ccc(cc3)Cl KM07227 Cc1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F KM03140 COc1ccc2c(c1)oc3ccc(cc3c2=O)CC(=O)OC RJC03494 CCCS(=O)(=O)c1cscc1NC(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C KM03053 CSc1nnc(n1c2ccc(cc2)OCc3ccccc3)c4ccco4 SPB07932 Cc1ccc(cc1)C(=O)NCC2COc3ccccc3O2 KM07126 Cc1ccc(cc1)C(=O)NC(=S)NCC2COc3ccccc3O2 KM07129 CC\1=NN(C(=O)/C1=N\Nc2ccc(cc2)Br)c3ccccc3 JFD02991 CCOC(=O)NC(=S)NCCCN1CC(OC(C1)C)C NH00505 Cc1cccc(c1)C(=N)NC(=O)c2cnccc2C(F)(F)F SPB07189 c1cc(ccc1SCC(=O)N2CCC(CC2)C(F)(F)F)Cl SPB07220 Cc1cccc(c1)c2nc(on2)NC(=O)O/N=C/c3ccccc3 SPB01254 Cc1cc(no1)NC(=O)NN2CCOCC2 SPB01258 Cc1cc(no1)NC(=O)NCc2cccnc2 SPB01260 CCNC(=O)N(c1ccccc1)c2ccccc2 KM07179 c1c(cc(c2c1CCO2)C(=O)N3CCOCC3)Br KM07180 c1ccc(c(c1)c2nc(no2)CS(=O)(=O)Cc3ccco3)Cl KM03126 c1cc(oc1)CS(=O)(=O)C/C(=N/OC(=O)Nc2ccc(cc2)Cl)/N KM03134 Cn1cc(cc1/C=C(\C#N)/S(=O)(=O)c2ccccc2)C(=O)c3ccc(cc3)Cl KM07225 Cn1c(c(cn1)C(=O)N)[N+](=O)[O-] KM03138 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2)OC)C#N RJC03431 Cc1csc(n1)c2c(c3ccccc3s2)O KM07120 Cc1ccc(cc1)NC(=S)NCC2COc3ccccc3O2 KM07125 Cc1ccc(cc1)S(=O)(=O)N=S(=O)(C)C KM03087 c1ccc(cc1)S(=O)(=O)CCSCC(=O)N/N=C/c2ccccc2Cl KM03088 c1cc(cc(c1)[N+](=O)[O-])c2cc[nH]n2 KM03091 Cc1cc(nc2c1c(nn2C)C)NNC(=S)NC KM04085 CSc1nccc(n1)c2cccs2 KM04089 Cc1cc(n(n1)S(=O)(=O)c2ccc(s2)c3nnc(n3C)SC)C KM04090 Cc1cc(no1)NC(=O)NNc2ccccc2 SPB01261 Cc1cc(no1)C(=O)N/N=C/C(C)(C)C SPB01265 CC(C)(C)NC(=O)c1cc(cc2c1OCC2)Br KM07186 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)Sc4ncc(s4)[N+](=O)[O-] SPB07951 Cc1cc(ccc1Cl)C(=O)c2cc3cc(ccc3o2)OC BTB02952 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCC(=O)c4ccc(cc4)Cl)c5ccco5 SPB07921 Cc1cc(ccc1Cl)c2csc(=N)n2c3ccc(cc3)Cl.Cl BTB03020 CC(=O)Nc1ccc(cc1Cl)C(F)(F)F SEW03073 CS(=O)(=O)c1ccsc1 KM05823 CS(=NC(=S)NC(=O)c1cnn2c1nc(cc2C(F)(F)F)C(F)(F)F)(=O)c3ccc(cc3)Cl KM05824 c1ccc(c(c1)C(=O)O)NCc2ccco2 SJC00396 CC(C)(C)NC(=O)c1ccc2c(c1)CCO2 KM07020 CSc1nccc(n1)c2ccc(s2)Br KM04249 CN1c2ccsc2C(=O)/C(=C\Nc3ccsc3C(=O)OC)/S1(=O)=O KM04247 CN1c2ccsc2C(=O)/C(=C/Nc3cccnc3)/S1(=O)=O KM04152 Cc1csc(n1)Cn2c(=O)c3ccccc3c(n2)CC(=O)NNC(=S)Nc4ccccc4 KM07240 CCOC(=O)N1CCN(CC1)CC(Cn2c(=O)c3c(ncn3C)n(c2=O)C)O RJC03498 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)SCC(=O)c4ccc(cc4)F SPB07952 c1cnc(cn1)c2nc(on2)CC(=O)NN KM08654 Cn1cc(c(n1)c2ccc(cc2)NC(=O)Nc3ccc(cc3)Cl)Br KM03069 Cn1cc(c(n1)c2ccc(cc2)NC(=O)Nc3ccccc3)Br KM03072 Cc1c(sc2c1C(=O)/C(=C\N(C)C)/S(=O)(=O)N2C)C KM07134 c1ccc(cc1)S(=O)(=O)CCSCC(=O)NNC(=O)c2ccc(cc2)Cl KM03102 c1ccc2c(c1)c(cc(n2)c3cccs3)N4CCCCC4 RJC03453 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)SCC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB07938 c1cc(ccc1CSc2[nH]c(=O)c3c(n2)CSC3)Cl KM07209 CCOC(=O)c1c2c(c(s1)SC)-c3c(cnc(n3)SCC(=O)Nc4ccc(cc4)Cl)CC2 KM04252 Cc1ccc(cc1)S(=O)(=O)Cc2c(cccc2Cl)Cl KM04254 CCOC(=O)c1cnc2c(c1Sc3ccc(cc3)Cl)cc(cc2F)F BTB03781 CC(=O)Nc1cc(ccc1C(=O)OC)Cl BTB07262 c1c(cc(c2c1c3c(cn2)c(=O)[nH][nH]3)F)F BTB04010 C/C(=N\NC(=S)NC(C)(C)C)/c1cc(cc(c1O)F)F BTB04136 Cc1c(c(ccn1)C(F)(F)F)c2nnc(o2)SCC(=O)c3ccc(cc3)Cl AW00229 c1ccc(cc1)Oc2c(cccn2)C(=O)NCCSc3ccccc3 BTB03479 c1cc(ccc1OC(=O)c2ccc3c(c2)CCO3)Cl KM07022 Cn1c(nnc1SCc2ccc(cc2)F)C3COc4ccccc4O3 KM07025 Cn1c(nnc1SCC(=O)Nc2ccccc2)C3COc4ccccc4O3 KM07028 c1ccc2c(c1)OCC(O2)CNC(=O)c3ccc(cc3)Cl KM07115 c1cc(c(cc1C(=O)Nc2ccc(c(c2)Cl)F)Cl)F BTB03719 Cc1csc(n1)Cn2c(=O)c3ccccc3c(n2)CC(=O)N/N=C/c4ccccc4 KM07214 Cc1nc(nc(n1)SC)N/C=C/2\C(=O)c3c(ccs3)N(S2(=O)=O)C KM04265 c1cc(c(cc1C(=O)Nc2nnc(s2)C(F)(F)F)Cl)F BTB03720 Cc1c(ncn1Cc2ccc(cc2)Cl)C(=O)N KM07243 CC(C)(C)NC(=S)N/N=C/c1ccccc1SC(C)(C)C BTB04000 CCOC(=O)N(c1ccccc1)c2ccccc2 KM07137 Cc1cc(ccc1Cl)c2csc(=N)n2c3c(cccc3F)F.Cl BTB03024 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCc4c(cccc4Cl)F)c5ccco5 SPB07944 CCOC(=O)c1c2c(nc3ccccc3n2)n(c1N)c4ccc(cc4)C RJC03481 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccc(nc3)Oc4ccc(cc4)C(C)(C)C BTB03884 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccc(nc3)Oc4c(cccc4Cl)Cl BTB03886 C/C(=N\NC(=S)NCC(C)(C)C)/c1cc(cc(c1O)F)F BTB04138 CC(C)(C)C(=O)NNC(=S)N BTB07411 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2Cl)OC)C(=O)OCC)C)C RJC03413 c1cc(cc(c1)Cl)Cn2cc(c(=O)[nH]c2=O)C#N KM09858 c1ccc(cc1)N2CCN(CC2)CCS(=O)(=O)c3ccc(cc3)F KM09865 c1ccc2c(c1)c(c(s2)c3nc(cs3)c4ccc(cc4Cl)Cl)O KM07121 CN1c2cc(ccc2-c3c(cnc(n3)SC)S1(=O)=O)C(=O)OC KM07037 CC(C)(C)C(=O)CSc1ncc2c(n1)-c3ccc(cc3N(S2(=O)=O)C)C(=O)OC KM07038 Cc1ccc(cc1)OC(=O)c2ccc3c(c2)CCO3 KM07042 Cc1ccc(cc1)C(=O)NC(=O)NCC2COc3ccccc3O2 KM07145 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccc(nc3)Oc4ccc(cc4Cl)Cl BTB03888 Cc1cc(cc(c1Cl)C)Oc2ccc(cn2)NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C BTB03890 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(nc3)Oc4c(cccc4Cl)Cl BTB03892 C/C(=N\NC(=S)NCC(C)(C)C)/c1cc(ccc1O)F BTB04140 Cc1cc(cc(c1)/N=C\2/NC(C(=C)S2)(C)C)C BTB04295 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCC(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)c5ccco5 SPB07923 CC(=O)c1cc2ccccc2oc1=O BTB03234 c1ccc(c(c1)c2nc(no2)c3ccc(cc3)Cl)NC(=O)c4ccc(c(c4)Cl)Cl BTB03478 CS(=NC(=O)c1cccnc1Oc2ccccc2)(=O)c3ccc(cc3)Cl KM02964 c1cc2c(cc1OC/C(=N/O)/N)non2 KM07268 CC(C)(C)NC(=S)N/N=C/c1ccc(c(c1)O)O BTB03916 CSc1nccc(n1)c2ccc(s2)S(=O)(=O)Nc3ccc(cc3)Cl KM04144 CSc1nccc(n1)c2ccc(s2)S(=O)(=O)Nc3cccc(c3)C(F)(F)F KM04146 c1cc(ccc1NC(=O)NCCSCc2csc3c2cc(cc3)Cl)Cl KM07354 CC1=C(C(C(=C(N1)C)C#N)c2cccs2)C#N RJC03421 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCc4cccc(c4)[N+](=O)[O-])c5ccco5 SPB07925 c1ccc(cc1)OC(=O)c2ccc3c(c2)scn3 KM07380 CC(=O)c1ccc2c(c1)CCO2 KM05976 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)Cl)CSCc3nc(cs3)c4ccc(cc4)Cl KM05962 Cc1cc(ccc1NC(=S)N2CCc3cc(c(cc3C2Cc4ccc(c(c4)OC)OC)OC)OC)Cl BTB00995 C1CN(CCC1C(=O)N)CCO KM08619 c1cc(ccc1NC(=S)NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)F KM05821 CC(=O)NC1CCN(CC1)C(=S)Nc2cc(ccc2Cl)Cl BTB01008 Cc1c(c(no1)c2ccccc2)C(=O)NC3CCSC3=O KM03960 COc1cccn(c1=O)Cc2nnc(o2)SCC(=O)c3ccccc3 KM07272 c1cc(cc(c1)SC(=O)c2csc(n2)c3ccc(cc3)OCc4ccc5c(c4)non5)C(F)(F)F KM07274 CCOC(=O)c1c([nH]c(=O)[nH]1)C KM07154 CN1c2ccsc2C(=O)/C(=C\Nc3cccc(c3)C(F)(F)F)/S1(=O)=O KM04148 CN1c2ccsc2C(=O)/C(=C\Nc3ccc(cc3)F)/S1(=O)=O KM04149 CN1c2ccsc2C(=O)/C(=C/Nc3cccc(c3)Cl)/S1(=O)=O KM04151 c1cc(sc1)C(=O)/C(=C/c2ccc(cc2)OC(=O)c3ccc(cc3Cl)Cl)/C#N KM06025 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(=O)Nc3ccc(cc3)Cl BTB07403 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2)O)C(=O)OC RJC03434 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCC(=O)c4ccc(cc4)C#N SPB07931 Cn1c(nnc1SCc2ccc(cc2Cl)Cl)Cc3c4ccccc4c(=O)n(n3)C KM07378 CCOC(=O)NC(=S)NC(C)(C)C NH00514 c1ccnc(c1)C(=N)NC(=O)c2cnccc2C(F)(F)F SPB07190 c1cc(ccc1SC(=O)N2CCOCC2)Cl SPB07203 CSc1nnc(s1)Sc2c(cc(cn2)Br)[N+](=O)[O-] SPB07426 c1cc(ccc1c2csc(n2)COc3ccc4c(c3)non4)Cl KM07277 c1ccc(c(c1)NS(=O)(=O)c2cccs2)SCc3ccc4c(c3)non4 KM07290 CC(C)(C)c1csc(n1)c2ccc3c(c2)non3 KM07316 COc1ccc(cc1)c2ccnc(n2)S KM04163 CN1c2ccsc2C(=O)/C(=C\Nc3ccncc3)/S1(=O)=O KM04154 c1ccc(cc1)NC(=O)ON=C2CC3CCCC(C2)N3Cc4cccs4 KM08828 Cn1c(nnc1SCc2ccccc2)Cc3c4ccccc4c(=O)n(n3)C KM07382 Cn1c(nnc1SCC(=O)c2ccc(cc2Cl)Cl)Cc3c4ccccc4c(=O)n(n3)C KM07385 c1cc(sc1)C(=O)Nc2c(cc(cc2F)F)C#N BTB03978 CCC(C)(C)NC(=S)N/N=C/c1ccccc1SC(C)(C)C BTB03999 Cn1c2c3cc(cc(c3ncc2c(=O)[nH]1)F)F BTB04001 c1cc(sc1)c2[nH]c(nn2)Sc3c(cc(cn3)Br)[N+](=O)[O-] SPB07417 CC(C)(C)c1ccc(cc1)c2nnc(n2CCCOC)Sc3c(cc(cn3)Br)[N+](=O)[O-] SPB07418 CC1=C(C(C(=C(N1)C)C#N)c2ccc(c(c2)OC)OC)C#N RJC03427 Cc1c(sc2c1-c3c(cnc(n3)SCC(=O)c4ccc(cc4)Cl)S(=O)(=O)N2C)C KM07151 c1cc2c(cc1C(=O)Nc3ccc(cc3Cl)Cl)scn2 KM07307 CCOC(=O)c1c(c2cccc(c2nc1SC)C(F)(F)F)N3CCOCC3 KM08800 c1ccc(cc1)n2c(=O)[nH]c(=O)c(n2)C#N KM08724 CCOC(=O)c1c(c(sc1N)C)C KM04171 c1cc(sc1)CSc2ccc(cc2[N+](=O)[O-])C(F)(F)F KM04173 CCOC(=O)c1c(c2cccc(c2nc1SC)Cl)O KM08730 CS(=O)(=O)NCCSCc1csc2c1cc(cc2)Cl KM07387 c1cc2c(cc1C(=O)O/N=C(/c3ccc(cc3Cl)Cl)\N)scn2 KM07390 c1ccc(c(c1)/C=C(/C#N)\C(=O)c2ccc(cc2)Cl)OCc3c(cccc3Cl)Cl KM05972 COC(=O)c1cc(c(nc1)Sc2[nH]c(nn2)c3ccccc3)[N+](=O)[O-] SPB07442 c1cc2c(cc1OCC#N)non2 KM07257 c1cc(cc(c1)SCC(=O)N2CCC(CC2)C(F)(F)F)C(F)(F)F SPB07222 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl KM03238 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cc(c(cc3NC(=O)C)Cl)F BTB03678 CCOC(=O)c1c2c(c(s1)/S(=N/S(=O)(=O)c3ccc(cc3)Cl)/C)C=CCC2 KM06074 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NOC(=O)c3ccc(cc3)Cl KM04311 COC(=O)c1ccc(cc1)Oc2c(=O)c3ccc(cc3oc2C(F)(F)F)O BTB14910 c1cc(ccc1C2SCCS2)OCC(=O)NNC(=O)C(Cl)Cl SPB01294 c1cc(ccc1C(=O)OCCSc2c(ccs2)[N+](=O)[O-])Cl KM07412 Cc1c(sc2c1C(=O)/C(=C\Nc3ccc(cc3)OC)/S(=O)(=O)N2C)C KM04334 CC(C)(C)NC(=S)N/N=C\c1cccc(c1OCc2ccccc2)OC BTB03911 CC(C)(C)NC(=S)N/N=C/c1c2ccccc2ccc1O BTB03912 c1ccc(cc1)SCc2nc(no2)c3cccc(c3)[N+](=O)[O-] BTB02936 CC1(CC(=O)C=C(S1)SCc2c(cccc2Cl)Cl)C KM03953 c1cc(c(c(c1)Cl)Oc2ccc(cc2)S(=O)(=O)Oc3ccc(cc3)Cl)[N+](=O)[O-] BTB02920 COc1ccc2cc(oc2c1)C(=O)c3ccc(c(c3)Cl)Cl BTB02922 c1cc(c(cc1C(=O)c2cc3cc(ccc3o2)Cl)Cl)Cl BTB02923 CC(=O)OCc1ccccc1S(=O)(=O)c2ccccc2COC(=O)C BTB14936 C1C2CC3(CC1CC(C2)(C3)O)CCC(=O)O BTB14959 CCCCC#Cc1cc(cnc1)C(=O)NNC(=O)c2ccccc2 KM09462 CC1(Cc2c(c(sc2Cl)SC)/C(=N\O)/C1)C KM05979 CN1CCN(CC1)c2ccccc2/C=C/3\c4ccccc4NC3=O SEW05754 CC(C)(C#C)NS(=O)(=O)c1ccc(cc1)Oc2c(cccc2Cl)[N+](=O)[O-] BTB02916 Cc1cc(cc(c1Cl)C)Oc2ccc(cn2)NC(=O)Nc3c(onc3c4c(cccc4Cl)Cl)C BTB03885 CC(C)S(=O)(=O)/C(=C(/N1CCCC1)\SC)/C#N KM02932 CC(C)(C)c1ccc(cc1)CSc2nnc(n2c3ccc(cc3)OCc4ccccc4)c5ccco5 SPB07926 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCc4ccc(cc4)Cl)c5ccco5 SPB07927 Cc1cc(no1)C(=O)NNC(=S)SC SPB01229 c1cc(ccc1CSc2[nH]c3cc(c(cc3n2)F)Cl)[N+](=O)[O-].Br BTB03704 CS(=NC(=O)c1ccc(s1)c2ccccn2)(=O)c3ccc(cc3)Cl KM03114 COC(=O)c1ccc(s1)c2ccccn2 KM03116 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3Sc4ncc(s4)[N+](=O)[O-] SPB07894 CC1(Cc2c(c(n3c(n2)cc(n3)c4cccs4)SC)C(=O)C1)C KM02940 c1cc(ccc1c2nnc(o2)c3ccc(cc3)Cl)Cl MBE00287 CC(C)S(=O)(=O)c1cc(sc1SC)NC(=O)Nc2cccc(c2)C(F)(F)F KM04057 CN1c2ccsc2C(=O)/C(=C\Nc3ccccc3Cl)/S1(=O)=O KM04150 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NNS(=O)(=O)c3ccc(cc3)Cl KM04051 c1ccc(c(c1)C(=O)Nc2cc(c(cc2NC(=O)c3ccccc3Cl)Cl)F)Cl BTB03692 CC(C)(C)c1cc([nH]n1)C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] SPB01230 CC(C)(C)c1cc([nH]n1)C(=O)N/N=C/N(C)C SPB01232 c1cc(ccc1c2csc(n2)c3ccc(c(c3)Cl)F)Cl.Br BTB03709 c1cc(ccc1C(=N)N)C(F)(F)F.Cl SPB01314 Cn1c(nnc1SCc2cccc(c2)C#N)C(F)(F)F KM03118 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(nc3)Oc4ccc(cc4)C(C)(C)C BTB03891 CC(C)(C)NC(=S)N/N=C/c1cccc(c1O)O BTB03915 CC(=O)Nc1c(cc(cc1F)F)C#N BTB03955 CSc1nccc(n1)c2ccc(s2)S(=O)(=O)N3CCCCC3 KM04142 Cn1c(cnc1SCC(=O)Nc2cccc(c2)C(F)(F)F)C(=O)OC KM05892 CC1(CCc2cc(ccc2O1)c3ccnc(n3)SCC(=O)OC)C KM05857 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccccn2)C(=O)OC RJC03438 CSc1c(cn(n1)c2ccccc2)C(=O)Nc3ccc(cc3)Cl KM08787 CCOC(=O)c1cc(n[nH]1)C(C)(C)C SPB01225 CCOC(=O)c1c(nsc1N)C KM04205 c1ccnc(c1)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM04209 COCc1cc(nc(n1)c2ccc(cc2)C(F)(F)F)O SPB01316 c1ccc(c(c1)Oc2ccc(cc2[N+](=O)[O-])C#N)Cl SPB01319 c1cc(oc1)CS(=O)(=O)Cc2nc(on2)c3ccc(cc3)Cl KM03123 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=C(\C#N)/C(=O)c3ccc(cc3)Cl KM04296 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=C(\C#N)/C(=O)c3cccs3 KM04297 Cc1c(c(n(n1)S(=O)(=O)c2ccc(s2)c3ccnc(n3)SC)C)Br KM04156 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)Nc3ccccc3Cl KM04063 CC(=O)O/N=C/1\CC(Cc2c1c(sc2Br)SC)(C)C KM04066 CC1(C=Cc2cc(ccc2O1)/C(=N/OC(=O)Nc3cccc(c3)C(F)(F)F)/N)C KM06986 CC1(C=Cc2cc(ccc2O1)/C(=N/OC(=O)Nc3ccc(cc3Cl)Cl)/N)C KM06987 c1cc(ccc1c2csc(n2)c3ccc(c(c3)Cl)F)F.Br BTB03710 Cc1c(c(n(n1)Cc2nnc(n2C)SCC(=O)c3cccc(c3)[N+](=O)[O-])C)[N+](=O)[O-] KM04213 Cc1ccc(cc1)S(=O)(=O)CCN(C)Cc2cccnc2 KM04113 Cc1c2c(c(sc2sc1C(=O)/C=C/N(C)C)Br)C KM04116 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=C(\C#N)/S(=O)(=O)c3cccc(c3)Cl KM04285 c1cc2c(cc1n3c(=O)[nH]nc3Sc4ncc(s4)[N+](=O)[O-])OCCO2 SPB07895 c1cc(cc(c1)[N+](=O)[O-])CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4 SPB07896 Cn1cc(cc1/C=C(\C#N)/C(=O)c2ccco2)C(=O)c3ccc(cc3)Cl KM07224 CC(C)S(=O)(=O)c1cc(sc1SC)NC(=O)Nc2ccc(cc2)Cl KM04058 c1cc(ccc1S(=O)(=O)CCN2C(=O)CSC2=O)Cl KM04061 CN1c2ccsc2C(=O)/C(=C\Nc3ccccn3)/S1(=O)=O KM04153 c1ccc(cc1)C#Cc2ccc(o2)C(=O)NNC(=O)Nc3ccccc3 KM08656 c1ccc(cc1)C#Cc2ccc(o2)C(=O)NNC(=O)Nc3cc(cc(c3)Cl)Cl KM08657 c1ccc(c(c1)/C=C(/C#N)\C(=O)c2cccc(c2)C(F)(F)F)OCc3c(cccc3Cl)Cl KM05971 CCOC(=O)c1c-2c(c(s1)SCc3ccccc3)S(=O)(=O)N(c4c2scc4)C KM04215 Cc1cc(nc2c1c(nn2C)C)n3c(cc(n3)c4cccc(c4)C(F)(F)F)N KM04217 Cc1c(c(n(n1)Cc2nnc(n2C)SCC(=O)C(C)(C)C)C)[N+](=O)[O-] KM04218 CC(C)(C)c1cc(cc(c1)NC(=O)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4)C(C)(C)C SPB07897 C/C(=N\OCC(=O)O)/c1ccc(cc1)Cl KM05916 CS(=NS(=O)(=O)c1ccc(s1)c2ccccn2)(=O)c3ccccc3 KM04077 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N=S(=O)(C)c3ccc(cc3)Cl)C(F)(F)F KM04078 Cc1ccc(cc1)NC(=O)c2ccc3c(c2)CCO3 KM07003 COc1ccc2c(c1)CCC3C2=NN(C3)c4ccccc4 KM07006 c1cc(sc1)c2nnco2 KM04120 CN1c2ccsc2C(=O)CS1(=O)=O KM04121 Cc1c(c(n(n1)Cc2nnc(n2C)SCC(=O)Nc3cccc(c3)C(F)(F)F)C)[N+](=O)[O-] KM04220 Cc1c(c(n(n1)Cc2nnc(n2C)SCC(=O)Nc3ccccc3)C)[N+](=O)[O-] KM04221 CSc1c(cc(s1)C(=O)O)c2nc(cs2)c3ccc(cc3)Cl KM04122 c1ccc(c(c1)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4)Cl SPB07898 c1cc(sc1)C(=O)/C(=C/c2ccsc2Sc3ccc(cc3)Cl)/C#N KM05913 Cc1cc(n(n1)S(=O)(=O)c2ccc(s2)c3ccnc(n3)SC)C KM04155 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3cscc3S(=O)(=O)C(C)C KM03054 Cc1c(c(on1)C)S(=O)(=O)N=S(=O)(C)c2ccc(cc2)Cl KM04161 CN(CCS(=O)(=O)c1ccc(cc1)Cl)Cc2cccnc2 KM04162 c1cc(sc1)c2ccnc(n2)S KM04074 CC1(Cc2c(c(sc2c3ccn(n3)C(=O)Nc4cccc(c4)Cl)SC)/C(=N/OC)/C1)C KM04069 CCOC(=O)CNS(=O)(=O)c1ccc(s1)c2cc(n(n2)C)C(F)(F)F KM04082 c1ccc(cc1)C#Cc2ccc(o2)C(=O)Nc3ccccc3 KM08671 COc1ccccc1NC(=O)c2ccc(o2)C#Cc3ccccc3 KM08672 c1cc(sc1)/C=N/NC(=O)CSCc2nc(cs2)c3ccc(cc3)Cl KM05992 CCCn1c(=O)c(nn(c1=O)c2ccccc2)C#N KM08767 Cc1c(c(n(n1)Cc2nnc(n2C)SCc3ccc(cc3)Cl)C)[N+](=O)[O-] KM04226 CCOC(=O)c1c(c(sc1N(C)S(=O)(=O)C)C)C KM04237 c1ccc(c(c1)/C=C(\C#N)/C(=O)c2cccs2)OCc3c(cccc3Cl)Cl KM05994 c1cc(ccc1Sc2c(ccs2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl)Cl KM05917 c1cc(ccc1NC(=O)/N=S/2\CCC3(C2)OCCO3)OC(F)(F)F KM05940 Cn1c(nnc1SCC(=O)c2ccccc2)CSCc3nc(cs3)c4ccccc4 KM05942 Cc1ccc(cc1)C(=O)OCc2cn(c3c2cc(cc3)[N+](=O)[O-])Cc4ccccc4 RH01268 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)OS(=O)(=O)c3ccccc3Cl KM05806 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)OS(=O)(=O)c3ccc(cc3)Cl KM05789 COc1cc(cc(c1OC)OC)C(=O)NC(=S)NC(=O)N BTB00525 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCCc4c3ccc(c4)OC BTB00794 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)OC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM05791 CN1c2ccccc2-c3c(c(sc3C(=O)Sc4ccccc4)SC)S1(=O)=O KM04135 CN1c2ccccc2-c3c(c(sc3C(=O)NCC4CC4)SC)S1(=O)=O KM04137 c1cc(ncc1C(F)(F)F)N2CCSCC2 KM05926 Cn1c(cc(n1)c2ccc(s2)c3ccnc(n3)SCC(=O)c4ccc(cc4)Cl)C(F)(F)F KM05996 Cn1c(cc(n1)c2ccc(s2)c3ccnc(n3)SCC(=O)c4ccccc4)C(F)(F)F KM05997 c1c(cc(cc1C(F)(F)F)S(=O)(=O)/N=S\2/CCC3(C2)OCCO3)C(F)(F)F KM05937 CCOC(=O)c1c(c(sc1NS(=O)(=O)C)C)C KM04174 COc1ccccc1C2CCN(CC2)C(=O)CSc3nnc(s3)NC(=O)c4cccnc4Oc5ccccc5 RH01267 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCC(=O)Nc4ccccc4C(F)(F)F)c5ccco5 SPB07918 CCCn1c(=O)c(nn(c1=O)c2ccccc2)/C(=N/O)/N KM08771 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Nc2c(cc(cn2)C(F)(F)F)Cl KM08777 CC(=O)N1CCSC1C(=O)NN KM06004 Cn1c(cc(n1)c2ccc(s2)c3ccnc(n3)SCC(=O)Nc4ccccc4)C(F)(F)F KM06001 c1cc(cc(c1)S(=O)(=O)NNC(=O)CSCc2nc(cs2)c3ccc(cc3)Cl)C(F)(F)F KM06011 c1ccc(cc1)c2csc(n2)CSCc3nnc(n3c4ccc(cc4)Cl)S KM05948 c1ccc(cc1)SCC(=O)c2ccc(s2)CC(=O)O KM05951 C(CCC(=O)O)C/C(=N/O)/C(=O)N KM05923 c1cc(ccc1S(=O)(=O)N=S2CCN(CC2)c3ccc(cn3)C(F)(F)F)Cl KM05936 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)CSCc3nc(cs3)c4ccc(cc4)Cl KM05949 c1ccc(cc1)C#Cc2cc(cnc2)NC(=O)N3CCCC3 KM08630 c1ccc(cc1)S(=O)(=O)C2=CCS(=O)(=O)C2 KM05800 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)OC(=O)Nc3ccc(cc3)OC(F)(F)F KM05802 Cc1ccc(cc1)NC(=S)NNC(=O)c2c(c3ccccc3s2)Cl BTB00810 Cn1c(nnc1SCC(=O)Nc2ccccc2)CSCc3nc(cs3)c4ccccc4 KM05945 COc1ccc(cc1)S(=O)(=O)NNC(=O)CSCc2nc(cs2)c3ccc(cc3)Cl KM06012 CCOC(=O)CSc1c([nH]c2c1cccc2)C KM06016 c1cc(cc(c1)NC(=S)NC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)C(F)(F)F KM05819 CC(C)(C)CNC(=S)N/N=C/c1cc(cc(c1O)I)I BTB04125 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccccc3C(=O)NNc4cc(cc(c4)Cl)Cl BTB04945 Cn1c(cc(n1)c2ccc(s2)C(=O)N(C)C)C(F)(F)F KM03003 c1ccc(c(c1)C(=O)Nc2ccc(cc2)N3CCC(CC3)n4cccc4)Cl KM08700 c1ccc(cc1)C(=O)Nc2ccc(cc2)N3CCC(CC3)n4cccc4 KM08701 Cc1ccc(cc1)SCC(=O)c2ccc(s2)CC(=O)O KM05953 c1c(cnc(c1Cl)N2CCSCC2)C(F)(F)F KM06020 c1cc(ccc1/C=C(\C#N)/C(=O)c2ccc(cc2)Cl)OC(=O)c3ccc(cc3)Cl KM06022 c1ccc(cc1)c2csc(n2)CSCC(=O)NNC(=O)Nc3ccccc3 KM06023 c1ccc(cc1)NC(=O)c2[nH]ccn2 KM08733 c1ccnc(c1)S(=O)(=O)/C(=C/N2CCC(CC2)n3cccc3)/C#N KM08634 c1cc(cc(c1)Cl)N2CCN(CC2)CCCSCC(=O)NNC(=O)Nc3ccc(cc3)Cl KM08643 CCOC(=O)NC(=O)/C(=N/Nc1cccc(c1)C(F)(F)F)/C#N KM08740 CCOC(=O)NC(=O)/C(=N/Nc1ccc(cc1)OC)/C#N KM08741 c1ccc2c(c1)OCC(O2)CNS(=O)(=O)c3cccc(c3)C(F)(F)F KM07132 CC(C)N(Cc1ccc(cc1)N(C)C)C(=S)Nc2ccc(cc2)Cl BTB01074 c1ccc(cc1)C(=O)N/N=C/c2cc(ccc2N3CCCC3)[N+](=O)[O-] JFD03002 c1ccc(cc1)C(=O)/C(=C/N2CCC(CC2)n3cccc3)/C#N KM08708 CCOC(=O)C(=C(Nc1ccc(cc1)Cl)SCC(=O)Nc2ccc(cc2)C(C)C)C(=O)OCC KM08719 c1ccc(cc1)C#Cc2ccc(o2)C(=O)O KM08625 CC(C)(C)S(=O)(=O)/C(=C/N1CCC(CC1)n2cccc2)/C#N KM08635 c1ccn(c1)C2CCN(CC2)CCS(=O)(=O)c3ccc(cc3)F KM08637 c1ccc(c(c1)C2CC(=CC(=S)S2)N3CCCCC3)Cl KM04187 COC(=O)c1cc(c(nc1)Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)[N+](=O)[O-] SPB07443 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(c(s3)C(=O)C)C KM07149 CCOC(=O)c1c(c2cc(ccc2nc1SC)Cl)O KM08720 c1c(nc2c(cnn2c1C(F)(F)F)/C(=N/O)/N)C(F)(F)F KM03006 c1cc2c(cc1c3nc(cs3)C(=O)Sc4ccc(cc4Cl)Cl)non2 KM07346 c1ccc(cc1)SC(=O)c2ccc3c(c2)scn3 KM07381 CCOC(=O)c1c(c2cc(ccc2nc1SC)Cl)N3CCOCC3 KM08801 CCOC(=O)c1c(c2cccc(c2nc1SC)C(F)(F)F)N3CCCC3 KM08803 c1ccc(cc1)NC(=O)c2ccc3c(c2)scn3 KM07379 CC1(C(CCC1(C)C(=O)N2CCCCC2)C(=O)N3CCCCC3)C BTB14916 CCOC(=O)COc1ccc2c(cc(=O)oc2c1)c3ccccc3 BTB14927 c1cc(cc(c1)n2c(=O)[nH]c(=O)c(n2)C#N)C(F)(F)F KM08742 CSc1c(cc(s1)C(=O)Nc2cccc(c2)Cl)c3nc(cs3)c4ccc(cc4)Cl KM04196 Cc1c2c(c(sc2sc1c3ccn(n3)C)Br)C KM04198 Cn1c(cnc1SCc2c(cccc2Cl)Cl)C(=O)OC KM05881 Cn1c(cnc1SCc2ccc(cc2)[N+](=O)[O-])C(=O)OC KM05882 Cn1cnc(c1Sc2ccc(cn2)C(F)(F)F)[N+](=O)[O-] KM05884 COc1ccc(cc1)OC(=O)c2csc(n2)COc3ccc4c(c3)non4 KM07320 Cc1ccc(cc1)S(=O)(=O)/N=S\2/CCCSC2 KM03008 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)Cl KM03010 c1cc(ccc1OC(=O)c2csc(n2)COc3ccc4c(c3)non4)Cl KM07323 Cc1cc(n2c(n1)c(c(n2)C(C)(C)C)Cl)C KM07375 c1ccc(cc1)n2c(=O)n(c(=O)c(n2)C#N)Cc3ccc(cc3)Cl KM08746 CCOC(=O)c1c(c2cc(ccc2nc1SC)Cl)Sc3ccc(cc3)C KM08758 c1ccc(cc1)CN2C3CCCC2CC(=NO)C3 KM08808 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N=S(=O)(C)c3ccc(cc3)Cl KM03042 CCOC(=O)c1c(c2cccc(c2nc1SC)Cl)Oc3cccc(c3)Cl KM08810 c1cc(cc(c1)Cl)N2CCN(CC2)CCCSCC(=O)N/N=C/c3ccc(cc3)Cl KM08645 c1ccc(cc1)C#Cc2ccc(o2)C(=O)NN KM08646 COc1ccc(cc1)n2c(=O)[nH]c(=O)c(n2)C#N KM08743 CCOC(=O)c1c(c2cccc(c2nc1SC)C(F)(F)F)O KM08747 c1ccc(cc1)NC(=S)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F AW00565 c1cc(cc(c1)O)/C=N/CCNc2nccc(n2)C(F)(F)F AW00573 c1ccc(cc1)SC(=O)c2csc(n2)c3ccc4c(c3)non4 KM07347 c1cc(ncc1[N+](=O)[O-])Sc2[nH]c(nn2)N BTB07991 Cn1c(nnc1SCC(=O)c2ccccc2)Cc3c4ccccc4c(=O)n(n3)C KM07384 CNC(=O)c1ccc(s1)c2cc(nn2C)C(F)(F)F KM03033 COC(=O)c1cccc2c1c(ccc2)Sc3ccccc3C#N BTB14933 c1cc2c(=O)ccoc2cc1OC(=O)c3ccc(cc3Cl)Cl KM07405 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3SCC(=O)Nc4ccc(cc4)Cl)c5ccco5 SPB07922 CCCCOC(=O)c1ccc(s1)c2ccccn2 KM03117 CN1c2ccsc2C(=O)/C(=N\Nc3ccccc3Cl)/S1(=O)=O KM04203 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])Sc3ccc(cc3)Cl BTB07537 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N=S(=O)(C)c3ccccc3 KM03041 Cc1c(c(n(n1)Cc2nnc(n2C)SCc3c(cccc3Cl)F)C)Br KM03046 Cc1c(c(n(n1)Cc2nnc(n2C)SCc3ccccc3Cl)C)Br KM03047 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N=S(=O)(C)c3ccc(cc3)Cl KM02809 CC(C)CSc1c(c(c(s1)C(=O)O)c2ccc(cc2)Cl)C#N KM02822 CC(C)S(=O)(=O)/C(=C(/N1CCCCC1)\SC)/C#N KM02933 CC(C)CSc1c(c(cs1)c2ccc(cc2)Cl)C#N KM02825 Cc1cc(no1)NC(=O)c2ccc3c(c2)scn3 KM07386 CC12CCC3C(C1CCC2C(=O)COC(=O)CCC(=O)O)CCC4=CC(=O)CCC34C NRB03870 Cc1cc(no1)COC(=O)Nc2ccc(cc2)Cl SPB01234 CCCn1c(=O)c(nn(c1=O)c2cccc(c2)C(F)(F)F)/C(=N/O)/N KM08774 CCCn1c(=O)c(nn(c1=O)c2ccc(cc2)OC)C#N KM08775 COc1ccccc1NC(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM06069 CS(=O)(=O)N1CCN(CC1)c2cc(nc3c2cccc3)C(F)(F)F KM08877 c1cc(ccc1Sc2c(cc(s2)S(=O)(=O)N)[N+](=O)[O-])Cl KM08878 CC(C)(C)c1cc([nH]n1)C(=O)N/N=C/c2cc(cc(c2O)Br)Br SPB01231 CC(=O)CSc1c(c(c(s1)C(=O)C)c2ccccc2)C#N KM06102 Cc1cc(nn1C)C(=O)O/N=C/c2ccccc2Cl SPB01253 c1ccc-2c(c1)CCc3c2nc4ccccc4c3N5CCOCC5 RJC03449 CC(=O)c1ccc(s1)C#CCOC(=O)Nc2ccccc2 KM08995 CC(C)(C(=O)N(C)c1ccccc1)Oc2cc(n(n2)C)C(F)(F)F BTB09358 CCCCCCCc1c(c2cccc3c2n(c1=O)c4c3cccc4)O BTB10330 COC(=O)C1=C(CSC1)NNc2c(cc(cn2)Cl)C(F)(F)F KM08885 CN(C)C(=O)c1ccc2c(c1)scn2 KM07393 Cn1c(c(c(n1)c2ccccc2)C#N)S(=O)(=O)C KM03078 c1ccc(cc1)S(=O)(=O)CCSCC(=O)NN KM03083 c1cc(ccc1c2csc(n2)COc3ccc4c(c3)non4)[N+](=O)[O-] KM07309 Cn1c(c(cn1)C(=O)NC(=O)Nc2ccc(cc2)F)[N+](=O)[O-] KM03145 Cc1cc(no1)C(=O)N/N=C/c2cc(c(c(c2)Br)O)Br SPB01263 Cc1cc(no1)C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] SPB01264 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)NC2CCN(CC2)Cc3ccccc3 KM08887 Cc1cc(no1)C(=O)NNC(=O)Nc2ccc(cc2)Cl SPB01200 CCOC(=O)c1cc(n[nH]1)C SPB01217 c1cc(oc1)CS(=O)(=O)/C(=C/Nc2ccc(cc2)Cl)/C#N KM03084 CC(C)(C)NC(=S)Nc1cc(ccc1N2CCCCC2)C(F)(F)F BTB03529 CC(C)(C)SC(=O)c1cccnc1SCCS(=O)(=O)c2ccccc2 KM06256 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])Oc3ccc(cc3)Cl BTB07536 CC(=O)c1ccc(s1)C#CCOC(=O)c2ccc(cc2)Cl KM09006 c1cc(sc1)CN2C3CCCC2CC(=NOC(=O)c4ccc(cc4)F)C3 KM08839 COC(=O)c1ccc(cc1Cl)[N+](=O)[O-] KM08842 CCCCCCc1c(c2cccc3c2n(c1=O)c4c3CCCC4)O BTB10363 CC(C)NC(=O)NC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl SPB01192 CC(C)S(=O)(=O)/C(=C/Nc1ccc(cc1)Cl)/C#N KM03157 CCOC(=O)c1cc(on1)C SPB01195 c1cc(cc(c1)N2C(=O)C3N(C2=S)CCS3)C(F)(F)F KM08954 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM04281 c1ccc(cc1)C(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F KM08927 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)SCC(=O)Nc4ccc(cc4)C(F)(F)F SPB07941 c1ccc(cc1)c2c(snn2)N SPB07968 c1ccc(cc1)NC(=O)CSCC(=O)N/N=C/c2ccccc2Cl KM09004 c1ccc(cc1)CN2C3CCCC2CC(=NOC(=O)Nc4ccc(cc4)Cl)C3 KM08844 CSc1c(cn(n1)c2ccccc2)C(=O)Sc3cccs3 KM08846 Cc1c2c3c(cnc2n(n1)C)c(=O)[nH]n3C KM08897 Cc1ccc(cc1)NC(=S)NCc2cccnc2 DSHS01288 CC(=O)c1cc2c(s1)SCC(=O)N2 KM08900 c1cc(ccc1OCC(=S)N)Cl SPB01323 c1cc(cc(c1)Cl)N/C=C(\C#N)/S(=O)(=O)Cc2ccco2 KM03093 c1cc(ccc1CSc2ccc(cc2)Cl)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F KM03153 Cc1c(sc2c1C(=O)CS(=O)(=O)N2C)C KM04248 Cc1ccc(cc1)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(F)(F)F KM03174 CC1(Cc2c(c(sc2Br)SC)/C(=N/OC(=O)c3ccc(cc3)Cl)/C1)C KM04080 c1ccc(cc1)S(=O)(=O)CCSCC(=O)NNS(=O)(=O)c2ccc(c(c2)Cl)Cl KM03097 c1ccc(cc1)S(=O)(=O)CCSCC(=O)NNC(=O)c2ccccc2Cl KM03101 CC(=O)c1ccc(s1)C#CCOC(=O)c2cccs2 KM09011 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=O)Nc2ccccc2 KM08989 c1cc2c(cc1Cl)c(cs2)CSCCNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM07397 c1ccc(cc1)S(=O)(=O)CCSCC(=O)N/N=C/c2ccc(cc2)Cl KM03089 c1ccc(cc1)S(=O)(=O)CCSCC(=O)N/N=C/c2ccsc2 KM03090 CCOC(=O)c1cnc(nc1C(F)(F)F)Sc2ccc(c(c2)Cl)F GK02973 CN1c2ccsc2C(=O)/C(=N\Nc3ccsc3C(=O)OC)/S1(=O)=O KM04246 c1ccc(c(c1)SCc2ccc(cc2)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl KM03161 c1cc(ccc1CSc2ccc(c(c2)Cl)Cl)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F KM03162 COC(=O)c1cscc1OC(=O)c2ccc(cc2)C(F)(F)F KM03167 COC(=O)C(Cc1csc2c1cc(cc2)Cl)NC(=O)c3ccccc3 KM08960 COC(=O)C(Cc1csc2c1cc(cc2)Cl)NC(=O)c3ccc(cc3)C(F)(F)F KM08961 c1c(c(sc1S(=O)(=O)N)N2CCCC2)[N+](=O)[O-] KM08941 CN(C)/C=C/C(=O)c1cc(ccc1SC)[N+](=O)[O-] KM03212 COc1ccc(cc1c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] KM03214 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2c(nc3ccccc3n2)Nc4ccc(cc4)Cl RJC03486 CSc1ccc(cc1c2ccn(n2)S(=O)(=O)C)[N+](=O)[O-] KM03281 c1cc(ccc1S(=O)(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl KM06043 Cc1c(c2ccccc2[nH]1)Sc3ccc(cc3)Cl KM06044 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)OC(C)C KM07463 CCOC(=O)c1c(nsc1NN=C(C#N)C(=O)C(C)(C)C)C KM04405 CCOC(=O)c1ccc(cc1)n2c(=O)ccs2 KM04416 CC(=O)c1cc(ccc1Sc2ccc(cc2)Cl)[N+](=O)[O-] KM03192 c1cc(sc1)Sc2ccc(cn2)C(F)(F)F KM04211 c1ccc(cc1)C2CC(=O)C=C(S2)SCC(=O)Nc3ccc(cc3)Cl KM04266 Cc1cc(nc2c1c(nn2C)C)N/N=C/c3ccc(cc3)Cl KM04103 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)SC SPB07940 C/C(=N/O)/c1ccc(cc1)OCCOc2ccc(cc2)C#N RJC03471 CC(C)(C)NC(=O)COc1cc(n(n1)C)C(F)(F)F BTB09355 CCOC(=O)Cn1c(=O)c2cnc3c(c2n1C)c(nn3C)C KM08998 c1cc(ccc1c2nc(c(o2)N)C#N)C(F)(F)F SEW05762 CSc1c(cn(n1)c2ccccc2)C(=O)Nc3ccccc3 KM08834 CSc1c(cn(n1)c2ccccc2)C(=O)Nc3cccc(c3)C(F)(F)F KM08835 CC(C)(C)c1c(c2nc(cc(n2n1)N(C)C)C(F)(F)F)I KM07429 Cc1cc(n(n1)CCS(=O)(=O)c2ccc(cc2)Cl)C KM04179 c1ccc(cc1)OC(=O)NC(=S)Nc2ccccc2OC(F)(F)F KM04258 c1cc(sc1)C/C(=N/OC(=O)c2ccc(cc2)Cl)/N SPB07947 CC(C)S(=O)(=O)c1cc(sc1)C(=O)OC KM03273 CCOC(=O)c1c2c(c(s1)SC)C(=O)CCC2 KM03288 Cn1c(nnc1SCc2cccc(c2)c3nc(on3)c4ccc(cc4)Cl)C(F)(F)F KM03148 COc1ccc(cc1c2cc[nH]n2)[N+](=O)[O-] KM03165 CC(=O)c1cc(c(s1)Sc2ccc(cc2)Cl)[N+](=O)[O-] KM03202 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)NC(=O)Nc3cccc(c3)C(F)(F)F KM04181 Cc1c(c(n(n1)CCS(=O)(=O)c2ccc(cc2)Cl)C)Br KM04184 c1ccc(cc1)OC(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM04223 CC(C)(C)c1cccc(c1)NC(=S)N2CCSCC2 NH00686 CC1=C(C(C(=C(N1)C)C#N)c2ccccc2)C#N BTB11137 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)Nc2cc(ccc2Cl)Cl KM03236 CC(C)(C)c1cc2nc(cc(n2n1)NN)C(F)(F)F KM07431 CC(c1ccc2c(c1)OCCO2)NC(=O)c3cc(c(c(c3)OC)OC)OC SW00134 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCC(=O)c4ccccc4 SPB07861 c1cc(ccc1Sc2ccc(cc2c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl)[N+](=O)[O-])Cl KM03277 COc1ccc(cc1)c2ccnc(n2)SC KM04183 CCOC(=O)c1c-2c(c(s1)SCc3ccc(cc3)Cl)S(=O)(=O)N(c4c2scc4)C KM04216 Cc1c2c(c(sc2sc1c3cc[nH]n3)Br)C KM04193 CCSc1c2c(c(s1)C(=O)OC)CC(CC2=O)(C)C KM03232 CCCCCCCCCCCc1nnc(n1C)SCc2ccc(cc2)Cl SPB01436 CS(=N/C=C(\C#N)/C(=O)c1ccc(cc1)Cl)(=O)c2ccc(cc2)Cl KM03291 c1cc2c(cc(nc2c(c1)Br)C(F)(F)F)O KM07477 c1cc2c(cc(nc2c(c1)Br)C(F)(F)F)Oc3ccc(cc3)F KM07484 c1cc2c(cc1c3nc(cs3)C(=O)Oc4ccc(cc4Cl)Cl)non2 KM07342 CC12CCC3c4ccc(cc4CCC3C1CCC2=O)N NRB04207 CC(=O)Nc1ccc(cc1)/C=C(\C#N)/C(=O)N RB00034 CCOC(=O)/C(=C\c1ccncc1)/C#N RB00247 Cn1cc(cc1/C=C(\C#N)/S(=O)(=O)c2cccs2)C(=O)c3ccc(cc3)Cl KM07228 Cc1c(c(no1)c2ccc(cc2)Cl)C(=O)C SPB04957 Cc1c(c(no1)c2ccccc2)C(=O)N=S(=O)(C)C KM03263 c1cc(oc1)CS(=O)(=O)Cc2nc(cs2)C(=O)N/N=C/c3ccc(cc3)Cl KM03266 c1cc(ccc1C(=O)n2ccc(n2)c3cc(ccc3Sc4ccc(cc4)Cl)[N+](=O)[O-])Cl KM03271 CSc1c(cn(n1)c2ccccc2)C(=O)Oc3ccc(cc3)Cl KM08849 CCOC(=O)c1ccc(c(c1)NC(=O)C(Cl)(Cl)Cl)N2CCCCC2 DSHS01057 Cc1nc(cs1)c2ccc3c(c2)CCC(=O)N3 BTB09232 c1cc(cc(c1)[N+](=O)[O-])c2c(c[nH]n2)Br KM03193 CSc1c(cc(s1)C(=O)Nc2ccccc2Cl)c3nc(cs3)c4ccc(cc4)Cl KM04195 CN(C)c1ccc(c(c1)Cl)C2Nc3ccccc3C(=O)N2 DSHS00673 Cn1c(nnc1SCC(=O)N)CSCc2nc(cs2)c3ccc(cc3)Cl KM05985 CCOC(=O)c1c2c(c(s1)/S(=N/S(=O)(=O)c3cccc(c3)Cl)/C)C=CCC2 KM06081 c1cc(sc1)C(=O)NOc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] BTB09588 Cn1c(nnc1SCC(=O)Nc2ccc(cc2Cl)Cl)Cc3c4ccccc4c(=O)n(n3)C KM07389 CCCCc1ccc(cc1)NC(=O)N=S2CCN(CC2)C(=O)c3ccc(cc3)Cl KM06246 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/OC(=O)Nc3ccccc3 KM04376 c1ccc2c(c1)c(n[nH]2)Oc3ccc(cn3)[N+](=O)[O-] BTB08565 c1ccc2c(c1)C(=C(CCN2S(=O)(=O)c3ccc(cc3)Cl)C#N)O BTB08585 c1cc(ccc1C(=O)NNC(=O)c2ccc(cc2)OC(F)(F)F)C(F)(F)F SPB03439 c1ccc2c(c1)OCC(O2)CSCCOC(=O)Nc3ccc(cc3)OC(F)(F)F KM07252 Cc1ccc(cc1)SC(=O)N2CCOCC2 SPB07204 CSc1ccc(cc1c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl)[N+](=O)[O-] KM03272 CCOC(=O)c1c2c(c(s1)SCc3ccccc3)C(=O)CC(C2)(C)C KM03283 c1cc(sc1)c2nc(cc(n2)O)C(F)(F)F RF01778 c1cc(ccc1S(=O)(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)Cl KM06062 CS(=O)(=O)n1ccc(n1)c2cccc(c2)[N+](=O)[O-] KM03194 CCN(c1ccccc1)C(=S)Nc2ccc(cc2)C SW00056 c1cc(oc1)CS(=O)(=O)CC(=S)N KM03209 Cn1c(cc(n1)c2ccc(s2)c3ccnc(n3)SCc4ccccc4)C(F)(F)F KM05989 c1ccc(cc1)C(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM06053 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Nc2ccccc2 KM08765 CCOC(=O)/C(=C/c1ccc(cc1C(C)(C)C)c2nccs2)/C#N KM04346 Cc1c(sc2c1C(=O)/C(=C\Nc3ccccn3)/S(=O)(=O)N2C)C KM04348 Cc1c(sc2c1C(=O)/C(=C\Nc3cccnc3)/S(=O)(=O)N2C)C KM04349 CC(=O)N1CSCC1C(=O)NNS(=O)(=O)c2ccc(cc2)Cl KM06093 CC(C)(C)c1ccc(cc1)NC(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl KM06178 c1cc(sc1)S(=O)(=O)n2ccc(n2)c3ccc4c(c3)CCO4 KM06207 c1cc(ccc1NC(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)Cl KM06066 c1cc(c(c(c1)Cl)SC(=O)N2CCOCC2)Cl SPB07205 Cc1ccc(cc1)SCC(=O)N2CCC(CC2)C(F)(F)F SPB07221 CCCCC#Cc1cc(cnc1)C(=O)N/N=C/c2ccc(cc2)C(F)(F)F KM09457 CCCCC#Cc1cc(cnc1)C(=O)N/N=C/c2cccc(c2)OC KM09458 COc1ccc(cc1)NC(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM06068 CCCCCCCc1c(c2cccc3c2n(c1=O)c4c3CCCC4)O BTB10329 CC(C)Oc1cc(nc2c1cc(cc2)CSCCO)C(F)(F)F KM07489 CCOC(=O)c1c(c2cccc(c2nc1SC)Cl)Sc3c(cccc3Cl)Cl KM08778 CC1c2cc(ccc2N(C1=O)C)S(=O)(=O)N3CCOCC3 KM04371 Cc1c(c(c([nH]1)C)C(=O)OC)/C=C(\C#N)/C(=O)c2ccc(cc2)Cl KM08858 c1cc(ccc1NC(=O)N=S2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C#N)Cl KM06205 COc1ccc(cc1)Nc2c(nc3ccccc3n2)NS(=O)(=O)c4ccccc4 RJC03492 CN1CCN(CC1)c2c(cc(s2)S(=O)(=O)N)[N+](=O)[O-] KM08943 Cn1c(cc(n1)OS(=O)(=O)c2ccc(cc2Cl)Cl)C(F)(F)F BTB09223 c1ccc(cc1)NNC(=O)c2cccs2 BTB08638 c1cc(ccc1/C=N/Oc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])C(F)(F)F BTB09581 c1cc(sc1)CN2C3CCCC2CC(=NOC(=O)c4ccc(cc4)Cl)C3 KM08831 c1ccc(cc1)NC(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F KM08837 CC(C)(C)c1c(c2nc(cc(n2n1)OC)C(F)(F)F)Br KM07421 c1cc(ccc1c2nc(cs2)C(=O)Sc3ccc(cc3Cl)Cl)OCc4ccc5c(c4)non5 KM07273 c1cc(ccc1C(=O)N2CCS(=NS(=O)(=O)c3ccc(cc3)Cl)CC2)Cl KM05847 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2Cl)O)C(=O)OCC)C)C RJC03429 C#CCSc1n[nH]c(=O)n1c2ccc(cc2)OCc3ccccc3 SPB07928 c1cc(c(cc1C#N)[N+](=O)[O-])N2CCSCC2 KM06160 c1cc(ncc1C(F)(F)F)SCc2ccc(o2)C(=O)O KM06169 Cc1c(sc2c1C(=O)/C(=C\Nc3ccccc3Cl)/S(=O)(=O)N2C)C KM04332 CC(C)(C)/C(=N\Oc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/c2ccccc2 NRB02470 Cc1c(sc2c1C(=O)/C(=C\Nc3ccc(cn3)Cl)/S(=O)(=O)N2C)C KM04396 CC(C)(C)c1cc2nc(cc(n2n1)N(C)C)C(F)(F)F KM07416 CCCn1c(=O)c(nn(c1=O)c2ccccc2)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N KM08790 CCCn1c(=O)c(nn(c1=O)c2ccccc2)/C(=N/OC(=O)Nc3ccc(cc3)OC(F)(F)F)/N KM08791 c1cc(ccc1C(=O)N=S2CCN(CC2)C(=O)c3ccc(cc3)Cl)Cl KM06132 c1cc(c(cc1Cl)N)C(=O)N2CCSCC2 KM06158 COc1ccc(cc1)NC(=S)Nc2ccc(cc2)OCc3ccccc3 SPB07934 CC(C)(C)c1cc2[nH]c(cc(=O)n2n1)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM06224 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=C(\C#N)/S(=O)(=O)C KM04283 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F KM08992 c1ccc(cc1)CN2C3CCCC2CC(=NOC(=O)c4ccccc4)C3 KM08832 c1cc(oc1)CS(=O)(=O)/C(=C/c2ccc(cc2)Cl)/C#N KM03086 c1ccc(cc1)/C(=N/OC(=O)c2ccc3c(c2)scn3)/N KM07394 COc1cc(nc2c1cc(cc2)Br)C(F)(F)F KM07395 CSc1c(cn(n1)c2ccccc2)C(=O)N3CCOCC3 KM08857 CCOC(=O)C1=C(C(=O)N(C1)C(C)(C)C)Nc2ccc(cc2)OC(=O)C KM05900 CCSc1nccc(n1)c2ccc3c(c2)CCC(O3)(C)C KM05858 CC1(Cc2c(c(sc2Cl)S(=O)C)C(=O)C1)C KM05861 CCSCc1cc(nc(n1)c2ccc(cc2)C(F)(F)F)O SPB01334 CN(C)C(=O)c1cccnc1SCCS(=O)(=O)c2ccccc2 KM06218 Cc1cc(cc(c1O)C)c2c3ccccc3c(=O)n(n2)C BTB08278 c1cc2c(nc1)n3ccsc3nc2=O.Cl BTB08368 Cc1c(cc(c(n1)SCCNS(=O)(=O)c2cccc(c2)C(F)(F)F)C#N)c3csc(n3)C BTB09501 Cn1c(cc(n1)OCC(=O)N(C)c2ccccc2)C(F)(F)F BTB09356 CC(C)(C)c1c(c2nc(cc(n2n1)OC)C(F)(F)F)I KM07422 CC(C)(C)c1c(c2nc(cc(n2n1)N(C)C)C(F)(F)F)Br KM07427 CN1CCN(CC1)c2cc(nc3c2cccc3)c4cccnc4 RJC03446 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3Sc4ncc(s4)[N+](=O)[O-])c5ccco5 SPB07935 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)/C=C(/C#N)\S(=O)(=O)c4ccccc4 KM09000 c1ccc(cc1)c2nc(c(o2)N)C(=S)N SEW05766 COc1ccc(cc1)c2nc(no2)COc3ccc4c(c3)non4 KM07442 CCSc1cc(nc2n1nc(c2Cl)C(C)(C)C)C(F)(F)F KM07443 CSc1c(cn(n1)c2ccccc2)C(=O)Sc3ccccn3 KM08847 Cc1ccc(cc1)SC2CN(C2)C(c3ccccc3)c4ccccc4 KM08894 c1ccc(cc1)C(c2ccccc2)N3CC(C3)Sc4nc5ccccc5s4 KM08895 c1cc2c(cc1C(=O)O)scn2 CC05901 c1ccc(c(c1)OCC(=S)N)Cl SPB01326 c1ccc(cc1)S(=O)(=O)CCSCC(=O)NNS(=O)(=O)c2ccc(s2)Cl KM03098 c1ccc(cc1)NC(=O)NNC(=O)CSCCS(=O)(=O)c2ccccc2 KM03099 c1cc(cc(c1)Cl)OCC(=S)N SPB01327 CCSCc1cc(nc(n1)c2ccc(cc2)C(F)(F)F)OC(=O)N(C)C SPB01338 Cc1ccc(cc1)S(=NC(=O)CO/N=C(\C)/c2ccc(cc2)Cl)(=O)C KM05964 Cn1ccc(n1)c2cccc(c2)NC(=O)Nc3ccccc3 KM03079 c1ccc(cc1)c2cc3[nH]c(cc(=O)n3n2)c4cc(cc(c4)C(F)(F)F)C(F)(F)F KM06223 CCC(CNCCO)Nc1nc2c(n1C)c(=O)n(c(=O)n2C)C RJC03501 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NO KM04276 COC(=O)c1ccc(nc1)N/C=N/O BTB08862 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl KM08876 CCCCOC(=O)CCCSc1c(cc(c(n1)C)c2csc(n2)C)C#N BTB09635 CCOC(=O)C(C(c1ccco1)NC(=S)N)C(=O)C(F)(F)F BTB09804 CC(C)(C)c1cc2nc(cc(n2n1)C#N)C(F)(F)F KM07435 Cc1nc(no1)c2cccc(c2)CSc3nnc(n3C)C(F)(F)F KM03150 c1ccc(cc1)S(=O)(=O)CCSCC(=O)NNC(=O)Nc2ccc(cc2)Cl KM03100 CCN(CCS(=O)(=O)c1ccc(cc1)C)C(=O)c2ccc(s2)c3cc(nn3C)C(F)(F)F KM03106 COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F KM08925 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)c4ccc(cc4)Cl KM08926 Cc1c2c(c(sc2sc1c3c(cn(n3)C)Br)Br)C KM04267 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=C(\C#N)/C(=O)c3cccc(c3)C(F)(F)F KM04301 c1cc(ccc1C2OCCO2)C(=S)N KM03256 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N=S(=O)(C)C KM03262 CSc1c(cn(n1)c2ccccc2)C(=O)N3CCCC3 KM08855 CSc1c(cn(n1)c2ccccc2)C(=O)N3CCCCC3 KM08856 Cn1c(nnc1SCc2cccc(c2)/C(=N\OC(=O)Nc3ccc(cc3)Cl)/N)C(F)(F)F KM03141 CCOC(=O)CNC(=O)C(CC(=O)N)NC(=O)OC(C)(C)C KM03183 c1cc(c(cc1C(=O)NC(=O)N2CCCC2)[N+](=O)[O-])Oc3cc(cc(c3)Cl)Cl SPB01193 Cc1cccc(c1)c2nc3cccc(c3c(=O)o2)F BTB04365 c1cc2c(c(c1)F)c(=O)oc(n2)c3ccc(cc3Cl)Cl BTB04366 c1ccc(cc1)C#Cc2ccc(o2)C(=O)Sc3ccc(cc3)Cl KM08668 CC(C)S(=O)(=O)c1c(n2c(cc(n2)c3ccccc3)nc1SC)N KM02977 CCCS(=O)(=O)c1cscc1NC(=O)c2c(onc2c3ccccc3Cl)C KM02979 c1ccc(cc1)C#Cc2ccc(cc2)c3ccn(n3)C(=O)c4ccc(cc4)Cl KM08986 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)SCC(=O)c4ccc(c(c4)Cl)Cl SPB07953 c1ccc(cc1)COc2ccc(cc2)NC(=S)NN SPB07960 c1ccc(cc1)COc2ccc(cc2)n3cnnc3S SPB07961 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)Nc4ccc(cc4)OC(F)(F)F KM08840 Cn1c2c3cccc(c3nc(c2c(=O)[nH]1)SC)Cl KM08890 COc1ccc(cc1)OC(=O)c2cn(nc2SC)c3ccccc3 KM08850 c1cc(cc(c1)Cl)OC/C(=N/O)/N SPB01345 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCC(=O)Nc4ccc(cc4)C(F)(F)F SPB07867 Cc1c(c(n(n1)Cc2nnc(n2C)SCC(=O)Nc3ccc(cc3)Cl)C)[N+](=O)[O-] KM04219 CCN(c1ccccc1)C(=S)Nc2cccc(c2)C(F)(F)F SW00052 CN1c2ccsc2C(=O)/C(=C\Nc3nc(nc(n3)SC)C4CC4)/S1(=O)=O KM04264 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)c4c(cc(cn4)Cl)C(F)(F)F KM08931 c1cc(ccc1c2csc(n2)CSCC(=O)NNS(=O)(=O)c3ccc(cc3)Cl)Cl KM06010 CC(C)S(=O)(=O)c1cc(sc1)C(=O)O KM03293 CC(C)S(=O)(=O)c1cc(sc1)NC(=O)Nc2ccc(cc2)Cl KM03301 Cc1ccc(c2c1CCC2)Oc3c(cc(cn3)C(F)(F)F)Cl BTB09387 CC(=O)c1cc(c(s1)SCc2ccc(cc2)Cl)[N+](=O)[O-] KM03206 Cc1csc2c1c(c(s2)c3ccnc(n3)SCc4ccccc4)C KM04319 CC1c2cc(ccc2N(C1=O)C)S(=O)(=O)Nc3ccc(cc3Cl)Cl KM04325 Cc1c(c(n(n1)Cc2nnc(n2C)SCc3c(cccc3Cl)F)C)[N+](=O)[O-] KM04224 CCOC(=O)c1c(n(/c(=N\N=C(C)C)/s1)C)C SPB01411 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Nc2ccccc2C(F)(F)F KM08773 c1cc2c(c(c1)F)c(ncn2)O BTB04061 c1cc(c(cc1F)F)NC(=O)CSc2ccc(cn2)[N+](=O)[O-] BTB04070 C/C(=N\NC(=S)NC(C)(C)C)/c1cc(ccc1O)F BTB04139 c1ccc(cc1)Oc2c(cccn2)c3nc4cccc(c4c(=O)o3)F BTB04364 CC(=O)c1ccc(s1)C#CCOC(=O)Nc2cc(cc(c2)Cl)Cl KM08996 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N=S(=O)(C)C KM03247 CCCCNC(=O)N1CCN(CC1)c2cc(nc3c2cccc3)C(F)(F)F KM08852 CNC(=S)NNC(=O)CSCCS(=O)(=O)c1ccccc1 KM07452 CC(C)(C)c1c(c2nc(cc(n2n1)N(C)C)C(F)(F)F)Cl KM07428 CSc1c(cc(s1)C(=O)N2CCCCC2)c3nc(cs3)c4ccc(cc4)Cl KM04234 CCCCCCCCCCCC(=O)NN SPB01420 CCCCCCCCCCCc1nnc(n1C)S SPB01425 CCOC(=O)c1cnc([nH]1)SCC(=O)c2ccc(cc2)Cl KM06212 c1ccc(cc1)C(=O)C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl SEW04330 c1ccn2c(c1)c[nH]c2=S BTB04390 Cn1c2c(cc(s2)C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N)c(n1)C(F)(F)F GK02730 CCOC(=O)c1c[nH]c(n1)S KM06163 c1cc(ncc1C(F)(F)F)SCc2ccc(o2)C(=O)NN KM06170 Cc1c(c(sc1NC(=O)Nc2ccccc2)S(=O)(=O)C)C=C KM03723 c1cc2c(c(c1)F)c(=O)oc(n2)c3c(cccc3F)F BTB04368 CSc1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB05275 Cc1cc(nc2c1c(nn2C)C)NNC(=O)c3ccccc3Cl KM04177 c1ccc(cc1)NC(=O)CSCC(=O)N/N=C/c2cccs2 KM09005 CCOC(=O)c1c-2c(c(s1)SC)S(=O)(=O)N(c3c2cccc3)C KM03284 COc1ccc(cc1)C(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM06054 c1ccc(cc1)C(=O)NCc2cccs2 KM04419 c1ccc(cc1)S(=O)(=O)NCc2cccs2 KM04420 CS(=O)(=O)NCc1cccs1 KM04421 c1cc(cc(c1)[N+](=O)[O-])c2ccn(n2)C(=O)c3ccc(cc3)Cl KM03200 c1cc(ccc1C(=O)NC(=S)Nc2ccc(cc2)F)C(F)(F)F SPB01430 CN1c2ccsc2C(=O)/C(=N\Nc3cccc(c3)C(F)(F)F)/S1(=O)=O KM04204 Cc1cc(nc2n1nc(c2Cl)C3CC3)C(F)(F)F KM07363 Cn1c(nnc1S)Cc2c3ccccc3c(=O)n(n2)C KM07366 c1cc(c(cc1[N+](=O)[O-])C#N)Oc2ccc3c(c2)non3 KM08809 CN1c2ccsc2-c3c(c(sc3C(=O)O)SC)S1(=O)=O KM04318 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCC(=O)c4ccc(cc4)Cl SPB07864 COc1ccc(cc1)S(=O)(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl KM06046 CC(C)(C)c1ccc(cc1)S(=O)(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl KM06047 CCOC(=O)c1c2c(c(s1)/S(=N/S(=O)(=O)c3ccccc3)/C)C=CCC2 KM06083 Cc1cc(nc2c1c(nn2C)C)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM04178 c1ccc(cc1)n2c(nnc2Sc3c(cc(cn3)Br)[N+](=O)[O-])O SPB07420 COC(=O)c1cc(c(nc1)Sc2nnc(n2CC=C)O)[N+](=O)[O-] SPB07448 CC(C)c1ccc(cc1)n2c(nnc2Sc3c(cc(cn3)C(=O)OC)[N+](=O)[O-])c4ccc(cc4)C(C)(C)C SPB07444 c1ccc(c(c1)SCc2cccc(c2)C(=O)CC#N)Cl KM05872 CCOC(=O)c1c2c(c(s1)/S(=N/C(=O)Nc3ccc(cc3)Cl)/C)C=CCC2 KM06072 CC1(C2CCC1(c3c2c(n(n3)c4ccccc4)C(F)(F)F)C)C BTB14906 Cc1csc2c1c(c(s2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4Cl)Cl)C KM04328 CN1c2ccsc2C(=O)/C(=C\Nc3ncccn3)/S1(=O)=O KM04188 c1ccc(cc1)SCC(=S)N KM04192 c1cc(ccc1NC(=O)c2csc(n2)COc3ccc4c(c3)non4)Cl KM07322 CCOC(=O)c1c(c2cccc(c2nc1SC)C(F)(F)F)Oc3ccc(cc3)OC KM08811 COc1ccc(cc1)NC(=O)CSc2c(c(cc(c2Cl)Cl)Cl)Cl KM08813 c1cc2c(cc1c3ccnc(n3)S)CCO2 KM06173 CC(=O)n1ccc(n1)c2cccc(c2)[N+](=O)[O-] KM03107 c1cc(sc1)C(=O)n2ccc(n2)c3ccc4c(c3)CCO4 KM06208 Cc1csc2c1c(c(s2)c3ccnc(n3)SCC(=O)NCC=C)C KM04337 CCOC(=O)c1c2c(c(s1)/S(=N/C(=O)c3ccccc3)/C)C=CCC2 KM06085 Cc1c(c(c2n1CSC2)C(=O)OC)C(=O)OC KM06088 CCOC(=O)c1c2c(c(s1)/S(=N/C(=O)c3ccc(cc3)Cl)/C)C=CCC2 KM06057 CCCCCc1ccc(cc1)NC(=O)NNc2cc(ccc2Cl)Cl BR00031 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)O KM07408 c1cc(ccc1NC(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl KM06094 CSc1c(cc(s1)C(=O)Nc2cccc(c2)C(F)(F)F)c3nc(cs3)c4ccc(cc4)Cl KM04194 CSc1c(cc(s1)C(=O)N2CCOCC2)c3nc(cs3)c4ccc(cc4)Cl KM04197 Cn1c(=O)c2ccccc2c(n1)CC(=O)NN KM07355 c1cc(ccc1C(=O)CSc2[nH]c(=O)c3c(n2)CSC3)Cl KM07359 c1cc(ccc1Oc2cc(nc3c2ccc(c3)Cl)C(F)(F)F)F KM07487 Cc1ccc(cc1)c2cc(nc(c2C#N)OC)c3ccc(cc3OCc4ccc(cc4)F)OCc5ccccc5 FM00001 COc1c(c(c2c(n1)-c3ccccc3CC2)c4ccc5ccccc5c4)C#N FM00015 CCOC(=O)c1c2c(c(s1)/S(=N/S(=O)(=O)c3ccccc3Cl)/C)C=CCC2 KM06075 CCOC(=O)c1c2c(c(s1)/S(=N/S(=O)(=O)c3ccc(cc3)C)/C)C=CCC2 KM06080 c1cc(ccc1[N+](=O)[O-])OC(=O)c2csc(n2)COc3ccc4c(c3)non4 KM07324 CCCCNC(=O)NNC(=O)CSCc1nc(cs1)c2ccccc2 KM06091 c1cc(ccc1c2nc(cs2)C(=O)N3CCOCC3)OCc4ccc5c(c4)non5 KM07269 c1cc(oc1)CS(=O)(=O)C/C(=N/O)/N KM03112 c1ccc(cc1)CSc2nccc(n2)c3ccc4c(c3)CCO4 KM06184 c1ccc(c(c1)Oc2ccc(cc2[N+](=O)[O-])/C(=N/O)/N)Cl SPB01320 CC1(Cc2c(c(sc2Cl)SC)/C(=N/OCC(=O)Nc3ccccc3)/C1)C KM06193 c1ccc(cc1)COC(=O)N2C(CNC2=O)C(=O)O KM08977 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCNCC3 KM08985 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Nc2cccc(n2)C(F)(F)F KM08783 CCOC(=O)c1c(c2cccc(c2nc1SC)Cl)N3CCCCC3 KM08784 c1ccc(cc1)CN2C3CCCC2CC(=NOC(=O)c4ccc(cc4)F)C3 KM08830 CCOC(=O)c1cc(nn1C(=O)c2ccccc2Cl)C SPB01242 CCOC(=O)c1cc(nn1C(=O)c2c(cccc2Cl)F)C SPB01243 Cc1c(c(c([nH]1)C)C(=O)OC)/C=C(\C#N)/C(=O)c2ccc(cc2)OC KM08859 Cc1c(c(c([nH]1)C)C(=O)OC)/C=C(\C#N)/C(=O)c2cccc(c2)C(F)(F)F KM08862 c1ccc(cc1)C(=O)CSc2[nH]c(=O)c3c(n2)CSC3 KM07360 c1cc(ccc1S(=O)(=O)N2CCSC2C(=O)NN)Cl KM05903 CS(=O)(=O)/C(=C/c1ccsc1Sc2ccc(cc2)Cl)/C#N KM05910 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Nc2c(cc(cn2)Cl)C(F)(F)F KM08782 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc(c(c2)Cl)F)Oc3ccc(cc3Cl)Cl CD08946 c1c(cc(cc1Cl)Cl)OCC(=S)N SPB01328 CCCCc1ccc(cc1)NC(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM06247 c1ccc(cc1)S(=O)(=O)CCSc2c(cccn2)C(=O)Oc3ccc(cc3Cl)Cl KM06252 CCOC(=O)c1c(c(sc1NC=C(C(=O)NC(=O)OCC)C(=O)NC(=O)OCC)C)C KM08764 c1cc(ccc1C(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)Cl KM06052 Cn1cnc(c1Sc2cccs2)[N+](=O)[O-] KM06089 c1ccc2c(c1)CCN(C2)/C=C(\C#N)/C(=O)c3cccs3 KM06107 CCCCCCCCCCCc1nnc(n1C)SC SPB01435 c1cnc(nc1C(F)(F)F)NCC/N=C/c2cc(cc(c2)F)F AW00569 c1cc(ccc1NC(=O)N2CCN(CC2)c3c(nccn3)C#N)Cl KM09018 c1cc(ccc1NC(=O)N2CCN(CC2)c3c(nccn3)C#N)OC(F)(F)F KM09019 c1cc(c(c(c1)Cl)Cn2c(nnn2)c3ccc(cc3)Cl)Cl GK02986 c1cnccc1C2=NNC(C2)(C(F)(F)F)O KM08939 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/OC(=O)c3ccccc3Cl KM04374 c1ccc(c(c1)C(=O)ONC(=O)CC2C(=O)Nc3ccccc3S2)Cl KM04364 c1ccc2c(c1)NC(=O)C(S2)CC(=O)NOC(=O)c3cccc(c3)C(F)(F)F KM04365 Cc1c(sc2c1C(=O)/C(=C\Nc3ncccn3)/S(=O)(=O)N2C)C KM04447 Cn1c(cc(n1)OCC(=O)O)C(F)(F)F BTB09348 Cn1c(cc(n1)OCC(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F BTB09350 Cc1c(snn1)C(=O)N=S(=O)(C)c2ccccc2 KM03268 COC(=O)C(Cc1csc2c1cc(cc2)Cl)NC(=O)c3ccc(cc3)Cl KM08959 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)c4cccs4 KM08928 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)c4ccc(cn4)C(F)(F)F KM08930 CSc1c(c(n[nH]1)NS(=O)(=O)c2ccc(cc2)Cl)c3ccccn3 PD00196 Cc1csc2c1c(c(s2)c3ccnc(n3)SCC(=O)NCc4ccccc4)C KM04359 CCOC(=O)c1c2c(c(s1)SC(C)C)C(=O)CC(C2)(C)C KM03258 c1ccc(cc1)C(c2ccccc2)N3CC(C3)OC(=O)Nc4ccc(cc4)OC(F)(F)F KM08871 Cc1c(snn1)C(=O)N=S(=O)(C)C KM03269 c1cc(oc1)CS(=O)(=O)Cc2nc(cs2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl KM03270 c1ccc(cc1)C2CC(=O)C=C(S2)SCC(=O)c3cccc(c3)[N+](=O)[O-] KM04384 c1ccc(cc1)/C=N/NC(=O)CSC2CN(C2)C(c3ccccc3)c4ccccc4 KM09064 CC(C)(C)c1csc(n1)c2c3c(c(s2)SC)C(=O)CCC3 KM04388 C/C(=N\O)/c1csc(n1)c2ccccc2 SPB03579 c1cc(cc(c1)NC(=O)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F)C(F)(F)F SPB06947 COc1cscc1C(=O)N/N=C/c2ccc(cc2)Cl KM04460 Cc1c2c(c(sc2sc1c3ccnc(n3)SCc4ccccc4)Br)C KM04466 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)SCC=C SPB07943 c1ccc(cc1)C(=O)O/N=C(/Cc2cccs2)\N SPB07946 CC1c2cc(ccc2N(C1=O)C)C(=O)C KM04293 c1cc(ccc1Sc2ccc(cc2c3cc[nH]n3)[N+](=O)[O-])Cl KM03216 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)CS(=O)(=O)Cc3ccco3 KM03219 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC=C)Br)C KM04458 CCn1c(cc(n1)C)C(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F SPB02531 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/Nc3ccc(cc3F)F KM04361 CC(C)(C(=O)O)Oc1cc(n(n1)C)C(F)(F)F BTB09345 c1cc(ccc1C2CC(=CC(=S)S2)N3CCCCC3)Cl KM04450 c1cc(ccc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)OC(F)(F)F KM04452 Cn1c(c(c(n1)c2ccc(s2)Br)Br)C(F)(F)F KM03211 Cn1c(cc(n1)c2ccc(s2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)Cl)C(F)(F)F KM06002 CC(C)(C)NC(=O)C(C)(C)Oc1cc(n(n1)C)C(F)(F)F BTB09360 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC(=O)Nc4ccc(cc4Cl)Cl)Br)C KM04467 CC(=O)c1ccc(s1)C#CCOC(=O)c2ccc(cc2)C(F)(F)F KM09010 Cn1cccc1c2nnc(n2c3ccc(cc3Cl)Cl)S CD10614 CNC(=S)NNC(=O)CC1C(=O)Nc2ccccc2S1 KM07424 CCOC(=O)c1c[nH]c(n1)SCC KM06183 CCCn1c(=O)c2c([nH]cn2)n(c1=O)c3ccccc3C KM09936 CC(C)(C)C(=O)CSC1=CC(=O)CC(S1)c2ccccc2 KM04401 CS(=O)(=O)c1c(c(n[nH]1)c2ccccc2)C#N KM00790 Cc1ccc(cc1)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F SPB06950 CSc1nc(n(n1)c2cc(ccn2)C(F)(F)F)N SPB06891 CSc1nc(n(n1)c2c(cccn2)C(F)(F)F)N SPB06892 c1cc(sc1c2ccno2)C(=S)N SEW02270 CN1C(=O)c2cccc3c2c(ccc3)C1=O NRB04170 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)N2CCc3c2cccc3 KM05385 c1ccc(cc1)C#Cc2ccc(cc2)c3ccn(n3)C(=O)c4cccs4 KM09012 C/C(=N\O)/C12CC3(CC(C1)(CC(C3)(C2)C)C)C BTB14969 c1cc(cc(c1)NC(=S)NC(=O)c2ccc(cc2)C(F)(F)F)C(F)(F)F SPB01431 c1ccc2c(c1)c(=O)n3n(c2=O)CC=CC3 KM07482 c1ccc(cc1)c2csc(n2)CSCC(=O)NNC(=O)Nc3ccc(cc3)Cl KM06090 c1ccc(cc1)NC(=O)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F SPB06945 Cc1cc2ncc(c(n2n1)C)c3cnc(nc3)SCCS(=O)(=O)c4ccc(cc4)Cl KM04766 Cc1c(cnn1c2c(cc(cc2Cl)Cl)Cl)c3ccn[nH]3 CD10635 Cc1ccc(cc1)N2CCN(CC2)CCCCCC(=O)OC RH00937 COc1c(c(cc(n1)c2ccccc2)c3ccc4c(c3)OCO4)C#N FM00020 CCSc1cc(nc2n1nc(c2)C(C)(C)C)C(F)(F)F KM07426 c1cc(c(nc1)SCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)C(=O)NCc3cccs3 KM06189 CC1=Cn2c(=O)c3ccccc3c(=O)n2C1 KM07445 COc1cc(c(cc1OC)[N+](=O)[O-])CC/N=C/c2ccccc2O CD03598 c1ccc(cc1)CN\2C(=CS/C2=C(/C#N)\C(=O)N)c3ccc(cc3)Br DP00032 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC(=O)c4ccc(cc4Cl)Cl)Br)C KM04495 c1ccc(cc1)N2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM09015 c1cnc(c(n1)C#N)N2CCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl KM09016 c1ccc(cc1)C\2=NOC(=O)/C2=C\c3ccc(cc3)Cl BTB06169 c1ccc(cc1)Sc2ccc(cc2[N+](=O)[O-])S(=O)(=O)Nc3ccc(c(c3)C(F)(F)F)Cl DSHS00919 Cc1c(sc2c1C(=O)/C(=C\Nc3ccncc3)/S(=O)(=O)N2C)C KM04350 Cc1csc2c1c(c(s2)c3ccnc(n3)SCC(=O)c4ccccc4)C KM04353 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/Nc3ccccn3 KM04360 c1ccc(cc1)N2CCN(CC2)CCCCCC(=O)O.Cl RH00938 Cc1c(cnn1c2c(cc(cc2Cl)Cl)Cl)c3ccnc(n3)N CD10638 c1cc(c(cc1NS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F)Cl)Cl MWP00979 CCN(CC)C(=O)Sc1nc2cc(ccc2s1)Cl SPB01397 Cn1c(c(nc1Sc2cccs2)C#N)C#N KM07475 c1cc(ncc1C(F)(F)F)Sc2cc(nc3c2c(cc(c3)Cl)Cl)C(F)(F)F KM07476 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=O)Nc2cc(cc(c2)Cl)Cl KM08991 COC(=O)C(Cc1csc2c1cc(cc2)Cl)NC(=O)c3cccs3 KM08962 c1c(cc(c2c1nc(cc2O)C(F)(F)F)Cl)Cl KM07464 c1ccc2c(c1)[nH]c(n2)[C@H]([C@H](c3[nH]c4ccccc4n3)O)O BTB14921 CS(=NS(=O)(=O)c1ccc(cc1)OC(F)(F)F)(=O)c2ccc(cc2)Cl KM04440 c1ccc(c(c1)/C=N/NC(=O)c2cc(=O)nc3n2ccs3)Cl KM04506 COC(=O)c1cnn2c1nc(cc2C(F)(F)F)C(F)(F)F KM06153 c1cc(c(c(c1)Cl)Cn2nc(nn2)c3c(cccc3Cl)Cl)F GK02981 c1ccc(cc1)Cn2c(nnn2)c3ccc(cc3)Cl GK02982 CC1(Cc2c(c(sc2c3ccnc(n3)SC)SC)C(=O)C1)C KM04358 Cn1c(cnc1SCc2ccc(cc2)Cl)C(=O)N/N=C/c3ccc(cc3)Cl KM06100 COc1ccc(cc1)C(=O)/C(=C/N2CCc3ccccc3C2)/C#N KM06113 c1cc(sc1)CN2C3CCCC2CC(=NOC(=O)Nc4ccc(cc4)SC(F)(F)F)C3 KM08872 CCSc1cc(nc2n1nc(c2Br)C(C)(C)C)C(F)(F)F KM07436 c1cc2c(cc(nc2c(c1)OC(F)(F)F)C(F)(F)F)O KM07449 c1cc(ccc1c2n[nH]nn2)[N+](=O)[O-] GK02978 c1ccc2c(c1)C(=C3c4ccccc4C(=O)c5c3cccc5)c6ccccc6C2=O BTB15056 C=CCNc1nc(cs1)c2ccccc2.Br CD00254 CN(C)/C=C/C(=O)c1ccc2c(c1)CCO2 KM06148 COc1ccc(cc1)NC(=S)NNC(=O)CSCC(=O)Nc2ccccc2 KM09024 CCOC(=O)CSc1nccc(n1)c2c(c3c(csc3s2)C)C KM04344 c1cc(ccc1/C=N/NC(=O)c2cc(=O)nc3n2ccs3)Cl KM04415 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=S)Nc2ccccc2 KM09022 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F KM08924 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)c4cccc(n4)C(F)(F)F KM08932 CN(C)/C=C/C(=O)c1ccc(s1)C#N KM04274 c1ccc(cc1)C(c2ccccc2)N3CC(C3)Sc4ccc(cc4)Cl KM08893 CCOC(=O)c1c(c2cccc(c2nc1SC)Cl)N(C)CCO KM08899 Cc1c2c3c(cnc2n(n1)C)c(=O)n(n3C)Cc4ccc(cc4)Cl KM08912 CCOC(=O)C(=CNc1nc(cs1)c2cc(c(=O)[nH]c2C)C#N)C(=O)OCC BTB09200 c1cc(c(c(c1)Cl)Cn2nc(nn2)c3c(cccc3Cl)Cl)Cl GK02983 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)N KM04438 Cc1cc(nc(n1)N/C=C/2\C(=O)c3c(c(sc3N(S2(=O)=O)C)C)C)C KM04448 C/C(=N\O)/C(=O)c1ccccc1 GK02977 Cc1ccc(c(c1)Cn2c(=O)c3cnc4c(c3n2C)c(nn4C)C)C KM08913 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F KM04362 Cc1c(c(no1)c2ccccc2Cl)C(=O)N=S(=O)(C)C KM03261 CCC(C)Sc1c2c(c(s1)C(=O)OCC)CC(CC2=O)(C)C KM03264 CSc1c(c(n[nH]1)NS(=O)(=O)c2cccc(c2)C(F)(F)F)c3ccccn3 PD00203 COc1cscc1C(=O)NNC(=O)c2cccc(c2)C(F)(F)F KM04435 COc1cscc1C(=O)NN KM04436 CC(=O)ONC(=O)c1ccc(cc1)[N+](=O)[O-] KM03226 c1ccc(cc1)c2csc(n2)CS(=O)(=O)Cc3ccco3 KM03223 Cc1c2c3c(cnc2n(n1)C)c(=O)n(n3C)Cc4ccccc4 KM08914 Cc1ccc(cc1)C(=O)CSc2nnc(n2c3ccc(cc3)OCc4ccccc4)C SPB07937 CC1(CC(=O)C(C(=O)C1)SC(F)(F)F)C RJC03464 CSc1c(c(c(s1)C(=O)NC2CC2)c3ccc(cc3)Cl)C#N KM04256 c1cc(cc(c1)[N+](=O)[O-])c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl KM03195 Cc1ccc(c2c1CCC2)Oc3c(cc(cn3)Cl)C(F)(F)F BTB09401 CCOC(=O)c1c(nsc1N/N=C(\C#N)/C(=O)c2ccc(cc2)Cl)C KM04403 C1C2CC34CC5(C2=NNC5=O)CC1C3=NNC4=O BTB14947 CCOC(=O)c1c2c(c(s1)SC)/C(=N\OC)/CCC2 KM04461 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)S(=O)(=O)Nc4nccs4 DSHS00193 c1cc(ncc1C(F)(F)F)Sc2c(cc(s2)S(=O)(=O)N)[N+](=O)[O-] KM08935 Cc1c(snn1)C(=O)N/N=C/c2ccc(s2)[N+](=O)[O-] CD09192 CCCCc1c(c2cccc3c2n(c1=O)c4c3CC(CC4)C)O BTB10442 Cn1c2c(cc(s2)C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N)c(n1)C(F)(F)F GK02697 c1cc(ccc1CSc2nnc(s2)c3ccc(cn3)C(F)(F)F)Cl SPB06949 CC(C)(C(=O)Nc1ccc(cc1Cl)Cl)Oc2cc(n(n2)C)C(F)(F)F BTB09346 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)Nc2cccc(c2)C(F)(F)F KM03241 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC(=O)NCC=C)Br)C KM04480 CC(=O)c1cc(c(s1)Sc2cccc(c2Cl)Cl)[N+](=O)[O-] KM03205 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H]([C@H](O1)F)OC(=O)C)OC(=O)C)OC(=O)C NRB05159 Cn1c(nnc1S)CSc2ccccc2 KM04428 CCCCCCc1c(c2cccc3c2n(c1=O)c4c3cccc4)O BTB10368 CCCSc1c2c(c(s1)C(=O)OC)CC(CC2=O)(C)C KM03235 c1ccc(cc1)C(c2ccccc2)N3CC(C3)OC(=O)Nc4cc(cc(c4)Cl)Cl KM08870 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC(=O)NC(C)C)Br)C KM04474 c1ccc(cc1)S(=O)(=O)CCSc2c(cccn2)C(=O)Sc3ccc(cc3Cl)Cl KM06253 c1cc(c(nc1)SCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)C(=O)Oc3ccc(cc3Cl)Cl KM06254 Cc1ccc(cc1)C(=O)NNC(=O)CSC2CN(C2)C(c3ccccc3)c4ccccc4 KM09096 c1ccnc(c1)c2c(nnc(n2)c3ccc(cn3)C(F)(F)F)c4ccccn4 SPB06961 CC1(Cc2c(c(sc2Br)SC)C(=O)C1)C KM03644 CS(=NC(=O)c1ccc(cc1)OC(F)(F)F)(=O)c2ccc(cc2)Cl KM04485 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC(=O)NCc4ccccc4)Br)C KM04489 c1cc(cc(c1)NC(=O)/C=C/c2ccc(s2)c3cccs3)C(F)(F)F SEW02639 Cc1ccc(cc1)S(=O)(=O)Nc2c(nc3ccccc3n2)Nc4ccc(cc4)O RJC03489 Cc1csc2c1c(c(s2)c3ccnc(n3)SCC(=O)c4ccc(cc4Cl)Cl)C KM04367 C=CCSc1nnc(s1)c2ccc(cn2)C(F)(F)F SPB06952 c1cc(ccc1C(=O)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F)Cl SPB06953 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC(=O)Nc4ccccc4)Br)C KM04475 Cc1c2c(c(sc2sc1c3ccnc(n3)SCC(=O)Nc4cccc(c4)C(F)(F)F)Br)C KM04476 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)NNC(=O)Nc4ccccc4 KM08918 c1cc(c(nc1)SCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)C(=O)Nc3ccc(cc3Cl)Cl KM06159 Cc1c(c(c(c(c1C)C)C#CCOC2CCCCO2)C)C CD08945 c1cc(cnc1)c2nc(cs2)C(=O)NN MWP00333 CC1(CC(=O)O1)C23CC4CC(C2)CC(C4)C3 BTB14978 Cc1cccc(c1)OS(=O)(=O)c2c(c(sc2C(=O)OC)C(F)(F)F)c3ccccc3 SEW03500 Cc1c(c(c2n1CCS2)C(=O)O)C(=O)O KM06117 Cc1cc(c(cc1Sc2cc(c(cc2C)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F)C(C)(C)C)C(C)(C)C)Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB07504 COc1ccc(cc1)NC(=O)CSc2[nH]c(=O)c3c(n2)CSC3 KM07376 CCCCc1ccc(cc1)C(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM06235 Cc1ccc(n1CCN2CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F)C SEW04386 c1cc(ccc1C(=O)NCCSc2ccc(cc2)Cl)[N+](=O)[O-] BTB02956 c1ccc(cc1)c2c(nnc(n2)c3ccc(cn3)C(F)(F)F)c4ccccc4 SPB06959 CC(C)(C(=O)Oc1ccc(cc1Cl)Cl)Oc2cc(n(n2)C)C(F)(F)F BTB09357 CC(C)(C(=O)N(C)C)Oc1cc(n(n1)C)C(F)(F)F BTB09359 CO/N=C/1\CCCc2c1c(sc2C(=O)N/N=C/c3ccc(cc3)Cl)SC KM04499 CC1(CC(=O)C=C(S1)SCc2ccc(cc2)[N+](=O)[O-])C KM04508 CC(=O)c1ccc(s1)C#CCO KM08978 CCSc1ccc(cn1)/C(=N/OC(=O)c2cccs2)/N SEW04435 CCSc1ccc(cn1)/C(=N/OC(=O)C(C)(C)C)/N SEW04438 CCSc1ccc(cn1)/C(=N/OC(=O)c2cccc(c2)C(F)(F)F)/N SEW04439 Cc1c2c(n(n1)c3ccccc3)OC(=C(C2c4ccc(cc4)[N+](=O)[O-])C#N)N BTB14982 C1CC2(CCCC(C1)(C2)C(=O)O)C(=O)O BTB15000 CS(=NC(=O)c1ccc(cc1)OC(F)(F)F)(=O)c2ccccc2 KM04484 CS(=NC(=O)c1ccccc1OC(F)(F)F)(=O)c2ccc(cc2)Cl KM04486 C/C(=N\OCC(=O)Nc1ccc(cc1)OC)/c2ccc(cc2)Cl KM06123 c1cc(ccc1S(=O)(=O)N=S2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C#N)Cl KM06181 c1ccc(cc1)NC(=O)N2CCN(CC2)c3c(nccn3)C#N KM09017 CC(=O)n1ccc(n1)c2ccc(cc2)C#Cc3ccccc3 KM09008 c1cc2c(cc1Br)c(cc(n2)C(F)(F)F)O KM07368 Cn1c(c(nc1Oc2ccc(cc2Cl)Cl)C#N)C#N KM07472 Cc1c(c(nc(n1)C)NCc2ccccc2)Oc3ccc(cc3Cl)Cl SPB05824 Cn1c(cnc1SCc2ccc(cc2)Cl)C(=O)N/N=C/c3ccccc3Cl KM06124 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)/C=C(/C#N)\S(=O)(=O)c4ccccn4 KM08993 CC(=O)c1ccc(s1)C#CCOC(=O)Nc2ccc(cc2)OC(F)(F)F KM08997 Cc1ccccc1NC(=S)NCc2cccnc2 DSHS01294 Cc1c2c(n(n1)c3ccccc3)OC(=C(C2c4ccc(cc4)F)C#N)N BTB15009 Cc1ccc(cc1)NC(=S)N(CCC#N)CCc2ccccn2 DSHS01295 CC(C)CC(C(=O)OC)NS(=O)(=O)c1ccc(s1)c2nnc(n2C)SC KM04497 CNC(=S)NNC(=O)CSc1cccs1 KM04500 c1ccc(c(c1)C(F)(F)F)Oc2cc(nc3c2c(cc(c3)Cl)Cl)C(F)(F)F KM07480 COCCCn1c(nnc1S)c2ccc(cc2)C(F)(F)F SPB01426 c1ccc(cc1)S(=O)(=O)n2ccc(n2)c3ccc4c(c3)CCO4 KM06195 c1c(c(sc1S(=O)(=O)N)N2CCOCC2)[N+](=O)[O-] KM08942 c1ccc(cc1)S(=O)(=O)CCSc2c(cccn2)C(=O)Nc3ccc(cc3Cl)Cl KM06154 c1cc(ccc1NC(=O)CSc2c(c(cc(c2Cl)Cl)Cl)Cl)Cl KM08814 c1c(cc(cc1Cl)Cl)OCC#N SPB01308 C1CC23CC4=NNC(=O)C41CC2=NNC3=O BTB14985 Cc1c(cccc1Cl)NC(=S)NCc2cccnc2 DSHS01289 CC12CC3(CC(C1)(CC(C2)(C3)CCO)C)C BTB14993 Cc1cccc(c1NC(=S)NCc2cccnc2)C DSHS01292 Cn1c(cnc1SCc2ccc(cc2)Cl)C(=O)N/N=C/c3cccs3 KM06129 CCCCSc1c2c(c(s1)C(=O)OCC)CCCC2=O KM03285 CCOC(=O)c1c2c(c(s1)SC(C)C)C(=O)CCC2 KM03286 CN(C)c1c(c(c(c(c1Cl)Cl)Cl)Cl)Cl BTB15017 COC(=O)C1=C(CSC1)Nc2ccc(cc2)O KM04507 Cc1cc(c2ccc(nc2n1)N)O KM03366 CN1CCN(CC1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM09013 Cc1cc(ccc1NC(=S)N2CCC(CC2)NC(=O)C)Cl BTB01007 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=S)Nc2ccc(cc2)Cl KM09023 Cc1c2c3c(cnc2n(n1)C)c(=O)n(n3C)Cc4ccccc4Cl KM08906 Cn1c2c3cccc(c3nc(c2c(=O)n1Cc4ccccc4)SC)Cl KM08963 CCOC(=O)c1c[nH]c(n1)S(=O)(=O)CC KM06185 c1ccc(cc1)S(=O)(=O)CCSc2c(cccn2)C(=O)O KM06149 c1cc(cc(c1)[N+](=O)[O-])NC(=O)C23CC4CC(C2)CC(C4)C3 BTB15010 Cc1ccc(cc1)S(=O)(=O)NC(=O)Oc2ccc(cc2)Oc3ccc(cn3)C(F)(F)F SEW06392 CO/N=C/1\CCCc2c1c(sc2C(=O)NN)SC KM04492 COc1cccc(c1)NC(=S)N=S(=O)(C)c2ccccc2 KM04501 c1cc(sc1)/C=N/NC(=O)c2cc(=O)nc3n2ccs3 KM04503 c1cc(cc(c1)[N+](=O)[O-])C(=O)CC2(c3cc(ccc3N(C2=O)CN4CCOCC4)Br)O BTB02025 CCOC(=O)c1c2c(c(s1)SCc3ccc(cc3)Cl)C(=O)CC(C2)(C)C KM03297 c1cc(c(cc1Cl)C2CCCCC2)Oc3ccc(cn3)NC(=O)C4CC4C(=O)O BTB09404 c1ccc(cc1)c2nnc(o2)c3ccncc3 DP01996 Cc1c(sc2c1C(=O)/C(=N\Nc3cccc(c3)C(F)(F)F)/S(=O)(=O)N2C)C KM04354 CS(=NS(=O)(=O)c1ccc(cc1)OC(F)(F)F)(=O)c2ccccc2 KM04441 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl KM08933 c1c(c(sc1S(=O)(=O)N)N2CCNCC2)[N+](=O)[O-] KM08944 CC(=O)c1ccc(cc1)C#Cc2ccccc2 KM08946 CN(C)/C=C/C(=O)c1ccc(cc1)C#Cc2ccccc2 KM08947 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)SCC(=O)Nc4ccc(cc4)OC SPB07950 C=CCSc1nnc(n1c2ccc(cc2)OCc3ccccc3)c4ccco4 SPB07939 Cc1csc2c1c(c(s2)c3ccnc(n3)SCC(=O)NC(C)C)C KM04411 COC(=O)CSC(=O)NC(=O)c1ccccc1Oc2ccc(cc2Cl)Cl CD09005 Cc1ccc(cc1)CC2=NC(=O)/C(=C/C(=O)OC)/S2 BTB05071 c1cc2c(cc1c3ccnc(n3)S)OCCO2 FM00176 c1ccc(cc1)c2ncc(s2)C(=O)c3ccc(cc3)Cl BTB04699 c1ccc(cc1)C(=O)/C(=C/c2cc(cs2)Br)/C#N CD09047 Cc1c(c(c([nH]1)C)C(=O)OC)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM08863 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)C(F)(F)F)C(F)(F)F KM09135 COc1ccc(cc1)CC2=NC(=O)/C(=C/C(=O)OC)/S2 BTB05072 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(nccn3)C#N KM09045 c1cc(ccc1F)S(=O)(=O)N2CCN(CC2)c3c(nccn3)C#N KM09047 CS(=NC(=O)Nc1ccc(cc1)OC(F)(F)F)(=O)c2ccccc2 KM04380 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3cc(ccc3Cl)Cl RH00742 c1cc(sc1)CNC(=O)C23CC4CC(C2)CC(C4)C3 CD09028 CC1(OC(=O)C(=C2CCCCCN2)C(=O)O1)C CD10642 c1ccc(c(c1)C(=O)NC(=O)Nc2cc3cc(ccc3oc2=O)[N+](=O)[O-])Cl BTB03417 c1cc(cnc1)C(=N)NS(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3)[N+](=O)[O-])Cl BTB04670 c1cc(ccc1Sc2ccc(cn2)[N+](=O)[O-])Cl BTB07158 c1cnccc1CCNC(=O)C(Cl)Cl BTB03465 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CCCCO RH00930 CNC(=O)NNc1nccc(n1)c2cccnc2 MWP01008 Cc1c2ccccc2sc1CC(=O)Nc3ccccc3C(F)(F)F MWP00212 COC(=O)c1cccc(c1F)C(=O)OC CD10531 c1ccc(cc1)C(=O)O/N=C(/CC2CC2(Cl)Cl)\N CD10677 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCCCCNC2=O CD11519 c1ccc(cc1)C2=CCN(CC2)CCCCN3C(=O)c4cccc5c4c(ccc5)C3=O RH00936 c1ccc(cc1)c2c(n(nn2)c3ccc(cc3F)F)CSCC(=O)Nc4ccc(cc4)Cl CD08739 c1cc2c(cc1[N+](=O)[O-])cc(c(=O)o2)NC(=O)c3ccc(cc3Cl)Cl BTB03412 COc1ccccc1N2CCN(CC2)C(=O)/C=C/c3ccc(c(c3)OC4CCCC4)OC BTB13413 c1c2c(cc(c1Cl)Cl)n(cn2)CCCCO SPB07625 Cc1c2cc(ccc2sc1C(=O)CC#N)Cl MWP00552 c1ccc(cc1)CN2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)F KM08981 c1ccc(cc1)C#Cc2ccc(cc2)c3ccn[nH]3 KM08948 c1cc(ccc1N2C(=O)C3N(C2=S)CCS3)Cl KM08953 c1cc(cnc1)c2ccnc(n2)SCC3=NN(C(=O)C3)c4ccc(cc4)Cl MWP01044 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)c3ccccc3O CD08789 Cc1cc(cc2c1C(=O)/C(=C\c3ccccc3O)/S2)Cl CD09056 c1ccc2c(c1)cc(o2)C(=O)O CC06601 CCOC(=O)c1csc(n1)N/N=C/2\CCCc3c2cccc3 FM00302 CCOC(=O)c1csc(n1)N/N=C/2\CCc3c2cccc3 FM00304 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3cc(c(cc3C)Cl)C RH00744 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3cccc(c3)C(F)(F)F RH00747 Cc1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2)Oc3c(cncc3Cl)Cl)\N SPB07107 CN(C)/C=C/C(=O)c1ccsc1 KM04514 c1ccn(c1)c2ccsc2C(=O)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD08797 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)Oc3ccc(cc3)Cl KM04513 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)/C=C(/C#N)\S(=O)(=O)c4cccs4 KM09001 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)Nc2cccc(c2)[N+](=O)[O-] KM03246 c1c(sc(n1)Sc2nnc(s2)SCC3CC3)[N+](=O)[O-] SPB07212 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3nnc(s3)NC(=O)c4ccccc4F RH00783 Cn1cc(c(n1)c2cccc(c2)NC(=O)Nc3ccc(cc3)OC(F)(F)F)Br KM04515 CSc1c(c(n[nH]1)NS(=O)(=O)c2ccccc2Cl)c3ccccn3 PD00200 COC(=O)c1ccccc1SC(CC(=O)c2ccccc2)c3ccc(cc3)F PD00283 CCOC(=O)Cc1cc(=O)n2c([nH]1)cc(n2)C(C)(C)C KM09502 c1ccc(cc1)C(=O)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F SPB06954 c1cc(cc(c1)F)C(=O)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F SPB06955 c1cc(ccc1C#N)C(=O)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F SPB06956 CSc1nnc(s1)Sc2ncc(s2)[N+](=O)[O-] SPB07211 Cc1c(sc(n1)C(=O)Nc2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)Cl SEW04642 Cc1c(sc(n1)C(=O)Nc2ccc(cc2)OC)C(=O)Nc3ccc(cc3)OC SEW04644 c1cc(ccc1NC(=O)NC(=O)C23CC4CC(C2)CC(C4)C3)Cl CD09060 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2ccc(s2)C#CCC3CCCCC3 KM08967 CCOC(=O)CSc1c2c(c(s1)C(=O)OCC)CCCC2=O KM03289 CCOC(=O)c1csc(n1)CS(=O)(=O)Cc2ccco2 KM03255 c1cc(oc1)CS(=O)(=O)Cc2nc(cs2)C(=O)NN KM03257 CCOC(=O)c1csc(n1)N/N=C/2\CCCc3c2ccc(c3)OC FM00295 Cc1c(nns1)C(=O)Oc2ccccc2c3nnco3 SEW04581 c1cc(cc(c1)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl)C(F)(F)F SEW04768 c1ccc(cc1)C#Cc2ccc(cc2)c3ccn(n3)S(=O)(=O)c4ccccc4 KM08988 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(nccn3)C#N KM09046 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4cccs4 KM09067 COc1ccc(cc1OC2CCCC2)/C(=N/OC(=O)c3ccccc3)/N KM09585 c1cc(sc1)c2nc(sn2)Sc3nnc(n3c4ccc(cc4)Cl)O SPB07008 c1cc(sc1)c2nc(sn2)Sc3[nH]c(nn3)c4ccc(cc4)Cl SPB07013 Cc1ccc(cc1)N2CCN(CC2)CCCCCC(=O)O RH00941 CC(C)(C)S(=O)(=O)C/C(=N/OC(=O)c1cc(oc1C(F)(F)F)c2ccc(cc2)Cl)/N SEW04774 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)NNC(=O)c4ccc(cc4)Cl KM09094 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)NNC(=O)c4cccs4 KM09097 CCOC(=O)NC(=S)Nc1cccc(n1)C MH00409 CCOC(=O)c1c2c(c(s1)SCc3c(cccc3Cl)Cl)C(=O)CC(C2)(C)C KM03298 CCOC(=O)c1c2c(c(s1)SCc3c(cccc3Cl)F)C(=O)CC(C2)(C)C KM03302 c1cc(c(c(c1)Cl)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F)Cl SPB06951 c1ccc(c(c1)NC(=O)CSc2nnc(s2)c3ccc(cn3)C(F)(F)F)Cl SPB06946 CCOC(=O)Cc1cc(=O)n2c([nH]1)cc(n2)c3ccccc3 KM09464 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)O/N=C(/c3ccc(cc3)Cl)\N)Cl SEW04772 Cc1ccc(cc1NC(C#N)c2ccccc2)Cl S12558 CC(C)(C)c1cc2nc(cc(n2n1)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl)C(F)(F)F KM09123 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)Cc3nc(no3)c4cnccn4 KM09232 c1cc(ccc1C2c3ccsc3CCN2C(=O)Nc4ccc(cc4)Cl)Cl SEW01025 CN(C)/C=C/C(=O)c1cc(sc1Cl)Cl CD09177 Cc1cc(no1)NC(=O)CC#N CD09191 Cc1c(snn1)C(=O)N/N=C/c2ccccc2Cl CD09187 CCCCc1ccc(cc1)NC(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl KM06245 c1cc(ncc1C(F)(F)F)c2nnc(s2)SCC(=O)N SPB06978 Cc1c(c(no1)c2c(cccc2Cl)F)NC(=O)N(C)c3c4c(nn3C)CCCC4 BTB07102 CC(C)(C)c1csc(n1)Cc2ccc(cc2)c3csnn3 SEW01317 c1ccc(cc1)C(c2ccccc2)N3CC(C3)OC(=O)Nc4ccccc4 KM08868 c1ccc(cc1)C(c2ccccc2)N3CC(C3)OC(=O)Nc4ccc(cc4)Cl KM08869 CCc1c(nc2c(ccc(c2n1)OC)OC)CC BTB05245 c1c(cc(c(c1[N+](=O)[O-])N2CC3CCC(C2)CC3)[N+](=O)[O-])C(F)(F)F BTB02570 Cc1ccc(cc1)Sc2ccc(cn2)[N+](=O)[O-] BTB07159 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)NNC(=O)Nc4cc(cc(c4)Cl)Cl KM08920 COc1ccc(cc1)/C=N/NC(=O)CSC2CN(C2)C(c3ccccc3)c4ccccc4 KM09065 c1cc(c(nc1)SCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)C(=O)Sc3ccc(cc3Cl)Cl KM06255 CSc1ccc(cc1)Oc2ccc(cn2)[N+](=O)[O-] KM06261 c1cc(sc1)C(=O)/C(=C/c2cc(cs2)Br)/C#N CD09048 c1cc(ccc1NC(=O)C23CC4CC(C2)CC(C4)C3)F CD09044 CCOC(=O)Cc1cc(=O)n2c([nH]1)cc(n2)C KM09487 c1ccc(cc1)C(=O)C2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW04329 CS(=O)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F KM06265 Cc1c(c(c(c(c1C)C)C#CCO)C)C CD08965 Cc1c(c(on1)C)S(=O)(=O)N2CCC(CC2)C(=O)c3ccccc3 SEW04331 Cc1ccc(n1CCN2CCN(CC2)C(=O)c3ccc(cc3)Cl)C SEW04385 c1cc(ccc1c2[nH]c3ccc(cc3n2)N)c4[nH]c5ccc(cc5n4)N SPB07727 Cc1c(c(nc(c1C#N)SCc2c(cccc2Cl)F)C)Cc3c(cccc3Cl)F CD09503 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)CS(=O)(=O)c3ccc(cc3)Cl SEW04354 c1cc(c(cc1C(F)(F)F)Cl)NS(=O)(=O)c2cc(ccc2OCC(F)(F)F)C(F)(F)F SEW04487 c1ccc(cc1)N2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)F KM08982 CC(=O)c1ccc(s1)C#CCOC(=O)Nc2ccc(cc2)Cl KM08984 CNC(=O)NNC(=O)c1csc(n1)Cc2ccsc2 MWP00378 c1ccc(cc1)c2cc(sc2C(F)(F)F)/C=C/C(=O)c3ccc(cc3)Cl SEW03689 c1ccc(cc1)c2cc(sc2C(F)(F)F)/C=C/C(=O)c3cccs3 SEW03693 Cc1cccc(c1n2c(n[nH]c2=S)C3CC4CCC3O4)C RDR03506 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=S)NCc3ccccc3 RH00588 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=S)NC(C)c3ccccc3 RH00594 c1cc(ccc1c2csnn2)/C(=N/OC(=O)c3csnn3)/N SEW01061 Cc1nc(cs1)c2nnc(n2CCCOC)S SPB02439 COc1ccc(cc1)/C=N/NC(=O)CSCC(=O)Nc2ccccc2 KM09003 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)Sc3ncc(s3)[N+](=O)[O-] SPB07213 c1ccc(cc1)SC(C(=O)NCCNc2c(cc(cn2)Cl)C(F)(F)F)(F)F RDR03667 Cc1ccc(cc1)/C(=C/2\C=C(/C(=N/O)/C=C2Cl)Br)/C#N JA00164 COc1ccc(cc1OC2CCCC2)NC(=O)Nc3cccc(c3)C(F)(F)F KM09605 COc1ccc(cc1OC2CCCC2)C(=O)NC(=O)Nc3ccc(cc3)Cl KM09606 CCCCCCNC(=S)NNC(=O)COc1ccc(c2c1CCC2)C RH00592 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=S)NC3CCCCC3 RH00593 Cn1c(nnc1S)CSc2cccs2 KM04509 CCOC(=O)c1c(c(c(s1)SCc2ccccc2)S(=O)(=O)C(C)C)N KM03290 c1ccc2c(c1)nc(o2)SCCC(=O)N3CCc4c3ccc(c4)[N+](=O)[O-] RH00461 CCc1cc(c(c(c1)CC)NC(=S)Nc2ccc(cc2Cl)C)CC BTB02079 c1cc2c(cc1[N+](=O)[O-])CCN2C(=O)CCSc3cc(ccc3Cl)Cl RH00460 COc1ccc(cc1OC2CCCC2)C(=O)NC(=O)Nc3ccccc3 KM09607 COc1ccc(cc1OC2CCCC2)c3nc(on3)c4cccs4 KM09630 CSc1ccc(cc1c2c(c[nH]n2)Br)[N+](=O)[O-] KM03292 COc1ccc(cc1OC2CCCC2)NC(=O)Nc3cc(cc(c3)F)F KM09600 COc1ccc(cc1)NC(=O)NC(=O)c2ccc(c(c2)OC3CCCC3)OC KM09608 c1ccc(cc1)Cn2c(nnn2)c3cc(cc(c3)Cl)Cl GK02987 CCCCCCCCCCCC(=O)c1ccccc1 CD08624 COc1ccc(cc1OC2CCCC2)c3nc(on3)c4ccc(cc4)Cl KM09631 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3cc(ccc3OC)OC RH00743 CCOC(=O)C1=C(OCC1=O)Nc2ccccc2 KM07656 CCOC(=O)C1=C(OCC1=O)Nc2ccc(cc2)OC KM08751 CC1=N/C(=C(\C#N)/C(=O)C)/SC1 CD09244 Cc1ccc(cc1)C(=O)OCc2ccccc2Sc3cccc4c3c(ccc4)C(=O)NC BTB14930 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/OC(=O)c3ccc(cc3)Cl KM04379 COc1ccc(cc1OC2CCCC2)C(=O)NC(=O)Nc3cccc(c3)C(F)(F)F KM09609 COc1ccc(cc1OC2CCCC2)c3nc(on3)c4ccccc4 KM09621 CSc1c(c(nc2c1c(c(s2)C(=O)c3ccc(c(c3)Cl)Cl)N)N)C#N RH00575 CN1c2ccccc2C(=O)C(=C3SCCCS3)S1(=O)=O KM08648 Cc1c(ccc2c1cccc2)CC#N NRB05223 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NC(=O)NC CD10049 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NC(=O)Nc3ccccc3 CD10050 CCOC(=O)c1cc2c(c(sc2nc1C(F)(F)F)C(=O)OCC)NC(=O)c3ccc(cc3)Cl SPB07268 CCOC(=O)c1cc2c(c(sc2nc1C(F)(F)F)C(=O)OCC)NC(=O)C SPB07269 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC(=O)C34CC5CC(C3)CC(C5)C4 CD09057 Cc1cc(cc2c1C(=O)/C(=C\c3cc(cs3)Br)/S2)Cl CD09064 c1ccc(cc1)c2csc(n2)NN=C3C4CC5CC(C4)CC3C5 FM00228 COc1ccc\2c(c1)CCC/C2=N\N=C(/N)\SC FM00243 Cc1c(snn1)c2nc(cs2)C(=O)C SPB03839 CCOC(=O)c1cc2c(c(sc2nc1C(F)(F)F)C(=O)OCC)NC(=O)c3cccc(c3)C(F)(F)F SPB07271 COc1ccc(c(c1)OC)NC(=O)Nc2ccc(c(c2)OC3CCCC3)OC KM09604 COc1ccc(cc1OC2CCCC2)/C(=N/OC(=O)c3ccc(cc3)Cl)/N KM09617 CNC(=S)NNC(=O)c1csc(n1)c2cccnc2 MWP00426 c1cc(c(nc1)SC/C(=N/O)/N)C(F)(F)F SPB03897 c1ccc2c(c1)c(=O)nc([nH]2)N BTB05782 Cc1cc(cc(c1OC(=O)Nc2ccc(cc2)Cl)C)c3c4ccccc4c(=O)n(n3)C BTB08291 Cc1ccc2c(c1)CCCN2CCn3c(=O)c4cc(ccc4[nH]c3=O)C P00168 Cc1cc2c3c(c1)c(c(c(=O)n3CCC2)c4ccccc4)OC(=O)c5cc(cc(c5)C(F)(F)F)C(F)(F)F RH00706 Cc1cc(c(c(c1)C)C(=O)Oc2c3cc(cc4c3n(c(=O)c2c5ccccc5)CCC4)C)C RH00708 Cc1ccc2c(c1)c(cs2)CC#N MWP00140 Cc1c[nH]nc1c2ccccc2 CD09683 c1cc(ccc1c2c[nH]c(=S)[nH]2)Br.Cl FM00285 c1cc(ccc1c2cc(c(o2)C(F)(F)F)c3nc(no3)c4ccc(cc4)Cl)Cl SEW04787 c1ccc\2c(c1)CCC/C2=N\Nc3nc(cs3)C(=O)NN FM00306 c1cc(cc(c1)C(F)(F)F)c2nc(on2)c3cc(oc3C(F)(F)F)c4ccc(cc4)Cl SEW04790 c1ccc(c(c1)C(=O)NNC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F)Cl KM09386 CCOC(=O)c1csc(n1)c2cccnc2 MWP00332 CC(=O)c1ccc(o1)c2ccc(cc2F)F CD10801 COc1cccc(c1SC)OC CD11814 c1ccc(cc1)N2C(=O)CC(=N2)CS(=O)(=O)c3ccc(cn3)C(F)(F)F BTB08007 COc1ccc(c(c1)[N+](=O)[O-])N BTB07533 c1ccc(cc1)NC(=O)O/N=C/c2ccc(o2)c3ccc(cc3F)F CD10915 c1ccc(cc1)c2cc3ccccc3n2CCCCO SPB07631 c1ccc(cc1)c2nc3ccccc3n2CCCCO SPB07628 Cc1cccc(c1F)C(=O)O CD10965 CSc1c(c(n[nH]1)NC(=O)c2cccs2)c3ccccn3 PD00192 c1cc(c(c(c1)C(=O)N2CCCCC2)F)C(=O)N3CCCCC3 CD10534 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3c(cccc3C#N)C#N CD10977 Cc1c(cnn1c2cccc(c2C#N)Cl)C(=O)C CD09783 c1cc(c(cc1C(F)(F)F)N)Oc2ccc(cc2Cl)Cl BTB02738 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3nnc(s3)NC(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F RH00782 c1ccc(c(c1)c2nnco2)OC(=O)c3ccc(cc3)Cl SEW04580 CNC(=O)n1c(ccn1)c2ccc(o2)c3ccc(cc3F)F CD10932 CCOC(=O)c1cc2c(c(sc2nc1C(F)(F)F)C(=O)OCC)NC(=O)c3ccc(cc3)OC SPB07270 c1cc(cnc1)c2nc(cs2)CC(=O)NNC(=O)c3ccc(cc3)C(F)(F)F MWP00495 c1ccc(c(c1)c2nnco2)OC(=O)c3ccc(cc3)C(F)(F)F SEW04613 Cc1c(sc(n1)C(=O)Nc2ccccc2)C(=O)Nc3ccccc3 SEW04643 Cc1nc(c(s1)C(=O)Sc2cccc(c2)C(F)(F)F)C(F)(F)F SPB07344 c1cc(sc1)/C(=N/OC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl)/N SEW04773 CCOC(=O)C/C(=N\NC(=O)N)/C(F)(F)F CD09105 CSc1nc(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)N SPB06893 c1cc(sc1)c2nc(on2)c3cc(oc3C(F)(F)F)c4ccc(cc4)Cl SEW04788 c1ccc2c(c1)c(c[nH]2)C3=NCCCCN3 NH00203 CNC(=O)O/N=C(/Cc1csc2c1cccc2)\N MWP00249 COc1ccc(cc1OC2CCCC2)NC(=O)Nc3ccc(cc3)OC(F)(F)F KM09603 COc1ccc(cc1)NC(=O)c2cn(nc2SC)c3ccccc3 KM08836 c1cc(ccc1C(=O)NNC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F)Cl KM09378 c1cc(cc(c1)C(F)(F)F)/C(=N/OC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl)/N SEW04775 COc1ccc(cc1OC2CCCC2)/C(=N/OC(=O)Nc3ccccc3)/N KM09561 COc1ccc(cc1OC2CCCC2)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N KM09583 Cc1c(cn(n1)C(=O)Nc2ccccc2)c3ccc4c(c3)OCO4 CD09697 c1cc2c(cc1/N=C/c3cc(cc(c3O)Cl)Cl)COCO2 BTB01303 c1cc(cc(c1)[N+](=O)[O-])c2c[nH]c(=S)[nH]2.Cl FM00284 c1cc2c(cc1c3ccnc(n3)N)OCCO2 FM00174 Cc1cc(cc(n1)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C(F)(F)F CD10773 CCCNC(=O)NNC1=NCCc2c1cccc2 MWP01096 c1cc2c(cc1c3ccc(c(n3)S)C#N)OCCO2 FM00189 Cc1cc2c(cc1C)nc([nH]2)CCCO BTB05699 Cc1nnc(s1)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC BTB04908 c1cc(cnc1)C2CCCN2C(=S)Nc3ccc(cc3Cl)Cl CD10375 CCOC(=O)c1c(c(nc(n1)C)Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)C SPB07262 c1cc(cc(c1)C(F)(F)F)C(=O)N/N=C(/c2cnccn2)\N SPB07154 CCOC(=O)c1c(c(nc(n1)C)Sc2[nH]c(nn2)c3ccccc3)C SPB07260 Cc1ccc(cc1)SC(=O)c2c(nc(s2)C)C(F)(F)F SPB07343 CCOC(=O)c1c(c(nc(n1)C)Sc2[nH]c(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C SPB07263 Cc1nc(c(s1)C(=O)Sc2ccccc2)C(F)(F)F SPB07342 c1cc(ccc1C(=O)/C=C\2/NCCS2)Cl PD00060 Cc1nc(nc(n1)SC)N/C=C(\C#N)/S(=O)(=O)c2ccccc2Cl KM01059 c1c(c(=O)[nH]c(=O)[nH]1)[N+](=O)[O-] SB01199 CCOC(=O)c1cnc2c(ccc(c2c1Sc3ccc(cc3)Cl)F)F BTB08659 CCOC(=O)CNC(=O)c1cccnc1Oc2ccc(cc2)C BTB08772 CNC(=O)Nc1c(c(n[nH]1)SC)S(=O)(=O)c2ccc(cc2)Cl KM01270 COc1ccc(cc1OC2CCCC2)NC(=O)Nc3ccc(c(c3)OC4CCCC4)OC KM09599 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc(cc3)Cl)Cl SEW04769 c1cc(oc1)CNC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl SEW04770 Cc1nc(c(c(n1)SC)C#N)c2ccccc2 KM00817 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N3CCc4c(ccs4)C3C DFP00164 Cc1c(c(c(c(c1C)C)C(=O)c2ccc(cc2)NC(=O)c3c(c4ccccc4s3)Cl)C)C CD01924 CSc1c(c(nn1CC(=O)NN)c2cccs2)C#N KM00917 Cc1ccc(c(c1)C)NC(=S)Nc2cc(ccc2NC(=O)C)OC BTB00544 CC(C)(C)c1ccc(cc1)c2c(c(no2)SC)C#N KM00895 CC1c2ccsc2CCN1C(=O)NC(=O)c3ccccc3Cl DFP00204 CN1c2ccc(cc2C(=O)N(CC1=O)C3CCCCC3)Cl DP01023 c1cc(c(c(c1)C(=O)O)Br)C(=O)O NRB00681 CC(C)C1=CC(=O)n2c3ccccc3nc2C1(C)C CD01635 COc1ccc(c(c1)C(=O)c2ccc(cc2)N)OC CD02057 c1ccc(cc1)C2CC(=O)CC(=O)C2 CD11369 Cc1c(c(c(c(c1C)C)C(C)OC(C)c2c(c(c(c(c2C)C)C)C)C)C)C CD01808 Cc1cc(c2c(c1)CC(/C(=N/NC(=O)c3ccc(cc3)N(C)C)/C2=O)(C)C)C CD02787 c1cc(ccc1CS(=O)(=O)/C(=C/N2CCOCC2)/C#N)Cl KM01086 c1ccc(cc1)C2=N/C(=C/c3cccs3)/C(=O)O2 RB00124 Cc1cc(c2c(c1)CC(/C(=N/NC(=O)CCc3ccc(cc3)O)/C2=O)(C)C)C CD02776 CC(C)C(=O)C(C)(C)c1[nH]c2ccccc2n1 CD01628 CC(C)Sc1nnc(n1C)S BTB08587 c1ccc(cc1)c2cc3nc4c(c(n3n2)O)CN(C4=O)C5CCCCC5 KM00418 COc1ccc\2c(c1)CCC/C2=N\Nc3nc(cs3)C(=O)NN FM00305 Cc1cc(cc(c1OCC(=O)NNS(=O)(=O)c2ccc(cc2)F)C)c3c4ccccc4c(=O)n(n3)C BTB08310 CC(c1c(cccc1OC)OC)(C(OC)OC)O CD11875 COc1ccc(cc1OC2CCCC2)/C(=N/OC(=O)c3cccc(c3)C(F)(F)F)/N KM09618 CN(C)c1c(c(ncn1)Oc2cccc(c2)C(F)(F)F)[N+](=O)[O-] KM09431 CN(C)c1c(c(ncn1)Oc2ccc(cc2)Cl)[N+](=O)[O-] KM09432 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CCC(=O)O CD04187 CS(=O)(=O)c1csc(c1Cl)C(=O)Nc2ccccc2Cl KM02082 CC(C)(C)SCCN/C(=N\c1cccc(c1)F)/c2cccc(c2)Cl BTB06318 c1ccc(cc1)C(=O)NCc2c(cccc2Sc3ccc(cc3)Cl)F CD11863 CC(=O)c1ccc(cc1)Oc2c(cccc2C#N)C#N CD12000 CC(C)(C)c1ccc(cc1)c2c(c(no2)SC)C(=O)N KM01493 Cc1c(c(n(n1)c2ccccc2)O)C(=O)c3c(noc3C)C BTB07775 c1ccc(cc1)C(=O)c2c(nn(c2O)c3ccccc3)CS(=O)(=O)c4ccc(cn4)C(F)(F)F BTB08027 Cc1c(c(n(n1)C(C)(C)C)NC(=O)c2ccc(cc2)Cl)Br KM00094 CCOC(=O)c1c(nc(n1c2ccccc2OC)SC)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl SEW00088 c1ccc(cc1)C(C#N)NC(=S)Nc2cccc(c2)Cl KM00056 c1cc(ncc1[N+](=O)[O-])SC2=NCCS2 BTB07602 CCOC(=O)c1c(nc(n1Cc2cccs2)SC)NC(=O)c3cccs3 SEW00103 COc1cccc(c1)NC(=S)N RB00291 CCOC(=O)c1ccc(cc1)Nc2nc(cs2)c3cc(cc(c3OC)Cl)Cl RDR02045 Cc1c(c(no1)c2ccccc2)C(=O)NN CD02805 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(=S)Nc3nc(cs3)c4ccccc4 CD02479 CC(=O)c1ccccc1OCC(=O)O CD02486 COc1cccc(c1)Nc2c(c(c(s2)C(=O)c3cc4cc(ccc4o3)Cl)N)C#N DP02061 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NC(=S)Nc2ccc(cc2)F S06212 COc1ccc2c(c1)c(c(s2)C(=O)OC)Cl BTB10140 Cc1ccc(cc1[N+](=O)[O-])NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C BTB01419 C/C=C(\c1ccccc1)/C(=O)O NRB02306 c1cc(cc(c1)N2C(=O)CC(=N2)CS(=O)(=O)c3ccc(cn3)C(F)(F)F)C(F)(F)F BTB08036 C#Cc1cccc(c1)NC(=O)c2ccc(cc2)Cl S09462 CC1CN(CC(O1)C)C(=O)NC(=O)c2ccc(cc2)c3csnn3 SEW01138 CN(C)/C=C\1/C(=O)c2ccccc2CS1 CD11403 c1cc(c(c(c1/N=C\2/NCCS2)Cl)Cl)Cl S05573 CSC1=C(C(=O)NC2(S1)CCCCC2)C#N CD04066 Cc1cccc(c1Nc2nc3c(cc(c(c3s2)C)C)C)C RDR00014 CSc1nc(c(n1Cc2ccco2)C#N)NC(=O)c3ccc(o3)[N+](=O)[O-] SEW00123 c1ccc(c(c1)C2=NCCCN2)SCc3cc(cc4c3OCOC4)Cl.Cl CD03447 c1ccc(cc1)S(=O)(=O)/N=C(\NNC(=S)Nc2cccc(c2)F)/N3CCCC3 CD03650 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2C)NC(=O)C BTB01422 c1ccc(cc1)c2cc(=S)ss2 S04601 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2c(c(c(c(c2F)F)C(=O)O)F)F BTB08329 c1cc(c(c(c1)F)C(=O)NN)F CD04003 c1ccc(cc1)S(=O)(=O)c2cscc2NS(=O)(=O)c3ccccc3C(F)(F)F KM01808 c1cc(c(cc1n2c(nnc2S)CC#N)Cl)Cl CD02884 c1ccc(c(c1)/C=N/OCc2csc(n2)c3ccc(cc3)Cl)OC(F)(F)F SEW02220 CCCCOC(=O)c1ccc(s1)c2cc(nn2C)C(F)(F)F KM03036 CC(C)C(=O)Nc1c(n(c(n1)SC)Cc2ccco2)C#N SEW00124 CSc1nc(c(n1Cc2ccco2)C#N)NC(=O)c3ccc(cc3)Cl SEW00126 c1cc2c(cc1CCCC(=O)O)OCO2 BTB10687 c1ccc2c(c1)cccc2/C=N/NC(=S)Nc3ccccc3F RB00281 c1ccc2c(c1)c(=O)n(nn2)c3ccc(c(c3)Cl)Br RB00240 COC(=O)CNC(=O)C1c2ccccc2Oc3c1cccc3 BTB10310 Cc1cc(cc(c1)Br)Br CD03137 Cc1cc(nc2c1c(nn2C)C)n3c(cc(n3)C)C KM04104 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C(=N/OCc3ccc(o3)C(=O)OC)/N SEW01764 c1ccc(c(c1)N)SC(C[N+](=O)[O-])c2c(cccc2Cl)Cl S10370 c1cc(c(c(c1)Cl)C2CC(=O)N(C(=O)C2)c3cc(cc(c3)Cl)Cl)Cl S08428 c1cc(c(cc1Cl)Cl)C2CC(=O)N(C(=O)C2)c3cc(cc(c3)Cl)Cl S08434 CC1(Cc2csc(c2/C(=N/OC(=O)NC)/C1)SC)C KM03898 Cc1c(c(c2c(c1C)[nH]c(n2)/C(=C/c3ccc(cc3)Cl)/NC(=O)c4ccccc4)C)C S05721 c1cc(ccc1/C=N/NC(=O)c2cnco2)OC(F)(F)F SEW02548 c1cc(c(cc1F)F)N/N=C\2/CCSc3c2ccs3 SEW01796 CN1c2ccccc2-c3c(sc(c3S1(=O)=O)SCC#N)C#N KM03866 c1cc(ccc1c2ncc3c(n2)-c4ccsc4SC3)C(=O)N SEW01901 c1ccn(c1)CC2CCN(CC2)C(=O)c3ccc(c(c3)Cl)Cl CD03789 c1cc(ccc1n2c(nnn2)/C=C/N(CCO)CCO)Br BTB11588 c1cc(sc1)SC(=O)C2CC3CCC2C=C3 SEW02103 c1cc(c(c(c1)Cl)C2CC(=O)N(C(=O)C2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl S08443 Cc1cc(ccc1NC(=S)OC)Cl CD03990 CSc1c(c(on1)c2ccc(s2)S(=O)(=O)N3CCCCC3)C#N KM03970 Cc1ccc(cc1)/C=C(/c2[nH]c3c(c(c(c(c3n2)C)C)C)C)\NC(=O)c4ccccc4 S05725 Cc1c(cc2c(c1NC(=O)c3ccccc3Cl)C(CC2(C)C)(C)C)N4CCCC4 CD03951 Cc1cc(=O)n2c([nH]1)cc(n2)c3cc(c(s3)C(F)(F)F)c4ccccc4 SEW03413 CC1(Cc2c(c(sc2[N+](=O)[O-])SC)C(=O)C1)C KM03494 c1ccc(cc1)c2c(nnn2c3ccc(cc3)[N+](=O)[O-])C(=O)N4CCCCC4 CD04663 c1cc(cc(c1)Cl)Nc2c(c(c(s2)C(=O)c3cc4cc(ccc4o3)Cl)N)C#N DP02062 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)OCC)c3ccccc3)C KM05018 CC1(Cc2c(c(sc2c3ccn(n3)S(=O)(=O)c4ccc(c(c4)Cl)Cl)SC)C(=O)C1)C KM03426 CN(C)C(=O)Oc1cccc(c1)N SEW00299 CC1(Cc2c(c(sc2c3ccn(n3)C(=O)NC)SC)C(=O)C1)C KM03436 Cn1ccc(n1)c2cccc(c2)NC(=O)Nc3ccc(cc3)Cl KM03080 c1cc2c(cc1Cl)-c3c(cc(s3)C(=O)NN)CS2 SEW01689 CNC(=O)N(CCS(=O)(=O)c1ccc(cc1)Cl)Cc2cccs2 KM03779 Cc1cc(nc2c1c(nn2C)C)NNC(=O)NC KM04084 C1C2CC3CC1[C@H](C(C2)[C@H]3O)C(=O)O NRB01775 c1csc2c1cc(s2)C(=O)O SEW01633 c1cc(c(c(c1)Cl)/C=C/2\C(=O)NC(=S)N2)Cl S10180 c1cc(sc1)CCNC(=O)c2ccc(cc2)Cl S10251 c1cc(sc1)c2ccc(s2)/C=C/C(=O)N3CCOCC3 SEW02634 COc1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4ccccc4 BTB11250 Cc1c(c(c2c(c1C)[nH]c(n2)/C(=C/c3cc(c(c(c3)OC)OC)OC)/NC(=O)c4ccccc4)C)C S05720 COc1cccc(c1)Oc2ccccc2C(=O)O CD04050 c1cc2c(cc1Cl)-c3c(cno3)CS2(=O)=O SEW01877 CCOC(=O)/C(=C/c1cccn1c2cccc(c2)SC)/C#N CD04385 Cc1cc(cc(n1)Oc2ccc(cc2)c3ccnc(n3)N)C(F)(F)F SEW01841 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=C/C(=N/O)/N CD04728 CCc1c(c2ccccc2oc1=O)O BTB11213 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)/N=S/3\CCC4(C3)OCCO4 KM06233 Cc1cc(nc2c1c(nn2C)C)n3c(c(c(n3)C)Br)C KM04125 C/C(=C\c1ccc(o1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F)/[N+](=O)[O-] CD04334 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)S KM04540 c1ccn(c1)CC2CCN(CC2)C(=S)Nc3cccc(c3)Cl CD03790 c1cc(ccc1S(=O)(=O)Cc2nc(no2)/C=C/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl CD04853 c1ccn(c1)CC2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl CD03788 c1cc(cc(c1)S(=O)(=O)CCSc2c(cccn2)C(=O)NCc3cccs3)C(F)(F)F KM06287 CC(=O)c1c(c(c(s1)SCCS(=O)(=O)c2ccccc2)C#N)c3ccccc3 KM05464 c1cc(ccc1OCc2ccsc2CNS(=O)(=O)C(F)(F)F)Cl SEW02528 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(c(cc3Cl)Cl)C(F)(F)F CD04430 CSc1c(c(c(s1)C(=O)NCC2CC2)c3ccc(cc3)Cl)C#N KM01231 Cc1ccc(cc1)S(=O)(=O)OCC23CCC(CC2)(CC3)OS(=O)(=O)c4ccc(cc4)[N+](=O)[O-] NRB02199 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nc(cs3)c4cc(c(s4)C(F)(F)F)c5ccccc5 SEW03096 c1cc(ccc1c2csnn2)C(=O)O CC16401 c1ccc2c(c1)C(=O)N(C2=O)SSN3C(=O)c4ccccc4C3=O BTB11006 CS(=NC(=S)Nc1ccc(cc1)Br)(=O)c2ccccc2 KM04502 c1cc(ccc1Sc2c(cncc2Cl)Cl)Cl RF01292 Cc1c(c(no1)c2c(cccc2Cl)F)/C(=N/O)/N RF00760 CC(C)C12CC3CC(C1)CC(C3)(C2)Br NRB01922 c1ccc2c(c1)CSCC2=O CD04109 c1cc(c(c(c1)F)C#N)N2CCOCC2 CD05368 c1cc(sc1)CCNC(=O)c2cccs2 S10258 c1cc(sc1)CCNC(=O)c2ccc(cc2Cl)Cl S10261 COc1cc(c(cc1OC)[N+](=O)[O-])/C=C/[N+](=O)[O-] S10284 CC1(CC2=C(Cc3cc(ccc3O2)Br)C(=O)C1)C CD04620 Cc1c(c(no1)c2ccccc2)C(=O)NCCc3cccs3 S10260 c1ccc2c(c1)c(nc3n2nnc3C(=O)N4CCCC4)N CD05133 Cc1c(cn[nH]1)c2nnnn2c3ccc(cc3)OC BTB11253 c1ccc(cc1)c2c3c(sc2C(F)(F)F)sc(n3)N SEW03170 c1ccc2c(c1)CC(C2)C(=O)O KM06597 CS(=N/C=C(\C#N)/S(=O)(=O)c1ccc(cn1)C(F)(F)F)(=O)c2ccsc2 KM05869 c1ccc2c(c1)nc(s2)/C=N/OCc3ccc(cc3)Cl SEW03006 c1ccc2c(c1)OCC(O2)C(=O)Sc3cccs3 KM06645 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])/C=C/C#N CD05536 c1ccc(cc1)c2c3c(sc2C(F)(F)F)sc(n3)NC(=O)c4ccc(cc4)Cl SEW03226 Cc1cc(c(c(c1)C)S(=O)(=O)O)C.c1c(cnc(c1Cl)N2CCS(=N)CC2)C(F)(F)F KM06021 c1ccc(cc1)c2nc3c(o2)c4ccccc4[nH]c3=O BTB11086 c1ccc(cc1)C2C(=Nc3cc(cc(c3N2c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C(F)(F)F)C(F)(F)F)c5ccccc5 S11340 Cc1c(c(n(n1)Cc2nnc(n2C)S)C)[N+](=O)[O-] KM04186 CCOC(=O)c1c2c(c(s1)SC)-c3c(cnc(n3)SCC(=O)C(C)(C)C)CC2 KM04240 c1ccc(cc1)c2c(snn2)C(=O)N CD05540 COc1ccc(cc1)NCCC#N EN00151 c1ccc(cc1)CCSc2ccc3c(c2[N+](=O)[O-])nsn3 KM06793 C/C(=C\c1c(ccs1)OC)/[N+](=O)[O-] SEW02942 CSC(=NS(=O)(=O)c1ccc(c(c1)Cl)Cl)SC CD05550 c1cc(c(c(c1Cl)Cl)Cl)I SEW04070 c1ccc(c(c1)CNc2[nH]nc(n2)N)OC(F)(F)F SEW02235 c1ccc(cc1)c2c(snn2)/C(=N/O)/N CD05542 CCOC(=O)c1cnc2ccc(cn2c1=O)C(F)(F)F SEW02295 c1cc(sc1)c2[nH]c(nn2)S SPB00125 c1ccc(cc1)C(=O)CSc2[nH]c(nn2)C(F)(F)F SPB00207 COc1cc(cc(c1)NCN2C(=O)CCC2=O)C(F)(F)F CD04595 c1cc2c(cc1Cl)c(nc3n2nnc3C(=O)N)N CD06386 CC(C)NC(=O)Nc1nc2c(c(sc2s1)C(F)(F)F)c3ccccc3 SEW03225 Cc1cc(ccc1NCN2C(=O)CNC2=S)Cl S10232 CN1c2ccccc2/C(=N/Nc3cccc(c3)C(F)(F)F)/C1=O KM04493 c1ccc2c(c1)nnc3n2cnn3 BTB10859 c1ccc(cc1)Oc2c(nccn2)C#N KM06166 CC1=CS/C(=C(\C#N)/C(=O)c2ccccc2Cl)/N1c3ccccc3Cl RF02505 COc1cccc(c1)CNC2CS(=O)(=O)CC2O.Cl SEW03566 COC(=N)c1c(nccn1)SCc2ccc(cc2Cl)Cl KM06394 Cc1ncc(c(n1)CN(C)C)c2nnnn2c3ccccc3 BTB12043 Cn1c(nnc1S)CSCc2nc(cs2)c3ccc(cc3)Cl KM05912 CCC(=O)c1ccc(cc1O)OC(=O)C BTB12503 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCC(=O)NC(C)C KM04572 COc1ccc(cc1)C(=O)N=S(=O)(C)c2ccsc2 KM05754 CC1(Cc2c(cnc(n2)SCC(=O)c3ccc(cc3)Cl)C(=O)C1)C KM04710 CCOC(=O)c1c2c(sc1N)CCC2 NRB02041 CSc1c(c(n[nH]1)N)c2ccc(cc2)[N+](=O)[O-] EN00085 c1cc(ccc1OCCC(=O)O/N=C(/c2ccc(o2)[N+](=O)[O-])\N)F SEW01467 CCN(CC)c1ccc(cc1)NN=C2C(=O)N(C(=O)N(C2=O)C)C NRB02953 c1cc2c(c(c1)Cl)c(nc3n2nnc3C(=O)N)N CD07368 c1cc(sc1)CNC(=O)c2cc(ccc2O)Br CD06840 c1ccc(cc1)C(CNC(=O)c2ccc(cc2)C(F)(F)F)c3c[nH]c4c3cccc4 SEW04401 Cn1ccc(n1)c2nc3ccccc3s2 SEW02853 Cc1c(c(c(=O)n(c1c2ccccc2)c3ccccc3)C(=O)C)O NRB02899 c1ccc2c(c1)nc(s2)c3ccn(n3)C(=O)c4cccs4 SEW02855 c1ccc(cc1)c2c(csc2C(F)(F)F)NC(=O)c3ccc(s3)[N+](=O)[O-] SEW03209 CCOC(=O)CCc1c2c([nH]c1C(=O)OCC)CNC(=O)C2 NRB02790 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)Cl)/C(=O)N2c4cc(cc(c4)C(F)(F)F)C(F)(F)F S11513 c1ccc2c(c1)CC/C(=C\c3csc4c3cccc4)/C2=O S12897 C(CC(=O)O)C(CCC(=O)O)C(=O)O NRB02462 Cc1ccc(cc1)NC(=O)N=S2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C#N KM06191 c1ccc(cc1)S(=O)(=O)OC[C@H]2CC3CCC2C=C3 BTB12743 c1ccc(c(c1)C(F)(F)F)n2c(nnc2Sc3cc(ccn3)C(F)(F)F)O SPB03223 CCOC(=O)c1nc(no1)c2cccc(c2)n3cccc3 SPB01498 c1ccc(cc1)c2c(csc2C(F)(F)F)NC(=N)N3CCCCC3 SEW03480 Cn1c2ccccc2nc1N3C(=O)c4cccc5c4c(ccc5N(C)C)C3=O BTB11700 CCN(CC)c1c(c(nc(n1)c2ccc(cc2)Cl)N(CC)CC)Cl CD07166 Cn1c(nnc1SCc2ccc(cc2)Cl)Cn3cccc(c3=O)OC KM07215 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC(=O)c3c(cccc3F)F CD05888 Cc1csc(n1)Cn2c(=O)c3ccccc3c(n2)CC(=O)NNS(=O)(=O)c4ccccc4 KM07232 CC(=O)Nc1cccc(c1)OCCOc2cccc(c2)NC(=O)C BTB12341 CN(C)c1ccc2c3c1cccc3C(=O)N(C2=O)c4ccccc4 BTB11675 COCCCNC(=O)c1c2nc(c3cc(ccc3n2nn1)Cl)N CD06390 COCCCNC(=O)c1c2nc(c3c(n2nn1)cccc3Cl)N CD07371 CCOC(=O)c1cc(nn1C(=O)C)c2ccc(s2)Cl SPB05161 CC(C)(C)C(=O)OC12C=CC(O1)C3C2C(=O)N(C3=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F S12600 COc1ccc(cc1NC(=C2C(=O)c3ccccc3C2=O)C#N)Cl S12611 Cc1coc2cc(ccc2c1=O)[N+](=O)[O-] BTB12534 c1ccc(cc1)C(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl KM06042 CN(C)/C=C/C(=O)c1c(cccc1F)F CD07340 c1ccc(cc1)OCCCCC(=O)CCCCOc2ccccc2 NRB02433 CCOC(=O)c1cc(nn1C(=O)c2ccc(cc2)Cl)c3cccs3 SPB04184 CCCCOc1cc(nc2c1cc(cc2)CS(=O)(=O)c3nc4ccccc4s3)C(F)(F)F KM07525 CC1(NC(=O)C(=C(S1)SC)C#N)C CD07740 c1ccc(cc1)C/N=c/2\n(c(=O)ss2)Cc3ccccc3.Br NRB03114 CSc1c(c2nc(cc(n2n1)C(F)(F)F)C(F)(F)F)C(=O)NCC(=O)O KM07430 CC(C(c1cccc(c1)OC)c2c(n(c(=O)n(c2=O)C)C)N)[N+](=O)[O-] S13304 c1cc(ccc1C(=N)N)Cl.I CD07981 Cc1c(c(c(c(c1C)C)CN2CCOC(C2C)c3ccccc3)C)C CD00970 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2cc(ccc2OC)Br)N S13301 c1cc(ccc1C(=N)N)C(=O)N.Cl SB00616 CCOC(=O)c1cc(=O)n(c2c1c(=O)oc3c2cccc3)C NRB03953 c1cc(ccc1NC(=S)NC2CCCCC2)S(=O)(=O)N3CCCCC3 CD00893 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3ccc(cc3)OC(F)(F)F S13899 c1cc2c(cc1Br)C3(C(=O)N2)OCCO3 S13952 CC(=O)CSC(=S)N1CCSCC1 CD08205 CN(C)/C=N/S(=O)(=O)c1cc(ccc1OC)OC CD07548 c1cc(c(c(c1)Cl)OCC(CN)O)Cl CD07138 c1cc2c(cc1Cl)c(cs2)CN3C(=O)C=CC3=O S13356 Cc1c(nnn1c2cccc(c2)C#C)C(=O)C CD08025 CC1(COC(=N1)c2ccccc2COC(=O)c3ccc(cc3)C(C)(C)C)C S13773 Cc1ccc(cc1)c2cc([nH]n2)NC(=O)C3Cc4ccccc4C3 KM06998 c1ccc2c(c1)c(cc(n2)c3cccc(c3)N)C(=O)O NRB03638 CNc1c(c(ncn1)Oc2ccsc2C(=O)OC)[N+](=O)[O-] KM07927 c1cc(c(c(c1)Cl)CO/N=C(/CN2CCSCC2)\N)Cl CD08424 Cc1c(nnn1c2ccccc2Oc3ccc(cc3Cl)Cl)C(=O)O CD08437 CC(C)Oc1ccc(cc1)/C=N/CCNc2nccc(n2)C(F)(F)F AW00567 c1cc(ccc1c2nc(on2)CN/N=C/c3ccc(c(c3)O)O)Cl CD02968 C1CCC(C1)N2CNC(=S)NC2 ML00416 c1ccc(cc1)C(=O)NC23CC4CC(C2)CC(C4)C3 BTB15007 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4cc(cc(c4)Cl)Cl NH00470 Cc1cc(c(c(c1)CO)OC)CO BTB14913 c1cc(ccc1c2cc([nH]n2)C(F)(F)F)Br BTB14920 CCOc1ccsc1C(=O)Nc2cc(ccc2F)F GK02494 c1ccc(cc1)C/C(=N/O)/N S01215 c1cc(c(cc1)Oc2c(cc(cc2)Cl)Cl)c3nc(nc(n3)NC(=O)/C=C/c4sccc4)NC(=O)/C=C/c5sccc5 MBE00012 c1ccc2c(c1)C(=O)C(C(=O)N2)(F)Cl NRB04833 COc1ccc(cc1OC)C(=O)Nc2ccccc2Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00755 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(c(c3)F)F DSHS00814 c1cc(ccc1NC(=S)N2CCC=CC2)S(=O)(=O)N3CCCCC3 CD00833 CCCCCCCCOS(=O)(=O)c1cc(ccc1OC)OC NH00269 CCOC(=O)c1cnc(nc1C(F)(F)F)Sc2ccc(cc2)Cl GK02953 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccc(cc2)C(C)C GK02954 CCCCNC(=O)Nc1nc(nc(n1)NC(=O)NCCCC)c2ccccc2Oc3ccc(cc3Cl)Cl MBE00024 COc1cc(ccc1O)CC(C(=O)O)N RJC01251 c1cc(sc1)c2c(cnc(n2)c3ccncc3)C#N CD08036 c1cc(ccc1c2c(c3ccc(cc3o2)S(=O)(=O)N4CCCCC4)Cl)S(=O)(=O)N5CCCCC5 S12979 c1ccc(cc1)c2ccc(cc2)C3C4C(=NN3)C5CCN4CC5 DSHS00399 Cn1c2c(cnc(n2)c3ccccc3Cl)c(=O)n(c1=O)C S13820 c1c(csc1[N+](=O)[O-])C2N3C(OCC3(CO2)CO)c4cc(sc4)[N+](=O)[O-] S13239 C1C(C1(Cl)Cl)C(=O)N BTB12878 c1ccc(cc1)C(=O)CN2C(=O)c3ccccc3C2=O S00647 COC(=O)CCN1CCc2c1ccc(c2)/N=N/c3ccc(cc3)C#N JFD03382 CCOC(=O)c1c(c(c(s1)N)C#N)C JFD03385 CCCn1c(nnc1S)Cc2ccc(c(c2)Cl)Cl SPB07980 CC1=N/C(=C\c2cccs2)/C(=O)O1 SPB07994 CCOC(=O)NNC(=O)NCCCc1ccc2ccc3cccc4c3c2c1cc4 JFD03484 CC1=N/C(=C\c2ccccc2Br)/C(=O)O1 SPB07999 CC(=O)N/C(=C\c1ccc2ccccc2c1)/C(=O)O SPB07988 CCOC(=O)c1csc(n1)c2cc(cc(c2)Br)Br SEW05758 c1c(cc(cc1Br)Br)C(=O)NC(=O)N2CCOCC2 SEW05764 Cc1c(c(c(s1)NC(=O)C)C(=O)OC)[N+](=O)[O-] JFD03387 C/C(=N\Cc1cc(ccc1)C/N=C(/c2c(cccc2)O)\C)/c3c(cccc3)O S03762 COC(=O)c1c(ccs1)N2C(=O)C=CC2=O GK01179 CC(=O)c1ccc(cc1)Oc2ccc(c(n2)Oc3ccc(cc3)C(=O)C)[N+](=O)[O-] SEW05763 CCO/C(=N/c1ccc(cc1)OC(F)(F)F)/SCC(=O)C(C)(C)C S13614 c1ccc(c(c1)C2C(CCC(=O)N2C3CCCCC3)C(=O)O)Cl CD01076 c1ccc2c(c1)cc(o2)CC(=O)NCc3ccc(cc3)F S14513 c1ccc(cc1)c2csc(n2)N CD00472 Cc1c(c(no1)c2ccccc2)C(=O)O CC00501 Cc1ccc(c(c1)C)c2nnc(o2)c3ccncc3 DP01997 c1cc(ccc1S(=O)(=O)Nc2ccc(c(c2)F)F)Br DSHS00759 CN1C(=S)S/C(=N/OC(=O)c2ccc(cc2)Cl)/C(N1)c3ccccc3 MBE00210 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(C)(C)C#C DSHS00840 c1cc(c(cc1Cl)Cl)S(=O)(=O)N2CCN(CC2)c3c4ccsc4ncn3 GK02965 C1CCN(C1)/C(=N\O)/c2c(non2)N RJC01203 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK02952 Cc1ccc(cc1)N(C2CS(=O)(=O)C=C2)C(=O)c3cc(cc(c3)[N+](=O)[O-])[N+](=O)[O-] JFD03013 c1c(nc(nc1O)N)C(F)(F)F RJF00185 c1cc(c(cc1n2c(=O)[nH][nH]c2=S)Cl)Cl NH00306 c1ccc(cc1)Sc2c(nc3n2cccc3)c4ccc(cc4)Br JFD03014 Cc1ccccc1NC(=O)CC#N DP00170 CC(C)(C)C(=O)NC(=S)Nc1ccc(cc1)C(F)(F)F NH00480 c1cc2c(c(c1)[N+](=O)[O-])nc[nH]2 RJC00582 C1CCN(C1)c2nc(nc(n2)N)N RJF00288 Cc1cn(nc1O)Cc2ccccc2 XBX00058 CCCCCCCCCCCCCCOS(=O)(=O)c1cc(ccc1OC)OC NH00271 c1cc(oc1COCOCc2ccc(o2)C(=O)O)C(=O)O NH00375 c1ccc2c(c1)c(n[nH]c2=O)c3cc(cc(c3)Cl)Cl NH00466 c1cc(c(cc1Cl)Cl)NC(=S)N2CCCN(CC2)c3nccc(n3)C(F)(F)F AW00564 c1cc(ccc1NNC(=S)N)S(=O)(=O)N PD00389 CC1=N/C(=C\c2cc(cc(c2)F)F)/C(=O)O1 SPB08017 c1cc(cc(c1)[N+](=O)[O-])C(=O)NN BTB09282 c1cc(cc(c1)n2c(n[nH]c2=S)c3ccco3)C(F)(F)F ML00353 CCC12CC3CC(C1)(CC(C3)(C2)NC(=O)C)C(=O)O BTB15004 c1ccc(cc1)/C=C/C=C/2\c3ccccc3NC2=O CD00743 C/C(=N\NC(=O)N)/c1ccccc1OCC(=O)O CD02489 COc1ccc\2c(c1)CCC/C2=N\c3ccccc3C(F)(F)F JFD02876 c1ccc(cc1)CNC(=O)NCCCCCCNC(=O)NCc2ccccc2 JFD03439 c1ccc(cc1)c2c3ccc(cc3oc-4cc(=O)ccc24)O JFD03443 CCCC(C1C(=O)CC(CC1=O)(C)C)C2C(=O)CC(CC2=O)(C)C JFD03444 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccc(cc2)C GK02962 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC GK02964 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCc4cccc(c4)C(F)(F)F SPB07877 CC(C)N(CCC#N)CN1C(=O)c2ccccc2C1=O SW00047 c1cc(c(cc1Cc2nnc(o2)S)Cl)Cl SPB07982 CC(=O)OCc1cccc2c1c(ccc2)Sc3ccccc3C(=O)Nc4ccccc4 BTB14931 C/C(=N\NC(=S)NC1CC2CC1C=C2)/c3ccccc3OCC(=O)O CD02502 C1CC2CCCC(C1)(C2)C(=O)NN BTB14987 CC12CCCC(C1)(CCC2)C(=O)N BTB14988 c1ccn2c(c1)nc(c2Sc3ccc(cc3)[N+](=O)[O-])c4ccc(cc4)Br JFD03011 c1c(cc(c(c1C(F)(F)F)C(=O)N)C(F)(F)F)C(F)(F)F JFD03020 CCCCCCCCCCOS(=O)(=O)c1cc(ccc1OC)OC NH00267 CC1CC(CC(C1)(C)C)NC(=O)c2cc(c(c(c2)OC)OC)OC NS00114 CCCCCC(=O)Nc1nc-2c(s1)Cc3c2cccc3 RH01311 CCCNC(=S)NNC(=O)Cc1ccc(c(c1)Cl)Cl SPB07997 CC(=O)Nc1ccc(cc1)/C=C(/C(=O)O)\NC(=O)C SPB08014 COC(=O)C12CCC3(C(C1)(CCC24SCCS4)C(=O)OC)SCCS3 BTB14945 CCOC(=O)NC(=S)NC(=O)C(C)(C)C NH00483 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4ccc(c(c4)Cl)F NH00493 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)C)C JFD02936 CC(C)CC(C(=O)O)NC(=O)C(CCC(=O)N)NC(=O)CNC(=O)C(C(C)C)NC(=O)OCC1c2ccccc2-c3c1cccc3 JFD02944 COC(=O)/C(=C/c1ccc(c(c1)[N+](=O)[O-])N2CCCC2)/C#N RH01317 c1cc(ccc1CC(=O)NN)[N+](=O)[O-] RH01329 c1ccc(cc1)C(=O)NNC(=O)CSCc2cccc3c2cccc3 RH01590 Cc1nc(cs1)c2nc(cs2)C(=O)NN(S(=O)(=O)C)S(=O)(=O)C SPB07818 c1cc(ccc1NCCC#N)/N=N/c2ccc(cc2)Cl JFD03380 CC(C)(C)[C@H]1COC(=N1)CC2=N[C@H](CO2)C(C)(C)C JFD02840 CC(C)(C)OCC(C(=O)NC(Cc1ccccc1)C(=O)NC(CCC(=O)N)C(=O)NC(CCC(=O)OC(C)(C)C)C(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4 JFD02945 Cc1cc(c(c(c1S(=O)(=O)NC(=N)NCCCC(C(=O)NC(Cc2ccccc2)C(=O)O)NC(=O)C(CCC(=O)N)NC(=O)C(C(C)OC(C)(C)C)NC(=O)C(CCC(=O)OC(C)(C)C)NC(=O)C(C)NC(=O)OCC3c4ccccc4-c5c3cccc5)C)C)OC JFD02950 Cc1c(c(on1)C)c2nnc(o2)c3ccc(cc3)Cl SEW05986 Cc1c(c(on1)C)c2nnc(o2)c3ccc(cc3)C(F)(F)F SEW05987 Cc1c(c(on1)C)c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05989 c1cc(c(cc1[N+](=O)[O-])CO)N2CCOCC2 RH01303 C1CCc2c(c(nc(n2)N)C(F)(F)F)C1 BTB15062 Cc1cc(c(n1c2ccccc2)C)C(=O)Nc3ccc(cc3)Cl SP00296 Cc1cc(c(n1Cc2cccs2)C)C(=O)Nc3ccc(cc3)Cl SP00298 Cc1ccc(cc1)NC(=O)C23CC4CC(C2)CC(C4)C3 BTB15011 C1CC2CC1C(C2C(=O)O)C(=O)O BTB15020 c1c(c(cc(c1Cl)Cl)Cl)Cl BTB15025 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2nnc(s2)SCC(=O)Nc3ccc4c(c3)OCO4 RH01565 c1c(cc(cc1C(F)(F)F)C(F)(F)F)Cc2[nH]nnn2 SPB07972 Cc1ccc(cc1)C(=O)CC(c2ccsc2)Sc3ccc4ccccc4c3 S11229 CC(=O)c1cc(no1)c2c(cccc2Cl)Cl SPB07990 Cc1c(c[nH]n1)c2nc(no2)c3ccc(cc3)Cl CD09798 c1ccc(cc1)c2c(cn(n2)c3ccccc3)C4N(C(=O)CS4)CCO BTB15006 c1cnc(cc1C(=O)O)c2cc(ccn2)C(=O)O JFD02898 Cc1c(c(on1)C)S(=O)(=O)NCc2cccs2 SEW05836 CC(C)(C)c1cc(n(n1)c2ccc(cc2)[N+](=O)[O-])C(C)(C)C SEW05841 CC(C)(C)C(=O)NC(=S)Nc1cccc(c1)C(F)(F)F NH00482 c1ccnc(c1)CNC(=S)Nc2cccc(c2)F NH00501 CCC(=O)N/N=C(\C)/c1ccc(cc1)Oc2ccccc2 RH01251 c1cc(ccc1c2cc(nc(n2)N)C(F)(F)F)Br BTB14922 c1ccc(cc1)c2cc(nc(n2)N)C(F)(F)F BTB14923 c1ccc(cc1)Cn2cc(c3c2ccc(c3)[N+](=O)[O-])CO RH01230 CC(=O)NC12CC3(CC(C1)(CC(C3)(C2)C)C)C BTB14972 COC(=O)C12CCCC(C1)(CCC2)C(=O)O BTB14975 c1cc(sc1)C(=O)Nc2ccc(cc2OC(F)(F)F)Cl SEW05844 COc1ccc2c(c1)oc(c(c2=O)Oc3ccc(cc3)C(=O)OC)C(F)(F)F BTB14911 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCC(=O)c4ccc(cc4)C(F)(F)F SPB07865 Cc1ccc(cc1)NC(=O)Nc2cc(cc(c2)Cl)Cl SEW05821 c1cc(cc(c1)S(=O)(=O)N2CCCCC2)C(F)(F)F GK02824 CN1CCN(CC1)c2ccccc2/C=N\Nc3cc(ccc3Cl)Cl SEW05753 Cc1c(c(n[nH]1)c2ccc(cc2O)O)Oc3ccc(cc3)F BTB14912 c1cc\2c(cc1)/C(=N/O)/C/C2=N\O JFD03516 Cc1cc(cc(n1)n2c(c(cn2)/C(=N/OC(=O)c3ccccc3)/C)C)C(F)(F)F CD11716 c1ccn(c1)CC2CCCN(C2)S(=O)(=O)c3cc(sc3Cl)Cl CD09949 CC1(C\2CCC1(C(=O)/C2=C\c3ccccc3)C)C BTB14917 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccc(cc2OC)OC GK02959 CC(CCc1ccccc1)NC(=O)C JFD03491 c1cc(nc(c1)CSc2ccc(c(c2)Cl)Cl)CSc3ccc(c(c3)Cl)Cl JFD02905 CC(=O)Oc1ccc(cc1)CC2C(=O)NC(=O)S2 JFD02851 c1ccc(cc1)[C@@H]2[C@@H](OC(=N2)CC3=N[C@@H]([C@@H](O3)c4ccccc4)c5ccccc5)c6ccccc6 JFD02847 c1cc(ccc1/C=N/CCNc2nccc(n2)C(F)(F)F)OC(F)(F)F AW00575 CN1CCN(CC1)c2ccccc2/C=N\Nc3c(cc(cn3)C(F)(F)F)Cl SEW05771 COc1ccc(cc1)c2nc3ccccc3s2 JFD02885 COC(=O)/C(=C/c1ccc(c(c1)[N+](=O)[O-])N2CCOCC2)/C#N RH01315 CCN(c1ccccc1)C(=S)Nc2ccccc2OC SW00053 c1cc(c(cc1C(F)(F)F)c2ccc(o2)C(=O)O)Cl JFD02875 CCN(CC)c1ccc(c(c1)NC(=O)N)/N=N/c2ccc(cc2)N(C)C JFD03405 CN1CCCc2c1ccc(c2)/N=N/c3ccccc3C#N JFD03406 CN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)Br JFD03407 c1ccc(cc1)NC(=O)Nc2ccccc2C(=O)O P00255 c1ccc-2c(c1)CCc3c2nc(s3)/N=C/c4ccc5c(c4)OCO5 RH01321 Cc1cc(=O)n(cn1)C(C(=O)c2ccccc2)NC(=O)c3ccccc3 BTB14956 c1c(c(c(c(c1I)Cl)Cl)Cl)Cl BTB15047 Cc1c(c(c(c(c1Br)Br)Br)Br)Br BTB15048 c1ccc(c(c1)NC(=S)NCc2ccccn2)Cl NH00507 CCOC(=O)c1csc(n1)N RH01231 COC(=O)C12CCC(=O)C(C1)(CCC2=O)C(=O)OC BTB14979 Cc1ccc(cc1)/N=N/c2ccc3c(c2)CCN3CCC(=O)OC JFD03381 c1cc(c(cc1CO)[N+](=O)[O-])N2CCCC2 RH01300 CC(CCO)(C12CC3CC(C1)CC(C3)C2)O BTB14986 Cc1c(c(on1)C)C(=O)NCc2c(cccc2Cl)F SEW05854 Cc1c(c(on1)C)S(=O)(=O)N(C)Cc2ccccc2 SEW05822 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)OC SEW05823 c1c(cc(c(c1/C=N/NCCO)O)Cl)Cl BTB03981 c1cc(ccc1C#N)/N=N/c2ccc3c(c2)CCCN3CCC#N JFD03378 c1ccc2c(c1)c(cs2)CCNC(=S)Nc3ccc(cc3)Cl S10770 c1cc(c(c(c1)Cl)CSC(=N)N)F.Cl S11211 c1ccc(c(c1)c2ccc(o2)C=C(C#N)C#N)C(F)(F)F JFD02882 Cc1ccccc1NC(=O)c2cc(n(c2C)c3ccccc3)c4ccccc4 SP00341 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)Nc4ccc(cc4)OC SP00352 Cc1c(cc(n1c2ccccc2)c3ccc(cc3)Cl)C(=O)Nc4ccccc4 SP00356 COC(=O)c1ccc(s1)c2ccccc2 SEW05850 CC(=O)N/C(=C\c1ccccc1Br)/C(=O)O SPB08006 CC(C)(C)OC(=O)Nc1ccc(cc1)CC(=O)O NRB00846 COc1ccc(cc1)NC(=O)c2ccccc2Sc3ccccc3CO BTB14929 CCOC(=O)/C(=C/c1ccc(s1)OC)/C#N S11311 c1ccc2c(c1)C(OC2=O)CC(=O)c3ccc(s3)Cl S11459 CC12CCC(=O)C=C1C[C@H](C3C2[C@@H](CC4(C3CC[C@@]45CCC(=O)O5)C)O)C(=O)OC JFD02853 Cc1ccc(cc1Cl)OCC(=O)O JFD02894 c1cc(cc(c1)C(F)(F)F)c2ccc(o2)c3cccc(c3)C(F)(F)F JFD02901 c1cc(ccc1NC(=S)NC2CCCC2)S(=O)(=O)N3CCCCC3 CD00808 CC1=N/C(=C\c2ccc(cc2)NC(=O)C)/C(=O)O1 SPB08010 CC(C)[C@H]1COC(=N1)c2cccc(n2)C3=N[C@H](CO3)C(C)C JFD02892 c1cc(c(c(c1)Cl)CSC(=N)N)Cl.Cl S11212 c1ccc(cc1)N2C(=O)c3cccc4c3c(ccc4N5CCSCC5)C2=O JFD03396 c1ccc-2c(c1)CCc3c2sc(c3C#N)N JFD03398 C=CCNC(=S)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl SEW06070 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2)[N+](=O)[O-])C(=O)OC RJC03441 CC1(C(C(=O)NC(=O)C1C#N)C#N)c2cccc(c2)OC SPB07986 Cc1c2ccccc2sc1/C=C\3/C(=O)OC(=N3)C SPB07992 CC(c1ccccc1)NC(=O)C JFD03490 Cc1cccc(c1C)NC(=O)C JFD03467 c1c(cc(c(c1Cl)n2c(=O)c(c(cn2)N3CCOCC3)Cl)Cl)C(F)(F)F SEW05767 C/C(=N\NC(=O)N)/c1ccccc1[N+](=O)[O-] SEW05772 C1C2CC3(CC1CC(C2)(C3)Cl)CC(=O)O BTB14958 c1cc(ccc1NC(=O)C23CC4CC(C2)CC(C4)C3)Br BTB14962 CC(C)C12CC3CC(C1)CC(C3)(C2)C(=O)NN BTB14966 Cc1cc(nc(n1)C(C)C)O BTB14961 C1C2CC3C(=NNC3=O)C1CC4=NNC(=O)C24 BTB14946 c1cc(ccc1F)S(=O)(=O)Nc2ccc(c(c2)F)F DSHS00758 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)Cl GK02955 Cc1ccsc1/C=C\2/C(=O)OC(=N2)C SPB07993 c1cc(ncc1C(F)(F)F)N2CCN(CC2)c3cnn(c(=O)c3Cl)c4c(cc(cc4Cl)C(F)(F)F)Cl SEW05768 Cc1cccc(c1NC(=S)N(CCC#N)C(C)C)C SW00049 Cc1c(c(on1)C)C(=O)O/N=C(/c2ccc(cc2)OC(F)(F)F)\N SEW05971 c1c(cnc(c1Cl)N2CCN(CC2)C(=O)/C=C/C(=O)O)C(F)(F)F SEW05973 c1cc(c(nc1)N2CCN(CC2)C(=O)c3cc(cc(c3)Cl)Cl)C(F)(F)F SEW05975 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2cccc(c2)Cl GK02956 CC12CC3(CC(C1)(CC(C2)(C3)O)C)C BTB14983 CC(C)(C)c1ccc(cc1)c2nnc(o2)S SPB07975 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)C(C)(C)C SEW05831 c1cc(ccc1c2csc(n2)c3cc(cc(c3)Br)Br)Cl SEW05780 c1cc2c(c(c1)F)c(ncn2)N SEW05781 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW05976 CC(C)(C)SCc1cccc(c1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05980 CC(C)(C)c1ccc(cc1)NC(=O)CSc2n[nH]c(=O)n2c3ccc(cc3)OCc4ccccc4 SPB07874 CS(=O)(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl SEW05984 Cc1c(c(on1)C)c2nnc(o2)c3ccc(cc3)OC(F)(F)F SEW05985 COC(=O)CCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)[N+](=O)[O-] JFD03383 c1cc(c(cc1Cl)Cl)c2ccno2 SEW05782 CCOC(=O)c1cnn(c1C)c2ccc(cc2)N SEW05794 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C(=O)/C=C/C(=O)O SEW05982 c1ccc2c(c1)Nc3ccc(cc3S2)C#N JFD02913 COC(=O)c1c2c(sc1N)CCC2 JFD03400 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC(Cc4c[nH]cn4)C(=O)NC(CCC(=O)N)C(=O)N5CCCC5C(=O)O JFD02942 c1ccc(cc1)COc2cccc(c2)C=C(C#N)C#N PD00354 Cc1ccc(cc1C)C(=O)c2c(ccc3c2cccc3)C JFD03464 CCc1cc(c(s1)N)C(=O)OC JFD03393 CC12CC3CC(C1)CC(C3)(C2)OC(=S)SC BTB14951 C1C2CC3(CC1CC(C2)(C3)Br)CCC(=O)O BTB14952 c1ccc(cc1)/C=N/CCNc2nccc(n2)C(F)(F)F AW00574 c1ccc(cc1)c2nc3cc(ccc3c(=O)o2)Cl S01228 c1ccc(cc1)C\2=NOC(=O)/C2=C\c3ccc(cc3Cl)Cl BTB06170 c1cc(c(cc1Cl)Cl)C(=O)NCCSC(=O)c2ccc(cc2Cl)Cl BTB09422 CCC(C)C(C(=O)O)NC(=O)C(CC(C)C)NC(=O)C(CC(=O)N)NC(=O)C(CCC(=O)OC(C)(C)C)NC(=O)C(C)NC(=O)C(CC(=O)OC(C)(C)C)NC(=O)OCC1c2ccccc2-c3c1cccc3 JFD02949 CC(C)C12CCCC(C1)(CCC2)C(=O)O BTB14973 C/C(=N/O)/C12CCC(C1)CC2 BTB14974 CC(=O)NC12CC3CC(C1)(CC(C3)(C2)C(=O)O)C BTB14976 c1ccc(c(c1)C#N)c2ccccc2C#N BTB14940 CCN(c1ccccc1)C(=S)Nc2c(cccc2C)C SW00057 C/C(=N/O)/C12CCCC(C1)CCC2 BTB14977 c1ccc(c(c1)NC(=O)NCCNc2ccc(cn2)C(F)(F)F)Cl AW00693 COc1ccc(cc1)c2cc(n3c(n2)cc(n3)c4cccs4)C(F)(F)F KM10411 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4cccc(c4)[N+](=O)[O-] KM10416 Cc1ccc2c(c1)nc([nH]2)SCC(=O)NCCSCc3ccco3 KM10409 Cc1c(ccc(n1)C(F)(F)F)C(=O)O/N=C(/c2cnccn2)\N AW00758 Cc1cc(on1)C(=O)NC(Cc2c[nH]c3c2cccc3)C(=O)OC RH01588 CCc1ccc(cc1)NC(=S)Nc2cc(cc(c2)C)C K00007 Cc1c(c(on1)C)c2nc(no2)c3cccc(c3)C(F)(F)F SEW05990 c1ccc(c(c1)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)O SEW05991 Cc1c(snn1)C(=O)Nc2cccc(c2)N SEW05857 c1cc(cc(c1)OCC(CNCCNc2nccc(n2)C(F)(F)F)O)C(F)(F)F AW00699 c1ccc2c(c1)c(cc(n2)c3cccnc3)N4CCOCC4 RJC03447 Cc1ccccc1NC(=O)c2cc(n(c2C)c3ccccc3)C(C)(C)C SP00312 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3ccccc3)C(F)(F)F GK03151 Cn1c(ccn1)NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N GK03150 Cc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)Cl GK03147 Cc1c(c(on1)C)C(=O)Oc2ccc(cc2)F SEW05859 CC(C)(C)c1ccc(cc1)NC(=O)c2ccc(s2)C(C)(C)C SEW05861 Cc1cc(c(n1Cc2cccs2)C)C(=O)Nc3ccc(cc3)OC SP00307 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)Nc3ccc(cc3)Cl SP00309 COc1ccc(cc1OC)C(=O)NC2CCCCC2 JFD02683 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW05995 COC(=O)CSc1[nH]c2ccccc2n1 JFD02859 COc1cc(cc(c1OC)Br)/C=C/C(=O)NCC(=O)O JFD02869 Cc1cc(cc(c1)NC(=O)c2cc(n(c2C)c3ccccc3)C(C)(C)C)C SP00317 CN(C)CCNc1cc(nc2c1cccc2)c3cccs3 RJC03452 CC(C)COc1ccc(cc1)/C(=N\O)/c2ccccc2 RJC03469 c1ccc(cc1)OCC(=O)NN RH01330 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3cccc(c3)Br RH01580 CC(C)(C)C(=O)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06071 Cc1c(c(on1)C)C(=O)Oc2ccc(cc2)C(C)(C)C SEW05870 c1cc(c(cc1[N+](=O)[O-])CO)N2CCCC2 RH01306 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)/C=C(\C#N)/C(=O)O JFD02863 CCN(CC)CCNc1cc(nc2c1cccc2)c3cccs3 RJC03454 CCCCCCCCCCOc1ccc(cc1)/C(=N\O)/c2ccc(cc2)C RJC03470 c1ccc(cc1)n2c(c(c3c2nc4ccccc4n3)C#N)N RJC03473 c1c(cc(cc1Br)Br)C(=O)NC(=O)N2CCCCC2 SEW05796 CCOC(=O)CNC(=O)/C=C/c1cc(c(c(c1)Br)OC)OC JFD02870 CC(=O)N/C(=C\C=C\c1ccccc1)/C(=O)O SPB08005 CC(=O)N/C(=C\c1ccc(cc1)C#N)/C(=O)O SPB08008 CC(=O)N/C(=C\c1ccc(c(c1Cl)OC)OC)/C(=O)O SPB08015 COC(=O)/C(=C\c1cc(ccc1N2CCOCC2)[N+](=O)[O-])/C#N RH01312 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)C(F)(F)F SEW05825 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)Cl SEW05827 c1cc(c(cc1S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl)Cl SEW05996 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW05997 c1ccc(c(c1)c2ccc(o2)/C=C(\C#N)/C(=O)O)C(F)(F)F JFD02884 CC1=N/C(=C\c2ccc(c(c2Cl)OC)OC)/C(=O)O1 SPB08011 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)O)Br SP00273 c1cc(ccc1NC(=O)NC(=O)c2cc(cc(c2)Br)Br)Cl SEW05797 Cc1cc(c(cc1NC(=O)c2ccccc2)OC)N SB01964 CCOC(=O)/C(=N\Nc1ccccc1)/c2csc(n2)Nc3ccc(cc3)OC JFD02975 COC(=O)C12CC3CCC(C1=O)CC(C2)(C3=O)C(=O)OC BTB14995 CC12CCCC(C1)(CCC2)C(=O)NN BTB14996 CCOC(=O)/C(=N\Nc1ccccc1)/c2csc(n2)Nc3ccc(cc3)C JFD02977 Cc1c(c(on1)C)C(=O)Nc2ccccc2 SEW05824 CC(=O)N/C(=C\c1ccc(cc1)OC(F)(F)F)/C(=O)O SPB08016 COc1ccc(cc1)n2c(nnc2SCC(=O)c3ccc(cc3)[N+](=O)[O-])c4ccncc4.Br.Br ML00376 c1cc(ccc1CNC(=S)N)F PD00384 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2OC(F)(F)F)Cl)F SEW05846 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2Cl)C(F)(F)F SEW05849 CCN(c1ccccc1)C(=S)Nc2ccc(cc2)OC SW00055 CN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)OC JFD03409 c1cc(ccc1/N=N/c2ccc3c(c2)CCCN3CCC#N)Br JFD03410 CC(C)CC(C(=O)NC)NC(=O)OC(C)(C)C JFD02956 Cc1ccc(cc1)S(=O)(=O)OCC(C(=O)OC)NC(=O)OC(C)(C)C JFD02959 c1cc2c(cc1Br)/C(=N/NC(=S)N)/C(=O)N2 RH01310 c1c(nc(s1)N)CSC(=[NH2+])N.Cl.[Cl-] CD04923 c1ccc(c(c1)n2c(nnc2SCC(=O)c3cccc(c3)[N+](=O)[O-])c4ccco4)Cl.Br ML00340 COc1ccc(cc1)n2c(n[nH]c2=S)c3cc(c(c(c3)OC)OC)OC ML00366 c1cc(ccc1CNC2=NC(CS2)(CO)CO)F PD00386 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW05998 Cc1c(nc(s1)c2ccc(cc2)Cl)CC(=O)NN SEW05808 Cn1cnc2cccc(c2c1=N)F SEW05811 Cc1ccc2c(c1)nc-3c(n2)-c4cccc5c4c3ccc5 JFD02984 c1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4ccccc4F JFD03046 c1ccc2c(c1)nc(c(n2)N/N=C\c3ccc(cc3)Cl)/C=C/c4cccs4 JFD03050 c1cc(ccc1C(=O)Nc2ccc(cc2OC(F)(F)F)Cl)Cl SEW05833 Cc1c(c(on1)C)C(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl SEW05834 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)C(C)(C)C SEW05835 c1cc(sc1/C=N/NC(=O)N)Cl SEW05783 c1c(ccc(c1)/N=N/c2ccc(cc2)[N+](=O)[O-])Nc3ccc(cc3)/N=N/c4ccc(cc4)[N+](=O)[O-] JFD03379 c1ccc(cc1)CNCC(Cn2c3ccc(cc3c4c2ccc(c4)Cl)Cl)O JFD02972 c1ccc(cc1)C(=O)C/C(=C\C(=C\2/C(=O)N=C(S2)N3CCCC3)\c4ccccc4)/c5ccc(cc5)Cl JFD03036 c1cc(ccc1c2c(cno2)c3nnnn3c4ccc(cc4)Cl)Cl JFD03043 Cc1c(c(on1)C)S(=O)(=O)N(C(C)C)C(C)C SEW05828 COc1cccc(c1)C(=O)Nc2ccc(cc2OC(F)(F)F)Cl SEW05832 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW05999 c1ccc2c(c1)c(cs2)CNC(=S)NCC3CC3 PD00402 c1c(cc(c(c1/C=N/CC2CC2)O)I)I PD00407 CCNC(=O)C(CC(C)C)NC(=O)OC(C)(C)C JFD02957 CC(C(C(=O)O)NC(=O)C(CSC(C)(C)C)NC(=O)OCC1c2ccccc2-c3c1cccc3)OC(C)(C)C JFD02954 CC(c1ccccc1)NC(=S)N/N=C/c2cc(cc(c2O)Cl)Cl RDR00802 Cc1cccc(c1NC(=S)NC(C)(C)CO)C RDR00460 c1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4ccc(cc4)F JFD03041 c1ccc(cc1)n2c(nnn2)c3cnoc3c4ccc(cc4F)F JFD03044 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)Cl SEW05838 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)O)C.CN1c2ccccc2C(=NC(C1=O)N)c3ccccc3 RJC03401 Cc1c(c(on1)C)C(=O)Nc2ccccc2OC(F)(F)F SEW05847 C/C(=N\c1ccccc1C(F)(F)F)/c2cccs2 JFD02891 COc1cc2c(c(c1)OC)C(OC2=O)OC JFD02895 C1CC2(CCC1C2)C(=O)NO BTB14998 C1CC2(CCCC(C1)(C2)Br)C(=O)N BTB15002 Cc1ccc(cc1)S(=O)(=O)c2ccc(c(c2)N)Cl RH01322 Cc1c(c(on1)C)S(=O)(=O)NCc2ccccn2 SEW05839 Cc1c(c(on1)C)S(=O)(=O)N2CCSCC2 SEW05840 Cc1cc(no1)NC(=O)c2c(noc2C)C SEW05842 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)C#N SEW05843 c1cc(ccc1C/N=C/c2cc(cc(c2O)I)I)F PD00408 CC1(C2CC3CC(C2)CC1C3)O JFD03015 Cc1c(c(on1)C)C(=O)N2CCSCC2 SEW05869 CC(C)(C)c1ccc(s1)C(=O)Nc2ccccc2OC(F)(F)F SEW05871 c1ccc2c(c1)[nH]c(=O)c(n2)/C=C/c3cccs3 JFD03047 c1ccc(cc1)/C=N\Nc2c(nc3ccccc3n2)/C=C/c4cccs4 JFD03049 CC1=C(C(C(=C(N1)C)C#N)c2ccccc2OC)C#N RJC03425 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2Cl)Cl)C#N RJC03426 c1c(cc(c(c1Cl)n2c(=O)c(c(cn2)N3CCCC3)Cl)Cl)C(F)(F)F SEW05792 CCN(CC)c1cnn(c(=O)c1Cl)c2c(cc(cc2Cl)C(F)(F)F)Cl SEW05793 CCOC(=O)COc1ccc2c(c1)oc(c(c2=O)Oc3ccc(cc3)C(=O)OC)C(F)(F)F BTB15058 c1ccc2c(c1)CC(NC2)C(=O)O.Cl JFD02927 CN1CCN(CC1)c2ccccc2/C=N\NC(=S)N SEW05759 c1cc2ccc3cccc4c3c2c(c1)cc4CCCn5c(=O)[nH][nH]c5=O JFD03446 COC(=O)/C(=C\c1cc(ccc1N2CCCCC2)[N+](=O)[O-])/C#N RH01313 C1CC2CCCC(C1)(C2)C(=O)NO BTB14971 COC(=O)C12CCC3(CC(C1=O)(CC(C2)(C3=O)C(=O)OC)C(=O)OC)C(=O)OC BTB15019 C(CSc1nnc(s1)S)Sc2nnc(s2)S JFD03130 c1cc(oc1)CSCCNC(=O)C2CCC2 KM10312 CCOC(=O)c1cc(n(c1C)CCSC)C(C)(C)C SP00337 CCOC(=O)c1cc(n(c1C)c2ccccc2)c3ccc(cc3)Cl SP00339 c1cnc(nc1C(F)(F)F)NCCNC2CCCCC2O AW00719 Cc1c(ccc(n1)C(F)(F)F)C(=O)NNC(=S)Nc2ccc(c(c2)Cl)F AW00720 CC1=C(C(C(=C(N1)C)C(=O)OC)c2cc(c(c(c2)OC)OC)OC)C(=O)OC RJC03432 C1CCc2c(c(n[nH]2)C(F)(F)F)C1 BTB15061 COC(=O)/C=C/1\C(=O)NCCN1 PD00240 CCC1(COC2(c3cc(ccc3NC2=O)F)OC1)CC PD00487 CC1=CCC2C(C1)C(=O)N(C2=O)c3cccc(c3)SC PD00488 Cc1c(cc(o1)C(C)(C)C)c2c(c(sc2C(=O)OC)S(=O)(=O)C)C#N SP00278 c1ccc(cc1)C(=O)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4 SPB07862 c1cc(cc(c1)F)C(=O)CSc2nnc(n2c3ccc4c(c3)OCCO4)c5ccco5 SPB08065 COC(=O)c1c(ccs1)Oc2ccc(cc2NS(=O)(=O)c3ccc(cc3)C(F)(F)F)C(F)(F)F GK03087 CC1=C(C(C(=C(N1)C)C#N)c2ccc(o2)c3ccccc3C(F)(F)F)C#N RJC03419 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(c(c2)OC)OC)C(=O)OC RJC03420 CN1CCN(CC1)c2ccccc2C=C(C(=O)O)C(=O)O SEW05791 c1ccn(c1)c2ccc(cc2)c3cc(nc(n3)N)C(F)(F)F BTB14887 COc1ccc(cc1)c2cc(nc(n2)N)C(F)(F)F KM10314 c1ccc2c(c1)C(=O)C(=C(C#N)NCc3ccc(cc3)Cl)C2=O S13784 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)Nc4cccc(c4)[N+](=O)[O-] SP00366 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK03144 CCOC(=O)C1CCN(CC1)C(=O)C23CC4CC(C2)CC(C4)C3 SEW06076 COc1cccc(c1)C(=O)N2CCN(CC2)c3ccccc3OC SEW06079 c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3cc(c(s3)Cl)Br SEW06082 c1cc(ccc1/C=N/CCN2CCNC2=O)C#N PD00381 C1CC[C@H]2[C@H](C1)NC(=S)N2 JFD03427 Cc1ccc(cc1)S(=O)(=O)NCC=C JFD03429 COc1ccccc1c2nc3ccccc3s2 JFD02897 Cc1ccc(cc1)C(=O)NNC(=O)Cc2c(sc(n2)c3ccccc3)C RH01235 Cc1c(cc(n1c2ccccc2)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)C(F)(F)F SP00357 c1ccc(cc1)NC(=O)CC(=O)Nc2ccccc2 RH01334 CC1=C(C(C(=C(N1)C)C#N)c2ccc3c(c2)OCO3)C#N RJC03436 CCOC(=O)C1=C(NC(=C(C1c2ccccn2)C(=O)OCC)C)C RJC03439 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc3c(c2)OCO3)C(=O)OC RJC03440 c1ccn(c1)c2ccc(cc2)c3cc(n[nH]3)C(F)(F)F BTB15057 c1ccc(cc1)c2ccc(cc2)C(=O)O[C@H]3C[C@@H]4[C@H]([C@@H]3CO)CC(=O)O4 JFD02903 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)N4CCCC4 SP00367 Cc1c(cc(n1c2ccccc2)c3ccc(cc3)Cl)C(=O)Nc4ccc(cc4)Cl SP00381 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2c(nc3ccccc3n2)Nc4ccc(cc4)OC RJC03487 CC1CC(CC(C1)(C)C)N2CNC(=NC2)SCc3ccc(cc3)OC.Cl ML00411 c1c(cnc(c1Cl)N2CCN(CC2)C(=S)NC3CC4CC3C=C4)C(F)(F)F SEW06087 COC(=O)c1c(ccs1)Oc2ccc(cc2NS(=O)(=O)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F GK03143 c1ccc(cc1)/C=C/C=C/C=C/c2ccc3ccccc3c2 JFD03442 CCOC(=O)/C(=N/Nc1ccc(cc1)[N+](=O)[O-])/N2CC2 JFD03001 CCOC(=O)C1=C(NC(=C(C1c2cccs2)C(=O)OCC)C)C RJC03404 CCOC(=O)C1=C(NC(=C(C1c2ccc(o2)c3ccccc3C(F)(F)F)C(=O)OCC)C)C RJC03405 COC(=O)/C(=C\c1cc(ccc1N2CCCC2)[N+](=O)[O-])/C#N RH01314 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)N4CCOCC4 SP00358 CC1=NN(C(=O)C1)c2cccc(c2)S(=O)(=O)N RH01325 Cc1c(cc(n1CCSc2cc(nc3c2cccc3)C(F)(F)F)c4ccccc4)C(=O)O SP00360 c1cc(c(cc1CC(CO)C#N)[N+](=O)[O-])N2CCCCC2 RH01584 CC(c1ccccc1O)N(Cc2ccccc2)C(=S)Nc3c(cc(cc3Cl)Cl)Cl BTB00962 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)/C=C/C(=O)O)Cl GK03148 c1ccc(cc1)[C@@]2(C3C4CC5C3C(C6C5C4C62)(F)F)O RJC03412 c1ccc(cc1)S(=O)(=O)Nc2c(nc3ccccc3n2)Nc4ccc(cc4)Cl RJC03491 COC(=O)Cc1cccc2c1oc3ccccc3c2=O RJC03495 CCC(COC(=O)C)Nc1nc2c(n1Cc3ccccc3)c(=O)n(c(=O)n2C)C RJC03500 c1cc(c(nc1)Oc2ccc3c(c2)OCO3)C(=O)O TL00927 CC(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)O SPB08019 CC(=O)N/C(=C\c1cc(cc(c1)F)F)/C(=O)O SPB08021 CC(=O)N/C(=C\c1cccc(c1OC)OC2CCCC2)/C(=O)O SPB08022 c1c(c(c(c(c1Cl)Cl)Cl)Cl)Cl BTB15036 Cc1ccc(cc1)S(=O)(=O)N(Cc2ccccc2Cl)c3ccc(cc3C(=O)c4ccccc4)Br RJC03417 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccccc2OC)C(=O)OC RJC03418 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2)O)C#N RJC03422 CC(=O)Nc1nc-2c(s1)Cc3c2cccc3 RH01302 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC(=O)O RH01742 CC(=O)Oc1cc(cc(c1)OC(=O)C)C(=O)O JFD03438 c1ccc(cc1)CN2C(=O)CC(=O)N(C2=O)CCCCCCN3C(=O)CC(=O)N(C3=O)Cc4ccccc4 JFD03440 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(o2)c3ccccc3C(F)(F)F)C(=O)OC RJC03416 c1ccc(cc1)/C=N/c2ccc(cc2)F BTB00824 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2Cl)Cl)C(=O)OC RJC03423 CN(C)CCNc1ccc(c2c1nccc2)[N+](=O)[O-].Cl RJC03513 CCN(CC)CCNc1ccc(c2c1nccc2)[N+](=O)[O-].Cl RJC03514 CC(C)(C)c1ccc(s1)C(=O)N2CCCC2 SEW05874 CC(C)(C)c1ccc(s1)C(=O)N2CCCCC2 SEW05875 Cc1c(c(on1)C)C(=O)NCc2ccc3c(c2)OCO3 SEW05855 COc1ccc(cc1)n2c(nnc2SCc3ccc(cc3)Br)c4ccco4.Br ML00346 c1cc(c(c(c1)Cl)Cn2c(nnn2)c3ccc(cc3)[N+](=O)[O-])Cl GK02992 Cc1ccc(cc1)/C(=N/O)/c2ccc(cc2)OCC(C)C JFD03017 CC(C)COc1ccc(cc1)/C(=N\O)/c2ccc(cc2)OC JFD03018 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2Cl)O)C(=O)OC RJC03428 CC1=C(C(C(=C(N1)C)C#N)c2cc(c(c(c2)OC)OC)OC)C#N RJC03433 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccccc2)C(=O)OC RJC03435 CN(C)c1ccc(cc1C#N)/C=C\2/c3ccccc3NC2=O SEW05852 Cc1c(c(on1)C)C(=O)NCc2ccc(cc2)Cl SEW05853 c1cc(ccc1CCN2C(=O)CSC2=S)Cl PD00388 c1ccc(cc1)SCC(CNCCNc2nccc(n2)C(F)(F)F)O AW00696 Cc1cn(nc1C(F)(F)F)c2ccc(cc2NC(=O)C)[N+](=O)[O-] AW00698 Cc1ccc(cc1)Sc2c(cccn2)C(=O)N3CCC(CC3)c4ccccc4OC RH01577 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C/C(=N/O)/N SPB07978 CC1=N/C(=C\C=C\c2ccccc2)/C(=O)O1 SPB07998 CC1=N/C(=C\c2ccc3ccccc3c2)/C(=O)O1 SPB07987 COc1cccc(c1O)/C=C/2\C(=O)N(C(=S)S2)CCc3ccccc3 PD00378 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW05969 COc1ccc(cc1)c2c(c[nH]n2)/C=C(\C#N)/S(=O)(=O)C SEW05788 c1ccc2cc3c(cc2c1)c(cc(n3)c4c[nH]c5c4cccc5)C(=O)O S03067 CCOC(=O)c1cccc2c1c(ccc2)Sc3ccccc3C#N BTB14934 c1ccc(c(c1)CSC(=N)N)F.Cl S11206 Cc1cc(c(cc1Cl)C)SCc2ccc(cc2)F S11209 c1ccc2cc(ccc2c1)SC(CC(=O)c3ccc(cc3)Cl)c4ccsc4 S11227 CC(C)(C)c1ccc(s1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3Cl)Cl SEW05872 C1C2CC3CC1[C@@H](C(C2)C3=O)C(=O)O NRB01685 c1ccc2c(c1)c(cs2)CN3C(=O)CC4(CCCC4)CC3=O PD00391 CCOc1ccc(cc1)NC23c4ccccc4CCCC2C(=O)CS3 S15412 Cc1nc2cc3c(cc2s1)OCO3 JFD02992 c1ccn2c(c1)n[nH]c2=S JFD02994 Cc1c(c(on1)C)C(=O)Oc2ccc(cc2)[N+](=O)[O-] SEW05860 c1ccc(cc1)n2c(c(cn2)C#N)N BTB07733 Cc1nnc(s1)Sc2ccc(c(n2)Sc3nnc(s3)C)[N+](=O)[O-] RH01610 CN1CCCC12c3c(c4ccccc4[nH]3)CCN2.Cl.Cl RH01612 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2Cl)Cl)C(=O)OCC)C)C RJC03403 c1ccc2c(c1)c(ccn2)C(=O)O CC04601 COc1ccccc1NC(=S)NCc2csc3c2cccc3 PD00398 CC(C)(C)c1cc(n(n1)c2ccc(cc2)N)C(C)(C)C SEW05979 COC(=O)c1ccccc1c2c3ccc(cc3oc-4cc(=O)ccc24)O JFD03457 Cc1cn(nc1C(F)(F)F)S(=O)(=O)c2cn(nc2C(F)(F)F)C AW00701 CCCCc1ccc(c(c1)C)NC(=O)NCCNc2nccc(n2)C(F)(F)F AW00706 c1cc(c(c(c1)Cl)Cl)NC(=O)NCCNc2ccc(cn2)C(F)(F)F AW00707 c1cc(c(cc1Cl)Cl)CC(=S)N SPB07979 Cc1c(c(on1)C)c2nnc(o2)c3cccc(c3)Cl SEW05972 COc1ccc(cc1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05974 Cc1cc(c(c(c1)C)NC(=S)NCc2csc3c2cccc3)C PD00392 c1ccc2c(c1)cccc2/C=C/3\C(=O)N(C(=S)S3)CCc4ccc(cc4)Cl PD00396 CC(C)(C)C(=O)CSc1[nH]c(=O)c(c(n1)c2cccnc2)C#N S15224 CC(C)(C)c1ccc(s1)C(=O)Nc2cc(ccc2F)F SEW05863 Cc1c(c(on1)C)C(=O)Oc2ccc(cc2)Cl SEW05864 COC(=O)c1ccc(cc1)CSc2ccc(cn2)C(F)(F)F SEW05865 Cc1ccc(c(n1)S)C#N JFD02996 CNC(=S)NNS(=O)(=O)c1ccc(cc1)Cl RDR00444 CCOC(=O)C1=C(NC(=C(C1c2cccc(n2)C)C(=O)OCC)C)C RJC03410 COc1cc2c(cc1OC)C(NCC2)c3cc(ccc3N)Cl NRB01258 c1ccc2c(c1)c(cs2)CN(CN3C(=O)c4ccccc4C3=O)CN5C(=O)c6ccccc6C5=O PD00399 CCCCCSc1[nH]cnn1 RJC03578 CCc1cc2c(cc1OC(=O)C)occ(c2=O)c3nc4ccccc4s3 JFD02982 CCOC(=O)/C=C/c1ccc(cc1)OCc2ccccc2 JFD03474 c1ccc(cc1)COc2ccc(cc2)CCC(=O)O JFD03475 c1ccc(c(c1)c2nc3ccccc3s2)Cl JFD02907 COc1ccc(cc1OC)CCN2C(=O)c3cccc4c3c(ccc4Sc5ccccn5)C2=O PHG00261 CCCSc1ccc2c3c1cccc3C(=O)N(C2=O)CCc4ccc(c(c4)OC)OC PHG00235 COC(=O)C(Cc1c[nH]c2c1cccc2)NS(=O)(=O)c3cccc4c3non4 RH01614 c1cc(c(cc1CO)[N+](=O)[O-])N2CCOCC2 RH01301 Cc1ccc(c(n1)O)C(=O)O SB01990 Cc1ccc(cc1NC(=S)N(C)N)Cl S15298 Cc1ccc(cc1)C2C3=C(c4ccc(cc4CC3)OC)NC(=S)N2 S15331 Cc1cc(nc2c1c(c(s2)C(=O)NN)C)C JFD02979 c1ccc2c(c1)c3ccc(cc3oc2=O)OCC(=O)O JFD02981 c1cc(c(c(c1)Cl)Cl)NC(=O)N2CCCN(CC2)Cc3ccc(cc3Cl)Cl AW00692 c1ccc(cc1)CSc2[nH]c(=S)c(c(n2)c3ccc(cc3)Cl)C#N JFD03061 COc1ccc(cc1)c2c(c(=S)[nH]c(n2)SCc3ccccc3)C#N JFD03062 Cc1ccc(cc1Cl)/N=C/c2cc(c(c(c2)OC)OC)OC BTB00822 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CC(=S)N SPB07976 c1cc(ccc1OCC(CN2CCCN(CC2)c3nc4ccc(cc4s3)Cl)O)Br AW00751 c1ccc2c(c1)C3=Nc4ccccc4SC(C3CO2)c5ccc(cc5)C(F)(F)F S15531 COC(=O)c1c(ccs1)Oc2ccc(cc2NS(=O)(=O)c3ccc(cc3)C#N)C(F)(F)F GK03145 CCOC(=O)c1cc(n(c1C)CCCNC(=O)OC(C)(C)C)C(C)(C)C SP00320 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)Nc4ccc(cc4)Cl SP00333 c1cc(ccc1F)SCC(CNCCNc2nccc(n2)C(F)(F)F)O AW00694 c1cnc(nc1C(F)(F)F)NCCNC(=O)CSCC(=O)O AW00695 c1ccc2c(c1)nc(o2)SCC(=O)NCCSCc3ccco3 KM10408 COc1ccc(cc1)NC(=O)CSc2n[nH]c(=O)n2c3ccc(cc3)OCc4ccccc4 SPB07866 COc1cc(nc(n1)OC)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccco3 BTB15014 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)C SPB07983 CN(C)/C=C/C(=O)c1csc2c1cccc2 PD00387 Cc1ccc(cc1)S(=O)(=O)NCCNc2nccc(n2)C(F)(F)F AW00688 c1ccc(cc1)OCC(CNCCNc2nccc(n2)C(F)(F)F)O AW00689 c1cc(ccc1Oc2ccc(c(c2)C(F)(F)F)NC(=O)C(Cl)(Cl)Cl)Cl BTB02735 Cc1c(ccc(n1)C(F)(F)F)C(=O)Oc2ccc(cc2)OC(F)(F)F AW00741 c1cc(ccc1c2ncon2)[N+](=O)[O-] BTB04223 c1cc(oc1)c2cc(n3c(n2)cc(n3)c4ccco4)C(F)(F)F KM10319 c1cc(oc1)CSCCNC(=O)C2CCCCC2 KM10313 CC(C)(C)c1ccc(cc1)OCC(CNCCNc2nccc(n2)C(F)(F)F)O AW00705 c1ccc(cc1)NC2CS(=O)(=O)CC2O JFD03540 Cc1ccc(cc1)NC2CCS(=O)(=O)C2 JFD03541 Cc1ccc(cc1)NC2CS(=O)(=O)C=C2 JFD03542 Cc1c(ccc(n1)NC(=O)c2cnccn2)Br PD00486 c1csc(n1)c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F KM10397 c1ccc(cc1)CNC(=S)N2CCCC(=N2)c3ccc(cc3)F S15423 c1ccc(cc1)n2c(=O)c3ccccc3c(n2)c4cccc(c4)C(F)(F)F BLT00223 c1cc(c(c(c1)Cl)Cl)NC(=O)N2CCCN(CC2)Cc3ccc(cc3)F AW00703 c1cc(c(c(c1)Cl)Cl)NC(=O)NCCNc2nccc(n2)C(F)(F)F AW00704 c1ccc2c(c1)c(c(s2)C(=O)NNC(=S)N)Cl BTB04205 CN1C(=O)/C(=C\c2cccc(c2O)OC)/SC1=S PD00379 c1ccc(cc1)c2ccc(cc2)N3C(=O)C=CC3=O PD00489 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)Nc3c(cc(cc3Cl)Cl)Cl)C(F)(F)F GK03156 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK03153 COc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3ccccc3OC RH01581 CCCCc1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3ccccc3OC RH01608 c1cc(oc1C2Nc3c(c4c(s3)CCCC4)C(=O)N2)[N+](=O)[O-] RH01609 CNC(=S)C12CC3CC(C1)CC(C3)C2 RJC00965 c1cc(c(cc1NNC(=S)N)Cl)Cl PD00325 Cc1cc(no1)C(=O)NNC(=O)CSCc2cccc3c2cccc3 RH01597 c1ccc2c(c1)cccc2CSCC(=O)NNC(=O)c3ccc(cc3)[N+](=O)[O-] RH01595 CC(C)c1ccc(cc1)/C=C/c2[nH]c(nn2)SCc3cccc(c3)C(F)(F)F BLT00265 c1ccc2c(c1)cccc2CSCC(=O)Nc3ccc(cc3)C(F)(F)F RH01598 c1ccc(cc1)/C=C/C2=N/C(=C/c3cccc4c3cccc4)/C(=O)O2 PHG00745 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl RH01606 CNS(=O)(=O)c1ccc(cc1S(=O)c2ccccc2C(=O)O)C(F)(F)F RJC03547 c1ccc(cc1)N2C(C3C(O2)C(=O)N(C3=O)c4ccccc4Cl)c5cc(ccc5O)Br JFD03552 C=CCOc1cccc(c1)/C=C/2\C(=O)N(C(=S)S2)CCc3ccccc3 PD00380 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)N4CCCCC4 SP00413 CCCCc1ccc(cc1)C(=O)NNC(=O)CSCc2cccc3c2cccc3 RH01592 c1ccc2c(c1)cccc2CSCC(=O)NNC(=O)c3ccccc3Br RH01593 c1ccc2c(c1)cccc2CSCC(=O)NNC(=O)c3ccc(cc3)F RH01591 Cc1ccc(cc1)CSc2nnc(n2c3ccc4c(c3)OCCO4)c5ccco5 SPB08063 Cc1ccccc1Sc2ccccc2C(=O)O NRB00554 CN(C)CCC(=O)c1ccccc1 EN00044 COc1ccc(cc1)c2c(c[nH]n2)C=C(C#N)C#N SEW05799 c1ccc2c(c1)ccn2c3ccccc3C#N SEW05800 COc1ccc(cc1)c2c(c[nH]n2)/C=C\3/c4ccccc4NC3=O SEW05801 c1ccc2c(c1)c(cs2)C/N=C/c3cc(ccc3O)Br PD00390 Cc1ccc(o1)/C=C/2\C(=O)N(C(=S)S2)CCc3ccc(cc3)Cl PD00393 c1ccc2c(c1)C(=O)N(C2=O)CN(Cc3ccc4c(c3)OCO4)CN5C(=O)c6ccccc6C5=O PD00400 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)CSCc3cccc4c3cccc4 RH01596 CCOC(=O)Nc1cc(c(cc1C(=O)OC)OC)OC PD00490 COc1ccc(cc1)C(=O)CSc2c3ccccc3nc(n2)SCC(=O)c4ccc(cc4)OC PD00493 Cc1nc(cn1Cc2ccc(cc2)F)[N+](=O)[O-] RH01582 c1cc(ccc1OCCCCCOC(=O)c2ccc(cc2Cl)Cl)Cl RH01605 Cc1ccc(cc1)N2C(=O)C3C(N(OC3C2=O)c4ccccc4)c5ccc(cc5)F JFD03553 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN3CCN(CC3)c4cccc(c4)Cl)O JFD03558 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN3CCN(CC3)c4ncccn4)O JFD03559 c1ccc(c(c1)C(=O)O)SC2CC(=O)N(C2=O)c3ccc(cc3)OC(F)(F)F PD00397 Cc1c(ccc(n1)C(F)(F)F)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F AW00714 CCCSc1nnc(s1)S JFD03132 c1cc(c(cc1[N+](=O)[O-])CC(CO)C#N)N2CCCC2 RH01586 Cc1cc(ccc1[N+](=O)[O-])C2=NCCc3c2cc(c(c3)OC)OC BTB01887 c1[nH]c(nn1)SCCSc2[nH]cnn2 JFD03129 c1cc2c(cc1NC(=S)NCCNc3nccc(n3)C(F)(F)F)OCCO2 AW00709 Cc1c(ccc(n1)C(F)(F)F)NC(=O)c2ccc(cc2)C(F)(F)F AW00717 CC(C)(C)OC(=O)N/N=C\c1cccc2c1cccc2 AW00722 c1ccc(cc1)c2nc3c(n2O)CCCC3=O BTB15113 COc1ccc(cc1)S(=O)(=O)NC(Cc2c[nH]c3c2cccc3)C(=O)OC RH01579 c1cc(c(cc1CC(CO)C#N)[N+](=O)[O-])N2CCCC2 RH01583 COC(=O)C(Cc1c[nH]c2c1cccc2)NS(=O)(=O)c3cc(cc(c3)Cl)Cl RH01589 COC(=O)c1ccsc1NC(=O)CN2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl GK03083 CCOC(=O)c1cc(c(nc1C(F)(F)F)C)c2nc(cs2)c3ccccc3 AW00765 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN3CCCCC3)O JFD03561 c1ccc(cc1)C(=O)NC(=O)c2ccc(s2)c3ccc(cc3)Cl MBE00139 Cc1ccc2cc(ccc2[n+]1C)F.[I-] BTB02615 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3cc(cc(c3)Cl)Cl)Oc4ccc(cc4Cl)Cl MBE00146 COC(=O)C\1C(SC/C1=N\O)C(=O)OC BTB02636 CCOC(=O)c1cc(c(nc1C(F)(F)F)C)c2nc(cs2)C(=O)NN AW00732 Cc1cc(c(n1Cc2cccs2)C)C(=O)Nc3cccc(c3)OC SP00300 C/C(=N\N(C)C)/c1cc(cc(c1O)Cl)Cl BLT00271 Cc1c(c(on1)C)c2nnc(o2)c3ccc(cc3)OC SEW05988 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)C(=O)O SEW05992 c1ccc2c(c1)CC=C2C(=O)N SEW05817 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCCc2cccs2 AW00726 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)c2nnc(o2)S SPB08052 Cc1ccc(cc1)NC(=O)c2cc(n(c2C)Cc3cccs3)C SP00301 Cc1ccccc1NC(=O)c2cc(n(c2C)Cc3cccs3)C SP00302 c1cc(cc(c1)NC(=S)NNc2ccc(cc2[N+](=O)[O-])S(=O)(=O)NCc3ccco3)C(F)(F)F BLT00211 c1cc(cnc1)C(=O)NNC(=O)c2ccc(cc2)[N+](=O)[O-] BW00108 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CNCc3ccccc3)O JFD03568 c1ccc(cc1)Cc2cc(c(nc2N)N)Cc3ccccc3 JFD03571 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccccc3[N+](=O)[O-] BTB07053 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)c2nnc(n2CC3CCCO3)S SPB08097 c1ccc2c(c1)c\3c([nH]2)CCC/C3=N\O RH01623 CC(C)(C)NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2CN1C(=O)c3ccno3 SPB08050 COc1cccc(c1)C2CCN(CC2)C(=O)c3cccc4c3cccc4 RH01625 Cc1ccc(cc1)NC(=O)c2cc(n(c2C)c3ccccc3)C(C)(C)C SP00311 CSc1cccc(c1)NC(=S)NCc2ccc(cc2)F PD00382 CN(C)NC(=O)c1cc(c(c(c1)OC)OC)OC CD01642 c1cc(ccc1N2C(=O)CC(C2=O)SCCC(=O)O)OC(F)(F)F PD00410 c1ccc2c(c1)c(cs2)CNC(=S)Nc3cccc(c3Cl)Cl PD00412 COCCCNC(=S)Nc1ccc(c(c1)OC)OC RDR00224 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)N(C)CCC#N RDR00475 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2O)O RDR00472 COCCCNC(=S)Nc1cc(ccc1Cl)Cl RDR00398 Cc1ccc(c(c1)C)/N=C(/NCc2ccco2)\SC.I RDR00187 Cc1cc(cc(c1)NC(=O)c2cc(n(c2C)Cc3cccs3)C)C SP00306 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)Nc3ccccc3 SP00310 CC(=O)Nc1cccc(c1)OCCCN2C(=O)c3ccccc3C2=O RH01634 CC1(C2CCC1(c3c2c(c4ccccc4n3)N5CCN(CC5)C)C)C RJC03443 c1cc(ccc1CSC(=N)N)C#N.Br CD00460 Cc1ccc(cc1)c2csc(n2)C.Br CD00561 Cc1c(c(c(c(c1C)C)CC2CC/C(=C\C=C\c3ccccc3)/C2=O)C)C CD01824 c1cc(cc(c1)Cl)N2CCN(CC2)CN3CCN(CC3)c4cccc(c4)Cl JFD03585 COc1ccc(cc1/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])Br PHG00094 CCOc1cc(ccc1O)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00085 Cc1ccc(cc1)N(C2CS(=O)(=O)C=C2)C(=O)c3ccc(cc3)Cl RJC03592 CN1CCN(CC1)c2c3ccccc3nc-4c2CCc5c4cccc5 RJC03448 COc1ccc-2c(c1)CCc3c2nc4ccccc4c3N5CCOCC5 RJC03450 c1ccc2c(c1)c(cc(n2)c3cccs3)N4CCOCC4 RJC03451 Cc1cc(c(c(n1)S)C#N)C(F)(F)F RF01420 Cc1cc(nc2c1c3c(s2)c(=O)[nH]cn3)C JFD02961 COc1ccc(cc1)/C=N\Nc2c(nc3ccccc3n2)/C=C/c4cccs4 JFD03052 c1ccc2c(c1)nc(c(n2)Nc3cccc(c3)Cl)/C=C/c4cccs4 JFD03053 C1CCC2C(C1)N(C(=O)C(=O)N2O)O RJC03768 c1cn(c(=O)[nH]c1=O)[C@H]2C[C@@H]([C@H](O2)CO)O SB01981 CN(C)CCNc1cc(nc2c1cccc2)c3cccnc3 RJC03445 Cn1c(nnc1Sc2c(cccn2)[N+](=O)[O-])C(F)(F)F RH01390 Cc1c(cc(c(n1)OC)C#N)c2csc(n2)C BTB09217 Cc1ccc(cc1)n2c(c(c3c2nc4ccccc4n3)C#N)N RJC03474 c1cc(ccc1C2C3C(=NN2c4cc(ccc4Cl)Cl)C5CCN3CC5)C(F)(F)F PD00459 c1cc(ccc1NNC(=S)N)F PD00460 c1ccc(c(c1)NC(=O)NCCNc2nccc(n2)C(F)(F)F)Cl AW00708 CCCCCCCc1ccc(cc1)C(=O)NC(=S)Nc2cccc(n2)C BR00114 Cc1c(ccc(n1)C(F)(F)F)C(=O)Oc2ccc(cc2F)F AW00768 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2c3ccccc3Cl ML00361 c1cc(cc(c1)n2c(n[nH]c2=S)c3ccncc3)C(F)(F)F ML00384 Cc1ccc(c(c1)Cl)NC(=S)N(Cc2ccc(cc2)N(C)C)C(C)C BTB01073 Cc1ccc(cc1)Nc2c(nc3ccccc3n2)NS(=O)(=O)c4ccc(cc4)NC(=O)C RJC03485 Cc1ccc(cc1Cl)N2C(=O)CC(CC2=O)c3ccccc3 PD00464 c1ccc(cc1)C2CC(=O)N(C2=O)c3ccc(cc3)I PD00465 CC(C)(C)c1cc2nc(cc(n2n1)C(F)(F)F)c3ccc4c(c3)CCC4 KM10318 c1ccc-2c(c1)CCc3c2nc4cc(nn4c3C(F)(F)F)C5CC5 KM10320 c1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccccc3Cl JFD03027 c1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3F)F JFD03028 c1ccc(cc1)C(C(=O)O)Nc2ccc3c(c2)OCO3 PHG00362 CCN(CC)c1c(cc(c(n1)C)C#N)C(=O)OCC AW00725 Cc1nnc2n1nc(cc2)c3cccc(c3)N(C)C(=O)C SB02011 CCCCCCCc1ccc(cc1)C(=O)NC(=S)NCc2ccco2 BR00119 CCOC(=O)c1c2c(nc3ccccc3n2)n(c1N)c4ccc(cc4)Cl RJC03482 Cc1ccccc1n2c(n[nH]c2=S)c3ccccc3Cl BTB01269 c1ccc(cc1)CN\2C(=CS/C2=C(/C#N)\C(=O)N)c3ccccc3 DP00031 CC([C@H](/N=C/c1nc(ccc1)/C=N/[C@H](C(C)(C)C)CO)CO)(C)C JFD02837 c1ccc(cc1)C2CC(=O)N(C(=O)C2)c3ccc(cc3)Oc4ccc(cc4)Cl PD00463 c1cc2c(cc1C(=S)N)non2 KM06798 COC(=O)c1ccc2c(c1)nns2 KM10174 c1ccc2c(c1)C3(C(=O)N2)N(C(=O)CS3)c4ccc(cc4)F S11632 Cc1c(c(on1)C)C(=O)N(C)Cc2ccccc2 SEW05881 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)N SEW05885 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCc2ccc(c(c2)Cl)Cl AW00769 CCCCCc1ccc(cc1)C(=O)NC(=S)Nc2cccnc2 BR00118 c1cc(ccc1CCNC(=S)NN)Cl S09768 CCn1c2ccccc2c3c(c1=O)c(cc(=O)o3)O RJC03692 c1cc(cc(c1)[N+](=O)[O-])c2cc(n3c(n2)cc(n3)c4cccs4)C(F)(F)F KM10415 c1cc(oc1)CSCCNC(=O)CSc2nnc(s2)SCC(=O)NCCSCc3ccco3 KM10410 COc1ccc(cc1)Cn2c(=O)c3cc(c(cc3[nH]c2=O)OC)OC PD00500 Cc1ccc(cc1)NC(=O)c2cc(n(c2C)c3ccccc3)c4ccc(cc4)Cl SP00382 Cc1c(ccc(n1)C(F)(F)F)C(=O)Sc2ccccc2 AW00776 CCc1cc(c(s1)NC(=O)CSc2ccc(cc2)Cl)C(=O)OCC BTB05735 CC(C)C(=O)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06206 Cc1c(cc(n1CCSCCO)c2ccccc2)C(=O)O SP00349 CC(C)Nc1ccc(cc1[N+](=O)[O-])C#N KM10396 CCOC(=O)c1c(c2c(nc(nc2s1)SCc3ccccc3)c4ccc(cc4)Cl)N BTB15110 CCOC(=O)c1c(c2c(nc(nc2s1)SCc3ccccc3)c4ccc(cc4)OC)N BTB15111 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=S)Nc3ccc(c(c3)Cl)Cl)Cl GK03152 c1ccc(cc1)c2c(c3cc(ccc3[nH]c2=O)F)O RJC03694 CC1(C(=S)NC(N1O)c2ccccc2)C BTB15120 COc1ccc(c(c1)Sc2cc(c(cc2[N+](=O)[O-])Cl)n3cccc3)OC RH01732 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)c4ccc(cn4)C(F)(F)F)[N+](=O)[O-] SP00735 Cc1ccccc1NC(=O)c2cc(n(c2C)c3ccccc3)c4ccc(cc4)Cl SP00383 CCOC(=O)c1cc(n(c1C)CCNC(=O)OC(C)(C)C)c2ccccc2 SP00375 Cc1ccc(c2c1CCC2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F RH01741 CCOC(=O)c1cnc2c(ccc(c2c1O)C)C RH01740 c1cc2c(cc1NC(=O)c3cnccn3)OCCO2 PD00492 Cn1c2c(c(cc(n2)N(C)C)Nc3ccccc3)c(=O)n(c1=O)C RJC03657 CCO/C=C/1\C(=O)N(C(=S)S1)CCc2ccc(cc2)Cl PD00405 Cc1c(cnn1c2ccc(cc2)N)C(=O)O SEW05806 c1cc(ncc1[N+](=O)[O-])N/N=C/c2cc(cc(c2)Cl)Cl SEW05809 c1ccc(c(c1)C#N)N2CCOCC2 SEW05816 c1c(cc(cc1Br)Br)C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW05813 c1cc(ccc1c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F)Cl KM10398 c1ccc2c(c1)cccc2CNCCCC(=O)O.Cl RH01630 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-])C(F)(F)F GK03155 Cc1ccc(cc1)/N=C/2\NC(=O)C(S2)CC(=O)Nc3ccc(cc3)OC(F)(F)F PD00403 COc1ccc(cc1/N=C/2\NC(=O)C(S2)CC(=O)Nc3ccc(cc3)OC(F)(F)F)Cl PD00404 c1ccc2c(c1)C(=O)N(C2=O)CN(Cc3ccsc3)CN4C(=O)c5ccccc5C4=O PD00411 CCOC(=O)c1cc(c(nc1C(F)(F)F)C)/C(=N/O)/N AW00734 CCOc1c(c(=O)c1=O)Nc2cccc(c2)OC KM09707 Cn1cnc2c1c(=O)n(c(=O)n2C)CC(CN3CCN(CC3)CCO)O RJC03497 c1ccc2c(c1)c(cs2)C/N=C/c3cc(cc(c3O)I)I PD00406 c1ccc(c(c1)CN2C(=O)c3ccccc3C2=O)C#N PD00409 c1ccc2c(c1)/C(=N/NC(=S)N)/C(=O)N2 S15100 Cc1ccc(cc1)NC(=O)c2cc(n(c2C)c3ccccc3)c4ccccc4 SP00334 CCOC(=O)c1cc(n(c1C)CCCN2CCOCC2)c3ccccc3 SP00336 COC(=O)c1ccccc1C(=O)c2ccc(cc2)Cl S15078 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)N3CCOCC3)c4ccccc4 SP00338 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)NCCCN3CCOCC3 SP00343 Cc1c(ccc(n1)C(F)(F)F)C(=O)Oc2ccc(c(c2)Cl)Cl AW00755 Cc1c(c(c(c(c1C)C)CSC(=N)Nc2ccc(cc2)F)C)C.Cl CD02452 Cc1c(c(c(c(c1C)C)C(=O)CCc2cccc(c2)/N=C/c3cccs3)C)C CD02593 c1cc2c(ccc(c2nc1)NC34CC5CC(C3)CC(C5)C4)[N+](=O)[O-] RJC03517 c1cc2c(ccc(c2nc1)N3CCN(CC3)CCO)[N+](=O)[O-] RJC03520 CCOC(=O)c1nc2c(cc(s2)c3cccs3)nn1 BTB15100 C1CS(=O)(=O)CC1NC(=O)C23CC4CC(C2)CC(C4)C3 RJC03567 CCOC(=O)c1cc(c(nc1NCC=C)C)C#N AW00746 Cc1c(cc(c(n1)C(F)(F)F)C(=O)O)c2nc(cs2)c3ccccc3 AW00761 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)N3CCOCC3 SP00347 Cc1cc(cc(c1)NC(=O)c2cc(n(c2C)c3ccccc3)c4ccccc4)C SP00353 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N/N=C/c2ccc(cc2)N(C)CCC#N CD02026 C/C(=C\c1cc2ccccc2o1)/[N+](=O)[O-] S12819 COCCCNC(=S)N/N=C/c1ccccc1O CD02861 c1ccc(cc1)CN2C(=O)c3ccccc3S(=O)c4ccccc4S2(=O)=O RJC03538 c1cc(cc(c1)NC(=S)NNC(=O)c2cccnc2)C(F)(F)F BW00101 CN(C)c1ccc(cc1)/C=N/NC(=O)c2cccnc2 BW00102 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCc3ccccc3Cl AW00756 Cc1c(cc(n1c2ccccc2)c3ccc(cc3)Cl)C(=O)Nc4cccc(c4)OC SP00384 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)[N+](=O)[O-])c3ccccc3 SP00335 Cc1cccc(c1)NC2CS(=O)(=O)CC2O JFD03543 c1ccc(cc1)NC(=S)Nc2ccc(cc2)F BTB01552 c1cc(sc1)C(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SEW06072 c1ccc(cc1)/C=C/C(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SEW06074 Cc1cc(c(c(c1)C)C(=O)C2CCNCC2)C.Cl SEW06077 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3cccc(c3)Cl SEW06083 Cc1c(c(on1)C)c2nc(no2)c3ccc(cc3)OC(F)(F)F SEW06084 CC(C)c1ccc(cc1)/C=C/C(=O)Nc2cccc(c2)SC BLT00256 Cn1c2c(c3c(cc4ccc(cc4n3)Cl)c(=O)n2c5ccccc5)c(=O)n(c1=O)C RJC03671 Cn1c2c(c3c(cc4c(n3)cc(cc4Cl)Cl)c(=O)n2c5ccccc5)c(=O)n(c1=O)C RJC03672 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)Nc4ccccc4 SP00354 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN3CCN(CC3)c4ccccc4)O JFD03557 COC(=O)C(Cc1c[nH]c2c1cccc2)NS(=O)(=O)c3ccc(s3)CNC(=O)c4ccccc4 RH01652 c1ccc(cc1)N(CCc2ccccn2)S(=O)(=O)c3ccc(cc3)Cl.Cl BTB01647 Cc1cc(c2cc(ccc2n1)Cl)OCc3c(c(c(c(c3C)C)C)C)C BTB01323 CCc1ccc2c(c1)cc3c(n2)n(c(=O)n(c3=O)C)C RJC03656 c1cc(cc(c1)Cl)C(=O)NNC(=O)c2cccnc2 BW00106 Cn1c2c(c3c(c(=O)n2c4ccccc4)nc(o3)c5ccccc5)c(=O)n(c1=O)C RJC03668 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2c(nc3ccccc3n2)Nc4ccc(c(c4)O)C(=O)O RJC03488 c1cc2c(ccc(c2nc1)NCCCN)[N+](=O)[O-].Cl RJC03511 c1cc2c(ccc(c2nc1)NCCCCN)[N+](=O)[O-].Cl RJC03512 CN(C)CCCNc1ccc(c2c1nccc2)[N+](=O)[O-].Cl RJC03515 c1cc(oc1)CSCCNC(=O)c2ccc(cc2)Cl KM10290 CCOc1ccccc1NC(=O)NCCSCc2ccco2 KM10291 c1cc(oc1)CSCCNC(=O)c2cc(cnc2)Br KM10292 c1cc(cc(c1)[N+](=O)[O-])c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F KM10402 CCCCOC(=O)N/C=C\1/C(=O)c2ccccc2OC1=O S15529 CCOC(=O)c1c2cc(ccc2oc1c3ccccc3)OCC(=O)OC JFD02998 CNC(=S)N/N=C/c1ccc(cc1)N(C)CCC#N CD01324 C#CC1(CCCCC1)NC(=O)/C=C/C(=O)O CD01657 CN(C)c1ccc(cc1)C(=O)NNC(=O)/C=C\C(=O)O CD01837 CCC(CO)Nc1nc2c(n1Cc3ccccc3)c(=O)n(c(=O)n2C)C RJC03499 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN3CCOCC3)O JFD03560 c1ccc(cc1)COc2ccc3c(c2)cc([nH]3)C(=O)NN KM10298 c1cc(ncc1C#N)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06078 Cc1cc(no1)C(=O)N2CCN(CC2)c3ccccc3OC SEW06080 CC(c1ccccc1O)N(Cc2ccccc2)C(=S)Nc3ccc(c(c3)Cl)Cl BTB00965 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)C(Cl)Cl)Cl GK03146 COc1ccc(cc1)NNC(=S)N PD00457 c1ccc2c(c1)c(=O)[nH]c(n2)SCc3ccc(cc3Cl)Cl PD00037 c1ccc2c(c1)C(=O)N(C2=O)CN(CCC#N)C3CCCCC3 SW00051 c1cc2c(ccc(c2nc1)NCCNCCO)[N+](=O)[O-] RJC03516 COc1ccc(c(c1)OC)NC(=S)NNC(=O)Cn2nc(nn2)c3ccccc3Oc4ccc(cc4Cl)Cl MBE00151 c1cc(ccc1/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])O PHG00075 COc1ccc(cc1)/C(=C/c2ccco2)/C#N PHG00041 c1cc(ccc1CNC(=S)Nc2ccc(cc2F)F)F PD00385 CC(C)(C)c1ccc(s1)C(=O)N2CCOCC2 SEW05873 COc1cc(cc(c1)NC(=S)NC(=O)c2ccccc2)C(F)(F)F SEW05876 Cc1c(c(on1)C)S(=O)(=O)NCc2cc(c(c(c2)OC)OC)OC SEW05877 c1cc(cc(c1)[N+](=O)[O-])c2cc(n3c(n2)cc(n3)c4ccco4)C(F)(F)F KM10401 Cc1c2cc(ccc2sc1c3cc(n4c(n3)cc(n4)c5cccs5)C(F)(F)F)Cl KM10407 c1ccc(cc1)c2ccc(s2)C(=O)O CC10501 Cc1c(c(on1)C)C(=O)N(C(C)C)C(C)C SEW05868 c1ccc(cc1)/C=C/C(=O)NNC(=O)CSCc2cccc3c2cccc3 RH01594 CC(=O)N[C@@H](Cc1ccc(cc1)OC(F)F)C(=O)O SPB08036 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)OS(=O)(=O)c5ccc(cc5)Br RJC03677 Cc1cc(c(cc1Cl)C)S(=O)(=O)N2CCN(CC2)c3ccccc3OC SEW06091 CC(C)c1ccc(cc1)NNC(=S)N PD00466 CC(C)c1ccc(cc1)NN2C(=O)CC(C2=O)c3ccccc3 PD00467 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=O)c3ccc(s3)c4ccc(cc4)Cl MBE00137 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3cccc(c3)F)Oc4ccc(cc4Cl)Cl MBE00150 c1ccc(cc1)C(=O)NCCSCc2ccco2 KM10280 c1cc(oc1)CSCCNC(=O)Nc2ccc(cc2)OC(F)(F)F KM10283 c1cc2cc(ccc2nc1)C(=O)NNC(=O)c3cccs3 KM10279 COc1ccc(cc1OC)c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F KM10400 CC1(CCc2c1cc(cc2c3cc(n4c(n3)cc(n4)c5ccccc5)C(F)(F)F)C(C)(C)C)C KM10399 c1ccc(cc1)C(CC(=O)Nc2cccc3c2CCCC3)CC(=O)O PD00462 c1ccc-2c(c1)Cc3c2nc4cc(nn4c3C(F)(F)F)c5ccc(cc5)Cl KM10316 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3nccs3 KM10413 COc1ccc(cc1OC)c2cc(n3c(n2)cc(n3)c4ccco4)C(F)(F)F KM10412 c1ccc(cc1)C(CNCCNc2nccc(n2)C(F)(F)F)O AW00690 Cc1cn(nc1C(F)(F)F)c2c3c(csc3ncn2)c4ccccc4 AW00691 CNC(=O)NN(C)c1ccc(cc1[N+](=O)[O-])C(F)(F)F BTB02843 C/C(=N\NC(=S)Nc1cccc(c1)C(F)(F)F)/c2cc(ccc2O)Cl BLT00234 c1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4cccc(c4)F JFD03040 CN(C)c1ccc(cc1)/C=C/c2cc[n+](cc2)Cc3ccc(cc3)F.[I-] JFD02841 Cc1ccc2c(c1)c(no2)OC(=O)N(C)C RF01309 CC1(CCc2c1cc(cc2c3cc(nc(n3)N)C(F)(F)F)C(C)(C)C)C KM10323 c1cc(sc1)c2cc(nc(n2)N)C(F)(F)F KM10327 COc1c(csc1C(=O)NN)Br GK02578 Cc1ccc(cc1)C(=O)C2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] SEW05891 CC(C)(C)c1cc2nc(cc(n2n1)C(F)(F)F)c3cccc(c3)[N+](=O)[O-] KM10403 C#CC1(CCCCC1)NC(=O)NC(=O)c2c(cccc2F)F BTB03929 COC(=O)c1cccnc1SC BTB06827 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NNC(=S)NCC2CC2 SPB08098 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)O SP00294 c1ccc(cc1)S(=O)(=O)NCCNc2nccc(n2)C(F)(F)F AW00812 c1cc(oc1)C(=O)NCCNc2nccc(n2)C(F)(F)F AW00813 CN1C(=O)c2ccccc2Sc3cc(ccc3S1(=O)=O)[N+](=O)[O-] RJC03544 CN1C(=O)c2ccccc2S(=O)c3cc(ccc3S1(=O)=O)[N+](=O)[O-] RJC03545 CNS(=O)(=O)c1cc(ccc1S(=O)c2ccccc2C(=O)O)Br RJC03546 CC(C)(CC(=O)NCc1csc2c1cccc2)CC(=O)O S11718 COc1ccccc1c2c(c(=O)c3ccccc3o2)O S11912 Cc1ccc(cc1)S(=O)(=O)N/N=C(/c2ccccc2)\c3ccc(cc3)OCC(C)C RJC03575 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NN SPB08096 c1cc(ncc1[N+](=O)[O-])Oc2cc(cnc2)Cl BTB07421 c1cc(cnc1)NC(=S)NCC2CC2 AW00829 CCOC(=O)C1=C(N(C(=NC1c2ccccc2)SC)C(=O)Oc3ccccc3)C JFD03077 c1c(c(=O)[nH]c(=O)n1[C@H]2[C@@H](C([C@H](O2)CO)O)O)I RJC03215 Cc1ccc(cc1)S(=O)(=O)N=S(Cc2ccccc2)Cc3ccccc3 BTB15072 C/S(=N\S(=O)(=O)c1ccccc1)/c2ccccc2 BTB15073 Cc1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4ccccc4F RJC03523 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NNC(=S)c2ccc3c(c2)OCCO3 SPB08099 CCc1ccc(cc1)OCC(=O)N(C)C2CCS(=O)(=O)C2 RJC03572 c1ccc(cc1)CC2C(=O)N/C(=N\c3ccccn3)/S2 JFD03550 Cc1ccc2c(c1)/C(=c/3\c(=O)n4c5ccccc5nc4s3)/C(=O)N2 JFD03554 CCCCCSc1[nH]c(=O)cnn1 JFD03555 CNS(=O)(=O)c1ccccc1S(=O)(=O)c2ccccc2C(=O)O RJC03552 Cc1c2c(=S)[nH]cnc2on1 SPB05318 c1cc(cnc1)NC(=S)NCc2ccco2 AW00830 CCCCCCCc1ccc(cc1)C(=O)NC(=S)Nc2ncccn2 BR00115 CCCCCCCc1ccc(cc1)C(=O)NC(=S)Nc2ccccn2 BR00117 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3ccc(cc3)[N+](=O)[O-])/C(=O)N2c4ccccc4 RJC03654 c1ccc(c(c1)C(=O)O)Sc2ccccc2S(=O)(=O)N RJC03554 Cc1ccc(cc1)S(=O)(=O)N(CCc2ccccn2)c3ccc(cc3)C(C)C.Cl BTB01670 Cc1cc(c(c(c1)C)C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)C BTB07471 Cc1cc(c(c(c1)C)C(=O)NC(=O)Nc2c(cc(cc2F)F)F)C BTB07473 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cccc2F)F)OC)Br)Cl BTB07744 CC(C)c1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC)C(C)C BTB07758 C/S(=N\S(=O)(=O)c1ccc(cc1)Cl)/c2ccccc2 BTB15075 Cc1ccc(cc1)Sc2c(nc3n2cccc3)c4ccccc4 RJC03559 c1ccc(cc1)c2cn3cccnc3n2 RJC03560 CCCCCc1ccc(cc1)C(=O)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB05762 CC(C)c1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)C(C)C BTB07614 c1cc(ccc1F)SCC(CNCCNc2ccc(cn2)C(F)(F)F)O AW00788 c1ccc(cc1)CCCC(=O)O SB02007 COC(=O)c1ccccc1Sc2ccc(cc2)[N+](=O)[O-] BTB15079 Cc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC)Cl BTB07709 c1ccc(cc1)n2c(nnn2)c3cnc(nc3c4ccccc4F)N RJC03521 Cc1ccc(cc1)n2c(nnn2)c3cnc(nc3c4ccccc4F)N RJC03522 COc1ccc(cc1)OCC(=O)N SPB08002 c1ccc(cc1)CNC(=S)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl BTB02315 CSc1ccccc1NC(=S)NNC(=O)Cn2nc(nn2)c3ccccc3Oc4ccc(cc4Cl)Cl MBE00148 CC(=O)Nc1ccc(cc1)/C(=N/O)/N DP01430 CC12C(NC(=O)N1)(NC(=O)N2)C ML00405 Cc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)Cl BTB07616 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OC)Br)[N+](=O)[O-] BTB07702 c1cc(c(cc1Br)S(=O)(=O)[O-])I.[K+] RJC03549 c1ccc(cc1)n2c(nnn2)c3c[nH]c4c3cc(c(c4)Cl)Cl RJC03526 Cc1ccc(cc1)n2c(nnn2)c3cnc4ccccc4c3c5ccccc5 RJC03530 COc1cccc(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)OC BTB07451 CC(C)CN(CC(C)C)CC(Cn1cnc2c1c(=O)n(c(=O)n2C)C)O JFD03566 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CNc3ccc(cc3)OC)O JFD03567 C1COCCN1C2=NC(=O)CS2 RJC03533 CCCCNc1ccc2c3c1cccc3C(=O)N(C2=O)CCCC JFD03094 c1ccc2c(c1)C(=O)NS(=O)(=O)c3ccccc3S2(=O)=O RJC03556 c1cc(ccc1[N+](=O)[O-])OCC(CNCCNc2nccc(n2)C(F)(F)F)O AW00783 c1ccc(cc1)CN(c2cccc3c2cccc3)C(=O)Nc4ccccc4 JFD03581 COc1ccc(c(c1)/C=N/NC(=S)NCCc2ccccc2)OC ML00116 CCCN(CCC)CC(Cn1cnc2c1c(=O)n(c(=O)n2C)C)O JFD03564 COc1ccc(cc1)n2c(nnn2)c3cnc4ccccc4c3N RJC03532 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(Cn3cnc4c3c(=O)n(c(=O)n4C)C)O JFD03570 Cc1cc(c(n1Cc2ccncc2)C)C(=O)O SP00292 Cc1cc(c(n1Cc2cccs2)C)C(=O)O SP00291 COc1cccc(c1C(=O)NC(=O)Nc2c(cc(cc2Br)Br)Br)OC BTB07461 C#Cc1cccc(c1)NC(=O)c2ccc(o2)[N+](=O)[O-] BR00077 c1ccc2c(c1)cccc2NC(=O)NCCSCc3ccco3 KM10285 Cn1c2c(cc3ccc(cc3n2)OC)c(=O)n(c1=O)C RJC03679 Cc1ccc2c(c1)c(c[nH]2)c3nnnn3c4ccc(cc4)Cl RJC03527 c1ccc2c(c1)C(=O)NC3(O2)CCCCC3 JFD03575 Cc1nc2c(o1)c3c(n(c(=O)n(c3=O)C)C)n(c2=O)c4ccccc4 RJC03667 COc1ccc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC)Br BTB07611 c1ccc(cc1)C2=C(OC3(C2Oc4c(c(c(c(c4Cl)Cl)Cl)Cl)O3)c5ccc(cc5)F)c6ccccc6 S14410 c1c(ccc(c1)F)/C=C\2/C(=O)/C(=C/c3ccc(cc3)F)/CC2 S15057 c1ccc(cc1)N2CCN(CC2)CN3CCN(CC3)c4ccccc4 JFD03584 CCOC(=O)CSc1ccc2c3c1cccc3C(=O)N(C2=O)CCc4ccc(c(c4)OC)OC PHG00259 Cc1ccc(cc1)n2c(nnn2)c3cnc4ccccc4c3N RJC03529 CCOC(=O)n1c2ccccc2oc1=O JFD03573 c1ccc2c(c1)n(c(=O)o2)C(=O)c3ccc(cc3)Cl JFD03574 c1ccc(cc1)CSc2ccccc2C#N JFD03096 c1ccc(cc1)CSc2ccccc2C(=O)O JFD03098 CCc1ccc(cc1)/C(=C/C=C/c2ccccc2)/C#N PHG00906 c1ccc(c(c1)C2(CC2)C#N)C3(CC3)C#N RJC03712 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)c4ccc(cc4Cl)Cl SEW05927 c1cc(oc1)CSCCNC(=O)Nc2ccc(cc2F)F KM10274 Cc1ccc(cc1C)CC(C(=O)O)NC(=O)C SPB08101 Cc1c(c2ccccc2o1)CCOC(=O)c3ccc(cc3)Cl S11672 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC)Cl)Cl BTB07688 CC1c2nc3ccc(cc3n2CN(CO1)c4ccc(cc4)OC(F)(F)F)Cl S14871 CCCc1cnc(nc1)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)C AW00861 c1ccc(cc1)CCNC(=S)NCCNc2nccc(n2)C(F)(F)F AW00715 c1ccc(cc1)NC(=O)Nc2ccc3c(c2)cccn3 KM10297 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCSCc2ccco2 KM10286 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3ccc(nc3Sc4ccccc4)Sc5ccccc5 SEW05929 Cc1c(cc(n1CCSC)C(C)(C)C)C(=O)O SP00345 Cc1c(c(c(c(c1C)C)C(=O)C2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])C)C SEW05892 CC(=O)N(C)c1ccc(cc1F)F TL00933 c1cc(ccc1S(=O)(=O)C(F)F)Cl RJC03717 COc1cccc(c1)NC(=O)Nc2cc(cc(c2)OC)C(F)(F)F SEW05887 Cc1cc(cc(c1)N2C(=O)CSC2=S)C S04501 c1ccc2c(c1)ccn2CC(CNCCNc3nccc(n3)C(F)(F)F)O AW00718 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)O SP00370 COc1cc(cc(c1)NC(=S)Nc2ccc(cc2)Cl)C(F)(F)F SEW05886 c1ccc(cc1)C(=O)C2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] SEW05888 c1cc(ccc1C(=O)C2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])F SEW05890 COc1ccc(cc1)c2cc(n3c(n2)cc(n3)C4CC4)C(F)(F)F KM10405 CC(C)(C)c1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(c(c3)OC)OC KM10406 c1cc2c(cc1C(F)(F)F)nnn2C3CCNCC3.Cl KM10214 c1cc(ccc1C(=O)C2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])Cl SEW05889 c1ccc(cc1)CN2CCC(CC2)NCC(COc3ccc4c(c3)OCO4)O AW00809 c1cnc(nc1C(F)(F)F)NCCNC(=O)C2CC2 AW00811 c1ccnc(c1)Sc2cc(c(cc2[N+](=O)[O-])Cl)n3cccc3 RH01736 CCOC(=O)CSc1cc(c(cc1[N+](=O)[O-])Cl)n2cccc2 RH01725 C/C(=N/O)/c1ccc(cc1)OCc2ccccc2 RJC03570 c1ccc(cc1)C(=O)CSc2nnc(n2c3ccc4c(c3)OCCO4)c5ccco5 SPB08066 c1cc(oc1)c2nnc(n2c3ccc4c(c3)OCCO4)SCC(=O)Nc5cc(cc(c5)Cl)Cl SPB08067 c1cc(oc1)c2nnc(n2c3ccc4c(c3)OCCO4)SCC(=O)Nc5ccc(cc5)C(F)(F)F SPB08068 c1ccc(cc1)c2c(c(c(n(c2=O)c3ccccc3)c4ccccc4)C(=O)c5ccccc5)O JFD03074 c1cc(sc1)C(=O)NCCNc2nccc(n2)C(F)(F)F AW00810 COc1cc(cc(c1)NC(=S)Nc2cccc(c2)OC(F)(F)F)C(F)(F)F SEW05912 Cc1ccc(cc1)S(=O)(=O)/N=S(\C)/c2ccccc2 BTB15067 CCS(=NS(=O)(=O)c1ccc(cc1)[N+](=O)[O-])CC BTB15074 COc1ccc(c(c1)S(=O)(=O)NC2CCS(=O)(=O)C2)OC BTB04400 CC(C)(C)c1ccc(cc1)NC(=O)N2CCCN(CC2)Cc3ccccc3 AW00792 c1cnc(nc1C(F)(F)F)N2CCN(CC2)CCO AW00793 c1ccc2c(c1)ccn2CC(CNCCNc3c(cccn3)C(F)(F)F)O AW00794 c1ccc(cc1)CN2CCCN(CC2)C(=O)Nc3ccc(cc3)Cl AW00795 CC1CC(=O)Nc2ccccc2N1C(=O)c3cccc(c3)Cl BTB00661 CC(C)(C)c1ccc(cc1)C(=O)O/N=C/c2ccc3c(c2)OCO3 RH01635 c1ccc2c(c1)c(ccn2)c3[nH]c4ccccc4n3 JFD03535 C/C(=N/O)/c1ccc(cc1)OCCO RJC03571 Cc1ccc(cc1)S(=O)(=O)/N=S(/c2ccccc2)\C(C)C BTB15070 c1ccc(c(c1)C(=O)N)NCC(=O)c2ccc(cc2)Cl BTB01835 CC(=O)OC12CC3CC(C1)CC(C3)(C2)C(=O)O JFD03085 C1CC2(CCC1(CC2)C(=O)O)C(=O)O JFD03086 C1CC2(CCC1C2)C(=O)NN JFD03087 c1ccc(cc1)c2c(n3ccsc3n2)Sc4ccc(cc4)Cl RJC03561 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2ccc[nH]2 BTB07257 c1ccc(cc1)OCC(CNCCNc2ccc(cn2)C(F)(F)F)O AW00785 Cc1ccc(cc1)S(=O)(=O)NC(=O)c2ccccc2 RJC03536 Cc1ccc(c(c1)[N+](=O)[O-])/N=N/c2c(nn(c2C)S(=O)(=O)c3ccc(cc3)F)C BTB00972 CN1C(=O)c2ccccc2Sc3cc(ccc3S1(=O)=O)Cl RJC03534 c1ccc(cc1)S2=NS(=O)(=O)c3c2cccc3 RJC03539 COc1ccc(cc1OC)CCNS(=O)(=O)c2cc(ccc2Cl)Cl DP00370 COc1ccc(cc1OC)CCNS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DP00371 c1ccc(cc1)CN2CCCN(CC2)C(=S)NC3CCCCCCC3 AW00797 c1ccc(cc1)CC(=O)NN JFD03115 CCOC(=O)c1ccc(cc1)N(C)C JFD03116 c1cc(c(nc1)NCCNCC(COc2ccc(c(c2)Cl)Cl)O)C(F)(F)F AW00786 c1cc(ccc1S(=O)(=O)N2CCCN(CC2)Cc3ccc(cc3Cl)Cl)Cl AW00835 c1cc(c(nc1)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F AW00836 c1cc(c(c(c1)Cl)CSC(=N)Nc2ccc(cc2)F)Cl.Cl CD02448 c1cc(ccc1CNC(=O)c2ccc(cc2)Cl)/C(=N/O)/N CD02765 Cc1cc(cc(c1NC(=O)NC(=O)c2c(ccc(c2OC)[N+](=O)[O-])OC)C)Br BTB07587 C1CC2CC34CC5(C2=NNC5=O)CC1C3=NNC4=O JFD03114 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)[N+](=O)[O-])NC(=O)C JFD03095 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/NCc3cccnc3)/C(=O)N2C RJC03660 CC(C)N(Cc1ccc(cc1)N(C)C)C(=S)Nc2ccc(c(c2)Cl)Cl BTB01072 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2cccc(c2)SC CD02022 CCN(CC)C(=S)Nc1cccc(c1)SC CD02445 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC)Br BTB07615 c1ccc2c(c1)ccn2CC(CNCCNc3ccc(cn3)C(F)(F)F)O AW00787 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN(CC=C)CC=C)O JFD03565 COc1ccccc1NC(=O)N2CCCN(CC2)Cc3ccc(cc3)F AW00848 c1ccc(cc1)c2nc(sn2)n3ccc(n3)C(F)(F)F AW00849 CCCc1cnc(nc1)N2CCCN(CC2)C(=O)NS(=O)(=O)c3ccc(cc3)C AW00854 c1ccc2c(c1)c3c([nH]2)c4ccccc4n5c3nnn5 RJC03687 CC(C)c1ccc(cc1)N(CCc2ccccn2)S(=O)(=O)c3ccc(cc3)Cl.Cl BTB01644 c1cc(ccc1c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5c(c4)CCC5)Cl KM10315 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3ccc(cc3OC)Cl)/C(=O)N2C RJC03661 c1ccc(cc1)Sc2ccccc2CC(=O)O BTB15078 CCC(CO)NC(=O)c1cc(c(c(c1)OC)OC)OC JFD03583 c1cc(c(c(c1)Cl)Cl)/C(=N/O)/N SPB01106 c1c(ccc(c1)/C=N/N=C(N)N)/C=N/N=C(N)N JFD03117 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3cc(cc(c3)Cl)Cl)/C(=O)N2C RJC03659 COCCCNC(=S)N/N=C/c1cccc(c1O)OC CD02862 c1cc(c(cc1C(=O)Nc2ccc3c(c2)[nH]nn3)Cl)Cl BTB01511 Cc1ccc(cc1NC(=S)Nc2ccc(cc2)F)NC(=O)C BTB01564 Cn1c2c(cc3cc(c(cc3n2)Cl)Cl)c(=O)n(c1=O)C RJC03655 COc1ccc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC)[N+](=O)[O-] BTB07578 CSc1ccccc1N2C(=O)CSC2=S S03508 Cc1cc2nc-3c(c(n2n1)C(F)(F)F)CCc4c3cccc4 KM10304 c1cc2cc(ccc2nc1)NC(=O)Nc3ccc(cc3)Cl KM10296 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)Nc5cccc(c5)C(F)(F)F RH01721 c1cc(oc1)C(=O)NC2CCS(=O)(=O)C2 BTB04394 c1ccc2c(c1)C(=O)N(C2=O)CN(CCC#N)Cc3cccnc3 SW00099 c1ccnc(c1)CCN(CCC#N)C(=S)Nc2cccc(c2)C(F)(F)F DSHS01296 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccco4 KM10307 c1ccc-2c(c1)Cc3c2nc4cc(nn4c3C(F)(F)F)c5cccs5 KM10308 CCCN(CCC#N)C(=S)Nc1ccc(c(c1)C)C SW00081 Cn1c2c(cc3cc(ccc3n2)c4ccccc4)c(=O)n(c1=O)C RJC03669 COC(=O)C(Cc1ccccc1)(Cc2ccccc2)C#N RJC03713 c1ccc(cc1)S(=O)(=O)CC2CC2(Cl)Cl RJC03721 c1cc(ccc1S(=O)(=O)NC2CCS(=O)(=O)C2)Cl BTB04396 c1cc(c(c(c1)Cl)C(=O)NC2CCS(=O)(=O)C2)Cl BTB04395 Cc1cc(c(c(c1)C)CSCC(=O)N/N=C/c2ccccc2O)C BLT00124 c1cc(sc1)C(CC(=O)c2ccc(cc2)Cl)C(C#N)C#N S13524 c1ccc(cc1)c2ccc(cc2)C(=O)/C(=C/c3cccc(c3)[N+](=O)[O-])/C(=O)c4ccc(cc4)N PHG00883 COC(=O)C1CC2CC(C1=O)CC(C23SCCS3)C(=O)OC JFD03084 c1ccc2c(c1)c(cs2)CN.Cl CC12313 c1ccc(cc1)C2CC(=O)N(C(=O)C2)c3cccc4c3CCCC4 PD00473 Cc1c(cc(c(n1)C)C(=O)C)C#N AW00736 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)NCC=C RH01722 c1cc(ccc1NC(=O)c2c(nccn2)C(=O)O)Cl PD00078 c1cc(ccc1N2C(=O)c3c(nccn3)C2=O)Cl PD00081 Cc1cc(c(c(c1)C)CSCC(=O)NNC(=O)c2cccc(c2)Cl)C BLT00131 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2ccc(cc2)Br S13644 c1cc(cc(c1)S(=O)(=O)Nc2ccsc2C#N)C(F)(F)F GK02473 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)OC(=N2)c3ccccc3I PD00475 CC(C)c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccccc3I PD00477 Cc1c(cc(n1CCCNC(=O)OC(C)(C)C)C(C)(C)C)C(=O)O SP00329 Cc1c(ccc(n1)C(F)(F)F)C(=O)Sc2ccc(cc2)F AW00750 CC1CCC2=C(C3C4C(C2(C1)C5C3C(=O)N(C5=O)Cc6ccc(cc6)Cl)C(=O)N(C4=O)Cc7ccc(cc7)Cl)C S14001 COc1ccc(cc1)C(=O)NCc2csc3c2cccc3 PD00418 c1ccc2c(c1)c(cs2)CNC(=O)c3ccc(cc3)OC(F)(F)F PD00423 c1ccc2c(c1)c(cs2)CNC(=O)c3ccco3 PD00424 c1ccc2c(c1)-c3c(cccc3C(=O)NCCO)C2=O JFD03219 CC(C)c1nn(c(=O)o1)c2ccc(cn2)C(F)(F)F RF04836 c1ccc(cc1)S(=O)(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl CD11888 CC1SCC(=NO)CS1 CD09937 COc1cccc(c1C(=O)c2ccncc2)OC CD11873 c1cc(c(c(c1)Cl)CNS(=O)(=O)c2ccc(cc2)Cl)Sc3ccc(cc3)Cl CD11886 CCc1ccccc1NNC(=S)N PD00472 Cc1c(c(on1)C)C(=O)NCc2ccco2 SEW05937 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)Nc4cccc(c4)[N+](=O)[O-] SEW05923 CN(C)/C=C/C(=O)c1cc(ccc1Cl)Cl CD11985 c1ccc2c(c1)-c3c(cccc3C(=O)NCCCN4CCOCC4)C2=O JFD03218 c1cc(cc(c1)NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F)C(F)(F)F SEW06124 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OCC(CO)NC(=O)CNC(=O)OCC4c5ccccc5-c6c4cccc6 RJC03210 CC(C)(C)C(=O)N1CCN(CC1)c2c(cccn2)C(F)(F)F SEW05907 CC/S(=N\S(=O)(=O)c1ccc(cc1)C)/c2ccccc2 BTB15068 c1ccc2cc(ccc2c1)OCC#N RJC03730 COc1ccc(cc1OC)C2(CC2)C#N RJC03706 c1cc(c(cc1F)F)N2C(=O)CSC2=S S07780 CCCCNC(=O)c1cccc2c1-c3ccccc3C2=O JFD03220 c1cc(ccc1N)Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] JFD03224 Cc1ccc(c(c1)COc2ccc(nc2NC(=O)c3ccc(cc3)F)C)C RH01353 Cc1ccc(c(c1)COc2ccc(nc2NC(=S)NCc3ccccc3)C)C RH01356 Cc1ccsc1/C=C/2\C(=O)OC(=N2)c3ccccc3I PD00476 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)Nc4ccc(cc4)OC(F)(F)F SEW05921 c1ccc(c(c1)NC(=S)NNC(=O)CSc2nc3cccnc3s2)F RH01368 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2cc(cc(c2)OC)C(F)(F)F)C)C CD06614 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O SB00572 c1ccc(c(c1)C(=O)NCc2cccs2)O CD06824 CC(=O)c1ccccc1N2C(=O)CSCC2=O S12274 c1ccc(cc1)NC2=CC(=O)OC2 BTB11211 c1cc(c(c(c1)Cl)N2C(=O)CSC2=S)F S07614 COC(=O)c1ccc(cc1)CSc2ncccn2 SEW05879 c1ccc(c(c1)n2c(nnc2SCC(=O)c3ccc(cc3)F)c4ccco4)Cl.Br ML00342 CC(=O)Nc1ccc(cc1)OC(=O)C RH01347 CC(C)(C)c1ccc(s1)C(=O)Nc2ccc(cc2)C(F)(F)F SEW05894 COC(=O)c1ccc(cc1)CSc2ccccn2 SEW05898 Cc1c(c(on1)C)C(=O)Nc2ccc(nc2Sc3ccccc3)Sc4ccccc4 SEW05930 Cc1c(c(on1)C)C(=O)NCc2cccs2 SEW05932 Cc1c(c(on1)C)C(=O)O/N=C(/c2ccc(cc2)Cl)\N SEW05933 C#Cc1cccc(c1)NC(=O)Nc2c(cccc2Cl)Cl BTB04470 CCC/S(=N\S(=O)(=O)c1ccc(cc1)C)/c2ccccc2 BTB15069 CCCCN1CCCc2c1ccc(c2)/N=N/c3ccccc3 RJC03699 c1ccc2c(c1)c3ccc(cc3[nH]2)/N=N/c4ccc(cc4)[N+](=O)[O-] RJC03701 Cc1ccc(cc1)S(=O)(=O)N=S(c2ccc(cc2)C(=O)O)c3ccc(cc3)C(=O)O BTB15076 c1cc(c(nc1)N2CCN(CC2)C(=O)/C=C/C(=O)O)C(F)(F)F SEW05900 c1cc(c(nc1)N2CCN(CC2)C(=O)c3ccco3)C(F)(F)F SEW05901 c1cc(c(nc1)N2CCN(CC2)C(=O)C3CCC3)C(F)(F)F SEW05902 COc1ccc(cc1)NC(=O)c2ccc(s2)c3ccccc3 SEW05906 c1c(cc(cc1Cl)Cl)NC(=O)CSc2[nH]c(=O)c(c(n2)C3CCCCC3)C#N RH01391 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)Nc4ccc(c(c4)Cl)F SEW05924 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)c4ccc(cc4)Cl SEW05926 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)c4cccc(c4)OC(F)(F)F SEW05928 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccccc2OC RH01373 CCCCc1ccc(cc1)NC(=S)N2CCC(CC2)C(=O)OCC RH01375 c1ccc(cc1)COc2ccc(cc2)n3c(nnc3S)c4ccco4 SPB07881 CCOC(=O)c1c(sc(n1)c2ccccc2)c3cc[nH]n3 SPB04632 CC(C)(C)OC(=O)N[C@@H](Cc1cccc(c1)F)C(=O)O SB02000 c1ccc2c(c1)c(cs2)CNC(=O)C3CCCCC3 PD00419 COC(=O)c1ccc(cc1)CSc2ccccc2N SEW05880 COc1cc(cc(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)C(F)(F)F SEW05895 c1ccc(c(c1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F)C(=O)O SEW05899 CCCCc1ccc(c(c1)C)NC(=O)COc2cc(c3c(c2)OC(CC3=O)(C)C)C RH01357 c1cc2c(cc1F)nc(cn2)c3ccc(s3)Br RH01384 Cc1c(ccc2c1OC(CC2=O)(C)C)OCc3ccccc3F RH01387 COC(=O)c1ccc(cc1)CSc2ccc(cc2)Cl SEW05904 c1ccc2cc(ccc2c1)C(=O)NNC(=O)c3ccc(o3)[N+](=O)[O-] RH01369 Cc1cc(cc2c1C(=O)CC(O2)(C)C)OCC(=O)O RH01371 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccc(cc2C)Cl RH01372 COc1ccc(cc1OC)CC(=O)NNC(=S)Nc2ccc(cc2)F S09968 CC(C)(C)c1ccc(cc1)c2nc(nn2c3ccccc3)O S14744 c1cc(c(cc1F)F)c2ccc(o2)/C=N/O CD10726 c1ccc(c(c1)C(=O)N/N=C/c2ccc3c(c2)OCO3)[N+](=O)[O-] BLT00020 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccccc2C(F)(F)F RH01376 COc1ccc2c(c1)c(=O)c3ccccc3o2 JFD03171 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OC[C@@H]4C(C[C@@H](O4)n5cc(c(=O)[nH]c5=O)I)O RJC03231 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CC(=O)Nc3c(ccs3)C(=O)OC GK03124 Cc1ccc(cc1)Sc2ccc(cc2)[N+](=O)[O-] RH01338 c1cc(ccc1C(=O)C2CCN(CC2)C(=O)Nc3ccc(cc3)Cl)Cl CD10001 COC(=O)c1c(ccs1)Oc2ccc(cc2N3C(=O)c4ccccc4C3=O)C(F)(F)F GK02198 COc1ccc(cc1)N2C(=O)CSC2=S S02024 c1cc(c(nc1)N2CCN(CC2)C(=O)c3cccs3)C(F)(F)F SEW05903 CCC(c1ccccc1)/C(=N/Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])/c3cc(ccc3OC)OC BLT00012 CCOC(=O)c1c(c2c(nc(nc2s1)SCc3ccccc3)c4ccccc4)N BTB15109 Cc1ccc(c(n1)[N+](=O)[O-])OCC(=O)O RH01378 c1ccc(cc1)C(=O)c2cccc(c2)NC(=O)c3cccnc3Oc4ccccc4 RH01379 CC(C)C(=O)Nc1[nH]c(=O)c2c(n1)n(cn2)[C@H]3CC([C@H](O3)COC(c4ccccc4)(c5ccc(cc5)OC)c6ccc(cc6)OC)OC(=O)C RJC03228 CCCc1cnc(nc1)N2CCCN(CC2)S(=O)(=O)c3cc(c(cc3C)Cl)C AW00858 CCCc1cnc(nc1)N2CCCN(CC2)C(=S)Nc3ccc(cc3)C AW00859 Cc1ccc(cc1)S(=O)(=O)OC[C@@H]2C(C[C@@H](O2)n3cnc4c3nc([nH]c4=O)NC(=O)C(C)C)O BTB14740 COC(=O)Cc1ccccc1Sc2ccccc2[N+](=O)[O-] BTB15083 CC(=O)OC[C@@H]1[C@H]([C@H]([C@@H](O1)n2c(=O)[nH]c(=O)cn2)OC(=O)C)OC(=O)C RJC03208 CSc1nnc(n1NC(=N)c2cccc(c2)C(F)(F)F)SC SPB01379 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)Nc3ccc(cc3)F)C(F)(F)F GK03125 Cc1cccc(c1)C(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SEW06094 COc1ccc(cc1NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F)Cl SEW06096 c1cc(c(cc1F)F)NC(=O)Nc2ccc(cc2F)F CD10243 c1cc(c(c(c1NC(=O)NC2CCSC2)Cl)Cl)Cl CD10284 Cc1ccc(cc1)S(=O)(=O)OC[C@@H]2C(C[C@@H](O2)n3cc(c(=O)[nH]c3=O)C)OC(=O)C BTB14738 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CO)O RJC03216 COc1cccc(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC BTB07458 C=CCNC(=S)NNC(=O)c1ccco1 JFD03125 CC(C#N)(c1ccccc1)Nc2ccc(cc2)Cl JFD03064 CC(C)C(C)(C#N)Nc1ccccc1 JFD03068 CCCCc1c(=O)c2cnn(c2[nH]c1O)c3ccccc3 JFD03066 CC(C#N)(c1ccc(cc1)F)Nc2ccccc2 JFD03067 CCCc1cnc(nc1)N2CCCNCC2 AW00852 c1ccc(cc1)C(CC(=O)O)CC(=O)Oc2ccccc2N3CCCC3 PD00445 c1ccc(c(c1)C(=O)NC2CCSC2)NC(=O)c3cccc(c3)Cl CD10385 Cc1cn(c(=O)[nH]c1=O)[C@H]2CC([C@H](O2)COS(=O)(=O)c3ccccc3)OC(=O)C BTB14739 c1ccc(cc1)C[C@H](C(=O)O)N SB02005 COc1ccccc1NS(=O)(=O)c2ccccc2[N+](=O)[O-] BTB15095 COC(=O)c1cc2c3ccccc3[nH]c2c(n1)C(F)(F)F SEW02470 c1cc(sc1)c2ccn(n2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F AW00845 CS/C(=N/c1ccc(cc1)Cl)/N.I JFD03127 CN(C)/C=C(\C#N)/c1ccccn1 CD11581 Cc1c(c(on1)C)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N SEW05934 c1ccc(cc1)C(CC(=O)NCc2csc3c2cccc3)CC(=O)O PD00447 c1cc2c(c(c1)NC(=O)c3c(nccn3)C(=O)O)CCCC2 PD00441 c1ccc2c(c1)-c3ccccc3C(C2O)O BTB10563 CC(C)(C)OC(=O)Cn1ccc(=O)[nH]c1=O BTB15121 Cc1cc(cc2c1C(=O)CC(O2)(C)C)OCc3ccc(cc3Cl)Cl RH01361 COc1ccc(cc1)c2c(c(nc(n2)SCc3ccccc3)SC)C#N BTB15108 CC(C)c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PD00451 CC(C)c1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)C(C)C BTB07741 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW05936 CC(C)(C)CC(C)(C)NC(=O)c1cccc2c1-c3ccccc3C2=O JFD03213 c1ccc2c(c1)-c3c(cccc3C(=O)N(CCO)CCO)C2=O JFD03216 c1cc(ccc1C(F)(F)F)Oc2ccc(cn2)N BTB04659 c1cc(c(cc1Cl)Cl)/C=N/OCc2cc(sc2Cl)Cl CD11585 Cc1ccc(cc1Cl)NC(=O)CC(CC(=O)O)c2ccccc2 PD00456 Cc1c(nnn1c2ccc(cc2F)F)C(=O)C CD09885 Cc1c(cnn1c2ccccc2)c3ccnc(n3)NS(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F CD09915 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)Nc4cccc(c4)Cl SEW05922 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)NC(=O)c4cccs4 SEW05925 CC(C)(C)c1ccc(cc1)NC(=O)N2CCOCC2 S11993 c1cc(ccc1/C=C\2/C(=O)NC(=S)S2)O BTB01734 Cc1cc(cc(c1OCC(CNCCNc2nccc(n2)C(F)(F)F)O)Br)Cl AW00808 Cc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)C BTB07742 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)O KM03993 CCCS(=O)(=O)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06208 c1ccc2c(c1)cccc2CSCC(=O)NNC(=S)NC3CCCCC3 RH01651 c1cc2cccc3c2c(c1)C(=O)N(C3=O)CC4CCCO4 PHG00949 COc1ccc(cc1)NC(=S)NNC(=O)CSCc2cccc3c2cccc3 RH01649 CC(C(C)(C)C)NC=C(C#N)C#N CD11593 c1cc(c(cc1[N+](=O)[O-])CC(CO)C#N)N2CCCCC2 RH01640 CCc1ccc(cc1)N2C(=O)CSC2=S S03806 c1ccc2c(c1)cc3ccccc3c2/C=C/4\C(=O)OC(=N4)c5ccccc5I PD00474 CC(=O)NCc1c(cccc1Cl)Sc2ccc(cc2)Cl CD11893 CC1(OC(=O)C(=C2CCCN2)C(=O)O1)C CD11922 c1cc(ccc1C(F)(F)F)NC(=O)c2c(nccn2)C(=O)O PD00074 Cn1c(ccn1)N2C(=O)c3ccccc3C2=O GK03123 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2ccc3c(c2)non3 KM08482 CS(=NC(=O)c1cc(cnc1)C#Cc2ccccc2)(=O)c3ccccc3 KM08484 Cn1c(nnc1SCc2ccccc2Cl)c3cc(cnc3)C#Cc4ccccc4 KM08507 c1cc(c(cc1F)F)C(=O)C2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] SEW05893 COc1cc(cc(c1)NC(=O)Nc2cc(cc(c2)Cl)Cl)C(F)(F)F SEW05896 Cc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC)Cl BTB07693 Cc1cc(cc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC)C)Br BTB07703 C/C(=C\C(=O)c1cccc(c1F)Cl)/N(C)C CD12024 CN(C)/C=C(\C#N)/C(=O)c1cccc(c1)C(F)(F)F CD12056 CN(C)/C=C/C(=O)c1cc(ccc1SC)C(F)(F)F CD12061 Cc1cc(c(cc1Cl)C)S(=O)(=O)NCCNc2nccc(n2)C(F)(F)F AW00819 Cc1csc2c1[nH]c(=O)n(c2=O)CCSc3ccc(cc3)Cl S13664 CCCCc1ccc(cc1)n2c(nnc2S)CSCc3cccc4c3cccc4 RH01678 CC(CN1C(=O)c2cccc3c2c(ccc3)C1=O)O PHG00959 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OC)Cl)Cl BTB07692 C#Cc1ccc(cc1)NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB08524 COc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC)OC BTB07694 c1cc(cc(c1)NC(=O)N2CCSCC2)C(F)(F)F BTB04469 c1ccc(cc1)C(=O)NCCNc2nccc(n2)C(F)(F)F AW00814 c1ccc(cc1)NC(=O)N2CCCN(CC2)Cc3c(cccc3Cl)F AW00817 Cc1ccc(cc1)S(=NC(=O)c2cc(cnc2)C#Cc3ccccc3)(=O)C KM08511 c1cc2c(cc1[N+](=O)[O-])C(=O)N(C2=O)CNc3cc(cc(c3)C(F)(F)F)C(F)(F)F S05533 COc1ccc(cc1)n2c(nnc2S)CSCc3cccc4c3cccc4 RH01677 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)Cc4cccnc4)[N+](=O)[O-] PHG00990 c1ccc(cc1)/C=N/c2ccc(cc2C(F)(F)F)Br BTB02730 COc1cc(cc(c1)NC(=S)Nc2ccccc2OC(F)(F)F)C(F)(F)F SEW05914 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)/N=C/c4ccccc4O SEW05915 CCOC(=O)c1c(c(c(n1c2ccc(cc2)OC)C(=O)OCC)O)O BTB10018 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)O SP00293 c1ccc2c(c1)cccc2CSCC(=O)NNC(=S)NC3CC4CC3C=C4 RH01681 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3ccc(cc3OC)Br RH01683 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)/N=C/c4cc(ccc4O)Cl SEW05916 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)OCC)N)c3ccco3 KM03459 CC1CC(CC(C1)(C)C)NC(=S)NCc2csc3c2cccc3 PD00444 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cccc2F)F)OC)Br)[N+](=O)[O-] BTB07704 Cc1cc(c(c(c1)C)NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC)C BTB07706 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)OC)Br)[N+](=O)[O-] BTB07708 c1cc(cc(c1)Br)N2C(=O)CSC2=S S06616 c1ccc(cc1)CN2CCC(CC2)Nc3nccc(n3)C(F)(F)F AW00821 c1cc(cnc1)NC(=S)NCCNc2nccc(n2)C(F)(F)F AW00831 c1ccc2c(c1)cccc2CSCc3nnc(n3c4cccc(c4)C(F)(F)F)S RH01676 CC(=O)OCC(Cn1cnc2c1c(=O)n(c(=O)n2C)C)OC(=O)C RJC03218 c1ccc2c(c1)cc(s2)C(=O)Nc3cc(cc(c3)Cl)Cl BTB04207 Cc1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4ccc(cc4F)F RJC03524 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl)F CD06867 c1ccc(cc1)c2csc3c2c(ncn3)n4ccc(n4)C(F)(F)F AW00840 c1cc(ccc1CN2CCCN(CC2)C(=O)Nc3ccc(cc3)Cl)F AW00843 c1cc(sc1)c2ccn(n2)c3nccc(n3)C(F)(F)F AW00844 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OC4C[C@@H](O[C@@H]4CO)n5cnc6c5ncnc6NC(=O)c7ccccc7 RJC03225 c1ccc(cc1)COC(=O)N2CCC[C@@H]2C(=O)O SB02004 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)/N=C/c4cc(cc(c4O)Br)Br SEW05917 c1ccc(cc1)Sc2ccc(c(n2)Sc3ccccc3)/N=C/c4cc(cc(c4O)Cl)Cl SEW05918 COc1cc2c(cc1OC)C(NC(=O)C2)c3ccccc3Cl JFD03611 CC(=O)c1ccc(s1)c2cc(n(n2)C)C(F)(F)F KM03660 c1cc2c(cc1Cl)c3cc(ccc3n2CC(CN4CCCC4)O)Cl JFD03612 c1cc(ccc1CNC(=S)NNc2ccc(cc2)S(=O)(=O)N)F PD00433 c1ccc(cc1)C(=S)NCc2csc3c2cccc3 PD00438 Cc1ccc(cc1)S(=O)(=O)NCc2csc3c2cccc3 PD00452 c1ccc2c(c1)cc(s2)C(=O)N3CCCCC3 BTB04216 COc1cc(cc(c1O)/C=N/c2ccc(nc2Sc3ccccc3)Sc4ccccc4)Br SEW05919 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(nc2Sc3ccccc3)Sc4ccccc4 SEW05920 c1ccc(cc1)CN2CCC(CC2)NC(=S)Nc3cccnc3 AW00833 c1ccc(cc1)C(c2ccccc2)N3CC(C3)C(=O)O KM10090 c1c(c(=O)[nH]c(=O)n1[C@H]2C[C@@H]([C@H](O2)CO)O)Br RJC03234 c1ccc(cc1)C(=O)OC2CC2(Cl)Cl RJC03719 c1ccc(cc1)C2(CC2(Br)Br)c3ccccc3 RJC03723 CC(C)C\1C(NC(C/C1=N/O)c2ccccc2)c3ccccc3 RJC03604 CC\1C(NC(C/C1=N/O)c2ccc(cc2)OC)c3ccc(cc3)OC RJC03607 COc1ccc(cc1)C2=NNC(=O)CC2 RH01336 c1cc2c(cc1OCC(CN3CCCN(CC3)c4nc5ccc(cc5s4)Cl)O)OCO2 AW00837 c1cc(ccc1[N+](=O)[O-])OCC(CN2CCCN(CC2)c3nc4ccc(cc4s3)Cl)O AW00841 CC(C)(C)c1ccc(cc1)NC(=O)N2CCCN(CC2)Cc3ccc(cc3)F AW00842 c1ccc2c(c1)c(cs2)CNC(=O)c3c(nccn3)C(=O)O PD00453 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)Nc5cccc(c5)Cl RH01723 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OC[C@@H]4C(C[C@@H](O4)n5cnc6c5[nH]c(nc6=O)N)O BTB14725 CCCC\1C(NC(C/C1=N/O)c2ccccc2)c3ccccc3 RJC03602 CC\1C(N(C(C/C1=N/O)c2ccccc2)C)c3ccccc3 RJC03603 c1ccc(cc1)NC(=O)N2CCCN(CC2)Cc3ccc(cc3)F AW00847 Cc1cn(c(=O)[nH]c1=O)[C@H]2C[C@@H]([C@H](O2)CO)OS(=O)(=O)c3ccccc3 RJC03236 CC(C)(C)c1cc(c(s1)C#N)N GK02506 CCOc1ccsc1C(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N GK02540 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COC(c3ccccc3)(c4ccc(cc4)OC)c5ccc(cc5)OC)O RJC03217 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OCC(CO)NC(=O)OCC4c5ccccc5-c6c4cccc6 BTB14729 Cc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK03068 Cc1ccc(cc1Cl)NC(=S)Nc2ccc(c(c2)Cl)C BTB04725 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2N CD10046 COc1cc(cc(c1)OC)C(=O)NNC(=S)Nc2cccc(c2)Cl BLT00092 Cc1cc(cc2c1C(=O)CC(O2)(C)C)OCc3c(cccc3Cl)F RH01365 COc1cc(cc(c1OC)OC)N2C(=O)CSC2=S S03517 CC(C)c1ccc(cc1)NC(=S)NNC(=O)c2cc(cc(c2)OC)OC BLT00096 COC(=O)C/C(=C(\C#N)/C(=O)OC)/N BTB08631 c1ccc2c(c1)C(=O)C(=C(C#N)NCCC3=CCCCC3)C2=O S14004 CC(C)C[C@H](C(=O)O)NC(=O)[C@H]1CCCN1C(=O)OCc2ccccc2 JFD03176 CC(C)C[C@@H](C(=O)O)NC(=O)[C@H]1CCCN1C(=O)OCc2ccccc2 JFD03177 CC(C)(C)C(=O)Nc1cc(c(cc1Cl)Cl)Cl JFD03119 CCOC(=O)c1c(c2cc(ccc2s1)OC)Cl BTB10141 CC(C)(C)C(=O)Nc1ccc(nc1Sc2ccccc2)Sc3ccccc3 SEW05931 COC(CNC(=O)C(=O)Nc1ccc(cc1Cl)Cl)OC CD11584 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl)CC(=O)O PD00448 c1ccc(cc1)Cn2c(=O)c3c([nH]cn3)n(c2=O)c4cccc(c4)Cl KM09316 c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4cccc(c4)F KM09342 CCOC(=O)C1CCC(N1C(=O)Nc2ccc(cc2)Cl)C(=O)OCC KM09504 COc1ccccc1N2CCN(CC2)C(=S)Nc3ccc(cc3Cl)Cl SEW06128 c1cc(ccc1/C=N/OCc2cc(sc2Cl)Cl)[N+](=O)[O-] CD11591 c1cc(cc(c1)F)Nc2n[nH]c(=S)s2 K00098 COc1ccc(cc1)/C=N/NC(=S)Nc2ccc(cc2)F K00100 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3ccccc3SCCC#N CD03866 c1ccc(cc1)n2c(nnn2)c3cnn(c3C(F)(F)F)c4ccc(cc4)F JFD03617 Cc1ccc(cc1)n2c(nnn2)/C=C/N3CCN(CC3)c4cccc(c4)C(F)(F)F JFD03619 C1CCN(CC1)C(=O)C23CC4CC(C2)CC(C4)C3 SEW06092 CC(C)(C)OC(=O)NC(Cc1ccccc1)C(=O)N JFD03161 c1ccc(cc1)C(=O)Nc2ccc(c(c2)Cl)F RF04239 c1ccc(c(c1)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)Cl RF04807 c1ccc(cc1)c2c(cc(n(c2=O)c3ccccc3)c4ccc(cc4)F)O RJC03581 CC(C)c1cc(c(c(=O)n1c2ccc(cc2)Cl)c3ccccc3)O RJC03583 c1ccnc(c1)c2cnoc2N CD11596 c1ccc(cc1)CC(c2ccccc2)N3CNC(=S)NC3 ML00427 Cc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC)C BTB07707 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)COc3ccc(cc3)OC SP00452 COc1ccc(cc1)OCc2nc(cs2)c3ccc4c(c3)OCCCO4 SP00453 Cc1ccc(cc1)c2csc(n2)COc3ccc(cc3)OC SP00456 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)OC)Br)Cl BTB07753 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2)OCc3ccccc3)C#N JFD03268 c12c(sc(=O)s1)sc(=O)s2 RJC03593 CSc1c(sc(=S)s1)SC RJC03594 c1ccc(cc1)c2c(nc([nH]2)S)c3ccccc3 JFD03142 CCOC(=O)CSc1ccc2ccccc2n1 JFD03225 c1ccc2c(c1)-c3ccc(cc3C2=O)C(=O)c4ccccc4Br JFD03226 c1ccc2c(c1)CC(=O)NC2c3ccc(cc3)Cl JFD03229 c1cc(cc(c1)F)CSCc2c(cccc2Cl)F CD07577 COc1ccccc1NC(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F SEW06218 Cc1cc(cc2c1C(=O)CC(O2)(C)C)OCC(=O)Nc3ccc(cc3)Br RH01358 c1ccc(cc1)C(=O)c2cccc(c2)NC(=O)c3ccc(cc3)[N+](=O)[O-] RH01359 CN1CCC2(C(C1)N=NN2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)N4CCOCC4 CD04659 CC(C)(C)OC(=O)NC(Cc1ccccc1)C(=O)NC JFD03162 CC(C)(C)OC(=O)NC(Cc1ccccc1)C(=O)NCc2ccccc2 JFD03164 c1cc(ccc1C#N)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06102 COc1ccccc1N2CCN(CC2)C(=O)Nc3cccc(c3)Cl SEW06105 COc1cccc(c1C(=O)NN)OC CD11636 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)Cl CD11652 CC1=C(C(NC(=O)N1)c2ccc(cc2)OC)C(=O)C JFD03235 c1ccc2c(c1)ccc(c2c3c4ccccc4ccc3OC(=O)c5ccc(cc5)Cl)OC(=O)c6ccc(cc6)Cl JFD03237 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccnn2C GK03071 Cn1c(ccn1)N2C(=O)CCC2=O GK03072 c1cn(c(=O)nc1N)[C@H]2[C@H]([C@@H]([C@H](O2)CO)O)O BTB15125 CC(C)(C)NC(=O)[C@@H]1Cc2ccccc2CN1 SB01999 Cc1cc(nc(n1)NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)C BTB07754 CCCCc1c(cc(n(c1=O)Cc2ccccc2)c3ccccc3)O RJC03582 CCc1cc2c(cc1c3csc(n3)c4ccccc4)C(CCC2(C)C)(C)C SEW06098 CC(C(=O)N)NC(=O)OC(C)(C)C JFD03165 CCNC(=O)C(C)NC(=O)OC(C)(C)C JFD03167 CC(C(=O)NCc1ccccc1)NC(=O)OC(C)(C)C JFD03168 CC(c1n[nH]c(=S)n1CC=C)Oc2ccc(cc2)Cl JFD03202 CC(c1n[nH]c(=S)n1c2ccccc2)Oc3ccc(cc3)Cl JFD03203 CCn1c(n[nH]c1=S)C(C)Oc2ccc(cc2)Cl JFD03212 Cc1c(ccc2c1OC(CC2=O)(C)C)OCc3cc(cc(c3)C(F)(F)F)C(F)(F)F RH01389 Cc1ccc(c(c1)CSc2[nH]c(=O)c(c(n2)C3CCCCC3)C#N)C RH01393 CCCCSc1nnc(s1)S JFD03146 CC1(CCC(c2c1ccc(c2)c3csc(n3)c4ccc(cc4)C(C)(C)C)(C)C)C SP00389 CC(=O)NCc1c(cccc1N(C)C)N(C)C CD09518 Cc1ccc(cc1)N/C(=N/c2ccc(cc2)C)/SC JFD03238 C=CCn1c(n[nH]c1=S)Cc2ccc(c(c2)Cl)O JFD03199 Cc1cc(ccc1OCc2n[nH]c(=S)n2CC=C)Cl JFD03204 c1ccc(cc1)C(=O)NCc2csc3c2cccc3 PD00420 c1ccc2c(c1)c(cs2)CNC(=O)c3cccs3 PD00421 CC(C)(C)c1ccc(cc1)C(=O)NCc2csc3c2cccc3 PD00422 CC1C(N(C(C(C1(c2ccc(cc2)F)O)C)c3ccccc3)C)c4ccccc4 RJC03606 c1cc(ccc1N2C3(C4CC(C3N=N2)C5C4C=CC5)N6CCOCC6)[N+](=O)[O-] CD04643 c1cc(c(c(c1)F)C#N)NC(=O)c2ccc(cc2)Cl CD05874 CC1C(OCCN1CN2C(=O)c3ccccc3C2=O)c4ccccc4 NS00008 Cc1ccccc1/C=C/c2c[nH]c3c2cccc3 RJC03734 Cc1cc(c(c(c1)C)CSCC(=O)NNC(=O)Cc2ccccc2)C BLT00129 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nc(on2)CN3CCOCC3.Cl CD04490 Cc1ccc2cc(c(cc2c1)C)C JFD03643 c1ccc(cc1)c2c(nnn2c3cccc(c3)C(F)(F)F)C(=O)O CD04494 Cc1c(c(c(c(c1C)C)C(=O)C2CCN(CC2)C(=O)C)C)C CD10667 c1ccc(cc1)S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)Cc3cc(cc(c3)NS(=O)(=O)c4ccccc4)C(F)(F)F CD10713 COCCCNC(=O)C12CC3CC(C1)CC(C3)C2 CD08950 CCCCCSc1nnc(s1)S JFD03151 CCC/N=c\1/n(c(=O)ss1)CCC.Br RH01363 CCCCCCCCCCCCSc1[nH]cnn1 JFD03155 Cc1ccc(c(c1)COc2cc(c3c(c2)OC(CC3=O)(C)C)C)C RH01366 CCCCCCCCSc1[nH]cnn1 JFD03158 Cc1cc(c2ccccc2n1)NNC(=O)c3ccc(o3)[N+](=O)[O-] RH01370 Cc1cc(c(c(c1)C)NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)C BTB07745 c1cc(c(c(c1)Cl)CC(=O)NC(=O)Nc2ccc(cc2)Cl)F CD06475 c1ccnc(c1)c2nc(cc(n2)O)C(F)(F)F CD06646 c1ccc(cc1)NNC(=S)Nc2cccc(c2Cl)Cl K00050 COc1ccc(cc1)CC(=O)NNC(=S)Nc2ccccc2 JFD03205 Cc1ccc(cc1)C#Cc2ccc(cc2)C JFD03642 Cc1cnc(c(c1OC)C)CS(=O)c2[nH]c3cc(ccc3n2)OC KM07219 C/C(=N\NC(=O)N)/c1c(cccc1F)F CD04764 C1C2CC(C1C=C2)NC(=S)N CD04880 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3ccccc3C(=O)O)C(F)(F)F GK02211 Cc1cc(n(n1)c2c(cc(cc2Cl)Cl)Cl)C CD10090 CCOC(=O)C1CCN(CC1)C(=S)Nc2cccc(c2)Cl RH01396 CCCCCCCCCCCCSc1nnc(s1)S JFD03150 CCCCSc1[nH]cnn1 JFD03153 Cc1cc(cc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)C)Br BTB07748 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cccc2Cl)Cl)OC)Br)Cl BTB07750 COc1c(cc(c(c1C(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl)OC)Br)Cl BTB07752 Cc1c(c(no1)c2ccccc2)c3csc(n3)C SP00411 c1cc(ccc1/C(=N/OCc2cc(cc3c2OCOC3)Cl)/N)Cl CD06089 Cc1ccc(cc1)NS(=O)(=O)c2ccsc2C(=O)OC GK03165 c1ccc(cc1)n2c(nnc2S)Cc3nnc(n3c4ccccc4)S JFD03149 CC(c1n[nH]c(=S)n1CC=C)Oc2ccccc2c3ccccc3 JFD03211 Cc1ccc(cc1)NC(=S)Nc2cc(cc(c2)C)C K00006 Cc1cc(cc(c1)NC(=S)Nc2cccc(c2C)Cl)C K00005 COc1cc(cc(c1OC)OC)/C=N/NC(=O)c2ccccc2[N+](=O)[O-] BLT00017 Cc1c2c(cc(s2)C(C)(C)C)sc1C(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N GK03056 Cc1ccc(cc1)S(=NS(=O)(=O)c2ccc3c(c2)CCN3C(=O)C)(=O)C KM05470 CN(n1cnc2ccccc2c1=O)S(=O)(=O)c3cc(sc3Cl)Cl CD09572 c1cc(sc1)CNS(=O)(=O)CS(=O)(=O)NCc2cccs2 CD09636 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Br)Br)Br)OC)Br)Cl BTB07759 Cc1ccc(cc1)n2c(nnn2)c3cnn(c3C(F)(F)F)c4ccc(cc4)F JFD03618 COC(=O)CCN1CCc2c1ccc(c2)/N=N/c3ccc(cc3)Br JFD03627 CC(=O)Nc1ccn(c(=O)n1)[C@H]2CC([C@H](O2)COC(c3ccccc3)(c4ccc(cc4)OC)c5ccc(cc5)OC)OC(=O)C BTB14727 CC(=O)OCC(COC(=O)C)NC(=O)OCC1c2ccccc2-c3c1cccc3 BTB14728 Cc1ccc(cc1C)NC(=O)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl BLT00072 c1ccc(cc1)C(CC(=O)NCc2ccco2)CC(=O)O PD00454 Cc1ccc(cc1NC(=O)N2CCN(CC2)c3ccccc3OC)F SEW06101 COc1ccccc1N2CCN(CC2)C(=O)Nc3cc(ccc3OC)Cl SEW06106 c1cc(oc1)Cn2c(nnc2S)c3ccc(cc3Cl)Cl SPB06040 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccc(cc2)Br RH01397 c1ccc2c(c1)c(=O)c3cc(ccc3o2)OCCCCC(=O)O JFD03169 Cc1ccc(cc1)NC(=O)c2cccc3c2-c4ccccc4C3 BTB15086 CCOC(=O)CCCCOc1ccc2c(c1)c(=O)c3ccccc3o2 JFD03170 COc1ccc(cc1OC)CCNC(=S)NCCc2ccccc2 CD01627 c1ccc2c(c1)CC(=C2)N3CCN(CC3)c4ccc(cc4)Cl JFD03622 COC(=O)CCN1CCc2c1ccc(c2)/N=N/c3ccc(cc3)[N+](=O)[O-] JFD03624 Cc1c(c(sc1C(=S)N)SC)C(=O)C KM04561 CCOC(=O)NNC(=O)NCCCCCCNC(=O)NNC(=O)OCC RJC03753 COc1ccc(cc1OC)S(=O)(=O)N(CCC(=O)N)Cc2ccco2 KM09282 c1ccc(cc1)Cc2c(c3ccccc3oc2=O)Cl RJC03767 COC(=O)c1c(=O)c2cscc2[nH]c1C(=O)OC GK02293 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD03853 c1ccc(cc1)Oc2ccc(cc2)NC(=S)Nc3cccc(c3)C(F)(F)F CD03753 CCCCNC(=S)Nc1ccc(cc1)C(C)C CD03739 c1cn2c(nc1=O)O[C@@H]3[C@H]2O[C@@H]([C@H]3O)CO RJC03786 Cc1cc(c(c(c1)C)CC(=O)NNC(=S)Nc2cccc(c2)SC)C BLT00106 CC(Cc1ccc(cc1)C(C)(C)C)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00087 CS(=O)(=O)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06210 CC(=O)OCC(COC(c1ccccc1)(c2ccc(cc2)OC)c3ccc(cc3)OC)NC(=O)OCC4c5ccccc5-c6c4cccc6 BTB14730 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3ccc(c(c3)Cl)Cl SP00363 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl SEW06108 Cc1c(cccc1Cl)NC(=O)N2CCN(CC2)c3ccccc3OC SEW06110 COc1ccc(cc1OC)S(=O)(=O)N(CC#N)Cc2ccco2 KM09252 COc1ccc(cc1OC)C(=O)NCc2ccco2 KM09256 CC(=O)Nc1cc2ccccc2oc1=O PHG00456 c1ccc2c(c1)c(cc(n2)O)C(=O)O RF00768 CC(C)c1ccc(cc1)S(=O)(=O)N2CCC(CC2)c3ccccc3OC RH01642 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3ccc(cc3)OC(F)(F)F RH01615 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3ccc(cc3F)F RH01616 COC(CNC(=O)C(=O)Nc1ccccc1Oc2ccc(cc2Cl)Cl)OC CD11666 COC(CNC(=O)C(=O)Nc1cccc(c1)C(F)(F)F)OC CD11669 COc1cc(cc(c1)OC)N2C(=O)c3c(nccn3)C2=O PD00080 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc(c2C#N)F CD05875 c1ccc2c(c1)c(cs2)CNC(=S)Nc3ccc(cc3Br)F PD00417 CNc1cccc2c1C(=O)c3ccccc3C2=O BTB15210 COc1ccccc1N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl SEW06116 c1cc(c(nc1)N2CCN(CC2)C(=O)Nc3ccc(cc3F)F)C(F)(F)F SEW06117 COC(=O)CNS(=O)(=O)c1ccsc1C(=O)OC GK03166 Cc1ccc(cc1)CNC(=S)NN(C)C PD00443 COC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)C3CCCN3C(=O)OCc4ccccc4 JFD03178 c1ccc2c(c1)cccc2CSCc3nnc(n3c4ccccc4Cl)S RH01684 Cc1cccc(c1)n2c(nnc2S)CSCc3cccc4c3cccc4 RH01685 Cc1ccc(c(c1)NC(=S)Nc2cccc(c2)F)C S04596 c1ccc(c(c1)C2=NCCCN2)SCc3c(cccc3F)F.Br CD05710 CCc1cccc(c1NC(=O)c2cccc(c2)Cl)C(C)C CD06351 CCOC(=O)C(c1ccc(c(c1)OC)NC(=O)NC(C(F)(F)F)(C(F)(F)F)Oc2ccc(cc2)F)(C(F)(F)F)O RJC03644 Cc1ccc(cc1)c2csc(n2)CC#N SP00555 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2ccc(c(c2)F)F SP00560 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2ccc3c(c2)OCCCO3 SP00561 c1ccc2c(c1)C(=O)C(=C(C2=O)Cl)Oc3ccccc3Cl JFD03184 c1ccc(cc1)C(=O)Oc2cccc3c2C(=O)C=CC3=O JFD03185 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4c(cc(cc4Cl)C(F)(F)F)Cl SP00592 Cc1cc(cc(c1)NC(=S)Nc2cc(cc(c2)C)C)C K00028 c1ccc(c(c1)OCc2nc(cs2)c3ccc(cc3)C#N)Cl SP00595 c1ccc(c(c1)OCc2nc(cs2)c3ccc(cc3)[N+](=O)[O-])Cl SP00597 Cc1cccc(c1)N(C2=NCC(S2)(C)C)C(=O)Nc3cccc(c3)Cl RJC03649 CN(C(=O)CN1CCOCC1)n2cnc3ccsc3c2=O CD11816 c1ccc(cc1)c2ccc(cc2)C(=O)CSc3c4ccccc4nc(n3)SCC(=O)c5ccc(cc5)c6ccccc6 PD00468 c1ccc(cc1)c2ccc(cc2)C(=O)CSc3[nH]c(=O)c4ccccc4n3 PD00469 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])C#N JFD03267 c1ccc(c(c1)OCc2nc(cs2)c3ccc4c(c3)OCCCO4)Cl SP00584 Cc1ccc(c(c1)C)c2csc(n2)COc3ccccc3Cl SP00585 Cn1c(ccn1)NC(=O)c2ccccc2C(=O)O GK03118 CC(C)Cc1ccc(cc1)c2cc(c(s2)C(=O)N)NC(=O)c3ccc(cc3)Cl GK03116 Cc1ccc(cc1)SCCS(=O)(=O)c2ccc(cc2)F KM08610 COc1ccccc1N2CCN(CC2)C(=S)c3ccccc3OC(F)(F)F SEW06129 c1cc(ccc1/N=C/c2cc(cc(c2O)Cl)Cl)S(=O)(=O)/N=C/c3cc(cc(c3O)Cl)Cl K00088 C=CNC(=S)NNC(=O)COc1ccccc1 RH01342 c1ccc(cc1)n2c(nnn2)c3cnoc3c4ccc(c(c4)F)F JFD03623 c1cc(ccc1Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl CD04029 CN(C)c1c(cc(cc1F)C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F CD12063 Cc1ccc(c(c1)C)c2csc(n2)c3ccc(cc3)C(C)(C)C SP00368 c1cc(oc1)C(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SEW06093 COc1ccc(cc1)C(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SEW06095 c1c(cncc1C(=O)O)C#CCC2CCCCC2 KM08907 CCOC(=O)c1cnc2c(c1NNc3ccccc3)c(nn2C)C KM08910 COc1cccc(c1)C(=O)CC#N KM08917 CC(C#N)(c1cccnc1)Nc2ccccc2 JFD03190 CN1CCN(CC1)c2cc(nc3c2cccc3)c4ccncc4.Br.Br JFD03240 c1cc(cc(c1)N/N=C/c2cc(cc(c2O)Cl)Cl)C(F)(F)F DP02041 Cc1ccc(cc1)c2csc(n2)COc3ccccc3Cl SP00596 Cc1c2ccccc2sc1c3csc(n3)COc4ccccc4Cl SP00598 c1ccc(c(c1)OCc2nc(cs2)c3cccc(c3)F)Cl SP00599 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccc3OC SEW06099 COc1ccccc1N2CCN(CC2)C(=O)Nc3ccc(cc3)F SEW06100 CC(Cc1ccccc1)(C#N)Nc2ccc(cc2)Cl RJC03587 c1cc(ccc1C(=O)CCC(=O)c2ccc(cc2)F)F CD08839 c1ccc2c(c1)CC(=O)NC2c3ccc(cc3)Br JFD03230 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)CCC(=O)O)Cl GK03171 c1cc(sc1)/C=C/C(=O)Nc2ccc(c(c2)C(=O)O)N3CCOCC3 CD05899 c1cc(ccc1C(=O)/C(=N/Nc2ccc(cc2)Cl)/C#N)OC(F)(F)F KM04883 C(C(=O)O)Sc1nnc(s1)S BTB12604 c1cc2c(c(c1)F)C(=O)NC(N2)c3cc(cc(c3O)Cl)Cl BTB04354 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])/C=C/C(=N/O)/N CD05552 c1cc(cnc1)c2ccc(s2)C#CCO KM07808 CC1CCCC(N1c2ccc(cc2C(=O)O)NC(=O)c3cc(ccc3Br)OC)C CD07043 COc1ccc(cc1)C(c2ccccc2)(c3ccc(cc3)OC)OCC(COC(c4ccccc4)(c5ccc(cc5)OC)c6ccc(cc6)OC)NC(=O)OCC7c8ccccc8-c9c7cccc9 BTB14731 COC(=O)CCN1CCc2c1ccc(c2)/N=N/c3ccc(cc3)C(F)(F)F JFD03626 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2nc(cs2)c3ccc(c(c3)F)F SP00608 c1ccc(cc1)c2c(nnn2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)O CD04516 Cc1c2ccccc2sc1c3csc(n3)c4ccc(cc4)C(C)(C)C SP00374 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3cccc(c3)F SP00385 Cc1c2cc(ccc2sc1c3csc(n3)c4ccc(cc4)C(C)(C)C)Cl SP00378 c1c(c(sc1Cl)Cl)CN2CCSCC2 CD11568 COCCCNC(=S)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06229 CCOC(=O)c1cc(=O)c2cc(ccc2o1)Cl GK03126 CN(C)c1ccc(cc1C(=O)O)NC(=O)c2ccc(cc2)Cl CD06988 Cc1c(c(c(c(c1C)C)CO/N=C/c2ccccc2SC(C)(C)C)C)C CD07339 CC1CC(CN(C1)c2ccc(cc2C(=O)O)NC(=O)c3ccc(cc3)Cl)C CD07222 COc1ccccc1C(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK03078 Cc1nnc(n1c2ccc(cc2)OCc3ccccc3)S SPB07880 c1ccc(cc1)COc2ccc(cc2)NC(=S)NNC(=O)c3ccco3 SPB07858 CN(C)CC#Cc1cc(cnc1)C(=O)NN KM08392 Cc1ccc(cc1)S(=NS(=O)(=O)c2c(c(cs2)C(=O)OC)OC)(=O)C KM08428 Cc1cc(cc(c1)NC(=S)Nc2ccc(cc2)Cl)C K00009 Cc1cccc(c1C)/N=C/c2cc(cc(c2O)Cl)Cl K00011 CC(C)c1cc(c(c(c1)C(C)C)S(=O)(=O)OC[C@@H]2C(C[C@@H](O2)n3cnc4c3nc([nH]c4=O)NC(=O)C(C)C)O)C(C)C BTB14741 CCOC(=O)c1c(n[nH]c1/N=C/c2ccccc2[N+](=O)[O-])C JFD03607 CC(=O)/C(=C(/c1ccccc1)\N)/C(=O)OC CD06937 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)C(F)(F)F SP00387 CC(C)(C)OC(=O)N1CCN(CC1)CCNS(=O)(=O)c2ccc(cc2)Cl KM08239 CCCS(=O)(=O)C(C#N)c1ccccc1[N+](=O)[O-] KM08263 Cc1cc(ccc1N2C(=O)CC(C2=O)Sc3ccccc3N)Cl K00042 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)C(C)C)C K00043 Cc1c(c(c2c(c1C)[nH]c(n2)SCc3nc(no3)c4ccc(cc4)Cl)C)C CD04426 c1ccc(c(c1)/C=N/NC(=O)CC#N)O DP00079 c1cc(sc1)c2c(c(c(o2)N)c3ccc(cc3)C#N)C#N CD09249 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3ccc(cc3)Cl)C(F)(F)F GK03069 Cn1c(ccn1)NC(=O)CC#N GK03073 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccc(cc2)F RH01398 COc1ccc(cc1)C(=O)/C(=C/c2ccc(cc2)O)/C#N KM05987 CCCCc1ccc(c(c1)C)NC(=O)NCc2csc3c2cccc3 PD00440 CN1c2ccccc2-c3c(c(sc3C(=O)O)SC)S1(=O)=O KM03766 Cc1c(csc1S(=O)(=O)NNC(=O)C)S(=O)(=O)c2ccc(cc2)Cl KM03929 Cc1cc(cc(c1N2CCSCC2)C)[N+](=O)[O-] CD08207 CCOC(=S)SCc1cc(cc(c1)Br)Br CD08520 CC(C)(C)c1ccc(c(c1)[N+](=O)[O-])n2cccc2 CD08755 c1c(cnc(c1Cl)N2CCC(CC2)C(=O)NN)C(F)(F)F KM08264 c1cc(oc1)C(=O)NNC(=S)Nc2ccc3c(c2)OCCO3 SPB07860 c1cc(oc1)c2nnc(n2c3ccc4c(c3)OCCO4)S SPB07883 Cc1ccc(cc1)S(=O)(=O)Nc2ccc-3c(c2)Cc4c3ccc(c4)Br JFD03615 Cc1ccc(c(c1)C)c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F SP00427 c1ccc2c(c1)ccc3c2C(=O)CCC3 JFD03646 c1ccc(cc1)c2ccnc3n2nc(c3/N=N/c4ccccc4)N JFD03194 CCCCCCSc1[nH]cnn1 JFD03152 c1[nH]c(nn1)SCCCCSc2[nH]cnn2 JFD03156 c1[nH]c(nn1)SCCCCCCSc2[nH]cnn2 JFD03157 COc1ccc(cc1)n2c(nnc2SCC(=O)c3ccc(cc3)[N+](=O)[O-])c4cc(c(c(c4)OC)OC)OC.Br ML00369 Cc1c2c(cc(s2)C(C)(C)C)sc1C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N GK03057 Cc1c2c(cc(s2)C(C)(C)C)sc1C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N GK03058 c1ccc(cc1)C(=O)c2cccc(c2)NC(=O)c3c(cccc3Cl)F RH01380 CCOc1ccc(cc1)NC(=S)N2CCC(CC2)C(=O)OCC RH01381 Cc1c(c(c(c(c1C)C)S(=O)(=O)NC(=N)C)C)C CD06791 CC1CC(CC(C1)(C)C)N2CNC(=NC2)SCc3ccc(cc3)[N+](=O)[O-].Br ML00412 c1cc2ccc3cccc4c3c2c(c1)cc4NS(=O)(=O)c5ccc(cc5)[N+](=O)[O-] RJC03751 c1cc(c(c(c1)F)n2ccnc(c2=O)O)F CD11673 c1ccc(cc1)C2CC(=O)N(C(=O)C2)Cc3csc4c3cccc4 PD00455 c1cc(c(nc1)N2CCC(CC2)C(F)(F)F)[N+](=O)[O-] SPB06070 c1c(cc(cc1Cl)Cl)OC(=O)C23CC4CC(C2)CC(C4)C3 CD08966 Cn1c(ccn1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl GK03076 COC(=O)c1c(ccs1)Oc2ccc(cc2NS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F GK02105 CCn1c(cc(c(c1=O)C#N)C)O JFD03640 CC(c1ccccc1)NS(=O)(=O)c2ccc-3c(c2)C(=O)c4c3ccc(c4)S(=O)(=O)NC(C)c5ccccc5 BTB15085 Cc1nc(cs1)c2ccc(cc2)[N+](=O)[O-] SP00408 Cc1cn(c(=O)[nH]c1=O)[C@H]2C[C@@H]([C@H](O2)CO)OC(c3ccccc3)(c4ccc(cc4)OC)c5ccc(cc5)OC RJC03785 c1cc(sc1)C(=N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD06700 c1ccc(cc1)CCNC(=O)N RJC03754 CCOc1ccc(cc1)NC(c2ccccc2)C(=O)Nc3ccc(cc3)OCC PHG00222 Cc1ccc(cc1F)NC(=S)NC(C)(C)C K00016 c1cc(cc(c1)n2ccnc(c2=O)O)C(F)(F)F CD11680 CC(=O)c1ccc(o1)c2ccc(c(c2)Cl)Cl CD11756 CCOC(=O)NC(=S)NCc1ccco1 NH00497 COc1ccc(cc1)NC(=O)c2cccc3c2-c4ccc(cc4C3)I BTB15082 CCCc1cnc(nc1)N2CCCN(CC2)C(=S)Nc3ccc(cc3C)C AW00860 c1ccc2c(c1)c(cs2)CCOC(=O)c3ccc(cc3)Cl S11585 c1cc(ccc1C(F)(F)F)NC(=O)N2CCOCC2 S11994 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3ccc4c(c3)OCCCO4 SP00365 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3ccc(c(c3)F)F SP00361 CCOc1ccc(cc1)/C=N/NC(=O)c2c(onc2c3ccccc3)C CD03131 c1cc(ccc1C#N)C(=O)c2cc3cc(ccc3o2)[N+](=O)[O-] RH01758 COc1ccc(cc1)Oc2cccc(c2CNC(=O)c3ccccc3N)Cl CD11675 CC(=O)c1ccc(c(c1)/N=C/c2cccc(c2O)OC)Cl CD03529 c1cc(c(cc1O)O)/C=N/NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03361 CCC1=Nc2cccc3c2c(ccc3)N1 RJC03760 COc1ccc(cc1OC)S(=O)(=O)NCc2ccco2 KM09223 COc1ccccc1N2CCN(CC2)CCCC#N SEW06104 COC(C/N=C/c1cc(cc(c1O)Cl)Cl)OC BTB03997 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccccc2OC(F)(F)F RH01377 c1ccc2c(c1)c(cs2)CSCc3csc4c3cccc4 S11548 Cn1c(c(cn1)c2nc(cs2)c3ccc(cc3)Cl)/N=C/N(C)C CD09665 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)Br)Cl BTB07746 CC(C)C[C@@H](C(=O)O)NC(=O)[C@@H]1CCCN1C(=O)OCc2ccccc2 JFD03175 c1cc(ccc1C(=O)CO)Cl CD11832 CCCCc1ccc(cc1)NC(=S)NNC(=O)CSCc2cccc3c2cccc3 RH01650 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(cc3)F SEW06115 c1ccc2c(c1)cccc2CSCC(=O)NNC(=S)Nc3ccc(cc3)OC(F)(F)F RH01648 c1ccc2c(c1)cccc2CSCc3nnc(n3c4ccc(cc4)OC(F)(F)F)S RH01670 COc1cccc(c1)NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW06118 CCN(CC)C(=S)NC(=S)c1ccc(cc1)C JFD03610 c1cc(sc1)c2c(sc3c2c(c(s3)C#N)N)C#N KM03473 c1ccc(cc1)CC(c2ccccc2)C(=O)O JFD03600 c1ccc(cc1)c2ccc(cc2)C(=O)c3cc4cc(ccc4o3)[N+](=O)[O-] RH01748 COc1ccc(cc1)c2cc(n3c(n2)ccn3)C(F)(F)F KM10333 COc1ccc(cc1OC2CCCC2)S(=O)(=O)NCc3ccco3 KM09317 CC(=O)OC(C(C(=O)O)OC(=O)C)C(=O)Nc1ccc(cc1)Cl CD11884 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=S)Nc3ccccc3 CD05939 Cc1cc(c(c(c1)C)CC(=O)NNC(=S)Nc2ccc(cc2)C(C)C)C BLT00107 Cc1nc(cs1)c2ccc(cc2)Br.Br CD00564 C1CC(C(=O)C(C1)CCC(=O)O)CCC(=O)O RH01730 Cc1ccc(c2c1c(c(cn2)C(=O)O)O)C RH01747 c1cc(ccc1C(=O)c2cc3cc(ccc3o2)[N+](=O)[O-])F RH01759 CC(C)(C)NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2CN1C(=O)c3ccc(cc3)C(F)(F)F SPB08061 CCCCNC(=O)Nc1cc(cc(c1)C(C)(C)C)C(C)(C)C RF03348 CC(C)NC(=O)N(Cc1cccnc1)Cc2ccc(cc2Cl)Cl RF03486 COc1ccc(cc1)C(=O)c2cc3cc(cc(c3o2)Br)Br RH01771 Cc1c(ccc2c1OC(CC2=O)(C)C)OCc3cccc(c3)OC(F)(F)F RH01401 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])Sc2nnc(n2C)C(F)(F)F RH01403 Cc1cc(c(c(c1)C)COc2ccc3c(c2C)OC(CC3=O)(C)C)C RH01404 C=CCNC(=O)c1cccc2c1-c3ccccc3C2=O JFD03217 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F SP00448 CC(=O)Oc1ccc2ccccc2c1c3c4ccccc4ccc3OC(=O)C JFD03222 Cc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)Cl BTB07747 COc1ccc(cc1)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM09328 COc1ccc(cc1OC2CCCC2)S(=O)(=O)N(CCC#N)Cc3ccco3 KM09324 c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccc(cc4)F KM09337 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NNC(=S)CC2CCCO2 SPB08055 CC1=N/C(=C\c2ccc(cc2)Br)/C(=O)O1 SPB08058 Cc1ccccc1C(=O)Nc2ccc(cc2)Cl RF04238 CCOC(=O)c1c(n[nH]c1/N=C/c2ccc(c(c2Cl)OC)OC)C JFD03609 CC(C)(C)c1c(sc2c1c(c(s2)C#N)N)C#N KM03484 c1cc(ccc1c2ccc(o2)c3ccc(cc3)[N+](=O)[O-])[N+](=O)[O-] JFD03613 C/C(=N\Nc1ccc(cc1[N+](=O)[O-])S(=O)(=O)NCc2ccco2)/c3ccc(cc3)F BLT00212 COc1ccc(cc1OC)S(=O)(=O)NCc2ccccc2 KM09224 c1cc[n+](cc1)Cc2cc(cc3c2OCOC3)Cl.[Cl-] CD06087 Cc1c(c(c2c(c1C)[nH]c(n2)SCc3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C)C CD04434 CC1CCN(CC1)Cc2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F.Cl CD04499 CC(C(=O)NNC(=S)NC)Oc1ccccc1c2ccccc2 JFD03208 CC(c1n[nH]c(=S)n1c2ccccc2)Oc3ccccc3c4ccccc4 JFD03210 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl SEW06023 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4cccc(c4)C(F)(F)F KM09564 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)c3ccc(cc3)C4SCCS4 SP00526 C/C(=N\c1ccc(cc1)Cl)/c2ccsc2 JFD03183 CC(C)(C)NC[C@H](COCc1ccccc1)OC(=O)C(C(C(=O)O)OC(=O)c2ccccc2)OC(=O)c3ccccc3 BTB15163 c1cc2c(cc1N3C(=O)COCC3=O)OCO2 PD00481 COc1ccc(cc1)CS/C(=N/N)/N.Cl DP00933 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)[N+](=O)[O-])C(=O)OCC)C)C JFD03266 CC1CN=C(S1)N(c2ccc(c(c2)Cl)Cl)C(=O)Nc3ccc(cc3)Cl RJC03588 c1cc(cc(c1)Cl)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06027 CC(C)c1ccc(cc1)NC(=O)C(Cl)Cl CD04876 c1cc(c(c(c1)F)NC(=O)/C=C/C(=O)O)F CD04905 COc1ccc(cc1)n2c(nnn2)/C=C/N3CCN(CC3)c4cccc(c4)C(F)(F)F JFD03620 c1cc(sc1)SCC(=O)NN KM04491 c1cc(c(cc1F)F)NC(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00816 c1cc(c(cc1Cl)Cl)NC(=S)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00801 CC(=O)c1ccccc1OC(=O)c2c(cccc2Cl)Cl CD07364 CN(C)c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00671 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Br)Br)Cl RH01767 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Br)Br)F RH01770 c1cc(cc(c1)[N+](=O)[O-])C(=O)c2cc3cc(cc(c3o2)Br)Br RH01768 c1cc(ccc1OC(F)(F)F)S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl SPB08077 CC(C)c1ccc(cc1)NC(=O)c2cnccn2 PD00482 COC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)CN3CCOCC3 RH01711 Cn1c(ccn1)NC=C(C#N)C#N GK03137 c1cc(ccc1Oc2c(c(ccn2)C(F)(F)F)C(=O)NCc3ccc(cc3Cl)Cl)Cl RF05066 c1cc(ccc1NC(=O)c2c(ccnc2OCC(F)(F)F)C(F)(F)F)Cl RF05071 CC1c2cc(c(cc2CCN1)OC)OC BTB04350 CC1=C(C(C(=C(N1)C)C(=O)OC)c2cccc(c2)Cl)C(=O)OC JFD03271 CCC(C)NC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl BTB03775 c1c(cnc(c1C(F)(F)F)N2CCOCC2)[N+](=O)[O-] RF05250 C#CCOC(=O)Nc1cc(c(nc1)N2CCOCC2)C(F)(F)F RF05257 Cc1ccc(c(n1)[N+](=O)[O-])OC RH01350 Cc1cc(cc2c1C(=O)CC(O2)(C)C)OCC(=O)N(C)c3ccccc3 RH01351 CC(=O)Nc1c(c2c(s1)-c3ccccc3CC2)C#N JFD03630 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Sc2[nH]c(=O)c(c(n2)C3CCCCC3)C#N RH01386 c1c(cc(c(c1)/C=N/N=C/c2c(cc(cc2)O)O)O)O CD03162 CCOc1nn(c(=O)o1)c2c(cc(cn2)C(F)(F)F)Cl RF04958 COC(=O)NNc1cc(ccn1)C(F)(F)F RF04966 Cc1cc(cnc1c2ccccc2)C3CC=C(C(N3)c4ccccc4)C RJC03626 c1ccc(cc1)C2CC3CC(N2O3)c4ccccc4 RJC03627 CC1=C(C(C(=C(N1)C)C#N)c2cccc(c2)Cl)C#N JFD03273 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccccc3)C#N JFD03281 Cc1nnc(n1c2ccc3c(c2)OCCO3)SCC(=O)c4ccc(cc4)Cl SPB08071 c1cc(cc(c1)Cl)c2nnc(o2)c3cnc(cc3C(F)(F)F)Oc4ccc(cc4)Cl RF04843 CC(=O)O/N=C/c1c(c[nH]n1)Br RF04845 c1cc(c(cc1C(=O)NNc2ccc(cn2)C(F)(F)F)Cl)Cl RF04848 COc1ccccc1C(=O)NNc2c(cccn2)C(F)(F)F RF04872 COCCOc1c(cc(cn1)NC(=O)OCC#C)C(F)(F)F RF05258 CC(=O)O[C@@H]1[C@@H]2[C@H](O[C@@H]1C3COC(O3)(C)C)OC(O2)(C)C RJC03781 CC(=O)O[C@@H]1[C@@H]2[C@H](O[C@@H]1C(CO)O)OC(O2)(C)C RJC03782 CCN(CC)C1=NC(N=C(O1)c2cccc(c2)Cl)(C(F)(F)F)C(F)(F)F RJC03648 c1ccc(cc1)Cc2c(nc3ccccn3c2=O)O JFD03136 CC(c1ccc[n+](c1)C)OC(=O)c2cccc(c2)Cl.[I-] BW00063 Cc1ccc(c(c1)C)c2csc(n2)COc3ccc(cc3)OC SP00454 c1cc(c(nc1)n2c(=O)oc(n2)c3ccc(c(c3)Cl)Cl)C(F)(F)F RF04896 c1cc(cc(c1)C(F)(F)F)C(=O)NNc2cc(ccn2)C(F)(F)F RF04910 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4ccc(cc4)[N+](=O)[O-] KM09562 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)OCc3ccccc3)C(=O)OCC)C)C JFD03272 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(o3)c4ccccc4C(F)(F)F)C#N JFD03288 COc1ccc(cn1)NC(=O)OCC#C RF05237 Cc1ccc(c(c1)C)n2c(noc2=O)c3cnccc3C(F)(F)F RF05234 COCCOc1ccc(cn1)NC(=O)OCC#C RF05238 c1cc(c(nc1)NNC(=O)c2ccc(c(c2)Cl)Cl)C(F)(F)F RF04875 Cc1c(ccc2c1OC(CC2=O)(C)C)OCc3ccc(cc3Cl)Cl RH01388 CN(c1ccccc1)C(=O)CSc2[nH]c(=O)c(c(n2)C3CCCCC3)C#N RH01394 c1cc(ccc1NS(=O)(=O)c2ccsc2C(=O)O)Cl GK03169 c1cc(ccc1C(=O)c2cc3cc(ccc3o2)[N+](=O)[O-])OC(F)(F)F RH01749 Cc1cc(cc(c1CNC(=O)c2c(ccnc2OC)C(F)(F)F)Cl)Cl RF05061 c1cc(c(cc1Cl)Cl)CNC(=O)c2c(ccnc2OCC(F)(F)F)C(F)(F)F RF05062 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cc(c(c(c3)OC)OC)OC)C#N JFD03287 COc1ccncc1C(=O)Nc2cc(cc(c2)Cl)Cl RF05518 COC(=O)CSCCc1nc(cs1)c2ccc(cc2)[N+](=O)[O-] SP00455 c1cc(ccc1c2csc(n2)c3ccc(cc3)Cl)C(F)(F)F SP00442 c1cnc(c(c1C(F)(F)F)C(=O)N)O RF05026 COc1c(c(ccn1)C(F)(F)F)C(=O)NCc2ccc(c(c2)Cl)Cl RF05057 c1cc(ccc1[N+](=O)[O-])OCC(CN2CCCCC2)O AW00771 c1c(cnc(c1Cl)NCCCN)C(F)(F)F AW00789 COc1ccc(cc1)OCc2nc(cs2)c3ccc(cc3)C#N SP00469 CC(C)(C)NC(=O)N1CCN(CC1)c2c(cccn2)C(F)(F)F SEW06003 c1cc2c(cc1c3csc(n3)CC#N)OCCCO2 SP00553 c1cc(ccc1C2SCCS2)OCc3nc(cs3)c4ccc(c(c4)Cl)Cl SP00505 CCCCc1ccc(c(c1)C)NC(=O)CSc2[nH]c(=O)c(c(n2)C3CCCCC3)C#N RH01395 c1cc(c(cc1Cl)Cl)NC(=S)NNCCCO CD10428 CCCCNC(=O)N1CCC(CC1)C(=O)c2c(c(c(c(c2C)C)C)C)C CD10731 c1cc(ccc1CNC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD10739 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)OC2CCSC2 CD10756 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCc5c(cccc5Cl)F RH01756 c1ccc(cc1)Sc2c(c(ccn2)C(F)(F)F)C(=O)Nc3ccc(cc3)Cl RF05080 CCc1ccc(cc1)n2c(nnn2)SCC(=O)NCCSCc3ccco3 KM10420 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc3c(c2)OCCCO3 SP00638 CC(=O)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06001 Cc1ccc(cc1[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06002 c1ccc(cc1)CNC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06011 c1cc2c(cc1c3csc(n3)c4c(cc(cc4Cl)C(F)(F)F)Cl)OCCCO2 SP00541 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])N3CCOCC3 RH01761 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccccc2Cl)C(=O)OC JFD03301 c1cc(ccc1CCNS(=O)(=O)CS(=O)(=O)NCCc2ccc(cc2)Cl)Cl CD09635 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)CC#N SP00552 c1cc(oc1)CSCCNC(=O)CSC2=NCCS2 KM10423 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)c5ccc(c(c5)F)F RH01757 CN(C)c1ccc(cc1)C=C(c2ccc(cc2)N)c3ccc(cc3)N PHG00059 c1cc(ccc1Oc2c(c(ccn2)C(F)(F)F)C(=O)NCc3ccc(c(c3)Cl)Cl)Cl RF05067 CCSc1c(c(ccn1)C(F)(F)F)C(=O)NCc2ccc(c(c2)Cl)Cl RF05078 CCOC(=O)CN(C)S(=O)(=O)c1ccsc1C(=O)OC GK03167 c1ccc2c(c1)cccc2NC(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06004 Cc1ccc(cc1Cl)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06015 CCOC(=O)c1c(nc(c(c1c2ccc(c(c2)OC)O)C(=O)OCC)C)C JFD03207 CC(c1n[nH]c(=S)n1C)Oc2ccccc2c3ccccc3 JFD03209 COc1ccc(cc1)Oc2cccc(c2CNC(=O)Nc3ccccc3)F CD11676 COc1ccc(cc1)C(=O)NCc2c(cccc2F)Oc3ccc(cc3)OC CD11677 c1cc2c(cc1C(F)(F)F)NC(=O)c3c(ccs3)O2 GK03168 CN(C)/C=N/S(=O)(=O)c1ccccc1 CD09422 c1ccc(cc1)OS(=O)(=O)CS(=O)(=O)Oc2ccccc2 CD09448 Cc1c(c(n[nH]1)C)/N=N/c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03017 Cc1c(c(c(c(c1C)C)CNc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)C CD03318 Cc1ccc2c(c1)nc(o2)c3ccc(cc3)Cl S14587 CC1c2nc3ccc(cc3n2CN(CO1)c4ccc(cc4)Cl)Cl S14869 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(cc2)C#N SP00646 c1ccc2c(c1)c(=O)[nH]c(=O)[nH]2 JFD03657 CNC(=S)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl SEW06012 CC(C)c1ccc(c(c1)Br)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06014 Cc1ccc(cc1)OCC2CN(C(=O)O2)Cc3ccccc3 BTB15176 CC1=C(C(C(=C(N1)C)C#N)c2cc(ccc2OC)OC)C#N JFD03302 CCOC(=O)C1=C(NC(=C(C1c2ccccc2Cl)C(=O)OCC)C)C JFD03305 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)c3ccc(cc3)c4csnn4 SP00514 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])N3CCCC3 RH01762 c1cc(c(nc1)N)C(=O)NN KM07915 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)[N+](=O)[O-] SP00371 Cc1ccc(cc1)c2csc(n2)c3ccc(cc3)C(C)(C)C SP00369 Cc1c2ccccc2sc1c3csc(n3)COC(=O)C(C)(C)C SP00643 C/C=C/C(=O)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06211 Cc1c(c(no1)c2ccccc2)c3csc(n3)CS(=O)(=O)C(C)(C)C SP00655 CNC(=S)N1CCc2c3ccccc3[nH]c2C1C(F)(F)F SEW06214 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(c(c3)Cl)Cl SEW06019 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=S)Nc4ccc(cc4)OC(F)(F)F)C(F)(F)F SEW06215 CCCCCCCSc1[nH]cnn1 JFD03159 Cc1cc-2c(cn1)C(=O)c3c2cccc3 RJC03608 CN(C)C(=O)COc1ccc2ccccc2c1 BTB15178 CNC(=O)CCN(Cc1ccco1)S(=O)(=O)c2ccc(c(c2)OC)OC KM09287 CSc1ccc(cc1)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM09351 C/C(=N\OCc1cccc(c1)C(=O)O)/c2ccc(c(c2)OC)OC KM06675 c1c2c(cc(c1Cl)Cl)nc[nH]2 RH00899 Cc1cccc(c1)NC(c2ccccc2)C(=O)O PHG00303 COC(=O)CSc1c(cc(s1)S(=O)(=O)N)[N+](=O)[O-] KM08945 CCCn1c(=O)c2c(nc[nH]2)n(c1=O)c3ccc(cc3)Cl KM09088 Cc1cccc(c1)N/C(=N\O)/c2ccccc2 RF05109 Cc1cc(c(c(c1)C)SCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C SEW06221 c1cc(oc1C=C2C(=O)NC(=O)NC2=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04080 Cc1c2cc(ccc2sc1c3csc(n3)COc4ccc(cc4)C5SCCS5)Cl SP00859 Cc1c2cc(ccc2sc1c3csc(n3)c4c(cc(cc4Cl)C(F)(F)F)Cl)Cl SP00857 CCOC(=O)NN1C(=O)c2cccc3c2c(ccc3)C1=O PHG00955 c1ccc(cc1)C(c2ccccc2)NC(=O)c3c(nccn3)C(=O)O PD00498 c1ccc(cc1)NCC/N=C/c2cc(cc(c2O)I)I PD00502 c1ccc(cc1)C#Cc2ccc(o2)C(=O)O/N=C(/c3cccc(c3)C(F)(F)F)\N KM08680 CC(c1n[nH]c(=S)n1CC=C)Oc2ccc(cc2Cl)Cl JFD03198 CC1C(N(C(CC1(c2ccc(cc2)F)O)c3ccccc3)C)c4ccccc4.Cl RJC03612 c1ccc(cc1)c2noc(=O)n2c3cccc(c3)C(F)(F)F RF05128 c1ccc(cc1)n2c(noc2=O)c3cccc(c3)Cl RF05129 c1ccc(cc1)n2c(noc2=O)c3cccc(c3)C(F)(F)F RF05130 c1ccc(cc1)N2C(=NC3(N2)CCCC3)S CD04272 c1cc-2c(cc1[N+](=O)[O-])/C(=N\O)/c3c2c(cc(c3)[N+](=O)[O-])C(=O)N BTB15089 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)Br)[N+](=O)[O-] BTB07701 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cccc2Cl)Cl)OC)Br)[N+](=O)[O-] BTB07710 CS(=O)(=O)NCc1c(cccc1Cl)Sc2ccc(cc2)Cl CD11887 Cc1cc(on1)NC(=O)c2ccc3c(c2)non3 KM10426 c1ccc(cc1)CCNC(=O)c2ccc3c(c2)non3 KM10427 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3ccccc3C(=O)O)Cl GK03172 Cn1c(nnc1Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C(F)(F)F RH01407 Cc1c(ccc2c1OC(CC2=O)(C)C)OCC(=O)C RH01408 c1ccc(cc1)/C=C(\C#N)/C(=O)O JFD03250 Cc1ccc(cc1)/C=C(\C#N)/C(=O)O JFD03253 CC1C(NC(C(C1=O)C)c2ccc(cc2)OC)c3ccc(cc3)OC RJC03619 c1ccc(c(c1)C(F)(F)F)N/C(=N\O)/c2cccnc2 RF05153 CC1=C(CC(C(C1)C(=O)Nc2cc(cc(c2)OC)OC)C(=O)O)C PD00504 c1ccc(cc1)/C=C/C2=N/C(=C/c3ccccc3Cl)/C(=O)O2 PHG00762 CSc1ccncc1C(=O)Nc2ccc(cc2F)F RF05519 COc1ccncc1C(=O)Nc2ccc(cc2F)F RF05520 Cc1cc(cc(c1)Cl)NC(=O)c2cc(ccc2Br)OC RF00413 c1cc(ccc1C#N)c2csc(n2)c3ccc(cc3)C4SCCS4 SP00533 CN(C)c1ccc(cc1)NC(=S)NCc2csc3c2cccc3 PD00414 c1ccc2c(c1)c(cs2)CNC(=S)Nc3ccc4c(c3)OCO4 PD00415 c1ccc(cc1)N2C(=NC3(N2)CCCCCC3)S CD04273 c1ccc-2c(c1)Cc3c2nccc3 RJC03622 c1ccc(c(c1)OCc2nc(cs2)c3ccc(cc3)OC(F)F)Cl SP00712 COc1c(cc(cn1)NC(=O)OCC#C)C(F)(F)F RF05163 c1ccc(cc1)c2c(nnn2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NS(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F CD04709 COc1c(cc(c(c1C(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl)OC)Br)[N+](=O)[O-] BTB07711 CCOC(=O)C(C(=O)OCC)NC(=S)SC RF03735 c1ccc(c(c1)C(=O)NNc2ccc(cn2)C(F)(F)F)Cl RF04817 Cc1ccc(c(c1)C)c2csc(n2)CS(=O)(=O)C(C)(C)C SP00563 Cc1ccc(cc1)c2csc(n2)CS(=O)(=O)C(C)(C)C SP00564 COc1c(csc1S(=O)(=O)N=S(=O)(C)c2ccccc2)C(=O)OC KM08427 c1ccc2c(c1)c(cs2)CNC(=S)Nc3ccc(cc3)F PD00413 CCCCc1ccc(cc1)NC(=S)NCc2csc3c2cccc3 PD00416 Cc1nc(cn1CC/C(=N/O)/N)[N+](=O)[O-] RH01400 c1ccc2c(c1)ccc3c2cc(c(=O)o3)NC(=O)c4cccc(c4)Cl PHG00642 c1cc(ccc1C#N)c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F SP00444 c1cc(c(cc1C(F)(F)F)NC(=O)c2cc(cc3c2-c4ccc(cc4C3=O)[N+](=O)[O-])[N+](=O)[O-])Cl JFD03214 CC1(CCC(c2c1ccc(c2)c3csc(n3)c4c(cc(cc4Cl)C(F)(F)F)Cl)(C)C)C SP00753 CCC(C)c1ccc(c(c1)/C=N/Nc2ccccc2)O RF01411 COc1ccccc1N2CCN(CC2)C(=O)c3c(cccc3F)F SEW06026 CC(C(C(=O)NCc1ccccc1)NC(=O)OC(C)(C)C)OCc2ccccc2 JFD03353 CC(C)NC[C@H](COCc1ccccc1)OC(=O)C(C(C(=O)O)OC(=O)c2ccccc2)OC(=O)c3ccccc3 BTB15172 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3ccc(cc3)Cl)Cl GK03173 c1ccc(cc1)NC(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl CD11881 CCc1cccc(c1NC(=O)c2ccc(cc2)Cl)C(C)CC CD06347 COc1cc(c(cc1C=C(C#N)C#N)C(=O)OC)OC JFD03259 c1cc(c(c(c1)C(F)(F)F)C(=O)OCC(=O)c2ccc(cc2)Cl)C(F)(F)F CD04769 Cc1nnc(n1c2ccc3c(c2)OCCO3)SCc4c(cccc4Cl)Cl SPB08070 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)CS(=O)(=O)C(C)(C)C SP00562 COC(CNC(=O)C(=O)Nc1c(cccc1F)F)OC CD11665 CC(C)(C#Cc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/N=C/c2cc(cc(c2O)Cl)Cl CD04309 COc1ccc(cc1OC)/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00677 Cn1c(nnc1Sc2ccc(cn2)[N+](=O)[O-])C(F)(F)F RH01409 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)COc3ccc4c(c3C)OC(CC4=O)(C)C RH01410 c1ccc(cc1)N2C(=O)c3cccc4c3c(ccc4N5CCOCC5)C2=O JFD03661 c1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl SPB08076 c1cc(c(cc1F)F)CNS(=O)(=O)c2ccc(cc2F)F CD10759 CCc1cc2c(cc1C(=O)CSc3nnc(n3c4ccccc4)COc5ccc(c6c5CCC6)C)C(CCC2(C)C)(C)C RH01719 c1ccc(c(c1)C(=O)c2cc(ccc2NC(=O)CN3CCCCC3)Cl)Cl RH01772 CCOC(=O)[C@@H]1[C@H]([C@@H]([C@](CC1=O)(C)O)C(=O)OCC)c2ccccc2 BTB15191 COC(=O)CSCCc1nc(cs1)c2ccc(cc2)C#N SP00487 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(c(c4)Cl)Cl SP00488 c1cc(c(c(c1)Cl)CNC(=O)c2ccc(cc2)Cl)Sc3ccc(cc3)Cl CD11890 c1ccc2c(c1)c(cc(n2)c3ccccn3)C(=O)[O-].[Na+] JFD03243 c1ccc2c(c1)c(cc(n2)c3cccnc3)C(=O)[O-].[Na+] JFD03244 CCOC(=O)CNC(=O)CC(C)(C)C JFD03262 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc5c(c4)C(CCC5(C)C)(C)C SP00751 CC1(CCC(c2c1ccc(c2)c3csc(n3)COc4ccc(cc4)OC)(C)C)C SP00750 CCOC(=O)c1c(n[nH]c1N/N=C\c2c(cccc2Cl)Cl)C JFD03662 c1ccc2c(c1)c3ccccc3n2Cn4c5ccccc5c6c4cccc6 JFD03667 C#CCOC(=O)Nc1ccc(nc1)Oc2ccc(cc2)Cl RF05210 Cc1ccc(c(c1)NC(=S)Nc2cccc(c2)OC)C K00136 Cc1ccc(c(c1)NC(=S)Nc2cc(c(cc2Cl)Cl)Cl)C K00139 CCOC(=O)c1c(noc1C(F)(F)F)c2c(cccc2Cl)Cl CD06047 CCc1nc(cs1)c2ccc(cc2)Cl.Br CD06040 CN(C)S(=O)(=O)Nc1cccc(c1)C(F)(F)F CD06080 Cc1ccc(cc1C)c2csc(n2)CC#N SP00554 c1cc(ccc1C#N)c2csc(n2)CC#N SP00557 Cc1nc(cs1)c2ccc(c(c2)Cl)Cl SP00390 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)Cl)Cl)Cl SP00396 c1cc(c(cc1c2csc(n2)c3ccno3)Cl)Cl SP00619 c1cc(ccc1c2csc(n2)c3ccc(cc3)Cl)[N+](=O)[O-] SP00415 CCOC(=O)Cc1csc(n1)c2ccc(cc2)Cl SP00419 Cc1nc(cs1)c2ccc(cc2)C(F)(F)F SP00422 c1ccc2c(c1)-c3c(cccn3)C2=O RJC03623 c1ccc\2c(c1)-c3c(cccn3)/C2=C\O RJC03624 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCCN2CC(OC(C2)C)C)C)C CD06142 c1ccc(cc1)c2c(nnn2c3ccc(cc3F)F)C(=O)O CD06341 c1cc(ccc1C2SCCS2)OCc3nc(cs3)c4ccc(c(c4)F)F SP00567 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2ccc(cc2)C#N SP00570 c1cc(ccc1C2SCCS2)OCc3nc(cs3)c4ccc5c(c4)OCCCO5 SP00573 CC(=O)Nc1cc(c(cc1[N+](=O)[O-])OC)[N+](=O)[O-] BTB15208 CCNC(=O)C(Cc1ccccc1)NC(=O)OC(C)(C)C JFD03163 CC(C(=O)NC)NC(=O)OC(C)(C)C JFD03166 c1cc(ccc1c2csc(n2)CC#N)[N+](=O)[O-] SP00556 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2ccc(cc2)[N+](=O)[O-] SP00565 Cc1nc(cs1)c2cc(c(c(c2)C(C)(C)C)O)C(C)(C)C SP00398 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2nc(cs2)c3ccc4c(c3)OCCCO4 SP00610 c1cc(cc(c1)OC(F)F)c2csc(n2)c3ccc(cc3)Cl SP00657 CC1C(N(C(C(C1O)C)c2ccccc2)C)c3ccccc3 RJC03631 CCC1C(NC(C(C1=NO)CC)c2ccccc2)c3ccccc3 RJC03632 Cc1c(c(no1)c2c(cccc2Cl)Cl)CC#N CD06548 Cc1ccc2c(c1)CCC[N@@]2S(=O)(=O)c3c(c(c(c(c3C)C)C)C)C CD06604 CC1CCCCN1CCCNC(=O)Nc2ccc(cc2)Cl CD06642 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)c3ccno3 SP00621 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=S)Nc4cc(cc(c4)Cl)Cl)C(F)(F)F SEW06219 c1cc(cc(c1)OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)[N+](=O)[O-] SEW06220 c1cc(c(cc1C(F)(F)F)Cl)NN=C(C#N)C#N SEW06223 Cc1cc(c(c(c1CSc2ccccc2N)C)CSc3ccccc3N)C BLT00117 c1ccnc(c1)CCNC(=S)Nc2ccc(cc2)Cl BTB01498 c1cc(ccc1c2csc(n2)CC#N)C(F)(F)F SP00559 Cc1c2ccccc2sc1c3csc(n3)CC#N SP00558 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)COc3ccccc3Cl SP00583 c1cc(ccc1c2nc(cs2)c3ccc4c(c3)OCCCO4)Cl SP00405 Cc1c2cc(ccc2sc1c3csc(n3)c4ccc(cc4)C5SCCS5)Cl SP00532 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2cccc(c2)F SP00656 c1cc(cc(c1)C(F)(F)F)CSCc2nc(cs2)c3cccc(c3)OC(F)F SP00661 c1cc(ccc1c2csc(n2)CC#N)OC(F)F SP00709 CC1=C(C(C(=C(N1)C)C#N)c2ccc(c(c2)Cl)Cl)C#N JFD03292 c1cc2c(cc1c3csc(n3)c4ccno4)OCCCO2 SP00622 COc1cc(ccc1OCc2ccccc2)CCNC(=O)Cc3cccc(c3)Br BTB15209 c1ccc(c(c1)OCc2nc(cs2)c3ccc(c(c3)Cl)Cl)Cl SP00581 Cc1c2ccccc2sc1c3csc(n3)COc4ccc(cc4)C5SCCS5 SP00578 Cc1nnc(n1c2ccc3c(c2)OCCO3)SCC(=O)c4ccccc4 SPB08072 COC(=O)CSCCc1nc(cs1)c2ccc(c(c2)Cl)Cl SP00397 Cc1nc(cs1)c2ccc3c(c2)OCCCO3 SP00399 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)COc3ccc(cc3)C4SCCS4 SP00568 Cc1c2ccccc2sc1c3csc(n3)CS(=O)(=O)C(C)(C)C SP00569 c1cc(ccc1C#N)c2csc(n2)c3ccc(cc3)Cl SP00602 Cc1ccc(c(c1)C)c2csc(n2)c3ccno3 SP00623 Cc1c2ccccc2sc1c3csc(n3)CS(=O)(=O)Cc4cccc(c4)C(F)(F)F SP00614 c1cc(cc(c1)OC(F)F)c2csc(n2)c3ccc(cc3)C4SCCS4 SP00660 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(cc2)OC(F)F SP00658 COc1ccc(cc1)OCc2nc(cs2)c3ccc(cc3)OC(F)F SP00705 CC(C)OC(=O)Cc1csc(n1)c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F SP00651 c1ccc(c(c1)/C=C(\C#N)/c2[nH]c3ccccc3n2)Cl PHG00737 c1ccc2c(c1)[nH]c(n2)/C(=C/c3ccc(cc3)Cl)/C#N PHG00731 Cc1ccc(cc1)c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F SP00428 Cc1ccc(c(c1)N)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl BTB01502 c1ccc(cc1)C(=O)Oc2ccc(cc2)CC/C=C/CCc3ccc(cc3)OC(=O)c4ccccc4 RJC03731 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4ccno4 SP00631 c1ccc(cc1)C(=O)S[C@H]2CCC[C@@H]2C(=O)O RJC03738 COc1ccc(cc1OC)S(=O)(=O)N(CCC#N)Cc2ccccc2 KM09254 COc1ccc(cc1OC)S(=O)(=O)N(CCC#N)CCC#N KM09255 CCOC(=O)C(=CNc1ccc(cc1)OC(F)(F)F)C(=O)OCC KM09280 c1cc(sc1)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C#N SPB08105 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)Cl)Cl)Oc4ccc(cn4)C(F)(F)F SP00424 Cc1ccc(c(c1)NC(=S)Nc2cccc(c2Cl)Cl)C K00135 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2nc(cs2)c3cccc(c3)F SP00616 c1cc(ccc1c2csc(n2)c3ccno3)[N+](=O)[O-] SP00626 c1cc(ccc1Nc2n[nH]c(=S)s2)I S00988 c1cc(ccc1C#N)c2csc(n2)c3ccno3 SP00630 Cc1c2ccccc2sc1c3csc(n3)c4ccno4 SP00627 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)COC(=O)C(C)(C)C SP00637 COc1ccc(cc1OC)S(=O)(=O)NCCC#N KM09229 c1cc2c(cc1/C=C/[N+](=O)[O-])OCO2 RH01697 CC(C)N(CCO)S(=O)(=O)c1ccc(cc1)N RH01700 Cc1cccc(c1NC(=O)NCCCO)C RH01703 Cc1ccccc1NC(=O)c2cccc3c2cccc3 RH01699 c1ccc2c(c1)nnn2C(=O)c3ccc(c(c3)Cl)Cl K00111 COc1ccc(cc1)c2csc(n2)c3ccc(cc3)OC.Br ML00293 COc1ccc(cc1)c2nc(cs2)c3cccc(c3)[N+](=O)[O-].Br ML00289 Cc1ccc(c(c1)C)c2csc(n2)c3ccc(cc3)OC.Br ML00288 CC(C)Cc1ccc(cc1)c2cc(c(s2)C(=O)C)N GK03027 Cc1ccc(cc1)c2csc(n2)COC(=O)C(C)(C)C SP00640 c1ccc(cc1)C(c2ccccc2)NC(=O)CSCC(=O)O PD00497 c1ccc2c(c1)ccc3c2nc(cc3C(=O)O)c4cc(cc(c4O)Cl)Cl RB00362 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)NNC(=O)c3ccccc3 KM08458 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)NNC(=O)c3cccs3 KM08461 CC(=O)N/C(=C\c1ccc(c(c1)OC)OCc2ccccc2)/C(=O)O SPB08029 c1ccc2c(c1)CC(=O)NC2c3ccccc3Cl JFD03231 CC1(CCC(c2c1ccc(c2)c3csc(n3)COc4ccc(cc4)C5SCCS5)(C)C)C SP00756 CC1(CCC(c2c1ccc(c2)c3csc(n3)COc4ccccc4Cl)(C)C)C SP00757 COC(=O)CSCCc1nc(cs1)c2ccc(cc2)C(F)(F)F SP00464 CC(C)OC(=O)Cc1csc(n1)c2ccc(cc2)Cl SP00418 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccco2)C(=O)OC JFD03315 CN(CCOC(=O)Nc1ccc(cc1)Cl)c2cc(nc3c2cccc3)C(F)(F)F KM08439 CC(C)(C#Cc1ccc(cc1)C(=O)OC)O KM08162 Cn1c(=O)c(cn(c1=O)c2ccccc2)/C(=N/O)/N KM08163 COc1ccc(cc1OC)S(=O)(=O)NC2CCCc3c2cccc3 KM09289 Cc1ccc(cc1)S(=O)(=O)O.Cc1ccc(cc1)S(=O)(=O)OCC(CNC(C)(C)C)O BTB15170 CC(C)(C)NC[C@H](COCc1ccccc1)OC(=O)C(C(C(=O)O)OC(=O)c2ccccc2)OC(=O)c3ccccc3 BTB15173 Cc1ccc(c(c1)NC(=S)Nc2c(cccc2Cl)C)C K00138 c1ccc(cc1)CNC[C@@H](COCc2ccccc2)OC(=O)C(C(C(=O)O)OC(=O)c3ccccc3)OC(=O)c4ccccc4 BTB15159 c1ccc2c(c1)cccc2OCC(=O)O BTB15160 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4c(c5cc(ccc5s4)Cl)C SP00852 CC(C)Cc1ccc(cc1)c2cc(c(s2)C(=O)N)N GK03028 CC(=O)Oc1nc(n(n1)c2ccccc2)c3ccc(cc3)C(C)(C)C S14746 CC1=N/C(=C/c2ccc(c(c2)Cl)Cl)/C(=O)O1 PHG00465 COc1ccc(cc1)NC(c2ccccc2)C(=O)O PHG00312 CC(C)(C)OC(=O)N1CCN(CC1)CCNC(=O)Nc2cc(cc(c2)Cl)Cl KM08222 C[C@H](c1ccccc1)NC[C@@H](COCc2ccccc2)OC(=O)C(C(C(=O)O)OC(=O)c3ccccc3)OC(=O)c4ccccc4 BTB15164 Cc1ccc(c(c1)C)NC(=O)C KM08882 c1ccc2c(c1)CC(=O)NC2c3ccc(cc3Cl)Cl JFD03232 CC1CC2(CCCCC2)N(Cc3c1cccc3)C(=O)C RJC03616 c1ccc(cc1)c2noc(=O)n2c3cccc(c3)Cl RF05127 Cc1c2cc(ccc2sc1c3csc(n3)CS(=O)(=O)C(C)(C)C)Cl SP00858 CCOC(=O)C1C2c3ccccc3C(C1C(=O)OCC)c4c2cccc4 BTB15161 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)F)C(=O)OCC)C)C JFD03318 c1cc(ccc1C(=O)N)S(=O)(=O)N2CCOCC2 CD10807 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)NCc5ccccc5 RH01720 c1cc(cc(c1)C(F)(F)F)CSC(=O)c2ccc(c(c2)Cl)Cl CD10879 CSc1ncc2c(n1)ncnc2O KM08177 Cc1c2c(cc(nc2n(n1)C)C(F)(F)F)O KM08178 c1cc(c(cc1Cl)Cl)CSc2c(nccn2)C#N KM08268 Cc1cc(cnc1c2ccccc2)C3CN(C(C(=C3)C)c4ccccc4)C(=O)C RJC03611 CCOC(=O)C1CCN(C1=O)S(=O)(=O)Cc2ccccc2 JFD03236 c1cc2c(cc1/C=C(\C#N)/C(=O)O)OCO2 JFD03247 COc1ccc(cc1Cl)N/C(=N\O)/c2ccccc2 RF05143 c1cc(c(c(c1)Cl)Cl)c2noc(=O)n2c3cccnc3 RF05146 c1cc(ncc1C(F)(F)F)N2CCN(CC2)c3ccc(cn3)NC(=S)NCC4CCCO4 SEW06232 c1cc(c(cc1S(=O)(=O)N)Cl)Cl NH00305 COc1ccccc1N2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F SEW06109 c1cc(c(nc1)N2CCN(CC2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F SEW06119 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)Cc4ccco4)[N+](=O)[O-] PHG00992 CN(CCOC(=O)Nc1cc(cc(c1)Cl)Cl)c2cc(nc3c2cccc3)C(F)(F)F KM08432 CC1CC2(CCCCC2)NCc3c1ccc(c3)[N+](=O)[O-] RJC03617 CC(C(=O)NNC(=S)Nc1ccccc1)Oc2ccc(cc2)Cl JFD03201 c1ccn(c1)c2c(cc(cc2Cl)[N+](=O)[O-])Cl CD04202 COc1ccc(cc1)/C=C(\C#N)/C(=O)O JFD03251 c1cc(cc(c1)n2c(noc2=O)c3cccnc3)C(F)(F)F RF05162 c1ccc(c(c1)NC(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F)OC(F)(F)F SEW06233 c1cc(cc(c1)Cl)S(=O)(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SEW06234 c1ccc(cc1)/C=C/C2=N/C(=C/c3ccc(cc3)Cl)/C(=O)O2 PHG00757 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3cnn(c3C(F)(F)F)c4ccccc4)C(F)(F)F GK03134 Cn1c(ccn1)NC(=O)Nc2ccc(cc2)Cl GK03133 CC1=C(CC(C(C1)C(=O)Nc2ccc(cc2)I)C(=O)O)C PD00507 CC(C#N)(c1ccncc1)Nc2ccccc2 JFD03182 CN(C)CC#Cc1ccc(s1)c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl KM08338 c1ccc(cc1)C(c2ccccc2)N3CCC(CC3)OCCC(=O)N KM08347 c1cc(c(c(c1)F)C(=O)NNc2cccc(n2)C(F)(F)F)F RF05177 CCCC1C(NC(CC1=O)c2ccco2)c3ccco3.Cl RJC03641 c1ccc(cc1)CN2C(=O)c3cccc4c3c(cc(c4)[N+](=O)[O-])C2=O PHG00994 CC(C)(C)c1ccc(cc1)NC(=S)N2CCN(CC2)c3ccccc3OC SEW06127 CNc1ccc(cc1)C(=O)O JFD03586 CN(C)/C=C/C(=O)c1cccc(c1)F CD11986 CN(C)/C=C/C(=O)c1cccc(c1Cl)Cl CD11987 CN(C)/C=C/C(=O)c1ccc(c(c1)Cl)F CD12011 C=CCNC(=O)NC(=O)c1cc(sc1)[N+](=O)[O-] DFP00087 CCc1c(nc2ccccn2c1=O)O JFD03141 c1ccc2c(c1)c(c(c(=O)[nH]2)C(=O)Nc3ccc(cc3)Cl)O JFD03148 c1cc(cc(c1)NC(=O)c2c(c3cccc4c3n(c2=O)CCC4)O)C(F)(F)F JFD03180 c1cc(ccc1c2nc(cs2)c3ccc4c(c3)OCCCO4)C5SCCS5 SP00527 c1ccc2cc(ccc2c1)C3=NNC(C3)(C(F)(F)F)O KM10431 CC(C)Nc1ccc(cc1[N+](=O)[O-])C(=O)OC KM10432 CC(C)Oc1ccc(cn1)NC(=O)OCC#C RF05299 C#CCOC(=O)Nc1cc(cc(c1)Cl)Cl RF05393 Cc1ccc(n1c2ccc(cc2)/C=N/Nc3ccc(cc3Cl)C(F)(F)F)C SEW01686 c1ccc2c(c1)OS(=O)(=O)CS(=O)(=O)O2 CD10604 c1cc(c(c(c1)C#N)Oc2ccc(cc2)N)C#N CD10959 CCOC1=CC(=O)N(C1)CC#C CD11017 CN(C)/C=N/c1nc(nn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)SC SEW00538 CC(=O)N/C(=C\c1c[nH]c(n1)c2ccccc2)/C(=O)O SPB08028 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK03099 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)F)F)C(F)(F)F SP00497 c1ccc2c(c1)CCNC2c3ccco3.C(=O)(C(=O)O)O RH01698 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)N(C)c5ccccc5 RH01714 CN(C)C(=O)Oc1cc(=O)oc2c1cccc2 JFD03189 CN(C)CCNc1cc(nc2c1cccc2)c3ccncc3.Br.Br JFD03239 Cc1cccc(c1)C(=O)Nc2cc(c(cc2C(=O)OC)OC)OC GK03176 CC1(CCC(c2c1ccc(c2)c3csc(n3)c4ccc(cc4)Oc5ccc(cn5)C(F)(F)F)(C)C)C SP00749 Cc1cc(c(c2c1CCC2)OCC(=O)NN)Br RH01785 C#CCOC(=O)Nc1ccc(cc1Cl)Cl RF05398 CSc1ccncc1C(=O)Nc2cc(cc(c2)Cl)Cl RF05515 c1ccc2c(c1)[nH]c(n2)/C(=C/c3c(cccc3Cl)Cl)/C#N PHG00741 CCOc1ccc(cc1)/C=C(\C#N)/c2[nH]c3ccccc3n2 PHG00732 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Br)Br)OC(F)(F)F RH01775 c1cc(c(c(c1)Cl)NC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-])Cl DFP00185 c1c(csc1[N+](=O)[O-])C(=O)NC(=O)N2CCOCC2 DFP00189 c1cc(cc(c1)F)c2csc(n2)c3ccc(cc3)Cl SP00443 CC1(CCC(c2c1ccc(c2)c3csc(n3)c4ccc(cc4)C(F)(F)F)(C)C)C SP00760 c1cc(ccc1c2nc(cs2)c3ccc4c(c3)OCCCO4)C(F)(F)F SP00499 Cc1c2cc(ccc2sc1c3csc(n3)c4ccc(cc4)C(F)(F)F)Cl SP00782 COC(=O)c1c(ccs1)Oc2ccc(cc2NC=C(C#N)C#N)C(F)(F)F GK03139 Cc1ccccc1n2c(cc(=O)n(c2=O)CCc3ccccc3)N KM09782 c1c(cc(c(c1Cl)N)Cl)C(=O)Nc2cc(c(cc2Cl)Cl)Cl BTB03564 c1cc(ncc1C#N)N2CCCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl SPB08088 COc1ccc2c(c1)cc([nH]2)C(=O)OC RH01702 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=S)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F GK03101 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)Nc3ccc(c(c3)Cl)F)C(F)(F)F GK03110 CC1(CCC(c2c1ccc(c2)c3csc(n3)CC#N)(C)C)C SP00754 Cc1ccc(c(c1)C)c2csc(n2)c3ccc(cc3)C(F)(F)F SP00500 COC(=O)c1c(ccs1)NC(=O)c2ccc3c(c2)non3 KM10428 c1ccc(c(c1)n2ccnc2Sc3c(cccn3)[N+](=O)[O-])Cl CD09988 c1ccc(cc1)CN2CNC(=NC2)SCc3ccc(cc3)Cl.Cl DP01359 c1ccc2cc(ccc2c1)CC(C(=O)O)N SPB08030 c1cc(ccc1C[C@@H](C(=O)O)N)OC(F)(F)F SPB08032 c1ccc(cc1)CSCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06236 Cc1c(c(no1)c2ccccc2)C(=O)N3C[C@H]4CCCC[C@H]4C[C@H]3C(=O)NC(C)(C)C SPB08082 CC(C)Cc1ccc(cc1)C(C)C(=O)N SEW06238 CC(C)(C)NC(=O)CSc1nnc(o1)[C@H](Cc2ccccc2)NC(=O)OC(C)(C)C SPB08083 CCC(C)C(C(=O)O)NC(=O)C(C(C)C)NC(=O)OCc1ccccc1 BTB15185 CC(C)C(C(=O)NC(Cc1ccc(cc1)O)C(=O)O)NC(=O)OCc2ccccc2 BTB15187 CC\1(C2CCC(C2)(/C1=N/O)C)C RH01753 CN(C)C1=NC(N=C(O1)c2ccc(cc2)F)(C(F)(F)F)C(F)(F)F RJC03650 CCC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)O RJC03651 c1ccc(cc1)c2c(nc3ccccn3c2=O)O JFD03135 COc1ccccc1C2CCN(CC2)C(=O)c3cccc(c3)[N+](=O)[O-] RH01436 c1ccc(cc1)C(=O)N[C@@H](CCCNC(=N)N)C(=O)Nc2ccc(cc2)[N+](=O)[O-] RH01441 Cc1ccc(cc1)c2csc(n2)c3ccc(cc3)C(F)(F)F SP00501 Cc1c2cc(ccc2sc1c3csc(n3)COc4ccccc4Cl)Cl SP00860 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)c2nnc(o2)SCC(=O)Nc3cccc(c3)SC SPB08081 Cc1c2ccccc2sc1c3csc(n3)c4ccc(cc4)C(F)(F)F SP00504 c1ccc(c(c1)C(=O)Nc2ccc(cc2)F)C(=O)O RH01454 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Cl)Cl)Cl RH01784 c1ccc(c(c1)C(F)(F)F)Nc2nnc(s2)c3ccc(cc3)N RH01036 CNc1ccccc1C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl DP01760 COc1ccc(cc1)C2CC3CC(N2O3)c4ccccc4 RJC03618 COc1ccc(cc1)OCc2nc(cs2)c3ccc(cc3)C(F)(F)F SP00470 COc1ccc(cc1)OCc2nc(cs2)c3cccc(c3)F SP00471 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(cc4)C#N SP00495 c1ccc(c(c1)C(=O)NC(=O)NNc2c(cncc2Cl)Cl)Cl CD11293 c1ccc(cc1)CNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD11323 c1ccc(c(c1)C(=O)N)OCC2CC2 RH01448 COC(=O)C1C([C@H]2c3c(cccc3)[C@@H]1c4c2cccc4)C(=O)OC BTB15204 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2ccc(c(c2)Cl)Cl SP00436 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)F)F)Oc4ccc(cn4)C(F)(F)F SP00425 c1cc(c(cc1c2csc(n2)CC#N)F)F SP00551 c1cc(ccc1C#N)c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl SP00465 Cc1c(snn1)C(=O)N2C[C@@H]3CCCC[C@@H]3C[C@@H]2C(=O)NC(C)(C)C SPB08084 c1cc(ccc1SCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl SEW06237 CC1=C(CC(C(C1)C(=O)NCc2ccccn2)C(=O)O)C PD00503 CC(=O)N[C@@H](Cc1ccc(c(c1Cl)OC)OC)C(=O)O SPB08087 CN(C)c1cc(oc(=O)c1Cl)c2cccc(c2)Cl CD11180 c1ccc(cc1)CC(=O)NCC(=O)O BTB15198 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)F)F)C4SCCS4 SP00525 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)Cl)Cl)C4SCCS4 SP00524 c1cc(ccc1c2nc(cs2)c3ccc(cc3)[N+](=O)[O-])C4SCCS4 SP00530 c1cc2c(cc1)[C@H]3C(C([C@@H]2c4c3cccc4)CO)CO BTB15205 c1cc(ccc1c2nc(cs2)c3ccc(c(c3)Cl)Cl)C(F)(F)F SP00496 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(cc3)C(F)(F)F SEW06018 Cc1cc(cc(c1F)C)S(=O)(=O)N2CCN(CC2)c3ccccc3OC SEW06020 c1ccc(cc1)/C(=N/O)/Nc2cccc(c2)C(F)(F)F RF05111 CC(=O)NCc1c(cccc1Cl)Cl CD06827 CC1C(CC(NC1c2ccccc2)c3ccccc3)O.Cl RJC03635 CCCCCC\1C(N(C(C/C1=N/O)c2ccccc2)C)c3ccccc3 RJC03637 CC1C(CC(N(C1c2ccccc2)C)c3ccccc3)O.Cl RJC03638 CC(=O)Nc1cc(cc(c1)OC)OC RH01765 Cc1nc(cs1)c2ccc(cc2)OC(F)F SP00423 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(c(c2)Cl)Cl)C(=O)OC JFD03293 CCOC(=O)C1=C(NC(=C(C1c2ccc(c(c2)Cl)Cl)C(=O)OCC)C)C JFD03294 CNC(=S)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06230 CCC(C)CNC(=S)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06231 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3cc(c(c(c3)C(C)(C)C)O)C(C)(C)C SP00364 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3cccc(c3)[N+](=O)[O-] KM10421 c1ccc(cc1)C#CC2(c3ccccc3-c4c2cccn4)O RJC03613 Cc1ccc(cc1)S(=O)(=O)N2Cc3ccccc3C(CC24CCCCC4)C RJC03615 CCOC(=O)c1ccsc1NC(=O)c2ccc(cc2)C(F)(F)F GK03088 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(c(c4)F)F SP00489 COc1ccc(cc1)OS(=O)(=O)CS(=O)(=O)C CD11205 c1cc(c(c(c1)Cl)C#N)OCC(F)(F)F CD11416 CNc1ccc(cc1[N+](=O)[O-])C(F)(F)F TG00004 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3ccc(cc3)Oc4c(cccc4Cl)[N+](=O)[O-] RH01643 c1ccc(cc1)/C=C/C=C(\C#N)/c2[nH]c3ccccc3n2 PHG00723 COc1cc(ccc1O)/C=c\2/c(=O)n3c4ccccc4nc3s2 JFD03344 CC(C)(C)C(=S)Nc1cccc(c1)Cl RH01081 Cc1cc(ccc1[N+](=O)[O-])OCc2ccccc2 RH01502 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Br)Br)Br RH01776 CN(C)c1ccc(cn1)C(F)(F)F SEW06239 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(cc4)OC(F)F SP00706 Cc1csc(c1C(=O)c2ccccc2)NC(=O)c3ccco3 GK03159 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)/C(=N/O)/N)C(F)(F)F SEW06204 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(c(cs2)C)C(=O)c3ccccc3 GK03160 COc1ccccc1N2CCN(CC2)S(=O)(=O)c3ccc(s3)c4ccno4 SEW06021 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl SEW06024 CC(=O)Nc1cc(c(cc1C(=O)OC)OC)OC GK03178 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccccc2[N+](=O)[O-])C(=O)OC JFD03307 CCOC(=O)C1=C(NC(=C(C1c2cc(ccc2OC)OC)C(=O)OCC)C)C JFD03308 CC1=C(C(C(=C(N1)C)C#N)c2cccc(c2)OC)C#N JFD03312 CC1=C(C(C(=C(N1)C)C(=O)OC)c2cccc(c2)OC)C(=O)OC JFD03313 COc1ccc(cc1)C(=O)c2cc3cc(ccc3o2)[N+](=O)[O-] RH01763 CCOC(=O)C(=CNc1cc(ccc1C)C)C(=O)OCC RH01766 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4c(c5ccccc5s4)C SP00494 CC(C)(C)c1cc(n(n1)c2ccc(cc2)n3cccc3)C(C)(C)C SEW06007 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06013 CCOc1ccccc1Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4C KM09792 c1ccc(cc1)C(=O)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06017 CN(C)/C=C/C(=O)/C=C/c1ccc(cc1Cl)Cl CD11423 CCC1C(CC(NC1c2ccccc2)c3ccccc3)O.Cl RJC03639 CC1C(NC(C(C1=O)C)c2ccco2)c3ccco3.Cl RJC03640 c1cc(ccc1/N=N/c2ccc(cc2O)O)S(=O)(=O)[O-].[Na+] RH01442 c1cc(cc(c1)O)C2=NC(C(=O)Nc3c2cc(cc3)Cl)O RH01507 Cn1c2ccccc2c\3c1CCC/C3=N\O RH01516 c1ccc(c(c1)C(=O)NCc2c(cccc2Cl)Cl)NS(=O)(=O)c3ccc(c(c3)Cl)Cl CD07248 CC(C)(C)NC(=O)[C@@H]1C[C@@H]2CCCC[C@@H]2CN1C(=O)COc3ccc(cc3Cl)Cl SPB08060 CC(=O)Oc1cccc(c1)/C=C/2\C(=O)OC(=N2)/C=C/c3ccccc3 PHG00763 CCC(C)C(C(=O)NCc1ccccc1)NC(=O)OC(C)(C)C JFD03349 CC1=N/C(=C/c2ccccc2Cl)/C(=O)O1 PHG00463 c1ccc(cc1)CN2C(=O)c3cccc4c3c(ccc4Br)C2=O PHG00543 Cc1c2cc(ccc2sc1c3csc(n3)COc4ccc(cc4)OC)Cl SP00459 COC(=O)CSc1ccc(cc1[N+](=O)[O-])C(F)(F)F KM08211 Cc1ccc(c(c1)C)c2csc(n2)CS(=O)(=O)Cc3cccc(c3)C(F)(F)F SP00611 Cc1c(c(no1)c2ccccc2)c3csc(n3)CS(=O)(=O)Cc4cccc(c4)C(F)(F)F SP00618 CCOC(=O)c1c-2c(sc1N)Cc3c2cccc3 PD00510 Cc1c2ccccc2sc1c3csc(n3)c4ccc(cc4)c5csnn5 SP00518 c1ccc-2c(c1)CCc3c2nc(nc3C(F)(F)F)N KM10419 COC(=O)c1c(ccs1)Oc2ccc(cc2N3C(=O)CCC3=O)Cl GK03175 CC(C)(C)C(=O)Nc1cc(c(cc1C(=O)OC)OC)OC GK03177 c1cc(cc(c1)F)c2csc(n2)c3ccc(cc3)c4csnn4 SP00521 C(C[C@@H](C(=O)O)N)CNC(=N)N.Cl RH01444 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3c[nH]c4c3cccc4)C(=O)OC JFD03660 c1cc(ccc1c2csc(n2)COc3ccc(cc3)C4SCCS4)OC(F)F SP00711 c1cc(ccc1S(=O)Cc2ccsc2C(=S)N)Cl SEW01701 Cc1cc2c(nc1)CCCC2=O RH01541 c1cc(cnc1)C(=O)NC(=O)N RH01549 c1ccc(cc1)C(c2ccccc2)N3CC(C3)Oc4ccc(cc4)Cl RH01550 c1cc(ncc1C#N)N2CCCNCC2 SPB07871 Cc1cc(no1)NC(=O)c2ccc3c(c2)non3 KM10433 c1cc(oc1)CSCCNC(=O)CSc2ccc(cc2)Cl KM10438 CN1CC2CCC1C[C@@H](C2)NC(=O)c3ccccc3 RH01463 CN1c2ccccc2C(=NCC1=O)c3ccccc3 RH01461 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2cc(cc(c2)Cl)Cl SEW06242 c1cc(cc(c1)Cl)/N=C/c2ccc(cc2)[N+](=O)[O-] DFP00124 CC1=N/C(=C/c2ccc(cc2)OC)/C(=O)O1 PHG00453 c1ccc2c(c1)cccc2CSCc3nnc(o3)c4ccc(cc4)F RH01641 c1ccc2c(c1)cccc2CSCc3nnc(o3)c4ccc(cc4)[N+](=O)[O-] RH01718 Cc1cc([nH]n1)C(=O)NNS(=O)(=O)c2ccccc2 RF04907 c1ccc(c(c1)n2c(noc2=O)c3cccnc3)Cl RF05157 c1ccc(cc1)N/C(=N\O)/c2cccnc2 RF05159 Cc1cc(c(c(c1)C)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C SEW06025 CCN1CNC(=NC1)SCc2cccc(c2)C#N.Br DP01313 CCOC(=O)NC(=S)Nc1ccc(cc1)F RDR00202 c1ccn(c1)c2c(c(c(o2)c3cccs3)C#N)c4cc(cs4)Br CD09255 Cc1cc(no1)NC(=O)CCCCCN2CCOCC2 CD09286 CS(=O)(=O)CC(=O)NC1CCCCC1 CD11430 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)C#N SP00433 Cc1c2cc(ccc2sc1c3csc(n3)c4ccc(cc4)Oc5ccc(cn5)C(F)(F)F)Cl SP00432 CC(c1ccccc1)N2C(=O)CSC2=S RB00026 c1cc(ccc1OCCCCCCCCCCOc2ccc(cc2)Cl)Cl RH01708 COc1ccc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)Cl BTB07641 Cc1cc(cc(c1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C SEW06028 CC(C)NC(=O)N(Cc1ccccc1)Cc2cccnc2 RF03331 CNC(=S)N(Cc1ccc(cc1)Cl)Cc2cccnc2 RF03336 COc1ccc(c(c1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)OC SEW06029 c1ccc(cc1)Oc2c(c(ccn2)C(F)(F)F)C(=O)NCc3ccc(c(c3)Cl)Cl RF05065 CC1(CCC(c2c1ccc(c2)c3csc(n3)c4ccc(cc4)c5csnn5)(C)C)C SP00752 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4cccs4)[nH]cn3 KM09694 c1ccc(cc1)NC(=O)Oc2cccc(c2)N3CCOCC3 CD09599 Cc1c(c(n(n1)C)C)Nc2[nH]nc(n2)N CD09983 c1cc(c(cc1F)Br)NC(=S)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00802 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccccc3Cl)C(=O)OC JFD03321 c1ccc(cc1)c2c(c(=O)c3ccccc3s2)Cc4ccc(cc4)Cl JFD03337 COc1ccc(cc1OC)/C=C(\C#N)/C(=O)O JFD03245 COc1cc(cc(c1OC)OC)/C=C(\C#N)/C(=O)O JFD03246 COc1cc(ccc1O)C2=NC(C(=O)Nc3c2cc(cc3)Cl)O RH01508 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])C(=O)OC JFD03269 CCOC(=O)C1=C(NC(=C(C1c2cccc(c2)Cl)C(=O)OCC)C)C JFD03274 CC1=C(C(C(=C(N1)C)C#N)c2c(cc(cc2OC)OC)C(=O)OC)C#N JFD03276 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cc(c(cc3OC)OC)C(=O)OC)C#N JFD03296 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(c(c3)OC)OC)C#N JFD03297 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)N RH01773 COc1ccc(cc1OC)CCN2C(=O)c3cccc4c3c(cc(c4)[N+](=O)[O-])C2=O PHG00250 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)Nc3ccc(cc3)Cl)C(F)(F)F GK03091 c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Oc3c(cccc3C#N)C#N CD11030 Cc1ccc(cc1Cl)NC(=S)N2CCCN(CC2)c3ccc(cn3)C#N SPB08092 CNC(=S)N1CCCN(CC1)c2ccc(cn2)C#N SPB08093 c1ccc2c(c1)nnn2CC(=O)NCCSCc3ccco3 KM10440 CC1=C(C(C(=C(N1)C)C(=O)OC)c2cc(c(cc2OC)OC)C(=O)OC)C(=O)OC JFD03295 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cc(ccc3OC)OC)C#N JFD03298 c1ccc(cc1)c2c(c(=O)c3ccccc3s2)Cc4ccc(c(c4)Cl)Cl JFD03339 Cc1cccc(c1)NC(=O)Nc2cccc(c2)C RH01510 c1ccc(cc1)CNc2c[nH]c(=O)[nH]c2=O JFD03326 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)Cl)C(=O)C1)C JFD03322 Cc1cc(nc(n1)NC(=O)NC(=O)c2c(c(cc(c2OC)Br)[N+](=O)[O-])OC)C BTB07757 c1ccc(cc1)c2c(c(=O)c3ccccc3s2)Cc4ccc(cc4Cl)Cl JFD03338 Cc1ncc(n1CCOC(=O)c2ccc(cc2)Br)[N+](=O)[O-] JFD03331 c1ccc2c(c1)nc3n2c(=O)/c(=C/c4ccc(cc4)Br)/s3 JFD03332 CCOC(=O)CNC(=O)c1ccc(o1)c2cccc(c2)[N+](=O)[O-] JFD03260 Cc1ccc(cc1)C2C(=C(NC3=C2C(=O)CC(C3)(C)C)C)C#N JFD03280 c1cc(ccc1n2c(n[nH]c2=S)c3ccncc3)S(=O)(=O)N4CCCCC4 ML00389 CC(=O)/C(=C(\c1c(cccc1Cl)F)/N)/C(=O)OC CD06917 CCOC(=O)C1=C(NC(=C(C1c2ccc(cc2)C)C(=O)OCC)C)C JFD03282 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3)OC)C#N JFD03283 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccccc3[N+](=O)[O-])C#N JFD03309 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cccc(c3)OC)C#N JFD03310 CCOC(=O)C1=C(NC(=C(C1c2ccccc2[N+](=O)[O-])C(=O)OCC)C)C JFD03311 c1ccc(cc1)COC(=O)[C@H](c2ccccc2)O BTB15197 Cc1ccc(c(c1)C)c2csc(n2)COc3ccc(cc3)C4SCCS4 SP00574 Cc1ccc(cc1)c2csc(n2)COc3ccc(cc3)C4SCCS4 SP00575 c1cc(cc(c1)F)c2csc(n2)COc3ccc(cc3)C4SCCS4 SP00580 Cc1c(c2c(c(c1O)C)C[C@@]3(C(=O)C(=C(C(=O)[C@@]3(O2)C)C)C)C)C BTB15202 Cc1c2ccccc2sc1c3csc(n3)c4ccc(cc4)Oc5ccc(cn5)C(F)(F)F SP00431 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4ccc(cc4)Oc5ccc(cn5)C(F)(F)F SP00445 CC(C)OC(=S)Nc1cccc(c1)Cl RH01096 Cc1ccc(cc1)S(=O)(=O)OCC(CNC(C)(C)C)O JFD03221 CN(C)C(=O)COc1cccc2c1cccc2 JFD03304 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(c(c3)Cl)Cl)C#N JFD03303 CC1=C(C(C(=C(N1)C)C#N)c2ccco2)C#N JFD03314 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc(cc3)Cl JFD03329 c1ccc(cc1)C(=O)O/N=C(/c2ccc(cc2)S(=O)(=O)N3CCOCC3)\N CD10840 Cc1ncc(n1CCOC(=O)c2ccccc2)[N+](=O)[O-] JFD03333 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])Sc3nnc(s3)N RH01680 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)OC)[nH]cn3 KM09981 Cc1c(c(no1)c2ccccc2)c3csc(n3)CC#N SP00593 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4ccc(cc4)c5csnn5 SP00591 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3Cl)Cl)C#N JFD03285 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc4c(c3)OCO4)C#N JFD03286 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3)O)C#N JFD03289 CS(=O)(=O)Nc1ccc(cc1)Oc2c(cccc2C#N)C#N CD11008 c1ccc(cc1)n2c(nnc2Sc3c(cccn3)[N+](=O)[O-])CSCc4cccc5c4cccc5 RH01693 CN(C)c1ccc(cc1)/C=C(\C#N)/c2[nH]c3ccccc3n2 PHG00721 c1ccc(cc1)c2c3cc(ccc3[nH]c2C(=O)NN)[N+](=O)[O-] RH00983 Cc1nnc(n1c2ccc3c(c2)OCCO3)SCC(=O)Nc4ccccc4Cl SPB08073 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2nc(cs2)c3ccc(cc3)C(F)(F)F SP00615 c1ccc(cc1)c2c(c(=O)c3ccccc3s2)Cc4ccc(cc4)C#N JFD03341 COc1cccc(c1C(=O)Nc2cccc(c2)[N+](=O)[O-])O JFD03254 COc1ccc(cc1)CC2CCC(=NO)CC2 RH01513 CC1=C(C(C(=C(N1)C)C#N)c2ccc(o2)c3ccc(cc3[N+](=O)[O-])Cl)C#N JFD03278 CC1=C(C(C(=C(N1)C)C#N)c2c(cc(cc2OC)OC)C(=O)O)C#N JFD03279 CCc1ccc(cc1)C2C(=C(NC3=C2C(=O)CC(C3)(C)C)C)C#N JFD03316 CC1C(=C(NC(=C1C(=O)OC)C)C)C(=O)OC JFD03317 CC1=C(CC(=C(N1)C)C(=O)OC)C(=O)OC JFD03319 c1ccc2c(c1)[nH]c(n2)/C(=C/c3ccc4c(c3)OCO4)/C#N PHG00726 c1cc(sc1)c2c(c(c(o2)NC(=O)C(Cl)Cl)c3ccc(cc3)C#N)C#N CD09275 Cc1c(sc(c1O)C#N)C#N CD09940 c1cc(c(cc1F)F)S(=O)(=O)Nc2cc(cc(c2)NS(=O)(=O)c3ccc(cc3F)F)C(F)(F)F CD10920 c1cc(ccc1c2csc(n2)COc3ccc(cc3)C4SCCS4)C(F)(F)F SP00594 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccco4)[nH]cn3 KM09702 c1cc2c(c(c1)F)CNC(=N2)S CD10970 c1cc(c(c(c1)C#N)Oc2ccc(cc2)NS(=O)(=O)c3ccc(cc3F)F)C#N CD10972 c1cc(c(cc1Cl)Cl)NC(=O)NCCC2CC2(Cl)Cl CD10980 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2nc(cs2)c3ccc(c(c3)Cl)Cl SP00607 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)Cl)C(=O)O CD11064 CN(C)C(=O)c1c2ccccc2c(=O)n(n1)c3ccccc3 CD11091 CCOC(=O)Cc1csc(n1)c2ccc(cc2)Oc3ccc(cn3)C(F)(F)F SP00650 CC(C)c1ccc(cc1)/C=C(\C#N)/c2[nH]c3ccccc3n2 PHG00728 COc1ccc(c(c1)Cl)NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)c4ccccc4OC RH01695 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(c(c2)F)F SP00636 c1cc(ccc1c2csc(n2)c3ccno3)C(F)(F)F SP00632 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(c(c2)Cl)Cl SP00635 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2)[N+](=O)[O-])C#N JFD03265 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM09711 Cc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)NC4=C2C(=O)CC(C4)(C)C JFD03284 CN(C)c1ccc(cc1C(=O)O)NS(=O)(=O)c2ccccc2 CD06987 Cc1c(c(c(c(c1C)C)S(=O)(=O)N(Cc2c(cccc2Cl)Cl)Cc3c(cccc3Cl)Cl)C)C CD07068 c1cc(cc(c1)NC(=O)N(Cc2c(cccc2Cl)Cl)Cc3c(cccc3Cl)Cl)C(F)(F)F CD07072 CC(=O)CCc1ccc(c(c1)OC)OC(=O)c2ccccc2Cl CD07217 c1ccc2c(c1)[nH]c(n2)/C(=C/c3ccc(cc3)O)/C#N PHG00725 Cc1cc(c(c(c1)C)NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)c4ccccc4OC)C RH01688 Cc1ccccc1NC(=O)N2CCCN(CC2)c3ccc(cn3)C#N SPB08090 COc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)Oc3c(cccc3C#N)C#N CD10976 Cc1ccc(cc1)c2csc(n2)CS(=O)(=O)Cc3cccc(c3)C(F)(F)F SP00612 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2nc(cs2)c3ccc(cc3)[N+](=O)[O-] SP00613 COc1ccc(cc1)OCc2nc(cs2)c3ccc(c(c3)Cl)Cl SP00450 CN(C)c1cc(oc(=O)c1Cl)c2cc(sc2Cl)Cl CD11159 CN(C)/C=C/C(=O)c1cc(ccc1OCC(F)(F)F)OCC(F)(F)F CD11167 c1ccc(c(c1)n2c(noc2=O)c3c(cccc3F)F)Cl RF05134 COc1ccc(cc1Cl)n2c(noc2=O)c3ccccc3 RF05145 c1cc(ccc1c2csc(n2)c3ccc(cc3)C(F)(F)F)C(F)(F)F SP00507 c1cc(ncc1C#N)N2CCCN(CC2)C(=S)NC3CCCC3 SPB08094 Cn1c(ccn1)NC(=O)Nc2ccccc2 GK03132 c1cc(ccc1C(CC(=O)O)CC(=O)O)C(F)(F)F PD00506 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc5c(c4)OCCCO5 SP00515 Cc1cccc(c1)C(=O)NCC(=O)O RH01715 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)Nc5ccc(cc5)C6CCCCC6 RH01716 Cc1c(ccc(c1F)Cl)S(=O)(=O)N2CCOCC2 CD10884 Cc1c(c(no1)c2ccccc2)c3csc(n3)c4ccc(cc4)C5SCCS5 SP00606 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)CS(=O)(=O)Cc3cccc(c3)C(F)(F)F SP00609 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3)OCc4ccccc4)C#N JFD03290 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3c(cc(cc3OC)OC)C(=O)OC)C#N JFD03291 c1cc(c(cc1c2csc(n2)c3ccno3)F)F SP00620 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)Cc2nc(cs2)c3ccc(cc3)C#N SP00617 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3c(ccs3)Cl)C(F)(F)F GK03127 c1cc(c(cc1F)F)NC(=O)N2CCCN(CC2)c3ccc(cn3)C#N SPB08089 CCCCNC(=O)N1CCCN(CC1)c2ccc(cn2)C#N SPB08091 c1cc(ccc1c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)C(F)(F)F SP00466 Cc1c2ccccc2sc1c3csc(n3)COc4ccc(cc4)OC SP00458 Cc1nc(cs1)c2ccc3c(c2)C(CCC3(C)C)(C)C SP00748 COc1c(cc(cn1)C(F)(F)F)NC(=O)OCC#C RF05164 CC(C)(C)OC(=O)N[C@@H](Cc1ccccc1)C(=O)NNC(=S)Nc2ccc(c(c2)Cl)F SPB08054 Cc1ccc(cc1C)/C=C(\C(=O)O)/NC(=O)C SPB08059 Cc1c(cccc1Cl)S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl SPB08075 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(cc4)C(F)(F)F SP00522 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4cccc(c4)F SP00523 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)Nc5cccc6c5OCO6 RH01717 CC(C(C(=O)N)NC(=O)OC(C)(C)C)OCc1ccccc1 JFD03350 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=C/C(=O)NNC(=O)c4ccc(cc4)C(F)(F)F RH01689 c1cc2c(cc1F)cc([nH]2)C(=O)NN RH01694 c1cc(ccc1C(=O)NCCC2CC2(Cl)Cl)[N+](=O)[O-] CD10989 c1cc(cc(c1)F)c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F SP00449 COc1ccc(cc1)OCc2nc(cs2)c3ccc(c(c3)F)F SP00451 CC1=NN(C(=O)C1)c2ccc(cc2)F RH01710 CN(C)/C=C/C(=O)c1cccc(c1)C(F)(F)F CD11107 CN(C)/C=C/C(=O)c1ccc(cc1)C(F)(F)F CD11139 Cc1ccc2c(c1)c3c([nH]2)C(=O)NCC3 RH01706 c1ccc(cc1)N/C(=N\O)/c2cccc(c2)Cl RF05116 c1ccc(cc1)c2noc(=O)n2c3cccc(c3)[N+](=O)[O-] RF05124 CCC(C)C(C(=O)NC)NC(=O)OC(C)(C)C JFD03347 CCC(C)C(C(=O)NCC)NC(=O)OC(C)(C)C JFD03348 c1cc(c(cc1Cl)Cl)NC(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00804 c1ccc(cc1)n2c(noc2=O)c3cccnc3 RF05166 c1ccc(cc1)CNC(=S)NCc2ccccn2 NH00547 Cc1ccc(cc1)c2csc(n2)c3ccc(cc3)C4SCCS4 SP00529 Cc1c2ccccc2sc1c3csc(n3)c4ccc(cc4)C5SCCS5 SP00531 c1ccc(c(c1)S(=O)(=O)NC(=O)Nc2c(c(c(o2)c3ccco3)C#N)c4ccc(cc4)C#N)Cl CD09529 COc1cc(cc(c1OC)OC)c2nnc(n2c3ccccc3Cl)SCC(=O)c4ccc(cc4)Br.Br ML00364 CCOC(=O)c1cnn(c1N)c2ccccc2 RH01176 CCCc1c(nc2ccccn2c1=O)O JFD03140 CC1=C(CC2C(C1)C(=O)N(C2=O)c3cc(cc(c3)OC)OC)C PD00509 c1cc(ccc1c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F)OC(F)F SP00704 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc(cc4)OC(F)F SP00707 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2ccc(cc2)OC(F)F SP00710 COC(=O)c1c(ccs1)S(=O)(=O)Nc2ccc(cc2)Cl GK03163 Cc1ccccc1n2c(noc2=O)c3cccnc3 RF05155 c1cc(c(cc1F)F)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06030 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3OC)CCC(=O)C CD07225 CC(=O)CCc1ccc(c(c1)OC)OC(=O)N(C)C CD07244 Cc1ccc(cc1)c2csc(n2)c3ccc(cc3)c4csnn4 SP00517 Cc1c(ccc2c1OC(CC2=O)(C)C)OCC(=O)Nc3ccc(cc3)C(C)C RH01452 c1cc(ccc1C(c2cc3cc(ccc3o2)[N+](=O)[O-])O)F RH01806 Cc1ccc(cc1)c2nc(on2)c3c(noc3C)C SP00767 Cc1cccc(c1)c2nc(on2)c3c(onc3c4c(cccc4Cl)F)C SP00862 CC1(COC(=N1)c2c(ccs2)SC)C SEW03322 Cc1ccc(c(c1)COc2ccc(nc2[N+](=O)[O-])C)C RH01340 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)NCc2ccco2 PD00369 CC(C)(C)Oc1ccc(cc1)CC(CO)NC(=O)OCC2c3ccccc3-c4c2cccc4 RJC04069 c1cc(cc(c1)Cl)NC(=O)NCCSCc2ccco2 KM10259 COC(=O)c1ccccc1SC(CC(=O)c2cccnc2)c3ccc(cc3)F PD00285 CC(=O)N/C(=C/c1ccc2c(c1)OCO2)/C(=O)O SPB08079 Cc1cccnc1NC(=O)NC(=O)c2ccc(s2)C(C)(C)C MBE00199 COC(=O)c1ccccc1SC(=O)c2ccc(c(c2)Cl)Cl MBE00271 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)c2c(cccc2F)F SEW06061 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)c2ccc(cc2)C(C)(C)C SEW06064 Cc1ccccc1c2nnc(o2)c3cc(nn3Cc4ccc(cc4)F)C(C)(C)C SPB08128 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(o3)C4CC4 SPB08129 c1cc2c(cc1NC(=O)CSc3nnc(s3)N)OCO2 RH01468 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCCNc2cccc(n2)C(F)(F)F AW00883 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)CCO)[N+](=O)[O-] PHG00249 c1cc(cc(c1)Cl)NC(=O)Nc2nccc(n2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F CD11220 c1cc(sc1)CNC(=S)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00134 c1ccc2c(c1)[nH]c(n2)/C(=C/c3ccco3)/C#N PHG00740 CC(=O)n1c2ccccc2c3c1cccc3 JFD03694 COc1cc(c(cc1OC)NC(=O)c2ccc(cc2)Cl)C(=O)OC GK03095 C/N=C(/Nc1cccc(c1)Cl)\SC.I RDR00260 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2Br)OC RH01476 CC(=O)Nc1nnc(s1)CC#N RJC03905 CCOC(=O)c1cc2cc(ccc2[nH]1)F RH01167 Cc1c(c2cc(ccc2n1C3CC3)OC)C(=O)O RH01118 Cc1cc(c(c(c1)C)NC(=S)N2CCN(CC2)c3ccccc3OC)C SEW06131 Cc1cccc(c1NC(=S)NC(Cc2ccccc2)c3ccccc3)Cl RDR00559 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)N(C)C RDR00435 c1cc(oc1)CS(=O)(=O)Cc2nc(on2)c3ccc(cc3)OC(F)(F)F SP00639 c1cc(ccc1OC(=O)C2=Cc3cc(ccc3OC2)Cl)OC(F)(F)F RDR03734 Cc1cc(c(c(c1)C)NC(=S)NC(C)(C)CO)C RDR00463 c1ccc(cc1)/N=c\2/n(c(cs2)c3cccc(c3)[N+](=O)[O-])c4ccccc4.Br RH01789 c1cc(cc(c1)N2C(=O)C=CC2=O)C(=O)O PD00190 CC(=O)N(C)c1cccnc1 RH01105 c1ccc(c(c1)C(=O)c2cc(ccc2NC(=O)CN3CCOCC3)Cl)Cl RH01774 c1cc(cc(c1)Cl)CNC(=S)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00144 c1ccc(cc1)CNC(=O)c2ccc3c(c2)non3 KM10429 CC(C)c1ccc(cc1)NC(=S)NNC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00196 CCC(=O)NNC(=O)c1cccc(c1)[N+](=O)[O-] DFP00247 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])SCc3ccc(cc3Cl)Cl RH01791 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])SCc3ccc(c(c3)Cl)Cl RH01793 CCOC(=O)/C(=N/NC(=S)N)/C SEW00414 CC(C)Oc1ccccc1C(=O)N RH01673 CC(C)(C)c1ccc(cc1)NC(=S)Nc2ccc(cc2)C(C)(C)C BTB04724 Cc1cc(c(c2c1CCC2)OCC(=O)NNC(=S)NCC=C)Br RH01790 C1CCN(C1)C(=O)C23CC4CC(C2)CC(C4)C3 SEW06033 Cc1c2cc(ccc2sc1C3=NNC(C3)(C(F)(F)F)O)Cl KM10430 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Cl)Cl)F RH01783 Cc1csc(c1C(=O)c2ccccc2)N3C(=O)C=CC3=O GK03162 COc1ccc(c(c1)S(=O)(=O)c2ccc(cc2Cl)[N+](=O)[O-])OC CD06943 CN(c1ccc(cc1[N+](=O)[O-])Cl)/N=C/c2cc(cc(c2O)Cl)Cl CD06974 CC1CC(CN(C1)c2ccc(cc2C(=O)O)NS(=O)(=O)c3ccccc3)C CD07006 c1cc(cc(c1)Cl)C(c2cc3cc(ccc3o2)[N+](=O)[O-])O RH01796 CC(=O)c1ccc(cc1)NS(=O)(=O)C RH01411 c1cc(cc(c1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F SEW06043 c1cc2cccc3c2c(c1)COC(=O)c4cccc5c4c(ccc5)S3=O JFD03345 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3ccc(cc3)c4csnn4 SEW01041 Cc1cc(c(n1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C)C(=O)O SEW01089 c1ccc2c(c1)cccc2CSCC(=O)NNC(=S)Nc3ccccc3Cl RH01645 COc1cc(ccc1n2cccc2)[N+](=O)[O-] RH01657 COC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)c3c(cccc3Cl)Cl RH01656 CCCCOC(=O)/C=N/Nc1ccccc1 SEW00213 CCOC(=O)c1c(=O)[nH]c(=S)[nH]n1 SEW00445 CN(C)NC(=O)c1ccc(o1)Oc2cc(cc(c2)Cl)Cl SEW00467 CC1CN(CC(O1)C)c2ccc(cc2C(=O)O)N CD06922 CCc1cc2c(cc1c3csc(n3)c4ccc(cc4)Cl)C(CCC2(C)C)(C)C SEW06035 c1ccc2c(c1)ccc3c2cc(c(=O)o3)c4ccc(cc4)[N+](=O)[O-] PHG00093 Cc1cccc(c1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06040 CCOC(=O)/C(=N/NC(=O)OCC)/C(F)(F)F SEW00614 CCOC(=O)N/N=C(\C)/c1cccc(c1)NC(=O)C SEW00688 Cc1ccc(cc1)c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl SP00544 CC(=O)CCc1ccc(c(c1)OC)OC(=O)c2cccs2 CD07229 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3ccccc3NC(=O)c4ccccc4Cl CD07277 c1cc(c(cc1c2csc(n2)CC#N)Cl)Cl SP00549 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] SP00685 c1cc(ccc1c2nc(no2)CS(=O)(=O)c3ccc(cc3)F)OC(F)(F)F SP00702 c1cc(ccc1c2csnn2)OC(=O)c3ccc(o3)[N+](=O)[O-] SEW01119 c1cc(ccc1C(c2cc3cc(ccc3o2)[N+](=O)[O-])O)OC(F)(F)F RH01799 Cc1cc(ccc1Br)N2C(=O)C3CC=C(CC3C2=O)C PD00513 CC1=C(CC(C(C1)C(=O)Nc2ccc(cc2F)F)C(=O)O)C PD00515 COc1ccc(cc1)/C=C/2\C(=O)OC(=N2)/C=C/c3ccccc3 PHG00750 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)C PHG00469 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)c3cc(c(c(c3)OC)OC)OC PHG00786 CC(=O)Oc1ccccc1/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] PHG00485 CCOc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PHG00630 CCOC(=O)N/N=C(\C)/c1ccc(cc1F)F SEW00665 CCOC(=O)N/N=C(\C)/c1cc(cc(c1)C(F)(F)F)C(F)(F)F SEW00666 Cc1c(c(no1)c2c(cccc2Cl)Cl)CNC(=O)C CD07086 c1cc(c(cc1F)F)NC(=O)c2cc(cc(c2O)Cl)Cl CD07140 CC(=O)CCc1ccc(c(c1)OC)OC(=O)c2ccco2 CD07228 C1COCCN1C(=O)C23CC4CC(C2)CC(C4)C3 SEW06032 Cc1cccc(c1)C(=O)N2CCN(CC2)c3ccccc3OC SEW06051 CC(C(C(=O)NC)NC(=O)OC(C)(C)C)OCc1ccccc1 JFD03351 CCNC(=O)C(C(C)OCc1ccccc1)NC(=O)OC(C)(C)C JFD03352 CC(C)(C)c1ccc(cc1)NC(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00806 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)[N+](=O)[O-])C(C)(C)C SP00566 CC1=N/C(=C/c2ccc(c(c2)OC)OC)/C(=O)O1 PHG00459 Cc1ccc(c(c1)C)c2csc(n2)c3ccc(cc3)C4SCCS4 SP00528 Cc1nnc(n1c2ccc3c(c2)OCCO3)SCC(=O)Nc4cccc(c4)C(F)(F)F SPB08074 c1ccc(cc1)C(=O)NCC(CC(=O)O)O JFD03228 c1cc(c(c(c1)Cl)COCCOC(=O)Nc2ccc(cc2)Cl)F CD09577 Cc1c(sc(n1)C)c2ccnc(n2)N CD09763 CCCc1ccc(cc1)c2nc(no2)c3ccccn3 SP00713 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4ccccn4 SP00719 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)Cc4ccncc4)[N+](=O)[O-] PHG00253 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl SP00540 c1cc2c(cc1Br)[nH]c(=S)s2 BTB09236 c1cc(c(cc1c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)Cl)Cl SP00538 Cc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Cl)OC)C BTB07640 CN(C)c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PHG00603 COc1ccc(cc1Br)/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00684 Cc1ccc(cc1)SCC(=O)Nc2cc(on2)C CD09233 c1ccc\2c(c1)-c3ccccc3C(=O)/C2=C/O JFD03665 Cc1c(c(sc1C(=O)Nc2ccccc2)N)C(=O)N JFD03666 CCn1c(c(c(n1)C)Br)c2nc(no2)CS(=O)(=O)c3ccc(cc3)F SP00699 COc1ccc(cc1OC)c2nc(no2)CS(=O)(=O)c3ccc(cc3)F SP00689 COc1ccc(cc1OC)c2nc(no2)c3ccccn3 SP00716 CN(C)C=C1C(=O)CC(CC1=O)c2ccc(cc2)Cl CD09850 CCc1cc2c(cc1c3csc(n3)c4ccc(cc4)OC)C(CCC2(C)C)(C)C.Br ML00291 CN1C2CCC1CC(=NO)C2 RH01542 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)Cl)Cl)OC)Br BTB07607 CCc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Cl)OC)CC BTB07639 COc1ccc(c(c1)c2nc(no2)c3ccccn3)Br SP00717 CC(=O)/C=C(/NCCN/C(=C/C(=O)C)/c1ccccc1)\c2ccccc2 CD10205 C1C(C1(Cl)Cl)CSc2nnc(s2)N CD10264 Cc1c(c(nc(c1C#N)S)C)Cc2ccc(cc2Cl)Cl CD10290 CCn1c(c(c(n1)C)Br)c2nc(no2)c3ccccn3 SP00723 c1cc(c(c(c1)Cl)C#N)Sc2ccc(cc2)Cl CD11671 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)/C=C/C(=O)O)C(F)(F)F GK02212 Cc1ccccc1C(=O)NNC(=O)c2cc(nn2Cc3ccc(cc3)F)C(C)(C)C SPB08124 COc1cccc(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC BTB07456 CCCCOC(=O)c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Cl RJC03158 CS/C(=N\C#N)/N1CCN(CC1)/C(=N/C#N)/SC CD09954 C=C(c1ccccc1O)n2ccnc2 CD10003 COc1ccc(c(c1OC)Cl)/C=C/c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SP00724 c1cc(ccc1NC(=O)Nc2cc(sc2Cl)Cl)Cl CD10297 Cc1cc2c(cc1C)n(c-3nc(=O)[nH]c(=O)c3n2)CC(C(C(CO)O)O)O RH01439 COc1ccccc1N2CCN(CC2)C(=O)c3cccc(c3)[N+](=O)[O-] RH01437 CNc1c(nc(o1)c2ccccc2)C#N JFD03335 c1ccnc(c1)SCC(=O)Nc2ccc(c(c2)Cl)F CD11418 c1ccc2c(c1)c(c[nH]2)CC(C(=O)O)N RH01445 c1cc(ccc1C(=O)N[C@@H](CCC(=O)O)CC(=O)O)NCc2cnc3c(n2)c(nc(n3)N)O RH01440 Cc1cc(ccc1[N+](=O)[O-])C(=O)NNC(=S)NCc2ccccc2 RH00771 c1ccc(c(c1)/C=N/NC(=S)N)O CD02771 CCc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)Cl)OC)CC BTB07686 COc1c(cc(c(c1C(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl)OC)Cl)[N+](=O)[O-] BTB07715 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC)Cl)[N+](=O)[O-] BTB07716 c1cc(cc(c1)Oc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])N3CCOCC3 BTB06086 CC(=O)Nc1ccc(c(c1F)F)F RH00323 COc1ccccc1C2CCN(CC2)C(=S)Nc3cccc(c3)C(F)(F)F RH01412 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(cc4)[N+](=O)[O-] SP00493 c1ccc(cc1)NC(=O)Nc2ccccc2C(=O)NC3CCSC3 CD10362 COc1ccc(c(c1C(=O)NC(=O)Nc2nc(nc(n2)OC)OC)OC)Cl BTB07649 CCc1ccc(cc1)NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)c4ccccc4OC RH01713 c1cc(c(cc1F)F)S(=O)(=O)N CD10447 COc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)[N+](=O)[O-])OC)OC BTB07726 Cc1c(ccc2c1OC(CC2=O)(C)C)S(=O)(=O)OC RH01479 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(cc4C)C SP00491 CCCCc1ccc(cc1)NC(=S)N2CCC(CC2)c3ccccc3OC RH01421 CC(=O)N/C(=C/c1ccc(cc1)Br)/C(=O)O SPB08080 CC(C)(C)NC(=O)[C@H]1C[C@H]2CCCC[C@H]2CN1C(=O)C34CC5CC(C3)CC(C5)C4 SPB08085 CCOC(=O)C(=C/C=C(/c1ccccc1)\N(C)C)C(=O)OCC RH01802 CC(=O)c1ccc(cc1)NC(=O)OC2CCSC2 CD10864 c1cc(c(c(c1)Cl)c2nc(on2)c3ccc(cc3Cl)F)Cl SP00780 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)c4ccccc4)[N+](=O)[O-] SP00788 c1cc(ccc1C(=O)CCC#N)Cl SEW02405 CCOC(=O)CCc1c2ccccc2[nH]c1C(=O)OCC SEW02793 COC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)c3cc(cnc3)Br RH01654 COC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)c3cccs3 RH01653 Cc1cc(cc(c1)NC(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F)C GK03105 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)c2cccs2 SEW06058 c1cc(ccc1C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)Cl SEW06266 c1cc(ccc1CSc2c(c(sn2)SCc3ccc(cc3)Cl)C#N)Cl SEW00158 COc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)OC BTB07743 c1c(csc1[N+](=O)[O-])C(=O)NC(=O)NN2CCOCC2 DFP00186 c1c(csc1[N+](=O)[O-])C(=O)NC(=O)N2CCCCC2 DFP00190 Cc1c(c(c(c(c1C)C)CSC2=NCN(CN2)CCc3ccc(c(c3)OC)OC)C)C.Cl DP00930 Cc1c(cn(n1)S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3ccccc3 CD09352 CCCCNC(=O)Nc1ccccc1Oc2ccccc2 CD09554 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3)F)C#N JFD03320 c1cc(c(c(c1)Cl)CSC/C(=N\O)/NC(=O)N)F CD11203 C1CC2(CCC13OCCO3)OCCO2 RH01539 Cc1ccc(cc1)C(=O)OC[C@@H]2[C@H](C[C@H](O2)c3nnc4n3cccn4)OC(=O)c5ccc(cc5)C JFD03691 COc1ccc2c(c1)C=C/C(=N\O)/C2=O PD00162 Cc1c(ccc2c1OC(CC2=O)(C)C)OCC(=O)Nc3ccc(cc3C(=O)c4ccccc4Cl)Cl RH01480 CN1CC2CCC1C/C(=N/O)/C2 RH01458 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2ccc(cc2)Cl JFD03687 CCOC(=O)c1c(n[nH]c1/N=C/c2ccccc2Cl)C JFD03689 c1cc(c(cc1c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)F)F SP00539 COc1cc(cc(c1)NC(=O)c2ccc(o2)[N+](=O)[O-])C(F)(F)F CD11058 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)O CD11079 COc1ccc(c(c1)c2nc(no2)CS(=O)(=O)Cc3ccco3)Br SP00586 Cc1c(ccc2c1OC(CC2=O)(C)C)OCC(=O)NCC=C RH01453 c1cc(ccc1c2nc(cs2)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F SP00503 COc1ccc(cc1OC)c2nc(no2)c3ccccc3 SP00792 COc1cc2c(cc1OC)nc[nH]c2=O GK03131 c1[nH]c(=O)c2c3c(sc2n1)CCCC3 GK03180 c1cc(sc1)/C=C(\C#N)/C(=S)N RJC03935 c1ccc(cc1)c2c(c(=O)c3ccccc3s2)Cc4ccc(cc4)Br JFD03340 c1ccc(cc1)c2c(c(=O)c3ccccc3s2)Cc4ccc(cc4)[N+](=O)[O-] JFD03342 COc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Cl)OC)OC BTB07653 c1cc(ccc1C(=O)CC(c2ccc(c(c2)Cl)Cl)SCC(=O)O)Cl JFD03343 c1ccc(cc1)C2=CC(=NN=C(C2)c3ccc(cc3)F)c4ccc(cc4)F JFD03693 CN1C2C[C@@H](CC1CC2)NC(=O)c3ccc(cc3)[N+](=O)[O-] RH01475 c1ccc(cc1)c2c(n[nH]c2N)c3ccccc3 JFD03669 c1ccc2c(c1)c(c[nH]2)c3c(nc4ccccc4n3)O JFD03671 c1cc(ccc1C#N)c2csc(n2)c3ccc(cc3)C(F)(F)F SP00509 Cc1ccc(c(c1)C)c2csc(n2)c3ccc(cc3)c4csnn4 SP00516 CCCCCCCCCCCCCCCCCCN1CNC(=S)NC1 RH01217 CC1(CC(=O)c2ccc(cc2O1)S(=O)(=O)OC)C RH01451 Cc1cc(ccc1N/C(=N/CCCOC)/SC)Br.I RDR00200 CN(C)c1ccc(cc1)c2c(c(nc(c2C#N)OC)N)C#N RDR00294 COc1cc(c(cc1OC)NS(=O)(=O)c2ccc(cc2)Cl)C(=O)OC GK03098 COc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2C(=O)OC)OC)OC GK03103 c1cc(cc(c1)F)c2csc(n2)c3ccc(cc3)C(F)(F)F SP00508 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc(c(c4)F)F SP00513 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc(c(c4)Cl)Cl SP00512 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Cl)Cl)OC(F)(F)F RH01787 c1cc(ccc1C#N)c2csc(n2)c3ccc(cc3)c4csnn4 SP00519 c1cc(sc1)C/C(=N/OC(=O)Nc2cc(cc(c2)Cl)Cl)/N SPB08122 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/Cc4ccco4 JFD03323 c1ccc(cc1)CNc2c(nc(o2)c3ccccc3)C#N JFD03325 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)F)/C=c\4/c(=O)n5c6ccccc6nc5s4 JFD03328 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)OC CD11090 CN(C)/C=C/C(=O)c1cccc(c1)Cl CD11177 CCOC(=O)C(=CNc1ccc(c(c1)Cl)F)C(=O)OCC BTB03722 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NNC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB08126 CC(C)C(=O)NNC(=O)CCC(=O)NNC(C)C RH00982 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)C2CCCCC2 SEW06063 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3ccccc3OC SEW06056 Cc1ccc(cc1)C(=O)Nc2cc(c(cc2C(=O)OC)OC)OC GK03093 Cc1cc2c(nc1)CCCC2=O.Cl RH01668 COc1cccc(c1)C\2CCCC/C2=N/O RH01599 c1cc(cc(c1)F)c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl SP00548 c1ccc(cc1)C2(c3ccccc3NC2=O)O RH01632 c1cc(ccc1c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)[N+](=O)[O-] SP00545 Cc1ccc(c(c1)C)c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl SP00543 CN(C)/C=C/C(=O)c1ccc(cc1Cl)Cl CD11150 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NNC(=O)c3cccs3 SPB08123 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NNC(=O)C3CC3 SPB08125 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)N3CCOCC3)C(C)(C)C SP00546 CC(C)(C)NC(=S)N/N=C/c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB03753 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)c2ccc(cc2)C SEW06059 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C SEW06060 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)c2cc(c(c(c2)OC)OC)OC SEW06062 c1c(c(sc1Cl)Cl)S(=O)(=O)N2CCC(CC2)C(=O)N CD10887 c1cc(ccc1NC(=O)O/N=C/c2ccc(o2)c3ccc(cc3F)F)Cl CD10908 Cn1cccc1C2=C(C(C(=C(O2)N)C#N)c3ccc(cc3)C#N)C#N CD10912 Cc1ccc(cc1)C(=O)NCC(=O)O PHG00643 CCn1c(c(c(n1)C)Br)c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SP00741 COc1ccc(cc1OC)c2nc(no2)c3ccc(cc3)OC(F)(F)F SP00820 CCCc1ccc(cc1)c2nc(no2)c3ccc(cc3)OC(F)(F)F SP00819 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4ccc(cc4)OC(F)(F)F SP00822 CC(C)(C)c1cc(n(n1)Cc2ccccc2)c3nc(no3)c4ccccn4 SP00734 c1ccnc(c1)c2nc(on2)c3ccno3 SP00732 Cc1c(c(on1)C)c2nc(no2)CS(=O)(=O)c3ccsc3 SP00785 CN(C)c1cc(c(cc1[N+](=O)[O-])F)N2CCOCC2 BTB03943 c1cc(c(c(c1)Cl)CNC(=O)Nc2ccc(cc2)Cl)Sc3ccc(cc3)Cl CD11892 CSC(=CC(=O)c1cccc(c1F)Cl)SC CD12025 c1cc(ccc1CCc2ccc(cc2)F)F RH01540 CCOC(=O)C(=CNc1ccccc1OC)C(=O)OCC RH01543 CN(C)Cc1c[nH]c2c1cccc2 RH01548 c1cc(ccc1c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)OC(F)(F)F SP00743 CCCc1ccc(cc1)c2nc(no2)CS(=O)(=O)c3ccsc3 SP00784 c1ccc(cc1)CC(C(=O)O)NC(=O)c2ccc(cc2)Cl PD00480 c1ccc(cc1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06041 CN(C(=O)Nc1ccccc1)n2cnc3ccsc3c2=O CD11737 c1cc(c(cc1F)Cl)c2nc(no2)c3cnccn3 SP00843 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)c5ccccc5 RH01738 c1ccc(cc1)C(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl CD11889 c1ccc(c(c1)C(F)(F)F)NC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00078 CN(C)C(=O)C(=O)c1c[nH]c2c1cc(cc2)Br RH01535 c1cc(ccc1C(F)(F)F)N2C(=O)c3c(nccn3)C2=O PD00075 c1ccc(cc1)NC(=S)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00799 c1cc2c(cc1NC(=S)N3CCCN(CC3)c4ccc(cn4)[N+](=O)[O-])OCO2 AW00800 c1cc(c(cc1N/N=C/c2cc(sc2)[N+](=O)[O-])Cl)Br DFP00003 CC(C)NC(=O)c1ccccc1c2ccccc2C(=O)NC(C)C JFD02702 CC(C)(C)c1ccc(cc1)NC(=O)c2cnccn2 PD00483 Cn1c(ccn1)NC(=O)/C(=C/c2ccc(cc2)Cl)/C#N GK03140 c1cc(ccc1CS(=O)(=O)Cc2nc(on2)c3ccc(cc3)OC(F)(F)F)F SP00813 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3cccs3)C(F)(F)F GK03142 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)c5ccc(cc5)[N+](=O)[O-] RH01735 c1cc(cc(c1)Cl)CNC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00080 c1ccc(c(c1)CNC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-])Cl DFP00083 c1cc(ccc1/C=N/c2ccc(cc2)Cl)C#N DFP00122 Cc1c(oc(n1)C)c2ccnc(n2)N SEW01615 COC(=O)C1Cc2c3ccccc3[nH]c2C4(N1)CCN(CC4)Cc5ccccc5 RH01562 CC(C)NC(=O)NNc1ccc(cc1)c2csnn2 SEW01044 c1cc(ccc1Sc2nc3ccc(cc3s2)Cl)Cl SEW01267 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)CS(=O)(=O)Cc4ccc(cc4)F)[N+](=O)[O-] SP00801 Cc1ccc(cc1)N2C(=O)c3c(nccn3)C2=O PD00082 c1cc2c(cc1NC(=O)COCC(=O)O)OCO2 PD00479 c1cc(ccc1CS(=O)(=O)Cc2nc(on2)c3ccc(cc3Cl)F)F SP00814 COc1ccc(cc1)Oc2cccc(c2CNC(=O)Nc3ccc(cc3)Cl)Cl CD11661 COc1c(c(ccn1)C(F)(F)F)C(=O)NCc2ccc(cc2Cl)Cl RF05056 CC(C)(C)NC(=S)NNC(=O)c1ccc(s1)c2ccc(cc2)Cl MBE00142 CCCNC(=O)O/N=C/c1cc(sc1)[N+](=O)[O-] DFP00098 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc(cc4)C SP00492 CN(C)c1c(cc(cc1F)C(=O)NC(=O)NCc2cccnc2)F SEW01893 COC(=O)c1cc(n(n1)c2ccccc2C(F)(F)F)O SEW00036 CC(C)N/C(=N/C#N)/SC SEW00053 CSc1c(c(sn1)SC)C(=O)NC(=O)NNc2ccc(c(c2)Cl)F SEW00166 c1ccc(cc1)N(Cc2c(cccc2Cl)F)NC(=O)c3ccc(cc3)Cl BTB06007 c1cc(oc1)C(=O)O/N=C(/Cc2cccs2)\N SPB08119 Cc1ccc(cc1)S(=O)(=O)c2c(scn2)Sc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] DFP00111 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)Nc3cccc(c3)C(F)(F)F)C(F)(F)F GK03100 Cc1ccccc1c2c3ccccc3c(=O)[nH]n2 BLT00216 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(o3)c4cccs4 SPB08127 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3cc(ccc3Oc4ccsc4C(=O)OC)C(F)(F)F GK03141 c1ccc(cc1)C(=O)c2cc3cc(cc(c3o2)Cl)Cl RH01797 c1cc(ccc1CS/C(=N/N)/N)C#N.Br DP00938 c1cc(c(cc1CNC(=O)c2c(ccnc2OCC(F)(F)F)C(F)(F)F)Cl)Cl RF05063 Cc1cc(cc(c1CNC(=O)c2c(ccnc2OCC(F)(F)F)C(F)(F)F)Cl)Cl RF05064 COc1ccc(cc1OC)/C=N/NC(=S)Nc2ccc(cc2)F RDR00445 CCN(CC)CCNC(=S)Nc1ccc(cc1)F RDR00467 c1ccc2c(c1)c(n[nH]2)C(=O)NN RH01089 c1ccc2c(c1)c(=O)nc(o2)c3c(c4ccccc4s3)Cl DSHS00610 C1CCc2c(c(c(sc2=S)N)C#N)C1 SEW00179 COC(=O)c1c(n(nn1)c2ccc(c(c2)Cl)F)SCc3c(cccc3Cl)F SEW00189 c1ccc(c(c1)S(=O)(=O)c2cscc2NC(=O)c3ccc(cc3)C(F)(F)F)Cl KM01991 CSC(=C(C#N)S(=O)(=O)C)SC KM01993 CC(C)(C)c1cc(n(n1)c2ccc(cc2Cl)C(F)(F)F)C(C)(C)C SEW06557 c1ccc(c(c1)F)S(=O)(=O)CC#N KM02055 c1cc(c(c(c1)Cl)CN2CCCN(CC2)C(=O)Nc3ccc(cc3)Cl)F AW00697 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCCN(CC3)Cc4c(cccc4Cl)F AW00745 c1cc(ccc1/N=N/c2ccc3c(c2)CCCN3CCC#N)Cl JFD03373 c1ccnc(c1)SCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06248 c1ccc2c(c1)ccc3c2cc(c(=O)o3)NC(=O)c4cccc(c4)[N+](=O)[O-] PHG00686 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Br)C(=O)O RH01536 c1cc(c(c(c1)Cl)SCCC(=O)c2ccc(s2)Cl)Cl MWP00769 Cc1c(c(n(n1)C(=O)NC)C)Cc2csc3c2cc(cc3)Cl MWP00820 Cc1c2c(cc(s2)C(C)(C)C)sc1c3nc(no3)c4ccc(cc4)C(C)(C)C GK03108 COc1ccc(cc1)CNC(=C2C(=O)c3ccccc3C2=O)C#N S11375 c1ccc(c(c1)C(=O)Nc2ccc(cc2Cl)Cl)[N+](=O)[O-] PD00343 CC(CO)NC(=O)OCC1c2ccccc2-c3c1cccc3 RJC04070 COc1ccc(cc1)C2N(C(=O)CS2)CCN3C(SCC3=O)c4ccc(cc4)OC PD00259 CSc1c(c(nn1S(=O)(=O)c2ccccc2)N)c3ccccc3 PD00263 c1cc(cc(c1)/C(=N/O)/N)COc2ccc(cc2)Cl KM01644 CC(C)Oc1cc(ccc1OC)C(=O)N KM09984 Cc1ccccc1C(=O)N2CCC(CC2)c3ccccc3OC RH01521 COCCCNC(=S)Nc1ccc(cc1Cl)Br RDR00271 c1cc(c(c(c1)Cl)Cl)/N=C\2/N(C(=O)CS2)Cc3ccco3 RDR00181 COc1ccccc1C2CCN(CC2)C(=S)Nc3ccc(cc3)Br RH01416 COc1ccccc1C2CCN(CC2)c3c(cccn3)[N+](=O)[O-] RH01423 c1cc(ccc1C(CC(=O)Nc2ccc(cc2F)I)CC(=O)O)C(F)(F)F PD00524 c1ccc(cc1)n2c(c(cn2)C(=O)NCCSCc3ccco3)C(F)(F)F KM10382 c1ccc(cc1)C(=O)Nc2cccc3c2cccc3 JFD03702 c1cc(cc2c1cc(cc2S(=O)(=O)[O-])S(=O)(=O)[O-])O.[K+].[K+] JFD03705 Cc1ccc(cc1)C2=NN=C(C=C(C2)c3ccccc3)c4ccc(cc4)C RJC04073 c1ccc2c(c1)CC(=C2)N3CCN(CC3)c4cccc(c4)C(F)(F)F RJC04075 Cc1ccc(cc1)n2c(nnn2)c3cnoc3c4cccs4 RJC04078 Cc1cccc(c1)NC(=O)c2cccc3c2cccc3 RH01558 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F RH01425 c1cc2c(cc1Cl)C3=C(CS2(=O)=O)C(=O)CCS3 SEW02187 c1cc(sc1)c2ccc(s2)C(=O)NC(=O)Nc3ccc(cc3)Cl SEW02555 CC(=O)c1nc2ccccc2s1 SEW02805 c1ccn(c1)c2ccc(cc2)C(F)(F)F SEW06045 Cc1c2ccccc2oc(=O)c1C#N JFD03729 Cc1nc(c(o1)C(F)(F)F)C(=O)NN RF04175 Cc1cc(no1)NCc2ccc(cc2)Cl RF03190 Cc1cc(ccc1NC(=N)NN)Cl.I RDR00163 COc1cc(c(cc1OC)NS(=O)(=O)c2c(cc(cc2Cl)Cl)Cl)C(=O)OC GK03104 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=S)Nc3ccc(cc3)Cl)C(F)(F)F GK03113 c1ccc2c(c1)cccc2c3nnc(o3)CN4CCCCC4 RH01455 COc1ccccc1C2CCN(CC2)C(=O)c3ccc(cc3)F RH01500 c1cc(ccc1S(=O)(=O)Cc2ccsc2C(=S)N)Cl SEW01702 Cc1c(oc(n1)C)c2ccnc(n2)C34CC5CC(C3)CC(C5)C4 SEW01751 COc1ccccc1C(=O)O/N=C(/COc2ccc(cc2Cl)Cl)\N SEW01974 CC(C)(C)c1ccc(cc1)NC(=O)NC(=O)c2csc(n2)c3ccc(cc3Cl)C(F)(F)F SEW01981 c1cc(c(nc1)SC2CC(=O)N(C2=O)c3ccc(cc3)OC(F)(F)F)C(=O)O PD00434 c1ccc(cc1)C(CNCc2csc3c2cccc3)O PD00436 Cc1c(cccc1Cl)S(=O)(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK03086 CCc1cccc(c1NC(=O)c2cnccc2C(F)(F)F)C RF04400 COc1ccccc1C2CCN(CC2)C(=O)c3ccc(cc3)N RH01667 c1ccc(cc1)CN(CCc2c[nH]c3c2cc(cc3)C#N)Cc4ccccc4 RH01669 COc1ccc(cc1OC2CCCC2)/C=N/O KM09286 CCOC(CN(Cc1ccc(c(c1)OS(=O)(=O)c2ccc(cc2)C)OC)S(=O)(=O)c3ccc(cc3)C)OCC RH01525 CC1(COC(OC1)c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)c4ccccc4OC)C RH01497 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCc2ccccc2 AW00882 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccc(nc2C)C(F)(F)F AW00884 c1cc(ncc1C(F)(F)F)S(=O)(=O)/C(=C/c2ccsc2)/C#N RF04737 c1cc(c(cc1F)Cl)c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SP00744 c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccc(cc3)F RH01559 COC(=O)c1c(ccs1)NC(=O)c2ccccc2 KM10201 C[C@@]1\2CCC(C1)C(/C2=N\O)(C)C RH01602 COC(=O)C(Cc1c[nH]c2c1cccc2)/N=C/c3ccccc3 RH01601 c1cc2c(cc1/C=N/O)OCO2 RH01603 c1ccc(cc1)NC(=O)NCCSCc2ccco2 KM10244 c1ccc(cc1)COc2ccc(cc2)n3cnnc3SCC(=O)Nc4ccccc4 SPB08047 COc1ccc(cc1)C(=O)N2CCC(CC2)c3ccccc3OC RH01530 c1ccc(cc1)n2c(ncn2)c3csc(n3)c4ccncc4 MWP01168 c1ccc(cc1)Oc2ccc(cc2)OC(=O)c3cccc(c3)[N+](=O)[O-] RH01569 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4cc(c(c(c4)C(C)(C)C)O)C(C)(C)C SP00542 Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2C(=O)OC)OC)OC GK03096 CC(C)c1ccc(cc1)Nc2cc(nn2C)O JM00030 c1cc(ccc1c2c(=O)[nH]c(=S)[nH]n2)Cl JM00201 CC(C)(C(=O)O)Oc1ccc2ccccc2c1 JM00276 CC(CN1CCN(CC1)c2ccccc2OC)N(c3ccccn3)C(=O)C4CCCCC4 RH01665 CC(=O)N(CC(=O)Nc1ccccc1C(=O)c2ccccc2)O RH01546 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)/C=C/c3ccccc3 PHG00759 c1cc2c(cc(nc2c(c1)F)C(F)(F)F)Oc3ccc(cc3)Cl KM09577 CC(C)(C)c1cc(n(n1)c2ccc(cc2)NC(=O)COCC(=O)O)C(C)(C)C SEW06193 c1cc(c(cc1Cl)OC(F)(F)F)NS(=O)(=O)C(F)(F)F SEW03596 Cc1c(c(on1)C)c2nc(no2)CS(=O)(=O)c3ccc(cc3)F SP00687 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)c4ccccn4)[N+](=O)[O-] SP00683 c1cc(c(c(c1)Cl)CSc2ncnc(n2)N)Cl JM00332 CN(C)C(=O)Oc1nnc(n1c2cccc(c2)Cl)SCc3ccccc3 SPB00583 Cc1ccc(cc1)c2nc(on2)c3ccno3 SP00918 c1ccc(c(c1)c2cc(c(o2)C(F)(F)F)c3nc(no3)c4ccc(cn4)C(F)(F)F)Cl SP00920 c1ccc(cc1)COc2ccc(cc2)NC(=O)NC3Cc4ccccc4C3 KM10450 CS(=O)(=O)/C(=C/c1cccn1c2ccc(cc2)C(F)(F)F)/C#N SEW06156 c1ccc(cc1)CSc2nncn2c3ccc4c(c3)OCCO4 SPB08042 Cc1c(cccc1NC(=O)NCc2ccccc2)C(=O)OC KM09949 CCCCNC(=O)O/N=C(\C)/c1ccc2cc(ccc2c1)OC SEW04550 Cn1c(nnc1/C(=C/N(C)C)/C#N)c2ccccn2 SEW04594 c1ccc(cc1)n2c(nnc2S)CSCc3cccc4c3cccc4 RH01662 CC(C)(C)c1ccc(s1)C(=O)Nc2cccc(c2)C#C MBE00203 c1ccc(cc1)NC(=O)Nc2ccc(cc2[N+](=O)[O-])Cl MGH00136 C1CCN(CC1)C(=O)C(Cl)(Cl)Cl SEW00140 c1ccc(cc1)C2C(NNC2=O)c3ccccc3 RH01553 c1cc(cnc1)CNC(=S)SCc2cc(sc2Cl)Cl CD11546 c1ccc(cc1)COc2cnc(nc2O)S RH01628 CC(=O)Nc1cc2cc(cc(c2oc1=O)Br)Br PHG00462 Cc1c(cccc1SC)NC(=O)NCc2ccccc2 KM10217 c1ccc(cc1)COc2ccc(cc2)n3cnnc3SCC(=O)c4ccc(cc4)C(F)(F)F SPB08049 CC(C)c1ccc(cc1)NC(=O)CSc2nncn2c3ccc4c(c3)OCCO4 SPB08043 Cc1ccc(cc1)SCCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06142 c1ccc(c(c1)/C=C\2/c3ccccc3NC2=O)N4CCOCC4 SEW05391 CC(C)(C)C(=O)Nc1cccc(c1)C(F)(F)F SEW03569 CC(C)(C)S(=O)(=O)Cc1nc(on1)c2ccc(cc2Cl)F SP00970 Cn1c(c(cn1)Br)NC(=O)c2ccc(cc2)Cl GK03429 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)NN3CCOCC3)C SPB08263 CCCCC#Cc1ccc(o1)C(=O)NN KM09492 CCCCC#Cc1cc(cnc1)c2nnc(n2C)S KM09483 c1cc(ccc1c2csnn2)NNC(=O)Nc3ccc(cc3)Cl SEW01042 c1cc(ccc1c2csnn2)C(F)(F)F SEW00669 c1cc(ccc1c2csnn2)OC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW01115 CCCCCCC#Cc1cc(cnc1)C(=O)NN KM09453 Cc1ccc(c2c1CCC2)OCC(=O)NN RH00591 CCc1cc2c(cc1c3csc(n3)NC(=N)N)C(CCC2(C)C)(C)C SEW06148 CCOC(=O)c1c(c(=O)[nH]c(=O)[nH]1)[N+](=O)[O-] RH00063 Cc1c(ccc2c1OC(CC2=O)(C)C)O RH01364 c1cc(cnc1)c2ccnc(n2)S MWP00580 COc1ccc(cc1)C2c3ccsc3CCN2S(=O)(=O)c4ccc(c(c4)Cl)F SEW01490 Cc1c(oc(n1)C)c2ccn(n2)C(=O)c3ccc(cc3)OC SEW01593 c1cc(cc(c1)F)c2csc(n2)c3ccc(cc3)C4SCCS4 SP00535 Cc1c2ccccc2sc1c3csc(n3)c4c(cc(cc4Cl)C(F)(F)F)Cl SP00536 c1ccc(cc1)c2csnn2 SEW00610 CC(=O)Oc1ccccc1/C=C/2\C(=O)OC(=N2)c3cc(c(c(c3)OC)OC)OC PHG00790 CCOc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cc(c(c(c3)OC)OC)OC PHG00785 CN(C)/C=N/c1nc(nn1c2ccccc2)SC SEW00536 CN(C)/C=N/c1nc(nn1c2c(cc(cc2Cl)Cl)Cl)SC SEW00537 c1cc(ccc1/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl)Cl PHG00629 COc1cc(c(cc1OC)N2C(=O)CCC2=O)C(=O)OC GK03185 COc1cc(c(cc1OC)NC(=O)CCCC(=O)O)C(=O)OC GK03187 Cc1ccc(c2c1CCC2)OCC(=O)NNC(=S)Nc3ccc(cc3)C(C)C RH00603 CCOC(=O)c1csc(n1)c2ccncc2 MWP00353 c1cc(cc(c1)NC(=O)Nc2csc(n2)Cc3ccsc3)C(F)(F)F MWP00404 CNC(=S)NNC(=O)c1csc(n1)Cc2ccsc2 MWP00530 Cc1c(c(n(n1)C(=O)Nc2ccc(cc2Cl)Cl)C)Cc3csc4c3cc(cc4)Cl MWP00821 c1ccc(c(c1)CSCC/N=C/c2cc(cc(c2O)Cl)Cl)Cl SEW06549 c1ccc2c(c1)c3ccccc3n2CC(CN4CCCC4)O JFD03700 CC(C)c1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl RH02043 Cn1cc(cc1C(=O)OC)/C=N/Nc2ccc(cn2)[N+](=O)[O-] SEW06554 Cn1cnnc1SCc2cccc3c2cccc3 RH01487 CSc1c(cccc1NC(=O)/C=C\C(=O)O)C(F)(F)F SEW03656 c1cc(cc(c1)Cl)CN/C(=C(/C#N)\N)/C#N KM00239 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3F)F PD00512 COc1ccccc1N2CCN(CC2)C(=S)Nc3cccc(c3)C(F)(F)F SEW06130 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)C#N)C(F)(F)F SEW06135 c1cc(cnc1)c2nc(cs2)C(=O)NO MWP00598 COc1ccccc1C2CCN(CC2)C(=S)Nc3cccc(c3)Cl RH01417 COc1ccccc1C2CCN(CC2)C(=S)Nc3ccc(cc3)F RH01418 COc1ccc(c(c1)c2nc(no2)c3ccccc3)Br SP00793 Cc1c(c(on1)C)c2nc(no2)c3ccccc3 SP00791 CC1=C(CC2C(C1)C(=O)N(C2=O)c3ccc(cc3)I)C PD00516 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2ccc(cc2)C#N PD00518 COc1cc(cc(c1)OC)NC(=O)CC(CC(=O)O)c2ccc(cc2)C(F)(F)F PD00519 c1cc(c2c(ccc3c2c1CC3)Br)[N+](=O)[O-] PHG00560 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2cccs2 PD00520 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00683 COc1ccc(cc1OC)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] PHG00487 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] PHG00624 COc1ccc(cc1OC)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PHG00610 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OC)[N+](=O)[O-] BTB07588 c1cc(c(cc1Cl)Cl)OCc2nc(on2)COc3ccc(cc3Cl)Cl SEW00558 CC1C/C(=N\O)/c2cc(ccc2S1(=O)=O)Cl SEW00564 CCCCC#Cc1cc(cnc1)C(=O)Nc2ccc(cc2)Cl KM09468 Cc1c2ccccc2sc1CNC(=O)Nc3ccc(cc3)OC(F)(F)F MWP00832 CCCc1ccc(cc1)c2nc(no2)c3ccccc3 SP00790 COc1ccccc1C2CCN(CC2)C(=O)Nc3ccccc3C#N RH01419 c1cc(ccc1C#N)S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06259 CCn1c2ccccc2c3c1ccc(c3)[N+](=O)[O-] JFD03684 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2cccs2 JFD03685 c1ccc(cc1)S(=O)(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH02042 COc1cc(c(cc1OC)N2C(=O)c3ccccc3C2=O)C(=O)OC GK03186 COc1cc(c(cc1OC)N2C(=O)CCCC2=O)C(=O)OC GK03188 Cc1cc(ccc1Br)N2C(=O)CC3(CCCC3)CC2=O PD00655 c1cc(ccc1/C=C/C(=O)Nc2ccc(cc2)Cl)OC(F)(F)F SEW06330 Cc1c(c(on1)C)c2nc(no2)CSc3ccccc3N SEW06331 CC(=O)Oc1cccc(c1)[N+](=O)[O-] RH01460 c1cc(cc(c1)OS(=O)(=O)c2c(cc(s2)Br)Br)C(F)(F)F SEW02672 CCCCC1(C(=O)c2ccccc2NC1=O)Cc3ccccc3 JFD03675 COc1ccccc1N2CCN(CC2)C(=O)Nc3ccc(cc3)C(F)(F)F SEW06138 CCCc1ccc(cc1)c2nc(no2)c3ccc(cc3)C(F)(F)F SP00738 Cc1c(oc(n1)C)c2ccn(n2)C(=O)c3ccc(cc3)Cl SEW01594 Cc1c(c(nc(c1C#N)S)C)CCC#N RF00409 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)c2c(c3ccccc3s2)Cl BTB00343 CCCCNC(=O)O/N=C(/Cc1cccs1)\N SPB08120 c1cc(c(cc1Cl)Cl)/C=C/C#N SEW02065 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4cccc5c4non5 KM10254 c1ccc(c(c1)C(=O)O)SC(CC(=O)c2ccc(cc2)F)c3ccc(cc3)F PD00288 CC1=CCC2C(C1)C(=O)N(C2=O)c3cc(cc(c3)OC)OC PD00505 c1ccc(c(c1)CSCCNC(=O)c2cccs2)Cl SEW06541 CC(C)(C)c1cc(n(n1)c2ccc(cc2)C(=O)O)C(C)(C)C SEW06547 c1cc(cc(c1)Cl)NC(=O)c2cccs2 JFD02667 Cc1ccnc(c1)NC(=O)c2cccs2 JFD02669 CC(C(=O)Nc1ccc(cc1)Cl)Oc2ccc(cc2)Oc3ccc(cc3)C(F)(F)F SEW06334 Cn1ccc(n1)c2ccc(cc2)Br KM02317 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SPB08130 CCCCC1(C(=O)c2ccccc2N(C1=O)c3ccccc3)O JFD03679 COC(=O)c1ccc(cc1)CNC(=O)Nc2cccc(c2)SC KM10210 c1cc(n(c1)c2ccc(cc2)C(F)(F)F)/C=N/NC(=O)N SEW06159 CN(C)c1ccc(cc1C#N)/C=C(\C#N)/S(=O)(=O)c2ccccc2 SEW06144 CC(C)(C)c1ccc(cc1)C(=O)Nc2c(c([nH]n2)SC)c3ccccn3 PD00176 c1ccc2c(c1)c(cn2C(=O)C3CCC3)/C(=C/c4ccc(cc4)C(F)(F)F)/C#N PD00186 CC(C)(C)C(=O)Cn1c(=O)c2ccccc2nc1SC PD00220 CC(c1ccccc1)NC(=O)c2cccs2 JFD02668 c1ccc(c(c1)C(=O)Nc2ccccc2C(F)(F)F)I JFD02673 COc1ccc(cc1OC)C(=O)Nc2ccccc2 JFD02674 CCCCc1ccc(cc1)NC(=O)c2cc(c(c(c2)OC)OC)OC JFD02688 CC(=O)N(CC(=O)Nc1ccccc1C(=O)c2ccccc2)OC(=O)C JFD04008 CC1CN(CC(O1)C)c2cc(c(cc2F)[N+](=O)[O-])N(C)C BTB03947 COc1cc2c(cc1OC)C(NC(=O)C2)c3ccc(cc3)Cl JFD03699 c1cc(sc1c2cc(ccn2)C(F)(F)F)S(=O)(=O)N3CCCC3 SEW03893 c1ccc(c(c1)NC(=S)NCc2ccc(cc2)C#N)Cl CD01716 c1ccc(cc1)C(=O)NC(c2ccccc2O)C(c3ccccc3O)NC(=O)c4ccccc4 JFD03673 Cc1c(c(oc(=O)c1Br)C)C(=O)OC KM09771 c1cc(ccc1F)S(=O)(=O)Cc2nc(on2)c3ccno3 SP00693 COc1ccccc1NC(=O)c2ccc(c(c2)OC)OC JFD02675 COc1ccc(c(c1C(=O)NC(=O)Nc2ccc(c(c2)Cl)Cl)OC)[N+](=O)[O-] BTB07577 CCCc1ccc(cc1)S(=O)(=O)C[N+](=O)[O-] SPB03873 c1cc(ccc1c2cc(n(n2)c3ccc(cc3)F)NC(=O)C4CCC4)Cl SP00983 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cc(nn3c4ccc(cc4)F)c5cccs5 SP00995 c1cc(sc1)SC/C(=N/O)/N KM02320 CC1(C2CCC1(C(C2)N3CCNCC3)C)C.Cl.Cl RH01561 c1ccc(cc1)C2=CC(=NN=C(C2)c3ccc(cc3)Cl)c4ccc(cc4)Cl RJC04074 CCc1cc2c(cc1c3csc(n3)N)C(CCC2(C)C)(C)C SEW06147 c1ccc(cc1)C(CC(=O)O)N RH01533 COc1cc(c(cc1OC)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)OC GK03097 Cn1c2ccccc2c3c1CCC(C3=O)CN(C)C JFD04011 COc1cc(c(cc1OC)NC(=O)CCC(=O)O)C(=O)OC GK03182 c1cc(oc1)CSCCNC(=O)CSc2ccc(cc2)F KM10437 c1cc(oc1)CSCCNC(=O)CSc2cccs2 KM10445 COc1ccc(cc1)C(=O)c2cc3cc(cc(c3o2)Cl)Cl RH01786 Cc1cc(c(c2c1CCC2)OCc3nnc(n3CC=C)S)Br RH01795 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2ccc(cc2)C(C)(C)C SEW06245 Cc1ccc(cc1)C(=O)Oc2cccc3c2nccc3 SEW06247 Cc1cccc(c1)NC(=S)NNC(=O)CSCc2cccc3c2cccc3 RH01646 c1ccc(cc1)n2c(nnn2)c3cnoc3c4cccc(c4)Cl RJC04076 c1ccc(cc1)n2c(nnn2)c3cnoc3c4cccs4 RJC04077 CCOc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] PHG00623 c1cc(sc1)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] PHG00799 c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4 KM09689 COc1ccccc1N2CCN(CC2)CCCCNC(=S)Nc3cc(cc(c3)Cl)Cl SEW06198 COc1cc(c(cc1OC)NS(=O)(=O)c2ccc(c(c2)F)F)C(=O)OC GK03106 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2ccccc2OC(F)(F)F SEW06243 COc1ccccc1N2CCN(CC2)C(=O)c3cc(c(c(c3)OC)OC)OC SEW06049 COc1ccc(c(c1)c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Br SP00729 Cc1ccc(cc1)S(=O)(=O)N/N=C\2/CCCCCCCCCCC2CCC#N RH01478 c1ccc(cc1)CCCCN2CNC(=S)NC2 RH01222 CC(C)Cc1ccc(cc1)C(C)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06250 c1ccc(cc1)NC(=S)NNC(=O)CSCc2cccc3c2cccc3 RH01644 COC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)c3cccc(c3)[N+](=O)[O-] RH01655 c1cc(cc(c1)NC(=O)CSc2nncn2c3ccc4c(c3)OCCO4)C(F)(F)F SPB08044 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCC(CC3)c4ccccc4OC RH01519 c1ccc(cc1)C(=O)/C(=N/Nc2ccccc2)/C#N JFD03727 CC(=O)Oc1ccccc1/C=C/2\C(=O)OC(=N2)/C=C/c3ccccc3 PHG00751 CC(=O)Oc1ccccc1/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00688 CCOc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00682 CC(C)c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] PHG00488 COc1ccc(c(c1)NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)c4ccccc4OC)OC RH01573 CCc1cc2c(cc1c3csc(n3)c4ccc(cc4)C(C)(C)C)C(CCC2(C)C)(C)C SEW06151 COc1ccc(cc1OC)S(=O)(=O)N(CCCC#N)Cc2ccco2 KM09250 COc1ccc(cc1OC)S(=O)(=O)N(CCC#N)C2CCc3c2cccc3 KM09308 Cc1c(c(on1)C)C(=O)O/N=C(/c2cccc(c2)C(F)(F)F)\N SEW05949 c1ccc2c(c1)c(=O)n(c(n2)SCC(=O)c3ccc(cc3)Cl)CC(=O)c4ccc(cc4)Cl PD00227 CSc1nn(c(=S)s1)CSc2[nH]c(nn2)c3ccccc3F SPB03274 Cc1c(c(no1)C(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F)c3csc(n3)C SPB03396 Cc1c(c(on1)C)C(=O)Oc2cccc3c2nccc3 SEW06256 CC(C)Cc1ccc(cc1)C(C)C(=O)O/N=C(/c2ccc(cc2)Cl)\N SEW06199 Cc1ccc(cc1)/C(=N/OC(=O)C(C)c2ccc(cc2)CC(C)C)/N SEW06201 CC(C)Cc1ccc(cc1)C(C)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N SEW06202 Cc1cc(n(n1)c2ccc(cc2)n3cccc3C=C(C#N)C#N)C SEW04328 CCCc1ccc(cc1)c2nc(no2)c3ccc(cn3)C(F)(F)F SP00733 CCOC(=O)C1=c2n(c(=O)/c(=C\c3ccc(cc3)C(=O)OC)/s2)C(=C(C1c4ccc(cc4)C(=O)OC)C#N)N JFD03726 COc1ccc(c(c1)c2nc(no2)CS(=O)(=O)c3ccc(cc3)F)Br SP00690 c1cc2cccnc2c(c1)OC(=O)c3c(cccc3F)F SEW06251 COc1cccc(c1)C(=O)Oc2cccc3c2nccc3 SEW06253 COc1cc(c(cc1OC)NS(=O)(=O)c2ccc(cc2Cl)Cl)C(=O)OC GK03102 Cc1cccc(c1)c2nc(on2)c3cc(oc3C(F)(F)F)c4ccccc4Cl SP00943 Cc1ccc(c(c1)C)Nc2c(c(c(s2)C(=O)c3ccc(cc3)Br)N)C(=O)N DP00041 c1ccc(cc1)COc2ccc(cc2)n3cnnc3SCC(=O)Nc4cc(cc(c4)Cl)Cl SPB08048 c1ccc(cc1)CN2c3ccccc3C(C2=O)c4ccccc4 RH01003 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccc(cc2)[N+](=O)[O-] RH01406 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2Cl)N(C)C RDR00436 CCC1CS/C(=N/c2c(cccc2C)C)/N1 RDR00434 COc1ccc(cc1)NC(=S)NCCNC(=S)Nc2ccc(cc2)OC RDR00482 c1cc(ccc1NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)OC(F)(F)F SEW06042 CCOC(=O)c1cc(=O)c2ccccc2o1 GK03111 C[C@@]12CC(CCN1CCc3c2cccc3)O RH01470 c1cc(cc(c1)NC(=S)NCCNC(=S)Nc2cccc(c2)C(F)(F)F)C(F)(F)F RDR00485 CC(C)(CO)NC(=S)Nc1ccccc1F RDR00457 c1ccc2c(c1)cccc2c3nnc(o3)CN4CCOCC4 RH01488 CN1CCC2(CC1)c3c(c4ccccc4[nH]3)CC(N2)C(=O)OC RH01524 Cc1cc(n(n1)c2ccc(cc2)n3cccc3/C=C(/C#N)\S(=O)(=O)c4ccccc4)C SEW04339 c1ccc(cc1)C(=O)c2c(cc(cc2Cl)C(F)(F)F)Cl SEW05088 c1cscc1c2n[nH]nn2 SEW05173 c1cc2cccnc2c(c1)OC(=O)c3ccc(cc3)Cl SEW06254 c1c2c(nc3c1C(=O)CCC3)CCCC2=O RH01555 COc1ccccc1C2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] RH01430 Cn1c(nnc1S)c2ccc3c(c2)non3 KM09671 COC(=O)c1ccc2c(c1)cccn2 KM10245 CC(C)(C)c1ccc(cc1)NC(=O)NCCSCc2ccco2 KM10248 Cc1ccc(cc1NC(=O)N(Cc2ccccc2)C(=O)CC#N)SC KM10237 c1cc(n(c1)c2ccc(cc2)C(F)(F)F)C=C(C#N)C#N SEW06155 Cc1ccc(c2c1CCC2)OCC(=O)N/N=C/c3cccc(c3)OC RH00604 c1cc(ccc1c2c([nH]nn2)C#N)OC(=O)c3ccc(cc3)Cl SEW03772 CCCS(=O)(=O)c1ccc(cc1)[N+](=O)[O-] MWP00962 c1cc(c(cc1Cl)Cl)C2(CC2)/C(=N/O)/N SEW03871 Cn1cnc(n1)c2ccccc2NS(=O)(=O)c3ccc(cc3)Cl MWP01083 Cc1ccc(c(c1)C(=O)N/N=C/c2cccs2)[N+](=O)[O-] BTB01691 Cc1ccc(c(c1)C(=O)N/N=C/c2cccnc2)[N+](=O)[O-] BTB01690 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F GK03112 CCC\1(CCCC/C1=N\O)c2cccc(c2)OC RH01433 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SP00740 c1ccnc(c1)c2nc(on2)c3ccc(cc3Cl)F SP00737 c1cnoc1c2nc(no2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SP00739 CCOC(=O)c1ccccc1NC(=O)CN2CCOCC2 RH01149 c1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4cccs4 RH01153 Cc1c(cccc1Cl)NC(=O)NCCSCc2ccco2 KM10258 c1cc(oc1)CSCCNC(=O)Nc2ccc(cc2)Cl KM10260 COc1ccc(cc1NC(=O)NCCSCc2ccco2)Cl KM10251 CCOC(=O)N/N=C(\C)/c1ccc(cc1)Cl SEW03374 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=C/C(=O)NCc4ccccc4 RH01572 CCOc1cc(cnc1C(=N)N)C(F)(F)F SEW03911 CC(C)(C)OC(=O)NC(COCc1ccccc1)C(=O)NC RJC03774 c1cc(cc(c1)Oc2ccc(cn2)C(=O)NN)C(F)(F)F SPB03971 c1cc(c(cc1)O)/C=N/C(C(/N=C/c2c(cccc2)O)c3c(cccc3)O)c4c(cccc4)O JFD03677 c1cc(ccc1Oc2cc(nc3c2cc(cc3)Cl)C(F)(F)F)Cl KM09576 c1cc([nH]c1)C(CN)C(F)(F)F SEW04444 c1ccc(cc1)C(C(c2ccccc2)Nc3ccc(cc3)Cl)C(=O)c4ccccc4 SEW04923 c1ccc2c(c1)c(c[nH]2)CN3CCC(CC3)NC(=O)C4CCCCC4 RH01629 Cc1c(cc(o1)C(C)(C)C)c2nc(no2)c3ccc(cc3)OC(F)(F)F SP00823 c1ccc(cc1)SCCC(=O)c2ccc(s2)Cl MWP00770 COc1ccc(cc1)NC(=S)N2CCC(CC2)c3ccccc3OC RH01415 Cc1ccc(n1c2ccc(cc2)n3c(cc(n3)C)C)C SEW04172 c1cc2c(c(c1)F)c(c3c(n2)OCCC3)N SEW04213 COc1cccc(c1)Oc2ccc(cc2C(=O)OC)OC SEW06257 CC(C)(C)S(=O)(=O)Cc1nc(on1)c2cc(ccc2Oc3ccc(cc3)OC)[N+](=O)[O-] SP00968 c1cc(ccc1C(F)(F)F)S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06036 c1ccc(cc1)CNS(=O)(=O)c2ccc(cc2)Cl CD11324 CCOc1ccc(cc1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06037 COC(=O)c1ccccc1NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06038 c1ccnc(c1)c2nc(on2)C3CCC3 SP00721 CCOc1ccc(cc1)NC(=S)N2CCC(CC2)c3ccccc3OC RH01420 c1ccc(cc1)NC(=O)NNC(=O)c2ccc3c(c2)cccn3 KM10273 Cc1ccc(cc1NC(=O)NCc2ccccc2)SC KM10227 Cc1c(sc(n1)c2ccccc2)C(=O)/C=C/N(C)C SEW04135 Cc1cc(n(n1)c2ccc(cc2)n3cccc3)C SEW04171 c1ccc(c(c1)c2cc(c(o2)C(F)(F)F)c3nc(no3)c4cccs4)Cl SP00930 CS(=O)(=O)N1CCN(CC1)c2c(cccn2)C(F)(F)F SEW06264 Cn1c(c(cn1)Br)NC(=O)Nc2ccccc2 GK03235 c1ccc(c(c1)CSCCNS(=O)(=O)c2c(c(sc2Cl)Cl)Br)Cl SEW06560 CSCCC(CC(=O)O)NC(=O)c1cccs1 KM01570 Cc1c(csc1C(=O)NN)S(=O)(=O)c2ccc(cc2)Cl KM01373 c1cnoc1c2nc(no2)CS(=O)(=O)c3ccsc3 SP00917 Cc1ccc(n1c2ccc(cc2)/C=C/3\c4ccccc4NC3=O)C SEW06561 c1cc(cc(c1)C(F)(F)F)CSCCNC(=O)c2ccc(cc2)Cl SEW06562 Cc1c(c(on1)C)S(=O)(=O)N(Cc2ccc(cc2)OC)Cc3ccc(cc3)OC SEW04969 c1cc(ccc1C(=O)NCc2c(cc(cc2Cl)C(F)(F)F)Cl)C(F)(F)F SEW05111 CC(C)(C)OC(=O)NC(COCc1ccccc1)C(=O)N RJC03773 COc1ccc(cc1)OS(=O)(=O)c2c(cc(s2)Br)Br SEW02682 c1ccc2c(c1)c(c([nH]2)c3ccc(cc3)Cl)/C=N/O SEW03054 c1cc(ccc1c2nc(on2)c3ccc(cc3Cl)F)OC(F)(F)F SP00827 c1cc(c(cc1F)Cl)c2nc(no2)c3ccc(cn3)C(F)(F)F SP00831 CN(C)c1ccc(cc1C#N)/C=N/NC(=S)N SEW06145 COc1ccc(cc1OC)S(=O)(=O)N(CCC(=O)O)Cc2ccco2 KM09277 c1cc(oc1)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06265 CC(C)(C)C(=O)N1CCN(CC1)c2ccc(cn2)C(F)(F)F SEW06267 c1ccc(c(c1)C(=O)O)NCC(=O)O JFD03681 c1csc(c1)/C=C\2/C(=O)/C(=C/c3sccc3)/COC2 PD00648 CC(=O)N1CCC(CC1)c2nc(no2)c3cccs3 SEW06536 CCNS(=O)(=O)c1ccc(cc1)F CD11336 CCn1c(c(c(n1)C)Br)c2nc(no2)c3ccc(cn3)C(F)(F)F SP00830 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4ccc(cn4)C(F)(F)F SP00829 COc1ccc(cc1)Oc2cccc(c2CNS(=O)(=O)c3ccc(cc3)OC)Cl CD11663 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C4OCCCO4 RH01485 Cc1cc(n(n1)c2ccc(cc2)n3cccc3/C=C(/C#N)\C(=O)OC)C SEW04333 Cc1ccc(cc-2c(cc(c12)C#N)C)C(C)C SEW04828 CCOC(=O)/C(=N/NC(=O)OCC)/C SEW00613 COC(=O)/C(=C/c1cccn1c2ccc(cc2)C(F)(F)F)/C#N SEW06157 CC1(OC(=O)C(=Cc2cccn2c3ccc(cc3)C(F)(F)F)C(=O)O1)C SEW06158 COc1ccc(c(c1OC)Cl)/C=C/c2nc(no2)c3ccc(cc3)OC(F)(F)F SP00818 COc1cc2c(cc1OC)ncnc2Sc3ccc(cc3)Cl GK03232 c1nc2c(c3c(s2)CCCC3)c(n1)SCC(=O)NN GK03233 c1ccc2c(c1)CC(C2)NS(=O)(=O)c3cc(ccc3Cl)C(F)(F)F KM10507 COc1cc(c(cc1OC)NC(=O)c2ccccc2C(=O)O)C(=O)OC GK03184 CCCCC#Cc1ccc(o1)C(=O)O KM09503 Cc1ccc(n1c2cc(c(cc2C(=O)NN)OC)OC)C GK03223 COc1cc2c(cc1OC)ncnc2SCC(=O)NN GK03234 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=S)N SEW03586 Cc1cccc(c1)n2c(=O)c3c(cccc3F)oc2=O RDR03929 Cc1ccc(cc1)NC(=O)c2c(nccn2)C(=O)O PD00079 COc1cc2c(cc1OC)C(NC(=O)C2)c3ccc(cc3Cl)Cl JFD03698 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)I PD00508 c1cc(cc(c1)Cl)C(=O)OCCSc2ccc(cn2)Cl BTB08982 Cn1c(ccn1)NC(=O)/C(=C/c2cccc(c2)Cl)/C#N GK03074 c1ccc(cc1)C(=O)O/N=C(/COc2ccc(cc2Cl)Cl)\N SEW01975 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C(/COc2ccc(cc2Cl)Cl)\N SEW01976 CCn1c(c(c(n1)C)Br)c2nc(no2)c3cccc(c3)C SP00842 CC(C)(C)CN/C(=C(/C#N)\N=C\c1cccc(c1)Cl)/C#N KM00229 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)Nc3ccc(cc3)OC SP00315 c1cc(oc1)CSCCNC(=O)Nc2cc(cc(c2)Cl)Cl KM10261 CSc1ccc(cc1)NC(=O)NCc2cccnc2 PD00322 COc1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccc(cc3)OC)/CN(C2)Cc4ccccc4 PD00326 CCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)C(F)(F)F JFD03374 c1cc(cc(c1)/N=C/c2ccc(cc2)Cl)C(F)(F)F DFP00184 CC(C)NC(=O)O/N=C/c1cc(sc1)[N+](=O)[O-] DFP00099 c1cc(ccc1/C=N/c2cc(cc(c2)Cl)Cl)Cl DFP00123 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)c5ccc(cc5)F RH01737 Cc1ccc(cc1)S(=O)(=O)c2c(scn2)SCc3ccc(cc3Cl)Cl DFP00109 COc1ccc(cc1OC)S(=O)(=O)Nc2cccc(c2)c3nnco3 SEW01332 c1cc(ccc1CS(=O)(=O)CC(=O)NN)c2csnn2 SEW01532 CCNC(=O)C(COCc1ccccc1)NC(=O)OC(C)(C)C RJC03775 CC(C)(C)OC(=O)NC(COCc1ccccc1)C(=O)NCc2ccccc2 RJC03776 CC(C)(C)OC(=O)NC(CSCc1ccccc1)C(=O)N RJC03777 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SC RH01739 CC(C)COC(=O)c1cn(c2ccccc2c1=O)C3CCCCC3 RH01729 CC1(OC2[C@H](OC(C2O1)[n@]3cnc4c3ncnc4N)CO)C KM09669 CCc1cc2c(cc1c3csc(n3)c4ccc(cc4)F)C(CCC2(C)C)(C)C SEW06150 COc1ccccc1C2CCN(CC2)C(=S)Nc3ccccc3 RH01413 CSc1c(c(nn1S(=O)(=O)c2ccccc2)N)c3cccs3 PD00267 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)Nc3cccc(c3)[N+](=O)[O-] SP00316 CCCCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)Br JFD03371 c1ccc(cc1)COC(=O)NCC(=O)ON2C(=O)CCC2=O KM10114 Cc1c(c(n(n1)c2ccccc2)C)c3nc(no3)c4cccc(c4)Cl SEW04215 Cc1c(snn1)C(=O)N2CCN(CC2)c3ccccc3OC SEW06052 COc1ccc(cc1)OCCNC(=O)c2ccccc2C(F)(F)F SPB08254 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc(cc3)Cl)C SPB08259 COC(=O)c1c(ccs1)Oc2ccc(cc2N3C(=O)C=CC3=O)C(F)(F)F GK02199 COCCCNC(=S)N1CCN(CC1)c2ccccc2OC SEW06152 CC(C)(C)c1ccc(cc1)NC(=O)NC2Cc3ccccc3C2 KM10452 Cc1c2cc(ccc2sc1C(=O)/C(=C/c3ccccc3)/C#N)Cl MWP00553 c1ccc2c(c1)c(cs2)CNS(=O)(=O)c3ccc(cc3)F PD00429 Cn1c2c(cnc(n2)c3ccc(cc3)C(F)(F)F)c(=O)n(c1=O)C S13811 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4ccc(cc4)C(F)(F)F SP00849 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)c4cnccn4)[N+](=O)[O-] SP00847 c1cc(c(c(c1)Cl)CSCC(=O)NCCSCc2ccco2)F KM10380 COc1cccc(c1)SCC(=O)NCCSCc2ccco2 KM10381 c1ccc(cc1)CN2CCCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl AW00798 c1cc(c(cc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)Cl)Cl SEW06252 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccc4c(c3)OCO4 PD00514 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2ccc(c(c2)OC)OC PD00517 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)C4C5CC(C4C(=O)O)C=C5)C(F)(F)F SEW06165 CC(C)(C)NCC(COc1ccc(cc1)c2csnn2)O SEW01605 COc1ccc(cc1)C(=O)O/N=C(/COc2ccc(cc2Cl)Cl)\N SEW01973 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)CS(=O)(=O)Cc4ccco4)[N+](=O)[O-] SP00838 CC(C)Sc1ccc(cc1[N+](=O)[O-])C(=O)OC KM10168 CC(C)(C)OC(=O)NC1CCN(CC1)Cc2c(cccc2Cl)F AW01031 c1ccc(cc1)CN2CCCN(CC2)S(=O)(=O)c3ccc(cc3)Cl AW01033 CC(C)Sc1c(cc(cc1[N+](=O)[O-])[N+](=O)[O-])C(=O)O KM10145 c1cnc(nc1)N2CCNCC2.Cl JFD03711 c1ccc(cc1)[C@H](C(=O)O)N JFD03710 c1ccc(cc1)C(=O)N2CCN(CC2)CCOc3ccccc3 TB00002 Cc1c(c(=O)n(n1C)c2ccccc2)N/C(=C/C#N)/C JFD03827 CCCCN(CCCC)c1ccc(cc1)/N=N/c2ccc(cc2)[N+](=O)[O-] JFD03377 c1cc(ccc1/C=C/c2nc(no2)c3ccc(cc3)Cl)OC(F)(F)F SEW06324 c1ccc2c(c1)CC(C2)NS(=O)(=O)c3cccc4c3non4 KM10504 c1ccc2c(c1)c(c(c(=O)o2)Cc3c(c4ccccc4oc3=O)O)O PD00769 Cn1c(c(cn1)C(=O)O/N=C/c2ccc(cc2Cl)Cl)n3cccc3 GK03590 Cc1c(c(nc(n1)c2ccccn2)NC)Cl SEW02968 Cc1c(c(nc(n1)c2ccccn2)NCCc3ccccc3)Cl SEW02975 CCOC(=O)/C(=N/Nc1ccc(cc1)F)/C RH01820 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2cccs2 AW01048 c1ccc(cc1)C(=CN2CCC2)c3ccccc3 RH01823 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccccc3 GK03594 c1ccc2c(c1)c3c([nH]2)C4(CCCCC4)NCC3.Cl.Cl RH01529 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCCNC(=O)OC(C)(C)C AW00881 CC(C)(C)SCCC(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl SEW06168 c1ccc(cc1)CN2CCC(CC2)N3C(=O)C=CC3=O PD00549 Cc1ccc(n1c2cc(c(cc2C(=O)NNC(=O)c3ccccc3)OC)OC)C GK03216 c1cc(c(cc1F)Cl)c2nc(no2)CS(=O)(=O)c3ccsc3 SP00798 C/C(=C\C=C\c1ccccc1)/C=C/c2ccccc2 RJC03803 Cn1c(c(cn1)C(=O)O/N=C/c2c(cccc2Cl)F)n3cccc3 GK03591 Cn1c(c(cn1)C(=O)O/N=C/c2ccc(cc2)OC(F)(F)F)n3cccc3 GK03592 COc1ccccc1NC(=O)c2cc(c(c(c2)OC)OC)OC JFD02685 Cc1ccc(cc1C)n2c(cc(n2)c3ccc(cc3)OC(F)(F)F)NS(=O)(=O)c4cccc(c4)F SP01023 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NC(=O)c4cc(oc4C)c5ccc(cc5)Cl SP01027 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NC(=O)Nc4ccccc4C#N SP01028 COc1ccccc1N2CCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl SEW06137 CCC(C)CNC(=S)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl SEW06141 COc1ccc(c(c1)c2nc(no2)c3ccc(cc3)C(F)(F)F)Br SP00811 C=CCC1(CCCCC1)NCc2ccccc2 JFD03354 CC\1C(NC(C/C1=N/O)c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3)[N+](=O)[O-] JFD03367 Cc1c(c([nH]n1)c2c(nns2)C)C(=O)NN SPB02132 CCn1c(c(c(n1)C)Br)c2nc(no2)CS(=O)(=O)c3ccsc3 SP00794 CC(C)Cc1ccc(cc1)C(C)C(=O)O/N=C(/c2ccc(cc2)OC(F)(F)F)\N SEW06200 CC(C)Cc1ccc(cc1)C(C)C(=O)NNC(=O)c2ccccc2C(F)(F)F SEW06203 c1ccc(cc1)C(=O)/C(=N/Nc2ccccc2)/C=N/Nc3ccccc3 JFD03773 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NC(=O)Nc4ccc(cc4)OC(F)(F)F SP01029 c1cc(cc(c1)S(=O)(=O)Nc2cc(nn2c3ccc(cc3)I)c4cccs4)F SP01006 c1cc(ccc1OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl SEW06172 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccccc3OC SEW06050 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2ccc(cc2)Cl SEW06244 COc1ccc(cc1)NN=C(C#N)C#N PD00168 CNC(=O)NNC(=O)c1cccnc1 JM00237 CCn1c(cc(n1)C)/C(=N/OC(=O)c2ccc(cc2)C(C)(C)C)/N SPB01885 Cc1cccc(c1)c2nc(on2)c3ccc(c(c3)OC)OC SP00840 c1cc(ccc1c2nc(on2)c3ccc(cc3Cl)F)C(F)(F)F SP00845 c1cc(cc(c1)[N+](=O)[O-])NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW06197 c1cc(cc(c1)Cl)/C=C(\C#N)/c2cccc(c2)Cl RDR01477 CN(C)N1C(=O)c2cccc3c2c(ccc3)C1=O PHG00957 c1cc(ccc1/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-])Cl PHG00622 COc1ccc(cc1)C2=C(/C(=C/N3CCOCC3)/N=C2)[N+](=O)[O-] SEW04077 Cc1ccc(cc1)NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW06169 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc(cc3)F)Cl SEW05357 c1cc(n(c1)c2ccc(cc2)C(F)(F)F)/C=N/NC(=S)N SEW06164 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N3CCN(CC3)c4ccccc4OC SEW06153 Cc1c(sc(n1)c2cccnc2)C(=O)NN SPB02180 Cc1cc(n(n1)C(C)(C)C)C(=O)NN SPB03143 CN(C)/C=C/C(=O)c1cc(no1)c2ccc(cc2)Cl SPB05039 Cc1cccc(c1)c2nc(on2)c3ccc(cc3Cl)F SP00851 c1cc(c(c(c1)Cl)c2nc(on2)c3ccc(cc3)OC(F)(F)F)Cl SP00850 COc1ccc(cc1OC)c2cc(n3c(n2)cc(n3)c4cccs4)C(F)(F)F KM10334 Cc1c(c(on1)C)c2nc(no2)c3ccc(cc3)C(F)(F)F SEW05955 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3ccco3)C(F)(F)F GK03085 CC1=CC(=O)N(C1=O)c2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK02197 c1cc2cccnc2c(c1)OC(=O)c3cccs3 SEW06255 COc1ccc(c(c1)c2nc(no2)c3ccc(cn3)C(F)(F)F)Br SP00715 Cc1c(c(on1)C)c2nc(no2)c3ccc(cn3)C(F)(F)F SP00718 c1cc(cc(c1)Cl)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl SEW05355 C/C(=N\NC(=O)CC#N)/c1ccc(cc1)OC RJC03927 COc1ccc(cc1O)/C=N/NC(=O)CC#N RJC03929 c1cc2c(cc1c3cc(nc(n3)N)C(F)(F)F)OCO2 KM10341 c1cc2c(cc1c3cc([nH]n3)C(F)(F)F)OCO2 KM10339 CN1C2CCC1CC(C2)NCc3ccccc3 JFD04003 c1ccc(cc1)Cn2c(=O)c3ccccc3[nH]c2=O S12249 c1cc(ccc1F)SCCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06180 c1ccc(cc1)OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06181 CN(C)c1ccc(cc1C#N)/C=C\2/C(=NOC2=O)c3ccccc3 SEW06183 c1cc(ncc1C(F)(F)F)N2CCN(CC2)c3ccc(cn3)N SEW05965 COc1cc(cc(c1)OC)N2C(=O)CC(CC2=O)c3ccc(cc3)C(F)(F)F PD00525 CSc1cccc(c1)NC(=O)CC(CC(=O)O)c2ccc(cc2)C(F)(F)F PD00526 c1ccc(c(c1)c2nn(c(=O)o2)c3ccc(cn3)C(F)(F)F)Cl RF04824 COc1ccc(cc1)NC(=S)N/N=C/c2cccnc2 RDR01026 CC(C)(C)NC(=S)N/N=C/c1ccccc1Cl RDR01114 Cc1ccc(cc1F)NC(=O)/C=C/C(=O)O RDR01189 COc1ccc2cc(ccc2c1)c3cc(nc(n3)N)C(F)(F)F KM10342 COc1ccc(cc1S(=O)(=O)NCCSCc2ccco2)Cl KM10350 COc1ccc(c(c1)O)/C=N/CCc2cccs2 S12729 c1ccc2c(c1)cn(c2C#N)Cc3cccc(c3)Cl S12800 c1ccc2c(c1)cnn(c2=O)c3ccc(cc3)S(=O)(=O)N PD00585 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=N)N3CC(OC(C3)C)C CD07836 Cn1c(c(cn1)C(=O)O/N=C(\c2ccccc2)/c3ccccc3N)n4cccc4 GK03589 C=CCNC(=S)N1CCc2c3ccccc3[nH]c2C1C(F)(F)F SEW06188 C=CCC(c1ccco1)NCc2ccccc2 JFD03356 c1ccc(cc1)C2CC(CC3(N2)CCCCC3)O JFD03358 c1cc(sc1)/C(=N/OC(=O)/C=C/c2ccc(cc2)OC(F)(F)F)/N SEW06313 COc1ccccc1C2CCN(CC2)c3ccc(c(c3)C(F)(F)F)[N+](=O)[O-] RH01456 COc1ccccc1C2CCN(CC2)c3ccc(c(c3)OC)[N+](=O)[O-] RH01429 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3cc(oc3C(F)(F)F)c4ccccc4Cl SP00947 CN(C)/C=C\1/C(=NNC1=O)c2ccccc2 JFD03756 c1cc(oc1)CSCCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM10352 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2I JFD02699 Cc1cc(c(c(c1)C)NC2=NC(CS2)(CO)CO)C S13263 CCC(C(c1cc(cc(c1)OC)OC)c2c(n(c(=O)n(c2=O)C)C)N)[N+](=O)[O-] S13372 Cc1c(c(nc(n1)SCc2c(cccc2Cl)Cl)O)Oc3ccc(cc3)Cl SPB03978 Cc1c(c(on1)C)C(=O)NNC(=O)c2ccc(cc2)OC SEW05940 c1ccc2c(c1)c(cs2)CNC(=O)C3CC3 PD00425 Cn1c(ccn1)NS(=O)(=O)c2ccc(cc2)NC(=O)C(F)(F)F GK03077 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2Oc3ccsc3C(=O)OC)C(F)(F)F GK03080 COC(=O)c1c(ccs1)Oc2ccc(cc2NS(=O)(=O)c3ccc(cc3)F)C(F)(F)F GK02204 COc1ccccc1c2nn(c(=O)o2)c3c(cc(cn3)C(F)(F)F)Cl RF04867 Cc1cccc(c1)c2nc(on2)c3cc(ccc3Oc4ccc(cc4)OC)[N+](=O)[O-] SP00861 CCCc1ccc(cc1)c2nc(no2)c3c(cccc3Cl)Cl SP00876 c1cc(ccc1c2nc(on2)c3ccc(cc3)OC(F)(F)F)OC(F)(F)F SP00600 CC(C(=O)O)Oc1cccc2c1oc3ccccc3c2=O JFD02524 COc1ccc(cc1)CNC(=O)c2cc(c(c(c2)OC)OC)OC JFD02697 COc1ccccc1C2CCN(CC2)C(=O)c3ccccc3C(F)(F)F RH01520 CN(C)C(=O)Nc1cccc(c1Cl)Cl PD00551 c1ccc2c(c1)c(cs2)CCOC(=O)Nc3ccc(cc3)OC(F)(F)F S13509 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)N2CCOCC2 S13549 c1cc(c(nc1)N2CCN(CC2)C(=O)CCC(=O)O)C(F)(F)F SEW05945 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])C(F)(F)F SEW06258 CCCCC1(C(=O)c2ccccc2N(C1=O)C)O JFD03680 c1ccc(c(c1)CSCC/N=C/c2ccccc2O)Cl SEW06551 c1ccc(c(c1)CSCC/N=C/c2cc(ccc2O)Br)Cl SEW06552 COc1cc(c(cc1OC)NC(=O)/C=C\C(=O)O)C(=O)OC GK03181 CCCCCCC#Cc1cc(cnc1)c2nnc(n2C)SCC(=O)Nc3ccccc3 KM09563 CC1(COC(=N1)c2c(ccs2)C(=O)N(C3CCCCC3)C(=O)NC4CCCCC4)C SEW03528 CC1CC2C/C(=N\O)/CC1N(C2)C.Cl RH01457 CC(C)N(C(C)C)C(=O)c1ccccc1c2ccccc2C(=O)N(C(C)C)C(C)C JFD02704 Cc1ccc(cc1)S(=O)(=O)Nc2nnc(s2)SCC(=O)Nc3ccc4c(c3)OCO4 RH01526 Cc1cc(c(o1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl SEW05352 CN(C)C(=S)Cc1ccc(cc1)Cl S11336 c1cc(ccc1C(=O)NNC(=O)c2ccc(cc2Cl)Cl)OC(F)(F)F SPB03442 COc1ccc(cc1)/C=C\2/C(=O)NC(=S)S2 S13814 CC(C)(C)OC(=O)N1CCC(CC1)O AW00442 c1cc(ccc1C2=N/C(=C/c3ccc(c(c3)Cl)Cl)/C(=O)O2)Cl PHG00634 CC(C)(C)c1ccc(cc1)/N=C/c2ccccc2N3CCN(CC3)C SEW06320 c1cc(cc(c1)C(F)(F)F)C(=O)NNc2c(cccn2)C(F)(F)F RF04878 CC(=O)CCC(=O)c1cccs1 SEW06323 Cc1csc2c1ncnc2NC3CCN(CC3)Cc4ccccc4 GK03209 c1ccc2c(c1)c(=O)cc(o2)c3cccs3 RG00015 c1cc(ccc1CS(=O)(=O)Cc2nc(on2)c3ccno3)F SP00914 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)/C=C/c3ccc(c(c3Cl)OC)OC SP00884 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])CO RH01496 CCOC(=O)N1CCN(CC1)CN2CCCCC2=O SEW04877 CCOC(=O)c1c(c2c([nH]1)cc(cc2Cl)Cl)CCC(=O)O SEW06555 CC(C)n1c(cc(n1)C(C)(C)C)C(C)(C)C SEW06556 Cc1cc(cc(c1)NC(=S)NCCCCN2CCN(CC2)c3cccc(c3)Cl)C SEW06559 CCCCCCC#Cc1cc(cnc1)C(=O)NNC(=S)NC KM09539 CC(=O)N1CC(=O)N/C(=C/c2cccs2)/C1=O PD00646 CCOC(=O)c1cc2c(c(c1)CSc3ccc(cn3)C(F)(F)F)OCOC2 SEW03867 COc1cc(c(c(c1)Cl)NC(=O)c2cc(cc(c2)Cl)Cl)Cl SEW03925 Cc1ccc(c(c1)Br)NC(=O)CCS(=O)(=O)c2ccccc2 RDR03801 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4cccs4 KM10253 c1ccc2c(c1)cccc2CSCC(=O)NNC(=O)c3ccccc3Cl RH01532 c1ccc(c(c1)CSCCNC(=O)c2ccc(cc2)Cl)Cl SEW06543 CSc1cccc(c1)NC(=O)CC2(CCCC2)CC(=O)O PD00653 c1cc2c(cc1N3C(=O)CC4(CCCC4)CC3=O)OCO2 PD00656 c1ccc2c(c1)ccn2C(=O)c3ccccc3I RJC03789 Cc1c(cccc1)/C=C/C=C/C=C/c2c(cccc2)C RJC03802 Cc1ccc(c(c1)C(=O)OC)OCc2ccc(cc2)[N+](=O)[O-] MWP01112 Cn1c(nnc1SCc2c(cccc2Cl)F)c3ccc4c(c3)cccn4 KM10637 c1cc(sc1)c2cc(n(n2)c3ccc(cc3)F)NS(=O)(=O)c4cc(ccc4OCC(F)(F)F)OCC(F)(F)F SP01000 c1cc(sc1)c2cc(n(n2)c3ccc(cc3)I)N SP00965 c1ccc2c(c1)c(c[nH]2)CC(=O)O RH01882 CCOC(=O)c1cc(c(nc1Sc2ccccc2NC(=O)Nc3ccc(cc3)SC(F)(F)F)C)C#N AW00778 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)[N+](=O)[O-] S11495 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)Cl)/C(=O)N2CCc4csc5c4cccc5 S11515 CC(=O)SC1CC(=O)N(C1=O)c2ccc(cc2)C(F)(F)F S11810 Cc1ccc(cc1)C(=O)NCCSCc2ccccc2Cl SEW06539 COc1cc(c(cc1OC)NC(=O)c2ccc(cc2)Cl)C(=O)O GK03423 c1cc(cc(c1)C(F)(F)F)CSCCNC(=O)c2cccc(c2)OC(F)(F)F SEW06563 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3c(onc3c4ccccc4Cl)C GK03432 c1ccc(cc1)CN2CCC(=N2)c3ccco3.Cl.Cl MWP01200 c1cc2cc(ccc2nc1)C(=O)NNC(=O)c3ccc(cc3)Cl KM10272 CCc1cccc(c1NC(=O)c2ccccc2I)CC JFD02671 COc1cc(cc(c1OC)OC)C(=O)NCc2ccccc2 JFD02689 CCCCNC(=O)NCCSCc1ccco1 KM10247 Cc1cc2nccc(n2n1)c3ccccn3 JFD03788 C1CCC2C(C1)C3(C(=O)N2CCC#N)OCCO3 RH01566 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)n3c(cc(n3)C(C)(C)C)C(C)(C)C)C SEW06546 c1cc(c(cc1S(=O)(=O)CC#N)Cl)Cl KM01396 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccccc3 GK03428 Cn1c(c(cn1)Br)NC(=O)c2ccccc2 GK03430 CCCCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)C#N JFD03376 CCCc1ccc(cc1)c2nc(no2)c3cccc(c3)C SP00863 Cc1c(c(on1)C)c2nc(no2)c3c(cccc3Cl)Cl SP00877 C/C(=C/c1c2ccccc2[nH]c1c3ccc4ccccc4c3)/[N+](=O)[O-] RDR01167 COC(=O)c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4cccc(c4)S(=O)C KM10231 Cc1cc(ccc1NC(=O)NCCSCc2ccccc2Cl)F SEW06529 c1ccc(c(c1)CSCCNC(=O)Nc2cc(cc(c2)Cl)Cl)Cl SEW06530 COc1cccc(c1)c2coc3cc(ccc3c2=O)O JFD02642 COc1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3cccc(c3)SC)N KM10212 c1cc(ccc1CSc2nncn2c3ccc4c(c3)OCCO4)Cl SPB08041 Cc1c(c(sc1C(=O)O)SC)S(=O)(=O)c2ccc(cc2)Cl KM01691 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)n3c(cc(n3)C(C)(C)C)C(C)(C)C)c4ccccc4 SEW06548 COc1cc(cc(c1O)/C=N/CCSCc2ccccc2Cl)Br SEW06550 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3cc(ccc3Oc4ccc(cc4)OC)[N+](=O)[O-] SP00883 CCOC(=O)c1c2c(sc1n3c(ccc3C)C)CCCC2 GK03191 COC(=O)CCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)Br JFD03363 c1ccc\2c(c1)CCC(/C2=N\O)Cn3ccnc3 KM02341 Cc1cccc(c1)c2ncc(c(n2)N)S(=O)(=O)C(C)(C)C KM02737 c1ccc2c(c1)c(cc(n2)c3ccccn3)N4CCCCC4 JFD03601 COC(=O)c1c(ccs1)Oc2ccc(cc2NS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F GK02104 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H](C(O1)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC03797 Cn1c(c(cn1)C(=O)N2CCOCC2)n3cccc3 GK03613 CC(C)(C)S(=O)(=O)c1cnc(nc1N)c2ccc(cc2)Cl KM02739 CC(C)(C)c1cc2c(s1)c(ncn2)N3CCN(CC3)c4c5c(cc(s5)C(C)(C)C)ncn4 GK03615 CC(=O)c1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)Cl SJC00128 COc1ccccc1NC(=O)/C=C/c2ccccc2 RH01889 Cc1ccc(cc1)c2nc(on2)C S09146 CC(=O)CC(=O)Nc1ccc(cc1)Cl GK03631 c1ccc2c(c1)nnn2CN3CCN(CC3)CCO PD00639 c1ccc2c(c1)nnn2CN(CCCCCCO)Cn3c4ccccc4nn3 PD00641 CC(C)n1c2ccc(cc2nc1C(F)(F)F)C(=O)Nc3ccc(cc3)Cl KM10734 c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4ccccc4 GK03600 CC(=O)O[C@H]1[C@@H](O[C@@H]2COC(O[C@H]2C1=O)c3ccccc3)OC RJC03795 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)O CC07501 CCOC(=O)c1c(n[nH]c1N/N=C\c2ccccc2[N+](=O)[O-])C JFD03603 CSc1c(cc(s1)C(=O)N)C#N KM03390 Cc1ccc(cc1)C(=O)NNc2c3c(cc(s3)c4ccc(cc4)C(C)(C)C)ncn2 GK03574 CCOC(=O)CCc1ccc(c(c1)I)OCc2ccccc2 RJC03845 CC(=O)Oc1cc(c(c2c1C(=O)c3ccccc3C2=O)O)OC(=O)C RJC03847 c1ccc(cc1)N2CCN(C2c3ccc(cc3)[N+](=O)[O-])c4ccccc4 RJC04079 c1ccc(cc1)N2CCN(C2c3cccc(c3)[N+](=O)[O-])c4ccccc4 RJC04080 c1cc(c(nc1)N2CCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F SEW06196 c1cc(cc(c1)[N+](=O)[O-])C2=N/C(=C/c3ccc(c(c3)Cl)Cl)/C(=O)O2 PHG00685 c1cc(cnc1)C(=O)CC(=O)C(F)(F)F KM09597 COc1ccc(c(n1)N2CCOCC2)NC(=O)COCC(=O)O PD00773 c1cc(ccc1n2c(c(cn2)C(=O)n3c(c(cn3)C#N)N)C(F)(F)F)[N+](=O)[O-] GK03605 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H]([C@H](O1)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC03798 CC(=O)NNc1c2c(cc(s2)c3ccc(cc3)C(C)(C)C)ncn1 GK03575 CN(C)C(=O)Oc1ccnc(n1)SCc2ccc(cc2)[N+](=O)[O-] JM00427 Cc1cccc(c1)C(=O)Nc2cccc3c2cccc3 JFD02663 COc1ccccc1c2coc3cc(ccc3c2=O)OS(=O)(=O)C JFD02649 Cc1ccc(cc1)S(=O)(=O)/N=C/N(C)C JFD04017 c1ccc(c(c1)C(=O)O/N=C/c2ccc(c(c2)Cl)F)C(F)(F)F SEW02053 Cc1c(c(no1)/N=C/c2ccc(cc2)Cl)c3ccccc3 JFD03796 CCOC(=O)c1c(n[nH]c1N/N=C\c2ccc(cc2)N(C)C)C JFD03604 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H]([C@@H](O1)OC)OC(=O)C)OC(=O)C)OC(=O)C RJC03796 Cc1c(c(on1)C)C(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N SEW05953 Cc1c(c(on1)C)c2nc(no2)c3ccc(cc3)Cl SEW05954 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4ccncc4 KM09646 CC(C)(C)c1ccc(cc1)C(=O)OC2CN/C(=C/C(=O)OC)/C(=O)NC2 PD00246 c1ccc(cc1)C(=O)Cn\2c(=O)c3ccccc3o/c2=N\c4ccc(cc4)F PD00256 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCCSCc2ccco2 KM10332 c1ccc(cc1)C(CN)c2c[nH]c3c2cccc3 SEW04399 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)CS(=O)(=O)c4ccc(cc4)F)[N+](=O)[O-] SP00648 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW05964 COC(=O)C\1CSCC/C1=N\Nc2ccc(cc2Cl)Cl RF03874 COC(=O)c1ccc(cc1)Cn2c3ccccc3nn2 KM10336 c1cc(ccc1C2N(C(=O)CS2)CCN3C(SCC3=O)c4ccc(cc4)C(F)(F)F)C(F)(F)F PD00260 Cc1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc(c(c4)OC)OC KM10335 CC(c1ccc2cc(ccc2c1)OC)C(=O)NCc3ccccc3 S14048 c1ccc(cc1)N/N=C/c2cccnc2 S14682 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCN(C)C PD00768 Cc1c(c(on1)C)C(=O)NNC(=O)c2cccc(c2)Cl SEW05938 c1cc(ccc1c2nc(on2)c3ccc(cc3)OC(F)(F)F)C(F)(F)F SP00765 COc1ccc(cc1OC)c2nc(no2)c3ccc(cc3)C(F)(F)F SP00848 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)NN KM08334 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)NCCSCc3ccco3 KM10347 CN1C(C2CCCc3ccccc3C2=N1)c4ccc(cc4)OCC=C S14827 CC(C)c1ccc(cc1)C2C3CCc4ccccc4C3=NN2CCO S15444 c1cc(c(nc1)N2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F SEW06170 Cc1c(c(on1)C)C(=O)NNC(=O)c2ccc(cc2)OC(F)(F)F SEW05950 Cc1c(c(sc1C#N)C(=O)/N=C/N(C)C)C CD11485 Cc1ccc(cc1Cl)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] DFP00325 Cc1c(c([nH]n1)N)c2ccc(c(c2)OC)OC JFD03697 Cc1ccc(cc1)c2nc(on2)c3ccc(c(c3)OC)OC SP00768 Cc1ccc(cc1)c2nc(on2)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl SP00777 COc1cccc(c1)C(=O)NNc2cc(ccn2)C(F)(F)F RF04904 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCSCc3ccco3 KM10345 CC(C)C(C(=O)NC(c1ccccc1)c2ccccc2)NC(=O)OC(C)(C)C KM09634 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)CN4CCN(CC4)Cc5ccccc5 PD00770 c1cc(n(c1)c2ccc(cc2)C(F)(F)F)/C=N/Nc3c(cc(cc3Cl)C(F)(F)F)Cl SEW06163 c1ccc2c(c1)c(cs2)CNC(=O)c3ccc(cc3)Cl PD00426 CC1CC(CC(C1)(C)C)NC(=S)Nc2ccc(cc2F)I PD00437 CC(=O)/C(=C\N(C)C)/c1c(cccn1)[N+](=O)[O-] HC00038 c1cc(ccc1NC(=O)c2c(cc(cn2)C(F)(F)F)Cl)Cl HC00022 c1cc(c(c(c1)F)c2nn(c(=O)o2)c3cc(ccn3)C(F)(F)F)F RF04900 Cc1cccc(c1)c2nc(on2)c3ccc(cc3)OC(F)(F)F SP00772 Cc1ccc(cc1)c2nc(on2)c3ccc(cc3Cl)F SP00778 CC(C)C(C(=O)NCCc1ccc(c(c1)OC)OC)NC(=O)OCc2ccccc2 KM09529 c1ccc2c(c1)c(cs2)CC(=O)Nc3ccc(cc3)F S12322 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)C3CCN(CC3)Cc4ccccc4 PD00555 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc(cc3)OC(F)(F)F)Cl SEW05358 c1cc(c(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)[N+](=O)[O-])C(F)(F)F SEW05960 CC(=O)c1ccc(cc1)OCC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05962 c1ccc(c(c1)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl)Cl SEW05353 Cc1ccc(cc1)S(=O)(=O)C KM00234 c1ccc2c(c1)c(=S)c3ccccc3o2 KM10425 COc1cc(c(cc1OC)N2C(=O)C=CC2=O)C(=O)OC GK03183 COc1ccc(c(c1)c2nc(no2)CS(=O)(=O)c3ccsc3)Br SP00787 CCOC(=O)/C(=N/Nc1ccccc1)/C#N RJC03903 c1cc(cnc1)OCC2=NCCN2S(=O)(=O)c3ccc(cc3)Cl AW00875 c1cc(oc1)CSCCNS(=O)(=O)c2cc(ccc2Cl)C(F)(F)F KM10351 c1cc2cc(ccc2nc1)C(=O)NNC(=O)c3cc(cnc3)Br KM10366 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3ccc4c(c3)cccn4 KM10356 Cc1ccc(cc1)NC(=O)N(C)C PD00545 Cc1ccc(cc1Cl)NC(=O)N(C)C PD00550 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=N)N3CC(OC(C3)C)C CD07828 c1cc(cc(c1)[N+](=O)[O-])C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05952 Cc1ccc(cc1)S(=O)(=O)NNC(=O)CSc2c3c4c(sc3ncn2)CCCC4 GK03284 c1ccc(cc1)c2c(n3c4ccccc4sc3n2)Sc5ccc(cc5)[N+](=O)[O-] JFD03871 Cc1c(c(on1)C)C(=O)NNC(=O)c2ccc(cc2)[N+](=O)[O-] SEW05941 CS(=O)(=O)c1ccc(cc1)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM09363 Cc1ccc(cc1N2C(=O)CC(C2=O)Sc3ccccc3C(=O)O)F PD00544 Cc1cc(c2c(=O)cc(oc2c1)c3ccccc3Cl)C RG00029 CC(=O)c1ccccc1OC(=O)c2ccccc2Cl RG00031 Cc1ccc(cc1C)OCC(CNCc2ccccc2)O AW00824 Cc1ccc(cc1)N/N=C\2/C(=NN(C2=O)c3ccccc3)C RJC03910 c1cc(c(c(c1)Cl)Cl)n2ccnc2SCc3ccc(cc3)Br RDR01361 c1cc(oc1)CSCCNC(=O)C2CC2 KM10377 c1ccc2c(c1)C(=O)N(C2=O)CN(CCCn3ccnc3)CN4C(=O)c5ccccc5C4=O PD00556 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NN)C(F)(F)F JP00944 c1cc(ncc1C(F)(F)F)n2ccnc2 KM08003 Cc1cc(cc(c1)/C(=N/OC(=O)C(C)(C)C)/N)/C(=N/OC(=O)C(C)(C)C)/N SEW04022 c1cc(ccc1/C=C/C(=O)O/N=C(/c2ccc(cc2)Cl)\N)OC(F)(F)F SEW06312 c1cc2c(cc1NC(=O)CC3(CCCC3)CC(=O)O)OCO2 PD00652 CSc1cccc(c1)N2C(=O)CC3(CCCC3)CC2=O PD00654 c1cc(oc1)CS(=O)(=O)Cc2nc(on2)c3ccno3 SP00916 c1cc(sc1)c2nc(on2)c3ccno3 SP00921 COC(=O)c1ccc(c(c1)[N+](=O)[O-])NC2CCN(CC2)Cc3ccccc3 KM10495 COc1ccc(cc1)C(=O)NNC(=O)CSCc2cccc3c2cccc3 RH01522 CC(C)Sc1c(cccc1Cl)NC(=O)C KM10121 COc1cc(cc(c1)OC)NC(=O)NCCSCc2ccco2 KM10265 c1cc(n(c1)c2ccc(cc2)F)C(=O)NN SEW04689 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)SCc3cccc(c3)C(F)(F)F SPB02628 Cc1c(c(on1)C)S(=O)(=O)N2CC(OC(C2)C)C SEW05944 Cn1cc(cc1C(=O)OC)C=C(C#N)C#N SEW06318 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])/C=C/C(=O)Nc4ccccc4 RH01571 COc1ccc(cc1)Oc2ccc(cc2c3nc(no3)c4ccc(cc4)C(F)(F)F)[N+](=O)[O-] SP00463 C=CCn1c(nnc1SCc2c(cccc2Cl)F)c3ccc4c(c3)cccn4 KM10638 Cn1c(nnc1SCc2ccc(cc2)C(=O)OC)c3ccc4c(c3)cccn4 KM10639 CC(=O)Nc1ccc(cc1)S(=O)(=O)NC2Cc3ccccc3C2 KM10502 COc1ccc(cc1)C(=O)CSc2nnc(n2c3ccccc3)CSCc4cccc5c4cccc5 RH01744 c1ccc2c(c1)cccc2CN3CCNCC3 RH01495 CC(=O)Nc1ccc(cc1Cl)OC(F)(F)F SEW03526 Cc1ccc(cc1)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl SEW05354 COc1cc(c(cc1OC)NC(=O)c2ccc(cc2)OC(F)(F)F)C(=O)O GK03424 c1ccc(cc1)NC(=O)NC(CC(=O)O)c2ccsc2 MWP00999 Cc1ccc(cc1)C(=O)NCCSCc2cccc(c2)C(F)(F)F SEW06565 COc1ccc(cc1)C(=O)NCCSCc2cccc(c2)C(F)(F)F SEW06566 c1ccc(cc1)CN2CCC(CC2)NC(=O)CC3(CCCC3)CC(=O)O PD00657 c1cc(cc(c1)Cl)N2CCN(CC2)C(=O)/C=C/c3ccc(cc3)OC(F)(F)F SEW06328 CC(C)(C)SCC(=O)N1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl SEW06263 Cc1ccc(cc1NC(=O)NCc2ccc(cc2)OC)SC KM10229 c1cc(sc1)S(=O)(=O)N2CCN(CC2)c3ncccn3 KM10194 c1ccc(cc1)N/N=C\2/CCCC(=C2)O RH01130 c1ccc2c(c1)cccc2CSc3cccc(c3Cl)Cl RH01498 c1cc(ccc1/C=C/C(=O)NNC(=O)c2ccc(cc2)Cl)OC(F)(F)F SEW06315 Cc1ccc(c(c1)C(=O)NNC(=S)Nc2ccc(cc2)Cl)O MWP01117 CCNC(=O)NNc1c(cncc1Cl)Cl RF01336 Cc1ccc(cc1F)NC(=O)CCC(=O)O RDR01190 Cc1ccc(cc1C)n2c(cc(n2)c3ccc(cc3)OC(F)(F)F)NC(=O)C4CCC4 SP00980 c1cc(ccc1c2cc(n(n2)c3ccc(cc3)F)N)Cl SP00835 Cc1cc(ccc1NC(=O)/C=C/C(=O)O)I S01527 c1cc(ccc1NC(=O)c2ccc3c(c2)nns3)Cl KM10331 CC(C)(C)c1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)OC KM10270 c1ccc(cc1)CC(=O)NC2CCNCC2 RH00745 Cc1nc2ccc(cc2o1)NC(=O)NC(=O)c3ccccc3Cl MWP00035 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cc(cc(c3)Cl)Cl GK03427 Cc1cc(n(n1)C)NC(=O)C KM00491 Cn1c(c(c(n1)c2ccc(cc2)Cl)C#N)SC KM01186 CN(C)/C=C/C(=O)c1cccc(c1)[N+](=O)[O-] KM01905 c1cnc2nc(cn2c1)c3ccc(cc3)[N+](=O)[O-] JFD03857 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(cc2)[N+](=O)[O-] RF03087 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])N3CCCCC3 RH01746 Cc1c(c(c(c(c1C)C)S(=O)(=O)N2CCN(CC2)c3ccccc3OC)C)C SEW06053 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN(CC3)c4ccccc4OC SEW06054 CCN(CC)c1ccc(c(n1)N(CC)CC)NC(=O)c2ccc(cc2)Cl SEW06057 CNC(=S)N1CCN(CC1)c2ccccc2OC SEW06132 CC(C)(C)NC(=S)N1CCN(CC1)c2ccccc2OC SEW06133 COc1ccccc1N2CCN(CC2)C(=S)NCC=C SEW06134 CC(C)(C)c1ccc(cc1)CSc2nncn2c3ccc(cc3)OCc4ccccc4 SPB08045 c1ccc(cc1)COc2ccc(cc2)n3cnnc3SCc4c(cccc4Cl)F SPB08046 COc1ccc(cc1)C(=O)NCCSCc2ccccc2Cl SEW06542 c1ccc(cc1)CNC(=O)CSCSCC(=O)NCc2ccccc2 S12082 CCOC(=O)c1csc(n1)Cc2c3cc(ccc3sc2Cl)Cl MWP00306 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)F GK03431 CN1c2ccccc2C(=O)/C(=C/Nc3nc(nc(n3)SC)N(C)C)/S1(=O)=O KM01416 c1ccnc(c1)SCc2cccc(c2)C#N KM01444 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3c(cccc3F)F GK03433 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cccs3 GK03434 CC1C(NC(CC1=O)c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3)[N+](=O)[O-] JFD03368 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)c3ccc(cc3)I)NC(=O)C4CCC4 SP01013 Cc1cc(no1)c2c(c(nn2c3ccc(c(c3)Cl)F)C)C(=O)NC SPB05221 CCc1cccc(c1NC(=O)c2cc(c(c(c2)OC)OC)OC)CC JFD02696 c1ccc(cc1)N2CCN(CC2)CC(=O)N3CCN(CC3)c4ccccc4.Cl KM10246 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCCSCc3ccco3 KM10243 Cc1c(c(no1)c2ccccc2Cl)C(=O)NNC(=O)c3cc4c(s3)-c5ccccc5CC4 PD00647 c1cnc(nc1C(F)(F)F)N2CCC(CC2)NC(=O)Nc3c(cc(cc3Cl)Cl)Cl AW01038 Cn1c2c(c(c3c(n2)-c4ccccc4CC3)c5ccc(c(c5Cl)OC)OC)c(=O)n(c1=O)C PD00650 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)C(C)(C)C GK03437 c1ccc(cc1)N2CCN(C2c3ccc(cc3)Br)c4ccccc4 RJC04081 CC(C)CN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)OC JFD03369 c1cc(sc1)c2cc(n(n2)c3ccc(cc3)F)NS(=O)(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SP00999 c1cc(sc1)c2cc(n(n2)c3ccc(cc3)F)NS(=O)(=O)c4ccc(s4)c5cc(on5)C(F)(F)F SP00998 CCOc1ccccc1NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW06136 c1ccc2c(c1)[nH]c(n2)/C(=C/c3cc(ccc3O)Br)/C#N PHG00729 CCOC(=O)CSc1ccc(c2c1cccc2C(=O)O)C(=O)O PHG00530 CCCCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)[N+](=O)[O-] JFD03370 CC(C)c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00678 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCN RH01887 CCCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)C(F)(F)F JFD03375 CCOC(=O)c1ccc2c(c1)CC/C(=C\c3cccc(c3)Oc4ccccc4)/C2=O SEW03712 CCOC(=O)c1ccc2c(c1)CC/C(=C\c3ccc(cc3Cl)Cl)/C2=O SEW03713 c1cc(c(cc1F)F)N/N=C(\C#N)/S(=O)(=O)c2ccsc2 SEW03716 Cc1cc(cc(c1)N2CC(CC2=O)C(=O)O)C SEW06298 c1cc(ccc1/C=N/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl GK03595 CN1CCN(CC1)CC(=O)N2CCN(CC2)c3ccccc3 KM10743 COc1ccc(cc1)CNC(=O)Nc2ccccc2OC KM10510 c1cc(sc1)/C=N/OCCS(=O)(=O)c2ccc(cc2)Cl KM00956 c1ccnc(c1)S(=O)(=O)Cc2nc(on2)CSc3ccc(cc3)Cl KM01331 CCn1c(=O)c2ccccc2nc1S KM01332 CN1C(=O)Cc2ccccc2C1=O RJC04083 CC(C)(C)c1ccc(cc1)OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06171 Cc1ccc(n1c2cc(c(cc2C(=O)NNC(=O)c3ccco3)OC)OC)C GK03217 c1ccc2c(c1)ccn2CC(CN3CCN(CC3)Cc4c(cccc4Cl)F)O AW01028 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])c2csc(n2)N SEW03265 CCOc1c(cnc2c1sc(c2c3ccccc3)C(F)(F)F)C(=O)OCC SEW03277 Cc1nc(no1)c2cccs2 SEW03437 c1cc(c(cc1OC(F)(F)F)Cl)NS(=O)(=O)C(F)(F)F SEW03441 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)Nc2ccc(cc2)OCc3ccccc3 TB00029 c1cc(ccc1S(=O)(=O)CC#N)Br KM00667 CCCCCCCCCCCCCO JFD04053 COc1ccc(cc1)NC(=O)c2ccc(c(c2)OC)OC JFD02677 Cn1c(nnc1SCc2ccc(cc2)Cl)c3ccc4c(c3)cccn4 KM10472 c1cc(cc(c1)C(F)(F)F)C(=O)NCCSCc2ccc(cc2)Cl SEW06359 COc1cc(cc(c1)OC)NC(=O)NC2Cc3ccccc3C2 KM10468 c1cc(sc1)C(=O)NCCSCc2ccc(cc2)Cl SEW06364 Cc1cc(c(c(c1)Cl)OC(=O)c2ccccc2[N+](=O)[O-])Cl RDR01773 Cc1cc(c(c(c1)Cl)OC(=O)c2ccc(cc2)[N+](=O)[O-])Cl RDR01774 c1ccc(cc1)NC(=O)OC2CCCC2 RJC03811 CC(C)Cc1ccc(cc1)C(C)c2nnc(o2)c3ccc(cc3)Cl SEW06272 c1cc2cccnc2c(c1)OC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW06277 Cn1c2c(cn1)c(ncn2)n3c(c(cn3)C(=O)NNC(=O)c4ccco4)C(F)(F)F GK03619 COc1cccc(c1O)/C=N/CCNc2cc(ccc2OC)Cl PD00533 C/C(=N\O)/CS(=O)(=O)c1ccc(cc1)Cl KM01817 CC(C)(C)S(=O)(=O)C/C(=N/OC(=O)Nc1ccccc1)/N KM02223 c1ccnc(c1)C2NN=C(S2)S SPB06965 c1cc(oc1)CSCCNC(=O)CSc2nnnn2c3ccc(cc3)O KM10378 c1cc(c(nc1)N2CCCN(CC2)C(=O)/C=C/C(=O)O)C(F)(F)F AW01029 c1cc(c(cc1NN=C(C#N)C#N)C(F)(F)F)F SEW06190 c1cc(ccc1[N+](=O)[O-])OC(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW01030 c1cc2c(cc1NN=C(C#N)C#N)OCCO2 SEW06191 c1c(cc(cc1F)F)NN=C(C#N)C#N SEW06192 COc1cccc(c1NC(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F)Cl SEW06187 CC(C)Cc1ccc(cc1)C(C)c2nc(no2)c3ccc(cc3)C(F)(F)F SEW06275 c1cc2cccnc2c(c1)OS(=O)(=O)c3ccc(cc3C(F)(F)F)C(F)(F)F SEW06279 c1ccc(cc1)CNC(=O)NC(=O)CC(=O)O RJC03821 CCOC(=O)c1ccc(cc1)n2c(ccc2C)C RH01808 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)C=C(C#N)C#N SEW06335 Cc1ccc(cc1)S(=O)(=O)Oc2cccc3c2nccc3 SEW06303 c1cc(ccc1/C=C/C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)OC(F)(F)F SEW06305 CC1C(OCCN1C(=O)CCC(=O)N2CCOC(C2C)c3ccccc3)c4ccccc4 RB00386 c1cc(n(c1)c2ccc(cc2)C(F)(F)F)/C=C/3\CSc4ccc(cc4C3=O)Cl SEW06161 COCCCNC(=S)N/N=C/c1cccn1c2ccc(cc2)C(F)(F)F SEW06162 Cc1cccc(c1OC(=O)c2ccc(cc2Cl)Cl)C RDR01796 COc1cccc(c1)NC(=O)NC2Cc3ccccc3C2 KM10469 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3cccc(c3)C(F)(F)F)C SPB08260 c1cc(c(c(c1)Cl)CN2CCN(CC2)C(=O)c3cccs3)F AW01025 CCc1cc2c(cc1c3csc(n3)c4c(nns4)C)C(CCC2(C)C)(C)C SEW06177 Cc1ccc(c2c1CCC2)Oc3ccc(cc3NC(=O)c4c(onc4c5c(cccc5Cl)F)C)C(F)(F)F RH01811 c1cc(ccc1c2csnn2)N3CC(CC3=O)C(=O)O SEW06295 c1cc(ccc1NC(=O)C(C(C(=O)O)O)O)Cl JFD03881 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4cccc(c4)OC)[nH]cn3 KM10613 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)Cl)[nH]cn3 KM10634 c1ccc(cc1)C(=O)/C(=N/Nc2ccc(cc2)Cl)/S(=O)(=O)c3ccccc3 JFD03861 CC(C(=O)N1CCN(CC1)c2ccc(cn2)C(F)(F)F)Oc3ccc(cc3)Oc4ccc(cc4)C(F)(F)F SEW06314 COC(=O)/C=C/1\C(=O)NCCCN1 PD00252 c1cc(c(cc1Cl)N2C(=O)C=CC2=O)Cl S01374 COc1ccc(c(c1)S(=O)(=O)Nc2cccc(c2)C#C)OC CD07857 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4ccc(cc4)OS(=O)(=O)N(C)C SP00888 c1c(c(=O)[nH]c(=O)n1C2CCCO2)F JFD03885 Cc1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4cccc(c4)F JFD03870 CCCCNC(=O)NC1Cc2ccccc2C1 KM10451 c1ccc(cc1)NC(=O)NC2Cc3ccccc3C2 KM10455 CC1=C(CC2C(C1)C(=O)N(C2=O)c3ccc(cc3F)F)C PD00522 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)c3cc(cc(c3)Cl)Cl)C(F)(F)F GK03081 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CCCC(=O)O)C(F)(F)F SEW06178 CCCc1ccc(cc1)C(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl RH02035 CC(=O)Nc1ccc(cc1)OCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06182 Cn1c(c(cn1)Br)NC(=O)Nc2ccc(cc2)OC(F)(F)F GK03419 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3ccc(c(c3)OC)OC SP00886 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3cc(ccc3Br)OC SP00887 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3ccc(cc3)OC(F)(F)F SP00893 c1cc(ccc1/C=C/c2nnc(o2)c3ccc(cc3)Cl)OC(F)(F)F SEW06326 c1ccc(cc1)COc2ccc(cc2)CCC3OCCO3 RJC03842 c1ccc(cc1)COc2ccc(cc2)COCc3ccc(cc3)OCc4ccccc4 RJC03846 CC(=O)CCC(=O)c1ccco1 SEW06316 c1ccc(cc1)NC(=O)c2cc3c(s2)ccs3 SEW02087 CC(=O)N1CCC(CC1)C(=O)O/N=C(/c2ccc(cc2)Cl)\N SEW06317 c1cc2c(cc1Cl)C3=C(CS2(=O)=O)/C(=N/Nc4c(cc(cc4Cl)Cl)Cl)/CCS3 SEW02198 Cc1csc2c1c(ncn2)NC3CCN(CC3)Cc4ccccc4 GK03210 CCn1c(c(c(n1)C)Br)c2nc(no2)c3ccc(cc3)OS(=O)(=O)N(C)C SP00890 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)C3CCC3 SP00896 c1ccc2c(c1)CC(C2)NS(=O)(=O)c3ccc(s3)Br KM10505 Cc1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc(cc4)OC KM10328 c1cc(c(c(c1)Cl)c2csc(n2)N)F RF02502 Cc1ccc(cc1)NC(=O)c2ccc(cn2)C(=O)OC RF03167 c1ccc(cc1)c2ccc(cc2)C(c3cc4cc(ccc4o3)[N+](=O)[O-])O RH01805 CCn1c(c(c(n1)C)Br)c2nc(no2)c3ccc(cc3)C SP00775 COc1ccc(cc1)/C=N/NC(=O)c2cc3c(s2)-c4ccccc4CC3 PD00640 Cc1ccc(cc1)n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)OC)[nH]cn3 KM10635 c1cc(cc(c1)C(F)(F)F)C(=O)O/N=C/c2ccc(c(c2)Cl)F SEW02054 Cc1c(c(on1)C)c2nc(no2)c3ccc(cc3)OS(=O)(=O)N(C)C SP00895 Cc1cccc(c1)c2nc(on2)c3ccno3 SP00899 COc1ccc(cc1OC)c2nc(no2)c3cccs3 SP00904 COc1ccc(c(c1)c2nc(no2)c3cccs3)Br SP00905 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCCn3ccnc3 PD00548 c1ccc(cc1)CN2CCC(CC2)NC(=O)CSCC(=O)O PD00553 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)Cc3ccc(cc3)F AW01059 Cn1c(c(cn1)Br)NC(=O)c2cc(cc(c2)Cl)Cl GK03230 CC(=O)c1ccccc1N2C(=O)CC(C2=O)Sc3ccccc3N S12282 c1ccc2c(c1)c(cs2)CC(=O)Nc3ccc(cc3)I S12290 CCNC(=S)Nc1ccc(cc1Cl)Cl GK03237 CNC(=S)Nc1ccc(c(c1)Cl)Cl GK03242 Cc1cc(c(c(c1)C)NC(=S)NCc2ccco2)C GK03250 c1cc(sc1)c2cc(n(n2)c3ccc(cc3)I)NC(=O)C4CCC4 SP01005 c1cc(cc(c1)S(=O)(=O)N2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F)C(F)(F)F SEW02212 c1cc(ccc1C2c3ccsc3CCN2S(=O)(=O)c4ccc(cc4)Cl)OC(F)(F)F SEW02213 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccn2 JFD02695 CCn1c(c(c(n1)C)Br)c2nc(no2)c3cccs3 SP00910 CNC(=O)N(Cc1cccnc1)Cc2cccc(c2Cl)Cl RF03324 COc1cccc(c1c2nn(c(=O)o2)c3ccc(cn3)C(F)(F)F)OC RF04819 COc1cccc(c1)c2nn(c(=O)o2)c3c(cc(cn3)C(F)(F)F)Cl RF04850 COc1ccccc1c2nn(c(=O)o2)c3ccc(cn3)C(F)(F)F RF04866 COc1ccccc1C(=O)NNc2cc(ccn2)C(F)(F)F RF04903 CCn1c(c(c(n1)C)Br)c2nc(no2)c3ccc(cc3)C(F)(F)F SP00844 CCCc1ccc(cc1)c2nc(no2)c3ccc(cc3)OS(=O)(=O)N(C)C SP00885 CN1CCN(CC1)c2ccccc2/C=N/c3ccc(cc3)OC SEW06319 c1cc(sc1)c2ccc(s2)C#N SEW02204 c1cc(ccc1C2c3ccsc3CCN2C(=O)c4ccc(cc4)Cl)OC(F)(F)F SEW02205 c1cc(ccc1C2c3ccsc3CCN2C(=O)c4ccc(cc4)OC(F)(F)F)OC(F)(F)F SEW02206 c1cc(c(cc1[N+](=O)[O-])Cl)C(=O)NN GK03218 COc1ccc(cc1OC)C(=O)OCC(=O)c2ccc(cc2)Br JFD02705 CC(C)(C)c1ccc(c(c1)C(C)(C)C)Oc2ccc(cc2C(C)(C)C)C(C)(C)C JFD02709 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)c2ccccc2 AW01035 Cc1ccc(cc1)S(=O)(=O)NC(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F AW01039 c1cc(ccc1S(=O)(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl)Cl RH01890 c1cc(c(cc1S(=O)(=O)NC2CCCCC2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01061 Cn1c(c(cn1)Br)N2C(=O)CCC2=O GK03222 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)NCc3cccs3)C SPB08261 c1ccc(cc1)c2csc3c2c(ncn3)N4CCOCC4 AW01068 Cc1cc(c(c(c1)C)NC(=S)NC(CO)(CO)CO)C S13257 c1ccc2c(c1)c(cs2)CNC(=S)Nc3ccc(cc3)OC(F)(F)F S13584 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)c3ccc(cc3)S(=O)(=O)N)N SP00991 c1cnc(nc1C(F)(F)F)N2CCC(CC2)N3C(=O)CC4(C3=O)CCCC4 AW01230 c1ccc(cc1)C(=O)Oc2cc(=O)n3c4c2cccc4CCC3 RJC04082 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)Cc3c(cccc3Cl)F AW01041 CCOC(=O)NNc1cc(ccn1)C(F)(F)F RF04967 CCCCCCCCCCCC(=O)Nc1ccc(cc1)Cl RG00112 COc1ccc(cc1)n2c(cc(c2c3ccccc3)c4cccs4)c5ccc(cc5)Cl RG00099 COc1ccc(cc1)c2cc(n(n2)c3ccc(c(c3)Cl)Cl)NC(=O)C4CCC4 SP00987 c1cc(ccc1NC(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl AW00702 c1cc(ccc1NC(=O)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl AW00735 Cc1ccc(cc1C)n2c(cc(n2)c3ccc(cc3)OC(F)(F)F)NC(=O)Nc4ccccc4C#N SP01030 COc1ccc(cc1)c2cc(n(n2)c3ccc(c(c3)Cl)Cl)NS(=O)(=O)c4cccc(c4)F SP00988 CC(=O)c1cc2c(s1)-c3cc(ccc3SC2)Cl SEW02679 c1cc(ccc1c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)N)OC(F)(F)F SP01049 c1ccc(cc1)CN2CCC(CC2)NC(=O)COCC(=O)O PD00561 c1cc(ccc1COc2ccc(cc2)C#N)Cl RF01849 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)I)C SP01238 C1CCC(=NC2=C(CCCC2)C(=O)N)CC1 JFD03877 c1ccc(cc1)N2CCN(CC2)Cc3c[nH]c4c3cccc4 RJC03948 c1ccc(cc1)C(=C2C=CC3C2C4CCC3C4=C(c5ccccc5)c6ccccc6)c7ccccc7 JFD04031 CC1(C2CC1C(=O)/C(=C\c3ccccc3)/C2)C JFD04032 Cn1cc(cc1C(=O)OC)/C=C/C(=O)N(C2CCCCC2)C(=O)NC3CCCCC3 SEW06693 c1ccc(c(c1)NC(=O)CSc2ccccn2)Sc3nccc(n3)C(F)(F)F AW00932 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc4ccccc4c3 GK03420 c1ccc(cc1)Oc2ccc(cc2)NC(=O)c3cnccn3 PD00537 c1ccc(cc1)n2c(nnc2SCC(=O)c3ccc(cc3)C(F)(F)F)CSCc4cccc5c4cccc5 RH01743 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3cc(nn3c4ccc(cc4)F)c5cccs5 SP01004 c1cc(sc1)c2cc(n(n2)c3ccc(cc3)F)NC(=O)C4CCC4 SP00981 COc1ccc(cc1)c2cc(n(n2)c3ccc(c(c3)Cl)Cl)NC(=O)Nc4ccccc4C#N SP01003 c1cc2c(c(c1)C(=O)O)NC(=O)C2=O KM10113 Cn1c(nnc1S)Cn2cc(ccc2=O)C(F)(F)F SPB06511 CC(C)(C)c1ccc(cc1)c2nnc(o2)SCc3ccc(cc3)OC(F)(F)F SPB08253 Cn1c(c(cn1)C(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N)n3cccc3 GK03582 c1ccc(c(c1)/C=N/Nc2nc(cs2)c3ccc4c(c3)OCCO4)Cl SPB08258 Cn1c(c(cn1)C(=O)O/N=C(/c2ccccc2)\N)n3cccc3 GK03584 COc1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccc(cc3)OC(F)(F)F RH01927 c1ccc(cc1)OCCN2CCN(CC2)S(=O)(=O)c3ccccc3 TB00008 c1ccc(c(c1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4N)F KM09746 c1ccc(cc1)C(=O)Nc2ccc(c(c2)Cl)Cl SPB08366 c1cc(c(cc1C(=O)Oc2ccc(cc2Cl)Cl)Cl)Cl RDR01769 Cc1cc(c(c(c1)Cl)OC(=O)c2ccc(c(c2)Cl)Cl)Cl RDR01771 c1cc(cc(c1)S(=O)(=O)Cc2cc3c(o2)c(c(c(c3F)F)F)F)C(F)(F)F SEW03440 CC(C)Cc1ccc(cc1)C(C)c2nc(no2)c3ccc(cc3)Cl SEW06273 Cc1ccc(cc1)c2nc(on2)C(C)c3ccc(cc3)CC(C)C SEW06274 Cn1c(ccn1)NC(=O)Nc2ccc(cc2)OC(F)(F)F GK03280 COc1cc2c(cc1OC)ncnc2NCCCn3ccnc3 GK03281 CC(=O)n1cc(c2c1cccc2)/C=C/3\C(=O)OC(=N3)c4ccccc4 PD00564 Cc1ccc(cc1)N/N=C\2/CCCNC2=O RH01829 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CCOc3ccccc3 TB00009 c1ccc(cc1)OCCN2CCN(CC2)S(=O)(=O)c3ccc(cc3F)F TB00012 c1ccc(cc1)OCCN2CCN(CC2)C(=O)c3cccs3 TB00013 c1cc(sc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc(cc4)Cl KM10271 c1ccc(cc1)NC(=O)NCCSCc2ccccc2Cl SEW06531 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCSCc2ccccc2Cl SEW06532 CC(C)(C)c1cc(n(n1)c2ccc(cc2)C(=O)NN)C(C)(C)C SEW06534 COc1cc(cc(c1OC)OC)C(=O)Nc2ccc3c(c2)OCO3 JFD02694 CC1=C(C(C(=C(N1)C)C#N)c2ccccc2Cl)C#N JFD03361 COC(=O)CSCCS(=O)(=O)c1ccc(cc1)Cl KM01501 CCCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)C(=O)C JFD03364 c1cc(sc1)C(=O)NCCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F RH01914 COc1ccc(cc1)C(=O)Nc2ccc(nc2)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06369 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)CCO KM10548 c1cc(c(c(c1NC(=O)c2cnccn2)F)F)F PD00536 COC(=O)C(Cc1cc(c(c(c1)Br)O)Br)NC(=O)C(F)(F)F SB02026 CC(=O)Nc1cccc(c1)n2c(nnn2)S SB02024 c1cncc(c1C(=O)O)C(=O)O SB02021 COc1cc(ccc1OC(=O)c2cc(c(c(c2)OC)OC)OC)/C=N/c3cccc(c3)C(F)(F)F SJC00170 c1cc(cc(c1)OCc2ccc(cc2)c3ncns3)C(F)(F)F SEW01941 CCOC(=O)c1cnn(c1C(F)(F)F)C(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK03606 CCOC(=O)c1cnn(c1N)C(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK03608 CC(C(=O)N1CCN(CC1)Cc2ccccc2)Nc3ccccn3 RH01830 c1c(cnc(c1Cl)CN2CCSCC2)C(F)(F)F HC00017 Cc1c(c(n[nH]1)C)c2c(cccn2)[N+](=O)[O-] HC00027 COc1ccc(c(c1)Cn2cc(c(=O)c(c2)F)C(=O)OC)OC HC00063 Cc1ccc(cc1)SCc2cccc(c2)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06283 c1cc(cc(c1)Cl)c2nnc(o2)c3cccc(c3)Cl SJC00156 CC(=O)C(=NNc1ccccc1)C(=O)C SPB04418 Cc1ccc(cc1)CSc2nc(c(c(=O)n2C)Oc3cccc(c3)C(F)(F)F)C SPB04452 c1ccnc(c1)S(=O)CC#N KM01123 COc1cc(ccc1OC(=O)c2cc(c(c(c2)OC)OC)OC)/C=N/C(Cc3ccccc3)c4ccccc4 SJC00167 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2cnn(c2n3cccc3)C)/N GK03583 c1ccc(cc1)c2csc3c2c(ncn3)NCCCN4CCN(CC4)Cc5c(cccc5Cl)F AW01229 c1csc2c1/C(=N/O)/CCS2 SEW01960 CCCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)C JFD03366 CCOC(=O)c1c(c(sc1N)C)c2ccccc2 AW00937 Cn1c(ccn1)NC(=O)Nc2cccc(c2)Br GK03277 Cc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2Oc3ccc(c4c3CCC4)C)C(F)(F)F RH01809 CSc1cccc(c1)NC(=O)c2cnccn2 PD00534 Cc1ccc(cc1S(=O)(=O)Nc2cc(ccc2Oc3ccc(c4c3CCC4)C)C(F)(F)F)[N+](=O)[O-] RH01838 Cc1ccc(c2c1CCC2)Oc3ccc(cc3NC(=O)c4ccc(cc4)[N+](=O)[O-])C(F)(F)F RH01836 COc1cc(ccc1OC(=O)c2cc(c(c(c2)OC)OC)OC)/C=N/Cc3ccccc3 SJC00171 CNC(=S)Nc1ccccc1 GK03238 CNC(=S)NCc1ccco1 GK03240 CCNC(=S)Nc1ccc(cc1C)C GK03241 c1ccc(cc1)C2=N/C(=C/c3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)/C(=O)O2 SP01246 c1cc(cc(c1)Cl)c2c(nco2)C(=O)N SEW02026 C/C(=C\1/C(=O)OC(=N1)c2ccccc2)/N(C)C RH01794 CC(CCc1ccc(c(c1)OC)O)N.Cl RH01800 Cc1cccc(c1)n2c(n[nH]c2=S)CC#N HR00167 Cc1cc(c(cc1OC)I)OC RH01788 COc1cc2c(cc1OC)ncnc2SCC(=O)OC GK03211 c1ccc2c(c1)/C(=C/c3cccn3c4ccc(cc4)OC(F)(F)F)/C(=O)N2 SEW06340 Cc1c2ccccc2sc1C#N MWP00784 CSc1ccc(s1)/C=C/2\C(=O)OC(=N2)c3ccccc3 SP01245 c1cc(sc1C(=O)O)Cl KM03331 CCOC(=O)c1c(n[nH]c1N/N=C\c2ccccc2Cl)C JFD03605 CCOC(=O)c1c(n[nH]c1N/N=C\c2ccccc2O)C JFD03606 Cn1c(c(cn1)Br)NC(=O)/C=C/C(=O)O GK03274 CC(=O)c1cc(no1)c2cccc(c2)C(F)(F)F SPB05243 Cc1ccc(cc1)c2csc(n2)CN3CCN(CC3)c4cccc(c4)Cl SEW06668 Cc1ccc(c2c1CCC2)Oc3ccc(cc3NS(=O)(=O)c4ccc(cc4)Cl)C(F)(F)F RH01837 c1ccc(c(c1)S(=O)(=O)CC#N)Cl HC00106 c1cc(ccc1C(F)(F)F)n2c(=O)c(c(cn2)N3CCOCC3)Cl SP01248 Cc1ccc(n1c2cc(c(cc2NC(=O)Nc3ccc(cc3)Cl)OC)OC)C GK03246 Cn1c(c(cn1)Br)NC(=O)c2ccco2 GK03247 Cn1c(c(cn1)Br)NC(=O)CN2CCOCC2 GK03248 Cn1c(c(cn1)Br)NC(=O)CSc2ccc(cc2)Cl GK03249 CC(C)n1c2ccc(cc2nc1C(F)(F)F)C(=O)N3CCC(CC3)O KM10742 CCCCc1ccc(cc1)NC(=O)c2ccc(c(c2)OC)OC JFD02679 CN1c2ccc(cc2C(=O)NC1c3ccc(cc3)C#N)Cl BTB05561 CC(=O)Nc1ccc(cc1Cl)F BTB05770 Cc1nc(cs1)c2nnc(n2CCCOC)SCC(=O)Nc3ccc(cc3)C(C)C SPB02443 COc1ccc(cc1OC)C(=O)Nc2cccc(c2)Cl JFD02680 c1ccc2c(c1)c\3c([nH]2)CCC/C3=N\OC(=O)C4CCCCC4 RH01818 CCOC(=O)c1c(c(sn1)/C(=N/Nc2ccccc2)/C)N JFD04025 CCCCNC(=O)NCCNc1ccc(cn1)C(F)(F)F AW00876 c1ccc(c(c1)C(=O)O)SC2CC(=O)N(C2=O)c3cccc(c3)Br PD00543 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc4c(c3)OCO4 KM10361 COc1ccc(c(n1)N2CCC(CC2)C(=O)N)[N+](=O)[O-] PD00775 CC(C)n1c2ccc(cc2nc1C(F)(F)F)C(=O)NCc3ccncc3 KM10739 CC(C)n1c2ccc(cc2nc1C(F)(F)F)C(=O)N3CCCCC3 KM10741 CC(=O)/N=C\1/NC(=O)/C(=C\c2cccs2)/N1C PD00431 COc1ccccc1N2CCN(CC2)C(=S)Nc3cc(c(cc3OC)Cl)OC SEW06154 c1cc(ccc1C#N)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl SEW05362 CN(C)/C=C(\C#N)/C(=O)Nc1ccncc1 BTB06699 c1ccc(cc1)c2c3ccccc3nc-4c2Cc5c4cccc5 HR00184 c1ccc(cc1)COc2ccc(c(c2)/C=C\N3CCCC3)[N+](=O)[O-] RH01816 COc1ccc(cc1)C(=O)NCCCCN2CCN(CC2)c3cccc(c3)Cl SEW06341 c1ccc(c(c1)N)SCc2nc(on2)c3cccs3 SEW06345 Cn1c(ccn1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F GK03213 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NNC(=O)Nc3ccccc3 SPB08146 c1ccc2c(c1)C3(C4N2CC5(CCCCC5)CN4)OCCO3 RH01870 c1cc(cc(c1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F)CSc4ccc(cc4)Cl SEW06281 c1ccc2c(c1)CC(C2)NC(=O)Nc3ccc(cc3)OC(F)(F)F KM10471 COC(=O)CSc1ccnc2c1ccc(c2)Cl KM10729 Cc1ccc2c3c(cc(cc3sc2c1C)C)C RJC03812 Cc1cc(no1)C(=O)Nc2ccc(cc2)C(F)(F)F SPB03090 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NN SPB03095 c1cc(c(cc1Cl)Cl)OCc2n[nH]nn2 SPB03175 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2nnc(o2)c3cc(ccc3OCC(F)(F)F)OCC(F)(F)F SPB03391 CC(C)(C)c1cc2ccc3cc(cc4c3c2c(c1)cc4)C(C)(C)C JFD04029 c1cc(cnc1)/C=N/N2CC(=O)N(CC2=O)c3cc(cc(c3)Cl)Cl S14384 Cn1c(ccn1)NC(=O)c2cc(cc(c2)Cl)Cl GK03262 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(n3C4CCCCC4)S SPB08144 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2c3c(sc2n4c(ccc4C)C)CCCC3 GK03228 Cc1ccc(n1c2c(c3c(s2)CCCC3)C(=O)NNS(=O)(=O)c4ccc(cc4)C(F)(F)F)C GK03229 c1ccc2c(c1)CC(C2)NC(=O)c3ccc4c(c3)non4 KM10501 Cc1ccc(cc1)S(=O)(=O)NC(=O)NC2Cc3ccccc3C2 KM10470 c1ccc2c(c1)CC(C2)NC(=O)Nc3ccc(cc3)Cl KM10466 c1ccc2c(c1)CC(C2)NC(=O)Nc3cccc(c3)Cl KM10464 Cn1c(nnc1SCC(=O)NCc2ccccc2)c3ccc4c(c3)cccn4 KM10460 c1c(cc(cc1C(F)(F)F)SCc2c(cc(cn2)C(F)(F)F)Cl)C(F)(F)F HC00059 Cc1ccc(o1)c2ccccc2N JFD03365 COC(=O)c1cn(cc(c1=O)F)Cc2ccc(cc2)C(F)(F)F HC00065 c1cc(ccc1N/N=C/c2c(cc(cn2)C(F)(F)F)Cl)OC(F)(F)F HC00076 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3cccc4c3nccc4 SEW06269 c1cc(sc1C(=O)N)[N+](=O)[O-] RF01604 C[C@@]12CCC(C1(C)C)CC2NS(=O)(=O)c3ccc(cc3)F JFD04010 c1cc(ccc1C(=O)NNC(=O)CSc2c3c4c(sc3ncn2)CCCC4)Cl GK03255 c1ccc(c(c1)NC(=S)NN)Cl GK03258 Cc1c(ccc(n1)C(F)(F)F)C(=O)N2CCN(CC2)Cc3c(cccc3Cl)F AW00889 c1cc(ccc1OC(F)(F)F)SCC#N KM04648 Cc1ccc(n1c2cc(c(cc2C(=O)NNC(=O)c3cc(cc(c3)Cl)Cl)OC)OC)C GK03224 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)OC KM10385 c1ccc2c(c1)cccc2NC(=O)NC3Cc4ccccc4C3 KM10497 COc1ccc(cc1OC)C(=O)NC2Cc3ccccc3C2 KM10500 c1ccc(cc1)CN2CCC(CC2)Nc3c4c(cc(s4)c5ccccc5)ncn3 GK03585 Cn1c(nnc1SCc2ccc(cc2)OC(F)(F)F)c3ccc4c(c3)cccn4 KM10475 Cn1c(nnc1SCc2c(cccc2Cl)Cl)c3ccc4c(c3)cccn4 KM10476 c1ccc(c(c1)C(=O)NCCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F RH01895 Cc1ccc(cc1)/C(=N\N(C)C)/C(=O)C(F)(F)F HC00021 Cc1ccc(cc1)C(=O)C(C(F)(F)F)(O)O HC00034 CC(C)[C@@H](C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 SB01001 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5c(c4)OCO5 KM10375 COc1ccc(cc1)c2ccnc(n2)SCC(=O)NCCSCc3ccco3 KM10379 c1cc2c(cc1NC(=O)c3cnccn3)OCO2 PD00495 CCOC(=O)/C(=C\c1ccccc1N2CCN(CC2)C)/C#N SEW06332 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)S RH01691 Cc1cc(cc(c1)n2c(cc(n2)c3cc(oc3C)C(C)(C)C)NS(=O)(=O)c4cccc(c4)F)C SP01066 c1ccc(c(c1)c2cc(c(o2)C(F)(F)F)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)Cl SP00698 Cc1ccc(cc1)c2nc(on2)c3cc(nn3Cc4ccccc4)C(C)(C)C SP00776 Cc1ccc(cc1)c2nc(on2)c3cc(ccc3Br)OC SP00769 c1cc(ccc1c2cc(n(n2)c3cc(ccc3Cl)C(F)(F)F)N)OC(F)(F)F SP01076 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(ccc3Oc4ccsc4C(=O)OC)C(F)(F)F GK03200 CC(C)(C)c1cc2c(s1)c(ncn2)NC3CCN(CC3)Cc4ccccc4 GK03599 COc1cccc(c1)Nc2c3c(cc(s3)c4ccccc4)ncn2 GK03602 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3ccccn3 PD00772 Cn1c(c(cn1)Br)NC(=O)c2ccc(cc2Cl)F GK03438 c1ccc(cc1)CN2CCN(CC2)C(=S)c3ccccc3 PD00546 c1ccc(cc1)CN2CCC(CC2)NC(=O)/C=C\C(=O)O PD00547 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc(cc4)Cl KM10364 c1cc(ccc1c2cc(nc(n2)N)C(F)(F)F)Cl KM10417 Cc1ccc(cc1)SCC(=O)Nc2c(cnn2C)Br GK03260 c1ccc(c(c1)/C=N/Cc2csc3c2cccc3)O S14405 COc1ccc(cc1)C/N=C/c2ccc(cc2)C(F)(F)F S14632 c1ccc2c(c1)NC3(CCCCC3)C4CCCCC4=N2 S14810 c1cc(oc1)c2cc3nc4c(c(n3n2)C(F)(F)F)CCC4 KM10376 c1ccc2c(c1)ccc3c2cc(c(=O)o3)NC(=O)c4ccc(cc4)Cl PHG00635 CCn1c(c(c(n1)C)Br)c2nc(no2)c3cccc(c3)C(F)(F)F SP00653 c1cc(cc(c1)C(F)(F)F)c2nc(on2)c3ccc(cc3Cl)F SP00654 c1cc(cc(c1)S(=O)(=O)Nc2cc(nn2c3ccc(cc3)F)c4cccs4)F SP00990 c1cc(sc1)c2cc(n(n2)c3ccc(cc3)F)N SP00975 CCOC(=O)C(=CNNC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)[N+](=O)[O-])C(=O)OCC GK03607 CC(=O)N[C@@H](Cc1ccc(cc1)Br)C(=O)O SPB08166 c1cc(c(nc1)NCCN)[N+](=O)[O-] RH01896 CCCCc1ccc(c(c1)C)NC(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW01067 c1cc(oc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5c(c4)OCO5 KM10348 c1cc2c(c(c1)S(=O)(=O)NCCSCc3ccco3)non2 KM10346 Cn1c(nnc1SCc2ccccc2)c3ccc4c(c3)cccn4 KM10355 c1ccc(cc1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05947 CCCS(=O)(=O)c1cscc1NC=C(C(=O)OCC)C(=O)OCC KM02281 CC(C)(C)c1ccc(cc1)c2nnc(o2)Sc3cnc(s3)[N+](=O)[O-] SPB08252 COC(=O)CCC1CCC(C1=O)CCC(=O)OC RJC03996 c1cc(sc1)/C=N/Nc2nc(cs2)c3ccc4c(c3)OCCO4 SPB08256 c1cc(ccc1S(=O)(=O)Cc2nc(cs2)c3ccc4c(c3)OCCO4)Cl SPB08257 Cc1c(cc(c(n1)Sc2nccn2c3cc(ccc3Cl)Cl)C(=O)OC)C#N AW01040 c1ccc2c(c1)CC(C2)NC(=O)c3ccc(cc3)Cl KM10478 c1cc(ccc1C(=O)Nc2nc(cs2)c3ccc(cc3Cl)Cl)C(F)(F)F RH01899 c1cc(c(cc1F)F)c2nc(cs2)/C(=N/O)/N SPB02706 Cc1ccc(cc1)S(=O)(=O)NCCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F RH01900 c1cc(ccc1NC2=NC(CS2)(CO)CO)I PD00558 c1cc(c(cc1Cl)NC(=S)N/N=C/c2cc(c(c(c2)Br)O)Br)Cl RDR01122 COc1ccc(cc1Br)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)[N+](=O)[O-] PHG00625 COc1ccc(cc1)c2cc(n(n2)c3ccc(c(c3)Cl)Cl)N SP00832 c1cc2c(cc1C(=O)CC(=O)C(F)(F)F)OCO2 KM10326 c1cc(c(cc1OC(F)(F)F)Br)NC(=O)c2cnccn2 PD00496 CC(CCC(=O)NCCS(=O)(=O)[O-])C1CCC2C1([C@H](CC3C2[C@@H](CC4C3(CC[C@H](C4)O)C)O)O)C.[Na+] JFD03704 Cc1ccc(cc1C)n2c(cc(n2)c3ccc(cc3)OC(F)(F)F)N SP00973 Cc1ccc(cc1)c2nc(on2)c3cc(oc3C(F)(F)F)c4ccccc4Cl SP00701 CCCc1ccc(cc1)c2nc(no2)CS(=O)(=O)C(C)(C)C SP00866 COc1ccccc1NC(=O)NCCSCc2ccccc2Cl SEW06533 CCCCc1ccc(c(c1)C)NC(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F AW01034 c1cc(ccc1/C=N/NC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-])C#N GK03621 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3cccc(c3)OC GK03417 Cc1nc(no1)Cc2ccc(cc2)[N+](=O)[O-] GK03626 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3)OC(F)(F)F GK03418 CCOC(=O)NC(=S)Nc1ccc(cc1Br)C(C)(C)C RF01584 c1ccc(cc1)COC(=O)NC(CCC(=O)O)C(=O)O KM08087 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3cc(nn3c4ccc(cc4)F)c5cccs5 SP00996 c1ccc(cc1)NC(=O)O/N=C(/CS(=O)(=O)c2cccs2)\N KM02310 CC(C)S(=O)(=O)c1cnc(nc1N)c2ccc(cc2)Cl KM02605 c1cc(oc1)c2nnc(o2)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-] GK03611 CC(C(=O)NNC(=O)c1ccc(cc1)[N+](=O)[O-])Oc2ccc(cc2)Oc3ccc(cc3)C(F)(F)F SEW06349 COc1ccc(c(n1)N2CCOCC2)NC(=O)CSCC(=O)O PD00771 c1ccc2c(c1)CC(C2)NC(=O)CSCc3c(cccc3Cl)F KM10514 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=S)Nc3ccccc3)C RH01885 CCc1cccc(c1NC(=O)NC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C AW01077 c1ccc(cc1)/C=N/NC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-] GK03623 CCOC(=O)CSC(=S)NCc1ccc(cc1)F PD00636 CCOC(=O)CSC(=S)NCc1ccc(cc1)C PD00637 CCCOc1ccccc1/C=N/NC(=S)Nc2cccc(c2C)Cl RDR01216 CCc1ccc(cc1)NC(=S)NNS(=O)(=O)c2ccc(cc2)C RDR01254 COCCCn1c(=O)c2ccccc2nc1S RDR01273 c1ccc(c(c1)CSCCNC(=O)Nc2ccc(cc2)C(F)(F)F)Cl SEW06528 CCCCc1ccc(cc1)NC(=O)NCCSCc2ccco2 KM10249 CC(C)(C)c1cc2c(s1)c(=O)[nH]cn2 GK03190 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)N SP00993 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cc(nn3c4ccccc4)c5ccc(cc5)OC(F)(F)F SP01015 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3ccc(c(c3)Cl)N4C(=O)CC5(C4=O)CCCC5 AW01043 c1ccc2c(c1)CC(C2)NS(=O)(=O)c3cccc(c3)Cl KM10513 c1cc(ccc1NC(=O)NC(=O)c2ccc(s2)[N+](=O)[O-])F RF01668 CC(C)(C)c1cc(n(n1)c2ccc(cc2)/N=C\c3ccccc3O)C(C)(C)C SEW06578 CC(C)(C)c1cc(n(n1)c2ccc(cc2)N3CC(CC3=O)C(=O)O)C(C)(C)C SEW06580 c1cc(ccc1c2csc(n2)Nc3ccncc3)[N+](=O)[O-] SEW06581 COc1ccc(cc1S(=O)(=O)NC2Cc3ccccc3C2)Cl KM10511 c1ccc2c(c1)CC(C2)NS(=O)(=O)c3ccc(s3)Cl KM10512 c1cc(oc1)CSCCNS(=O)(=O)c2ccc(cc2)Cl KM10384 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4nccs4 KM10390 COc1ccc(cc1)CNC(=O)Nc2ccccc2SC KM10324 Cc1ccccc1NC(=O)NCc2cccc(c2)OC KM10516 Cc1ccc(cc1)NC(=O)Nc2ccc(nc2)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06368 Cn1c(nnc1SCC(=O)N2CCOCC2)c3ccc4c(c3)cccn4 KM10456 Cc1c(cccc1Cl)NC(=O)NC2Cc3ccccc3C2 KM10463 CC(=O)Nc1ccc2c(c1)COCO2 SEW03603 c1ccc(cc1)OCCN2CCN(CC2)C(=O)c3c(cccc3F)F TB00003 c1ccc(cc1)OCCN2CCN(CC2)C(=O)c3ccco3 TB00004 CCOC(=O)c1ccc2c(c1)CC/C(=C\c3ccc(cc3)F)/C2=O SEW03710 c1ccc(cc1)CN2CCN(CC2)Cn3c4ccccc4nn3 PD00638 c1cc(c(c(c1)Cl)CSc2nc(cc(n2)O)O)Cl GK03629 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RH02048 Cc1cc([nH]c1c2ccn(n2)C(=O)c3c(nns3)C)C SP01255 c1ccc2c(c1)nnn2C3CCN(CC3)C(=O)c4ccc(cc4)Cl KM10223 COC(=O)c1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3cccc(c3)SC)N KM10221 c1cc(cc(c1)Cl)NC(=O)Nc2cccc(c2)Cl KM10199 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCCNc2c(cccn2)C(F)(F)F AW00873 Cc1ccc(n1c2ccc(cc2)c3nnc(n3c4ccc(cc4)Br)S)C RH01921 CCOC(=O)C(=C1CCN(CC1)Cc2ccccc2)C#N AW00943 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01044 CC(C)(C)OC(=O)NCCNS(=O)(=O)c1ccc(c(c1)Cl)N2C(=O)CC3(C2=O)CCCC3 AW01045 c1cc(c(cc1S(=O)(=O)N2CCN(CC2)c3nccc(n3)C(F)(F)F)Cl)N4C(=O)CC5(C4=O)CCCC5 AW01046 CC(C)(C)c1ccc(cc1)CSc2nc(cc(n2)O)N GK03628 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)Cc5c(cccc5Cl)F AW01087 c1cc(c(cc1Cl)Cl)CSc2nc(cc(n2)O)N GK03630 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)CNc4ccc(c(c4)[N+](=O)[O-])C PD00569 c1cc2c(cc1C3=NNC(C3)(C(F)(F)F)O)CCCC2 SP01307 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl SP01058 c1ccc(c(c1)NC(=S)NC(=O)c2cc(sc2)[N+](=O)[O-])Cl DFP00129 COC(=O)C1N(CCS1)S(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F SP01064 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cccc(c3)[N+](=O)[O-] SP01068 CC(=O)Nc1c(cc(cc1Cl)OC)Cl SEW03939 CC(C)(C)OC(=O)NC1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl AW01032 Cn1cc(cc1C(=O)OC)/C=C(\C#N)/S(=O)(=O)c2ccccc2 SEW06342 Cc1c2cc(ccc2sc1CC(=O)OC)Cl MWP00256 C/C(=C\c1ccccc1)/c2ccc3ccccc3c2 RJC03898 c1cc(c(c(c1)Cl)/C=N/c2ccc(c(c2)Cl)Cl)Cl GK03597 c1cc(c(cc1/N=C/c2cc(cc(c2O)Cl)Cl)Cl)Cl GK03598 c1cc(ccc1CSCCNC(=O)C(Cl)Cl)Cl SEW06365 COc1ccc(c(n1)N2CCOCC2)NC(=O)CC3(CCCC3)CC(=O)O PD00774 CCOC(=O)C1CCN(CC1)c2cc(nc3c2cc(cc3)C)C(F)(F)F KM10697 CCc1c(nc2ccccc2n1)N3CCCC3 GK03497 c1cc2c(cc1C3=NNC(C3)(C(F)(F)F)O)OCCO2 SP01306 COc1cc2c(cc1OC)ncnc2NCc3cccc4c3OCO4 GK03624 Cc1cc(c(c(c1)C)Nc2nc3cc(cc(c3s2)C)Br)C RDR00017 CC1Cc2cc(ccc2O1)C3=NNC(C3)(C(F)(F)F)O SP01344 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccccc3 SP01060 CC(C)(C)C(=O)Nc1c(cnn1C)Br GK03275 CC1C(=O)N(/C(=N/N=C/c2cccc(c2)[N+](=O)[O-])/S1)C(C)(C)C RF01574 Cc1ccc(cc1n2c(cc(=O)n(c2=O)Cc3ccccc3)N)OC KM09943 CC(C)(C)OC(=O)NCC(=O)NNC(=S)Nc1ccccc1 KM10394 CC(C)(C)OC(=O)NCC(=O)NNC(=S)NCc1ccccc1 KM10393 CCCc1c(nc(nc1O)SCC(=O)c2cccc(c2)[N+](=O)[O-])C RDR01520 Cc1ccc(n1c2cc(c(cc2C(=O)O)OC)OC)C GK03194 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])NCCNC(=O)C2CCC2 RH01920 c1cc(sc1)C(=O)Nc2ccc3c(c2)c(c[nH]3)C#N SP01310 c1ccc(cc1)N/N=C/c2ccc(c(n2)SCc3ccc(cc3)Cl)C#N SPB04270 c1c(c(cc2c1OCCO2)Br)C3=NNC(C3)(C(F)(F)F)O SP01347 CC1(CCC(c2c1ccc(c2)C3=NNC(C3)(C(F)(F)F)O)(C)C)C SP01343 c1ccc(cc1)c2csc(c2C(=O)c3ccccc3)Nc4ccccc4 SP01067 Cc1c(cc(o1)C(C)(C)C)c2c(c(n(n2)c3ccccc3)SC)C#N SP01088 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCSC3C(=O)OC SP01090 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCN(CC4)Cc5ccc(c(c5)Cl)Cl AW00964 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cccc(c3)C(F)(F)F SP01071 Cc1c(c(nc(n1)C23CC4CC(C2)CC(C4)C3)O)Cl RF02109 c1cc(c(cc1c2nc(cs2)C34CC5CC(C3)CC(C5)C4)Cl)F SPB08336 c1cc(cc(c1)Cl)N/N=C/c2cccn2c3cc(cc(c3)Cl)Cl SEW03064 c1ccc2c(c1)c(c([nH]2)c3ccc(cc3)Cl)C=C(C#N)C#N SEW03041 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Oc3ccccc3 SPB08279 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Oc3cccc(c3)[N+](=O)[O-] SPB08281 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F RH01919 c1ccc(cc1)NC(=S)NCCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F RH01917 Cc1nc(c(c(n1)SC)C#N)c2cccc(c2)CSc3ccccc3 KM06007 Cc1c2cc(ccc2sc1c3cc([nH]n3)C(F)(F)F)Cl SP01356 COc1cccc(c1)C(=O)Nc2c3ccccc3[nH]n2 SP01362 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)C(F)(F)F SP01072 COCCCN\1C(=O)CS/C1=N\N=C\c2ccc(c(c2)Cl)Cl RDR00378 Cc1c(cc(o1)C(C)(C)C)c2c(c(n(n2)C)SC)C#N SP01094 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4cccnc4 KM09592 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3csc(n3)Cc4ccsc4 MWP00534 Cc1ccc(c(c1)C(=O)NNC(=S)Nc2ccccc2C(F)(F)F)O MWP01118 CC(C)(C)C(=O)OC/C(=N/OC(=O)c1ccc(cc1)[N+](=O)[O-])/N RF03004 CC(C)(C)C(=O)OCc1nc(on1)c2ccc(cc2)[N+](=O)[O-] RF03006 Cc1cc2nnc(c(n2n1)C)/C(=N/O)/N KM01347 c1ccnc(c1)SCc2cccc(c2)/C(=N/O)/N KM01464 CC1CCN(CC1)c2ccc(c(c2)Oc3nc4cc(ccc4s3)Cl)[N+](=O)[O-] BTB06103 Cc1c(c(n[nH]1)C)Sc2ccc(cn2)C(F)(F)F SPB04327 CC1(OC(=O)C(C(=O)O1)Cc2ccc(cc2)[N+](=O)[O-])C RH02122 COC(c1ccnc(n1)SCc2ccc(cc2Cl)Cl)OC SPB04442 Cc1c(c(nc(n1)N)O)Oc2cccc(c2)C(F)(F)F SPB04458 CCOC(=O)NC(=S)Nc1ccc(cc1Cl)C(C)(C)C RF01583 c1cc(sc1)CCNS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW00966 C/C(=N\NC(=O)CSC1CN(C1)C(c2ccccc2)c3ccccc3)/c4ccc(cc4)[N+](=O)[O-] KM09881 CCC(CO)NC(=S)Nc1c(cccc1Cl)Cl RDR00430 Cc1c2c(cnn(c2=O)C)c(n1CCSCc3c(cccc3Cl)Cl)c4ccccc4 SP01103 c1cc(c(c(c1)F)C(=O)Nc2cccnc2)F SPB08376 CSc1c(cn(n1)c2ccccc2)c3nc(cs3)C45CC6CC(C4)CC(C6)C5 SPB08337 c1cc(cc(c1)[N+](=O)[O-])/N=C\c2cc(cc(c2OS(=O)(=O)c3ccc(cc3)F)Cl)Cl SJC00194 COc1cc(c(cc1OC)NC(=O)CSCC(=O)O)C(=O)OC GK03195 CC(C)(C)NC(=O)N1CCC(CC1)Nc2nccc(n2)C(F)(F)F AW00887 COc1cccc(c1NC(=O)NC(=O)c2c(ccc(c2OC)Br)OC)OC BTB07625 CN(C)CCCN/C(=N\O)/c1ccc(cc1Cl)Cl CD05822 CSc1cccc(c1)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM09253 c1ccc2c(c1)CC(C2)NC(=O)Nc3cc(cc(c3)Cl)Cl KM10467 c1ccc2c(c1)CC(C2)NC(=O)Nc3ccc(cc3F)F KM10465 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCN(CC3)Cc4ccccc4 SP01096 Cc1c2c(cn[nH]c2=O)c(n1CCSCc3c(cccc3Cl)F)c4ccccc4 SP01098 CC(=O)O/N=C(/c1ccc(nc1)N2CCN(CC2)c3c(cccn3)C(F)(F)F)\N SEW06307 Cc1cc(c(c2c1sc(c2C(=O)Oc3ccccc3)C(=O)OC)C)Cl PD00008 COc1ccc(cc1)NC(=O)c2ccccc2 SPB08372 c1ccc2c(c1)CC(C2)NC(=O)C3CCCCC3 KM10490 CCOc1ccc(cc1)NC(=O)N/C=C/c2ccsc2 GK03203 Cc1ccc(cc1)NC(=O)N/C=C/c2ccsc2 GK03205 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(s2)C3=CCOc4c3cccc4)/C#N SEW03781 c1cnc(cc1C(F)(F)F)N2CCN(CC2)C(=O)/C=C/C(=O)O SEW03805 c1ccc(c(c1)NC(=O)c2ccc(c(c2)Cl)Cl)Cl BTB06186 Cc1ccc(cc1)C(=O)c2c(ccc3c2cccc3)C RJC03830 C/C(=C\c1ccccc1[N+](=O)[O-])/c2cc3ccccc3c4c2cccc4 RJC03831 Cn1c(ccn1)NC(=O)NC(=O)c2c(cccc2Cl)Cl GK03202 Cc1c(c(n(n1)CC(=O)NCCSCc2ccco2)C)Br KM10479 CC(C(=O)O)Oc1ccc(cc1)OC RDR02440 c1ccc(c(c1)NC(=O)c2c(cccc2F)F)Cl SPB08381 CCC1CS/C(=N/c2ccc(c(c2)Cl)C)/N1 RDR00431 C=CCNc1nccc(n1)C(F)(F)F AW00879 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)COC(=O)c4ccc(cc4)C(C)(C)C PD00124 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)COC(=O)c4ccc(cc4)OC PD00127 c1ccc(cc1)c2cc(n(c(=O)c2C#N)N)c3ccccc3 RH02137 COCc1cc(cc2c1OCOC2)C(=O)Nc3ccc(cc3)Cl SEW03869 Cc1cc(cc(c1)/C(=N/O)/N)/C(=N/O)/N SEW03984 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F SEW03958 Cn1c(ccn1)NC(=S)Nc2ccc(cc2)Cl GK03198 Cc1cc(c(cc1Cl)C)S(=O)(=O)N2CCCN(CC2)Cc3ccc(cc3F)Br AW00866 Cc1cc(n2c(n1)cc(n2)c3ccc(cc3)Cl)C KM10461 c1cc(ccc1NC(=O)N2CCCN(CC2)Cc3ccc(cc3F)Br)Cl AW00909 CC(C)(C)OC(=O)N1CCCN(CC1)C(=S)Nc2cccnc2 AW00916 CC(C)NC(=O)CSc1nnc(n1C)c2ccc3c(c2)cccn3 KM10459 Cc1cc(c(c(c1)C)C(=O)NCCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C RH01893 Cc1cc(c2ccccc2n1)Nc3ccc(cc3)C(=O)C RH01894 c1cc(ccc1c2nc3cc(ccc3o2)CN4CCCCC4)Cl PD00043 c1cc(c(nc1)NCCN2C(=O)CC3(C2=O)CCCC3)C(F)(F)F AW00897 c1ccc(cc1)SCC(CN2CCC(CC2)Nc3nccc(n3)C(F)(F)F)O AW00865 CCOC(=O)c1cc2c(c(c1)CSc3ccc(cc3)Cl)OCOC2 SEW03866 CCOC(=O)c1c(nc(s1)C2COc3ccccc3O2)C KM06899 Cc1cccc(c1)Oc2ccccc2OC RJC03838 c1ccc(cc1)C(=O)COC(=O)c2ccc3ccccc3c2O RDR01443 c1ccc(cc1)C(=O)COC(=O)c2c(cccc2Cl)Cl RDR01457 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCC(=O)c3ccc(cc3)Cl RDR01489 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)N RH01891 CC(=O)c1ccc(cc1)Nc2ccnc3c2ccc(c3)Cl RH01892 c1cc(c(cc1NC(=O)Nc2ccc(c(c2)Cl)Cl)Cl)Cl PD00552 c1cc(ccc1NC(=S)NC(CO)(CO)CO)I PD00557 CC(=O)c1ccc(cc1)OCC(CN2CCCN(CC2)C(=O)c3cccs3)O AW00868 Cc1c(c(nc2n1nc(c2)c3ccc(cc3)Cl)SC)C(=O)C KM02150 c1ccc2c(c1)CC(C2)NC(=O)c3cc(cnc3)Br KM10481 Cc1c(c(co1)c2cc(ccc2Cl)F)C(=O)NC3Cc4ccccc4C3 KM10482 Cc1cc(c(c(c1)C)OC2CN(C2)C(c3ccccc3)c4ccccc4)C RH01864 CCn1c(c(c(=O)n(c1=O)CC)C=C2C(=O)N(C(=O)N(C2=O)CC)CC)O.c1ccncc1 RJC03860 c1ccc(cc1)C(=O)N2c3ccccc3OCC2=O RJC03965 Cc1ccc(cc1)Sc2c3cc(c(cc3ncn2)OC)OC GK03225 COc1c2c3c(sc2ncn1)CCCC3 GK03226 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)N3C(=O)C=CC3=O GK03443 CC(=O)N1CC(=O)N/C(=C/c2ccc(cc2)OC)/C1=O PD00658 c1ccc(cc1)c2nc3ccccc3c(n2)O RH01897 c1cc(cnc1)C(=O)NNC(=S)NCc2ccc(cc2)Cl RDR01850 c1ccc(c(c1)C#N)S(=O)(=O)Nc2ccccc2[N+](=O)[O-] JFD03874 Cc1ccc(cc1Cl)NC2=NCCS2 JFD03875 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)C RH02142 c1cc(sc1)SCC2=CS(=O)(=O)c3c2cc(cc3)Cl KM08697 CCOC(=O)CSc1c(cc(s1)C(=O)C)[N+](=O)[O-] KM08884 c1ccc(cc1)S(=O)(=O)c2cc(sc2)NC(=O)c3cccc(c3)Cl KM05907 CN(CCCCCc1cccc(c1)OC)C(=O)N RH01862 c1ccc2c(c1)c(=O)cc(o2)n3ccc(n3)C(F)(F)F KM10519 CC(C)n1c2ccc(cc2nn1)C(=O)Nc3ccc(cc3)Cl KM10506 c1ccc(cc1)S(=O)(=O)NC2Cc3ccccc3C2 KM10503 c1ccc(cc1)CN2CCC(CC2)N3C(=O)c4ccccc4C3=O PD00554 Cc1ccc(n1c2cc(c(cc2C(=O)NNC(=O)C(C)(C)C)OC)OC)C GK03214 CC1CN(CC(O1)C)S(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01064 Cc1cc(c2ccccc2n1)N3CCN(CC3)C(=O)c4ccco4 RH02140 Cc1ccc(cc1Cl)NC(=O)NC PD00560 CC(=O)O/N=C(\c1cnn2c1nc(cc2C(F)(F)F)C(F)(F)F)/N KM03129 c1ccc(c(c1)Sc2ccc(s2)c3ccccn3)Cl KM05129 c1csc(c1[N+](=O)[O-])SCCO KM06260 Cc1cc(c(c(c1)C)S(=O)(=O)O)C.CS(=N)(=O)c1ccc(cc1)Oc2ccc(cn2)[N+](=O)[O-] KM06270 COc1ccc(cc1)c2cc(n3c(n2)cc(n3)c4ccccc4)C(F)(F)F KM10524 COc1cc(cc2c1oc(=O)c(c2)C(=O)O)Br RH01879 Cc1ccc(cc1)NCC(Cn2cnc3c2c(=O)n(c(=O)n3C)C)O RJC03969 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COc3ccc(cc3)Br)O RJC03973 Cc1ccc(cc1)c2nc(on2)c3c(onc3c4c(cccc4Cl)F)C SP00770 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4ccccc4 SP00865 c1ccc(c(c1)c2cc(c(o2)C(F)(F)F)c3nc(no3)c4ccc(cc4)C(F)(F)F)Cl SP00797 CC(C)(C)c1cc(n(n1)Cc2ccccc2)c3nc(no3)c4ccccc4 SP00870 c1c(cc(c2c1c3cc(cc(c3[nH]2)Br)Br)[N+](=O)[O-])Br RJC03993 c1cc(cnc1)NC(=O)COCC(=O)O PD00785 c1cc(sc1)SCc2nc(on2)COc3ccc(cc3Cl)Cl SP01268 CNC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F GK03644 c1cc(oc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5c(c4)CCC5 KM10520 c1ccc(cc1)NNC(=O)c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F KM05960 COc1ccc(cc1)c2c(c[nH]n2)/C=N/Nc3cnc4ccccc4n3 SEW06352 c1cc(ccc1C(F)(F)F)NC(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW01065 CC(C)n1c2ccc(cc2nn1)C(=O)O KM10480 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCC(CC3)c4ccccc4OC AW01004 CCCCCc1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW01005 c1ccc2c(c1)c(c[nH]2)C3CCNCC3 RH02036 c1cc(ccc1C2CC(=O)N(C2=O)c3ccc(cc3)I)[N+](=O)[O-] S12472 c1cc2c(nc1)C(=O)N(C2=O)c3ccc(cc3OC(F)(F)F)Br S13234 c1cc(ccc1/C=N/c2ccc(cc2)OC(F)(F)F)Cl JFD04057 CS/C(=N\S(=O)(=O)c1ccccc1)/NNc2ccccc2 CD03053 Cc1c(cc2c(c1N)C(CC2(C)C)(C)C)N3CCCC3 CD03838 c1cc(ncc1C(F)(F)F)S(=O)(=O)Cc2ccc(o2)C(=O)O KM06293 CS(=NS(=O)(=O)c1cc(sc1Cl)Cl)(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06566 COc1ccc(cc1)c2c(c[nH]n2)/C=N/NC(=O)c3cccnc3 SEW06355 COc1ccc(cc1)c2c(c[nH]n2)/C=N/NC(=O)c3ccc(cc3)Cl SEW06356 Cn1c(c(cn1)Br)N2C(=O)c3ccccc3C2=O GK03263 CCCc1cnc(nc1)NCCNCC(COc2ccccc2)O AW00939 Cc1csc([n+]1CCCOC)Nc2ccc(cc2)Cl.[I-] RDR00400 CC(C)(C)c1cc(n(n1)c2ccc(cc2)/N=C\c3cc(cc(c3O)Br)Br)C(C)(C)C SEW06579 Cn1c(=O)n(sc1=O)c2cccc3c2cccc3 PD00642 c1cc(c(c(c1)I)C#N)Cl CD07335 Cc1c(snn1)C(=O)Oc2ccc(cc2)c3c([nH]nn3)C#N SEW03778 c1ccc(c(c1)n2cc(c(n2)N)C#N)Cl CD11759 COc1ccc(cc1)c2c(c[nH]n2)/C=N/NC(=O)c3cccc(c3)[N+](=O)[O-] SEW06353 c1ccc(cc1)c2csc3c2c(ncn3)NC4CCN(CC4)c5c(cc(cn5)C(F)(F)F)Cl AW01085 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C KM10690 CS(=O)(=O)/C(=C/c1cccn1c2ccc(cc2)OC(F)(F)F)/C#N SEW06336 Cc1c(cc(n1CCCN2CCOCC2)c3ccccc3)C(=O)Nc4ccncc4 SP00867 c1ccc(c(c1)C(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F)C(=O)O AW00987 CCCNC(=O)NC1CCN(CC1)c2c(cc(cn2)C(F)(F)F)Cl AW01074 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)NCc4ccco4 SP00933 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)Nc4ccc(cc4)c5ccccc5 SP00936 c1cc(oc1)C(=O)N2CCN(CC2)c3nc(ns3)c4cccs4 SPB08325 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)Nc2ccc(cc2F)F AW00914 COc1ccccc1C2CCN(CC2)C(=S)Nc3cccnc3 AW00915 c1ccc(cc1)c2csc3c2c(ncn3)N4CCNCC4 AW01086 COc1ccc(cc1)OCC(CNCCNc2nccc(n2)C(F)(F)F)O AW00924 Cc1ccc(cc1)S(=O)(=O)NNC(=S)NC RDR00414 CC(=O)c1ccc(c(c1)/N=C/c2cc(cc(c2O)Br)Br)Cl SJC00146 Cn1c(ccn1)NC(=O)Nc2cc(cc(c2)Cl)Cl GK03276 COc1cc2c(cc1OC)ncnc2NC3CCN(CC3)Cc4ccccc4 GK03273 c1cc2c(cc1Cl)nc[nH]c2=O RH01844 CC1CCc2c3ccc4c(c3ccc2C1=O)CCC(C4=O)C RJC03881 c1ccc(cc1)C(=O)C2CCCCC2=O RJC03883 c1ccc(cc1)c2csc3c2c(ncn3)NCc4ccccn4 AW01070 c1ccc(cc1)CCNc2c3c(csc3ncn2)c4ccccc4 AW01071 Cc1ccc(cc1)NC(=O)c2cc3cccc(c3[nH]2)[N+](=O)[O-] SP00919 c1c(cnc(c1Cl)N2CCC(CC2)N)C(F)(F)F AW01072 c1ccc(cc1)C(=O)NNC(=O)Nc2ccccc2 RH01911 c1cc(ncc1C(F)(F)F)NCCNC(=O)/C=C/C(=O)O AW00918 c1cc(cnc1)CNS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01091 c1cc(c(c(c1)Cl)CN2CCN(CC2)S(=O)(=O)c3ccc(c(c3)Cl)N4C(=O)CC5(C4=O)CCCC5)F AW01092 CC(C)n1c2ccc(cc2nn1)C(=O)OC KM10473 Cc1c(c(on1)C)C(=O)N2CCN(CC2)CCOc3ccccc3 TB00005 c1cc2c3c(c(cc4c3c1CCC4)Br)CCC2 RJC03899 COc1cccc(c1)SCC(=O)NC2Cc3ccccc3C2 KM10537 COc1ccc(cc1)c2ccnc(n2)SCC(=O)NC3Cc4ccccc4C3 KM10538 COc1ccc(cc1)c2nc(cs2)c3ccc(cc3)c4ccccc4.Br ML00290 Cc1c(c(n(n1)c2ccccc2)C)c3nc(no3)c4ccc(cc4)C(C)(C)C SEW04216 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)Nc4ccc(cc4)OC(F)(F)F SP00939 COc1cccc(c1C(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl)OC AW01080 COc1ccc(c(n1)N2CCOCC2)NC(=O)c3c(nccn3)C(=O)O PD00778 Cc1ccc(c(c1)C)NC(=S)N2C(CCCC2C)C AW01105 CC(CN1CCN(CC1)c2ccccc2OC)Nc3ccccn3 RH01866 CNCCNS(=O)(=O)c1ccc(c(c1)Cl)N2C(=O)CC3(C2=O)CCCC3 AW01095 Cc1ccc(cc1)/C=N/c2ccc(cc2)C GK03639 CCc1c(nc2ccccc2n1)N3CCN(CC3)S(=O)(=O)c4ccccc4 GK03645 Cc1c(sc(n1)CN2CCN(CC2)c3ccccc3OC)C(=O)C SP01250 CC1(OC(=O)C(=Cc2cccn2c3ccc(cc3)OC(F)(F)F)C(=O)O1)C SEW06339 Cc1ccc(cc1)Oc2ccc(cc2)C RJC03896 Cc1ccc(cc1)C#Cc2ccc(s2)C#Cc3ccc(cc3)C RJC03873 Cn1c(ccn1)NC(=S)Nc2ccc(cc2OC(F)(F)F)Br GK03279 c1cc(c(cc1NC(=O)c2c(c(sn2)Cl)Cl)Cl)F SPB08359 c1cc(ccc1NC(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F)OC(F)(F)F AW01075 c1cc(ccc1C(F)(F)F)NC(=O)NC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW01076 Cc1cc(n(n1)c2ccc(cc2)n3cccc3/C=C(\C#N)/S(=O)(=O)C)C SEW04334 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(c(c3)OC)OC GK03440 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)CCC(=O)O GK03444 Cc1c(cccc1Cl)/N=C\2/N(C(=O)CS2)Cc3ccco3 RDR00184 c1cc(cc(c1)[N+](=O)[O-])/C=N/NC(=S)N RF01528 CC(C)(C)c1cc(n(n1)c2c(cc(cn2)C(F)(F)F)Cl)C(C)(C)C SEW06572 Cc1cc(no1)NC(=O)/C(=C/c2cccs2)/c3ccsc3 SEW02122 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F SEW02207 Cc1ccc(cc1N2CC(CC2=O)C(=O)O)F SEW06299 CC1CC(=O)c2c3n1cc(c(=O)c3cc(c2F)F)C(=O)O RJC04111 c1cc(ccc1S(=O)(=O)CCC\2CCCC/C2=N\Nc3ccc(cc3[N+](=O)[O-])C(F)(F)F)Cl KM05807 CC(=O)c1c(cc(s1)c2ccc(cc2)F)NS(=O)(=O)c3ccccc3 GK03710 COC(c1ccc2c(c(sc2n1)C(=O)Nc3ccccc3)N)OC SPB04341 CC(C)NC(=O)c1cnn(c1n2cccc2)C GK03652 c1cc(c(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F)C(F)(F)F SP01063 Cn1c(c(cn1)C(=O)NC2CCCCC2)n3cccc3 GK03653 c1cc(ccc1NC(=O)NCc2c(cc(cn2)C(F)(F)F)Cl)Cl SPB04616 c1c(ccc(c1)OC(F)(F)F)/C=c\2/[nH]c(=O)/c(=C\c3ccc(cc3)OC(F)(F)F)/[nH]c2=O PD00661 c1ccc(cc1)/C=C/C(=O)NNC(=O)c2cc3c(s2)-c4ccccc4CC3 PD00663 c1cc(ccc1C(=O)CSC(=S)N2CCSCC2)Cl RF02035 COc1cc(c(cc1OC)NS(=O)(=O)c2ccc(cc2)Cl)C(=O)O GK03506 CCCCc1ccc(cc1)NC(=O)N2CCC(CC2)NC(=O)OC(C)(C)C TB00036 c1ccc(cc1)c2cc(c3ccccc3n2)NCCN4CCCCC4 RH02141 c1cnc(cn1)NC(=O)CSCC(=O)O PD00780 CCOC(=O)N1CCN(CC1)c2cc(nc3c2cccc3Cl)C(F)(F)F KM10542 COc1ccc(cc1OC)c2cc(n3c(n2)cc(n3)c4ccccc4)C(F)(F)F KM10540 COC(=O)c1ccc(cc1)Cn2cnc3c2cccc3 KM10736 Cc1c(c(no1)c2c(cccc2Cl)F)c3nc(no3)c4cccs4 SP00906 Cc1ccc(cc1)S(=O)(=O)N/N=C(\CCC(=O)OC)/c2ccn(c2)S(=O)(=O)c3ccccc3 RH02224 COc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)OC RH01928 Cn1c(c(cn1)C(=O)Nc2ccc(cc2)OC(F)(F)F)n3cccc3 GK03587 Cn1c(c(cn1)C(=O)Nc2cccc(c2)OC)n3cccc3 GK03588 CCOC(=O)NC(=S)Nc1ccc(cc1)C(C)(C)C RF01582 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccccc3Cl SP01069 CC(C)(C)c1cc(n(n1)c2ccc(cc2)NS(=O)(=O)c3cc(c(s3)Cl)Br)C(C)(C)C SEW06576 COc1ccccc1N2CCN(CC2)C/C(=N/O)/N SEW06569 COCCCNC(=S)NNS(=O)(=O)c1ccc(cc1)Cl RDR00420 CCC(CO)NC(=S)Nc1ccc(c(c1)Cl)C RDR00429 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(cc2)Cl RF02976 c1cc(cc(c1)Cl)c2c(nco2)C(=O)O SEW02011 CCN(CC)S(=O)(=O)c1ccc(c(c1)Cl)N2C(=O)CC3(C2=O)CCCC3 AW01049 CCOC(=O)C1CCN(CC1)c2c3cc(c(cc3ncn2)OC)OC HTS00369 c1ccc2c(c1)c(=O)sc(n2)NC(=O)c3ccc(cc3)[N+](=O)[O-] HTS01330 c1cc(oc1)C(=O)Nc2nc3ccsc3c(=O)s2 HTS01331 CS(=N/C=C(\C#N)/C(=O)C1CC1)(=O)c2ccc(cc2)Oc3cccc(c3C#N)F KM06612 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4ccccn4 KM09598 Cc1c2c(c(=O)n(n1)c3cccc(c3)C(F)(F)F)nc(s2)c4ccccc4 SPB04781 CCc1cc2c(=O)[nH]cnc2s1 GK00218 c1ccc(cc1)CCNC(=S)Nc2ccc(cc2)Oc3ccc(cc3)Cl RDR00912 COC(=O)c1c(noc1C(=O)N/N=C/c2c(cccc2Cl)Cl)c3c(cccc3Cl)Cl RF02173 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)c2ccc(cc2Cl)Cl TB00028 COc1ccc(cc1OC)NC(=O)CC2(CCCCC2)CC(=O)O PD00713 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Oc3ccccc3)C SPB08329 CSc1ccccc1N2CC(CC2=O)C(=O)O SEW06300 CN1CCN(CC1)c2ccccc2/C=N/c3cc(cc(c3)Cl)Cl SEW06308 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)c3nc(on3)C(C)(C)C SEW02540 Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)c(c[nH]3)C#N SP01311 CC1(CCc2cc(ccc2O1)c3ccnc(n3)S)C KM05834 c1cc(ccc1C2CC(=O)N(C(=O)C2)c3ccc(cc3F)I)C(F)(F)F PD00531 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)C(C)(C)C SP01070 c1cc2cccnc2c(c1)OS(=O)(=O)c3ccc(s3)c4ccno4 SEW06304 Cc1ccc(cc1C)/N=C/c2ccc(cc2)N(C)C RDR01032 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCc3ccc(c(c3)OC)OC PD00779 COc1ccc(cc1OC)C(=O)NCc2ccccc2 JFD02681 Cc1cc(ccc1c2ccccc2)c3ccccc3 RJC03805 Cc1nc(cn1CC(=O)c2ccccc2)[N+](=O)[O-] RH02121 CCOC(=O)c1c(c2cc(ccc2nc1SC)Cl)N3CCN(CC3)C KM10533 c1cc(oc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc(cc4)Cl KM10528 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)c3ccc(cc3)OC(F)(F)F RH02049 c1cc2c(c(c1)NC(=O)CSCC(=O)O)CCCC2 PD00307 Cc1ccc(cc1)N2CC(CC2=O)C(=O)O SEW06286 CCc1c(nc2ccccc2n1)N3CCN(CC3)S(=O)(=O)c4c(cc(cc4C)Cl)C GK03646 Cc1cc([nH]c1c2ccn(n2)C(=O)c3cc(oc3C)c4ccccc4)C SP01252 CC(C)N(CCOC(=O)C)S(=O)(=O)c1ccc(cc1)NC(=O)C RH01858 Cc1c(ccc(n1)C(F)(F)F)C(=O)N2CCCCC2 AW00896 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccccn3 PD00528 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCCN(CC2)C(=O)c3ccc(o3)[N+](=O)[O-] AW00846 c1cc2c(cc1C#N)nns2 KM10536 COc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3cc(cc(c3)F)F RH02051 c1cc(cc(c1)Cl)S(=O)(=O)Nc2c(cccn2)OCc3cc(cc(c3)F)F RH02052 COc1ccc(cc1)/C=N/c2ccc(cc2)OCCCOc3ccc(cc3)/N=C/c4ccc(cc4)OC RDR01976 COc1ccc(cc1)N2CC(CC2=O)C(=O)O SEW06285 c1cc(cc(c1)[N+](=O)[O-])N2CC(CC2=O)C(=O)O SEW06292 CCOC(=O)COc1ccc(cc1)NC(=O)C(Cl)(Cl)Cl RDR02019 CCN(CC)c1cnn(c(=O)c1Cl)c2ccc(cc2)C(F)(F)F SP01249 c1cc2c(cc1Cl)c(c(s2)Cl)CC#N MWP00122 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2Cc4ccc(cc4)F)C(=O)O PD00668 c1cc(c(c(c1)Cl)CS(=O)(=O)CC#N)F SPB02475 CC(=O)NC(=O)NCc1ccccc1 RJC03822 c1ccc(cc1)C(c2ccccc2)N3C(=O)c4c(nccn4)C3=O PD00499 Cc1ccc(cc1C)C(=O)OCC(=O)c2ccc(cc2)Cl RDR01564 Cc1cc(ccc1NC(=S)N2CCCCCC2)Br RDR01585 CC(C)(C)c1cc(n(n1)Cc2ccccc2)c3nc(no3)c4ccc(cc4)OS(=O)(=O)N(C)C SP00891 CCCCCCCCCc1ccc(cc1)Nc2ccccc2C(=O)O JFD03882 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)c3ccc(cc3)Cl)F TB00019 c1cc(c(c(c1)F)C(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F)F TB00020 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)CCC3 PD00666 COc1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4cccc(c4)SC KM10213 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)NCCSCc3ccco3 KM10383 c1cc(ccc1c2cc(n3c(n2)ccn3)C(F)(F)F)Cl KM10518 c1cc(sc1)c2nnc(o2)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-] GK03612 CC(C(=O)NNc1cnc2ccccc2n1)Oc3ccc(cc3)Oc4ccc(cc4)C(F)(F)F SEW06351 c1cc(cc(c1)Cl)N2CCN(CC2)CC#N SEW06568 CCCc1ccc(cc1)c2nc(no2)c3cccs3 SP00868 CCn1c(c(c(n1)C)Br)c2nc(no2)c3ccccc3 SP00869 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl SP00892 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3ccno3 SP00901 Cc1cccc(n1)CC(c2ccccc2)(c3ccccc3)C(=O)OC JFD03880 CC(C)(C)c1ccc(cc1)C(=O)NNC(=S)Nc2ccc3c(c2)OCO3 TB00026 c1ccc(cc1)CN2CCC(CC2)NS(=O)(=O)c3cccs3 TB00033 Cc1cc(c(c(c1)C)CSCCNC2=CC(=O)CC(C2)c3ccc(cc3)Cl)C SEW06585 c1cc(oc1)CNC2=CC(=O)CC(C2)c3ccc(cc3)Cl SEW06587 CCCc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3cc(cc(c3)F)F RH02054 CCCc1cc(nc(n1)SCC(=O)NCCSCc2ccco2)O KM10389 COc1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3ccccc3SC)N KM10359 Cc1c(c(no1)C(=O)NNC(=O)Nc2cccc(c2)Cl)c3csc(n3)C SPB03395 c1ccncc1.C(=C1C(=O)NC(=S)NC1=O)c2c([nH]c(=S)[nH]c2=O)O RJC03826 CC1(CCc2c1cc(cc2c3cc([nH]n3)C(F)(F)F)C(C)(C)C)C KM10340 CS(=NC(=O)c1ccc2c(c1)snn2)(=O)c3ccccc3 KM10337 CN(C)S(=O)(=O)Oc1ccc(cc1)c2nc(on2)c3ccc(cc3Cl)F SP00894 COc1cc(cc(c1OC)OC)CCC(=O)O RDR01646 CCc1ccccc1NC(=S)NC(C)(C)CO RDR01687 c1cc(c(c(c1)Cl)OC(=O)c2ccc(c(c2)Cl)Cl)Cl RDR01770 c1(c(c(c(c(c1F)F)S(=O)(=O)N)F)F)F SEW04027 Cc1cn(nc1c2cccs2)S(=O)(=O)c3csc(c3Br)Cl SP01277 CC(C)n1c2ccc(cc2nc1C(F)(F)F)C(=O)N3CCOCC3 KM10740 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)c2c(cccc2F)F TB00038 c1ccc(cc1)CSCC(=O)NCCSCc2ccco2 KM10387 CC(C)(C)C(=O)NNC(=O)CSc1c2c3c(sc2ncn1)CCCC3 GK03268 Cc1ccc(cc1)/C(=C/c2ccc(cc2)Cl)/C#N SJC00404 Cc1cc(c(c(c1)C)NC(=O)CCC(=O)O)C SJC00441 Cn1c(c(cn1)C(=O)Nc2cccc(c2)F)n3cccc3 GK03614 CC(C)NS(=O)(=O)c1ccc(c(c1)Cl)N2C(=O)CC3(C2=O)CCCC3 AW01090 CCCCNS(=O)(=O)c1ccc(c(c1)Cl)N2C(=O)CC3(C2=O)CCCC3 AW01093 c1cc(ccc1c2nc(on2)c3ccno3)OC(F)(F)F SP00898 c1cc(ncc1C(F)(F)F)c2nc(on2)c3ccno3 SP00902 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=S)Nc3ccc(cc3)OC)C RH01888 c1ccc2c(c1)ncc(n2)N3CCC(CC3)C(=O)NC(=O)NCCCN4CCOCC4 SEW04046 Cc1cc(c(o1)C)C(=O)n2cc(c(n2)c3cccs3)C SP01276 c1cc(ccc1OCC#N)Br RJC03947 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)/C=N\c3cccc(c3)SC SJC00182 CC(C)(C)OC(=O)NCC(=O)NNC(=S)NCC=C KM10392 CC(C)(C)NC(=S)N/N=C/c1ccco1 SJC00395 Cc1ccc(cc1)/C(=C/c2cc(c(c(c2)OC)OC)OC)/C#N SJC00402 c1ccc(c(c1)C(=O)NCCNc2ccc(cn2)C(F)(F)F)C(=O)O AW00911 c1cc(oc1)CNC(=S)N GK03251 Cc1c(c2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)Cl)Cl KM10362 Cc1ccc(cc1)NC(=S)NNC(=O)c2ccc(cc2)n3c(ccc3C)C RH01886 c1ccc(cc1)/C=C\2/C=C(OC2=O)c3ccccc3 SEW04443 CC(=O)NC(Cc1ccc(cc1)OC(=O)C)C(=O)O KM08348 c1ccc2cc(ccc2c1)C(=S)N SPB07522 Cc1ccccc1NC(=O)c2cc(n(c2C)CCSC)c3ccccc3 SP00912 CCCCNc1c2c(csc2ncn1)c3ccccc3 AW01069 CCc1cccc(c1NC(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C AW01066 CN1c2ccsc2-c3c(cnc(n3)SCc4ccc(cc4)Cl)S1(=O)=O KM06797 c1cc(ccc1NC(=O)CCC(=O)O)F SJC00442 Cc1c(c(n(n1)c2ccccc2)N)c3ccccc3 RJC03975 CCOC(=O)c1cc(oc1/C=N/OC(=O)c2ccco2)c3ccc(cc3)Cl SP00953 Cc1c(c(c([nH]1)C)C(=O)OC)/C=N/OC(=O)c2ccco2 SP00959 Cc1c(c(c([nH]1)C)C(=O)OC)/C=N/OC(=O)c2cccs2 SP00958 c1ccc(cc1)OCCN2CCN(CC2)S(=O)(=O)c3ccccc3Cl TB00010 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CCOc3ccccc3 TB00011 CC(C)c1ccc(cc1)NC(=O)N2CCCN(CC2)CCOc3ccccc3 TB00014 Cc1c(c(n(n1)c2ccccc2)C)C(=O)N SEW04158 c1ccc(cc1)C(=O)Oc2cccc3c2cccc3 RJC03885 CSc1cccc(c1)/N=C\c2cc(cc(c2OS(=O)(=O)c3ccc(cc3)F)Cl)Cl SJC00192 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCN(CC4)c5nc6ccccc6s5 AW01058 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)Nc3cccc(c3)C(F)(F)F SP00913 COc1ccccc1NC(=O)NC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW01073 c1cc(ccc1NC(=O)Nc2ccc(cc2)Cl)OCC(CN3CCCCC3)O AW00910 c1ccc(cc1)CN2CCC(=NO)CC2.Cl RH01871 Cc1cccc(c1NC(=O)c2cccc3c2cccc3)C RH01869 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc4ccccc4c3 KM10365 c1cc(ccc1C(=O)OCCSC2CS(=O)(=O)c3c2ccc(c3)[N+](=O)[O-])Cl KM08383 CC(=O)OC[C@@H]1[C@@H]([C@@H]([C@H]([C@H](O1)Oc2c(c(c(c(c2Br)Br)Br)Br)Br)OC(=O)C)OC(=O)C)OC(=O)C RJC03890 c1cnc(nc1C(F)(F)F)N2CCC(CC2)NC(=O)/C=C/C(=O)O AW00984 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)Nc3ccccc3 SP00510 CC(C)(C)NC(=S)N/N=C/c1c[nH]nc1c2ccc(cc2)OC SEW06354 Cc1ccc(cc1)NC(=O)c2cc(n(c2C)CCSCc3c(cccc3Cl)F)c4ccccc4 SP00937 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCCC4 AW01078 Cc1ccc2c(c1)nc(cc2N3CC4CCC(C3)CC4)C(F)(F)F KM10696 CCCc1cnc(nc1)N2CCCN(CC2)C(=S)Nc3cccnc3 AW00925 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3Cl)F GK03439 c1cc(ccc1c2cc(n3c(n2)cc(n3)c4ccc(cc4)Cl)C(F)(F)F)Cl KM10484 c1cc(ccc1C2(CCN(CC2)S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F)O)Cl SP01056 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SP01057 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)Nc2ccc(c(c2)Cl)F TB00032 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCCCCCO PD00781 COc1ccc(cc1OC)S(=O)(=O)Nc2cc(c(cc2C(=O)OC)OC)OC GK03107 COc1cc(c(c(c1)Cl)NC(=O)c2ccc(cc2)Cl)Cl SEW03918 CCOC(=O)C(C#N)C(=O)c1c(onc1c2c(cccc2Cl)Cl)C CD05945 Cc1ccc(c(c1)C)Sc2cc(c(cc2N)C)C RJC03897 Cc1c2cc(ccc2sc1CC(=O)NN)Cl MWP00364 c1cc(sc1)c2nc(sn2)N3CCN(CC3)C(=O)c4cccs4 SPB08326 CN(Cc1ccccc1)C(=S)Nc2ccc(cc2)Cl GK03266 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NNC(=O)CSc2c3c4c(sc3ncn2)CCCC4)C(F)(F)F GK03265 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)Nc4ccc5c(c4)OCCO5 SP00934 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)Nc4ccccc4Cl SP00940 c1ccc(cc1)NC(=O)CCC(=O)O RH01868 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SP01051 c1cc2c(cc1F)c3c([nH]2)CN(CC3)S(=O)(=O)c4ccc(s4)c5cc(on5)C(F)(F)F SP01054 CC(=O)N1CC(=O)N/C(=C/c2ccco2)/C1=O PD00660 c1c(c(nc(n1)S)N)C#N KM08132 CC(=O)O[C@@H]1[C@H](O[C@@H]([C@@H]([C@H]1OC(=O)C)OC(=O)C)OC)CO RJC03791 CC(=O)O[C@@H]1[C@H](O[C@@H]([C@@H]([C@H]1OC(=O)C)OC(=O)C)OC)COC(c2ccccc2)(c3ccccc3)c4ccccc4 RJC03793 CC1=C(CC(C(C1)C(=O)Nc2ccc(nc2N3CCOCC3)OC)C(=O)O)C PD00776 c1ccc(cc1)N2CCN(CC2)C(=O)CN3CCCCC3 KM10735 Cc1ccc(n1c2ccc(cc2)c3nnc(n3c4ccccc4)S)C RH01912 c1ccc2c(c1)cnn(c2=O)CCOC(=O)c3cccs3 PD00599 CC1=C(CC(C(C1)C(=O)NCc2csc3c2cccc3)C(=O)O)C PD00601 c1ccc2c(c1)CC(C2)NC(=O)CSc3ccc(cc3)F KM10559 Cc1ccccc1C(=O)Nc2ccccc2F RDR01805 c1ccc(cc1)C#Cc2ccc(o2)C(=O)N3CCCC3 KM08687 CCC(C)c1ccccc1NC(=O)c2cc3cccc(c3[nH]2)[N+](=O)[O-] KM11032 Cc1cc(c2cc([nH]c2c1)C(=O)N(C)c3ccc(cc3F)F)C KM11034 c1ccc(c(c1)NC(=S)NCCNC(=S)Nc2ccccc2F)F RDR00564 Cn1c2cccc(c2c(n1)NC(=O)COCC(=O)O)F HTS00769 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCc3ccncc3 PD00786 Cc1cc(n(n1)c2cc(c(cc2Cl)S(=O)(=O)O)Cl)O RJC04098 c1cc(c(cc1[N+](=O)[O-])CO)N2CCN(CC2)c3ccc(cc3CO)[N+](=O)[O-] RH02175 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)N RH02176 Cc1cc(c2ccccc2n1)N3CCN(CC3)c4nc5cc(ccc5s4)Cl RH02177 CCOC(=O)/C(=C/Nc1cccc(c1)OC)/C#N RH02237 Cc1nc(cn1CC(c2ccc(cc2)Cl)O)[N+](=O)[O-] RH02226 c1ccc2c(c1)CC(C2)NC(=O)Cn3c4ccccc4nn3 KM10562 CS(=O)(=O)CS(=O)(=O)Oc1ccc(cc1Cl)Cl CD11199 COc1cc2c(cc1OC)ncnc2NCC=C GK03348 COc1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3ccccc3C(F)(F)F)N KM10585 COc1ccc(cc1)OCCNC(=O)c2c(cccc2Cl)F SPB08188 c1cc(c(cc1F)N)n2ccnc2 SS00044 COC(=O)C(Cc1c[nH]c2c1cccc2)N.Cl RH01792 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCc3ccccc3 PD00783 Cc1cc(=O)[nH]c(n1)c2ccccn2 RDR03731 Cc1c(c(nc(n1)c2ccccn2)N(C)Cc3ccccc3)Cl SEW02973 CO/N=C/c1nc2ccccc2s1 SEW03004 c1cc(c(cc1Cl)Cl)/C=C/2\COc3ccc(cc3C2=O)Cl SEW03023 c1ccc(cc1)C(=O)NC(CO)C(=O)O JFD03889 c1ccc2c(c1)ccc3c2[nH]c4c3ccc5c4cccc5 JFD03891 CN(C)c1cccc2c1cccc2S(=O)(=O)NN JFD03892 COc1ccc(cn1)NC(=O)c2cccs2 SPB08388 c1ccc2c(c1)CC(C2)NC(=O)CSc3ccc(cc3)Cl KM10560 c1ccc2c(c1)cc(o2)C(=O)CSc3[nH]c(=O)c4ccccc4n3 PD00722 CCc1ccc2c(c1)cc([nH]2)C(=O)N(C)c3ccc(cc3F)F KM11037 CC(C)(C)OC(=O)NCCNC(=O)C1CCN(CC1)c2nccc(n2)C(F)(F)F AW01261 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)c4ccc(cc4)F)[N+](=O)[O-] HTS00991 c1cc(c(c(c1)Cl)NS(=O)(=O)c2ccc(cc2)N)F CD05954 COc1cc(cc(c1OC)OC)CCC(=O)NNC(=O)C(F)(F)F SEW04146 c1cc(ccc1c2nc(cs2)C(=O)NN)C(F)(F)F RF04269 Cn1c(nnc1SCC#N)c2ccc3c(c2)cccn3 KM10643 c1cc(c(cc1S(=O)(=O)N2CCSCC2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01050 C=CCn1c(nnc1SCC#N)c2ccc3c(c2)cccn3 KM10644 Cn1c2c(cn1)c(ncn2)N3CCOCC3 GK03447 c1cc(ccc1CCC(=O)O)[N+](=O)[O-] RH02123 Cc1c(c2cc(ccc2[nH]1)C(C)C)CC(=O)O RH02124 CC(=O)/C(=C\N(C)C)/Sc1ccccc1 SPB04574 c1ccc(cc1)NC(=O)c2ccc(cc2)Br JFD03951 c1cc(cnc1)c2nc(cs2)C(=O)NNC(=O)c3ccc(cc3Cl)Cl MWP01177 COc1ccccc1NC(=S)N/N=C/c2ccc(c(c2)OC)O RDR00442 COc1ccccc1NC(=S)N/N=C/c2ccco2 RDR00443 c1ccc(cc1)C(=O)Nc2cccc(c2)Cl SPB08383 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccc(c(c2)F)F)C RJC04084 CC(C)(CO)NC(=S)Nc1cccc(c1)F RDR00453 Cc1ccc(cc1)n2cccc2 SEW04206 c1ccc(c(c1)CCOC(=O)c2ccc(cc2)C(F)(F)F)/C=C\[N+](=O)[O-] RH01876 CC(C(=O)Nc1ccc(cc1)OC)Oc2ccc(cc2)Oc3ccc(cc3)C(F)(F)F SEW06311 c1cc(oc1)CN2C(=O)CC(CC2=O)c3ccc(cc3)C(F)(F)F PD00539 Cc1c(c(n(n1)c2ccccc2)C)c3nc(no3)c4ccccc4 SEW04214 CCOC(=O)N1CCN(CC1)c2cc(nc3c2cccc3)C(F)(F)F KM10508 c1cc2c(c3c1c4c(cc3)C(=O)CCC4)CCCC2=O RJC03878 CSC(=N)Nc1csc(c1c2ccccc2)C(F)(F)F.I SEW03409 Cc1c(ccc(n1)C(F)(F)F)NC(=O)N2CCCN(CC2)Cc3c(cccc3Cl)F AW00927 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc4c(c3)c(c[nH]4)C#N SP01293 CCOC(=O)c1cnn(c1C(F)(F)F)c2ncc(c(n2)C(F)(F)F)C(=O)OC GK03738 c1ccc2c(c1)[nH]c(n2)COCC(=O)O PD00810 Cn1c2c(cn1)c(ncn2)NC3CCCCC3 GK03455 Cn1c(nnc1SCc2cc(cc(c2)F)F)c3ccc4c(c3)cccn4 KM10647 CC(C)(C)OC(=O)NCc1nnc(n1c2ccccc2)S KM10565 CC(C)CC(C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 RJC04010 CC(C)(C)c1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccccc4F)[nH]cn3 KM09822 CN(C)/C=C(\C#N)/S(=O)(=O)c1ccsc1 SEW04153 Cc1ccc(n1c2ccc(cc2)C(=O)NN)C RH01873 c1ccc(cc1)C(=O)NC(=S)NNc2c(cccn2)n3cccc3 SEW04277 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccco3 GK03425 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)c4c(cccc4Cl)Cl)[N+](=O)[O-] HTS01009 Cc1cc(=O)oc2c1c(cc(c2)O)O JFD03945 CCN(CC)C(=O)Cc1c2ccccc2sc1Cl KM07289 CC1(Cc2c(c(sc2C(=O)OC)SC)/C(=N\OC(=O)c3c(cc(cn3)C(F)(F)F)Cl)/C1)C KM07567 c1cc(c(cc1NC(=S)N/N=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl)Cl RDR00734 Cc1cccc(c1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3)C KM09959 c1ccc2c(c1)ccc(c2Br)C(=O)O JFD03900 CCCCCCCOc1ccc(cc1)C(=O)O JFD03907 Cc1c(sc(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)C(=O)/C=C/N(C)C SEW05036 CC(C)c1cc(c(c(c1)Br)NC(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F)Br AW01036 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)c2ccco2 AW01037 Cc1cc(no1)NC(=O)CC(CC(=O)O)c2ccc(cc2)C(F)(F)F PD00671 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2CC4CC4)C(=O)O PD00672 COc1ccccc1N2CCN(CC2)Cc3nc(cs3)c4ccc(cc4)[N+](=O)[O-] SEW06639 Cc1c(cccc1n2c(cc(=O)n(c2=O)Cc3ccccc3)N)C(=O)OC KM09979 CCOC(=O)c1c(n[nH]c1/N=C/c2ccncc2)C RJC04090 Cc1cc2[nH]nc(n2n1)c3ccccc3Cl RJC04094 CCOC(=O)c1c(n[nH]c1N/N=C/c2cccc(c2)O)C RJC04092 Cc1cc2[nH]nc(n2n1)c3ccc(cc3)C(F)(F)F RJC04093 Cc1ccc(cc1)C(=O)NNC(=O)c2ccc(cc2)n3c(ccc3C)C RH01935 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)C(=O)NN SPB08117 CC(C(=O)Nc1c(cccc1F)F)N2CCN(CC2)c3nccc(n3)C(F)(F)F AW00895 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccc(cc2)C(F)(F)F)C RJC04091 CC(c1ccco1)N(c2ccccn2)C(=O)c3c(c4ccccc4s3)Cl RJC04096 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)N3CCOCC3 SP00576 CN(c1cccc(n1)C(F)(F)F)/N=C/c2cc(c(s2)C(F)(F)F)c3ccccc3 SEW03692 c1ccc(cc1)c2cc(sc2C(F)(F)F)/C=C\3/CSc4ccc(cc4C3=O)Cl SEW03698 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCCCN.Cl PD00703 c1cc(ccc1N2CC(=O)N(CC2=O)CC3CC3)OC(F)(F)F PD00706 COc1c(c(cc(c1)/C=N/CCCN2CCN(CC2)CCC/N=C/c3cc(c(c(c3)OC)OC)OC)OC)OC CD01027 CC(C)(C)C(=O)NNC(=O)c1cccc(c1)[N+](=O)[O-] SEW06571 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)CC#N SEW06588 Cn1c(ccn1)NC(=O)NC(=O)c2c(cccc2F)F GK03204 Cn1c(c(cn1)Br)N GK03207 CCc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH01933 CC(C(=O)Nc1c(cccc1Cl)Cl)Oc2ccc(cc2Cl)Cl RDR02520 Cc1ccc(n1c2c(c3c(s2)CCCC3)C(=O)NN)C GK03208 CCOc1ccc(cc1)/C=N/NC(=S)Nc2cc(c(cc2OC)Cl)OC CD03236 c1ccc(cc1)C(=S)N2CCOCC2 S12105 c1ccc(cc1)C(=S)N2CCSCC2 S12106 CC(C)(C)C(=O)NNC(=O)c1ccc(o1)Oc2ccc(cc2)C3SCCS3 SPB02437 c1c(c(sc1Br)Br)CC(=O)NN SPB02938 Cc1c(c(on1)c2c(nns2)C)c3nc(no3)c4ccc(s4)[N+](=O)[O-] SPB03420 CC1=CC(=O)C(=CC1=O)C(C)C JFD03914 Cc1c(ccc(n1)C(F)(F)F)C(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl AW00871 c1cc(c(cc1OCC(CN2CCC(CC2)Nc3nccc(n3)C(F)(F)F)O)Cl)Cl AW00901 CCCc1cnc(nc1)NCCNCC(COc2ccc(c(c2)Cl)Cl)O AW00907 c1csc(n1)C2=NNC(C2)(C(F)(F)F)O KM10449 CCOC(=O)c1cc2c(ccnc2NCc3ccc(cc3Cl)Cl)nc1C(F)(F)F SPB04554 CCCc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3n4cccc4)[N+](=O)[O-] HTS01010 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3ccccc3C(F)(F)F)C RH01936 c1ccc(cc1)NC(=O)c2cccc(c2)C(F)(F)F SPB08373 CC(=O)c1c(cc(s1)c2ccccc2)NC(=O)c3ccc(c(c3)OC)OC GK03715 c1ccc(c(c1)CCOC(=O)c2ccc(cc2)Cl)/C=C\[N+](=O)[O-] RH01877 CCON1C(=O)c2ccccc2C1=O JFD03908 Cc1c(c(c2ccccc2n1)C(=O)O)O JFD03910 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2ccc(cc2)F S13215 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2c(cccc2Cl)F S13216 Cc1cccc(c1C)C(=O)Nc2cccnc2Oc3ccc(cc3)OC RH01908 CCOC(=O)c1cc(nn1Cc2c(cc(cc2C)C)C)C(C)(C)C SPB08109 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)c3nnc(n3c4ccccc4)S SPB08133 Cc1ccccc1C(=O)c2ccccc2C(=O)O BLT00214 CC1CN(CC(O1)C)c2c3c(ccs3)ncn2 GK00378 c1cc2c(nc1)ncn(c2=O)CCCN3CCOCC3 RJC03956 c1ccc(cc1)N2CCN(CC2)CCCOc3ccccc3C(=O)N RJC03957 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3cccc(c3)Br PD00538 c1cc(ccc1NC(=O)c2cnccn2)I PD00540 COc1cc(cc(c1)OC)NC(=O)c2cnccn2 PD00541 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)NNC(=S)NC3CCCCC3 SPB08143 c1cc(c(cc1I)I)NC(=O)/C=C/C(=O)O RDR02669 CC(=O)Oc1cccc2c1C(=O)C=CC2=O RJC03855 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3ccc(cc3F)Br KM06926 c1ccc2c(c1)c(c(s2)Cl)CC(=O)N3CCCCC3 KM07286 c1ccc(cc1)Oc2cc(nc3c2cccc3Br)C(F)(F)F KM07542 c1cc(cnc1)NC(=S)NCCCNc2c(cc(cn2)C(F)(F)F)Cl AW00919 c1ccc(c(c1)NC(=O)CN2CCOCC2)Sc3nccc(n3)C(F)(F)F AW00921 Cc1cc(ccc1NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Br RDR00491 Cc1ccc(n1c2c(c3c(s2)CCCC3)C(=O)NNC(=O)C(C)(C)C)C GK03227 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)c4c(cccc4F)F)[N+](=O)[O-] HTS01011 CN(C)c1ccc(cc1C#N)/C=N/c2ccc(cc2)OC SEW06309 COc1ccc(c(c1)S(=O)(=O)Oc2ccc3ccccc3c2I)OC RDR02614 c1ccc2c(c1)CC(N3C2=NCC3)(c4ccc(cc4)F)O JFD03924 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccnc3Oc4ccc(cc4)Cl RH01940 Cc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH01939 CCOC(=O)c1c(nc(s1)n2cccc2)C SPB02685 c1cc(ccc1N2C(=O)CC3(C2=O)CCCC3)Br AW00960 COc1ccccc1C2CCN(CC2)c3c4c(csc4ncn3)c5ccccc5 AW00962 Cn1c2c(cn1)c(ncn2)OC GK03449 CC(=O)c1ccc(cc1)N2C(=O)CSCC2=O PD00670 CC(C)(C)c1cc(n(n1)c2cnc3ccccc3n2)C(C)(C)C SEW06586 CC(=O)Nc1ncc(s1)[N+](=O)[O-] JFD03897 c1ccc2c(c1)ccc3c2cccn3 JFD03898 CCOC(=O)c1cc(nc(c1C#N)O)c2ccc(cc2)Cl RF01079 Cn1c(nnc1SCC(=O)N2CCN(CC2)c3ccccc3)CSc4ccnc5c4ccc(c5)Cl HTS01210 CC(=O)Oc1ccc(c2c1C(=O)c3ccccc3C2=O)OC(=O)C RJC03865 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COc3ccccc3)O RJC03972 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN3CCN(CC3)c4ccccc4OC)O RJC03971 CC(=O)Nc1ccc(c(c1)C(=O)O)O JFD03890 c1ccc(cc1)c2nc(on2)c3ccc(cc3Cl)F SP00872 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(C)(C)C)C(C)(C)C SEW06574 CC(C)(C)c1cc(n(n1)c2ccc(cc2)NC(=O)c3cccs3)C(C)(C)C SEW06575 Cc1ccc(cc1C)NC(=O)C(=O)N/N=C/c2ccc3c(c2)OCO3 BLT00075 c1ccc2c(c1)c3c(n(c2=O)Cc4ccc5c(c4)OCO5)-c6ccccc6C3=O PD00707 c1cc2c(cc1C3=NNC(C3)(C(F)(F)F)O)CCO2 SP01259 C1C2CC3CC1CC(C2)(C3)C4=NNC(C4)(C(F)(F)F)O SP01345 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)C(=O)NNC(=S)Nc3ccccc3 SPB08132 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)NN SPB08116 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/Cc3ccc(cc3)C(C)(C)C)\N RF01765 c1cc2c(cc(c(c2nc1)O)I)S(=O)(=O)O JFD03939 Cc1c2cnn(c(=O)c2c([nH]1)C)C SP01108 c1ccc(cc1)N/C=C\2/C(=O)c3ccccc3NC2=O RH01931 c1ccc2c(c1)ncn2CN3CCC(CC3)C(=O)N HTS00629 c1ccc(cc1)C(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS00725 CC(C)(C)c1ccc(cc1)C(=O)NCCSCc2ccc(cc2)Cl SEW06361 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)Nc4cccc(c4)C(F)(F)F SP00935 COc1cc(cc(c1OC)OC)C(=O)Oc2c(cc(cc2Cl)Cl)/C=N\c3cccc(c3)C(F)(F)F SJC00209 COc1cc(cc(c1OC)OC)C(=O)Oc2c(cc(cc2Cl)Cl)/C=N\c3cccc(c3)[N+](=O)[O-] SJC00210 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CNc3ccccc3OC)O RJC03970 CCn1cc(c(=O)c2c1nc(cc2)C)C(=O)O RJC03974 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCOCC3 SP01074 c1ccc(cc1)c2csc3c2c(ncn3)NC4CC4 AW00972 CCOC(=O)C1CCN(CC1)c2c3c(csc3ncn2)c4ccccc4 AW00969 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCN(CC4)c5ccc(cn5)C(F)(F)F AW00970 CC(C)c1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3cc(cc(c3)F)F RH02055 CCCCCc1ccc(cc1)C(=O)Nc2cccnc2Sc3ccc(cc3)C RH02058 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)Nc2cc(cc(c2)Cl)Cl TB00030 COc1ccc(cc1)OCc2nc(cs2)c3ccc4c(c3)OCCO4 SPB08262 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)Nc2ccc(cc2F)F TB00031 Cc1cc(c(cc1Cl)C)S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00953 CC(=O)c1ccc(cc1)NC(=O)CSCC(=O)O PD00665 c1ccc2c(c1)C(C(N(C2=O)Cc3ccc(cc3)F)c4ccncc4)C(=O)O PD00669 CCCc1ccc(cc1)S(=O)(=O)Nc2cccnc2Sc3ccc(cc3)C RH02053 c1cc(ccc1c2nnc(o2)c3cnn(c3C(F)(F)F)c4ccc(cc4)Cl)Cl HTS01028 COc1ccc(cc1OC)N2C(=O)CC3(CCCCC3)CC2=O PD00714 c1cc(c(cc1I)F)NC(=O)CC2(CCCCC2)CC(=O)O PD00716 Cc1cccc(c1OC(=O)c2cc(nn2Cc3c(cc(cc3C)C)C)C(C)(C)C)Cl SPB08330 c1cc(c(c(c1)Cl)Cl)C(=O)Nc2cccnc2 SPB08377 c1cc(ccc1CSCCNC(=O)c2ccc(cc2)Cl)Cl SEW06362 c1cc(c(c(c1)F)C(=O)Nc2ccc(cc2)C(F)(F)F)F SPB08378 c1ccc(cc1)NC(=S)NNC(=S)Nc2ccccc2 PD00334 COc1cc2c(cc1OC)C(=O)CC2 JFD03942 COC(=O)c1ccc(c(c1)CSc2ccc(cc2)Cl)O SPB04386 CSC(=N)NCc1ccco1.I SJC00409 c1ccc(c(c1)c2/c(=N/c3cc(cc(c3)Cl)Cl)/ssn2)Cl KM09244 Cc1c(c(ccn1)O)OCc2ccc(cc2Cl)Cl RF01757 c1cc(ncc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F SP01055 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)Cl SP01059 COC(=O)C1=C(CCS1)N GK02761 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F SP01080 c1cc(sc1c2cc(on2)C(F)(F)F)S(=O)(=O)N3CCC(CC3)O SP01082 c1ccc2c(c1)nc3c4cc(ccc4n(c3n2)C(=O)C5CCCCC5)F RH01990 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)CC(=O)NNC(=O)c2cccc(c2)Cl CD03714 c1ccc(cc1)N/N=C\2/CCCNC2=O RH01832 c1ccc(cc1)NCc2cccc3c2cccc3 RH01833 c1ccc(cc1)NC(=O)c2cccc3c2cccc3 RH01840 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06538 Cc1cc(c(cc1C)/N=C\c2cc(cc(c2OS(=O)(=O)c3ccc(cc3)F)Cl)Cl)C SJC00195 c1ccc(cc1)CN2c3ccccc3OCC2=O RJC03964 c1ccc2c(c1)N(C(=O)CO2)C(=O)c3ccc(cc3)Cl RJC03966 Cc1c(c(ccn1)O)OCc2ccc(cc2)Cl RF01787 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/Nc3c(cccc3Cl)Cl RF01915 COc1ccc(c(c1)C(=O)NC(=S)Nc2ccc(cc2)F)Br RDR02330 c1cc(c(cc1Br)C(F)(F)F)/C=C/C#N CD05663 CC([C@@H](C(=O)O)NC(=O)OC(C)(C)C)O RJC04002 Cc1c2c(cnn(c2=O)C)c(n1c3ccc(cc3)[N+](=O)[O-])c4ccccc4 SP01107 c1cc(ccc1SCC(=O)c2ccc3c(c2)OCCO3)Cl SPB08268 CC(C)(C)OC(=O)NC1CCNCC1 SPB07957 CS(=O)(=O)C(c1cc(cc(c1)C(F)(F)F)C(F)(F)F)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05923 COc1cccc(c1)c2nnc(o2)c3ccccc3NC(=O)c4ccc(cc4)F RH02149 CC(C)(C)C(=O)NC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F RF01488 Cc1ccc(cc1)C(=O)N2CCN(CC2)CC(=O)Nc3cc(sc3C(=O)C)c4ccc(cc4)F GK03727 c1ccc(cc1)c2cc(c(s2)C(=O)N)NC(=O)c3ccc(cc3)Cl GK03730 COc1ccccc1N2CCN(CC2)CCCCNC(=O)c3ccco3 SEW06462 Cn1cc(cc1C(=O)OC)/C=N/NC(=O)N SEW06460 Cc1ccc2c(c1)nc([nH]2)SCC(=O)NC3Cc4ccccc4C3 KM10556 c1ccc(cc1)CN2C(SCC2=O)c3cn(nc3c4ccc(cc4)Cl)c5ccccc5 RJC04007 CC(C)C(C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 RJC04008 c1cc(sc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4nccs4 KM10529 COc1cccc(c1)Oc2ccc(cc2C(=O)NN)OC SEW06282 Cc1cccc(c1)c2nc(no2)c3ccc(nc3)N4CCN(CC4)c5ccc(cn5)C(F)(F)F SEW06280 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCCC(=O)O PD00782 Cc1ccc(cc1)C(=O)CSc2nnc(o2)c3cc(nn3Cc4cccc(c4)C)C(C)(C)C SPB08341 Cc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)OC RH01924 Cc1cc(c(cc1C)/N=C\c2cc(cc(c2OC(=O)c3cc(c(c(c3)OC)OC)OC)Cl)Cl)C SJC00212 Cc1ccc(cc1)C(=O)Nc2cccnc2Sc3ccc(cc3)C RH02056 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccccc3OC(F)(F)F SP01075 c1ccc(cc1)CNS(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F SP01078 CCOC(=O)c1c(c(sc1NC(=O)c2cccs2)C)c3ccccc3 AW00968 c1cc(ccc1CNC2CCS(=O)(=O)C2)C(=O)O RJC04004 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)[N+](=O)[O-] GK03356 CC(C)Nc1c2cc(c(cc2ncn1)OC)OC GK03354 Cn1c(ccn1)NC(=O)c2ccccc2Cl GK03345 CCC(CO)NC(=S)Nc1c(cccc1C)C RDR00432 Cc1cc(ccc1NC(=S)N/N=C/c2ccc(cc2)N(C)C)Cl RDR00449 Cc1cc(n(n1)c2ccc(cc2)[N+](=O)[O-])C SEW04162 COc1cc(cc(c1OC)OC)CCc2nnc(o2)c3cccs3 SEW04160 c1cc(c(c(c1)Cl)Cl)SCc2nc(on2)COc3ccc(cc3Cl)Cl SP01266 c1ccc2c(c1)c(=O)sc(n2)NC(=O)c3ccco3 HTS01333 COc1cc2c(cc1OC)nc(sc2=O)NC(=O)c3ccco3 HTS01334 c1cc(oc1)C(=O)Nc2nc3c(cc(cc3Br)Br)c(=O)s2 HTS01335 COc1cc2c(cc1OC)nc(sc2=O)NC(=O)c3ccccc3 HTS01337 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl GK03426 Cc1ccsc1/C=C/c2ccnc(n2)Sc3c(cccn3)[N+](=O)[O-] MWP00699 CC(C)(C)c1cc(c(s1)C#N)/N=C/c2ccc(cc2)O GK02527 c1cc(c(c(c1)Cl)NC=C(C#N)C#N)F CD05981 Cc1ccc(cc1)S(=O)(=O)c2c(scn2)Sc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] DFP00110 c1ccc2c(c1)C3(C(=O)N2CCC#N)OCCO3 RH01855 Cc1c(sc(n1)c2ccccc2)C(=O)C SEW04061 c1cc(cc(c1)Cl)N2CCN(CC2)CCCn3cnc4c(c3=O)cccn4 RJC03951 c1cc(cnc1)CNC(=O)c2ccc(cc2)[N+](=O)[O-] RF00014 C1CCOC(C1)OCCCCSc2nnc(s2)N RH02167 CN(C)CCNc1c2c(csc2ncn1)c3ccccc3 AW00973 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCN(CC4)Cc5ccc(cc5)F AW00971 c1ccc2c(c1)CC(C2)NC(=O)CSc3nnc(s3)SCC(=O)NC4Cc5ccccc5C4 KM10557 c1cc(oc1)CNC(=O)/C=C/c2ccc(cc2)OC(F)(F)F SEW06458 c1cc(ccc1C(=O)COC(=O)CCC(=O)OCC(=O)c2ccc(cc2)C(F)(F)F)C(F)(F)F RF03433 c1ccc2cc(ccc2c1)c3csc(n3)N RDR01057 CC(C)(C)NC(=S)N/N=C/c1ccc(cc1)O RDR01063 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2ccc(c(c2)C)Br RDR01073 COc1cccc(c1)NC(=O)c2cnccc2C(F)(F)F RF04000 CCNC(=S)Nc1ccc(cc1)C(C)(C)C GK03643 c1ccc(c(c1)C(=O)NC(=O)C(=O)Nc2cc(cc(c2)Cl)Cl)Cl RF03990 CC(=O)c1coc2ccccc2c1=O SEW04752 c1cc(cc(c1)NC(=O)c2cccnc2)C(F)(F)F SPB08384 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCOCC3 KM10691 Cc1nc(cn1CC(c2ccc(cc2)F)O)[N+](=O)[O-] HTS00996 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3n4cccc4)[N+](=O)[O-] HTS00999 COc1ccc(cc1)C(=C2C=CC(=NO)C=C2)C#N S09951 c1ccc(cc1)C(=O)Nc2cc(cc(c2)Cl)Cl SPB08365 c1ccc(c(c1)NC(=O)c2cccnc2)F SPB08367 CCOC(=O)c1c2c(sc1NC(=O)CSCC(=O)O)CCCC2 GK03286 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)CNc4cc(cc(c4)C(F)(F)F)C(F)(F)F PD00571 Cc1ccc(c(c1)C)c2csc(n2)c3cnccn3 SEW06372 c1ccc(cc1)Cn2ccnc2 KM08030 CC(=O)c1c(cc(s1)c2ccc(cc2)F)NS(=O)(=O)c3ccc(cc3)Cl GK03714 COc1ccc(cc1OC)Cc2nnc(n2c3ccc(cc3)F)SCc4c(cccc4Cl)F PD00784 CCc1c(nc2ccccc2n1)N3CCN(CC3)C(=O)c4cccs4 GK03647 CCc1c(nc2ccccc2n1)N3CCN(CC3)C(=O)c4cc(cc(c4)Cl)Cl GK03648 c1cc(ccc1[N+](=O)[O-])OCC(CN2CCOCC2)O AW00890 Cc1cc(cc(c1Cl)C)OCC#N SPB02453 Cn1c(c(cn1)C(=O)Sc2ccc(cc2)Cl)n3cccc3 GK03651 Cc1ccccc1CS/C(=C/N(C)C)/C(=O)C SPB04575 c1cc(ccc1c2nc(nc(n2)O)c3ccc(cc3)Cl)Cl RF01842 c1ccc2cc(ccc2c1)c3cc([nH]n3)C(F)(F)F SP01371 Cc1c2cc(ccc2sc1C3=NOC(C3)(C(F)(F)F)O)Cl SP01381 c1cc(ccc1/C=C/C(=O)Oc2ccc(cc2)Cl)OC(F)(F)F SEW06456 CC(C)(C)OC(=O)NCC(=O)NNC(=S)NC1CC1 KM10563 c1cc(c(cc1Cl)NC(=S)NCc2ccncc2)Cl RDR00573 c1ccnc(c1)CCNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl GK01737 Cn1c2c(cc(s2)C(=O)Nc3ccc(cc3)F)c(n1)C(F)(F)F GK02659 Cc1csc2c1ncnc2N3CCN(CC3)C(=O)Nc4ccccc4 GK02682 CCOC(=O)/C(=C/Nc1cc(ccc1C)F)/C#N RH02230 COc1ccccc1C(=O)Nc2cccc(c2)C(F)(F)F SPB08385 c1c(cc(cc1C(F)(F)F)N)Cc2cc(cc(c2)N)C(F)(F)F CD03495 c1ccc2c(c1)ccc-3c2C(=O)c4c3cccc4 RJC03891 c1ccc2cc3c(ccs3)cc2c1 RJC03900 c1ccc2c(c1)c(cs2)CCOC(=O)c3ccc(cc3)C(F)(F)F S11586 Cc1ccc(cc1)N2C(=O)CC(C2=O)N3CCCCC3 S12350 CCOC(=O)c1ccc2c(c1)CC/C(=C\c3cccc(c3)C(F)(F)F)/C2=O SEW03711 Cc1ccc(cc1)NC(=O)CSCc2ccc(cc2)C#N CD01696 CCc1c(nc2ccccc2n1)N3CCN(CC3)C(=O)C(C)(C)C GK03501 Cc1cc(nc2n1nc(c2Cl)C(C)(C)C)C(F)(F)F KM06937 CC(C)(C)c1ccc(cc1)/C=N/NC(=O)CSC2CN(C2)C(c3ccccc3)c4ccccc4 KM09582 Cc1c(cc(n1CCCN2CCOCC2)c3ccccc3)C(=O)Nc4ccccc4 SP00944 c1cc(ncc1C(F)(F)F)N2CCN(CC2)CC#N SEW06589 c1ccc2c(c1)c(cc(n2)C(F)(F)F)Sc3cc(nc4c3cccc4)C(F)(F)F KM10483 CN(C)CC#Cc1cc(cnc1)C#N KM08401 C/S(=N\S(=O)(=O)c1cccc2c1nsn2)/c3c(cccn3)C(F)(F)F KM08403 CN(C)c1ccc(cc1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05894 c1cc(c(cc1C(F)(F)F)Cl)C(=S)N SEW01578 c1ccc(cc1)NC(=O)c2ccccc2C(=O)O RH01849 c1ccc(cc1)COC(=O)NC(CC(=O)N)C(=O)O KM08968 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)Nc2ccc(cc2)OC(F)(F)F AW01056 Cc1c2c(c(c(nc2n(n1)c3ccccc3)N)C#N)c4ccc(cc4)C(C)(C)C HTS00839 COc1ccc2c(c1)cc([nH]2)C(=O)N(Cc3ccccn3)Cc4ccccn4 HTS00777 c1ccc(c(c1)C(=O)Nc2ccc(cc2)C(=O)N)C(=O)O HTS00749 c1ccc(c(c1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4C(F)(F)F)F KM09743 CCNC(=O)Cc1c2ccccc2sc1Cl KM07287 CCC(=O)Nc1c2c(cccc2F)n(n1)C SP01357 Cc1ccc(cc1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3)C(=O)O KM10009 CC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)Cl GK03720 Cc1c(ccc(n1)C(F)(F)F)NC(=O)NCCNc2nccc(n2)C(F)(F)F AW00898 c1c(cc(cc1C(F)(F)F)N2C(=O)C=CC2=O)C(F)(F)F S04394 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccc(cc2)O)C RJC04089 CC(C)Sc1ccc(cc1[N+](=O)[O-])C#N KM10491 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCc4c(c5cc(ccc5[nH]4)F)C3 SP01077 Cc1c(cc(o1)C(C)(C)C)c2c(c(n(n2)c3ccc(cc3)F)SC)C#N SP01081 CCOC(=O)NN(c1c(c(c(c(c1C)C)C)C)C)C(=O)OCC CD08006 Cc1c(c(n(n1)C(C)(C)C)C)/C=N/O CD07395 Cc1ccc(cc1Cl)NC(=O)/C=C/C(=O)Nc2ccc(c(c2)Cl)C CD07695 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)Nc3ccc(cc3)OC(F)(F)F SP00688 Cc1c(cc(n1CCCN2CCOCC2)c3ccccc3)C(=O)Nc4cccc(c4)C(F)(F)F SP00692 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3cccc4c3cccc4 RH02068 Cc1ccc(cc1C)C(=O)Nc2cccnc2Oc3ccc(cc3)C(C)(C)C RH02069 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccccc3F RH02070 Cc1c(c(c([nH]1)C)C(=O)OC)/C=N/OC(=O)c2ccccc2 SP00957 CCOC(=O)c1cc2ccccc2[nH]1 RH01865 Cc1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc(cc4)Cl KM10486 CCOC(=O)CC(c1cc(c(c(c1)OC)OC)OC)Sc2ccccc2N PD00711 c1ccc2c(c1)c3c(n(c2=O)CC4CC4)-c5ccccc5C3=O PD00715 Cc1ccc(cc1)c2csc3c2c(ncn3)N4CCCC4 AW01140 CC(C)Cc1ccc(cc1)C(=O)C(C)N2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS01195 COc1ccc(cc1)c2ccnc(n2)SCC(=O)N3CCN(CC3)c4ccccc4 HTS01202 CC(C)(C)c1cc2nc(cc(n2n1)C(F)(F)F)c3ccc4c(c3)OCO4 KM10523 c1cc(sc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5c(c4)OCO5 KM10525 Cc1ccc(cc1)c2nnc(o2)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-] GK03610 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCC(CC3)C(=O)OCC KM10692 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCCCC3 KM10693 c1ccc(cc1)NC(=O)c2cccc(c2)Cl SPB08369 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccc(cc2)OC)C RJC04095 c1ccc(cc1)n2c(nnn2)SCC(=O)NC3Cc4ccccc4C3 KM10554 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)c3cccc4c3cccc4 RH02061 CCCCCCN1C(C(c2ccccc2C1=O)C(=O)O)c3c(cccc3Cl)F PD00708 COCCOc1ccccc1NC(=O)c2ccc(cc2)Cl CD05897 Cc1c(nc(s1)NC(=O)c2ccc(cc2)C(F)(F)F)c3ccc(cc3)CC(C)C HTS01182 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2C(=O)O)OC)OC GK03477 COc1cc2c(cc1OC)ncnc2Nc3ccccc3 GK03498 CCOC(=O)c1ccc(cc1)NC(=S)NC GK03278 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCCC3 SP01089 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)NC3CCN(CC3)Cc4ccccc4 SP01093 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)NCc3ccccc3 SP01095 c1cc(sc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5c(c4)CCC5 KM10541 COc1cccc(c1)NC(=O)c2ccccc2 SPB08379 c1cc(ccc1c2nc(cs2)C34CC5CC(C3)CC(C5)C4)OC(F)(F)F SPB08334 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)Nc3ccc4c(c3)OCCO4 SP00908 Cc1c(cc(n1CCCN2CCOCC2)c3ccccc3)NC(=O)c4ccc(cc4)Cl SP00924 Cc1cc(no1)c2nc(cs2)C34CC5CC(C3)CC(C5)C4 SPB08335 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C RH02151 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)/C=C/N(C)C RH02152 Cc1c(c2c(cn1)COC(OC2)C(C)C)O RJC03962 c1ccc2c(c1)c(c[nH]2)CCNC(=O)c3cccnc3 RJC03963 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCC(CC3)C(=O)O KM10700 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)Cc4ccccc4 KM10702 c1cc(ccc1F)SCC(CN2CCC(CC2)C(=O)N)O HTS00956 c1cnc(c(n1)C(=O)N2CCC(CC2)O)C(=O)O HTS01105 c1ccc2c(c1)CC(C2)NC(=O)CSc3nc4ccccc4o3 KM10555 CC(C)(C)c1cc2c(s1)c(ncn2)N3CCCCC3 GK03616 CC(C)(C)c1cc2c(s1)c(ncn2)N3CCSCC3 GK03617 c1ccc(cc1)c2csc3c2c(ncn3)NC4CCCCC4 AW01082 CC(C)Nc1c2c(csc2ncn1)c3ccccc3 AW01083 CC(=O)Nc1cccc(c1)OCCCNc2c3c(csc3ncn2)c4ccccc4 AW01084 COc1ccc(cc1OC)CCNC(=S)Nc2ccc(cc2)F S12453 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])OCCO CD08081 Cc1ccc(cc1)C(=O)CSc2[nH]c(=O)c3ccccc3n2 PD00038 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)N3CCCC3 SP00874 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)c3cccs3 RH02064 CCOC(=O)c1cc(oc1/C=N/OC(=O)c2ccccc2)c3ccc(cc3)Cl SP00951 c1cc2cc([nH]c2c(c1)[N+](=O)[O-])C(=O)Nc3ccc(cc3)Cl SP00945 CCCCCc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3cc(cc(c3)F)F RH02067 COc1ccc(cc1)c2cc(n3c(n2)cc(n3)c4ccc(cc4)Cl)C(F)(F)F KM10485 COc1cc2c(cc1OC)ncnc2Nc3cccc(c3)Cl GK03499 COc1cc2c(cc1OC)ncnc2Nc3ccc(c(c3)F)F GK03500 Cc1cc(cc(c1OCC(CN2CCC(CC2)C(=O)N)O)Br)Cl HTS00951 c1cc(c(cc1I)F)N2C(=O)CC3(CCCCC3)CC2=O PD00717 c1ccc2c(c1)CC(C2)NC(=O)CSc3cccs3 KM10561 COc1ccc(cc1OC)c2cc(n3c(n2)cc(n3)c4ccc(cc4)Cl)C(F)(F)F KM10544 CC(=CC(=O)NCCSCc1ccc(cc1)Cl)C SEW06363 c1ccc2c(c1)cccc2C(=O)NN JFD03929 CC1=NN(C(=O)C1[N+](=O)[O-])c2ccc(cc2)[N+](=O)[O-] JFD03931 c1cc(sc1)c2nc(sn2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl SPB08327 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Oc3cccc(c3)C(F)(F)F)C SPB08332 CC(C)c1ccc(cc1)n2c(=O)c3ccccc3cn2 PD00570 COc1cc(cc(c1OC)OC)C(=O)Oc2c(cc(cc2Cl)Cl)/C=N\c3cc(c(cc3OC)Cl)OC SJC00207 c1cc(ccc1CC(=O)O)Br TL00410 c1cc(c(cc1Cl)Cl)OCc2nc(no2)CSc3ccc(cn3)C(F)(F)F SP01273 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(nc3)OC SPB08387 c1ccc2c(c1)ccc(c2/N=N/c3ccccn3)O JFD03913 c1ccc2c(c1)C(C(N(C2=O)Cc3ccc(cc3)F)c4cccnc4)C(=O)O PD00719 c1ccc(cc1)CCn2c(=O)c3ccccc3cn2 PD00598 CC(=O)c1ccc(c(c1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)Cl SJC00125 CC(C)c1ccc(cc1)S(=O)(=O)Nc2cc(ccc2Cl)C(=O)C SJC00144 CCc1cccc(c1Nc2nc3ccc(cc3s2)C(C)C)CC RDR00125 CCc1cccc(c1Nc2nc3c(cc(c(c3s2)Cl)Cl)Cl)CC RDR00127 CSC1=C(C(=O)NC(S1)c2ccc3c(c2)OCO3)C#N CD04077 Cc1c(c(c(cn1)CSc2ccccc2/N=C/c3cc(cc(c3O)Cl)Cl)CO)O CD04097 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)Nc3ccc(cc3)c4ccccc4 SP00907 CN1C(=O)[C@@H](NC1=S)Cc2ccc(cc2)[N+](=O)[O-] KM10701 Cn1c(nnc1SCc2ccccc2)CNC(=O)c3ccccc3 KM10703 CN(C)CCNC(=O)COc1cc(nc2c1cccc2)c3ccccc3 RH02062 c1ccc2c(c1)CC(C2)NC(=O)C3CCC3 KM10489 c1cc(ccc1/C=C/C(=O)N2CCOCC2)OC(F)(F)F SP01235 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00826 CC1CC(CN(C1)c2ccc(cc2C(=O)O)N)C CD06942 c1cc(cc(c1)Cl)C(=O)NNC(=O)c2cccc(c2)Cl SJC00152 CCc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)OC RH01925 Cc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)C(C)(C)C RH01923 c1cc(c(nc1)Oc2ccc(cc2)Cl)N RH01922 CN(CCC#N)c1ccc(cc1)c2c(c(nc(c2C#N)OC)N)C#N RDR00291 CCCc1ccc(cc1)C(=O)Nc2cccnc2Sc3ccc(cc3)C RH02057 CSc1nn(c(=S)s1)CO SPB03207 COc1ccc(cn1)NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F SPB08389 Cc1ccc(cc1)SC(=O)c2cnn(c2n3cccc3)C GK03650 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F SP01084 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] RF01916 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccco3 RH01985 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=O)/C=C/C(=O)O CD02030 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Oc3ccc(cc3)NC(=O)C)C SPB08333 c1ccc2c(c1)c3c(n(c2=O)Cc4ccc(cc4)F)-c5ccccc5C3=O PD00709 COc1cc(cc(c1OC)OC)/C=C/C(=O)NCc2ccc3c(c2)OCO3 PD00712 c1ccc(cc1)OCCN2CCCN(CC2)C(=O)Nc3ccc4ccccc4c3 TB00015 c1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl RH02038 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)Nc3ccc(cc3)Cl SP00928 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)CSc3ccc(cc3)Cl GK03446 c1ccc2c(c1)NC(S2)c3ccc4c(c3)OCO4 SJC00336 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CNc3ccc(cc3)F)O RJC03968 c1ccc(cc1)c2ccc(cc2)c3nc4ccc(cc4o3)c5ccccc5 JFD03903 c1cc2ccc3cccnc3c2nc1.Cl JFD03909 C[C@]12CCC(C1)C(C2NS(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F)(C)C SP01079 CC(=O)N(c1ccccc1)/N=C/c2cc(n(n2)c3ccccc3)COC(=O)C RH01906 c1ccc(cc1)Cn2cc(c3c2ccc(c3)[N+](=O)[O-])/C=C/C#N RH01902 CCOC(=O)c1ccc(cc1)NC(=O)CC(C)(C)CC(=O)O PD00572 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3cccc(n3)C KM11018 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)CSCC(=O)O HTS01106 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NC(=O)CSCC(=O)O HTS01107 c1cc2c(cc1C(=O)N3CCOCC3)nns2 KM10653 Cc1ccc(cc1)c2nnn(n2)CC(=O)NNC(=O)N3CCOCC3 GK03461 Cc1cc(c2c(c1)cc([nH]2)C(=O)NCc3ccccc3)C KM11022 c1ccc2c(c1)ccn2CC(CN3CCC(CC3)NC4CCCCC4O)O AW00957 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CN4C(=O)c5ccccc5C4=O HTS00733 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)CC(C)(C)CC(=O)O HTS00491 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)NCCNc3c(cccn3)C(F)(F)F HTS00437 CCN(CC)c1ccc2cc(c(=O)oc2c1)C(=O)O RH02173 Cc1cc(c2ccccc2n1)N3CCN(CC3)CC(=O)c4ccc(cc4)OC RH02163 Cc1c(c([nH]c(=O)c1C#N)C)CC=C RH02164 c1cc(cnc1)c2cc(c(c(n2)O)C#N)C(F)(F)F RH02165 Cn1c(c(cn1)C(=O)NCC=C)n2cccc2 GK03655 c1ccc(cc1)C(=O)c2cccc3c2NCC3 SEW06375 c1cc(ccc1c2csc(n2)c3cnccn3)[N+](=O)[O-] SEW06377 c1ccc(cc1)CCNC(=O)c2ccc3c(c2)nns3 KM10651 c1cc2c(cc1C(=O)NCc3ccncc3)nns2 KM10652 COc1ccc(cc1)Oc2c(cccn2)NS(=O)(=O)c3ccc(c(c3)F)F RH01991 COc1ccc(cc1)Oc2c(cccn2)NS(=O)(=O)c3ccc(cc3)OC RH01992 Cn1c(ccn1)NS(=O)(=O)c2ccccc2 GK03355 Cc1cc(ccc1F)NC(=O)c2cc3cccc(c3[nH]2)[N+](=O)[O-] KM11027 CN(C)c1ccc(cc1)/C=N/NS(=O)(=O)c2ccc(cc2)Cl RDR00582 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)F GK03347 CC(C)n1c2ccccc2nc1S SPB02552 CCn1c(cc(n1)C)c2nnc(n2c3ccc(cc3)Cl)S SPB02501 COc1cc(cc(c1OC)OC)C(CC(=O)N2CCC(CC2)n3cccc3)CC(=O)O HTS00581 CCCCCc1ccc(cc1)S(=O)(=O)N2CCC(CC2)n3cccc3 HTS00591 c1ccn(c1)C2CCN(CC2)S(=O)(=O)c3cccc4c3non4 HTS00594 CCCCNC(=O)c1cc2cccc(c2[nH]1)[N+](=O)[O-] KM11025 c1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)SCC(COc3ccc(cn3)C(F)(F)F)O HAN00269 c1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)SCc3nc(on3)c4cccs4 SEW06389 Cc1ccc(cc1)C(=O)Nc2ccccc2SCc3nc(on3)c4cccs4 SEW06390 c1ccc2c(c1)ccn2CC(CSc3ccccc3NC(=O)c4ccc(cc4)Cl)O HAN00324 c1ccc2cc(ccc2c1)c3csc4c3c(ncn4)N5CCC(CC5)O HTS00420 c1ccc(cc1)c2nc(sn2)N3CCCN(CC3)C(=O)c4ccc(cc4)F HTS01147 c1ccc(cc1)CSc2ccc(cc2C#N)N RH02174 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2ccnn2C GK03349 c1cc(sc1)C(=O)N2CCCN(CC2)CC(COc3ccc(c(c3)Cl)Cl)O.Cl AW00362 c1ccc(cc1)CNC(=O)c2cc3cccc(c3[nH]2)[N+](=O)[O-] KM11020 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)CC4(CCCC4)CC(=O)O HTS00568 c1cc(ccc1OCC(CNCc2ccc3c(c2)OCO3)O)F HTS00692 c1ccc(cc1)CCNC(=O)c2cc3cccc(c3[nH]2)[N+](=O)[O-] KM11024 c1cc2cc([nH]c2c(c1)[N+](=O)[O-])C(=O)Nc3ccc4c(c3)OCO4 KM11028 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)Nc3cccc(c3C)Cl)C SEW06397 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)Nc3ccc(cc3)Cl)C SEW06398 CCOC(=O)c1c(noc1c2ccc(o2)Br)C JM00027 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)Nc2ccccc2OC AW01054 CCc1cccc(c1NC(=O)N2CCN(CC2)C(=O)OC(C)(C)C)C AW01055 CCOC(=O)c1c(n[nH]c1N/N=C/c2cccc(c2)Cl)C RJC04087 Cc1nc(cs1)c2nnc(n2C)SCc3nc(no3)c4ccc(cc4)C5SCCS5 HTS00221 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F HTS00228 Cc1cc(c2cc([nH]c2c1)C(=O)NCCc3ccccc3)C KM11026 Cc1nc(c(c(n1)O)[N+](=O)[O-])O RH02113 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(n3C4CCCCC4)SCC(=O)O SPB08186 c1ccc(cc1)c2c(oc(n2)CCC(=O)O)c3ccccc3 SS00042 CCOC(=O)CSc1nnc(n1C2CCCCC2)c3cc(nn3Cc4cccc(c4)C)C(C)(C)C SPB08185 CC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccccc3 GK03718 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)C)c3ccccc3 GK03719 c1cc(c(c(c1)Cl)CSCC(=O)c2ccc3c(c2)OCCO3)F SPB08269 c1cc2c(cc1C(=O)CSc3ccc(cn3)C(F)(F)F)OCCO2 SPB08274 CNC(=O)Nc1cccc(c1)c2cc(no2)c3c(cccc3Cl)Cl RF01983 CC(=O)Nc1cccc(c1)c2cc(no2)c3ccc(cc3Cl)Cl RF01994 CC(C)(C)OC(=O)NCc1nnc(n1CC=C)S KM10567 c1ccc2c(c1)C(=O)C(=Cc3ccc(s3)[N+](=O)[O-])C2=O PD00675 CC1=C(CC(C(C1)C(=O)Nc2ccc3c(c2)OCO3)C(=O)O)C PD00676 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2Cc4ccco4)C(=O)O PD00677 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)Nc3ccc(cc3)C(F)(F)F)C SEW06399 c1ccc2c(c1)C(=O)CCS2(=O)=O CD03987 Cc1cc(nc2c1ccc(=O)n2CC(=O)N/N=C/c3ccccc3Cl)C KM10860 CN(C)/C=C/C(=O)c1ccc(c(c1)Cl)Cl CD08596 COc1ccc(cc1)COc2cccnc2N RH02040 c1ccc2c(c1)nnn2CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS00730 c1ccc(c(c1)C(=O)N)NC(=O)c2c(nccn2)C(=O)O HTS00748 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)NCc3ccco3 SP00550 CCOC(=O)c1cc2c(nn(c2s1)C)C(F)(F)F GK02729 COC(=O)C1=C(CC(S1)c2ccccc2)N GK02762 CCOC(=O)NC(=S)N1CCOCC1 NH00193 c1cc(ccc1OC(F)(F)F)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl HTS01443 CC1CN(CC(O1)C)c2c3c(csc3ncn2)c4ccccc4 AW01100 c1cc(oc1)CNC(=S)N/N=C/c2ccc(c(c2)Cl)Cl RDR01356 Cc1c(cc(n1c2ccc(cc2)SC)c3ccccc3)C(=O)O SP01451 CC(=O)c1c(cc(s1)c2ccc(cc2)C(C)(C)C)N GK03407 c1ccc2c(c1)C(=O)N(C2=O)CCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F RH01946 CSc1nnc(n1CC=C)c2ccc3c(c2)cccn3 KM10642 CC(=O)CSc1nnc(n1CC=C)c2ccc3c(c2)cccn3 KM10645 Cn1c2c(cn1)c(ncn2)Sc3ccc(cc3)Cl GK03448 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=O)C(F)(F)F SEW06570 CCOC(=O)c1c(c(c(=O)n(n1)c2ccc(cc2)OC)C#N)C JFD03716 c1ccc(cc1)NC(=O)/C=C/C(=O)O S14473 Cc1ccc(cc1)S(=O)(=O)N/N=C(\C)/c2ccc(cc2)OC(=O)c3ccc(o3)Br JFD03979 CC(C)(C)c1ccc(cc1)c2nnc(o2)SC SPB08276 c1cc(ccc1NC(=S)NCC(=O)O)F RDR00799 CC(c1ccccc1)NC(=S)N/N=C/c2ccccc2O RDR00803 Cc1cc(c(c(c1)C)NC(=S)NC(=O)C(C)Oc2ccc(cc2)C(C)(C)C)C RDR02298 c1cc2c(cc1NC(=O)COCC(=O)O)OCCCO2 HTS00133 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCC3=CCCCC3 PD00789 Cc1ccc(cc1)C(=O)NN(C)c2ccc(cn2)[N+](=O)[O-] SP01284 CC1=C(CC2C(C1)C(=O)N(C2=O)C(Cc3ccccc3)C(=O)O)C PD00577 Cc1ccccc1NC(=O)c2cc(n(c2C)CCCN3CCOCC3)c4ccccc4 SP00700 c1cc(oc1)C(=O)NCCSCc2ccc(cc2)Cl SEW06366 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NN SPB03911 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)C(=O)O SPB08113 Cc1c(sc(n1)c2cnccn2)C(=O)C SEW06370 COC(=O)c1ccccc1NC(=O)CC2C(=O)NCCN2 HTS00378 Cc1ccc(cc1C)OCC(CNC2Cc3ccccc3C2)O HTS00966 COc1ccc(cc1OC)c2cn[nH]c2N JFD03989 Cn1c(nnn1)SCC(=O)NC2Cc3ccccc3C2 KM10549 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)c4cccc(c4)C(F)(F)F SPB08278 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)c4cnccc4C(F)(F)F SPB08283 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)c4c5c(csc5ncn4)c6ccccc6 AW01109 Cc1ccc(cc1)Sc2c(nc3n2cccn3)c4ccccc4 RJC04097 c1ccc(cc1)/C=C(\C#N)/c2[nH]c3ccccc3n2 PHG00718 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)NS(=O)(=O)c3ccc(cc3)C)C SEW06395 CCCCCCCCC1CCCC1N.Cl RJC04000 c1c2c(nc3c1CCCC3)CCCC2 JFD03985 COc1ccc(c(c1)NC(=O)C(=O)NCCc2ccccn2)OC JPV00089 COc1c(csc1Cl)C(=O)Nc2cc(c(cc2Cl)Cl)Cl KM00468 c1ccc(cc1)CN2CCC(CC2)NC(=O)C3CCN(CC3)c4nccc(n4)C(F)(F)F AW01262 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)Cc4ccc(cc4Cl)Cl SPB08285 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)CCn4c5ccccc5oc4=O SPB08286 Cc1c2cnn(c(=O)c2c(n1c3ccccc3)C)C SP01109 Cc1c2cnn(c(=O)c2c(n1Cc3cccs3)C)C SP01110 Cc1ccc(c(c1)[N+](=O)[O-])NN=C(C(=O)C)C(=O)C RH01930 c1ccc2c(c1)Nc3cc(ccc3S2)C(F)(F)F JFD03930 c1ccc(cc1)/N=c\2/[n-]n(c[n+]2c3ccccc3)c4ccccc4 JFD03932 c1cc2c(cc1Br)CC(C(=O)O2)C(=O)N3CCCCC3 RH01913 Cn1c(ccn1)NC(=O)Nc2cccc(c2)[N+](=O)[O-] GK03282 Cc1ccc(c(c1)C)NC(=S)N2CCC(CC2)Nc3nccc(n3)C(F)(F)F AW00877 CC(C(=O)Nc1c(cccc1F)F)Sc2nccn2c3cccc(c3Cl)Cl AW00904 COCCCNC(=S)NNC(=O)c1ccc(cc1)C(F)(F)F SPB01422 Cc1ccc2c(c1)cc([nH]2)C(=O)O JFD03921 CC[C@H]1[C@H](COC1=O)Cc2cncn2C.Cl JFD03923 Cc1nc(nc(n1)SC)N/C=C(\C#N)/S(=O)(=O)c2ccccc2 KM01107 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2ccc(o2)Oc3cccnc3 AW01257 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)c4ccc(cc4)C(F)(F)F SPB08288 COc1ccccc1OCc2nc(cs2)c3ccccc3 SPB08289 COc1ccc2c(c1)cc([nH]2)C(=O)Nc3nc4ccccc4s3 SP01205 Cc1cc(c2cc([nH]c2c1)C(=O)NCc3cc(ccc3Cl)Cl)C SP01177 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NNC(=O)Nc3cccc4c3cccc4 SPB08176 Cc1cc2c(cc1C)nc3c(n2)c4cc(ccc4[nH]3)F RH01951 c1ccc(c(c1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)Cl)Cl PHG00619 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)c3cccc(c3)Cl PHG00638 c1cc(cc(c1)[N+](=O)[O-])C2=N/C(=C/c3ccc(cc3)Cl)/C(=O)O2 PHG00681 c1ccc(cc1)CSc2c(ccc(n2)/C=N/c3ccc(cc3Cl)Cl)C#N SPB04382 c1ccc2c(c1)[nH]c(n2)c3cc4cc(cc(c4oc3=O)Cl)Cl PHG00770 CCCCNC(=O)NNC(=O)c1cc(nn1Cc2ccc(cc2)F)C(C)(C)C SPB08175 Cc1c(csc1C(=O)NCc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM01482 Cc1c(csc1C(=O)OCC=C)S(=O)(=O)c2ccc(cc2)Cl KM01513 c1cc(oc1)CNC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F AW01260 c1cnc(nc1C(F)(F)F)N2CCC(CC2)C(=O)N3CCSCC3 AW01258 Cc1cc(c2cc([nH]c2c1)C(=O)NC3CCCCC3)C KM11064 COc1ccc2c(c1)cc([nH]2)C(=O)NCc3cc(ccc3Cl)Cl SP01196 CC(=O)Oc1c(cc(cc1I)C(=O)OC)I RF04603 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2ccc(cc2)Cl)C)c3ccccc3)C SP01111 c1ccc2c(c1)CC(C2)NC(=O)CSC3=NCCS3 KM10558 c1ccc(cc1)CSCC(=O)NC2Cc3ccccc3C2 KM10545 COc1ccc(cc1)C(=O)NCCSCc2ccc(cc2)Cl SEW06358 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)Nc4ccc(cc4)Cl SP00926 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)Nc4ccccc4 SP00929 Cc1cc(c2ccccc2n1)N3CCN(CC3)CC(=O)N(C)c4ccccc4.Cl RH02147 COC(=O)c1ccccc1CS(=O)(=O)C CD05665 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C2(CC2)O CD05704 Cc1cc(c(c(c1)C)CSCCNC2=CC(=O)CC(C2)c3ccc(cc3)N(C)C)C SEW06603 Cc1cc(c2cc([nH]c2c1)C(=O)Nc3ccc4c(c3)OCO4)C SP01192 CCc1ccc2c(c1)cc([nH]2)C(=O)NCc3cc(ccc3Cl)Cl KM11001 CC(C)C(=O)NCc1ccc(cc1Cl)Cl RF04992 CC1CC(CC(C1)(C)C)NC(=S)N/N=C/c2cc(c(cc2OC)OC)OC PD00576 c1ccc(c(c1)NC(=O)/C=C/C(=O)O)F RJC04025 COc1cc(cc(c1OC)OC)C=C(C(=O)O)C(=O)O RJC04027 CC(=NNC(=S)Nc1ccc(cc1)Cl)C RDR00659 c1cc(sc1)C(=O)Nc2nnc(s2)C(C(C(F)(F)F)(F)F)(F)F SP01387 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)OC SP01349 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)S(=O)(=O)c4cc(cc(c4)Cl)Cl HTS01321 CCCCCCC\1C(CC/C1=N\O)C(=O)OC RJC04022 CCOC(=O)C(=Cc1cc(c(c(c1)OC)OC)OC)C(=O)OCC RJC04026 CCOC(=O)C(=Cc1ccc(cc1)NC(=O)C)C(=O)OCC RJC04028 c1ccc(cc1)/C(=N\O)/Nc2cc(cc(c2)Cl)Cl RF05106 CN(C)c1ccc(cc1)C2CC(=CC(=O)C2)NCCc3ccccn3 SEW06601 CN(C)c1ccc(cc1)C2CC(=CC(=O)C2)NCCSCc3ccc(cc3)F SEW06602 COc1ccc(cc1)C(=O)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS01191 Cc1cc(c2cc([nH]c2c1)C(=O)NCCN3CCOCC3)C KM11004 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)N3CCN(CC3)CCOC(=O)C4CC4 KM10566 c1cc(ccc1C(=O)c2[nH]ccn2)OC(F)(F)F HTS00475 c1cc(sc1c2csc(n2)c3cnccn3)Cl HTS00039 CC(C)n1c2ccc(cc2nc1C(F)(F)F)C(=O)O KM10492 Cc1cccc(c1)NC(=O)N(C)C PD00573 c1cc(ccc1C(=O)N)NC(=O)c2c(nccn2)C(=O)O HTS00750 c1cc(c(cc1F)F)NC(=O)/C=C/C(=O)Nc2ccc(cc2F)F CD07700 C/S(=N\C(=O)c1cccc2c1non2)/c3c(cccn3)C(F)(F)F KM08405 CCOC(=O)CSc1nc2cc(ccc2s1)Cl RH02145 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(o3)SCC(=O)c4ccc(cc4)Cl SPB08340 c1ccc(cc1)CN2CCC(CC2)/N=C\3/c4ccccc4NC3=O PD00567 c1ccc2c(c1)cnn(c2=O)CCO PD00568 c1ccc(cc1)C(=O)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS01188 CC(C(=O)c1ccc(cc1)c2ccccc2F)N3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS01189 COc1cc(cc(c1OC)OC)/C=N/N=C/c2ccccc2O RDR00882 Cc1c2ccccc2sc1C(=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS01198 Cc1c(nc(o1)c2ccccc2)C(=O)Nc3cc(ccc3Oc4ccc(cc4)OC)C(F)(F)F HTS00254 Cc1ccc(cc1)c2csc3c2c(ncn3)N4CCC(CC4)O HTS00419 CCOC(=O)c1ccc(cc1)N2C(=O)CC(CC2=O)(C)C PD00575 Cc1cccc(c1NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl)Cl HTS01150 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)NC(=O)Nc4ccc(cc4F)F)C(F)(F)F SEW06381 c1ccc(c(c1)CSCCNC2=CC(=O)CC(C2)c3ccc4c(c3)OCO4)Cl SEW06592 CN(C)c1ccc(cc1)C2CC(=CC(=O)C2)NCc3cccs3 SEW06600 Cc1cc(cc2c1c(cc(=O)o2)C)O RDR01465 CC(C)(C)c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4cccc(c4)OC GK03739 Cc1c(sc(n1)c2cccnc2)C(=O)N/N=C/c3ccccc3Cl SPB02285 CCCCNc1nc(cs1)c2ccc(cc2)[N+](=O)[O-].Br RDR01304 COc1cc(cc(c1)OC)C(=O)OCC(=O)c2ccccc2 RDR01496 CCCCCc1ccc(cc1)C(=O)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS01192 Cc1ccc(cc1)C(=O)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS01194 CC(C)(C)NC(=S)N/N=C/c1ccc(cc1)N(C)C RDR01152 c1ccc(cc1)C(=O)COC(=O)c2ccc(cc2)I RDR01538 Cc1ccc(cc1C)OCC(CN2CCC(CC2)C(=O)N)O HTS00965 Cc1cc(c(c(c1)C)C(=O)C2CCN(CC2)C(=O)c3ccc(cc3)C(C)(C)C)C SEW06384 Cc1cc(c(c(c1)C)C(=O)C2CCN(CC2)C(=O)c3cccs3)C SEW06385 COc1ccccc1NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl HTS01152 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)Cc2cc(cc(c2)F)F SEW06378 Cc1ccc(cc1NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl)F HTS01154 COc1cc2c(cc1OC)ncnc2Nc3ccc(cc3)OC(F)(F)F GK03504 CCc1c(nc2ccccc2n1)N3CCN(CC3)C(=O)Nc4ccccc4 GK03505 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)/C=N/c3cc(c(cc3OC)Cl)OC SJC00180 Cn1c(nnc1SCC(=O)c2ccc3c(c2)OCCO3)C(F)(F)F SPB08271 CSc1nnc(s1)SCC(=O)c2ccc3c(c2)OCCO3 SPB08272 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)c3ccco3 RH02060 c1ccc(cc1)CNC(=S)NC2CCCCC2 AW01174 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)C(C)(C)C RH02065 Cc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3cc(cc(c3)F)F RH02066 c1ccc2c(c1)C(=O)N(C2=O)CCCN3CCN(CC3)c4nccc(n4)C(F)(F)F AW01204 Cn1c2c(cn1)c(ncn2)NNS(=O)(=O)c3ccccc3 GK03510 c1cc(cc(c1)N)c2nnc(o2)/C=C/c3ccc(cc3)OC(F)(F)F SEW06640 CCCc1cc(nc(n1)SCC(=O)N2CCN(CC2)c3ccccc3)O HTS01205 c1cc(c(cc1OCC(CN2CCC(CC2)C(=O)N)O)Cl)Cl HTS00720 CC[C@H](C)[C@@H](C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 SB00966 CCCCc1ccc(c(c1)C)NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl HTS01157 CCC(=O)Nc1cc(cnc1OC)C(F)(F)F RF05138 CC(=O)N/C(=C/c1ccoc1)/C(=O)O SPB08160 c1cc2cccnc2c(c1)S(=O)(=O)NCC3CCCO3 HTS00640 Cc1c(c(c(o1)C)S(=O)(=O)NCC2CC2)C(=O)OC HTS01164 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)C2=CN3C=C(C=C(C3N2)Cl)C(F)(F)F AW01181 CCOC(=O)Cc1csc(n1)NC(=O)COCC(=O)O PD00808 CCCc1cc(nc(n1)SCc2ccc(cc2)Cl)O JM00414 Cc1c(ccc(n1)C(F)(F)F)NC(=O)C(F)(F)Sc2ccccc2 AW01180 CCOC(=O)Cc1csc(n1)NC(=O)CSCC(=O)O PD00796 CCN(CCC#N)C(=S)Nc1cccc2c1cccc2 SW00150 CCCc1cnc(nc1)N2CCSCC2 AW01190 CS(=O)(=O)NCCNc1cc(nc2c1cccc2)c3ccccc3 RH02047 CCOC(=O)C(C)Oc1ccc(cc1Cl)NC(=O)C(Cl)Cl RDR02169 c1cc(c(c(c1)Cl)CSc2nnnn2c3ccc(cc3)O)F KM10675 CCCc1c(cnn1c2ncc(c(n2)C(F)(F)F)C(=O)OC)C(=O)OCC GK03734 COC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccco2 GK03737 Cc1cn(c2c1cccc2)CCC(=O)NCc3ccc4c(c3)OCO4 HTS01097 CCN(c1ccccc1)/C(=N/c2ccc(cc2)Cl)/SC.I RDR02123 CC(C)(C)c1ccc(cc1)c2nnnn2c3ccccc3C(F)(F)F RF04558 COc1ccc(cc1)NC(=O)NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F RF04510 CCc1c(nc2ccccc2n1)N3CCN(CC3)C(=S)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F GK03507 Cn1c(nnc1SCc2ccccc2)CNC(=O)c3ccc(cc3)Cl KM10704 COc1ccc(cc1)Oc2c(cccn2)NC(=O)Nc3cccc(c3)C(F)(F)F RH01993 CCOc1cccc2c1oc(=O)c(c2)C(=O)O RH02235 CCc1c(nc2ccccc2n1)N3CCN(CC3)S(=O)(=O)c4cc(c(cc4Cl)Cl)Cl GK03649 Cc1ccc(cc1)Sc2cc(c(cc2[N+](=O)[O-])Cl)n3cccc3 RH02245 CC(C)(C)c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4ccc(cc4)OC(F)(F)F GK03740 Cc1ccc(cc1F)NC(=O)c2cc3c(cc(cc3[nH]2)C)C KM11006 Cc1cc(n2c(n1)cc(n2)c3ccccc3OC)C KM00105 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc(cc3F)I KM11010 COc1ccc(cc1)c2ccnc(n2)SCC(=O)c3ccc(s3)Cl HTS00632 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4ccc(cc4F)F HTS00665 c1ccc(cc1)N/N=C\c2ccnc(n2)SCc3ccccc3Cl SPB04196 Cc1c(sc(n1)COc2ccccc2OC)C(=O)C SPB08293 c1ccc2c(c1)cc(o2)/C(=N/O)/c3ccc(cc3)Cl DP02004 Cc1nc(nc(n1)NC(=O)NC(=O)c2c(ccc(c2OC)Cl)OC)C BTB07648 c1ccc2c(c1)ccc3c2C(=O)CCO3 DP01872 CNC(=O)n1c(c(c(n1)c2ccc(cc2)Cl)SC(=O)NC)SC RF04999 Cc1ccc(cc1)C(=O)CSc2ccc(cc2)Cl SPB04109 CSc1nc(cc(n1)O)O SPB07198 CC(C)(C)n1c(cc(n1)C2CC2)NC(=O)c3ccccc3 KM00287 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc(c(n3)C)Br KM11008 CCc1ccc2c(c1)cc([nH]2)C(=O)NCc3ccccc3 KM11009 c1cc(c(c(c1)Cl)CSc2ccc(cn2)C(F)(F)F)F PD00597 Cc1ccccc1S(=O)(=O)NNC(=O)c2cc(c(cc2n3c(ccc3C)C)OC)OC GK03319 Cc1ccc(n1c2ccc(cc2)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl)C RH01958 Cc1ccc(n1c2ccc(cc2)C(=O)NNS(=O)(=O)c3ccc(cc3F)F)C RH01960 Cn1c(nnc1SCc2ccccc2)CNC(=O)c3cccs3 KM10708 CCOC(=O)NNc1ccc(cn1)C(F)(F)F RF04826 COc1cccc(c1)c2cc3nc(cc(n3n2)c4cccs4)C(F)(F)F KM00401 c1cc(ccc1S(=O)(=O)c2cnc(nc2NC(=O)NS(=O)(=O)Oc3ccc(cc3Cl)Cl)N4CCCCC4)Cl KM00980 CCc1ccc2c(c1)cc([nH]2)C(=O)NC(C)COC KM11011 CCCc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)OC RH01987 Cc1ccc(cc1C)C(=O)NC[C@H]([C@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC04017 c1ccc(cc1)c2cc(c(c(n2)O)C#N)C(F)(F)F RH02143 c1cc(c(c(c1)F)/C(=N/O)/Nc2ccc(cc2)C(F)(F)F)F RF05122 c1cc(sc1)c2nc(sn2)N3CCN(CC3)S(=O)(=O)c4ccc(c(c4)F)F SPB08328 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(o3)SCC(=O)c4ccccc4 SPB08339 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F RH01943 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)CSCC(=O)O HTS01109 CC(C)(CC(=O)N1CCN(CC1)S(=O)(=O)c2cc(cc(c2)Cl)Cl)CC(=O)O HTS00430 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)c3c(nccn3)C(=O)O HTS01414 c1ccc2c(c1)cnn(c2=O)CCOC(=O)c3ccc(cc3)OC(F)(F)F PD00602 CCCCCc1ccc(cc1)C(=O)NC(=S)Nc2ccsc2C(=O)OC HTS01477 c1ccc(cc1)C2=Nc3ccccc3SC(C2)c4ccc5c(c4)OCO5 PD00600 c1cc(c(cc1Br)/C=N/c2c(c3c(s2)CCCC3)C(=O)N)O RJC04018 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc(cc3Br)F KM11012 CCc1ccc2c(c1)cc([nH]2)C(=O)NCCc3ccccc3 KM11014 Cc1ccccc1NN=C(C(=O)C)C(=O)C SPB06724 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=N)N3CCOCC3 CD07768 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccncc2)C RJC04085 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccccc2OC)C RJC04086 c1ccc2c(c1)c(=S)c3ccccc3[nH]2 JFD03915 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(O)Oc4ccc(c(c4)Cl)Cl HTS00718 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)C(=O)C4CCC4C(=O)O HTS01135 Cc1ccc(cc1)c2nnc(n2CC(OC)OC)S SPB04801 c1cnc(nc1C(F)(F)F)N2CCC(CC2)C(=O)N3CCN=C(C=C3)C(F)(F)F HTS01564 c1cc(cc(c1)[N+](=O)[O-])/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00672 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)c3ccccc3Cl RH02073 COc1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccco3 RH01986 CCOC(=O)COc1c(c(cc(n1)C)C(F)(F)F)C#N RH02148 CSc1ccc(s1)C(=O)N SEW03628 COC(=O)c1ccccc1SC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F MBE00268 Cc1ccc(n1CCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C RH01942 Cc1ccc(n1c2ccc(cc2)c3nnc(n3c4ccc(cc4)C(F)(F)F)S)C RH01944 CCNC(=S)N1CCOCC1 RDR01196 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)Nc3ccc(cc3)C(C)(C)C)C SEW06396 CC(=O)N/C(=C/c1ccc(c(c1)Cl)Cl)/C(=O)O SPB08040 c1ccc(cc1)n2c(nnn2)SCC(=O)N3CCN(CC3)c4ccccc4 HTS01209 c1cc(ccc1NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl)OC(F)(F)F HTS01156 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2cccnc2 S13213 CCOC(=O)Cn1c2ccc(cc2c3c1nc4ccccc4n3)F RH01989 c1cc(oc1)CNC(=S)NCc2ccncc2 RDR00772 Cc1cc(ccc1[N+](=O)[O-])Oc2ccccc2 RH02074 CCOC(=O)c1c2c(sc1/N=C/c3cc(c(cc3O)Br)Br)CCCC2 RJC04020 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)C(=O)c5cccs5 AW01106 c1ccc(cc1)c2csc3c2c(ccc3)N4CCN(CC4)C(=O)c5ccc(c(c5)Cl)Cl AW01107 CCOC(=O)COc1c(c(cc(n1)c2ccccc2)C(F)(F)F)C#N RH02158 c1ccnc(c1)/N=N/c2ccc(cc2O)O JFD03916 COc1ccc(cc1)Oc2ccccc2OC RJC03901 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)OC(F)(F)F SP01073 Cc1c(cc(o1)C(C)(C)C)c2c(c([nH]n2)SC)C#N SP01086 CCOC(=O)c1c2c(sc1NC(=O)/C=C/C(=O)O)CCCC2 GK03285 c1cc(c(cc1F)F)C(=O)N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl HTS01442 c1ccc(cc1)/C=C(\C#N)/c2cccc(c2)Cl PHG00573 Cc1ncc(c(n1)c2ccc(cc2)Cl)Sc3ccc(cc3)Cl SPB04322 Cc1c(c(c(c(c1C)C)CSC2=NCN(CN2)C)C)C.Cl DP01302 c1cc(ccc1NC(=O)NNC(=O)Nc2ccc(cc2)OC(F)(F)F)OC(F)(F)F HC00105 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)c4ccccn4 SPB08277 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCN(CC4)C(=O)c5cccs5 AW01256 c1cc(c(c(c1)Cl)CN2CCN(CC2)c3c4c(csc4ncn3)c5cccs5)F AW01112 CN(c1ccc(cn1)[N+](=O)[O-])NC(=O)c2ccc(cc2F)F SP01285 c1ccc(cc1)CCNc2nnns2 HTS00543 COc1ccc2c(c1)cc([nH]2)C(=O)NCCSCc3cccc(c3)C(F)(F)F HTS00335 COc1cc(cc(c1OC)OC)C(=O)Nc2cc3c4ccccc4ccc3oc2=O PHG00788 CC(=O)c1c(cc(s1)c2ccc(cc2)F)NC(=O)c3ccc(c(c3)OC)OC GK03707 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(sc2C(=O)C)c3ccc(cc3)F GK03708 Cc1cc(nc(c1C(=O)N)OC)C RH02222 Cc1cc(nc(c1C(=O)O)OC)C RH02223 CC1CN(CC(O1)C)c2c3cc(c(cc3ncn2)OC)OC GK03283 COc1ccccc1N2CCN(CC2)CCCCNC(=O)c3ccc(cc3)Cl SEW06310 Cc1ccc(cc1)S(=O)(=O)NCCCCN2CCN(CC2)c3ccccc3OC SEW06373 CCCCC1(C(=O)c2cccc3c2n(c4c3cccc4)C1=O)Cc5ccccc5 JFD03991 COc1cccc2c1oc(=O)c(c2)C(=O)O RH02228 c1cc(sc1)c2cc(c(c(=O)n2N)C#N)C(F)(F)F RH02208 COc1cc(cc(c1OC)OC)/C=C(\C#N)/c2ccccc2 RDR00958 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)COc4ccccc4OC SPB08284 CCCCC(=O)NCc1nc(no1)c2ccc(cc2)C(F)(F)F HTS00572 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N RF02365 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2ccc(cc2)Cl)c3ccccc3)c4ccccc4)C SP01115 CC(C)(C)c1ccc(cc1)C(=O)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW01232 Cc1c2c(cn[nH]c2=O)c(n1CCSCc3c(cccc3Cl)Cl)c4ccccc4 SP01087 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)N3CCN(CC3)CCO KM10547 c1cc2c(cc1c3cc(n4c(n3)cc(n4)C5CC5)C(F)(F)F)OCO2 KM10546 Cc1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccc5c(c4)CCC5 KM10539 Cc1c(cc(o1)C(C)(C)C)c2c(c(n(n2)c3ccc(cc3)I)SC)C#N SP01097 CCn1c(nnn1)SCC(=O)NC2Cc3ccccc3C2 KM10550 CCCc1c2cc(c(cc2cc(n1)O)OC)OC JFD03988 c1ccc(c(c1)/C(=C/c2ccc(cc2)Cl)/C#N)Cl RDR00959 Cc1c(cccc1Cl)NC(=S)N/N=C\c2cccc3c2cccc3 RDR01027 CN(CCOC(=O)Nc1ccccc1)c2cc(nc3c2cccc3)C(F)(F)F KM08433 Cc1ccc(cc1F)NC(=O)c2cc3cc(ccc3[nH]2)OC SP01201 COc1cc(c(cc1OC)NC(=O)Nc2cc(cc(c2)Cl)Cl)C(=O)OC GK03120 c1ccc2c(c1)c(nc(n2)SCC(=O)c3ccccc3Cl)SCC(=O)c4ccccc4Cl PD00578 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)c4nnc(o4)N RJC04005 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCCC4C(=O)O RJC04009 CC(C(=O)O)NC(=O)OCC1c2ccccc2-c3c1cccc3 RJC04012 c1cc(ccc1/C=C/C(=O)Nc2ccc3c(c2)c(c[nH]3)C#N)OC(F)(F)F SP01315 c1ccc(cc1)C(=O)Nc2nc3ccsc3c(=O)s2 HTS01324 CCCc1cc(nc(n1)SCC(=O)NC2Cc3ccccc3C2)O KM10551 c1ccc2c(c1)CC(C2)NC(=O)CSc3nnnn3c4ccc(cc4)O KM10552 COC(CNC(=S)Nc1cc(c(cc1Cl)Cl)Cl)OC RDR00361 Cc1nc(cn1CC(c2ccccc2)O)[N+](=O)[O-] RH02179 CNc1nnc(s1)C(C(C(F)(F)F)(F)F)(F)F CD05965 c1cc(sc1)C2CCCN2S(=O)(=O)c3ccc(cc3)Cl CD10415 Cc1cc(c(c(c1)C)S(=O)(=O)O)C.CS(=N)c1ccccc1 KM06877 COc1ccc2c(c1)cc([nH]2)C(=O)NCCN3CCOCC3 SP01231 c1c(cnc(c1Cl)/C=N/O)C(F)(F)F HC00130 CCOC(=O)c1c2c(sc1N3C(=O)CCC3=O)CCCC2 GK03303 CCOC(=O)c1c2c(sc1N3C(=O)CSCC3=O)CCCC2 GK03302 Cc1c2c(cn[nH]c2=O)c(n1c3ccc(cc3)[N+](=O)[O-])c4ccccc4 SP01104 COc1ccc(cc1)C(=O)Nc2cccnc2 SPB08374 c1ccc(c(c1)C(=O)Nc2ccccc2Cl)Cl SPB08375 COc1c(csc1S(=O)(=O)N=S(=O)(C)c2ccc(cn2)C(F)(F)F)C(=O)OC KM08430 Cn1ccnc1SCC(=O)NC2Cc3ccccc3C2 KM10553 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)C)C RH01938 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3ccc(cc3)OC(F)(F)F)C RH01937 Cc1ccc(cc1)n2c(nnc2S)c3ccc(cc3)n4c(ccc4C)C RH01934 Cn1c2c(cn1)c(ncn2)NCCO GK03458 Cc1ccc(cc1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3)OC KM09948 Cc1c(cccc1OC)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM10042 COc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc(cc3F)I SP01229 CN(c1ccc(cc1F)F)C(=O)c2cc3cc(ccc3[nH]2)OC SP01210 CCOC(=O)c1c(n(c(c1S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)c4ccccc4)c5ccccc5)C SP01126 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NS(=O)(=O)c3ccccc3C(F)(F)F RH02081 Cc1cc(c(c(=O)[nH]1)C#N)C(F)(F)F RH02138 c1cc(cnc1)C(=O)CC(=O)c2cccnc2 RH02159 Cn1c(c(cn1)C(=O)NN)n2cccc2 GK03656 Cc1csc2c1nc(sc2=O)NC(=O)c3ccco3 HTS01332 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3cccs3)C HTS00993 c1ccc(c(c1)C(=O)Nc2cccnc2Oc3ccc(cc3)Cl)C(F)(F)F RH01932 CCC(CO)NC(=S)Nc1c(cc(cc1C)C)C RDR00424 c1cc(c(cc1I)F)NC(=O)CC2(CCCC2)CC(=O)O PD00680 c1(nnc(s1)N)C(C(C(F)(F)F)(F)F)(F)F CD05830 Cc1cccc(c1)C2=N/C(=C/c3ccc(c(c3)OC)OC)/C(=O)O2 PHG00655 CCCn1c(=O)c2c(cc(o2)C)n(c1=O)c3ccccc3C KM10044 C#CCOC(=O)Nc1ccc(c(c1)Cl)Cl RF05392 Cc1cccc(n1)NC(=O)c2cc3cc(ccc3[nH]2)OC SP01203 CC(C)(C)NC1=NN=C(CS1)c2ccc(cc2)Cl RDR01015 c1ccc(cc1)C(CN2CCN(CC2)C(c3ccccc3)c4ccccc4)O HTS00724 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2cccc(c2)C(F)(F)F)c3ccccc3)c4ccccc4)C SP01130 CC(=O)Nc1cccc(c1)C(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F TB00021 CCC1(C(=O)C=CNC1=O)CC JFD03934 CCOC(=O)c1cc2c3ccccc3[nH]c2cn1 JFD03941 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)/C=N\c3cc(c(cc3C)C)C SJC00186 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CN4c5ccccc5C6(C4=O)OCCO6 HTS00636 CCC1CS/C(=N\c2ccc(cc2)OC)/N1 RDR00428 c1cc(oc1)c2nnc(o2)S RDR02072 Cc1ccc(c(c1)[N+](=O)[O-])OCC(CN2CCC(CC2)C(=O)N)O HTS00981 c1cc(ccc1C(=O)Nc2nc3ccsc3c(=O)s2)Cl HTS01471 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2ccc(cc2)C(F)(F)F)c3ccccc3)c4ccccc4)C SP01134 CCOC(=O)c1c(n(c(c1S(=O)(=O)N2CCSC2C(=O)OC)c3ccccc3)c4ccccc4)C SP01135 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2ccc(cc2)[N+](=O)[O-])c3ccccc3)c4ccccc4)C SP01136 CCOC(=O)c1cc2c(ccnc2N3CCOCC3)nc1C(F)(F)F HC00141 Cc1ccc(cc1)C(=O)Nc2cc(sc2C(=O)C)c3ccccc3 GK03723 COc1ccc(cc1)C(=C)c2ccccc2 CD01809 CC(C)(C)c1ccc(cc1)CSCCNC2=CC(=O)CC(C2)c3ccc4c(c3)OCO4 SEW06593 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)NS(=O)(=O)c4ccc(cc4)Cl)C(F)(F)F SEW06596 CCc1cccc(c1NC(=O)C(C)Oc2ccc(cc2)C(C)(C)C)CC RDR02523 Cc1c(c(ccn1)O)OCc2ccccc2 RF01681 c1cc(cc(c1)[N+](=O)[O-])C(CNCc2ccc3c(c2)OCO3)O HTS00989 c1cc(ccc1OCC(CN2CCC(CC2)C(=O)N)O)Br HTS01115 Cc1ccc(c(c1)[N+](=O)[O-])OCC(CNCc2ccc(cc2)OC)O HTS01124 CCOC(=O)c1c2c(sc1NC(=O)CCC(=O)O)CCCC2 GK03295 c1cc(ccc1C2(CCN(CC2)S(=O)(=O)c3ccc(c(c3)Cl)F)O)Cl HTS00195 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2ccc(cc2)C(C)(C)C)c3ccc(cc3)Cl)C SP01139 c1ccc(cc1)C(=O)NC(=S)Nc2cccc3c2non3 PD00673 c1cc(cc(c1)/N=C\c2cc(cc(c2OS(=O)(=O)c3ccc(cc3)F)Cl)Cl)C(F)(F)F SJC00193 COc1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccccc3C(F)(F)F RH01926 c1cc2c(cc1C(F)(F)F)nc(cc2O)C(F)(F)F KM09515 c1cc(ccc1S(=O)(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)Cl RDR00572 CC(C)NCC(COc1ccc(cc1)OC)O.Cl RDR02611 Cc1cccc(c1)N2CCN(CC2)CC#N SEW06597 c1cc(cc(c1)C(F)(F)F)CSCCNC2=CC(=O)CC(C2)c3ccc(cc3)Cl SEW06598 c1cc(cc(c1)C(F)(F)F)CSCCNC2=CC(=O)CC(C2)c3ccc4c(c3)OCO4 SEW06599 Cc1cc(cc(c1NC(=O)c2ccc(cc2)Cl)C)I RDR02686 c1cc(ccc1c2nc(on2)CNC(=O)c3ccc(cc3F)F)C(F)(F)F HTS00574 c1cc(ccc1c2nc(on2)CNC(=O)COCC(=O)O)C(F)(F)F HTS00584 c1cc(ccc1C(=O)NC(=O)NN2CCCCCC2)C(F)(F)F SPB01462 c1cc(sc1)c2nc(cs2)CC(=O)NN SPB02328 Cc1cccc(c1NC(=S)Nc2ccc(cc2C)Br)Cl RDR00557 CC(C)(C)NC(=O)Cn1ccc(n1)C(F)(F)F HAN00239 c1cc(cc(c1)Oc2cc(ccc2C(=O)O)[N+](=O)[O-])[N+](=O)[O-] HTS01386 COc1ccc(cc1OC)C(=O)N2CCN(CC2)c3c4c(cc(s4)c5ccccc5)ncn3 GK03666 c1cc(ccc1C(F)(F)F)NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl HTS01155 COC(CNC(=O)COc1ccc(cc1Cl)Cl)OC SPB01417 COc1cc2c(cc1OC)ncnc2NNC(=O)c3ccco3 GK03668 c1ccc2c(c1)c(=O)c3cc(ccc3o2)OCC(=O)O RJC02950 CCOC(=O)/C(=C/Nc1ccccc1)/C#N RH02239 c1ccc(cc1)COC(=O)N[C@@H](Cc2ccc(cc2)O)C(=O)O SB02038 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)c2ccco2 HTS00023 CCn1c(c(c(n1)C)[N+](=O)[O-])C(=O)Nc2ccccc2 SPB02908 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)Cl)OC(F)(F)F SPB03485 CCOC(=O)c1c(csc1NC(=O)Nc2ccc(cc2)Cl)c3ccco3 HAN00453 c1ccc(cc1)CNS(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 KM10752 c1cc(ccc1CSCCCNC(=O)c2ccc(cc2)Cl)F SEW06615 c1cc(cc(c1)OC(F)(F)F)C(=O)NCCSCc2ccc(cc2)F SEW06616 CC(C)(C)NC(=S)NNC(=O)c1ccncc1 DP01752 CC(C)(C)OC(=O)NCc1nnc(n1C)SCc2ccccc2 KM10577 c1ccc2c(c1)C(=O)N(C2=O)CN3CCC(CC3)C(=O)N HTS00732 c1ccc2c(c1)C(C(=O)N2)Cc3ccc(cc3)N CD01293 Cc1csc2c1nc(sc2=O)NC(=O)c3ccc(cc3)Cl HTS01472 c1ccc2c(c1)c(=O)sc(n2)NC(=O)c3ccc(cc3)Cl HTS01473 c1c(ccc(c1)Cl)[C@H]2CC[C@@H](CC2)C(=O)O SB02037 c1cc2cccnc2c(c1)S(=O)(=O)N3CCN=C(C=C3)C(F)(F)F HTS00235 c1c(c(sc1S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F)Cl)Br HTS00232 c1cc(oc1)c2nccs2 CD10225 Cc1nc(cs1)c2nnc(n2C)SCC(=O)c3ccc(cc3)F HTS00219 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2ccco2 SEW04440 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)C3CCC3 RJC03014 CCCCCCCc1ccc(cc1)C(=O)N/C(=N/c2ccccn2)/SC BR00129 COC(=O)C(CCSC)N.Cl KM01809 Cc1cc(nc(n1)Sc2ccccc2NC(=O)c3ccccc3)C(=O)OC SPB06392 CN(C)NC(=O)c1ccc(s1)[N+](=O)[O-] RF01653 c1ccc(cc1)CNC(=O)CSCCS(=O)(=O)c2ccccc2 KM01727 CN1CCN(CC1)c2c3cc(c(cc3ncn2)OC)OC GK03378 c1c(cc(cc1C(F)(F)F)S(=O)(=O)N/N=C/c2cc(cc(c2O)Cl)Cl)C(F)(F)F JP00945 c1cc(ccc1NC(=S)N2CCC(CC2)CCCC3CCN(CC3)C(=S)Nc4ccc(cc4)F)F JP00966 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4ccccc4C(=O)O HTS00567 CCOC(=O)Cn1c2ccccc2c3c1cccc3 RH01949 c1ccc(cc1)SCC(CNCc2ccc3c(c2)OCO3)O HTS00807 c1cc(ccc1NC(=O)Cn2ccc(n2)C(F)(F)F)Cl HAN00237 CC(C)(C)c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4cc(cc(c4)OC)OC GK03747 CC(=O)c1c(cc(s1)c2ccccc2)NC(=O)c3ccco3 GK03748 CC(=O)c1c(cc(s1)c2ccccc2)NC(=O)c3cccs3 GK03749 c1ccc(cc1)CCNS(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 KM11052 CC(COC)NC(=O)c1cc2cccc(c2[nH]1)[N+](=O)[O-] KM11030 CCCCNC(=O)c1cc2c(cc(cc2[nH]1)C)C KM11033 c1cc(ccc1C(F)(F)F)NC(=O)CSc2nncn2c3ccc(cc3)C(F)(F)F HTS00226 CC(C)(C)OC(=O)N1CCC(CC1)C(=O)N TL00951 Cc1ccc(cc1)Sc2c(cccn2)c3nnc(o3)C4CC4 HTS01015 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)O)Oc3ccccc3 SPB04144 COc1cc2c(cc1OC)nc(sc2=O)NC(=O)c3ccc(cc3)Cl HTS01474 Cc1c(c(on1)C)n2c(=O)n(c(=O)s2)c3ccc(cc3)F HTS01243 Cc1c(c(no1)c2ccccc2)C(=O)N3CCC(CC3)(c4ccc(cc4)Cl)O HTS00204 c1cc(ccc1C2(CCN(CC2)C(=O)C3CCCCC3)O)Cl HTS00205 Cc1cc(c(cc1Cl)C)S(=O)(=O)NCCNc2ccc(cc2[N+](=O)[O-])C(F)(F)F RH01953 CSc1c(c(sn1)SC)C(=O)Nc2ccc(cc2)c3csnn3 SEW00793 CCOC(=O)N/N=C(\C)/c1ccc(cc1)C#N SEW00981 c1cc(ccc1C(=O)Nc2cc3cc(cc(c3oc2=O)Cl)Cl)Cl PHG00712 CSc1nc(n(n1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)N JM00008 CCOC(=O)c1cc2c(s1)cc(cn2)C(F)(F)F HC00132 CC(=N)NC(=S)Nc1ccc(cc1)Cl JM00016 c1cc2c(ccnc2cc1Cl)N3CCN(CC3)C(=O)C4CCC4 KM11056 COC(=O)CCC(=O)c1ccn(c1)S(=O)(=O)c2ccccc2 RH02254 Cc1cc(c2cc([nH]c2c1)C(=O)NCc3ccccc3)C KM11036 CCCCCCCc1ccc(cc1)C(=O)N/C(=N/c2cccc(n2)C)/SC BR00127 COc1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4OC KM10578 Cc1ccc(n1c2ccc(cc2)C(=O)NNS(=O)(=O)c3cccc(c3)C(F)(F)F)C RH01950 CCSc1nc(nc(n1)O)c2ccc(cc2)Cl JM00164 CC(=O)NC(Cc1cc(c(c(c1)[N+](=O)[O-])O)[N+](=O)[O-])C(=O)O KM08324 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)c3c(nccn3)C(=O)O HTS01411 c1ccc(c(c1)C(F)(F)F)n2c(nnn2)c3ccc(cc3)F RF04543 c1ccc2c(c1)c(=O)n(c(n2)S)c3ccc(c(c3)Cl)Cl RDR01287 CC(=O)N1CCC(CC1)c2nc(no2)c3ccc(cc3)C(F)(F)F KM10800 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01110 Cc1nc(cs1)c2nnc(n2C)SCC(=O)Nc3ccc(cc3)C(F)(F)F HTS00222 CC(=O)C(=NNc1cccc(c1)C(F)(F)F)C(=O)C RH01956 Cc1ccc(cc1)S(=O)(=O)n2ccc3c2ccc(c3)N.Cl SS00046 CNC(=S)N(Cc1ccccc1)Cc2cccs2 RF03344 Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccccc3 SPB03009 Cc1c(c(on1)C)n2c(=O)n(c(=O)s2)CC3CC3 HTS01244 c1cc(c(c(c1)Cl)OC/C(=N/O)/N)Cl SPB02461 CCn1c2ccc(cc2nc1S)Cl SPB02590 CCC(C)c1ccccc1NC(=O)c2cc3c(cc(cc3[nH]2)C)C KM11040 Cc1ccc(n1c2c3c(cccc3F)n(n2)S(=O)(=O)C)C HTS01086 COc1ccc2c(c1)cc([nH]2)C(=O)NC3CCN(CC3)Cc4ccccc4 HTS01092 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(n3C4CCCCC4)SCc5c(cccc5Cl)F SPB08191 COc1ccc(cc1)NC(=O)C(C(=O)Nc2ccc(cc2)OC)C34CC5CC(C3)CC(C5)C4 JFD03972 Cc1cc(cc(c1OC(=O)c2cc(nn2Cc3ccc(cc3)F)C(C)(C)C)Cl)Cl SPB08280 c1ccc2c(c1)C3(C(=O)N2CN4CCN(CC4)CCO)OCCO3 HTS00590 CCN(CC)c1c2cnn(c2ncn1)C GK03454 CC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)OC GK03750 CC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F GK03752 CC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl GK03754 Cc1cc(c2c(c1)cc([nH]2)C(=O)Nc3ccc4c(c3)OCO4)C KM11038 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F HTS00060 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)c2cccs2 HTS00041 c1cc2cc([nH]c2c(c1)[N+](=O)[O-])C(=O)NCc3cc(ccc3Cl)Cl KM11039 Cc1cccc(c1)C2=N/C(=C/c3ccc(cc3)Cl)/C(=O)O2 PHG00659 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccccc2Cl RDR00405 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)C(=O)c4c(nccn4)C(=O)O HTS01136 CC(=O)c1csc(n1)c2ccc(nc2)OCC(F)(F)F SPB07471 c1cc(oc1)c2ccc(c(=O)[nH]2)C#N SPB07843 COc1c(csc1Cl)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM00466 COc1ccc(c(c1)NC(=O)c2csc(c2OC)Cl)OC KM00470 COC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccccc2 GK03735 COc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc4c(c3)OCO4 SP01198 c1ccc(c(c1)/C(=N/O)/C#N)Cl SPB00254 Cc1ccc(cc1)S(=O)(=O)Nc2ccnn2C GK03317 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)N)N GK03408 CC(C)(C)c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4ccccc4 GK03742 Cc1cc(c2cc([nH]c2c1)C(=O)N(C)c3ccc(cc3)Cl)C KM11043 Cc1cccc(n1)NC(=O)c2cc3cccc(c3[nH]2)[N+](=O)[O-] KM11044 COc1ccc2c(c1)cc([nH]2)C(=O)NCCc3ccccc3 SP01208 C1CCN(CC1)C(=O)C(C(=O)N2CCCCC2)C34CC5CC(C3)CC(C5)C4 JFD03973 Cc1cc(c(c(c1)C)C(=O)C2CCN(CC2)C(=O)c3ccc(cc3)Cl)C SEW06383 Cc1cc(c(c(c1)C)C(=O)C2CCN(CC2)C(=O)c3ccc(cc3)OC)C SEW06386 c1cc(oc1C(=O)NN)Oc2cc(cc(c2)Cl)Cl SPB03104 CC1=C(CC2C(C1)C(=O)N(C2=O)c3ccc4c(c3)OCO4)C PD00678 CC(C)(C)C(=O)CN1C(=O)c2ccccc2C1=O SP01116 CC(C#N)Oc1ccc(cc1Cl)Cl SPB00388 CC(=O)CN1C(=O)c2ccccc2C1=O SP01117 c1cc(oc1)CNC(=S)N/N=C/c2ccc(cc2)Cl RDR00736 Cc1cc(ccc1NC(=S)N/N=C/c2cc(cc(c2O)Cl)Cl)Br RDR00691 CN(C)/C=C(/C(=O)c1ccc(cc1)Cl)\Sc2ncccn2 SPB04169 CC(C)Cc1ccc(cc1)C(C)C(=O)NNC(=O)c2ccccc2Cl SEW06474 CN1c2ccccc2C(=O)/C(=C/Nc3nc(nc(n3)SC)C4CC4)/S1(=O)=O KM01417 Cn1c(cc(=O)n(c1=O)C)NCc2ccc(cc2)F PD00811 COc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccccc3Cl SP01197 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2cc(c(cc2n3c(ccc3C)C)OC)OC GK03306 Cc1cccc(n1)NC(=O)c2cc3c(cc(cc3[nH]2)C)C KM11005 COc1ccc(cc1OC)/C=C(\C#N)/S(=O)(=O)c2ccc(cn2)C(F)(F)F RF04734 CC(C)(C)c1cc([nH]n1)C(=O)NNS(=O)(=O)c2ccccc2 RF04979 Cc1cc(nc(n1)NC(=O)C)O RDR01727 c1ccc(cc1)/C=C/C2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)O2 PHG00752 Cc1c(c(nc(n1)c2cccnc2)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F)Cl AW01235 COc1ccc(cc1[N+](=O)[O-])/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00931 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)C(=O)O RJC04003 c1ccc(cc1)CON2C(=O)c3ccccc3C2=O TL00612 c1ccc(c(c1)C(=O)N2CCCN(CC2)c3c(cccn3)C(F)(F)F)C(=O)O AW00949 COC(=O)c1c(ccs1)S(=O)(=O)NNC(=O)c2ccc(cc2)[N+](=O)[O-] HTS00484 Cc1cc(c2cc([nH]c2c1)C(=O)Nc3ccc(cc3F)I)C KM11002 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc(c(c3)F)C KM11003 CC(C)(C)c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4ccc(cc4)I GK03744 Cc1cc(cc(c1)Nc2c3c(cc(s3)c4ccc(cc4)C(C)(C)C)ncn2)C GK03745 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCC(CC3)n4cccc4 HTS00663 Cc1c2cc(ccc2sc1c3cc(n(n3)C)C(F)(F)F)Cl SP01368 Cc1ccc(c(c1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)[N+](=O)[O-] BTB01500 Cc1ccc(c2c1CCC2)Oc3c(cccn3)C(F)(F)F BTB09399 CCCCCc1ccc(cc1)C(=O)NC(=S)Nc2c(cnn2C)C(=O)OCC HTS01482 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)ON=C2C3CC4CC(C3)CC2C4 JP00898 Cc1ccc(cc1)COc2ccc(cc2)I JP00917 CN(C)C(=O)Oc1ccnc(n1)SCc2c(cccc2Cl)F JM00429 c1ccc(cc1)c2cc(c3cc(ccc3n2)Br)C(=O)N BW00129 CSc1nc2ccc(cc2s1)NS(=O)(=O)c3ccc(s3)Br KM10779 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc4c(c3)sc(n4)SC KM10784 Cc1c2cc(ccc2sc1C(=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)Cl HTS01200 c1cc2c(cc1C(CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)O)OCCO2 HTS01384 CCCCCc1ccc(cc1)C(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS01385 COc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cc(c(c(c3)OC)OC)OC PHG00777 c1ccnc(c1)CCN2C(=O)c3cccc4c3c(ccc4Br)C2=O PHG01016 c1cc(ccc1OC(F)(F)F)S(=O)(=O)NNC(=O)CSc2c3c4c(sc3ncn2)CCCC4 GK03298 c1cc(ccc1c2csc(n2)c3cnccn3)Br SEW06388 CC(C)(C)OC(=O)NCc1nnc(n1C)SC KM10576 CCOC(=O)c1c(c(on1)C)/C(=N/Nc2ccccc2Cl)/C SPB04273 CSc1c(ccc(n1)/C=N/O)C#N SPB04451 Cc1c(c(nc(n1)N)O)Oc2ccc(cc2Cl)Cl SPB04466 CC(=O)NNC(=O)CSc1c2c3c(sc2ncn1)CCCC3 GK03297 c1ccc(c(c1)N)Sc2cc(c(cc2[N+](=O)[O-])Cl)Sc3ccccc3N JP00490 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)NC3CCN(CC3)Cc4ccccc4 KM10705 c1cc(cnc1)NC(=O)CC2(CCCCC2)CC(=O)O PD00723 CCc1c(nc2ccccc2n1)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl GK03509 CCCc1ccc(cc1)NS(=O)(=O)c2c(oc(c2C(=O)OC)C)C HTS01163 Cc1c(c(c(o1)C)S(=O)(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O)C(=O)OC HTS01166 Cc1csc2c1nc(sc2=O)NC(=O)c3ccc(cc3)C(C)(C)C HTS01340 CN(C1CCS(=O)(=O)C1)C(=O)c2ccc(o2)Br JFD03983 Cc1cc(c2ccccc2n1)N3CCN(CC3)C(=O)/C=C/C(=O)O RH02180 Cc1c(sc(n1)c2ccc(cc2)Cl)c3csc(n3)c4ccc(cc4)Cl RH02182 COc1cccc(c1)c2nn(c(=O)o2)c3cc(ccn3)C(F)(F)F RF04931 c1cc(c(cc1F)Cl)C(=O)Nc2nc3ccsc3c(=O)s2 HTS01483 c1ccc(cc1)c2cc(c(o2)NC(=O)c3cccs3)C#N HTS01247 Cc1cccc(c1)C(=O)Nc2ccc(c(c2)C)C RDR01924 Cc1cccc(c1)c2nc(cc(n2)OC(=O)N(C)C)C RDR02801 CCCCc1ccc(c(c1)C)NC(=O)Nc2ccc(cc2)N3CCN(CC3)C HTS01160 CC(c1cccnc1)OC(=O)c2ccc(cc2)[N+](=O)[O-] BW00058 C/C(=N\Nc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])/c2cccnc2 BW00069 c1csc2c1ncnc2NN3CCCCC3 GK03292 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCCCO SPB08211 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(O)Oc4cccc(c4)C(F)(F)F HTS00931 c1cc(ccc1c2nc(on2)CNC(=O)C3CCCCC3)C(F)(F)F HTS00573 c1cc(ccc1OCC(CNCc2ccc3c(c2)OCO3)O)OC(F)(F)F HTS01111 CCC(=O)NCc1ccc(cc1Cl)Cl RF04991 CCCCNC(=O)Oc1ccc(cc1)C2=NCCS2 SPB01403 CC(C)c1ccc(cc1)NC(=S)NC(=O)c2ccc(cc2)C(F)(F)F SPB01432 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccc(cc3)OC(F)(F)F RH02080 CCCN1C(C(c2ccccc2C1=O)C(=O)O)c3ccc(cc3)OC PD00679 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)c3cccc(c3)C PHG00661 c1cc(ccc1NC(=O)C(=O)Nc2ccc(cc2)Cl)Cl JFD03944 c1cc(c(cc1)O)/C=N/CC2CCC(CC2)C/N=C/c3c(cccc3)O JFD03947 c1ccc(cc1)c2c3cc(ccc3ncn2)Cl JFD03957 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2OC)/C=N/NC(=S)Nc3cc(ccc3Cl)Cl RDR01241 c1cc(cc(c1)Cl)C2=N/C(=C/c3ccc(c(c3)Cl)Cl)/C(=O)O2 PHG00641 c1cc(cc(c1)Nc2nnc(s2)c3cccnc3)C(F)(F)F BW00112 COc1ccc(cc1)c2ccnc(n2)SCc3ccc(cc3Cl)Cl KM10759 Cn1c(cc(=O)n(c1=O)C)N2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS01387 COc1ccc(cc1)COCC(CNC2Cc3ccccc3C2)O HTS00784 COc1ccc(cc1)c2ccnc(n2)SCc3cccc(c3)[N+](=O)[O-] KM10760 c1cc(c(c(c1)Cl)Cl)NC(=S)NCc2ccncc2 RDR00576 CC(C)(C)c1cc2c(s1)c(ncn2)N/N=C/c3ccc(cc3)OC GK03665 Cc1cc(c(cc1Cl)C)S(=O)(=O)NNc2c3c(cc(s3)C(C)(C)C)ncn2 GK03667 COC(=O)c1c(ccs1)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)N HTS01031 c1cc(ccc1NC(=O)Nc2ccc(cc2)F)F HTS00434 CCc1ccc2c(c1)cc([nH]2)C(=O)NCCN3CCCCC3 KM11041 c1cc2cc([nH]c2c(c1)[N+](=O)[O-])C(=O)Nc3ccc(cc3Br)F KM11042 Cc1cc(c2cc([nH]c2c1)C(=O)Nc3ccc(c(n3)C)Br)C KM11046 CC(C1CC2CCC1C2)NC(=O)C(C(=O)NC(C)C3CC4CCC3C4)C56CC7CC(C5)CC(C7)C6 BTB14793 Cc1cc(=O)oc(c1C(=O)O)C KM09734 Cc1ccccc1n2c(cc(=O)n(c2=O)Cc3ccc(cc3)C(=O)OC)N KM10011 c1cnc(cc1C(F)(F)F)NCCNc2nccc(n2)C(F)(F)F HAN00248 CC(C)Cc1ccc(cc1)C(C)C(=O)NNC(=O)c2cccc(c2)[N+](=O)[O-] SEW06478 Cc1ccc(n1c2ccc(cc2)C(=O)NNS(=O)(=O)c3ccc(cc3)OC)C RH01947 c1ccc(c(c1)N)SCC(COc2cccc(n2)C(F)(F)F)O HAN00268 CS(=O)(=O)Nc1ccccc1c2nnc(o2)Cc3cc(cc(c3)F)F SP01386 Cc1c(c(c(o1)C)S(=O)(=O)Nc2ccccc2)C(=O)OC SP01391 Cc1c(c(c(o1)C)S(=O)(=O)N(C)C)C(=O)OC SP01392 CC(C)(C)c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4cccc(c4)Br GK03743 c1ccc(cc1)CSC(=N)Nc2cc(ccc2Cl)Cl.Cl RDR01678 c1ccc(cc1)c2ccccc2CO JFD03959 Cc1cc(c(nc1)NC(=O)c2cc3cc(ccc3[nH]2)OC)Br SP01209 Cc1cc(nc(n1)C)NC(=O)c2cc3cc(ccc3[nH]2)OC SP01204 CCCCNC(=O)c1cc2cc(ccc2[nH]1)OC SP01207 COc1cc2c(cc1OC)ncnc2NC3CCCCC3 GK03357 CC(C)(C)OC(=O)Nc1cc(ccc1OC)C(=O)O SPB08147 c1cc(ccc1CCc2ccc(cc2)Cl)Cl KM09696 COC(=O)c1ccc(cc1)CSc2nnc(n2CC=C)c3ccc4c(c3)cccn4 KM10649 CCC(CO)NC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F RDR00561 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3c(cccc3F)F)Cl SEW06475 COc1ccc(cc1)C(=O)NCc2c(cccc2Cl)Oc3ccccc3 SEW06476 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3cccc(c3)C(F)(F)F)Cl SEW06477 c1cc(cc(c1)NC(=O)Cn2ccc(n2)C(F)(F)F)C(F)(F)F HAN00240 COc1ccc(cc1OC)/C=N/NS(=O)(=O)c2ccc(cc2)Cl RDR00583 c1cc(sc1C(=O)NC(=O)N2CCOCC2)[N+](=O)[O-] RF01665 Cc1ccc(cc1)NC(=O)NCc2ccc3c(c2)CCO3 SP01305 COc1ccc(cc1)c2ccnc(n2)SCc3c(cccc3Cl)F KM10763 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCCCOC RDR02536 CC(C)Nc1c2c3c(sc2ncn1)CCCC3 GK03360 c1cc(ccc1n2c(c(cn2)C(=O)NC3CCCCC3)C(F)(F)F)Cl GK01738 c1ccc(cc1)N2CC(OC2=O)COc3ccc(cc3)Br RDR03125 COC(=O)c1c(ccs1)NC(=O)CSCC(=O)O HTS00183 Cc1c(cccc1OC)NC(=O)NCc2ccccc2 KM10033 CCc1ccc2c(c1)cc([nH]2)C(=O)NCCN3CCOCC3 KM11016 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc(c(c3)C#N)C(F)(F)F KM11017 c1cc(ccc1F)SCC(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS00957 c1cc(ccc1n2c(nnn2)SCc3cc(cc(c3)F)F)O HTS00944 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)C(=O)c4cc(cc(c4)Cl)Cl GK03760 CCOC(=O)C1CCN(CC1)c2c3cnn(c3ncn2)C HTS00361 Cc1ccc(c(c1)NC(=S)Nc2ccc(cc2OC(F)(F)F)Br)n3cccc3 SEW06489 c1ccc2c(c1)C(=O)N(C2=O)CN3CCN(CC3)c4ccc(cc4[N+](=O)[O-])C(F)(F)F PD00814 Cc1c(c(n(n1)C)NCCCN2CCOCC2)[N+](=O)[O-] HTS00372 CC(C)(C)c1ccc(cc1)C(=O)Nc2nc3ccccc3c(=O)s2 HTS01341 CC(C)(C)c1ccc(cc1)C(=O)Nc2nc3cc(c(cc3c(=O)s2)OC)OC HTS01342 c1c(cn2cc(nc2c1Cl)C(=O)NN)C(F)(F)F RDR03772 c1cc(c(c(c1)F)c2nn(c(=O)o2)c3ccc(cn3)C(F)(F)F)F RF04829 Cn1cc(c(n1)NC(=O)/C=C\C(=O)O)Br GK02751 c1ccc(cc1)CNC(=O)c2ccc3c(c2)nns3 KM10650 Cc1ccc(cc1)c2nnn(n2)CC(=O)NNC(=O)C(C)(C)C GK03462 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc4c(c3)OCO4 KM11015 Cn1c2cccc(c2c(n1)NC(=O)/C=C/c3ccc(cc3)OC(F)(F)F)F SP01322 COc1ccc(c(c1OC)Cl)C(CC(=O)c2cccs2)Sc3ccccc3N HTS00615 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3cc(c4c(n3)c(cs4)C(=O)OC)C(F)(F)F GK03756 C1CC1c2nnc(s2)NC(=O)C3CC3 RH02253 COC(=O)c1c(ccs1)S(=O)(=O)NNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl HTS00402 Cc1cc(c(nc1)NS(=O)(=O)c2ccsc2C(=O)OC)Br HTS00126 CC(=O)c1ccc(cc1)OCC(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS00804 c1cc2c(cc1OCC(CN3CCC(CC3)C(=O)N)O)OCO2 HTS00797 COc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-] PHG00674 c1ccc-2c(c1)CCc3c2sc(c3)C(=O)O PD00589 CCC(Cn1c2c(nc1NCc3ccccc3)n(c(=O)n(c2=O)C)C)O RJC03326 c1ccc(cc1)CN2CCC(CC2)NC(=O)C3=Cc4cc(ccc4OC3)Cl HTS00418 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)C3CC3 RH02084 Cc1cc(nn1C(C)(C)C)C(=O)NNS(=O)(=O)c2ccc(cc2)C(C)(C)C HTS00054 c1ccc(c(c1)C(F)(F)F)NC(=O)c2cc(cc(c2)Cl)Cl RF04632 c1cc(ccc1CCNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)Cl GK01736 Cc1ccc(cc1)S(=O)(=O)Nc2csc(c2C(=O)Nc3ccc(cc3)OC)C HTS00467 c1cc(nc(c1)NCCNc2nccc(n2)C(F)(F)F)C(F)(F)F HAN00247 Cc1cc2nnc(c(n2n1)C)/C(=N\O)/C KM01319 c1ccnc(c1)S(=O)(=O)Cc2cccc(c2)C#N KM01557 c1ccc(cc1)COc2c3cccc4c3n(c(=O)c2[N+](=O)[O-])CCC4 BTB09650 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)COc3ccccc3)C RH01965 CCCc1ccc(cc1)C(=O)NNC(=O)c2ccc(cc2)n3c(ccc3C)C RH01966 CC(C)NC(=O)N(Cc1ccc(cc1)Cl)Cc2cccs2 RF03401 CC(C)(C)N\1C(=O)C(S/C1=N\N=C\c2cccc(c2)[N+](=O)[O-])c3ccccc3 RF01573 CC(=O)CC1(c2cc(ccc2NC1=O)F)O RH02231 Cc1ccc(cc1)c2csc3c2c(ncn3)NCCc4ccc(c(c4)OC)OC AW01197 c1ccc(cc1)OCC(CNCc2ccc3c(c2)OCO3)O HTS00938 c1ccc(cc1)c2c(snn2)C(=O)Oc3ccc(cc3)Cl CD05486 Cc1cc(cc(c1OCC(CNCc2ccc3c(c2)OCO3)O)Br)Cl HTS00950 c1cc(sc1)SCC(CNCc2ccc3c(c2)OCO3)O HTS00959 c1cc(cc(c1)C(F)(F)F)c2nn(c(=O)o2)c3ccc(cn3)C(F)(F)F RF04840 CCOC(=O)c1c(c(sc1N2C(=O)CC3(C2=O)CCCC3)C)c4ccccc4 AW00948 c1ccc2c(c1)cnn(c2=O)c3cc(ccc3Cl)Cl PD00582 Cn1c(nnc1SCC(=O)O)Cn2c3ccccc3c4c2cccc4 RH02088 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3ccco3 PD00682 c1cc(c(c(c1)F)C(=O)O)NC(=O)CSCC(=O)O HTS00456 COC(=O)c1c(cc(s1)S(=O)(=O)Nc2ccc(cc2)F)Cl HTS00468 Cc1cc(nn1C(C)(C)C)C(=O)NNS(=O)(=O)C HTS00061 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(COc4ccc(cc4)F)O HTS00701 CC(=O)c1ccc(cc1)OCC(CNCc2ccc3c(c2)OCO3)O HTS00801 CC(C)(C)OC(=O)NCc1nnc(n1C2CC2)S KM10564 CC(C)(C)OC(=O)NCc1nnc(n1C)SCC(=O)c2ccc(cc2)Cl KM10603 c1ccc2c(c1)CC(C2)NCC(COc3ccc(cc3)Cl)O HTS00976 c1cc(ccc1OCC(CNCc2ccc3c(c2)OCO3)O)Br HTS01114 COC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2cccs2 GK03733 c1cc(c(c(c1)Cl)c2nc(on2)C(=O)NN)F SPB00721 Cc1cc(c(cc1Cl)C)SCc2nc(no2)COc3c(cccc3Cl)Cl SPB03185 CC(C#C)OC(=O)Nc1cnccc1C(F)(F)F RF04724 Cc1c(c(n[nH]1)C)Sc2nnc(n2C)C(F)(F)F SPB03958 CCOC(=O)/C(=N\Nc1cccc(c1)Cl)/C(=O)CSc2ccc(cc2)Cl SPB04017 CCOC(=O)CNC(=S)SC RF02866 c1ccc(c(c1)C(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F)C(F)(F)F HTS00080 c1ccc(c(c1)C(=O)O/N=C(/c2cccc(c2)COc3ccc(cc3)Cl)\N)Cl KM01661 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)COCC(=O)O HTS00566 CCOC(=O)c1c(csc1NC(=O)CSCC(=O)O)C HTS00181 c1cc(sc1)CCN2C(=O)CC3(C2=O)CCCC3 AW00947 Cc1cc(c(c(c1)C)NC(=S)NC(=O)C(C)Oc2ccc(cc2)I)C RDR02299 c1cc(c(cc1CSc2nc3cc(ccc3c(=O)n2c4ccc(c(c4)Cl)Cl)Cl)Cl)Cl RDR01319 Cc1ccc(cc1C)OCC(CNCc2ccc3c(c2)OCO3)O HTS00967 Cn1c(c(c(n1)C(F)(F)F)/C=N/Nc2ccc(cc2)[N+](=O)[O-])O GK02661 c1cnc(cn1)c2nc(cs2)C34CC5CC(C3)CC(C5)C4 SPB08343 CCOC(=O)c1ccc(cc1)N2C(=O)CC3(C2=O)CCCC3 AW00951 c1cc(ccc1C(=O)NNC(=O)c2cnccc2C(F)(F)F)OC(F)(F)F SPB03470 Cc1c(snn1)c2nc(cs2)/C(=N/OC(=O)c3ccccc3)/C SPB03849 c1cc(ccc1N2CCOCC2)N3C(=O)c4ccncc4C3=O HTS00631 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)Nc3ccccc3Cl KM11054 CC1(CCC(=O)N(C1=O)c2ccc(cc2)N3CCOCC3)C HTS00599 CC(C)(CC(=O)NNc1c(cnn1C)C(=O)O)CC(=O)O HTS00091 CC(C)(C)c1[nH]c(nn1)Sc2c(cccn2)[N+](=O)[O-] SPB00540 Cn1c(nnc1SCC(=O)NNC(=O)c2ccc(cc2)Cl)Cc3ccsc3 SPB02394 c1cc(c(cc1c2nc(no2)CO)Cl)Cl RF03009 CC(C)(C)c1ccc(c(c1)Cl)NC(=O)NC RF01593 CC1([N+](=c2ccc(cc2=[N+]1[O-])[N+](=O)[O-])[O-])C RH02211 c1cc(c(cc1C#N)[N+](=O)[O-])Oc2ccc(cc2Cl)Cl SPB01876 C=CCn1c(nnc1S)O SPB01982 c1cc(ccc1F)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F HTS00231 COc1cn(nc(c1=O)C(=O)OC)c2cccc(c2)Cl SPB04024 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)C(=O)C5CC5 AW01108 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)N2CCN(CC2)c3c4c(csc4ncn3)c5ccccc5 AW01103 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)CSCC(=O)O HTS00490 Cn1c(ccn1)NC(=O)Nc2cccc(c2Cl)Cl GK03305 CN1CCN(CC1)c2ccc(cc2)NS(=O)(=O)c3cccc4c3non4 HTS00073 Cc1csc2c1nc(sc2=O)NC(=O)c3cccs3 HTS01346 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4cccc5c4non5 HTS00656 c1ccc2c(c1)cnn(c2=O)c3ccc(cc3)F PD00574 c1ccc(c(c1)/C=C(\C#N)/c2cccc(c2)Cl)Cl PHG00579 COc1ccc(cc1)/C=C(\C#N)/c2cccc(c2)Cl PHG00576 Cn1c2c(cn1)c(ncn2)NCC=C GK03453 CC(C)(C)c1cc(cc(c1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)C(C)(C)C KM00994 CCCS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/Nc2cccc(c2)OC KM00997 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(cc2)C(F)(F)F RF03255 c1cc2c(cc1NC(=O)CCC(=O)O)OCCCO2 HTS00135 Cc1cc(c2cc([nH]c2c1)C(=O)NC(C)COC)C KM11035 CC(C)(C)OC(=O)NCCNc1ccc(cc1N2C(=O)CC3(C2=O)CCCC3)C(F)(F)F AW00955 CC(C)(C)OC(=O)N1CCC(CC1)c2nc(cs2)c3ccc(s3)Cl HTS00074 CC(C)n1c2ccc(cc2[nH]c1=S)C(F)(F)F TG00015 c1cc(ccc1NC(=S)NCCNC(=S)Nc2ccc(cc2)Cl)Cl RDR00642 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3cc(ccc3Oc4ccc(cc4)OC)C(F)(F)F HTS00853 CN(C1CCS(=O)(=O)C1)C(=O)COc2ccc(cc2)Oc3ccccc3 JFD03976 c1cc(ccc1[N+](=O)[O-])OCCOC(=O)c2ccc(o2)Br JFD03978 Cc1cc(c(cc1Cl)C)S(=O)(=O)NNc2c3cnn(c3ncn2)C GK03511 CC(COC)NC(=O)c1cc2cc(ccc2[nH]1)OC SP01206 Cc1ccc(n1c2c(c3c(s2)CCCC3)C(=O)NNC(=O)c4ccc(cc4)Cl)C GK03315 Cn1c(ccn1)NC(=O)Nc2cc(cc(c2)OC)OC GK03304 COC(=O)c1ccccc1NC(=O)c2c(cccc2F)F GK03362 Cc1c(c(c(o1)C)S(=O)(=O)NC2CCCCCCCCCCC2)C(=O)OC HTS01161 CC1=C(CC(C(C1)C(=O)NCc2c(cccc2Cl)F)C(=O)O)C HTS00875 c1ccc(c(c1)NC(=O)c2cc3cccc(c3[nH]2)[N+](=O)[O-])Cl KM11050 c1ccc2cc(ccc2c1)S(=O)(=O)NCCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F RH01941 c1cc2cccnc2c(c1)Oc3ccc(cc3)[N+](=O)[O-] SEW06400 CCCCNC(=S)NNC(=O)CNC(=O)OC(C)(C)C KM10568 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)C)c3ccc(cc3)F GK03711 c1cc(sc1)c2nc(on2)C(=O)NN SPB00568 c1ccc2c(c1)C(=O)N(C2=O)CCCN3CCN(CC3)Cc4c(cccc4Cl)F AW01111 c1ccc2c(c1)cccc2/C=C/3\C(=O)OC(=N3)c4cccc(c4)[N+](=O)[O-] PHG00669 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3cccs3 RH02072 Cc1ccc(n1c2cc(c(cc2C(=O)NNS(=O)(=O)c3ccc(cc3)Cl)OC)OC)C GK03307 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(c(c2)OC)OC RH01957 Cc1cc(c2c(c1)cc([nH]2)C(=O)Nc3ccc(cc3Br)F)C KM11047 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3ccc(cc3)CN4Cc5c(n(c(=O)n(c5=O)C)C)NC4 PD00727 COc1ccc(cc1OC)CCN2C(=O)/C(=C\c3ccccc3C(=O)O)/SC2=S PD00728 Cc1ccc(cc1)S(=O)(=O)N/N=C(\C)/c2ccc(cc2)OCCOc3ccc(cc3)[N+](=O)[O-] JFD03984 Cc1c(c(c(o1)C)S(=O)(=O)N2CCCC2)C(=O)OC SP01384 c1ccc(cc1)NC(=O)n2c(ccn2)c3ccc(cc3Cl)[N+](=O)[O-] MWP00482 c1ccc(c(c1)C(=O)O)SCC(=O)c2ccc(cc2)Cl JP00881 c1cc2c(ccnc2cc1Cl)SCC(=O)NN KM10748 c1ccc2c(c1)ncn2Cc3ccc(cc3)C(=O)O KM10745 c1cc(c(nc1)N2CCN(CC2)CCCCNS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F SEW06485 COc1ccc2c(c1)c(cc(n2)c3ccccc3)O RH02079 COC(=O)c1cnc(nc1C(F)(F)F)n2c(c(cn2)C#N)N GK03746 CCOC(=O)c1c(n(c(c1S(=O)(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F)c4ccccc4)c5ccccc5)C SP01128 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2ccc(cc2)OC(F)(F)F)c3ccccc3)c4ccccc4)C SP01132 c1cc(sc1)c2ccnn2C(=O)c3cccs3 SEW06463 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3cc(c(cc3Cl)Cl)Cl GK03369 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)NC(=O)C GK03370 CC(=O)c1c(cc(s1)c2ccc(cc2)F)NC(=O)c3cccs3 GK03713 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)NC(=O)c4cccs4)C(F)(F)F SEW06379 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)c3nnc(o3)Cc4cc(cc(c4)F)F SP01361 Cc1c(ccc(n1)NC(=O)c2cc3cc(ccc3[nH]2)OC)Br KM11000 COc1cc(c(cc1OC)NC(=O)Nc2cccc(c2)Cl)C(=O)OC GK03122 CCN(CC)c1c2c(ccs2)ncn1 GK03311 Cn1c(ccn1)NC(=O)Nc2cccc(c2)Cl GK03313 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl GK03318 Cc1cccc(c1)C2=N/C(=C/c3cccc(c3)[N+](=O)[O-])/C(=O)O2 PHG00650 Cc1cccc(c1)C2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)O2 PHG00654 c1nc(c2c3c(sc2n1)CCCC3)NCCCN4CCOCC4 GK03364 CCN(CC)c1c2c3c(sc2ncn1)CCCC3 GK03363 COC(=O)c1ccccc1NC(=O)c2ccccc2Cl GK03366 Cc1cc(ccc1S(=O)(=O)Nc2ccnn2C)Br GK03367 c1cc(oc1)CNC(=S)NNC(=O)c2cc(nc(c2)OCC(F)(F)F)OCC(F)(F)F SPB06654 CC(C)(CO)NC(=S)Nc1cc(ccc1Cl)Cl RDR00439 Cc1cccc(c1C)NC(=S)N/N=C\c2cccc3c2cccc3 RDR00634 COc1ccc(cc1)C(C[N+](=O)[O-])Sc2cccc(c2)N PD00790 COc1ccc(cc1)OCCNC(=O)c2ccc(cc2)OC(F)(F)F SPB08192 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccccc3Cl SP01195 COc1ccc2c(c1)cc([nH]2)C(=O)NCc3ccccc3 SP01230 COc1ccc(cc1)Oc2c(cccn2)NS(=O)(=O)c3ccc(cc3)Cl RH01994 c1ccc(c(c1)NC(=S)NCCNC(=S)Nc2ccccc2Cl)Cl RDR00652 c1ccc(c(c1)/C=N/NC(=O)N)Cl RDR00524 Cc1cc(on1)NC(=O)Nc2c(c(cs2)S(=O)(=O)c3ccc(cc3)Cl)C KM01767 CC(C)(C)S(=O)(=O)/C(=C/NN1CCCCC1)/C#N KM02641 c1c(cc(cc1C(F)(F)F)S(=O)(=O)/C(=C/NN2CCOCC2)/C#N)C(F)(F)F KM02644 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccccc3SCc4nc(on4)c5cccs5 SEW06471 CC(C)Cc1ccc(cc1)C(C)C(=O)O/N=C(/c2cccs2)\N SEW06473 CC(C)Cc1ccc(cc1)C(C)C(=O)O/N=C(/c2cccc(c2)Cl)\N SEW06472 CCOc1c(nc(c(c1c2cccc(c2)[N+](=O)[O-])OCC)C)C RJC04019 c1cc(ccc1C#N)S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl HTS01140 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccc(cc3n4cccc4)[N+](=O)[O-])F HTS00284 Cc1c(snn1)C(=O)NN(C)c2cnc3ccccc3n2 SP01278 CN(c1ccc(cn1)[N+](=O)[O-])NC(=O)c2c(cccc2Cl)F SP01290 COC(=O)C1CCc2ccccc2N1.Cl SPB08364 COc1ccc2c(c1)cc([nH]2)C(=O)NCCN3CCCCC3 SP01232 c1ccc(cc1)SCCN(CN2C(=O)c3ccccc3C2=O)CN4C(=O)c5ccccc5C4=O PD00604 c1ccc2c(c1)c(cs2)c3csc(n3)N PD00608 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2cccc(c2)[N+](=O)[O-])c3ccccc3)c4ccccc4)C SP01131 CCOC(=O)c1c(n(c(c1S(=O)(=O)N2CCN(CC2)Cc3ccccc3)c4ccccc4)c5ccccc5)C SP01137 Cn1c(c(c(n1)N)C#N)SC KM02074 COc1ccccc1N2CCN(CC2)CC(=S)N SEW06467 CC(=O)c1ccc(cc1)OCc2cccc(c2)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06468 CCOc1cccc(c1)NC(=O)c2c(oc(n2)C)C(F)(F)F RF04220 Cc1cc(c2ccccc2n1)N3CCN(CC3)CC(=O)c4ccccc4 RH02166 Cc1cc(c2ccccc2n1)N3CCN(CC3)CC(=O)c4ccc(cc4)Cl RH02168 c1ccc(c(c1)/C(=N/O)/Nc2ccccc2Cl)Cl RF05131 CC(C)Cn1c(nnc1S)Cn2c3ccccc3c4c2cccc4 RH01998 Cn1c(ccn1)NS(=O)(=O)c2cccc(c2)Cl GK03353 c1ccc(cc1)COC(=O)N[C@@H](CC(=O)N)C(=O)O SB02036 Cc1cccc(c1)C(=O)Nc2nnc(s2)C(C(C(F)(F)F)(F)F)(F)F SP01390 c1ccc2c(c1)nc(c(n2)NCCO)NCCO RH02243 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)cc[nH]3 SP01378 CCOC(=O)c1c(n(c(c1S(=O)(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F)c4ccc(cc4)Cl)c5ccccc5)C SP01142 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2ccc(cc2)Cl)c3ccc(cc3)Cl)C SP01143 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4ccccc4 HTS00650 c1cc2cccnc2c(c1)S(=O)(=O)NCc3cccs3 HTS00646 COc1ccccc1CNS(=O)(=O)c2cccc3c2nccc3 HTS00643 Cn1c(cc(n1)O)C(=O)N/N=C/c2ccc(cc2)[N+](=O)[O-] JM00220 CC(C)Cc1ccc(cc1)C(C)C(=O)NNC(=O)c2ccc(cc2Cl)Cl SEW06479 c1cc(cc(c1)C#N)CSc2nccc(n2)O JM00411 c1ccc(cc1)c2nc([nH]n2)O JM00247 c1ccc2c(c1)cccc2CN3CCCN(CC3)C(=S)NC4CC4 AW01234 Cc1ccc(cc1)C(=O)Nc2nc(c(s2)C)c3ccc(c(c3)Cl)C HTS00992 Cc1c(c(c(c(c1C)C)CNC(=O)c2ccccc2)C)C CD01127 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(sc2C(=O)N)c3ccccc3 GK03726 c1ccc2c(c1)nnn2CN3CCC(CC3)(c4ccc(cc4)Cl)O HTS00731 CC/C(=C/c1ccc(c(c1)OCc2ccccc2)OC)/[N+](=O)[O-] PD00611 COc1cccc(c1)C(=O)Nc2nnc(s2)C(C(C(F)(F)F)(F)F)(F)F SP01389 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2ccccc2)c3ccc(cc3)Cl)C SP01138 CCOC(=O)c1c(oc(c1S(=O)(=O)NCc2ccccc2)c3ccc(cc3)Cl)C SP01140 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2cccc(c2)C)c3ccc(cc3)Cl)C SP01141 c1cc(ccc1c2nc(on2)CNC(=O)CSCC(=O)O)C(F)(F)F HTS00583 CSC(=N)Nc1ccc(cc1)F.I RDR00489 c1ccc(cc1)c2c(csc2C(F)(F)F)N SEW03133 CCOC(=O)c1cc2c(c(c1)CSc3cccc(c3)C(F)(F)F)OCOC2 SEW03868 CC(C)(C)OC(=O)NCc1nnc(n1C)SCc2c(cccc2Cl)F KM10588 CC(C)(C)OC(=O)NCc1nnc(n1C)SCc2ccc(cc2)C(=O)OC KM10589 c1cc(sc1)c2cc(n3c(n2)cc(n3)c4ccc(cc4)Cl)C(F)(F)F KM10596 c1ccc(cc1)CN2CCN(CC2)c3cccc4c3cc[nH]4.Cl.Cl RH02255 Cc1c(c(c(o1)C)S(=O)(=O)N2CCOCC2)C(=O)OC SP01415 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CCC(=O)NN RJF02208 c1cc(oc1)CNS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01147 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)CC(=O)Nc5ccc(cc5)Br AW01148 CC(=O)c1c(cc(s1)c2ccc(cc2)C(C)(C)C)NC(=O)c3ccc(cc3)Cl GK03524 CCc1ccc(c(c1)CC)OC(=O)c2cc(nn2Cc3ccc(cc3)F)C(C)(C)C SPB08349 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(o3)SCC(=O)Nc4cccc(c4)C(F)(F)F SPB08350 c1cc(ccc1C(=O)CSc2nncn2c3ccc(cc3)C(F)(F)F)F HTS00223 c1cc(ccc1/C=N/NC(=O)N)Cl RDR00526 COc1ccc(cc1)C2=C(/C(=C/N3CCCCC3)/N=C2)[N+](=O)[O-] SEW04075 Cc1c(c(n(n1)c2ccccc2)C)c3nnc(o3)c4ccc(cc4)Cl SEW04237 c1cc(cc(c1)NC(=S)N2CCCC2)C(F)(F)F SEW04258 c1ccc(cc1)NC(=O)CSCCS(=O)(=O)c2ccccc2 KM01724 Cc1nc(nc(n1)SC)N/C=C(\C#N)/C(=O)c2ccco2 KM01105 CCOC(=O)NS(=O)(=O)c1ccccc1Cl KM01664 CC(=O)C(C(=O)C)Sc1nnc(n1C)C(F)(F)F SPB03955 Cc1c(c(c(c(n1)S)C#N)c2cccs2)C(=O)C SPB07034 Cc1nc(nc(n1)OC)N/C=C(\C#N)/C(=O)C2CC2 KM01711 c1ccc(cc1)CN2CCC(CC2)Nc3c4c(ccs4)ncn3 GK03288 c1ccc(c(c1)NC(=O)CCCC(=O)O)SCc2nc(on2)c3cccs3 SEW06424 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)Nc3ccc(cc3F)I KM11063 Cc1ccc(cc1)Sc2c(cccn2)n3c(ccc3C)C RH02103 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3cc(oc3C(F)(F)F)c4ccc(cc4)C(F)(F)F HTS01354 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS01359 c1ccc(c(c1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4F)F KM09716 Cc1cc(no1)N(Cc2ccc(cc2)Cl)C(=O)c3ccc(cc3)Cl RF03234 Cc1c(c(n(n1)C(C)(C)C)C)/C=N/OC(=O)Nc2cccc(c2)C(F)(F)F CD07444 c1cc(c(c(c1)Cl)C#N)NC2CCSC2 CD10423 COC(c1c(cnn1c2c(cc(cc2Cl)Cl)Cl)C(=O)OC)OC SPB04910 COc1ccccc1N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00463 c1cc(ccc1C(F)(F)F)NC(=O)c2ccc3c(c2)nns3 KM10600 COc1cc(cc(c1)OC)NC(=O)c2ccc3c(c2)nns3 KM10601 Cc1nc(cs1)c2ccc(s2)/C(=N/O)/N KM02732 Cc1cc(no1)NCc2cccc(c2Cl)Cl RF03210 CC(=O)OCC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F RF03375 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3ccccc3F HTS00930 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2N SPB07539 CN(C)CCCNc1ccc(c(c1C#N)N2CCOCC2)[N+](=O)[O-] CD07398 CC(C)(C)C(=O)Nc1cc(c(cc1C(=O)O)OC)OC GK03479 CC(C)(C)c1ccc(cc1)c2nc(cs2)C34CC5CC(C3)CC(C5)C4 SPB08313 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11062 CCOC(=O)CSc1c(c(nc(n1)c2ccccc2OC)C)C(=O)C SPB05495 CCOC(=O)c1c(c2c(nc(nc2s1)c3ccccc3OC)C)C SPB05496 c1cc(oc1)/C=N/OCCS(=O)(=O)c2ccc(cc2)Cl KM00960 COc1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4Cl KM10622 c1c(cc(c2c1[nH]c(c2CCC(=O)O)C(=O)O)Cl)Cl SEW06645 CCOC(=O)c1ccc(c(c1)OCCOC)OCCOC GK03508 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C#N GK03375 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4cccc5c4nccc5 HTS00660 Cc1c(c(n(n1)C(C)(C)C)C)/C=N/OC(=O)Nc2ccc(c(c2)Cl)Cl CD07457 CC(=O)Oc1c(cc(cc1Br)/C=C(\C#N)/C(=O)OC)OC RH02197 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)N3CCN(CC3)c4ccnc5c4ccc(c5)Cl KM11070 CS(=O)(=O)Nc1ccc2c(c1)c(c[nH]2)C#N SP01397 c1c(cc(c(c1Cl)C(=O)O)Cl)C(=O)O SEW04506 COc1ccc(cc1)C(=O)NCCSCc2ccc(cc2)F SEW06617 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])Sc3ccc(cc3)C(F)(F)F RH02091 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)NN3CCCCC3)Cl SPB02097 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3c(cccc3Cl)F PD00818 COc1ccc(cc1)Cn2c-3c(c4ccccc4c2=O)C(=O)c5c3cccc5 PD00732 Cc1cccc(c1)C2=N/C(=C/c3ccc(c(c3)Cl)Cl)/C(=O)O2 PHG00664 c1csc2c1ncnc2NCCCN3CCOCC3 GK03291 c1ccc(c(c1)/C=N/Nc2cc(ccc2Cl)Cl)C(=O)O PD00581 c1cc(cc(c1)NC(=O)NC(=O)c2csc(n2)c3ccc(cc3Cl)C(F)(F)F)C(F)(F)F SEW01979 Cn1c(nnc1SCC(=O)c2ccc(cc2)F)CSc3ccnc4c3ccc(c4)Cl HTS00156 c1cnc(cn1)c2ncc(c(n2)N)C#N HTS00174 CN(C)c1ccc(cc1)n2c(nnn2)SCc3ccc(c(c3)Cl)Cl HTS00698 c1cc2c(ccnc2cc1Cl)N3CCN(CC3)C(=O)C4CCCCC4 KM11066 Cc1c(c(c(o1)C)S(=O)(=O)NCc2ccco2)C(=O)OC SP01408 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nnc(s3)NC(=O)c4ccco4 SP01409 Cc1cccc(c1)C2=N/C(=C/c3ccc(cc3)OC)/C(=O)O2 PHG00652 c1ccc(c(c1)C(=O)Nc2cccnc2Sc3ccc(cc3)Cl)Cl RH02096 c1cc(c(nc1)Sc2ccc(cc2)Cl)NC(=O)C3CC3 RH02097 Cc1c(c(n[nH]1)C)Oc2ccc(cc2)Cl SPB03996 CC(=O)/C(=N\Nc1ccc(cc1)C(F)(F)F)/C(=O)c2ccccc2 SPB04010 c1cc(c(cc1S(=O)(=O)NN)Cl)Cl SPB07955 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2Cl)Cl SPB07973 CN(CCO)c1nc2cc(ccc2s1)Cl TG00093 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)C(F)(F)F SPB04108 c1cc(ccc1c2csc(n2)CO)[N+](=O)[O-] RF03095 c1ccc(cc1)c2cc(c(s2)C(=O)N)NC(=O)c3cccs3 GK03729 c1ccc(cc1)SCC(CN2CCC(CC2)C(=O)N)O HTS00808 Cc1c(snn1)C(=O)Nc2ccccc2SCc3nc(on3)c4cccs4 SEW06425 Cn1c(nnc1SCC(=O)NNC(=O)c2c(cccc2Cl)F)Cc3ccsc3 SPB02395 Cc1nc(cs1)C(=O)NNC(=S)NC SPB02302 CCCc1ccc(cc1)C(=O)Nc2ccc(c(c2)C(=O)OC)N3CCOCC3 HTS01360 COC(c1ccnc(n1)SCc2ccccc2Cl)OC SPB04194 c1cc(c(cc1c2csc(n2)CO)Cl)Cl RF03063 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)C(=O)c4cccs4 GK03758 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2C4CCN(CC4)Cc5ccccc5)C(=O)O PD00736 Cc1ccc(cc1)CSC(=N)N.Cl S01709 COc1ccc(cc1Br)/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PHG00632 c1ccc2c(c1)C(=O)N(C2=O)c3ccc4c(c3)c(c[nH]4)C#N SP01404 CC1CCC(/C(=N/NC(=O)CC#N)/C1)C(C)C DP00093 c1ccnc(c1)CNC(=O)c2ccc(cc2)[N+](=O)[O-] DP01792 Cc1c(cccc1Cl)S(=O)(=O)Nc2ccnn2C GK03325 COc1ccc(cc1OCc2ccccc2)/C=C/3\C(=O)OC(=N3)c4ccccc4 PD00586 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4c(nccn4)C(=O)O HTS01070 Cc1c(sc(n1)COc2ccc(cc2)C3SCCS3)C(=O)NN SPB01947 Cc1c(n(c(c1S(=O)(=O)c2ccccc2)N)CCc3ccncc3)C SPB02266 CCOC(=O)/C(=C/Nc1ccc(cc1Br)F)/C#N RH02252 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)C(=O)Nc4ccccc4 GK03761 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2csc(n2)CO RF03118 CSc1nc(nc(n1)SCC2=C(N3C(C(C3=O)NC(=O)Cc4ccccc4)SC2)C(=O)O)N RF03184 Cc1c(cccc1Cl)NC(=S)N2CCCCC2CCN3CCCCC3 BTB01749 c1ccc2cc(ccc2c1)C3=NOC(C3)(C(F)(F)F)O SP01379 Cc1ccc(cc1)C(=O)NNC(=O)c2c3c(sc2n4c(ccc4C)C)CCCC3 GK03322 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3ccccc3Cl HTS00921 c1cc(c(cc1Cl)Cl)OCCC#N SEW04636 Cc1c(sc(n1)c2ccc(s2)c3cccs3)C(=O)C SEW04843 Cn1c(ccc1S(=O)(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O)C(=O)OC HTS01078 Cc1c(c(on1)c2cc(cc(c2)Cl)Cl)C(=O)OC SPB02359 CC1CC(CC(C1)(C)C)NC(=S)N/N=C/c2ccc(c(c2)OCc3ccccc3)OC PD00820 Cc1c(cnn1c2ccccc2)c3ccnn3C(=O)c4ccco4 SP01325 COc1ccc(c(n1)N2CCOCC2)[N+](=O)[O-] PD00792 c1cc(ccc1C(=O)CSc2nc3cc(ccc3o2)Cl)F HTS01255 Cc1cc(cc2c1c(cc(=O)o2)C)OC(=O)c3ccccc3Cl RDR01470 CCN(CC)CC(COc1cc(ccn1)C(F)(F)F)O HAN00201 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Nc3ccc(c(c3)C(=O)OC)N4CCOCC4 HTS00926 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Nc3ccc(c(c3)OC4CCCC4)OC HTS01366 CC(=O)Nc1nc2cc(c(cc2c(=O)s1)OC)OC HTS01604 c1ccc(cc1)C(=O)Oc2cc(=O)n(c3c2cccc3)c4ccccc4 JFD03990 Cc1ccc(c2c1CCC2)Oc3ccc(cn3)C(F)(F)F BTB09400 c1cc(ccc1NC(=O)n2c(ccn2)c3ccc(cc3Cl)[N+](=O)[O-])Cl MWP00485 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2c(cc(o2)c3ccccc3)C#N HTS01248 c1ccc2c(c1)cc(o2)C(=O)CSc3nc4cc(ccc4o3)Cl HTS01256 Cc1ccc(cc1Cl)S(=O)(=O)Nc2cc(sc2C(=O)C)c3ccccc3 GK03753 CC1(OC(=O)C(C(=O)O1)Cc2ccc(c(c2Cl)OC)OC)C RH02249 c1ccc2cc(ccc2c1)c3cc(n4c(n3)cc(n4)c5ccco5)C(F)(F)F KM10594 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3c(cccc3Cl)Cl HTS00929 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc(c(c3)C(=O)OC)N4CCOCC4 HTS00927 c1ccc(cc1)n2c(c(cn2)C(=O)N3CCN(CC3)c4ccnc5c4ccc(c5)Cl)C(F)(F)F KM11073 c1cc(ccc1Nc2ccnc3c2ccc(c3)Cl)OC(F)(F)F KM11074 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)C(=O)c3cccs3)C(=O)OC HTS01541 COCCOc1cc2c(cc1OCCOC)ncnc2N3CCC(CC3)C(=O)O HTS00373 Cc1nc(cn1CC(c2ccc(cc2)OC)O)[N+](=O)[O-] RH02184 c1ccc2cc(ccc2c1)C(=O)N3CCN(CC3)c4ccnc5c4ccc(c5)Cl KM11083 c1cc2c(ccnc2cc1Cl)N3CCN(CC3)C(=O)c4cc(cc(c4)Cl)Cl KM11091 Cc1c(snn1)C(=O)Nc2c3c(cccc3F)n(n2)C SP01319 c1cc(sc1)c2cc(c(c(n2)OCC(=O)c3ccc(cc3)Cl)C#N)C(F)(F)F RH02189 c1ccc(cc1)CN2CC(OCC2)CN3CCN(CC3)c4ncc(cc4)C(F)(F)F.C(=C/C(=O)O)\C(=O)O.C(=C/C(=O)O)\C(=O)O HTS01388 Cc1c(nc(nn1)SC)O SPB01522 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C(/c3cc(c(c(c3)Br)OC)Br)\N SPB00198 CNC(=S)N(Cc1cccnc1)Cc2cccc(c2Cl)Cl RF03338 c1cc(c(c(c1)Cl)CSc2nc(cc(n2)O)N)Cl GK03672 c1cc(ccc1S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl)Br KM11076 CCOC(=O)C1CCN(CC1)c2c3c(c(cs3)C)ncn2 HTS00362 CC(C)(C)c1cc2c(s1)c(ncn2)N3CCN(CC3)C(=O)c4ccc(c(c4)OC)OC GK03640 CC(C)(C)c1cc2c(s1)c(ncn2)NNC(=O)c3ccc(c(c3)OC)OC GK03664 c1cc(cc(c1)NC(=S)NNS(=O)(=O)c2ccc(cc2)Cl)C(F)(F)F RDR00708 CC(=O)Oc1ccccc1/C(=C/C=C(c2ccccc2)c3ccccc3)/N4CCCCC4 RF01255 Cc1c(ccc(n1)C(F)(F)F)C(=O)N2CCN=C(C=C2)C(F)(F)F HTS01563 c1cc(c(c(c1)Cl)C2=N/C(=C/c3ccc(c(c3)Cl)Cl)/C(=O)O2)Cl RDR00698 CC(C)(C)OC(=O)Nc1ccc(cc1C(=O)O)Br SPB08275 c1cc2c(cc1/N=C\3/N4CCCCC4CS3)OCO2 HTS00189 c1ccc(cc1)C(=O)Nc2nc3ccccc3c(=O)s2 HTS01336 CCOC(=O)C(c1ccc(cc1)OCc2ccccc2)C(=O)OCC KM10096 CSc1nc2ccc(cc2s1)NC(=O)c3ccc4c(c3)nns4 KM10780 CC(C)(C)c1cc(n(n1)c2cc(ccc2Cl)Cl)C(C)(C)C SEW06605 CNC(=S)NCc1cccnc1 RDR00588 CN(C)c1ccc(cc1)/C=N/NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl RDR00607 c1ccc2c(c1)c(=O)[nH]c(n2)SCc3cccc(c3)F PD00040 C/C=C/C(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl KM11095 COc1ccc(cc1)C(=O)COc2c(c(cc(n2)c3ccccc3)C(F)(F)F)C#N RH02191 c1ccc(cc1)c2cnc(o2)c3ccccc3C(F)(F)F SPB01766 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)Cc3ccccc3)C(=O)OC HTS01539 Cn1c(ccc1S(=O)(=O)NCc2ccccn2)C(=O)OC HTS01542 c1cc(ccc1C2OCCO2)/C(=N/O)/N KM01110 COc1ccc(cc1)C(=O)N=S2CCN(CC2)C(=O)c3ccc(cc3)Cl KM06139 CS(=N/C=C(\C#N)/S(=O)(=O)c1ccc(cn1)C(F)(F)F)(=O)c2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-] KM06758 CSc1nc2ccc(cc2s1)NC(=O)c3ccccc3C(F)(F)F KM10777 CSc1nc2ccc(cc2s1)NC(=O)c3cccs3 KM10778 Cc1c(snn1)C(=O)NN(C)c2ccc(cn2)[N+](=O)[O-] SP01288 c1ccc(cc1)C2=N/C(=C/c3ccc(c(c3)[N+](=O)[O-])Oc4c(c(c(c(c4Cl)Cl)Cl)Cl)Cl)/C(=O)O2 RDR00621 c1ccc(cc1)c2nc(nc(n2)O)c3ccccc3 RF01839 CN(C)C(=O)Oc1nnc(n1c2cccc(c2)Cl)SCc3ccc(cc3Cl)Cl SPB00585 c1ccc2c(c1)c(no2)CC(=O)O KM10833 CCOC(=O)c1c2c(sc1N)CN(CC2)C AW01200 Cc1c(sc(n1)c2ccc(cc2)Cl)C(C)O RH02169 COc1ccc(cc1)c2ccnc(n2)SCc3ccccc3 KM10764 c1cc(sc1)C(=O)Nc2nc3ccsc3c(=O)s2 HTS01345 COc1cc2c(cc1OC)nc(sc2=O)NC(=O)c3cccs3 HTS01348 Cn1c2c(cn1)c(=O)sc(n2)NC(=O)c3ccccc3 HTS01338 Cc1cc(c2cc([nH]c2c1)C(=O)Nc3ccccc3Cl)C SP01190 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)N(C)c4ccccc4 RH02181 CCCCNC(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl HTS01153 Cc1ccc(c(c1)[N+](=O)[O-])n2cccc2/C=C(\C#N)/S(=O)(=O)C SEW06610 c1cc(sc1)C(=O)Nc2ccc3c(c2)CS(=O)(=O)C3 KM10786 Cn1c(=O)c(nn(c1=S)C)c2ccc(c(c2)Cl)Cl SPB07806 CC(C)n1c(nnc1SC(C)C)O SPB01458 Cn1c(cc(n1)O)C(=O)N/N=C/c2ccc(cc2)Cl JM00219 Cn1c(cc(n1)O)C(=O)N/N=C/c2ccccc2 JM00218 Cn1c(nc(n1)c2ccccc2)O JM00241 c1cc(ncc1C(F)(F)F)N2CCN(CC2)S(=O)(=O)c3ccsc3C(=O)O HTS00471 c1csc(c1S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(=O)O HTS00470 COc1ccc(cc1OC2CCCC2)NC(=O)C3CC3 HTS00323 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2nc3ccsc3c(=O)s2 HTS01618 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2nc3cc(c(cc3c(=O)s2)OC)OC HTS01651 Cc1c(cc(o1)S(=O)(=O)Nc2cccc(c2)c3cnco3)C(=O)OC HTS00155 c1cc(ccc1C(=O)CSc2nnnn2c3ccc(cc3)O)F HTS00798 CC(=O)c1ccc(cc1)OCC(CN2CCN(CC2)C(c3ccccc3)c4ccccc4)O HTS00800 Cc1c(c(c(o1)C)S(=O)(=O)NN(C)c2ccc(cn2)[N+](=O)[O-])C(=O)OC SP01300 c1cc(ccc1c2csc(n2)Nc3ccncc3)Br SEW06612 c1cc2c(cc1Cl)nc([nH]2)C(C(c3[nH]c4ccc(cc4n3)Cl)O)O SPB07799 Cc1ccc(cc1)C(=O)Nc2c3c(cccc3F)n(n2)C SP01314 Cn1c(cc(n1)O)C(=O)NN JM00213 CN(C)NC(=O)NC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl SPB01191 CCN(CC)c1ccc(cc1[N+](=O)[O-])C#N SPB01194 c1cc(sc1)C(=O)Nc2nc3c(cc(cc3Br)Br)c(=O)s2 HTS01349 c1ccc2c(c1)C(=O)N(C2=O)Cc3nc(no3)c4ccc(cc4)C(F)(F)F KM10767 COc1ccc(cc1)C(C[N+](=O)[O-])Sc2ccc(cc2)N PD00791 Cc1nnc(s1)NC(=O)c2cc(ccc2NC)Cl DP01421 Cc1c(c(c(c(c1C)C)CN)C)C.Cl DP01201 CCOC(=O)/C(=C/c1ccc(c(c1)OCc2ccccc2)OC)/C#N PD00587 Cc1ccccc1S(=O)(=O)Nc2ccnn2C GK03326 Cn1c(ccn1)NS(=O)(=O)c2ccc(cc2)[N+](=O)[O-] GK03327 Cn1c(=O)c(nn(c1=S)C)c2ccc3ccccc3c2 SPB07816 Cn1c2cccc(c2c(n1)NC(=O)c3c(nsc3SC)SC)F SP01324 Cc1ccc(cc1)c2nnn(n2)CC(=O)NNS(=O)(=O)c3ccccc3 GK03483 Cc1cc(c(c(c1)C)SCCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C SEW06487 c1ccc(c(c1)NC(=O)COCC(=O)O)SCc2nc(on2)c3cccs3 SEW06488 Cc1nc(cs1)c2nc(cs2)c3ccc(s3)Cl HTS00040 c1cc(cc(c1)OC(F)(F)F)C(=O)NCCS(=O)(=O)Cc2ccc(cc2)F SEW06624 c1cc(c(c(c1)Cl)C(=O)NCCS(=O)(=O)Cc2ccc(cc2)F)F SEW06625 COc1ccc(cc1)C(=O)NCCS(=O)(=O)Cc2ccc(cc2)F SEW06626 Cn1cccc1CN(Cc2ccc(cc2)OC)S(=O)(=O)c3ccc(cc3)F HTS00338 c1ccc2c(c1)cc(o2)c3csc(n3)c4cccs4 HTS01586 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)Nc2ccc(cc2F)F HTS00059 c1cc(cc(c1)S(=O)(=O)Oc2c(cccn2)C(F)(F)F)F SPB08432 c1cc(c(nc1)OS(=O)(=O)c2ccc(cc2)C(F)(F)F)C(F)(F)F SPB08433 C=CCNc1c2c3c(sc2ncn1)CCCC3 GK03332 Cn1c(=O)c(nn(c1=S)C)c2cccc(c2)C3OCCO3 SPB07829 Cn1c2cccc(c2c(n1)NC(=O)c3c(cccc3Cl)F)F SP01320 Cn1c2cccc(c2c(n1)NC(=O)c3cccc(c3)OC)F SP01321 CN1CCN(CC1)c2c3c4c(sc3ncn2)CCCC4 GK03372 CCn1c(cc(n1)C)/C(=N/OC(=O)c2cc(cc(c2)Cl)Cl)/N SPB01883 c1cc(c(cc1CO)[N+](=O)[O-])Oc2cc(cc(c2)Cl)Cl SPB01952 c1ccnc(c1)C(=O)CC(=O)c2ccccn2 RH02194 COc1ccccc1C2C(CC(=O)O2)C(=O)Oc3c(cc(cc3Cl)F)Cl BTB09439 CCOc1c(cc(cn1)NC(=O)OCC#C)C(F)(F)F RF05275 CC(C)Sc1nnc(n1c2ccccc2)O SPB00864 c1cc(ccc1C2=NCCS2)OC(=O)c3ccc(cc3)Cl SPB01400 CC(C)(C)c1ccc(cc1)NC(=O)Cc2cc(cc(c2)F)F SEW06430 c1cc(c(c(c1)Cl)C(=O)Nc2ccc(cc2)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F)F SEW06431 COc1ccc(cc1)C2c3ccsc3CCN2C(=O)Nc4cc(cc(c4)Cl)Cl SEW06420 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)C(=S)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F GK03781 CC(C)Cc1ccc(cc1)C(C)c2nc(cs2)c3ccc(cc3)[N+](=O)[O-] SEW06619 COc1ccc(cc1)C(=O)NCCCCN2CCN(CC2)c3c(cccn3)C(F)(F)F SEW06484 c1cc(n(c1)CCCn2ccnc2)C=C(C#N)C#N SEW04456 c1ccc2c(c1)C(=O)N(C2=O)c3ccc(cc3)n4c(cc(n4)C(F)(F)F)C(F)(F)F SEW04525 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)OC(F)(F)F)F SPB03440 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)OC(F)(F)F)C(F)(F)F SPB03522 Cn1c(cc(=O)n(c1=O)C)NC2CCN(CC2)Cc3ccccc3 PD00816 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)C(=O)Nc4ccc(cc4)F GK03763 Cc1ccc(c(c1)NC(=S)NC(=O)c2ccccc2)n3cccc3 SEW06490 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl)C(F)(F)F HTS01450 c1ccnc(c1)CNS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01158 Cc1cc2nc(cc(n2n1)C)C(F)(F)F KM02422 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COC(=O)c3cccnc3)O RJC03294 Cc1cc(c2ccccc2n1)Nc3ccc(cc3)OC(F)(F)F KM11110 c1ccc(cc1)CC(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F KM11111 Cc1c(cco1)C(=O)/C(=C/N=S(=O)(C)c2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-])/C#N KM06770 c1ccc(c(c1)Nc2ccnc3c2ccc(c3)Cl)Cl KM11071 c1nc(c2c3c(sc2n1)CCCC3)N4CCCC4 GK03374 CN(C)/C=C(/C(=O)c1ccc2c(c1)OCCO2)\Sc3ccc(cc3)Cl SPB08300 c1cc(sc1)c2nc(sn2)N3CCN(CC3)C(=O)c4ccc(cc4)OC(F)(F)F SPB08310 Cc1ccc(cc1F)NC(=S)N(C)C RJF00535 CC(C)(C)C(=O)CSc1nnnn1c2ccc(cc2)N(C)C HTS00699 c1cc(ccc1c2nc(cs2)c3ccc(s3)Cl)Oc4ccc(cn4)C(F)(F)F HTS00033 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4ccc(cc4)Cl HTS00654 c1cc(cc(c1)Cl)C(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS00678 COc1cccc(c1)c2c(c([nH]n2)SC)C#N KM00803 Cc1c(c(on1)c2c(cccc2Cl)F)C(=O)NCCOc3ccc(cc3)OC SPB08196 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C(=O)C3CCC3C(=O)O HTS00262 CC(C)(CC(=O)N1CCN(CC1)c2nc3ccc(cc3s2)Cl)CC(=O)O HTS01133 Cc1cc(no1)C(=O)Nc2cc(cc(c2)Cl)Cl SPB03612 Cc1ccc2c(c1)nc([nH]2)SCC(=O)N3CCN(CC3)c4ccccc4 HTS01207 c1cc2c(cc1F)nc([nH]2)C(C(c3[nH]c4ccc(cc4n3)F)O)O SPB07800 c1cc2c(cc1Cl)sc(n2)N3CCN(CC3)CC#N SPB07564 COc1ccc(cc1)C2C(c3ccccc3C(=O)N2Cc4ccc(cc4)Cl)C(=O)O PD00735 CC(=O)Nc1cscc1S(=O)(=O)c2ccccc2 KM01794 CCCc1ccc(cc1)S(=O)(=O)NNC(=O)c2ccc(cc2)n3c(ccc3C)C RH01961 CCS(=O)(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl KM11068 c1cc2c(ccnc2cc1Cl)N3CCN(CC3)S(=O)(=O)c4ccc(s4)Br KM11069 CC(C)(C)NC(=O)c1cc(ccc1NC)Cl DP01666 Cc1ccccc1NC(=O)c2ccc3c(c2)nns3 KM10599 c1cc(c(c(c1)Cl)Cl)n2cc(nn2)COC(=O)c3c(cccc3F)F SEW04504 COc1cc(cc(c1OC)OC)C2C(c3ccccc3C(=O)N2Cc4ccc(cc4)F)C(=O)O PD00688 CCOc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)C PHG00660 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N)CC(=O)O RJC03311 COC(=O)CSc1c2c(ccs2)ncn1 GK03289 c1csc2c1ncnc2NCCCn3ccnc3 GK03290 Cc1cc(ccc1NC(=O)OC(C)(C)C)Br SPB08149 Cc1c(c(no1)c2ccccc2)c3nc(no3)CSc4ccc(cn4)C(F)(F)F SEW06649 Cc1cc(cc(c1)NC(=S)N2CCc3c(ccs3)C2c4ccc(cc4)OC)C SEW06403 COc1ccc(cc1)C2c3ccsc3CCN2C(=S)Nc4ccc(cc4)OC(F)(F)F SEW06404 CN(C)c1ccc(cc1)n2c(nnn2)SCc3ccc(cc3)OC(F)(F)F HTS00696 CS(=O)(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl KM11061 Cc1ccc(cc1Cl)Nc2cc(nn2C)O JM00146 CC(C)NC(=O)N(Cc1cccc(c1Cl)Cl)Cc2cccs2 RF03396 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)O SPB03031 COc1cc2c(cc1OC)ncnc2N3CCCC3 GK03373 COc1cccc(c1)n2c(=O)c3ccccc3[nH]c2=S SEW04475 Cc1ccc(cc1)Sc2c(cccn2)NS(=O)(=O)c3ccc(cc3)C(C)C RH02095 CCCc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH01967 c1ccc(c(c1)C(=O)Nc2cccnc2Oc3ccc(cc3)Cl)Cl RH01968 CC(C(=O)Nc1cc(cc(c1)Cl)Cl)N2CCCC2 SEW04560 Cc1c(c(c(o1)C)S(=O)(=O)NCc2ccc(cc2Cl)Cl)C(=O)OC HTS01167 CSCc1nnc(o1)c2cccc(c2)[N+](=O)[O-] SEW06644 c1cc(ccc1C#N)OC(=O)c2ccc(o2)Br JFD03980 CC(=O)c1ccc(cc1)OC(=O)Cc2cc(cc(c2)F)F SEW06405 c1cc(oc1)CNC(=O)Cc2cc(cc(c2)F)F SEW06406 Cc1ccc(c(c1)NC(=O)c2cccc(c2)C(F)(F)F)n3cccc3 SEW06407 C=CCn1c(nnc1S)c2ccc3c(c2)cccn3 KM10631 Cc1c(c(on1)C)c2c(c(no2)C)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F SPB02418 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)O)Oc3ccc(cc3)OC SPB04150 Cn1c(ccn1)NC(=O)c2c(cccc2OC)OC GK03320 Cn1c(ccn1)NS(=O)(=O)c2ccc(cc2)F GK03323 CCCCNc1nc(cs1)c2cc(cc(c2OC)Cl)Cl RDR02044 c1ccc(cc1)CN2CCC(CC2)Nc3c4c(csc4ncn3)c5ccccc5 AW00944 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCCCCO SPB08212 c1ccc2c(c1)-c3ccccc3C2COC(=O)NCCCCCCO SPB08213 Cc1c(c(c(o1)C)S(=O)(=O)NCc2cccs2)C(=O)OC SP01412 COc1ccccc1N2CCN(CC2)CC#N SEW06412 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2cc(n(c2)C)C(=O)OC SEW06413 c1cc2c(ccnc2cc1Cl)Nc3ccc(cc3F)I KM11072 COc1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc(c(c3)C(=O)OC)N4CCOCC4 HTS01352 Cc1c(c(=O)[nH]c(=S)[nH]1)Oc2ccccc2 SPB04136 Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc(cc3)Cl SPB03011 c1ccnc(c1)S(=O)(=O)Cc2nc(cs2)C(=O)NN SPB02238 Cc1ccc(c(c1)C)NC(=O)c2ccc(o2)Br JFD03982 c1cc(sc1)c2nc(no2)N3CCCCC3 KM10804 CCOC(=O)/C(=C/Nc1ccccc1OC(F)(F)F)/C#N RH02236 c1ccc2c(c1)cccc2C(=O)Nc3cccnc3Sc4ccc(cc4)Cl RH02117 Cn1cc(cc1C(=O)OC)/C=N/NC(=S)N SEW06414 c1ccc2c(c1)c(c[nH]2)C(c3ccccn3)O HTS01389 c1cc(ccc1c2nc(on2)CNC(=O)Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F HTS01222 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3cc(oc3C(F)(F)F)c4ccccc4Cl HTS01353 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(c(c3)C(=O)OC)N4CCOCC4 HTS01357 CC(C)(C)OC(=O)NCc1nnc(n1C)SCc2c(cccc2Cl)Cl KM10587 c1c(c(sc1Br)Br)CC(=O)N SPB02305 CNC(=S)NNC(=O)Cc1ccsc1 SPB02358 CSc1nc(n(n1)c2cc(cc(c2)Cl)Cl)N JM00004 Cc1c(c(c(o1)C)S(=O)(=O)N2CCCCC2)C(=O)OC SP01406 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2nc3cc(ccc3o2)Cl HTS01257 CC(C)(C)c1csc(n1)NNC(=O)c2ccc(cc2)Cl HTS01570 c1cnc(c(n1)C(=O)N2CCCCCC2)C(=O)O HTS01068 Cc1cc(cc2c1c(cc(=O)o2)C)OC(=O)c3ccc(cc3)Cl RDR01469 CC(C)(C)OC(=O)NCc1nnc(n1C)SCc2cc(cc(c2)F)F KM10590 CC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccc(c(c3)OC)OC GK03751 CC(C)c1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)C(=O)OC)N3CCOCC3 HTS01362 CCOC(=O)c1c(nc(s1)COc2ccccc2OC)C SPB08301 CSc1nc(n(n1)c2ccccc2)N JM00001 COc1ccc(cc1)CN(Cc2ccc(cc2)OC)S(=O)(=O)c3ccc(c(c3)Cl)Cl SEW04967 Cc1c2ccccc2sc1C3=NNC(C3)(C(F)(F)F)O SP01376 Cc1nc(cs1)c2nc(cc(n2)O)COC SPB03571 CCOC(=O)c1c[nH]c2cc(nn2c1=O)C3CC3 KM00819 Cc1cc(c2ccccc2n1)N3CCN(CC3)C(=O)Nc4ccc(cc4F)F HTS01445 c1cc2c(cc1CNC(=O)CC34CC5CC(C3)CC(C5)C4)OCO2 HTS01100 c1ccc(cc1)C(CNCc2ccc(cc2)F)O HTS00621 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)CCO)C(=O)OC HTS01076 CNC(=S)N(Cc1ccc(cc1)Cl)Cc2cccs2 RF03339 C=CCn1c(nnc1SCC(=O)NCc2ccccc2)c3ccc4c(c3)cccn4 KM10655 Cc1ccc(c(c1)C)Nc2ccnc3c2ccc(c3)Cl KM11081 Cc1ccc(cc1)C(=O)Nc2cc(ccc2Oc3ccc(cc3)OC)C(F)(F)F HTS00851 COc1ccc(cc1)Oc2ccc(c(c2)NC(=O)C3CCC3C(=O)O)C(F)(F)F HTS00259 COc1ccc(cc1)C(=O)COc2c(c(cc(n2)c3cccs3)C(F)(F)F)C#N RH02188 CC(C)(C)c1cc2c(s1)c(ncn2)NNC(=O)c3cccs3 GK03671 c1cc(ccc1C(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O)F HTS01393 c1cc(c(c(c1)Cl)OC(=O)c2ccc(cc2Cl)Cl)Cl RDR01801 Cc1cc(c(c(c1)C)C(=O)Nc2ccc(c(c2)C(=O)OC)N3CCOCC3)C HTS00923 CCOC(=O)CSc1nnc(n1C)c2ccc3c(c2)cccn3 KM10660 C=CCn1c(nnc1SCc2ccc(cc2)Cl)c3ccc4c(c3)cccn4 KM10656 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)C(=O)OC HTS01079 Cn1c(ccc1S(=O)(=O)NCc2ccc3c(c2)OCO3)C(=O)OC HTS01535 c1cc(ccc1NC(=N)NC#N)Cl JM00246 c1cc(c(c(c1)Cl)C#N)n2ccnc2 RF00701 CCOC(=O)c1c(c(nc(c1Cl)C(C)(C)C)O)C#N RF01229 CC(C)(C)C(=O)NC(=O)Nc1ccccc1C(F)(F)F RF01486 c1cc(ncc1[N+](=O)[O-])N2CCN(CC2)C(=O)C3CCC3C(=O)O HTS00263 Cc1c(c(on1)C)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11085 CCn1cc(c(cc1=O)C(F)(F)F)C(=O)N(C)c2ccc(cc2)Cl RF04780 c1ccc2c(c1)cccc2/C=N\NC(=S)Nc3cccc(c3Cl)Cl RDR01025 Cc1c(cccc1Cl)NC(=S)N2C(CCCC2C)C RDR01212 Cc1ccc2c(c1)n(c(=O)o2)C(=O)C RH02170 CC(=O)Nc1ccc(cc1C#N)C(C)(C)C RF01512 c1ccc(cc1)C(CN2CCC(CC2)C(=O)N)O HTS00628 C/C(=N\OC(=O)c1ccccc1Cl)/CS(=O)(=O)c2ccc(cc2)Cl KM01837 Cn1c(nnc1SCc2cccc(c2)/C(=N/OC(=O)c3ccc(cc3)Cl)/N)C(F)(F)F KM03139 CN1CCN(CC1)C(=O)COc2cc(nc3c2cccc3)c4ccccc4.C(=C/C(=O)O)\C(=O)O RH02100 c1cc(ccc1COc2ccc(cc2)c3nc(on3)C4CC4)Cl RF01869 c1cc(ccc1C2=CSC(=C(C#N)C#N)S2)Cl RF01950 c1ccc(c(c1)/C=C/2\C(=O)NC(=S)S2)C(=O)O PD00729 c1ccc2cc(ccc2c1)c3cc(n4c(n3)cc(n4)c5ccc(cc5)Cl)C(F)(F)F KM10597 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)NC(=O)Nc4ccc(cc4)Cl)C(F)(F)F SEW06481 Cc1cc(ccc1Br)NC(=O)c2cc3c(s2)-c4ccccc4CC3 PD00605 CC(=O)Nc1nc2ccccc2c(=O)s1 HTS01603 c1ccc2c(c1)c(=O)[nH]c(n2)c3c(nccn3)C(=O)O HTS01065 c1ccnc(c1)CNc2[nH]nc(n2)N RF02198 c1cc(ccc1C(=O)NCC#N)Cl RF02552 c1ccc2c(c1)c(c(s2)Cl)CC(=O)N3CCCC3 KM07288 c1ccc2c(c1)c(c3ccccc3n2)C(=O)N KM08233 c1ccc(cc1)C#Cc2cc(cnc2)C#N KM08442 Cc1c(nc(s1)NC(=O)C2CCC2C(=O)O)CC(=O)OC HTS00266 COc1ccc(cc1)Oc2ccc(cc2NS(=O)(=O)c3cccs3)C(F)(F)F HTS00255 CCC(=O)N(C)c1nc(cs1)c2ccc(s2)Cl HTS00243 Cn1c2c(cn1)c(ncn2)NNC(=O)CCC(=O)O GK03521 CCOC(=O)c1cnn(c1N)c2c3cnn(c3ncn2)C GK03523 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/OC(=O)Nc3c(cccc3Cl)Cl RF01903 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)SC RH02172 c1cc2c(cc1CNC(=O)c3ccc(c(c3)Cl)Cl)CCO2 SP01303 c1cc(c(cc1F)Cl)C/C(=N/O)/N TL01010 c1cscc1Cc2nnc(o2)S SPB02523 CC(C)(C)C(=O)OC/C(=N/OC(=O)c1ccccc1)/N RF02985 C1CCNCC1.C1CCN(CC1)C(=S)S KM03887 c1ccc(cc1)n2cc(c(=O)[nH]c2=O)C#N KM08134 c1cc(ccc1NC(=O)O/N=C(/c2cnn3c2nc(cc3C(F)(F)F)C(F)(F)F)\N)Cl KM03095 Cc1ccc(cc1)/C(=N/OC(=O)c2ccc(o2)C#Cc3ccccc3)/N KM08681 c1cc(c(c(c1)F)/C=N/O)F RF00368 CC1CN(CC(O1)C)c2c3c4c(sc3ncn2)CCCC4 GK03368 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3cccc(c3)Cl GK03371 CCC1CS/C(=N\c2c(cc(cc2C)C)C)/N1 RDR00427 c1ccc2cc(ccc2c1)c3cc(n4c(n3)cc(n4)C5CC5)C(F)(F)F KM10598 c1cc(cnc1)N2C(=O)CC3(CCCCC3)CC2=O PD00730 c1ccc2c(c1)c(=O)n(c(n2)S)CC3CC3 RJF01259 CC(=O)N1CCC(CC1)c2c[nH]c3c2cccc3 RH01995 COc1ccc(cc1)CNC(=O)Nc2ccccc2C#N KM10616 c1cc(c(c(c1)F)c2csc(n2)N)F RF02538 CC(C)Sc1cc(c2cc(ccc2n1)Br)C#N RF01108 CC(C)(C)C(=O)OCC(=O)c1ccc(cc1)C(F)(F)F RF03421 CC(C)CC(C(=O)N/N=C/c1cccs1)NC(=O)Cc2ccsc2 KM02910 Cc1c(c(sc1C(=O)O)SC)C(C)O KM09403 c1cc(ccc1OCC(CN2CCC(CC2)C(=O)N)O)F HTS00693 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(on3)C GK03365 Cc1cc(ccc1NC(=O)NC(=O)c2c(cccc2F)F)/N=N/c3cccc(c3)C(F)(F)F BTB06673 Cc1c(sc(n1)N2CCOCC2)C(=O)C SEW03933 CCOC(=O)NC(=S)NCCC1CCNCC1 NH00418 CCOC(=N)c1ccc(c(c1)Cl)F.Cl RJF00463 c1cc(cc(c1)C(F)(F)F)CSCCN2C(=O)CCC2=O SEW06653 c1ccc2c(c1)C(=O)N(C2=O)CCSCc3cccc(c3)C(F)(F)F SEW06654 CCOC(=N)c1cccc(c1)C(F)(F)F.Cl RJF00590 CCn1c(cc(n1)C)c2nnc(o2)S SPB02756 c1cc(ccc1n2ccc(=O)c(n2)c3cc[nH]n3)F SPB02820 CC(C)(C)OC(=O)Nc1cc(n(c1)C)C(=O)O SPB08449 c1cc(c(cc1F)Cl)CC(=O)N TL01011 c1c(c(sc1Cl)Cl)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F HTS00233 c1ccc2c(c1)cc(o2)C(=O)CSc3nncn3c4ccc(cc4)C(F)(F)F HTS00224 c1cc(c(nc1)Sc2ccc(cc2)Cl)NC(=O)c3ccc(cc3)C(F)(F)F RH02101 Cc1nc(cn1CC=C)[N+](=O)[O-] RH02102 c1cc(ccc1[N+](=O)[O-])S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11059 c1cc(c(cc1Cl)Cl)NC(=O)N2CCC(C(=C2)C(=O)N)C(F)(F)F RF04555 c1ccc(c(c1)c2nnnn2c3ccccc3C(F)(F)F)Cl RF04546 CC(=O)N1C(CC(=N1)c2ccco2)c3ccc(cc3)Br RJC04104 CC(=O)N1C(CC(=N1)c2ccc(cc2)OC)c3ccc(cc3)Cl RJC04106 Cc1ccc(n1c2cc(c(cc2C(=O)NNC(=O)C(C)C)OC)OC)C GK03393 CC(C)(C)OC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl AW00959 CC(=O)CCC(=O)OCC(=O)c1ccc(cc1)C(F)(F)F RF03432 Cc1nc(cn1CC(=O)c2ccc3c(c2)OCCO3)[N+](=O)[O-] HTS01291 c1cc(ccc1Sc2c[nH]nc2c3ccc4c(c3)OCCO4)Cl SPB08304 c1cc(ccc1c2nc(cs2)C34CC5CC(C3)CC(C5)C4)Cl SPB08305 CS(=O)(=O)/C(=C/c1c(ccs1)Cl)/C#N SEW06621 Cc1c2c(c(cnc2n(n1)C)C(=O)O)O KM05117 CSc1c2c(c(s1)C(=S)N)CCCC2=O KM03868 Cc1csc(n1)c2ccc(cc2)c3csnn3 SEW01082 Cc1ccc(c2c1cccc2)S(=O)(=O)Nc3ccc(c(c3)C(=O)OC)N4CCOCC4 HTS01361 c1ccc(cc1)S(=O)(=O)N[C@@H](Cc2ccc(cc2)[N+](=O)[O-])C(=O)O SPB08302 c1cc(c(c(c1)Cl)C(=O)NCCSCc2ccc(cc2)F)F SEW06618 CC(=O)C(Cc1ccc(cc1)[N+](=O)[O-])(Cc2c(cccc2Cl)F)C(=O)C CD07605 CC1=NN=C(C1(CC#C)Cc2c(cccc2Cl)F)C CD07631 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)C(=O)c5c(cccc5Cl)Cl AW01160 c1ccc2c(c1)CCC(=C2)N3CCN(CC3)c4ccc(c(c4)Cl)Cl HTS01275 c1ccc2c(c1)CCC(=C2)N3CCN(CC3)c4cccc(c4)C(F)(F)F HTS01276 CSc1nc(n(n1)c2c(cc(cc2Cl)Cl)Cl)N JM00003 c1cc(sc1C(=S)N)[N+](=O)[O-] RF01687 CC(C)(C)c1ccc(c(c1)Br)NC(=O)NC RF01594 CCOC(=O)/C=C/1\NC(=O)CS1 JP00167 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)c3cc(cc(c3)Cl)Cl GK03537 CC(=O)Nc1cc(sc1C(=O)OC)c2ccc(cc2)C(C)(C)C GK03538 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2c(cc(cc2Br)C(C)C)Br)C SEW06455 CSc1c(c(on1)c2ccc(cc2)Cl)C(=O)NC(=O)Nc3ccccc3Cl KM01576 Cc1cccc(c1/C=N/Nc2ccc(cc2)c3csnn3)Cl SEW00961 CCCSc1c(cccn1)C(=O)NCc2ccc3c(c2)OCO3 PD00694 Cc1cccc(c1NC(=O)c2cnc(cc2C(F)(F)F)NC3CCCCC3)C RF04439 Cc1cccc(c1NC(=O)c2cnc(cc2C(F)(F)F)SCC(=O)OC)C RF04444 c1ccc(cc1)CC2CCN(CC2)S(=O)(=O)c3ccc(cc3)F HTS00835 COc1ccc(cc1)n2c(nnn2)c3c[nH]c4c3cc(cc4)F HTS01272 c1cc(ccc1n2c(nnn2)c3c[nH]c4c3cc(cc4)F)Br HTS01274 Cc1ccc(n1c2ccc(cc2)C(=O)ON3C(=O)CCC3=O)C RH02007 COc1ccc(cc1)NC(=O)c2ccc(o2)S(=O)(=O)N3CCOCC3 HTS00431 c1cc(ccc1NC(=O)O/N=C/2\CCCCC2Cn3ccnc3)Cl KM02531 COC(=O)c1c(ccs1)N/N=C(\C#N)/S(=O)(=O)C KM03703 c1cc(ncc1C(=S)N)n2cncn2 SPB07242 CCOC(=O)CSc1nccc(n1)c2c(nc(s2)c3ccc(cc3)Cl)C RH02262 Cc1cc(no1)C(=O)N[C@@H](C(C)C)C(=O)OC SPB08428 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4)C(=O)OC HTS01077 Cn1c(ccc1S(=O)(=O)NC2Cc3ccccc3C2)C(=O)OC HTS01532 c1cc(cc(c1)N2CCN(CC2)c3nc(cs3)c4ccc(cc4)Cl)C(F)(F)F HTS01261 CC(C)(C)C(=O)Nc1c2c(cccc2F)n(n1)C SP01340 c1ccc(cc1)CN2CCC(CC2)Oc3cc(nc4c3cccc4F)C(F)(F)F KM10661 COc1ccc(cc1)c2ccnc(n2)SCC(=O)N3CCOCC3 KM10776 c1ccc2c(c1)c(=O)c(co2)N3CCN(CC3)S(=O)(=O)c4cccc5c4non5 HTS00152 c1ccc(cc1)CN2CCN(CC2)C(=O)c3cc4c(s3)-c5ccccc5CC4 PD00616 c1ccc(cc1)c2cc(nc(n2)SCC(=O)c3ccc(s3)Cl)O HTS01201 CC(C)(C)C(=O)Nc1ccsc1C(=O)OC HTS00507 CC(C)(C)c1ccc(c(c1)NC(=O)C(Cl)Cl)NC(=O)c2ccco2 RF01740 CS(=NC=C(C#N)C#N)(=O)c1ccc(cc1)Cl KM02952 CC(=O)OC1CCN(CC1)c2cc(nc3c2c(cc(c3)Cl)Cl)C(F)(F)F KM10663 c1ccc(cc1)NC(=O)NC2CCCC2 KM10666 c1cc(sc1)c2nc(no2)CO RF04231 CCOC(Cc1nnc(n1C)S)OCC SPB05196 CCOC(=O)c1cc(c(cc1NS(=O)(=O)c2ccc(cc2)C)OCCOC)OCCOC GK03806 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)NC(Cc2ccc(cc2)[N+](=O)[O-])C(=O)O SPB08316 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)NS(=O)(=O)c4ccccc4 SS00021 c1ccc(cc1)C(C2CCCC2)C(=O)Nc3cccnc3Sc4ccccc4 RH02094 c1ccc2c(c1)C(C3(CCCCC3)N(C2=O)C4CCCCC4)C(=O)O PD00689 c1cc(c(cc1NC(=O)/C=C/C(=O)Nc2ccc(c(c2)Cl)F)Cl)F CD07704 Cc1ccc(cc1)n2c(nnn2)c3cnc(nc3C(F)(F)F)N HTS01264 Cc1ccc(cc1)c2c(cno2)c3nnnn3c4ccc(cc4)Cl HTS01267 c1cc(ccc1C(=O)NNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)OC(F)(F)F HTS00504 Cc1c(c(n(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)C)C(=O)N SEW05009 CC\1=NN(C(=O)/C1=N\Nc2ccccc2)c3c(cc(cc3Cl)C(F)(F)F)Cl SEW05017 CS(=O)(=O)/C(=C/Nc1ccc(cc1)OC(F)(F)F)/C#N KM03580 CCOC(=O)N/N=C(\C)/c1ccc(cc1)[N+](=O)[O-] SEW00751 Cc1c(c(nc(n1)SCC(=O)c2ccccc2)O)Oc3ccc(cc3)Cl SPB03982 CCCCc1ccc(cc1)C(=O)NCCNC(=O)c2ccc(cc2)CCCC HTS00375 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(cc2)OC(F)(F)F HTS00049 c1cc(ccc1NC(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)F BTB06284 Cc1cc(c2ccccc2n1)N3CCN(CC3)CC(=O)Nc4ccc5c(c4)OCCO5.Cl RH02193 CCOc1cc(c(cc1N2CCOCC2)OCC)NS(=O)(=O)CC SS00015 c1cc(c(cc1S(=O)(=O)/C(=C/NCc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl)Cl KM01948 COc1ccc2c(c1)cc([nH]2)C(=O)N3CCCN(CC3)Cc4ccc(cc4)F HTS00779 Cc1ccc(cc1)S(=NC(=O)Nc2ccc(cc2)Cl)(=O)C KM02834 Cc1c(cc(o1)S(=O)(=O)Nc2ccsc2C(=O)OC)C(=O)OC HTS00509 c1cc(c(nc1)NS(=O)(=O)c2ccc(c(c2)F)F)OCc3cc(cc(c3)F)F RH02083 CC1=C(CC(C(C1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl)C(=O)O)C PD00681 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3cccnc3 PD00683 c1ccc(c(c1)c2csc(n2)c3ccc(cc3)Cl)Cl.Br RDR02368 Cc1ccc(n1c2cc(c(cc2C(=O)NNS(=O)(=O)C)OC)OC)C GK03308 CC(=O)Oc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cc(c(c(c3)OC)OC)OC PHG00778 Cn1c(ccc1S(=O)(=O)N2CCC(CC2)O)C(=O)OC HTS01536 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2ccc(n2C)C(=O)OC HTS01538 Cc1csc2c1nc(sc2=O)NC(=O)c3ccc(cc3Cl)F HTS01484 c1cc(sc1)c2nc(cs2)C(=O)NN SPB02133 c1ccc(cc1)OC/C(=N/O)/N SPB02646 c1cc(ccc1c2csc(n2)NNC(=O)c3ccc(cc3)Cl)F HTS00813 c1cc(ccc1S(=O)(=O)CC(=O)NO)Cl KM02107 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)C4CCCCC4)[N+](=O)[O-] HTS00278 CSc1c(c(cs1)c2cccs2)CNC(=O)c3ccccc3Cl KM02202 COC(=O)c1c(ccs1)N/C=C(\C#N)/C(=O)c2cccs2 KM03698 Cn1c(nnc1Sc2c(cccn2)[N+](=O)[O-])Cn3c4ccccc4c5c3cccc5 RH02089 COc1ccc2c(c1)cc([nH]2)C(=O)N3CCCN(CC3)Cc4ccccc4 HTS00775 Cn1c(ccn1)NS(=O)(=O)c2ccc(cc2)OC GK03382 c1ccc2c(c1)cc(o2)C(=O)CSc3nnnn3c4ccc(cc4)O HTS00941 CN(C)c1ccc(cc1)n2c(nnn2)SCC(=O)c3ccc(cc3)F HTS00788 CC(C)(C)C(=O)CC1(c2cc(ccc2NC1=O)Br)O SPB00595 CCOC(=O)/C(=C/c1ccc(cc1)Cl)/[N+](=O)[O-] SPB00667 CC(=O)NC1=NN(C(S1)c2ccccc2)C(=O)C RJC04099 COc1ccc2c(c1)cc([nH]2)C(=O)N3CCCN(CC3)C(=O)c4cccs4 HTS01110 c1ccc(c(c1)C(=O)Oc2ccc(cc2)C3=NCCS3)Cl SPB01401 CS(=NC(=O)Nc1ccccc1)(=O)c2ccccc2 KM02835 Cc1c(cc(o1)S(=O)(=O)Nc2ccsc2C(=O)O)C(=O)O HTS01026 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(CSc4ccc(cc4)F)O HTS00958 Cc1cc(cc(c1OCC(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O)Br)Cl HTS00953 c1c(cc(c(c1Cl)CN)Cl)C(F)(F)F.Cl SEW05112 c1ccc2c(c1)c(c-3c(n2)CSc4c3cc(cc4)Cl)C(=O)O SEW05167 c1ccc2c(c1)C(=C(C2=O)c3cc(cc(c3)Cl)Cl)O SEW05448 Cc1ccc(c(c1)[N+](=O)[O-])n2cccc2C(=O)C(F)(F)F SEW06608 COc1cccc(c1)NC(=O)Nc2ccc(nc2)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06611 Cc1csc2c1c(c(s2)C(=O)CC(=O)C(F)(F)F)C SP01416 COC(=O)c1ccc(o1)S(=O)(=O)NCc2ccco2 SP01417 COC(=O)c1c(ccs1)NS(=O)(=O)c2cc(cc(c2)Cl)Cl HTS01021 CCOC(=O)CSc1c(c(c(s1)C(=O)OCC)c2cccs2)C#N KM03460 Cc1ccc(c2c1cccc2)S(=O)(=O)n3c4cccc(c4c(n3)n5c(ccc5C)C)F HTS01082 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)C SS00011 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl)C#N KM11078 Cc1csc2c1c(ncn2)N3CCC(CC3)C(=O)O HTS00368 CN(C)c1ncc(c(n1)C(F)(F)F)C(=O)Nc2cc(c(cc2C(=O)OC)OC)OC HTS00371 Cc1ccc(cc1)S(=NS(=O)(=O)c2ccc(cc2)OC)(=O)C KM02836 CS(=NS(=O)(=O)c1ccc(cc1)Cl)(=O)c2ccccc2 KM02840 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(COc4ccc(cc4)Cl)O HTS00974 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3cccs3 PD00684 CC1=C(CC2C(C1)C(=O)N(C2=O)c3ccc(cc3)Oc4ccc(cc4)Cl)C PD00686 c1ccc(cc1)c2nc(cs2)C(=O)Nc3cc(cc(c3)Cl)Cl SPB02929 Cc1c(c(on1)c2c(nns2)C)C(=O)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N SPB03416 c1ccc(cc1)c2csc3c2c(ncn3)NCCNc4c(cccn4)C(F)(F)F AW00979 c1cc(ccc1SCc2ccc(cc2Cl)[N+](=O)[O-])Cl SPB01537 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NC(=O)c3c(nccn3)C(=O)O HTS01412 CC(C)(C)n1c(c(c(n1)c2ccc(cc2)Cl)C#N)N SS00047 CC(C)(C)OC(=O)NCC1CCNCC1 SPB08455 Cc1csc2c1nc(sc2=O)NC(=O)c3ccc(cc3)OC(F)(F)F HTS01596 c1c(cc(c2c1nc(cc2N3CCC(CC3)O)C(F)(F)F)Cl)Cl KM10664 c1cc2c(cc(nc2c(c1)F)C(F)(F)F)N3CCN(CC3)CCOC(=O)C(F)(F)F KM10665 c1cc(cc(c1)C(=O)O)CSc2cccs2 KM02425 COc1ccc(c(c1)[N+](=O)[O-])NN=C(C#N)C#N SEW00893 c1ccn2cc(nc2c1)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RDR02796 CC(C)S(=O)(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl KM11077 Cc1c(c(c(o1)C)S(=O)(=O)NC(C)(C)C)C(=O)OC SP01407 CC(C)(C)c1cc2c(s1)c(ncn2)NNC(=O)c3ccco3 GK03670 CCOC(=O)COc1c(c(cc(n1)c2cccs2)C(F)(F)F)C#N RH02185 c1ccc(cc1)c2cc(c(c(=O)n2N)C#N)C(F)(F)F RH02186 COc1ccccc1NC(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS01221 COC(=O)c1ccc(o1)S(=O)(=O)N2CCOCC2 SP01418 CCOC(=O)c1csc(n1)NC(=O)C RH02257 c1c(cc(cc1Cl)Cl)OCc2cc(no2)C(=O)NN SPB01290 CCC(CO)NC(=S)Nc1ccsc1C(=O)OC GK03767 Cn1c(ccn1)NC(=O)c2ccc(c(c2)Cl)Cl GK03341 Cc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2C(=O)O)OC)OC GK03466 Cn1c2c(cn1)c(ncn2)Sc3cccc4c3cccc4 GK03468 COc1cc(c(cc1OC)NS(=O)(=O)c2ccc(cc2)F)C(=O)O GK03467 COc1c(cc(s1)/C=N/O)Br KM01074 Cc1ccc(c(c1)[N+](=O)[O-])OCC(CN2CCN(CC2)c3nc(ns3)c4ccccc4)O HTS01118 Cc1c(nc(s1)NS(=O)(=O)c2ccc(cc2)OC(F)(F)F)CC(=O)OC HTS00842 Cc1c(nc(s1)NC(=O)c2ccccc2)CC(=O)OC HTS00035 CC(=O)c1c(ccs1)NC(=O)CC(C)(C)CC(=O)O HTS00503 c1c(cc(c2c1scc2N)Cl)C(F)(F)F SEW03146 COc1ccc(cc1)OCCC(=O)NN CD01747 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(on3)C GK03321 Cc1ccc(cc1)CSc2ccc(cc2)[N+](=O)[O-] PD00594 c1cc2cccnc2c(c1)Oc3ccc(cc3)NC(=O)c4cccs4 SEW06444 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2ccccc2)C SEW06447 CCCCCCCCCC(=O)n1c2ccc(cc2c3c1nc4ccccc4n3)F RH02009 c1cc(ccc1F)SCCNC(=O)NCCO PD00610 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)OC(F)(F)F)[nH]cn3 KM10607 CC(C(C(=O)O)Nc1ccccc1CC(=O)OC(C)(C)C)O RJC04029 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)NC3CCCCC3 KM11104 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)NCCN3CCOCC3 KM11105 c1ccc2cc(ccc2c1)S(=O)(=O)N3CCN(CC3)c4ccnc5c4ccc(c5)Cl KM11089 c1cnc(cn1)NC(=O)COCC(=O)O PD00793 CCOC(=O)COc1c(c(c(c(n1)C)CC=C)C)C#N RH02187 c1ccc(cc1)C(=O)COc2c(c(cc(n2)c3cccs3)C(F)(F)F)C#N RH02190 c1cc(oc1)C(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11090 Cc1c2cc(ccc2sc1C(=O)COc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N)Cl RH02192 Cc1cc(c2cc([nH]c2c1)C(=O)Nc3ccc(cc3)OC(F)(F)F)C KM11065 COc1cccc(c1)c2cc3[nH]c(cc(=O)n3n2)c4ccccc4 KM00288 c1ccc(cc1)Cn2cc(c3c2ccc(c3)[N+](=O)[O-])Cc4cc(n[nH]c4=O)c5ccc(cc5)F HTS01403 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4ccc(cc4n5cccc5)[N+](=O)[O-] HTS01310 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3ccccc3 HTS00919 c1ccc(cc1)CC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11098 Cc1cc(c2ccccc2n1)Nc3ccccc3 KM11101 c1ccc(c(c1)NC(=S)N2CCCCC2)F SEW04275 Cc1csc(c1NC(=O)C(C)(C)C)C(=O)OC HTS00508 Cc1ccc(cc1)c2c(cno2)c3nnnn3c4ccc(cc4)C HTS01265 c1ccc(cc1)C2CC(CC3(N2)CCCC3)O RJC03989 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)CSCC(=O)O HTS01108 Cc1csc2c1c(=O)sc(n2)NC(=O)c3ccccc3 HTS01032 c1cc2c(cc(nc2c(c1)F)C(F)(F)F)N3CCN(CC3)CCO KM10654 C=CCn1c(nnc1SCc2ccccc2)c3ccc4c(c3)cccn4 KM10659 C=CCn1c(nnc1SCC(=O)Nc2ccccc2)c3ccc4c(c3)cccn4 KM10658 CC(C)NC(=O)CSc1nnc(n1C)CNC(=O)OC(C)(C)C KM10610 c1cc2c(cc1Cl)nc(o2)SCC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS01258 c1cc2c(cc1C(=O)C3CCC3)CCC2 SEW04500 COc1ccc2cc(ccc2c1)c3ccno3 SEW04501 Cc1ccc(cc1)c2csc3c2c(ncn3)NCc4ccco4 AW01152 COc1ccc(c(c1)OC)NS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01153 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01154 c1ccc2c(c1)c(=O)sc(n2)NC(=O)c3ccc(cc3Cl)F HTS01485 COc1cc2c(cc1OC)nc(sc2=O)NC(=O)c3ccc(cc3Cl)F HTS01486 c1cc(ccc1C(=O)Nc2nc3ccsc3c(=O)s2)F HTS01494 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)C4CCCCC4 HTS00652 c1ccc(c(c1)NS(=O)(=O)c2ccsc2C(=O)O)N3CCCCC3 HTS00474 CC1=CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)N4CCOCC4 HTS00600 c1ccc(cc1)C(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS00598 c1ccc2c(c1)c(c(c(=O)o2)CC(=O)c3ccccc3O)O HTS00005 c1ccc(c(c1)NS(=O)(=O)c2ccsc2C(=O)O)N3CCOCC3 HTS00473 COC(=O)c1cc(ccc1N2CCOCC2)NS(=O)(=O)c3ccc(cc3)F HTS00303 CN1CCN(CC1)c2ccc(cc2)NS(=O)(=O)c3ccsc3C(=O)OC HTS00072 Cc1cc(c(c(c1)C)CSCCNC(=O)NC(C)(C)C)C SEW06448 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2ccc(cc2)OC(F)(F)F)C SEW06450 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F)C(=O)OC HTS01554 Cc1ccc(cc1)c2csc3c2c(ncn3)N4CCNCC4 AW01150 Cc1ccc(cc1)c2csc3c2c(ncn3)N4CCOCC4 AW01151 CC(C)(C)S(=O)(=O)/C(=C/NNS(=O)(=O)c1ccc(c(c1)Cl)Cl)/C#N KM01898 c1ccc(cc1)C(CNCc2ccco2)O HTS00626 c1cc(c(c(c1)Cl)CSc2ccc(cc2)[N+](=O)[O-])F PD00588 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)/N=S/2\CCC3(C2)OCCO3 KM05934 c1cc(cc(c1)Br)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11099 CC1(c2ccccc2N3C1(NC(=O)C3)/C=C/c4ccc(cc4)F)C RJC04037 c1cc(ccc1CSCCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)Cl SEW06486 Cc1cccc(c1)Nc2c3cc(c(cc3ncn2)OC)OC GK03474 c1ccc(cc1)SCC(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS00810 Cc1c(c(nc(n1)c2cccnc2)N3CCCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl AW01129 CN1CCN(CC1)c2ccc(cc2)NC(=O)c3ccc(cc3F)F SS00020 CCCSc1cc(c(cn1)C(=O)Nc2ccc(cc2)Cl)C(F)(F)F RF04414 CSc1c(c(n2c(n1)cc(n2)c3ccc(cc3)Cl)N)S(=O)(=O)c4ccc(cc4)Cl KM02065 CC(C)S(=O)(=O)c1cscc1NC(=O)c2ccccc2Cl KM02177 CC(=O)N1C(CC(=N1)c2ccccc2O)c3ccc(cc3Cl)Cl RJC04102 Cc1csc(c1c2nc3ccccc3s2)NC(=O)C(F)(F)F HTS00386 CCCCCc1ccc(cc1)C(=O)Nc2nc3c(cc(cc3Br)Br)c(=O)s2 HTS01481 COc1ccc(cc1OC2CCCC2)NS(=O)(=O)c3ccc(cc3)F HTS00320 c1cc(ccc1F)S(=O)(=O)Nc2ccc3c(c2)OCO3 HTS00315 COc1ccc(c(c1OC)Cl)/C=C/C(=O)Nc2ccc(nc2)Oc3ccc(cc3)Cl HTS00305 Cn1cc(cc1C(=O)OC)/C=N/NC(=O)c2cccc(c2)[N+](=O)[O-] SEW06434 Cn1c2c(cn1)c(ncn2)N3CCCC3 GK03470 COc1ccc(cc1)Oc2ccc(cc2NS(=O)(=O)c3cccc4c3non4)C(F)(F)F HTS00256 Cc1c(nc(o1)c2ccccc2)C(=O)Nc3nc(c(s3)C)CC(=O)OC HTS00253 Cc1c(nc(s1)NS(=O)(=O)c2cccc(c2)C(F)(F)F)CC(=O)OC HTS00841 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2 HTS00383 COc1ccc(cc1)Oc2c(cccn2)NC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RH01999 c1ccc(cc1)c2csc3c2c(ncn3)NCCCn4ccnc4 AW01118 c1cc(c(c(c1)Cl)CN2CCN(CC2)CCCNc3nccc(n3)C(F)(F)F)F AW01119 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(sc2C(=O)OC)c3cccs3 GK03698 COC(=O)c1c(cc(s1)c2cccs2)NS(=O)(=O)c3ccccc3 GK03699 Cc1c(c(c(n1C)C)S(=O)(=O)N)C(=O)OC SP01165 CCOC(=O)c1c(n(c(c1S(=O)(=O)N2CCOCC2)C)c3ccccc3)C SP01167 CC1(c2ccccc2N3C1(NC(=O)C3)/C=C/c4ccc(cc4)N5CCOCC5)C RJC04038 c1c(cc(cc1C(F)(F)F)C(F)(F)F)CCC#N CD07888 c1cc(c(nc1)Sc2cccs2)C(=O)Nc3ccc(cc3F)F KM02412 Cc1ccc2nc(c(c(=O)n2c1)/C=N/Cc3ccco3)NCc4ccco4 RJC03979 COc1ccc(c(c1C#N)N2CCOCC2)[N+](=O)[O-] CD07399 c1cc2c(cc1Cl)cc(c(=O)o2)C(=O)O RH02219 CC(C)(C)OC(=O)NCc1nnc(n1C)SCc2ccc(cc2)OC(F)(F)F KM10586 Cn1c(ccn1)NC(=O)C2CCCCC2 GK03336 CNc1cc(c(cn1)C(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F RF04421 CC(C)(C)OC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01156 COC(=O)/C(=C/c1cccn1CCCn2ccnc2)/C#N SEW04562 c1cc2c(cc1NS(=O)(=O)c3ccc(s3)Br)CS(=O)(=O)C2 KM10785 Cc1c(snn1)C(=O)n2c(ccn2)c3cnn(c3C)c4ccccc4 SP01327 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4c5c(csc5ncn4)c6ccccc6 AW01159 COc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3n4cccc4)[N+](=O)[O-] HTS01007 COCCOc1ccccc1NC(=S)NNC(=O)c2ccc(cc2)[N+](=O)[O-] GK03686 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)C3Cc4ccccc4C3 PD00800 c1ccc2c(c1)c(=O)c(c[nH]2)c3nnnn3c4ccc(cc4)Cl HTS01263 c1cc(sc1)c2nc(cs2)c3ccc(cc3)F HTS01587 COCC(=O)Nc1cc(c(cc1C(=O)OC)OC)OC GK03376 c1cc(ccc1NC(=O)c2ccc(o2)S(=O)(=O)N3CCOCC3)Cl HTS00425 c1cc(ccc1NC(=O)c2ccc(o2)S(=O)(=O)N3CCOCC3)OC(F)(F)F HTS00424 c1cc(ccc1NC(=O)c2ccc(o2)S(=O)(=O)N3CCOCC3)F HTS00421 CC(C)(C)c1ccc(cc1)S(=O)(=O)Nc2ccnn2C GK03377 COC(=O)c1c(cc(s1)c2cccs2)NC(=O)c3ccco3 GK03701 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2cccc(c2C)Cl)C SEW06454 CC(=O)Nc1cc(sc1C(=O)N)c2ccc(cc2)C(C)(C)C GK03535 c1ccc(c(c1)/C=N/c2c(c3c(s2)CCCC3)C(=O)N)Cl RJC04031 c1cc(ccc1c2csnn2)c3nc(on3)c4ccc(cc4)Cl SEW01077 CCOC(=O)N/N=C(/c1ccc(cc1)/C(=N/NC(=O)OCC)/C)\C SEW01074 c1ccc(cc1)Cn2ccc3c2ccc(c3CC#N)[N+](=O)[O-] SP01336 Cn1c2cccc(c2c(n1)NC(=O)c3ccco3)F SP01339 Cc1c(ccc(n1)C(F)(F)F)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 HTS00674 COc1ccc(cc1)C(=O)Nc2cc(ccc2Oc3ccc(cc3)OC)C(F)(F)F HTS00863 COC(=S)Nc1cc(cc(c1)Cl)Cl NH00699 c1ccc(cc1)CN(Cc2cccnc2)C(=O)c3ccc(cc3)Cl RF03281 c1cn(cn1)CCCNc2c3c4c(sc3ncn2)CCCC4 GK03333 c1nc(c2c3c(sc2n1)CCCC3)NC4CCCCC4 GK03334 Cn1c(ccn1)NC(=O)c2ccccc2 GK03335 CN1CCN(CC1)C(c2cccs2)N3CCN(CC3)C PD00612 Cc1c(c(c(o1)C)S(=O)(=O)Nc2ccccc2SCc3c(cccc3Cl)F)C(=O)OC HTS01460 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3NS(=O)(=O)c4ccccc4 SPB07791 Cc1c(c(n(n1)C(C)(C)C)C)/C=N/OC(=O)Nc2ccc(cc2)OC CD07460 c1c(csc1/C=N/O)Cl CD07676 COc1cc(cc(c1OC)OC)C/N=C/c2cc(c(c(c2)OC)OC)OC SEW04987 c1csc2c1ncnc2N3CCOCC3 GK03785 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)[N+](=O)[O-] SS00006 Cc1c(cnn1c2ccccc2)c3ccnn3C(=O)c4cccs4 SP01341 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl HTS01138 COc1ccc(cc1S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl)Cl HTS01139 c1cc(ccc1C(=O)NNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)Cl HTS00505 CC(C)NC(=O)c1ccccc1N KM09493 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C RH02002 c1nc(c2c3c(sc2n1)CCCC3)NCCO GK03331 CS(=NS(=O)(=O)c1ccc(c(c1)Cl)Cl)(=O)c2ccccc2 KM02837 CN1CCN(CC1)c2ccc(cc2)NC(=O)c3ccccc3Cl SS00002 c1cc2c(cc1C3=NNC(C3)(C(F)(F)F)O)OCO2 KM10713 COc1cc(c(cc1OC)NC(=O)c2ccccc2)C(=O)O GK03478 Cc1c(c2c(s1)c(cc(n2)OC)C(F)(F)F)C(=O)OC GK03800 CCOC(=O)c1cc(c(cc1NS(=O)(=O)c2ccc(cc2)Cl)OCCOC)OCCOC GK03801 CCOC(=O)c1cc(n(c1C)N(C)c2cc(ccn2)C(F)(F)F)C SEW04421 c1ccc(cc1)c2csc3c2c(ncn3)NCCN AW00963 c1cc(ccc1CC(C(=O)O)NS(=O)(=O)c2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] SPB08317 c1ccc(cc1)CC2CCN(CC2)C3=Cc4ccccc4C3 HTS01269 CSc1c(c([nH]n1)N)S(=O)(=O)c2ccc(cc2)Cl KM01037 C1CSCc2c1nc(nc2O)C3CC3 RF03876 COC(=O)c1ccccc1NC(=S)NNC(=O)c2ccc(cc2)[N+](=O)[O-] GK03689 Cc1csc(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl SEW05044 Cc1ccc(c(c1)NC(=O)c2c(onc2c3c(cccc3Cl)Cl)C)n4cccc4 SEW06416 COc1cc(c(cc1OC)NC(=O)c2ccccc2)C(=O)OC GK03383 c1ccc2c(c1)C(C(N(C2=O)Cc3ccc(cc3)F)c4cccs4)C(=O)O PD00690 Cc1cc(ccc1Br)NC(=O)C KM10161 c1cc(sc1)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11084 c1cc(ccc1OC(F)(F)F)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11086 c1ccc(cc1)C(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11087 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2cc(ccc2OC)Cl HTS00050 CC(C)(C)OC(=O)C(C)(C)Sc1nnc(s1)N RH02005 Cc1cccc(c1NC(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4)Cl HTS00667 CCCCNC(=O)N1CCN(CC1)C(c2ccccc2)c3ccccc3 HTS00668 COCC(=O)/C(=N\Nc1cccc(c1)Cl)/C(=O)OC SPB04023 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl GK03757 COc1cc(c(cc1OC)NC(=O)Nc2ccccc2)C(=O)OC GK03293 COc1cc(c(cc1OC)NC(=O)Nc2ccc(cc2)F)C(=O)OC GK03294 Cn1c(=O)c(nn(c1=S)C)c2ccc(cc2)C(F)(F)F SPB07820 Cc1cc(nc(c1C#N)OCC(=O)Nc2ccccc2)C HTS01404 COc1ccc(cc1)Nc2nc([nH]n2)N TG00127 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01163 COC(=O)c1cc(=O)c2cc(ccc2[nH]1)NC(=O)c3ccc(cc3)OC(F)(F)F SEW04939 c1cc(c(c(c1)Cl)/C=C/c2ccnn2C(=O)c3cccs3)Cl SP01328 CC(C)(C)OC(=O)n1ccc2c1ccc(c2)Br RH02183 c1cc(sc1)S(=O)(=O)Cc2ccc(cc2)Cl KM02264 c1cc(cc(c1)/C(=N/OC(=O)Nc2ccc(cc2)Cl)/N)CSc3cccs3 KM02351 c1ccn(c1)C2CCN(CC2)C(=O)CC3(CCCC3)CC(=O)O HTS00582 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4ccc(cc4F)F HTS00653 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4cccc(c4)C(F)(F)F HTS00659 c1cc(c(c(c1)Cl)SC(=O)c2ccc(cc2)OC(F)(F)F)Cl SPB03553 Cc1ccc(cc1)Sc2c(cccn2)NS(=O)(=O)c3ccc(cc3)C RH02093 Cc1ccc(n1c2c3c(cccc3F)n(n2)S(=O)(=O)c4cccc5c4nccc5)C HTS01083 Cc1ccc(n1c2c3c(cccc3F)n(n2)S(=O)(=O)c4ccc(c(c4)OC)OC)C HTS01089 c1cc(ccc1Nc2nnns2)F HTS00547 c1cc(c(c(c1)Cl)Cl)Nc2nnns2 HTS00546 Cn1c(cc(=O)n(c1=O)C)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] HTS00865 Cc1ccc(n1c2c3c(cccc3F)n(n2)S(=O)(=O)c4ccccc4)C HTS01085 CC(C)(C)c1ccc(cc1)S(=O)(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O HTS00210 COc1ccc(cc1OC2CCCC2)NC(=O)c3ccccc3C(F)(F)F HTS00326 CC(C)N(C(C)C)C(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl KM11096 CN(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11097 Cc1c(ccc(n1)C(F)(F)F)C(=O)N2CCC(CC2)n3cccc3 HTS00673 CC1(CC2CC1C=C2)C(=O)O RH02006 COc1ccc(cc1)Oc2c(cccn2)NC(=O)c3cccc4c3cccc4 RH02008 c1cc(ccc1SCc2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)Cl SEW05046 Cc1cc(no1)NCc2cccnc2 RF03209 c1ccc-2c(c1)CCc3c2sc(c3)C(=O)NNC(=O)C4CCC4 PD00819 COc1ccccc1OCC(=O)N SPB08038 CC(=O)c1ccc(cc1)OCC(CN2CCC(CC2)C(=O)N)O HTS00802 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(CSc4ccccc4)O HTS00806 c1ccc2c(c1)CC(C2=O)Sc3nnnn3c4ccc(cc4)O HTS00942 CC(=O)Nc1ccc(cc1)/N=N/c2cccc(c2)Cl BTB06644 c1ccc2c(c1)c(=O)n(c(n2)SCC(=O)c3ccc(cc3)F)c4ccc(c(c4)Cl)Cl HTS00686 CC(C)(C)NC1=C(C(=O)NC(S1)c2ccccc2O)C#N CD07641 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])Sc3ccc(cc3Cl)F RH02090 c1cc2c(cc1Nc3ccnc4c3ccc(c4)Cl)OCO2 KM11079 Cc1ccc(cc1F)Nc2ccnc3c2ccc(c3)Cl KM11080 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)c3cccs3 SS00013 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3ccc(cc3)F PD00613 Cc1cc(ccc1Br)N2C(=O)CSC23c4ccccc4NC3=O PD00615 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4cccc(c4)Cl HTS00677 CCCCCc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 HTS00658 c1cc(ccc1c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)Cl SEW05043 COc1ccc(cc1)n2c(nnn2)c3c[nH]c4c3cc(cc4)Cl HTS01271 c1ccc2c(c1)c(c(cn2)c3nnnn3c4ccc(cc4)Cl)N HTS01281 c1cc(ccc1n2c(nnn2)c3cnc4cc(ccc4c3N)Cl)F HTS01282 COc1cccc(c1NC(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F)Cl HTS00414 CCOC(=O)C1CCN(CC1)c2cc(=O)n(c(=O)n2C)C HTS00864 c1ccc(cc1)Oc2c(cccn2)C(=O)NCCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F RH01964 Cc1csc2c1nc(sc2=O)NC(=O)c3ccc(cc3)F HTS01495 CN1CCc2c(sc3c2c(=O)sc(n3)NC(=O)c4ccc(cc4)OC(F)(F)F)C1 HTS01600 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)Cc3ccc(cc3)F)C(=O)OC HTS01540 CC(C)(C)c1ccc(cc1)c2cc([nH]n2)N KM00336 Cc1nccc(n1)c2cccc(c2)[N+](=O)[O-] KM02121 Cc1cc(oc(=O)c1)C(=O)N SEW01574 c1cc(ccc1CSc2nnnn2c3ccc(cc3)O)OC(F)(F)F HTS00945 c1cc(cc(c1)[N+](=O)[O-])C(CN2CCC(CC2)C(=O)N)O HTS00990 COC(=O)c1cc(sc1)[N+](=O)[O-] SEW03128 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)SC[C@@H](C(=O)O)NC(=O)OCC4c5ccccc5-c6c4cccc6 SB02035 COc1cc2c(cc1OC)ncnc2NNC(=O)c3cccs3 GK03669 COc1ccc2c(c1)cc([nH]2)C(=O)NCCCn3ccnc3 HTS01091 COc1ccc2c(c1)cc([nH]2)C(=O)NCCNc3cccc(n3)C(F)(F)F HTS01094 COc1ccc(cc1)COCC(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS00786 Cn1cc(cc1C(=O)OC)/C=C/2\CSc3ccc(cc3C2=O)Cl SEW06428 CC(C)(C)NC(=O)N1CCc2c(ccs2)C1c3ccc(cc3)OC SEW06429 c1ccc(c(c1)NC(=S)NNC(=O)c2ccc(cc2)[N+](=O)[O-])Cl GK03676 COc1ccc2c(c1)cc([nH]2)C(=O)NCc3ccc4c(c3)OCO4 HTS01090 COc1ccc(cc1S(=O)(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O)Cl HTS00196 CC(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl KM11088 Cc1cc(c2ccccc2n1)Nc3ccc(cc3F)I KM11094 c1cc(ccc1S(=O)(=O)Cc2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)Cl SEW05047 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)CC(COc4ccc(cc4)F)O HTS01130 c1ccc(cc1)CC2CCN(CC2)S(=O)(=O)c3cc(sc3Cl)Cl HTS00833 Cn1c(ccc1S(=O)(=O)N2CCC(CC2)C(=O)N)C(=O)OC HTS01073 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)C)C(=O)OC HTS01074 Cn1c(ccc1S(=O)(=O)N2CCCCCC2)C(=O)OC HTS01075 Cc1c(sc(c1c2ccn(n2)S(=O)(=O)c3cc(ccc3Cl)Cl)SC)C#N KM03668 CC(C)(C)OC(=O)NCc1nnc(n1C)SCC(=O)Nc2ccccc2 KM10582 COc1ccc(cc1)COCC(CN2CCC(CC2)C(=O)N)O HTS00783 CCOC(=O)Cn1c(=O)c(cc(n1)c2ccc(cc2)F)Cc3ccccc3 HTS01410 COc1ccc(cc1OC)C(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH01983 c1ccc2c(c1)cccc2C(=O)Nc3cccnc3Oc4ccc(cc4)Cl RH01984 C[C@@H](c1ccccc1)Nc2c3cc(c(cc3ncn2)OC)OC GK03379 c1cnccc1c2nc(cs2)C(=O)NN MWP00354 c1cc(ccc1c2nc(cs2)C34CC5CC(C3)CC(C5)C4)C(F)(F)F SPB08314 COc1ccc(cc1)Oc2ccc(cc2NC(=O)c3ccc(cc3)F)C(F)(F)F HTS00848 c1csc2c1nc(sc2=O)NC(=O)C3CCC3 HTS01611 c1c(cc(c2c1c(=O)sc(n2)NC(=O)C3CCC3)Br)Br HTS01615 CCC(=O)N1CCN(CC1)c2ccnc3c2ccc(c3)Cl KM11107 Cc1ccc(cc1)n2c(nnn2)c3cnoc3c4ccc(cc4)F HTS01266 c1cc(cc(c1)Cl)NC(=S)Nc2ccc(nc2)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06480 c1ccc2c(c1)c(nc(n2)C(F)(F)F)O RH01963 Cc1cc(c2ccccc2n1)OCC(=O)Nc3ccc4c(c3)OCO4 HTS00868 Cc1ccc(c2c1c(ccn2)OCC(=O)N(c3ccccc3)C4CCCCC4)C HTS00869 Cc1cc(c2ccccc2n1)OCC(=O)Nc3ccc(cc3)OC(F)(F)F HTS01178 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)C(=O)NNC(=S)NC SPB08173 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3 HTS00912 c1cc(ccc1OCC(CN2CCN(CC2)c3nc4ccc(cc4s3)Cl)O)F HTS01132 Cc1ccccc1C(=O)Nc2nc3c(csc3c(=O)s2)C HTS01500 Cc1ccccc1C(=O)Nc2nc3c(cc(cc3Br)Br)c(=O)s2 HTS01593 c1cc(ccc1C(=O)Nc2nc3ccsc3c(=O)s2)OC(F)(F)F HTS01595 Cc1cc(c2ccccc2n1)Nc3ccccc3Cl KM11102 Cc1c(nc(s1)c2ccc(cc2)Cl)c3ccc(cc3)CC(C)C HTS00858 c1cc(ccc1c2csc(n2)N3CCN(CC3)c4ccc(cc4)Cl)Cl HTS01262 c1cc(ccc1c2nc(on2)CNC(=O)Nc3ccc(cc3F)F)C(F)(F)F HTS01220 c1c(cnc(c1N2CCCC2)C(=S)N)C(F)(F)F SEW03743 CC(C)(C)C(=O)Nc1ccc(c(c1)OC)Br SEW03860 CCOc1cc(cnc1/C(=N/OC(=O)NC)/N)C(F)(F)F SEW03907 Cc1csc2c1ncnc2N3CCC(CC3)C(=O)O HTS00364 c1cc(sc1c2csc(n2)NC(=O)C3CCC3C(=O)O)Cl HTS00261 c1ccc(cc1)c2csc3c2c(ncn3)NCCNC(=O)CCC(=O)O AW00999 Cn1c(nnc1S)Cn2c3ccccc3c4c2cccc4 RH02011 Cc1ccc(cc1C)C(=O)Nc2cc(ccc2Oc3ccc(cc3)OC)C(F)(F)F HTS00258 COC(=O)c1cccc(c1)CN2CCN(CC2)c3c4c(csc4ncn3)c5ccccc5 AW01131 CCCc1cnc(nc1)N2CCN(CC2)c3c4c(csc4ncn3)c5ccccc5 AW01134 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3ccc(c(c3)Cl)N4C(=O)CC5(C4=O)CCCC5 AW01144 c1cc(cc(c1)F)c2c(cno2)c3nnnn3c4ccc(cc4)Cl HTS01268 c1ccc(cc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS01395 c1cc(c(c(c1)Cl)/C=N/OC(=O)Nc2ccc(cc2)Cl)Cl RF01985 CN1CCN(CC1)CC(c2ccccc2)O HTS00727 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCc3ccc(cc3)Cl PD00606 c1ccc(cc1)CN2CCN(CC2)CN3C(=O)c4ccccc4C3=O PD00607 CC1(OC(=O)C(=Cc2ccc(c(c2)OCc3ccccc3)OC)C(=O)O1)C PD00609 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccccc3C(F)(F)F RH01981 COc1ccc(cc1)CNC(=O)Nc2ccccc2Cl KM10592 c1cc(ccc1n2c(c(cn2)C(=O)NNC(=O)C3=Cc4cc(ccc4OC3)Cl)C(F)(F)F)Cl HTS00409 Cc1csc(c1NC(=O)C2=Cc3cc(ccc3OC2)Cl)C(=O)OC HTS00405 COc1ccc(cc1OC2CCCC2)NC(=O)C3CCCCC3 HTS00329 CN(C)S(=O)(=O)Nc1ccccc1 KM09705 c1cc(cnc1)CN2CCC(CC2)C(=O)NN KM09939 c1ccc(cc1)C(CN2CCC(CC2)(c3ccc(cc3)Cl)O)O HTS00726 c1ccc2c(c1)C(=O)N(C2=O)CN3CCC(CC3)(c4ccc(cc4)Cl)O HTS00735 c1cnc(c(n1)C(=O)N2CCC(CC2)C(=O)N)C(=O)O HTS01066 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc(c(c3)C(=O)OC)N4CCOCC4)C HTS00925 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3c(cccc3Cl)F HTS00928 Cc1ccc2c(c1)C(C3(N2CC(=O)N3)/C=C/c4ccc(cc4)Br)(C)C RJC04039 c1ccc(cc1)c2cc([nH]c(=O)c2C#N)c3ccccc3 JFD03993 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C#N)Cl SPB01032 CCC(=O)Nc1cc(cc(c1)C)C RH02000 c1cc2c(cc1C(=O)N3CCCC3)nns2 KM10678 c1cc(cc(c1)NS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4)C(F)(F)F AW01157 CCC(C)Sc1cc(c(cn1)C(=O)Nc2c(cccc2C)C)C(F)(F)F RF04425 CCOC(=O)c1c(nc(s1)N)C RF02301 COc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11100 Cc1ccc(cc1F)Nc2cc(nc3c2cccc3)C KM11103 c1cc(sc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS01397 Cn1c(ccn1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl GK03361 c1cc(ccc1n2c(c(cn2)C(=O)NC3CC3)C(F)(F)F)Cl GK01739 COc1cc(c(cc1OC)NC(=O)c2ccccc2Br)C(=O)OC GK03385 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3Cl)F GK03388 Cc1ccc(cc1)Sc2c(cccn2)NS(=O)(=O)c3ccc(cc3)F RH02111 c1ccc2c(c1)CCN(C2)c3cc(nc4c3cccc4Cl)C(F)(F)F KM10574 c1ccc(cc1)CNc2c(cccn2)[N+](=O)[O-] KM10676 Cc1nc(cs1)C(=O)/C=C/N(C)C SPB03610 c1cc2c(cc1C(=O)N3CCN(CC3)c4ccnc5c4ccc(c5)Cl)OCO2 KM11106 Cc1ccc(c(c1)C)Nc2cc(nc3c2cccc3)C KM11109 Cc1ccc(cc1)c2csc3c2c(ncn3)N4CCc5ccccc5C4 AW01149 Cc1cc(ccc1Br)N2C(SCC2=O)c3cccnc3 PD00629 CCOC(=O)CSC(=S)NCc1ccccc1 PD00632 c1ccc-2c(c1)CCc3c2sc(c3)C(=O)NN PD00633 c1cc(c(c(c1)Cl)Cl)NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)Cl RDR00727 CC(C)(C)OC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(cc2)Cl AW01172 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2cccs2 HTS00043 COc1cc(c(cc1OC)NC(=O)CN2CCOCC2)C(=O)OC GK03491 COc1cc(c(cc1OC)NC(=O)CN2CCNCC2)C(=O)OC GK03492 c1cc2c(cc1CNc3nccc(n3)C(F)(F)F)OCO2 AW00986 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3c4c(cc(s4)c5ccc(cc5)C(C)(C)C)ncn3 GK03770 c1ccnc(c1)Sc2c3c(ccs3)ncn2 GK03339 CN1CCN(CC1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Br SS00024 Cc1ccc(cc1)c2nnn(n2)CC(=O)NNC(=O)c3ccco3 GK03485 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)N2CCCCC2 AW01126 Cc1cccc(c1NC(=O)c2c(ccnc2SCCN(C)C)C(F)(F)F)C RF04609 c1cc(c(cc1I)F)N2C(=O)CC3(CCCC3)CC2=O PD00696 CC(=O)Nc1cccc(c1)OCCCN2Cc3c(n(c(=O)n(c3=O)C)C)NC2 PD00698 Cc1ccc(cc1)S(=O)(=O)NNc2c3cnn(c3ncn2)C GK03490 CNC(=O)NC(=O)c1cnccc1C(F)(F)F RF04467 c1cc(c(cc1OCC(F)(F)F)C(=O)NC(=O)Nc2c(cc(cc2F)F)F)OCC(F)(F)F RF04588 c1cc(sc1)c2nc(cs2)c3ccc4c(c3)OCCO4 SPB08223 CC(C)(CC(=O)N1CCN(CC1)c2cc(nc3c2cccc3)C(F)(F)F)CC(=O)O HTS01453 c1ccc2c(c1)nnn2CN3CCC(CC3)C(=O)N HTS00728 Cc1ccc2cc(ccc2n1)NC(=O)c3ccccc3 RH02205 Cc1ccc2cc(ccc2n1)NC(=O)c3ccc(cc3)C(C)(C)C RH02207 c1cc(c(cc1[N+](=O)[O-])/C=C\2/C(=NNC2=O)N)N3CCOCC3 RH02220 c1cc(ccc1OC(F)(F)F)S(=O)(=O)Nc2c(ccs2)C#N GK03772 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(o3)SCC(=O)Nc4ccccc4Cl SPB08351 c1ccc(c(c1)C(=O)N)NC(=O)c2cccs2 RH02030 CC(C)C(=O)n1c2ccc(cc2c3c1nc4ccccc4n3)F RH02031 Cc1cc(nn1C(C)(C)C)C(=O)NNS(=O)(=O)c2ccc(cc2)F HTS00063 Cc1cc(c2ccccc2n1)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl HTS00068 Cc1cc(c2ccccc2n1)N3CCN(CC3)S(=O)(=O)c4ccccc4 HTS00069 Cc1c(cc(o1)C(C)(C)C)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SP01211 Cc1c(cc(o1)C(C)(C)C)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SP01212 Cc1ccc(cc1)SCC(=O)Nc2cc(c(cc2C(=O)OC)OC)OC GK03493 C=CCC1(CCCCC1)NCCc2ccccc2.Cl RJC03988 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3nc(cs3)C(C)(C)C CD08375 Cn1c(ccc1S(=O)(=O)NC2CCN(CC2)Cc3ccccc3)C(=O)OC HTS01531 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=N)N3CCCC3 CD07791 Cc1c(c(c(c(c1C)C)CN2CCSCC2)C)C CD07855 c1ccc(cc1)c2c(snn2)C(=O)NNC(=O)c3ccco3 SP01308 CCOC(=O)c1c(c(sc1NC(=O)CCC(=O)O)C)c2ccccc2 AW01011 c1cc(sc1)c2csc3c2c(ncn3)N4CCN(CC4)c5nccc(n5)C(F)(F)F AW01013 c1cc(c(cc1Cl)Sc2c3c(ccs3)ncn2)Cl GK03791 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCC(CC2)C(=O)OCC)C#N SPB08421 Cc1cc(no1)C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F SPB08440 Cc1c(c(nc(n1)c2ccccn2)N3CCCN(CC3)Cc4ccc(cc4Cl)Cl)Cl AW01237 CC(CNc1c2c(csc2ncn1)c3ccccc3)O AW01133 CC(C)N1CCN(CC1)c2c3c(csc3ncn2)c4ccccc4 AW01135 CCOC(=O)c1c2c(sc1NC(=O)CN3CCCCC3)CCCC2 HTS01896 Cc1ccc(cc1NC(=O)N2CCN(CC2)c3cccc4c3ccc(n4)C(F)(F)F)F HTS01458 c1cc(sc1)C(=O)c2ccc(cc2)Cl SEW04625 c1ccc(c(c1)C(=O)NNc2nc(cs2)c3cccc(c3)[N+](=O)[O-])Cl CD03335 CC(=O)c1c(cc(s1)c2ccccc2)NC(=O)c3ccccc3 GK03768 CC(=O)c1c(cc(s1)c2ccccc2)NC(=O)c3ccc(cc3)OC(F)(F)F GK03769 COc1ccc(cc1)S(=O)(=O)Nc2c(ccs2)C#N GK03771 c1ccc(cc1)c2c(oc(n2)Sc3cc(c(cc3[N+](=O)[O-])Cl)n4cccc4)c5ccccc5 RH02106 Cc1nc(cn1CC(=O)c2ccc(cc2)c3ccccc3)[N+](=O)[O-] HTS01003 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)c4ccc(cc4)OC(F)(F)F)[N+](=O)[O-] HTS00292 COC(c1c(cnn1c2ccc(cc2F)F)C(=O)OC)OC SPB05109 CN1CCN(CC1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)F SS00025 CN(C)/C=C/C(=O)C12CC3CC(C1)CC(C3)C2 SPB08306 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)c3c4c(csc4ncn3)c5ccccc5 AW01130 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)C(=O)Nc3ccc(c(c3)C(F)(F)F)Br HTS01947 Cc1ccccc1C(=O)Nc2ccc3c(c2)ccc(n3)C RH02206 CCc1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4C KM10792 CCn1c(cc(n1)C)C(=O)OCC(=O)c2ccc(cc2)Cl HTS01506 Cc1c2c(onc2c(=O)n(n1)c3ccc(cc3)C(C)(C)C)C HTS01320 CSc1cccc(c1)NC(=O)CN2CCN(CC2)CC(=O)Nc3cccc(c3)SC HTS01903 Cc1ccc2cc(ccc2n1)NC(=O)c3ccco3 RH02213 CCOC(=O)c1cc2c(n1C(=O)OC(C)(C)C)cc(cc2Cl)Cl RH02215 CCOC(=O)C1CCN(CC1)c2c3c(csc3ncn2)C HTS00365 CN1CCN(CC1)c2ccc(cc2)NC(=O)c3ccccc3 SS00003 CCCCCCCCCCCC(=O)Nc1cc(c(cc1Cl)Cl)Cl RG00118 c1cnc(nc1C(F)(F)F)N2CCC(CC2)NC(=S)NC3CC3 AW01026 COc1ccc(cc1OC)C(=O)Nc2cc(sc2C(=O)N)c3ccccc3 GK03725 Cn1cc(nc1)S(=O)(=O)Nc2cc(sc2C(=O)OC)c3cccs3 HTS01041 COC(=O)c1c(cc(s1)c2cccs2)NS(=O)(=O)c3cc(sc3Cl)Cl HTS01042 c1cc(ccc1C(F)(F)F)NC(=O)CSc2nnnn2c3ccc(cc3)O HTS01668 Cn1c(ccc1S(=O)(=O)NCc2ccco2)C(=O)OC HTS01747 c1cc(c(cc1S(=O)(=O)Nc2ccc(cc2Cl)Cl)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01146 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)NCc3cccs3 HTS01371 c1ccc(cc1)/C(=C/Sc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N)/O HTS01848 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl)C(=O)OC HTS01548 COC(=O)c1cccn1c2ccc(cc2)F SEW04661 c1ccc(cc1)C(=O)c2cccn2S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW04641 CCOC(=O)c1cc(c(nc1C(F)(F)F)C)C(=S)N AW00991 c1c(cc(c(c1[N+](=O)[O-])N/N=C/c2cc(cc(c2O)Cl)Cl)[N+](=O)[O-])C(F)(F)F CD03421 c1cc(sc1)S(=O)(=O)N2CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl HTS01448 Cn1cccc1CN(Cc2ccc(cc2)OC)S(=O)(=O)c3ccccc3 HTS00761 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCOc2ccc(cc2)OC SPB08199 CN(C)c1ccc(cc1)n2c(nnn2)SC3Cc4ccccc4C3=O HTS00787 CN(C)c1ccc(cc1)n2c(nnn2)SCc3ccc(cc3)Cl HTS00697 CC(C)c1ccc(cc1)NC(=O)CSc2nnnn2c3ccc(cc3)O HTS01666 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)COCC(=O)O HTS01719 Cc1ccc(cc1)c2csc3c2c(ncn3)N4CCCCC4 AW01141 c1cc(nc(c1)NCCNS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4)C(F)(F)F AW01143 COc1ccccc1NS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01145 Cn1c(ccc1S(=O)(=O)NNC(=O)COc2ccc(cc2)OC(F)(F)F)C(=O)OC HTS01546 Cc1ccc(cc1)C(=O)Nc2cc(sc2C(=O)OC)c3cccs3 GK03696 c1cc(c(cc1[N+](=O)[O-])Cl)n2c(=O)n(c(=O)s2)CC3CC3 HTS01835 CN(C)/C=N/c1nnc(s1)SCC(=O)c2ccc(cc2)Cl HTS01503 COc1ccc(cc1OC)C2CC(=O)c3c2cc(c(c3)OC)OC HTS01505 c1ccc2c(c1)cccc2CN3CCCN(CC3)C(=O)Nc4ccc(cc4)Cl AW00996 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3c(cccc3F)F)C HTS01286 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(c(cc2C(=O)O)OC)OC GK03530 Cc1ccc(cc1)c2csc3c2c4nnnn4cn3 AW01169 COc1cccc(c1C(=O)N2CCN(CC2)c3c4c(csc4ncn3)c5ccccc5)OC AW01170 COc1ccc(cc1)C(=O)Nc2ccc(c(c2)C(=O)OC)N3CCOCC3 HTS00917 Cc1c(c(c2c(c1C)[nH]c(n2)SC)C)C CD04437 c1cc(sc1)S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl HTS01323 COc1ccc(c(c1OC)Cl)C2OCCCO2 HTS00065 c1ccc2c(c1)CC(C2)n3c(=O)n(sc3=O)c4ccc(c(c4)Cl)F HTS01580 Cc1ccc(cc1C)C(=O)NC2(C(=O)c3ccccc3C2=O)O HTS01852 Cc1ccc(cc1)S(=O)(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH02019 Cc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl RH02026 c1cc(oc1)CS(=O)(=O)Cc2nc(cs2)c3ccc4c(c3)OCCO4 SPB08228 Cc1nc(cn1CC(=O)c2ccc3c(c2)OCCCO3)[N+](=O)[O-] RH02258 Cn1c(ccc1S(=O)(=O)N(Cc2ccccn2)Cc3ccccn3)C(=O)OC HTS01743 c1c(cc(cc1C(F)(F)F)S(=O)(=O)N)C(F)(F)F CD03372 Cc1cc(ccc1Nc2nnns2)Cl HTS00549 c1ccc2c(c1)C(=O)N(C2=O)CCCSc3nccn3c4cc(ccc4Cl)Cl AW00978 c1ccc(cc1)c2csc3c2c(ncn3)N4CCC(CC4)C(=O)O AW00983 CCCc1ccc(cc1)C(=O)Nc2nc(c(s2)C)c3ccc(c(c3)Cl)C HTS01287 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3ccc(cc3)C(F)(F)F)C HTS01288 Cc1csc(c1c2nc3ccccc3s2)NC(=O)C HTS00384 c1ccc2c(c1)/C(=N/O)/CCS2(=O)=O CD04025 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)c3ccc(cc3)C(C)(C)C HTS01050 c1cc(oc1)CNC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00084 COc1ccc(cc1OC)C(=O)Nc2cc(sc2C(=O)OC)c3cccs3 GK03697 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)c3cccc(n3)C(F)(F)F)C(=O)OC HTS01550 c1cc(ccc1c2nnc(o2)SCC3CC3)Cl SPB08233 COc1cc(cc(c1)NC(=O)c2cccc(c2)C(F)(F)F)C(F)(F)F.Cl CD03641 c1c(cc(c2c1nc(cc2N3CCC(=O)CC3)C(F)(F)F)Cl)Cl KM10686 CC(C)(C)c1c(c(n[nH]1)C(C)(C)C)Cc2c(cccc2Cl)F SEW06632 CC(C)(C)C(=O)C(Cc1c(cccc1Cl)F)C(=O)C(C)(C)C SEW06633 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NC3CC3 HTS00915 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3ccc(cc3)F HTS00916 Cc1cc(c(c(c1)C)C(=O)N2CCN(CC2)c3ccc(cc3n4cccc4)[N+](=O)[O-])C HTS00286 CC(C)(C)c1ccc(cc1)NC(=O)/C=C/c2ccc(cc2)C(=O)C(F)(F)F SEW06497 c1cnccc1c2cc([nH]n2)C(F)(F)F KM09522 c1ccc(c(c1)CN(C(=O)CC#N)C(=O)NC2CCCCC2)F KM09710 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc(cc3)C(C)(C)C SPB08238 c1ccc(c(c1)C(=O)O)n2cccc2C(=O)O SEW05149 CS(=NS(=O)(=O)NC(=O)Nc1cccc(c1)C(F)(F)F)(=O)c2ccccc2 KM05902 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)C(=O)Nc3ccccc3 SPB08246 c1cc(sc1c2csc(n2)c3ccsc3)Cl HTS00038 c1cc2c(cc1c3nc(cs3)c4ccc(s4)Cl)CCO2 HTS00037 c1cc2c(cc1Cl)nc(o2)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS01561 Cc1cccc(c1)S(=O)(=O)Nc2nc(c(s2)C)CC(=O)OC HTS00843 CSc1c(cn(n1)c2ccccc2)C(=O)ON=C3CC4CCCC(C3)N4Cc5ccccc5 KM08829 c1cc2c(cc1[N+](=O)[O-])COCO2 SEW03597 c1cc(ccc1c2nc(cs2)CSc3ccc(cc3)Cl)Cl CD03336 CC(C)(C)OC(=O)NCc1nnc(n1C)SCC(=O)NCc2ccccc2 KM10583 Cc1cccc(c1)NC(=O)NCc2ccc(cc2)OC KM10591 Cn1c2cccc(c2c(n1)NC(=O)C3CCC3C(=O)O)F HTS00766 Cc1c2ccccc2sc1C(=O)COc3c(c(cc(n3)c4cccs4)C(F)(F)F)C#N RH02195 c1ccc(cc1)NC(=O)CSCC(=O)NN KM08976 c1cc(cc(c1)C(F)(F)F)c2ccnc3n2nc(c3)/C(=N/OC(=O)c4cccc(c4)C(F)(F)F)/N SEW04865 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)c4ccccc4 KM10683 Cc1c(nc(s1)NC(=O)c2ccc(cc2)OC)CC(=O)OC HTS00862 c1cc(sc1)c2ccc(s2)/C=C/3\COc4c(cc(cc4F)F)C3=O SEW05378 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Nc2ccnn2C GK03391 CC1(CC2=C(C(C(=C(O2)N)C#N)c3ccc(c(c3)OCc4ccccc4)OC)C(=O)C1)C PD00592 CC(C)(C(=O)OCC(=O)c1ccc(cc1)Cl)O RF03424 CCNC(=O)N(Cc1ccccc1)Cc2cccnc2 RF03427 c1ccc(cc1)CN2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F KM10629 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)C)C SP00967 CN(/C=C\c1cc(ncc1)c2nccc(c2)/C=C\N(C)C)C RJC04049 c1ccc(cc1)CNC(=S)Nc2ccc(nc2)N3CCN(CC3)c4c(cccn4)C(F)(F)F SEW06438 COc1ccc(cc1)C2c3ccsc3CCN2C(=S)Nc4ccc(cc4)OC SEW06439 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS00675 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(CSc4cccs4)O HTS00961 Cc1ccc(cc1)Sc2nc3ccc(cc3s2)Cl SEW01266 COc1ccc(cc1OC)S(=O)(=O)N2CCC(CC2)Cc3ccccc3 HTS00834 CC(CSc1ccc(cc1)Cl)C(=O)O SEW01350 COc1ccc(cc1)C(=O)NCCc2cccs2 SEW01481 c1ccc(cc1)S(=O)(=O)/C(=C/c2ccc(cc2)OCc3cc(cc(c3)F)F)/C#N SEW06627 CS(=O)(=O)/C(=C/c1ccc(cc1)OCc2cc(cc(c2)F)F)/C#N SEW06628 COc1cc(c(cc1OC)NC(=O)CSc2ccc(cc2)Cl)C(=O)OC GK03494 CN1CCN(CC1)c2cc(nc3c2cc(cc3)F)C(F)(F)F KM10688 Cc1ccc(n1c2c(c3c(s2)CCCC3)C(=O)NNC(=O)c4ccccc4)C GK03402 CCN1CCC(CC1)(C#Cc2ccccc2)O RJC03985 c1ccc(cc1)c2nc(sn2)N3CCCN(CC3)C(=O)c4ccc(cc4F)F HTS01148 c1ccc(cc1)C(CNCc2cccs2)O HTS00624 c1ccc2c(c1)CC(=C2)N3CCN(CC3)CCO HTS01270 c1cc(nc(c1)Oc2ccc(cc2)Cl)NS(=O)(=O)c3ccc(cc3)F HTS00313 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccc(c(c3)OC)OC RH01979 Cc1ccc2c(c1)C(C3(N2C)CCCC(=O)N3)(C)C RJC04042 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCN3CCCCC3 SPB08429 CC(C)NC(=O)CSc1nnc(n1CC=C)c2ccc3c(c2)cccn3 KM10657 c1cc(c(c(c1)Cl)CSCCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)F SEW06508 c1cc(sc1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F SEW06504 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 HTS00649 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCc3nc(no3)c4ccc(cc4)C(F)(F)F HTS00662 C/C(=N\NC(=S)N)/COc1ccc(cc1)c2csnn2 SEW01197 CC(C)NC(=O)c1cc(nn1Cc2ccc(cc2Cl)Cl)C(C)(C)C SPB08249 Cc1cc(nn1C(C)(C)C)C(=O)Nc2ccccc2 SPB08251 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(on3)C)C GK03410 CCCSc1c(cccn1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl PD00699 CCCSc1c(cccn1)C(=O)Nc2ccc(cc2)OC(F)(F)F PD00700 CCOC(=O)NNC(=S)Nc1ccccc1N2CCOCC2 SPB07667 c1ccc2c(c1)c(c[nH]2)CCNC(=O)CC(CC(=O)O)c3ccc(cc3)C(F)(F)F PD00593 CCCc1ccc(cc1)C(=O)Nc2cccnc2Oc3ccc(cc3)C(C)(C)C RH01980 Cc1ccccc1NC(=O)NCc2ccc(cc2)Cl KM10710 Cc1nc(cn1CC(=O)c2ccc(cc2)Cl)[N+](=O)[O-] RH02128 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2ccc(cc2F)F)C SEW06449 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2ccccc2OC)C SEW06452 c1ccc(c(c1)NC(=S)Nc2ccccc2F)F SEW04256 CCOC(=O)C(=NNc1ccc(cc1[N+](=O)[O-])OC)C(=O)OCC SEW01554 c1ccc(cc1)C(C2CCCC2)C(=O)Nc3cccnc3Sc4ccc(cc4)Cl RH02118 c1cc(sc1)c2nc(sn2)N3CCN(CC3)C(=O)c4ccc(cc4Cl)F SPB08320 CCOC(=O)c1c(n(c(c1S(=O)(=O)N)C)c2ccccc2)C SP01164 c1cc(c(cc1Cl)C2CCCCC2)Oc3ccc(cn3)NC(=O)C4CCCCC4 HTS00901 Cc1ccc2c(c1)C(C(=N2)C)(C)C.Cl RJC04033 COc1ccc(c(c1OC)Cl)/C=C/C(=O)Nc2ccc(c(c2)C(=O)OC)N3CCOCC3 HTS00924 CS(=N/C=C(\C#N)/S(=O)(=O)c1ccc(cn1)C(F)(F)F)(=O)c2ccc(cc2)Oc3cccc(c3C#N)F KM06611 Cn1c2c(cn1)c(ncn2)O/N=C(/c3cc(cc(c3)C(F)(F)F)C(F)(F)F)\N GK03532 COc1ccccc1N2CCN(CC2)CCCCNS(=O)(=O)c3ccc(c(c3)Cl)Cl SEW06441 Cn1cc(cc1C(=O)OC)/C=N/NC(=S)NC2CC3CC2C=C3 SEW06443 c1ccc(cc1)c2csc(n2)CSCC(=O)NNC(=S)Nc3ccc(cc3)Cl KM05943 CSC(=CC(=O)c1nccs1)SC SEW02761 c1cc(c(cc1F)Cl)S(=O)(=O)N SEW03823 Cc1ccc(cc1Cl)NC(=O)Nc2ccc(c(c2)Cl)C PD00701 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3)F GK03413 c1ccc2c(c1)ccn2c3ccc(cc3)[N+](=O)[O-] SEW06426 Cn1cc(cc1C(=O)OC)/C=C\2/c3ccccc3NC2=O SEW06435 COc1ccc(cc1)c2cc3c([nH]2)c4ccccc4oc3=O PD00833 Cc1ccc(c(c1)Cl)C(=O)C(C)c2c(c3ccccc3oc2=O)O PD00834 c1ccc2c(c1)c(c(c(=O)o2)CC(=O)c3ccc(cc3)C(F)(F)F)O PD00837 Cc1ccc(cc1F)c2nc(cs2)c3ccc4c(c3)OCCO4 SPB08219 Cn1c(ccc1S(=O)(=O)N(C2CCCCC2)C3CCCCC3)C(=O)OC HTS01745 CC(C)(C)C(=O)Nc1c(c(nn1C)C(F)(F)F)c2ccc(cc2)Br HTS00348 CCc1cccc(c1NC(=O)Nc2c(cnn2C)Br)C GK03412 Cn1c(c(cn1)Br)NC(=O)Nc2cccc3c2cccc3 GK03414 CCOC(=O)c1ccc(cc1)n2c(cc(n2)C(C)(C)C)C(C)(C)C SEW06520 Cc1c(c(c(n1C)C)S(=O)(=O)N2CCOCC2)C(=O)OC SP01171 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)OC GK03396 c1ccc(cc1)CNCC(c2ccccc2)O AW00958 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3)Cl GK03401 CS(=N/C=C(\C#N)/C(=O)c1cccs1)(=O)c2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-] KM06753 CC1(c2ccccc2N3C1(NC(=O)CC3)/C=C/c4cccs4)C RJC04041 CN1CCN(CC1)S(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 KM10747 c1ccc(cc1)CN2CCC(CC2)(C#Cc3ccccc3)O RJC03986 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2ccc(cc2)Cl)C SEW06446 c1cc2c(c(c1)S(=O)(=O)NCCSCc3c(cccc3Cl)F)non2 HTS01722 CCCCNC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(on2)C GK03403 Cc1cc(cc(c1)NC(=O)Nc2c(cnn2C)Br)C GK03411 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2cccc(c2)C(F)(F)F SP01217 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nc(cs3)c4ccc5c(c4)OCCO5 SPB08222 Cc1ccc2c(c1)C(C3(N2CC(=O)N3Cc4ccccc4)C)(C)C RJC04036 c1ccc(cc1)c2csc(n2)CC#N RJC03997 Cc1ccc(cc1)C(=O)N2CCN(CC2)CC(=O)Nc3cc(sc3C(=O)N)c4ccccc4 GK03775 Cc1ccc(cc1)C(=O)N2CCN(CC2)CC(=O)Nc3cc(sc3C(=O)C)c4ccccc4 GK03776 c1cc(ccc1CC(=O)NCCNC(=O)/C=C/C(=O)O)O AW01196 COc1cc(c(cc1OC)NC(=O)c2ccco2)C(=O)O GK03481 COc1cc(c(cc1OC)NC(=O)c2cccs2)C(=O)O GK03482 CC(C)(C)OC(=O)C(C)(C)ONC(=O)Nc1ccc(cc1)Cl RF04666 c1cc(ccc1/C=N/c2ccc(cc2)OCC(CN3CCCCC3)O)Cl AW01127 COc1ccc(c(c1)OC)CNC(=O)c2cnc(cc2C(F)(F)F)OC RF04460 COc1cc2c(cc1OC)C(=O)CC2c3ccccc3 HTS01504 c1ccc(c(c1)C(F)(F)F)n2c(nnn2)c3ccc(cc3F)F RF04544 CCOC(=O)c1c(csc1NC(=O)c2cccs2)c3ccc(cc3)Br AW01138 C=CCC1(CCCCC1)NC2CCCCC2.Cl RJC03987 c1cc(ccc1C#N)N2CCN(CC2)C(=O)c3ccc(cc3)OC(F)(F)F SPB08308 Cc1nc(cn1CC(=O)c2ccc3c(c2)OCO3)[N+](=O)[O-] HTS01298 c1cc(sc1)c2ccnn2C(=O)Cc3cc(cc(c3)F)F SEW06417 c1cc(sc1)C(=O)Nc2ccc(cc2)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW06432 Cn1c(ccc1S(=O)(=O)NCCc2ccccc2OC)C(=O)OC HTS01742 Cc1ccc(c(c1)NC(=O)Nc2cccc(c2)C(F)(F)F)n3cccc3 SEW06510 c1ccc2c(c1)nc3c4cc(ccc4n(c3n2)CC(=O)NN)F RH02022 CC(C)Cc1ccc(cc1)C(C)c2nnc(o2)c3cccc(c3)[N+](=O)[O-] SEW06521 c1cc(sc1)SCCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06522 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)CCSc2cccs2)/N SEW01792 CSC(=N)Nc1ccc(c(c1)Cl)Cl.I RDR00795 c1cc(ccc1N2CC(=O)N(CC2=O)Cc3ccc4c(c3)OCO4)OC(F)(F)F PD00693 c1cc(ncc1C(F)(F)F)N2CCN(CC2)CC(c3cc(no3)c4cc(cc(c4)Cl)Cl)O HTS01400 CC(C)Nc1nccc(n1)C(F)(F)F AW00985 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)C(=O)Nc3ccc(cc3)F HTS00394 CCOC(=O)CN(c1ccc(cc1)F)C(=O)c2c(onc2c3ccccc3Cl)C PD00692 Cc1ccc(cc1)Sc2c(cccn2)NS(=O)(=O)c3ccc(cc3)Cl RH02105 c1cc(ccc1C(C[N+](=O)[O-])Sc2ccc(cc2)N)F PD00794 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)OCC)C#N SPB08424 Cc1ccc(cc1)Sc2c3c(ccs3)ncn2 GK03792 CC(C)Oc1c2ccc(cc2sc1C(=O)OC)Cl RH02264 Cc1nc(cs1)C23CC4CC(C2)CC(C4)C3 SPB08312 CN1CCN(CC1)c2ccc(cc2)NS(=O)(=O)c3cccc(c3)C(F)(F)F SS00029 CC(C)(C)C(=O)N1CCN(CC1)c2c3c(csc3ncn2)c4ccccc4 AW01136 c1ccc2c(c1)OCC(O2)C(=O)Nc3cccc(c3)c4cnco4 HTS01992 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)/C=C/C(=O)O HTS01716 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)c2ccc(nc2C)C(F)(F)F HTS01575 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F HTS01576 c1cc2c(ccnc2cc1Cl)N3CCN(CC3)C(=O)CSCC(=O)O HTS01446 Cc1c(c(c(o1)C)S(=O)(=O)NCc2ccc3c(c2)OCO3)C(=O)OC HTS01715 c1ccc-2c(c1)CCc3c2sc(c3)C(=O)Nc4cccnc4 PD00617 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCN(CC3)c4nc5ccc(cc5s4)Cl AW00952 Cn1c2c(cn1)c(ncn2)NN3C(=O)CCC3=O GK03525 Cc1c(sc(n1)c2c(cc(cc2Cl)C(F)(F)F)Cl)C(=O)C SEW05034 Cc1ccc(cc1)Sc2c(cccn2)NC(=O)Cc3ccccc3 RH02087 COc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl RH02029 Cc1cc(no1)c2c(c(no2)C)C(=O)O SPB03205 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NCCN3CCOCC3 SPB08418 Cc1cc(nc(n1)Sc2ccccc2NC(=O)Nc3ccc(cc3)Cl)C(=O)OC SPB06397 c1cc(c(cc1NS(=O)(=O)c2cc(sc2Cl)Cl)C(F)(F)F)Br HTS01950 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)c3cc4ccccc4o3)C HTS01989 Cc1c(c(nc(n1)c2ccccn2)N3CCN(CC3)c4c5c(csc5ncn4)c6ccccc6)Cl AW01132 CC(C(=O)c1ccc(cc1)c2ccccc2F)N3CCN(CC3)c4ccc(cc4)C#N HTS01294 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3nc(cs3)c4ccccc4 HTS01312 c1ccc(cc1)CN2CCC(CC2)NC(=O)CC34CC5CC(C3)CC(C5)C4 HTS01101 CCCc1cnc(nc1)N2CCCN(CC2)S(=O)(=O)c3ccc(n3C)C(=O)OC HTS01547 CC(=O)c1c(cc(s1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)OC(F)(F)F GK03773 c1cc(ccc1S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl)Cl AW00954 c1ccc(c(c1)C(C[N+](=O)[O-])Sc2ccc(cc2)N)C(F)(F)F PD00795 COC(=O)c1ccc(o1)S(=O)(=O)N2CCCC2 SP01419 COc1cc(c(cc1Cl)OC)NC(=S)NNC(=O)c2ccc(cc2)[N+](=O)[O-] GK03675 CC(=O)c1ccc(cc1)NC(=O)CN2CCN(CC2)CC(=O)Nc3ccc(cc3)C(=O)C HTS01197 CCOC(=O)/C(=C/Nc1ccc2c(c1)OCO2)/C#N RH02199 Cc1cc(c(c(n1)OC)C#N)C(F)(F)F RH02201 c1ccc(c(c1)NC(=O)CSc2nnnn2c3ccc(cc3)O)Cl HTS01667 CN(C)/C=C/C(=O)C(c1ccccc1)c2ccccc2 CD11347 Cc1ccc(c(c1)NC(=O)Nc2ccccc2C(F)(F)F)n3cccc3 SEW06502 c1ccc2c(c1)cccc2c3cc([nH]n3)C(F)(F)F SP01352 COc1ccc(cc1OC2CCCC2)NC(=O)c3cccs3 HTS01369 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)N SEW04679 COC(=O)c1cccn1c2ccccc2[N+](=O)[O-] SEW04688 c1cc2c(cc1Cl)sc(n2)N3CCCN(CC3)S(=O)(=O)c4cc(c(cc4Cl)Cl)Cl AW00977 c1ccc(cc1)c2csc3c2c(ncn3)NCCNC(=O)/C=C/C(=O)O AW00981 COC(c1c(cnn1c2ccccc2)C(=O)OC)OC SPB05108 c1ccc(cc1)C2=NN=C(C=C(C2)c3ccc(cc3)Cl)c4ccccc4 HTS01278 Cc1cn(c2c1cccc2)CCC(=O)Nc3ccc(cc3)n4ccc(n4)C(F)(F)F HTS01432 CC(=O)c1ccc(cc1)OCC(CN2CCN(CC2)Cc3c(cccc3Cl)F)O AW01238 CN(C)c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3ccccc3Cl HTS01662 CC(C)(C)c1cc2c(s1)c(ncn2)NNS(=O)(=O)c3ccc(n3C)C(=O)OC HTS01558 Cc1c2c3ccccc3ccc2oc1C(=O)c4ccc(cc4)OC RH02210 CSc1cccc(c1)NC(=O)CN2CCOCC2 HTS01904 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)CN3CCOCC3 HTS01901 CC(C)(C)OC(=O)NCCNS(=O)(=O)c1ccc(n1C)C(=O)OC HTS01741 c1ccn(c1)c2ccc(cc2)/N=C\c3ccc(cc3)F SEW04793 COc1cc(c(cc1OC)[N+](=O)[O-])CC(=O)NN SEW04626 COc1cccc(c1NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl)Cl HTS00415 Cc1c(nc(s1)NS(=O)(=O)c2ccc(cc2)OC)CC(=O)OC HTS00844 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3ccc(cc3)OC)C HTS01285 c1cc2c(cc1C(=O)Nc3c(ccs3)C#N)CCO2 HTS00389 CN(C)c1ccc(cc1)n2c(nnn2)SCC(=O)c3ccc4c(c3)OCO4 HTS01659 COc1ccc(cc1)OCCNC(=O)c2ccco2 SPB08207 Cc1ccc(cc1)C(=O)Nc2ccc(c(c2)C(=O)OC)N3CCOCC3 HTS00918 COc1ccc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)Br BTB07608 c1cc(c(nc1)Oc2ccc(cc2)Cl)NS(=O)(=O)c3ccc(cc3)Cl RH02017 c1cc(c(nc1)NC(=O)c2cc(cc(c2)Cl)Cl)OCc3ccc(c(c3)Cl)Cl RH02024 c1ccc(c(c1)C(=O)N(Cc2cccnc2)Cc3ccc(cc3Cl)Cl)C(=O)O RF03580 CC1(OC(=O)C(=Cc2ccc(c(c2Cl)OC)OC)C(=O)O1)C RH02203 CCOC(=O)N1CCN(CC1)c2cc(cc(n2)C(F)(F)F)C(F)(F)F SPB08425 Cn1c(ccc1S(=O)(=O)NCCOC)C(=O)OC HTS01752 Cn1c(ccc1S(=O)(=O)NCc2ccc(cc2)OC)C(=O)OC HTS01754 COC(=O)c1ccc(n1c2ccc(cc2)F)/C=N/Nc3c(cccn3)[N+](=O)[O-] SEW04815 Cc1ccc(cc-2c(cc(c12)/N=N/c3ccccc3)C)C(C)C SEW04857 Cc1c(c(c(c(c1C)C)CSc2nnc(n2c3ccc(cc3)OC)CC#N)C)C CD02680 c1ccc(cc1)n2c(nnn2)c3cnc4ccccc4c3N HTS01279 c1ccc2c(c1)c(c(cn2)c3nnnn3c4ccc(cc4)F)N HTS01280 Cc1csc2c1ncnc2NCCCN3CCOCC3 HTS00106 c1cc(ccc1n2c(nnn2)SCC(=O)c3ccc4c(c3)OCO4)O HTS01664 COC(=O)c1c(cc(s1)c2cccs2)NC(=O)/C=C\C(=O)O HTS01037 CCOc1ccccc1N2CCN(CC2)C(=O)c3cc4cc(ccc4[nH]3)OC HTS01093 c1cc(cc(c1)Cl)S(=O)(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O HTS00212 Cc1ccc(c(c1)NC(=O)C)OCC(=O)c2ccc(cc2)OC RH02202 CC(C)c1ccc(cc1)S(=O)(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH02015 COc1ccccc1NS(=O)(=O)c2ccc(s2)Cl KM01052 CCCS(=O)(=O)/C(=N/Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C#N KM01567 c1ccc(cc1)CN(Cc2cccs2)C(=O)c3ccc(cc3)Cl RF03298 Cc1ccc2cc(ccc2n1)NC(=O)c3cccs3 RH02214 Cc1ccc(n1c2ccc(cc2)n3cccc3)C SEW04800 c1ccc(cc1)c2csc3c2c(ncn3)N4CCC(CC4)NC5CCCCC5O AW00995 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Nc3ccccc3Cl SPB08241 Cc1ccc(cc1)/N=C/c2ccc(cc2)Cl SEW04894 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Nc3cccc(c3)C(F)(F)F SPB08242 c1cc2c(cc1C(=O)N3CCCCC3)nns2 KM10684 CS(=O)(=O)c1ccc(cc1)C(=O)Nc2cccc(c2)Cl TG00187 Cc1cc(c2ccccc2n1)OCC(=O)N(c3ccccc3)C4CCCCC4 HTS01171 Cc1ccc(c2c1c(ccn2)OC(C)C(=O)N3CCN(CC3)c4ccccc4OC)C HTS01173 CC(C)(C)OC(=O)N1CCC(CC1)Nc2ccc(cc2)OC CC00005 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3cccs3 HTS00920 CCOC(=O)C1CCN(CC1)c2ccc(cn2)[N+](=O)[O-] SPB08216 c1cc(ccc1c2nc(cs2)c3ccc4c(c3)OCCO4)C(F)(F)F SPB08221 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)c4cccc(c4)Cl)[N+](=O)[O-] HTS00283 CC(C)(C)C(=O)N1CCN(CC1)c2ccc(cc2n3cccc3)[N+](=O)[O-] HTS00285 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)F)c4ccc(c(c4)Cl)Cl HTS00683 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3cccc(c3)OC(F)(F)F SPB08237 CSC(=NS(=O)(=O)c1ccccc1)SC CD03004 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)C(=O)Nc3cccc(c3)Cl SPB08247 CCOC(=O)c1c(c2cc(ccc2nc1SC)Cl)N3CCCCCC3 KM10687 c1cnc(c(n1)C(=O)N2CCN(CC2)CCO)C(=O)O HTS01069 c1cc(oc1C(=O)N2CCOCC2)S(=O)(=O)N3CCOCC3 HTS00432 Cc1ccc(cc1)S(=O)(=O)Nc2csc(c2C(=O)O)C HTS00435 Cc1cn(c2c1cccc2)CCC(=O)Nc3ccc(cc3)OC HTS01098 COc1ccc(cc1OC)CC(=O)NNC(=S)NCC2CC2 PD00799 c1cc(ccc1C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3)F HTS00909 c1cc2c(cc1c3csc(n3)CC#N)OCCO2 SPB08214 c1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3n4cccc4)[N+](=O)[O-] HTS00280 c1ccc(cc1)c2cc(nc(n2)SCC(=O)N3CCOCC3)O HTS00688 c1ccc2c(c1)c(=O)n(c(n2)SCC(=O)c3ccc(s3)Cl)c4ccc(c(c4)Cl)Cl HTS00685 Cc1c(c(no1)c2ccccc2)CO CC00509 CCC(C)c1ccc(cc1)NC(=O)c2cc(nn2Cc3ccc(cc3)F)C(C)(C)C SPB08243 c1c(cc(c(c1[N+](=O)[O-])NCCN)[N+](=O)[O-])C(F)(F)F CD03702 CCc1cccc(c1NC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(on3)C)C GK03399 Cc1csc2c1c(=O)[nH]c(n2)CN3CCOCC3 GK03784 CCCc1c(cnn1c2cc(cc(c2)Cl)Cl)C(=O)O SP01487 c1ccc2c(c1)cnn(c2=O)CCOC(=O)c3ccc(cc3Cl)F PD00595 COc1cccc(c1)Cn2c-3c(c4ccccc4c2=O)C(=O)c5c3cccc5 PD00705 c1cc(sc1)C(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F AW01007 CCCCCC(=O)n1c2ccc(cc2c3c1nc4ccccc4n3)F RH02010 CCC(C)Nc1c2cc(c(cc2ncn1)OC)OC GK03387 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCC(CC2)c3nc(no3)c4ccc(cc4)Cl SEW06515 COc1ccc2c(c1)cc([nH]2)C(=O)N3CCC(CC3)Cc4ccccc4 HTS00776 Cn1c(ccn1)NC(=O)c2ccc(cc2)F GK03342 Cc1ccc(n1c2c3c(cccc3F)n(n2)S(=O)(=O)c4cccc5c4non5)C HTS01081 COc1ccc(c(c1)SCCC(=O)O)OC SEW01631 c1cc2c(cc1NCC(=O)c3cc4cc(ccc4o3)Cl)OCCCO2 HTS00130 c1cc(c(cc1Cl)Cl)CSc2c3c4c(sc3ncn2)CCCC4 GK03392 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)c3ccc(cc3)C SS00008 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)N3CCN(CC3)Cc4ccccc4 SS00010 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)Cc3ccccc3 SS00012 COc1cc(c(cc1OC)CO)CC(=O)NN CD01926 CC12CCCCC1=[N+](c3c2cccc3)C.[I-] RJC04034 CC1(c2ccccc2N3C1(N(C(=O)C3)CC=C)C)C RJC04035 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)C4CC4)[N+](=O)[O-] HTS00281 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)c3nc4ccc(cc4s3)Cl)F HTS01137 Cn1cc(cc1C(=O)OC)/C=N/NC(=O)c2cccnc2 SEW06436 c1cc(oc1)C(=O)N2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F SEW06507 CC(C)(CC(=O)Nc1c2ccccc2n(n1)C)CC(=O)O HTS00773 c1cc(cc(c1)NC(=O)c2ccc(cc2)[N+](=O)[O-])c3nnco3 SEW01219 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3cccnc3 SPB08239 Cc1c(oc(n1)C)c2ccn(n2)S(=O)(=O)c3ccccc3Cl SEW01592 Cc1c(c(on1)C)C(=O)n2ccc(n2)c3c(nc(o3)C)C SEW01595 c1ccc(cc1)c2c(nnn2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NC(=O)Nc4c(n(nn4)c5cc(cc(c5)C(F)(F)F)C(F)(F)F)c6ccccc6 CD05765 c1ccc(cc1)CN2CCN(CC2)c3c(cccn3)[N+](=O)[O-] SS00004 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccccc3 GK03397 CCOc1cc(c(cc1N2CCOCC2)OCC)NS(=O)(=O)C SS00014 c1cc(oc1)C(=O)N2CCN(CC2)c3ccc(cc3)C#N SPB08324 CC(=O)N1C(CC(=N1)c2cccc(c2)[N+](=O)[O-])c3ccccc3 RJC04103 Cc1ccc(cc1)C2=NN(C(C2)c3ccc(cc3Cl)Cl)C(=O)C RJC04105 COc1ccc(cc1OC)S(=O)(=O)N(CCC#N)C2CCCc3c2cccc3 KM09301 c1ccc(cc1)C2C3COc4ccccc4C3=NN2c5ccccc5 RJC04108 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)c3nnc(n3c4ccccc4)SC SPB08183 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)c3nnc(n3c4ccccc4)SCC#C SPB08184 CCOC(=O)N/N=C(\C)/c1c(cc(o1)C)C SEW00668 Cc1c(c(sc1C(=O)OC)SC)S(=O)(=O)c2ccc(cc2)Cl KM01675 Cc1ccc(cc1)n2c(nnn2)c3ccccc3C(F)(F)F RF04538 Cc1csc(c1N(C)C)C(=O)NN GK03384 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(on3)C GK03389 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cnn(c3C(F)(F)F)c4ccc(cc4)[N+](=O)[O-] GK03390 CC(C)C(=O)NNC(=O)CSc1c2cc(c(cc2ncn1)OC)OC GK03394 CCSc1c2c3c(sc2ncn1)CCCC3 GK03400 CC(C)(C)OC(=O)NC1CCN(CC1)c2nccc(n2)C(F)(F)F AW00950 Cc1ccc(cc1)N/N=C(\C#N)/C(=O)c2ccccc2OC(F)(F)F KM04881 c1ccc2c(c1)ncc(n2)N3CCC(CC3)C(=O)NC(=O)N4CCCC4 SEW04047 c1ccc(c(c1)C(F)(F)F)NC(=S)N2CCCC2 SEW04263 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11057 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)c4ccnc5c4ccc(c5)Cl KM11058 CC(C)(CC(=O)Nc1c2c(cccc2F)n(n1)C)CC(=O)O HTS00774 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)c3nc(no3)c4ccc(cc4)Cl SEW06516 c1cc(sc1)C(=O)N2CCC(CC2)c3nc(no3)c4ccc(cc4)Cl SEW06518 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)c3nnc(n3C)S SPB08174 Cc1c(c([nH]c1c2ccccc2)C(=O)OC)C(=O)OC SEW01736 Cn1c(c(cn1)Br)NC(=O)Nc2ccc(cc2)Cl GK03409 CCOc1cc(c(cc1N2CCOCC2)OCC)NS(=O)(=O)C(C)C SS00016 Cc1ccc(cc1)N/C=C(\C#N)/C(=O)c2ccccc2OC(F)(F)F KM04811 CCOc1c2cc(c(cc2ncn1)OC)OC GK03398 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCNc2c(cc(cn2)C(F)(F)F)Cl AW01171 c1ccc(c(c1)C#N)n2cccc2 CD03418 C/C=C/C(=O)Nc1ccc(cc1)N2CCN(CC2)C SS00030 CCOC(=O)N/N=C/1\CCCc2c1cccc2 SEW00611 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCC(CC3)c4nc(no4)c5ccc(cc5)Cl SEW06513 Cc1ccc(c(c1)NC(=S)Nc2ccc(cc2)C(C)(C)C)n3cccc3 SEW06500 Cc1ccc(c(c1)NC(=S)Nc2c(cccc2Cl)C)n3cccc3 SEW06501 c1cc(c(nc1)NS(=O)(=O)c2ccc(cc2)Cl)OCc3ccc(c(c3)Cl)Cl RH02027 c1cc(c(nc1)NS(=O)(=O)c2ccc(cc2)Br)OCc3ccc(c(c3)Cl)Cl RH02028 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc(s4)Cl.Br HTS00030 CCOC(=O)c1c(oc(c1S(=O)(=O)N2CCOCC2)C)C SP01170 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)C(=S)NC5CCCCCCC5 AW01175 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)C(=O)CCC(=O)O AW01176 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3ccc4c(c3)OCO4 PD00691 Cc1ccc2cc(ccc2n1)NC(=O)Cc3ccccc3 RH02217 c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4cccc(c4)Br KM09362 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3c(onc3c4c(cccc4Cl)Cl)C)C HTS01309 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4nc(ns4)c5cccs5 SPB08309 Cc1ccc(cc1)c2nnco2 SEW01491 COC(=O)c1cc(ccc1N2CCOCC2)NS(=O)(=O)c3cccc(c3)Cl HTS01363 c1c(cc(cc1Cl)Cl)S(=O)(=O)N2CCN(CC2)C(=O)CSCC(=O)O HTS01170 c1ccc2c(c1)CCC2NCC(COc3ccc(cc3)c4csnn4)O HTS03852 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)NCc3cccnc3 HTS03713 CC(=O)c1ccc(c(c1)C(=O)NC2(C(=O)c3ccccc3C2=O)O)O HTS01851 CCOc1cc(c(cc1N2CCOCC2)OCC)NS(=O)(=O)c3ccc(cc3)OC HTS00117 CN1CCN(CC1)c2ccc(cc2)NC(=O)c3ccco3 SS00027 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)c3ccc(cc3F)F SS00031 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)c3ccco3 SS00032 c1ccc(cc1)COc2ccc3c(c2)cc([nH]3)C(=O)O KM10299 c1ccc2c(c1)C3(C(=O)N2CN4CCCCCC4)OCCO3 HTS00589 Cc1cc(ccc1NC(=O)CC(C)(C)CC(=O)O)C(C)(C)C HTS02062 CC(c1ccccc1)NS(=O)(=O)c2ccc(cc2)c3cc(sc3C(F)(F)F)C(=O)OC HTS03717 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnn3C(=O)Nc4ccc(cc4)C(C)(C)C HTS04114 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(c(c2)C#N)C(F)(F)F SP01219 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)S(=O)(=O)c4ccccc4OC(F)(F)F HTS00114 COc1cc(cc(c1OC)OC)C(CC(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F)CC(=O)O HTS00585 c1ccc(cc1)c2cc3c(s2)c(ncn3)NCc4ccc5c(c4)OCO5 HTS00601 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3coc4ccccc4c3=O HTS00149 CC(C)(C)C(=O)Nc1c(c(nn1C)C(F)(F)F)c2cccc(c2)C(F)(F)F HTS00350 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)sc(n3)SC KM10783 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCCN(C)C AW01002 CN(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C(F)(F)F HTS00119 c1cc(ccc1OCc2nc(cs2)c3ccc4c(c3)OCCO4)Cl SPB08229 CC(C)(C)c1ccc(cc1)/C(=N/Oc2c3cnn(c3ncn2)C)/N GK03544 CC(C)(C)OC(=O)NCCNC(=O)c1cccs1 AW01248 c1ccc2c(c1)c(=O)c(co2)N3CCCCC3 HTS00122 Cc1cccc(c1)NC(=O)c2cc(oc2C)C(C)(C)C SP01216 COc1ccc(cc1)C2C3CSc4ccccc4C3=NN2c5ccccc5 RJC04109 COc1cccc(c1)CC(=O)NCCCNc2c(cc(cn2)C(F)(F)F)Cl AW01179 Cc1nc(cs1)c2ccc(cc2)NC(=O)Cc3cccc(c3)OC AW01185 COc1cc(cc(c1OC)OC)/C=C/2\CCc3ccccc3C2=O PD00619 CCOC(=O)N/N=C(\C)/c1ccc(cc1)C(F)(F)F SEW00664 c1ccc(c(c1)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-])Cl SEW00905 c1ccc(c(c1)C(F)(F)F)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] SEW00906 c1ccc(cc1)CNC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] SEW00907 c1cc(c(nc1)Oc2ccc(cc2)Cl)NS(=O)(=O)c3ccc(cc3)C(F)(F)F RH02018 Cc1cc(c2ccccc2n1)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)F HTS00070 CCOC(=O)C(C1Cc2ccccc2C1=O)(C(=O)OCC)O HTS00078 CCOC(=O)c1cc(c(cc1NS(=O)(=O)c2cn(cn2)C)OCCOC)OCCOC HTS00093 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)N3CCOCC3 SPB08240 Cc1c(cc(o1)C(C)(C)C)C(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SP01213 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccccc2 SP01214 COC(=O)c1c(cc(s1)c2cccs2)NC(=O)c3cccs3 GK03704 Cn1c(nnc1SCc2ccccc2)CNC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM10711 Cc1cc(cc(c1)N2C(=O)CC(C2=O)Sc3ccccc3C(=O)O)C PD00829 CCOC(=O)c1cc(c(nc1NCc2ccc3c(c2)OCO3)C)C(=O)OC AW01009 CCOC(=O)c1c(c(sc1NC(=O)c2ccco2)C)c3ccccc3 AW01010 CC(C)(C)[C@H]1COC(=N1)C(C)(C)C2=N[C@H](CO2)C(C)(C)C RJC04047 Cc1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccc(cc3)OC HTS01630 Cc1cccc(c1)CSc2nnc(n2c3ccc4c(c3)OCO4)c5ccc(cc5)C(C)(C)C HTS02051 c1cc2c(cc1C(=O)O)nsn2 CC09201 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)OC)c3cccs3 GK03702 c1ccc(cc1)C2=NNC(C2)(C(F)(F)F)O KM10712 c1ccc(cc1)C(=O)CSc2nccc(n2)c3cccs3 HTS04397 c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cccs3 HTS04399 CC(=O)NC(=O)/C(=C/NCc1cccs1)/C#N KM09185 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)c3ccccc3 SS00018 Cc1c(nc(s1)C)CC(=O)O TL01023 CNC(=O)NNc1ccc(cc1)c2csnn2 SEW01043 CCOC(=O)N/N=C(\C)/c1ccc(cc1)Br SEW01073 c1ccnc(c1)c2ccc(s2)CO CC02209 c1cc(c(cc1C(F)(F)F)Cl)/C=C/[N+](=O)[O-] SEW01610 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(ccc3N4CCc5ccccc5C4)C(F)(F)F HTS01380 CSc1cccc(c1)NC(=O)CSCc2ccc(cc2)Cl HTS01908 CCc1ccc(cc1)NC(=S)NNC(=O)C(C)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01890 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCc3ccc(c(c3)Cl)Cl PD00804 COc1ccc(c(c1OC)Cl)/C=C(\C#N)/C(=O)OC RH02221 C/C(=N\OC(=O)c1ccco1)/c2ccccc2O CD03672 Cc1cc(nc(n1)Sc2ccccc2NC(=O)c3ccc(cc3)OC)C(=O)OC SPB06394 CCOc1cc(c(cc1N2CCOCC2)OCC)NC(=O)C(C)(C)C SS00017 CC(=O)Nc1c(ccs1)C#N GK03793 COC(=O)/C=C(/c1ccccc1)\n2cnc3c2cccc3 KM10810 c1cc(ccc1C(=O)NNc2c3c(ccs3)ncn2)Cl GK03797 CCOC(=O)/C(=C/Nc1cc(ccn1)C)/C#N RH02198 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCCCN3C(=O)c4ccccc4C3=O AW01027 Cc1c(oc(n1)C)/C(=N/O)/C SEW01646 c1cc(ccc1OCc2ccsc2C#N)Cl SEW01661 c1ccc(cc1)CCN2CCCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl HTS01808 c1cc(ccc1S(=O)(=O)Cc2ccsc2C#N)Cl SEW01664 CCOC(=O)c1c(c(sc1Nc2ccccc2)[N+](=O)[O-])N SEW01715 c1ccc2c(c1)cc(o2)C3=NNC(C3)(C(F)(F)F)O KM10716 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)NCc2ccco2)C)C CD03694 Cn1c(c(cn1)C(=O)O)NNC(=O)CCC(=O)O GK03789 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CC(=O)Nc3cc(sc3C(=O)N)c4ccccc4 GK03794 Cc1ccc(cc1)Sc2c(cccn2)C(=O)OC RH02266 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)c3ccccc3 HTS01628 c1ccc(cc1)c2nnc(o2)C(=O)NC(=O)N3CCOCC3 SEW01682 CCOC(=O)/C(=C\c1ccc(cc1)n2c(ccc2C)C)/C#N SEW01692 CC(C)(C)c1cc(n(n1)C(=O)c2ccc(cc2)Cl)C(C)(C)C SEW06667 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CC(=O)Nc3cc(sc3C(=O)C)c4ccccc4 GK03795 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3c4c(cc(s4)c5ccc(cc5)C(C)(C)C)ncn3 GK03796 CCCc1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccc(cc3)OC HTS01430 Cc1cc(no1)NC(=O)CC2(CCCCC2)CC(=O)O PD00737 Cc1ccc(cc1)Sc2c(cccn2)c3nnc(o3)c4ccccc4 HTS01016 c1ccc(cc1)c2cc(c(c(n2)S/C=C(/c3cc4ccccc4o3)\O)C#N)C(F)(F)F HTS01845 Cc1c(c(nc(n1)c2ccccn2)N3CCOCC3)Cl AW01183 c1cc2c(cc1Cl)-c3c(c(n[nH]3)N)CS2 SEW01734 Cn1c2c(cn1)c(ncn2)N/N=C/c3ccccc3 GK03551 Cn1c2c(cn1)c(ncn2)n3c(c(cn3)C#N)N GK03552 Cc1c(c(no1)c2ccccc2)c3nc(no3)CSc4[nH]c5ccccc5n4 SEW06661 Cc1cn(c2c1cccc2)CCC(=O)NCc3c(cccc3Cl)F HTS01431 Cc1cn(c2c1cccc2)CCC(=O)Nc3c4ccccc4n(n3)C HTS01435 Cc1cn(c2c1cccc2)CCC(=O)Nc3c4c(cccc4F)n(n3)C HTS01436 Cc1c(snn1)C(=O)NC2CCN(CC2)Cc3ccccc3 HTS01676 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)c3ccccc3 HTS01627 Cc1ccccc1n2c3c(c(=O)n(c2=O)CCc4ccccc4)[nH]cn3 KM09803 COc1ccc(cc1)NC2CCN(CC2)Cc3ccccc3 SPB08401 CC(C)(C)NC(=S)NC1CCN(CC1)Cc2ccccc2 SPB08441 COc1c(c(ccn1)C(F)(F)F)C(=O)NC(=O)Nc2ccc(cc2)Cl RF04651 c1ccc(c(c1)C(F)(F)F)n2c(nnn2)c3ccc(cc3Cl)Cl RF04541 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)[N+](=O)[O-] RJC04055 COC(=O)c1c(cc(s1)c2cccs2)NC(=O)CSCC(=O)O HTS01470 COc1ccc(cc1)Oc2ccc(cc2NC(=O)c3ccc(cc3)OC(F)(F)F)C(F)(F)F HTS00852 c1ccc(cc1)c2cc(c3ccccc3n2)NCCN RH02021 COc1cccc(c1)NC(=O)c2cc(c(c(c2)OC)OC)OC JFD02686 c1ccc2c(c1)c(cc(n2)C(F)(F)F)OCC(=O)Nc3ccc4c(c3)OCO4 HTS01177 Cc1c(c(nc(n1)c2cccnc2)N3CCCN(CC3)Cc4ccc(cc4)F)Cl AW01182 c1cc(ccc1Oc2nccc(n2)C(F)(F)F)I AW01189 c1ccc2c(c1)[nH]c(n2)c3cccc(c3)NC(=O)c4ccc(cc4)F HTS00908 COc1ccc(cc1)c2csc(n2)CN3CCN(CC3)c4ccccc4OC SEW06634 COc1c(c(ccn1)C(F)(F)F)C(=O)Nc2ccc(cc2Cl)Cl RF04601 c1cc(c(c(c1)F)NC(=O)NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)F RF04587 Cc1cccc(c1n2c(=O)n(c(=O)s2)CC3CC3)Cl HTS01833 Cc1c(cc(o1)c2ccccc2)C(=O)Nc3ccc(cc3)C(C)(C)C SP01185 Cc1c(cc(o1)c2ccccc2)C(=O)Nc3cccc(c3)C(F)(F)F SP01186 c1ccc(cc1)CCN2CCCN(CC2)S(=O)(=O)c3cc(sc3Cl)Cl HTS01807 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)COCC(=O)O HTS01455 Cc1c(c(c(o1)C)S(=O)(=O)NCc2csc3c2cc(cc3)Cl)C(=O)OC HTS01712 CNC(=S)N(Cc1ccccc1)Cc2cccnc2 RF03337 c1cc(cc(c1)OCNCCCCCCO)[N+](=O)[O-] RH01969 C1CC(=C(C(=O)C1)Br)O RH01970 c1cnc(c(c1O)[N+](=O)[O-])O SPB07414 c1ccc(c(c1)OCc2nc(on2)C(=O)NN)Cl SPB01580 c1cc2c(cc1F)c(cc(n2)C(F)(F)F)N3CCOCC3 KM10689 c1cc(ccc1c2nc(cs2)c3ccc4c(c3)OCCO4)Oc5ccc(cn5)C(F)(F)F SPB08220 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)Nc4ccc5c(c4)OCO5 HTS00241 c1cc(sc1)C(=O)Nc2ccc(c(c2)C(F)(F)F)Br HTS01941 c1ccc(cc1)Cc2cc(nn(c2=O)CCC(=O)O)c3ccc(cc3)F HTS01683 Cn1c(ccc1S(=O)(=O)NCCNc2c(cc(cn2)Cl)C(F)(F)F)C(=O)OC HTS01544 c1ccc2c(c1)C(C3CCCCC3(O2)N4CCCC4)O CD03662 c1ccc(cc1)c2csc3c2c(ncn3)NCCNS(=O)(=O)c4ccc(cc4)Cl AW01015 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)N4CCN(CC4)c5ccccc5 HTS01212 c1ccc(cc1)N2CCN(CC2)C(=O)CN3CCCCCC3 HTS01217 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS01219 Cn1c2c(c(cc(n2)c3cccc(c3)F)c4ccc(cc4)F)c(=O)n(c1=O)C PD00622 COc1cc(cc(c1OC)OC)c2c3c(nc(c2C#N)OC)-c4ccccc4CC3 PD00623 c1cc(ccc1C(=O)Nc2ccc(c(c2)C(F)(F)F)Br)C(F)(F)F HTS01946 COc1ccc(cc1OC)S(=O)(=O)Nc2ccc(c(c2)C(F)(F)F)Br HTS01949 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)c3ccc4c(c3)OCO4)C HTS01981 c1ccc2c(c1)cc(o2)/C(=C/Sc3c(c(c4c(n3)CCCC4)C(F)(F)F)C#N)/O HTS01849 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])C(=O)OC HTS01551 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)Cc3cccc(c3F)Br)C(=O)OC HTS01553 Cn1c(ccc1S(=O)(=O)NNC(=O)c2ccc(cc2)Cl)C(=O)OC HTS01555 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3ccc(c(c3)OC)OC)C RH01972 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccccc3Cl RH01978 c1cc(c(cc1NC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F)C(F)(F)F)Br HTS01942 c1ccc2c(c1)OCC(O2)C(=O)Nc3ccc(c(c3)C(F)(F)F)Br HTS01945 Cc1cc(nn1C(C)(C)C)C(=O)NNS(=O)(=O)c2ccccc2C(F)(F)F HTS00056 COc1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc(cc3)F HTS01772 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc(cc3)F)C HTS01775 COc1ccccc1N2CCN(CC2)Cc3nc(cs3)c4ccc(cc4)Br SEW06523 COc1ccccc1NC(=O)N2CCCN(CC2)C(=O)c3cccs3 AW01018 c1ccc(cc1)c2csc3c2c4nnnn4cn3 AW01020 c1ccc(cc1)c2csc3c2c4nncn4cn3 AW01021 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)NCCCOC)C)C CD03695 CSc1c(cccn1)C(=O)NC2(C(=O)c3ccccc3C2=O)O HTS01952 CCOC(=O)/C(=C/Nc1ccc(cc1)F)/C#N HTS00300 COc1ccc(cc1)c2[nH]c(=O)nc(n2)c3ccncc3 NH00333 c1c(cc(cc1Cl)Cl)C(=S)NN NH00518 c1cc2cccnc2c(c1)S(=O)(=O)NCc3nc(no3)c4ccc(cc4)C(F)(F)F HTS00571 CCn1c(nnn1)SCC(=O)N2CCN(CC2)c3ccccc3 HTS01208 c1ccc2c(c1)c(nc(n2)c3cccs3)O RH02025 c1cc(sc1)c2nnc(o2)c3ccc(cc3)C(F)(F)F SEW06524 c1ccc2c(c1)cccc2/C=C/3\C(=O)C4CCN3CC4 PD00628 Cc1ccc(cc1C)/N=c\2/n(c(c(s2)NC(=O)C)c3ccc4c(c3)OCO4)C(=O)C CD03952 c1ccc(cc1)c2csc3c2c(ncn3)N4CCc5ccccc5C4 AW01167 CCCCCc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)OC(C)(C)C AW01115 CC(C)(C)NC(=O)N1CCN(CC1)c2c3c(csc3ncn2)c4ccccc4 AW01168 Cn1c2c(cn1)c(ncn2)N3CCN(CC3)C GK03471 C=CCn1c(nnc1SCc2c(cccc2Cl)Cl)c3ccc4c(c3)cccn4 KM10674 CCOC(=O)C1CCN(CC1)Cc2cccc(c2)NC(=O)c3cccs3 SPB08435 CCOC(=O)C1CCN(CC1)Cc2cccc(c2)NC(=O)c3cc(on3)C SPB08436 CCOC(=O)C1CCN(CC1)Cc2c(cccc2Cl)F SPB08224 Cc1c2c(ncnc2sc1c3ccccc3)O AW01166 Cc1cc(nn1C(C)(C)C)C(=O)NN SPB08431 Cc1cc(nn1C(C)(C)C)C(=O)NNS(=O)(=O)c2ccc(c(c2)OC)OC HTS00062 c1cc(sc1c2csc(n2)c3ccno3)Cl HTS00075 CC(C)(CC(=O)NNc1ccc(cc1)S(=O)(=O)N)CC(=O)O HTS04421 COc1ccc(cc1)CC2CCC3(CC2)NC(=O)c4ccccc4O3 HTS00605 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)S(=O)(=O)c4cccc(c4)Br HTS00124 c1ccc(cc1)c2csc(n2)CC(=O)N SB02074 c1ccc2c(c1)CC3C2=Nc4ccccc4SC3c5ccc(cc5)F JFD02639 CCOC(=O)C1CCN(CC1)Cc2cccc(c2)NC(=O)c3ccco3 SPB08437 C1C(CSc2c(sc(=S)s2)S1)O JFD04066 c1cc2cccc3c2c(c1)C(=O)C34OCCS4 JFD04068 CCS(=O)(=O)c1ccc(c(c1)NC(=O)Nc2ccccc2OC)O HTS04080 c1cc(c(c(c1)Cl)CSCCNC(=O)c2c(nccn2)C(=O)O)F HTS04413 Cc1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccc(cc3)Br HTS01637 CCCCCc1ccc(cc1)S(=O)(=O)Nc2cccnc2Oc3ccc(cc3)Cl RH02020 CN(C)c1c(cc(cc1F)C(=O)NC(=O)NC2=NCCS2)F SEW01895 Cc1cc(nc(n1)C)NC(=O)c2cc(oc2C)C(C)(C)C SP01221 c1cc(sc1)C(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl HTS00115 Cn1c2c(c(cc(n2)c3ccc(cc3)OC)c4ccc(cc4)OC)c(=O)n(c1=O)C PD00618 CCOC(=O)[C@H](C(C)C)NS(=O)(=O)c1cc(ccc1OC)Cl HTS00168 CC1(c2ccccc2N(C13C=Cc4c5ccccc5ccc4O3)CCC(=O)N)C RJC04043 CC1(c2ccccc2N3C14CC(C3C(=O)NC(C)(C)C)c5c6ccccc6ccc5O4)C RJC04044 CCc1ccc(cc1)C(=O)Nc2c(cc(cn2)C)Br HTS04002 c1ccc(cc1)N(C2CCCCC2)C(=O)CN3CCN(CC3)CCCc4c[nH]c5c4cc(cc5)F HTS01687 c1ccc(cc1)CNC(=O)C2CCC(N2)C(=O)NCc3ccccc3 KM09489 c1cc2c(c(c1)S(=O)(=O)NCc3nc(no3)c4ccc(cc4)C(F)(F)F)non2 HTS00175 CCc1ccc(cc1)C(=O)Nc2ccc(c(c2)NS(=O)(=O)C)C HTS04131 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)c2c(onc2c3ccccc3)C HTS04134 Cn1c2c(cn1)c(ncn2)O/N=C(/c3ccc(cc3)C(F)(F)F)\N GK03531 CN1CCN(CC1)CN2c3ccccc3C4(C2=O)OCCO4 HTS00588 CC(C)NC(=O)CSc1nnc(n1c2ccc3c(c2)OCO3)c4ccc(cc4)C(C)(C)C HTS02056 c1cc(ccc1c2nc(on2)C3CCNCC3)Cl.Cl SEW06344 c1ccc2c(c1)nc3c4cc(ccc4n(c3n2)C(=O)c5cccs5)F RH02032 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4ccc(cc4)OC(F)(F)F KM09565 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2ccc(cc2)C(C)(C)C)c3ccccc3)c4ccccc4)C SP01133 CN(C)CCCNc1c(c(c(s1)c2ccccn2)[N+](=O)[O-])[N+](=O)[O-] CD08052 CC12c3ccccc3CCN1CC(=O)N2 RJC04046 CSc1nc2ccc(cc2s1)NS(=O)(=O)c3ccc(cc3)[N+](=O)[O-] KM10781 COc1c(cc(cn1)C(=O)NN)[N+](=O)[O-] SPB07425 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCCNCC2)C#N SPB07872 CCOC(=O)c1c(c(c([nH]1)COC(=O)C)C(=O)C)C SB02046 c1ccc(cc1)SCCC(=O)c2cccs2 MWP00746 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc(cc3)SC(F)(F)F)Cl MWP00966 CCCCC#Cc1ccc(o1)C(=O)NNC(=S)NC KM09613 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cc(nn3c4ccc(cc4)I)c5cccs5 SP01017 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2cccc(c2)C(F)(F)F)c3ccc(cc3)C)C SP01153 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2ccc(cc2)OC(F)(F)F)c3ccc(cc3)C)C SP01154 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2ccc(cc2)C(F)(F)F)c3ccc(cc3)C)C SP01155 c1ccc2c(c1)cc3ccccc3c2C4=NNC(C4)(C(F)(F)F)O SP01413 c1cc(sc1c2ccn[nH]2)[N+](=O)[O-] CD08139 c1cc(ccc1NC(=O)Nc2ccc(c(c2)C(F)(F)F)Br)F HTS01940 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC(=O)Nc5ccccc5Cl HTS02057 COc1c(csc1Br)C(=O)NNC(=O)c2cccs2 KM00636 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(sc2C(=O)OC)c3ccc(cc3)C(C)(C)C GK03527 c1cc(ccc1S(=O)(=O)NNc2c3c(ccs3)ncn2)Cl GK03804 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cc(nn3c4ccc(c(c4)Cl)Cl)c5ccc(cc5)OC SP00979 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3cc(nn3c4ccc(cc4)I)c5cccs5 SP01018 c1cc(cc(c1)Cl)CNC(=O)NC(=O)c2ccc(cc2)c3csnn3 SEW01150 c1cc(ccc1CC(=S)N)c2csnn2 SEW01314 CCOC(=O)c1c(oc(c1S(=O)(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)c4ccccc4)C SP01156 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2ccc(cc2)Cl)C)C SP01159 CCOC(=O)c1c(oc(c1S(=O)(=O)Nc2ccccc2)C)C SP01162 c1cc2c(cc1/C=C/C3=NNC(C3)(C(F)(F)F)O)OCO2 SP01459 CN1C(CC(=N1)c2coc3c2cccc3)(C(F)(F)F)O SP01462 c1ccc(cc1)NC(=O)Nc2ccc(c(c2)C(F)(F)F)Br HTS01938 CSc1nc(sn1)SC CD08326 CC(C)(C)c1csc(n1)Sc2c(cccn2)[N+](=O)[O-] CD08394 CC(=O)N1CCN(CC1)c2ccc(cc2)O SB02047 c1csc(c1C#N)NC(=O)CSCC(=O)O GK03787 Cc1ccc(n1c2c3c(cccc3F)n(n2)S(=O)(=O)c4cccc(c4)C(F)(F)F)C HTS01087 Cc1cc(c2ccccc2n1)N3CCN(CC3)C(=O)Nc4c(cccc4Cl)OC HTS00413 c1cc(cc(c1)NC(=O)C(Cl)(Cl)Cl)c2ncon2 SEW01245 Cc1cc(ccc1NC(=N)NC(=N)N)Br.Cl RJF00555 Cc1ccccc1NC(=N)NC(=N)N.Cl RJF00571 CCOC(=O)c1c(oc(c1S(=O)(=O)N2CCOCC2)c3ccc(cc3)C)C SP01168 c1ccc2c(c1)cc(s2)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS03780 Cc1cc(nc(n1)Sc2ccccc2NC(=O)C)C(=O)OC SPB06395 Cc1cc(nc(n1)Sc2ccccc2NC(=O)c3ccc(cc3)Cl)C(=O)OC SPB06393 CC(C)NC(=O)N(Cc1ccccc1)Cc2cccs2 RF03402 c1csc2c1ncnc2NNC=C(C#N)C#N GK03805 c1ccc(cc1)CCNc2c3c(ccs3)ncn2 GK03340 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)C4CCCCC4 KM11112 CCOC(=O)c1cc(c(cc1NS(=O)(=O)c2ccsc2C(=O)OC)OCCOC)OCCOC GK03807 c1cc(ccc1c2nc(on2)CCOc3ccc(cc3)F)C4SCCS4 SEW01469 COc1cc(ccc1OC(=O)/C=C/c2cccs2)/C=N/c3ccc(c(c3)Cl)F RJF01286 CCOC(=O)c1c(n(c(c1S(=O)(=O)N2CCOCC2)c3ccccc3)c4ccccc4)C SP01172 Cc1c(cc(o1)c2ccccc2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl SP01180 CC(C)NC(=O)N(Cc1cccnc1)Cc2cccs2 RF03414 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NS(=O)(=O)c3ccccc3F HTS01048 CC(C)(CC(=O)Nc1ccc(c(c1)C(F)(F)F)Br)CC(=O)O HTS01932 CCNC(=O)N(Cc1ccc(cc1)Cl)Cc2cccnc2 RF03395 CCOC(=O)N1CCN(CC1)c2cc(=O)n(c(=O)n2C)C HTS01405 c1ccc(cc1)N2CCN(CC2)C(=O)CN3CCOCC3 HTS01213 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)c2cccs2 AW01024 Cc1cc(n(n1)c2c(cccn2)[N+](=O)[O-])C SEW04734 CCOC(=O)CN1CCN(CC1)c2ccc(cn2)[N+](=O)[O-] HTS00856 CCc1cccc(c1NC(=S)NCCC(=O)O)C RJF01736 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS01367 COc1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)NCc3cccs3 HTS01773 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)O/N=C(/c3ccc(cc3)C(C)(C)C)\N HTS00477 c1ccc2c(c1)C(=O)N(C2=O)c3c(ccs3)C#N GK03808 CN(C)c1ccc(cc1)n2c(nnn2)SCC(=O)c3ccccc3 HTS01663 CC(C)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS00012 c1cc(ccc1NC(=O)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)OC(F)(F)F HTS00014 Cc1ccc2c(c1)c(c(s2)C3=NNC(C3)(C(F)(F)F)O)C SP01414 CC1(CCC(=O)c2c1c(sc2SC)C3=NNC(C3)(C(F)(F)F)O)C SP01411 c1ccc(c(c1)N)Sc2c(cc(cn2)[N+](=O)[O-])C(F)(F)F SPB07559 COc1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc4c(c3)OCO4 HTS01774 c1ccc(c(c1)C(=O)O)NC(=O)c2cccs2 HTS00441 CC(C)(CC(=O)N1CCN(CC1)c2nc(ns2)c3ccccc3)CC(=O)O HTS01126 CC(C)Cc1ccc(cc1)C(=O)C(C)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] HTS00860 Cn1c(ccc1S(=O)(=O)N)C(=O)O SP01488 CC(C)(C)C(=O)N(Cc1cccnc1)Cc2cccs2 RF03361 CC(C)NC(=O)N(Cc1cccnc1)Cc2cccc(c2Cl)Cl RF03387 c1cc(ccc1NC(=O)N2CCC(C(=C2)C(=O)N)C(F)(F)F)Cl RF04552 CCSc1cc(c(cn1)C(=O)Nc2ccc(cc2)Cl)C(F)(F)F RF04413 c1cc2c(cc1NC(=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)OCO2 HTS00021 Cc1nc(nc(n1)NC(=O)NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F)C RF04517 c1ccc2c(c1)Nc3cc(ccc3S2)C4=NNC(C4)(C(F)(F)F)O SP01458 Cc1cc2ncc(c(n2n1)C)C3=NNC(C3)(C(F)(F)F)O SP01460 CC1=CSC2C1C(=C(S2)C3=NNC(C3)(C(F)(F)F)O)C SP01461 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)c3nc(no3)c4ccc(cc4)C(C)(C)C HTS00478 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2nnnn2c3ccc(cc3)O HTS01665 Cc1ccc(cc1)S(=O)(=O)Oc2cc(ccc2C)C RDR01000 CNC(=S)Nc1ccc(cc1)F RDR01003 Cc1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccccc4SC)[nH]cn3 KM09772 Cc1c(snn1)C(=O)NC2Cc3ccccc3C2 HTS01675 CCN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)NC RF04438 COC(=O)CSc1cc(c(cn1)C(=O)Nc2ccc(cc2)Cl)C(F)(F)F RF04442 CCOC(=O)c1c2c(sc1NC(=O)CN3CCOCC3)CCCC2 HTS01898 Cc1ccc2c(c1)c(c(s2)C3=NN(C(C3)(C(F)(F)F)O)C)C SP01463 c1cc(c(cc1NC(=O)c2c(nccn2)C(=O)O)C(F)(F)F)Br HTS01935 CC(C)c1ccc(cc1)N2C(C3CCc4ccccc4C3=N2)c5cc(c(c(c5)OC)OC)OC PD00627 CC(=O)N1CC(=O)N/C(=C\c2cccnc2)/C1=O PD00630 COC(=O)c1ccccc1Sc2c(nc3n2cccn3)c4ccccc4 HTS01508 CC(C)c1cc(c(c(c1)C(C)C)Sc2c(nc3n2cccn3)c4ccccc4)C(C)C HTS01509 CSCC(Cn1c(=O)c2ccccc2cn1)O PD00590 COc1ccc2c(c1)occ2CC(=O)O KM10844 c1cc2c(cc1CNCC(COc3ccc(c(c3)Cl)Cl)O)OCO2 AW01006 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)c4ccc(cc4)C#N SPB08321 c1cc(ccc1C#N)N2CCN(CC2)C(=O)c3ccc(cc3Cl)F SPB08322 CCOC(=O)c1cccc(c1)n2c(=O)n(c(=O)s2)C3Cc4ccccc4C3 HTS01585 Cc1ccc(cn1)C(=O)NC2(C(=O)c3ccccc3C2=O)O HTS01957 COc1ccccc1NC(=O)Nc2ccc(c(c2)C(F)(F)F)Br HTS01936 COc1ccc(cc1NC(=O)Nc2ccc(c(c2)C(F)(F)F)Br)Cl HTS01937 c1ccc(c(c1)C(F)(F)F)NC(=O)Nc2ccc(c(c2)C(F)(F)F)Br HTS01939 CSC(=N)Nc1cccc(c1Cl)Cl.I RDR00797 COc1ccc(cc1)c2c(nn3c2[nH]c(cc3=O)c4ccccc4)C(F)(F)F HTS01428 Cc1ccc(c(c1)NC(=O)c2cc(oc2C)C(C)(C)C)OC SP01218 c1ccc(cc1)c2cc(c(c(n2)SCC(=O)c3ccccc3)C#N)C(F)(F)F HTS01844 COc1cscc1C(=O)NC2(C(=O)c3ccccc3C2=O)O HTS01858 c1cc(ncc1C(F)(F)F)N2CCN(CC2)Cc3cc(cc4c3OCOC4)Cl HTS01691 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cccc3c2nccc3 HTS00641 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NS(=O)(=O)c3ccc(cc3)Cl HTS01047 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)c3ccc(cc3)F HTS01049 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)N2CCCC2 AW01001 Cc1c(cc(o1)c2ccccc2)C(=O)Nc3ccc(cc3)[N+](=O)[O-] SP01182 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCC2CC2 AW01003 Cc1c(cc(o1)c2ccccc2)C(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F SP01179 Cc1ccc(cc1)NC(=O)c2cc(n(n2)C(C)(C)C)C SPB08204 Cc1c(c(n(n1)c2ccccc2)O)C(=O)c3ccccc3 JFD03992 c1cc(sc1)C(=O)N2CCN(CC2)c3ccc(cc3)C#N SPB08323 c1cc(ccc1/C(=N\O)/Cn2nc(nn2)N3CCCC3)Cl.Cl RJF00360 CC(C)(C)NS(=O)(=O)c1ccc(n1C)C(=O)OC HTS01750 Cn1c(ccc1S(=O)(=O)NCc2ccccc2)C(=O)OC HTS01753 CC(C)(CC(=O)N1CCN(CC1)Cc2c(cccc2Cl)F)CC(=O)O HTS01678 c1ccc(cc1)c2ccccc2NC(=O)CSCC(=O)O HTS04386 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2)OC SP01222 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc3c(c2)OCO3 SP01223 Cn1c2c(cn1)c(ncn2)O/N=C/c3ccc(cc3Cl)Cl GK03545 COc1ccc(cc1)OCCNC(=O)c2cccs2 SPB08208 CCOC(=O)N1CCN(CC1)C(=O)c2c(onc2c3ccccc3Cl)C PD00840 c1cc(cc(c1)NC(=O)c2ccc(cc2)C(F)(F)F)c3cnco3 HTS01993 c1ccc2c(c1)C(=O)C(C2=O)(NC(=O)c3ccccn3)O HTS01955 c1ccc2c(c1)CC3C2=Nc4ccccc4SC3c5ccc(cc5)Cl JFD02641 CC(C)(C)c1ccc(cc1)c2nnc(o2)SCC(=O)c3ccccc3 SPB08250 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)NCc3ccco3 SPB08244 c1cc2c(cc1Cl)C=C(CO2)C(=O)NCCNc3c(cc(cn3)C(F)(F)F)Cl AW01265 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@@H]1C(=O)NCc3cccs3 SPB08446 c1cc(ccc1c2nc(cs2)c3ccc4c(c3)OCCO4)OC(F)(F)F SPB08215 c1cc(ccc1/C=N/Nc2nc(cs2)c3ccc4c(c3)OCCO4)C#N SPB08217 COc1cc(c(cc1OC)NC=C(C#N)C#N)C(=O)OC HTS00455 COc1ccc(cc1)C(=O)N2CCC(CC2)c3nc(no3)c4ccc(cc4)Cl SEW06512 c1cc(ccc1c2nc(on2)C3CCN(CC3)C(=O)c4ccc(cc4)Cl)Cl SEW06514 c1cc(oc1)CNC(=S)NC2CC2 RJF00375 Cc1c(nc(nc1O)SC)COC RJF00530 CCOC(=O)[C@H](C(C)C)NS(=O)(=O)c1ccc(c(c1)Cl)F HTS00169 c1ccc2c(c1)c(=O)c(co2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)F HTS00148 c1cnc(nc1)SCC(=O)Nc2ccc(cc2)Cl HTS04457 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NCN3C(=O)c4ccccc4C3=O HTS00495 c1cc(ccc1C(F)(F)F)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03696 CC(=O)c1c(cc(s1)c2ccc(cc2)C(C)(C)C)NC(=O)c3cc(cc(c3)Cl)Cl GK03534 c1c(cc(c(c1[N+](=O)[O-])N2CCOCC2)[N+](=O)[O-])Cl MGH00044 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)/C=C/C(=O)O AW01214 COC(=O)CNC(=O)c1c(cnc(n1)SC)Cl SPB08356 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2csnn2 SEW00673 Cc1cc(nn1C(C)(C)C)C(=O)NNS(=O)(=O)c2cccc(c2)Cl HTS00055 Cc1c(c(no1)c2ccccc2)CN3CCOCC3 HTS04318 c1cc2c(cc1C(=O)N3CCN(CC3)C(=O)c4ccc5c(c4)CCO5)CCO2 HTS00388 CCN(CC)c1ccc(cc1)NC(=O)c2c(onc2c3c(cccc3Cl)F)C HTS04534 Cc1ccc2c(c1)n(c(=O)o2)CC(=O)c3ccc(cc3)F HTS04187 Cc1cc(on1)NC(=O)c2cc(oc2C)C HTS04339 Cc1csc2c1ncnc2Sc3ccccc3NS(=O)(=O)c4ccsc4C(=O)OC HTS00120 c1ccc2c(c1)CC(C2)n3c(=O)n(sc3=O)c4ccc(cc4Cl)[N+](=O)[O-] HTS01584 Cc1nc(cs1)c2cc3cc(ccc3o2)Cl HTS00544 CCCc1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccc(cc3)Br HTS01638 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc4c(c3)OCO4 HTS01370 CC(C)(C)C(=O)NCc1ccc(cc1)c2csnn2 SEW00913 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)Nc2ccc(cc2)C(F)(F)F HTS00004 c1ccc(cc1)NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F HTS02559 c1cc(c(cc1C(F)(F)F)NC(=O)Nc2ccc(cc2Cl)Cl)N3CCOCC3 HTS02561 Cn1c(nnc1SCC(=O)c2cccc(c2)[N+](=O)[O-])c3ccco3 HTS02851 c1ccc2c(c1)cc(s2)C(=O)NCc3ccc4c(c3)OCO4 HTS01770 CCOC(=O)c1c(c2cc(ccc2[nH]1)[N+](=O)[O-])CCC(=O)O SEW06679 c1cc(c(c(c1)Cl)CSCCNC(=O)Nc2ccc(cc2)OC(F)(F)F)F HTS01724 c1cc(cnc1)C2N(CCCN2Cc3ccc(cc3)Cl)Cc4ccc(cc4)Cl HTS01039 CC(C)(C)c1cc2c(s1)c(ncn2)NCc3ccc4c(c3)OCO4 HTS00630 CC(C)(C)c1ccc(cc1)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03699 c1cc(ccc1NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)OC(F)(F)F HTS03709 Cc1cc(c(o1)C)C(=O)Nc2ccccc2N3CCOCC3 HTS04340 Cc1cc(c(o1)C)C(=O)Nc2ccccc2 HTS04342 Cn1c(ccc1S(=O)(=O)NCCc2ccccc2OC)C(=O)O HTS01755 c1cc(c(cc1C(F)(F)F)NS(=O)(=O)c2cc(sc2Cl)Cl)N3CCOCC3 HTS02571 Cc1cc(no1)C(=O)Nc2c3c(cccc3OC)n(n2)C HTS02614 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2c3ccccc3n(n2)C HTS00332 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)C4CC(=O)N(C4=O)c5cc(cc(c5)C)C PD00763 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)C4CC(=O)N(C4=O)c5cc(ccc5F)F PD00764 Cn1cccc1CN(Cc2ccc(cc2)OC)C(=O)c3cc4cc(ccc4[nH]3)OC HTS00003 c1ccc(cc1)CCNC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] SEW00908 c1cc(cnc1)/C=N/c2ccc(cc2)c3csnn3 SEW01006 COc1ccc(cc1OC)C(=O)N2CCC(CC2)C(=O)O HTS00873 Cn1c(nnc1SCc2c(cccc2Cl)F)CSc3ccnc4c3ccc(c4)Cl HTS00159 Cc1ccc2c(c1)CCCN2CC(=O)c3ccc4c(c3)OCCO4 HTS02135 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3c(onc3c4c(cccc4Cl)Cl)C HTS00445 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)CCc4ccccc4 HTS01827 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)Cc3c(c4ccccc4oc3=O)O PD00835 Cc1cc(nn1C(C)(C)C)C(=O)NNS(=O)(=O)c2cccc3c2nccc3 HTS00064 COc1ccc2cc(ccc2c1CC#N)Br SB02088 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC5CC5 HTS02048 Cc1ccsc1CNC(=O)Nc2ccc(cc2)F HTS04010 Cc1ccsc1CNC(=O)Nc2ccc(cc2)C(C)(C)C HTS04011 Cc1ccsc1CNS(=O)(=O)c2ccc(cc2)F HTS04013 c1ccc(cc1)CCN2CCN(CC2)S(=O)(=O)c3ccc4c(c3)OCCO4 HTS01826 c1cc(ccc1NC(=O)C2=Cc3cc(ccc3OC2)Cl)n4ccc(n4)C(F)(F)F AW01266 COc1ccc(cc1)C(=O)COc2cc(=O)oc3c2cccc3 PD00825 COc1ccc(cc1)C(=O)Cc2c(c3ccccc3oc2=O)O PD00826 CC(C)(CC(=O)Nc1ccccc1N2CCCCC2)CC(=O)O HTS00163 CN(c1ccccc1)C(=O)CN2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] HTS00007 Cc1csc(c1c2nc3ccccc3s2)N GK03755 Cc1csc(c1c2nc3ccccc3s2)NS(=O)(=O)c4ccc(cc4)Cl HTS00390 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc(cc4)Cl SEW01081 CN1CCN(CC1)c2ccc(cc2)NS(=O)(=O)c3ccccc3 SS00022 CCOc1cc(c(cc1N2CCOCC2)OCC)NS(=O)(=O)c3ccccc3 SS00023 CC(C)(C)C(=O)Nc1c(c(nn1C)C(F)(F)F)c2ccc(cc2)F HTS00351 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)c3ccccc3 HTS01625 c1cc2c(nc1)sc(n2)Sc3c(cccn3)NC(=O)c4ccc(cc4)F HTS01778 c1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc(cc3)F HTS01794 c1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccncc3 HTS01796 c1cc2c(cc1NC(=O)CSCC(=O)O)OCCCO2 HTS00132 CC(C)(CC(=O)Nc1ccc2c(c1)OCCCO2)CC(=O)O HTS00134 c1ccc2c(c1)c(c(c(=O)o2)CC(=O)c3ccc4c(c3)OCCO4)O PD00836 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CC3CCCO3 PD00839 c1ccc(cc1)CCN2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F HTS02016 c1ccc(cc1)CCN2CCN(CC2)C(=O)Nc3ccc(cc3F)F HTS02017 COCCOc1c(cc(cn1)NC(=O)CSCC(=O)O)C(F)(F)F HTS01968 c1ccc(cc1)CCN2CCCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F HTS01811 CCCCCCCC1C(=O)/C(=C/c2ccc(cc2)/C=C\3/C(=O)C(CC3)CCCCCCC)/CC1 S15337 Cc1cc(c(o1)C(F)(F)F)NC(=O)NCCCN2CCOCC2 HTS04302 c1ccc(cc1)N2CCN(CC2)C(=O)CSc3nccs3 HTS01822 c1ccc(cc1)CCN2CCN(CC2)S(=O)(=O)c3cccc4c3nccc4 HTS01824 COC(=O)c1cc2c(s1)ccs2 SEW02080 c1ccc(cc1)CCN2CCN(CC2)S(=O)(=O)c3cccc(c3)C(F)(F)F HTS01828 c1ccn(c1)C2CCN(CC2)C(=O)COCC(=O)O HTS00580 Cn1c(ccc1S(=O)(=O)Nc2ccsc2C(=O)OC)C(=O)OC HTS01534 Cn1c(ccc1S(=O)(=O)NNC(=O)c2c(c3c(ccs3)[nH]c2=O)O)C(=O)OC HTS01559 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)CCc4ccccc4)C(F)(F)F HTS02012 COc1ccc(cc1NC(=O)N2CCN(CC2)CCc3ccccc3)Cl HTS02013 C1COC2(O1)CSc3c(sc(=S)s3)SC2 JFD04067 CCc1c2cc(c(cc2cc(n1)O)OC)OC JFD04072 Cc1cc(ccc1NC(=O)CSCC(=O)O)C(C)(C)C HTS01966 c1ccc(cc1)CCN2CCCN(CC2)C(=O)Nc3ccc(cc3)F HTS01812 Cn1c2cccc(c2c(n1)NC(=O)CC34CC5CC(C3)CC(C5)C4)F HTS01642 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)NC(=O)Nc3ccc(cc3)F HTS01919 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)NC(=O)Nc3ccccc3 HTS01920 CCOc1cc(c(cc1N2CCOCC2)OCC)n3cccc3 SS00033 CCOc1cc(c(cc1N2CCOCC2)OCC)n3c(ccc3C)C SS00034 CC(C)(C)c1ccc(cc1)NC2CCN(CC2)Cc3ccccc3 SPB08400 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)CCO)C(=O)O HTS01760 c1ccc2c(c1)cc(s2)C(=O)N3CCN(CC3)c4ccccn4 HTS01767 c1cc(oc1)c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NC(=O)C4CCC4 SP01019 c1ccc(cc1)C(=O)Nc2ccc3c(c2)OCCO3 HTS01865 COc1ccc(cn1)NC(=O)CSCC(=O)O HTS01969 Cn1c(ccc1S(=O)(=O)Nc2ccc(cc2)N3CCOCC3)C(=O)OC HTS01533 Cn1c(ccc1S(=O)(=O)N(Cc2ccccc2)Cc3ccccc3)C(=O)OC HTS01744 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC(=O)N5CCOCC5 HTS02054 Cc1c2cc(ccc2sc1C(=O)/C(=C\c3ccc(cc3)OC)/C#N)Cl MWP00555 c1cc(c(cc1F)F)SCCC(=O)c2ccc(s2)Cl MWP00771 Cc1ccc2c(c1)CCCN2CC(=O)c3ccc(cc3)OC HTS02134 CC(=O)c1ccc(c(c1)NC(=O)Nc2ccc(cc2)Cl)Cl SEW06664 Cn1c2c(cn1)c(ncn2)NNS(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F GK03553 c1ccc(c(c1)C(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F)C(=O)O HTS00597 c1cc(c(c(c1)F)C(=O)Nc2ccc3c(c2)OCCO3)F HTS01868 c1cc(ccc1c2cc(n(n2)c3ccc(cc3)I)N)Cl SP00985 c1ccc(cc1)CCN2CCN(CC2)C(=O)Nc3ccccc3 HTS02018 c1ccc(cc1)CCN2CCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl HTS02020 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCc5ccc(cc5)C#N HTS02052 CN1C(=S)S/C(=N/OC(=O)c2ccc(cc2)Cl)/C(N1)c3ccc(cc3)Cl MBE00221 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)Cc4cccc(c4)C(=O)N5CCC(CC5)O HTS01624 COC(=O)c1ccccc1NC(=O)c2cccs2 HTS00440 Cc1nc2ccc(cc2o1)NC(=O)NC(=O)c3c(cccc3F)F MWP00036 c1ccc(cc1)CCN2CCCN(CC2)S(=O)(=O)c3cccc(c3)C(F)(F)F HTS01804 c1cc(c(c(c1)Cl)C(=O)Nc2ccc3c(c2)OCCO3)F HTS01871 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)c3cc(no3)c4ccccc4 HTS02152 CN1C(=S)S/C(=N/OC(=O)c2ccc(cc2)Cl)/C(N1)c3cccc(c3)OC MBE00225 c1ccc2c(c1)cccc2NC(=O)Nc3c(cccn3)OCc4ccc(c(c4)Cl)Cl HTS04540 Cc1ccc2c(c1)n(c(=O)o2)CC(=O)c3ccc(cc3)OC HTS04188 c1ccc(cc1)C(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl HTS04452 c1cc(cc(c1)NC(=N)NC(=N)N)C(F)(F)F.Cl RJF00541 CCCCCc1ccc(cc1)S(=O)(=O)Nc2cc(ccn2)C HTS02250 c1ccc2c(c1)cc(o2)c3csc(n3)c4ccc(s4)c5ccno5 HTS02299 Cc1c(cn(n1)C)/C=N/Nc2c3cnn(c3ncn2)C GK03554 CCOC(=O)c1cnn(c1C(F)(F)F)c2c3cnn(c3ncn2)C GK03555 CCOC(=O)c1cc(c(cc1NS(=O)(=O)c2cccc3c2nccc3)OCCOC)OCCOC HTS00095 c1ccc(c(c1)C#N)NC(=O)Nc2cc(nn2c3ccc(cc3)I)c4cccs4 SP01007 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc4c(c3)OCCO4)Cl HTS01869 Cc1ccc(cc1)C(=O)CSc2nnn(n2)c3cccc(c3)NC(=O)C HTS02150 COc1ccc(cc1)C(=O)Nc2cccc(c2)c3[nH]c4ccccc4n3 HTS01781 c1cc(sc1)c2ccnc(n2)SCC(=O)N3CCOCC3 HTS04401 CC(C)NC(=O)CSc1nccc(n1)c2cccs2 HTS04404 c1cc(ccc1c2c(c([nH]n2)N)C#N)Cl CC00044 CCCCc1ccc(cc1)C(=O)NC(=S)Nc2cc(nn2c3ccc(cc3)I)c4ccc(cc4)Cl SP01065 c1cc(ccc1NC(=O)Nc2nnc(s2)C3CC3)OC(F)(F)F HTS03431 c1cc(ccc1/C(=C/Sc2c(c(c3c(n2)CCCC3)C(F)(F)F)C#N)/O)F HTS01847 Cc1cc(nc(c1C#N)OCC(=O)Nc2ccc(cc2)Oc3ccccc3)C HTS01682 CCCCc1ccc(cc1)C(=O)Nc2c(ccs2)C#N HTS00436 Cc1c(cc(o1)c2ccccc2)C(=O)Nc3ccccc3Cl SP01184 Cc1c(cc(o1)c2ccccc2)C(=O)N3CCSC3C(=O)OC SP01188 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCN(CC3)CCc4ccccc4 HTS01806 c1cc(ccc1n2c(c(cn2)C(=O)NCCN3CCNC3=O)C(F)(F)F)Cl HTS02484 CCN(CC)c1ccc(cc1)NC(=O)c2cc(sc2Cl)Cl HTS04531 COc1ccc(cc1)c2ccnc(n2)SCC(=O)Nc3ccccc3 HTS00595 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cc(nn3c4ccc(cc4)F)c5ccc(cc5)Cl SP01036 CNC(=S)NCCc1ccccc1 RDR01004 CCS(=O)(=O)c1ccc(c(c1)NC(=O)Nc2cccc3c2cccc3)O HTS04076 CCS(=O)(=O)c1ccc(c(c1)NC(=O)Nc2ccc(cc2)OCc3ccccc3)O HTS04077 CCCCNC(=S)NCC1CC1 RJF01271 Cc1nc(cn1CCc2nc(on2)c3ccc(cc3)F)[N+](=O)[O-] HTS01909 COc1cc(cc(c1OC)OC)CN2CCCN(C2)Cc3cc(c(c(c3)OC)OC)OC HTS01914 CCOC(=O)c1c(nc(s1)CN2CCN(CC2)c3cccc(c3)Cl)C SEW06658 c1ccc2c(c1)c(cs2)C(=O)O CC12301 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)Nc4ccc(cc4C(=O)c5ccccc5Cl)Cl HTS04396 Cc1ccc(cc1C)n2c(cc(n2)c3ccc(cc3)OC(F)(F)F)NC(=O)Nc4ccc(cc4)OC(F)(F)F SP01024 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04036 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04037 c1ccc(cc1)c2c(n3cccnc3n2)Sc4ccc(cc4)[N+](=O)[O-] RJC04056 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2)[N+](=O)[O-] SP01215 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(n3C4CCCCC4)SCc5ccccc5 SPB08206 Cc1cccc(c1)n2c(=O)c3ccccc3cn2 PD00624 Cc1cc(cc(c1)NC(=S)NCCCCN2CCN(CC2)c3ccccc3OC)C SEW06498 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)c3cccc(c3)[N+](=O)[O-])C HTS01982 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)Nc3ccccc3Cl)C HTS01984 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)Nc3ccc(cc3)C(F)(F)F)C HTS01985 Cc1cc(c(o1)C(F)(F)F)NC(=O)NCc2c(cccc2Cl)Oc3ccccc3 HTS04308 Cc1cc(c(o1)C(F)(F)F)NC(=O)NCc2ccccc2 HTS04310 COCc1cc(nc(n1)SCC(=O)N2CCOCC2)O HTS02437 COCCOC(=O)c1c(nccn1)C(=O)Nc2ccccc2 HTS03750 CCCNC(=O)Nc1cc(ccc1O)S(=O)(=O)CC HTS04079 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(sc2C(=O)N)c3ccc(cc3)C(C)(C)C GK03561 Cc1ccc(cc1)CN2CC(CC2=O)C(=O)O SEW06669 c1cc2c(cc1CN3CC(CC3=O)C(=O)O)OCO2 SEW06670 Cc1cc(c(o1)C(F)(F)F)NC(=O)Nc2ccccc2 HTS04303 Cc1cc(c(o1)C(F)(F)F)NC(=O)NCc2ccc3c(c2)OCO3 HTS04304 Cc1cc(c(o1)C)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS04332 c1ccc(cc1)c2ccccc2NC(=O)c3cccs3 HTS04382 c1c(cc(cc1Cl)Cl)NC(=O)/C=C/C(=O)O RJF00738 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)C(=O)O SP01358 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)N)NC(=O)c3cc(cc(c3)Cl)Cl GK03559 c1ccc(cc1)CN2CCN(CC2)c3ccccc3CO SEW06511 c1cc(cc(c1)[N+](=O)[O-])c2nnc(o2)Cc3cc(cc(c3)F)F SEW06503 CCOC(=S)Nc1cccc2c1cccc2 NH00643 CNC(=S)Nc1cc(cc(c1)Cl)Cl RJF00131 Cc1cc(c(o1)C)C(=O)Nc2ccccc2C(C)C HTS04346 Cc1cc(c(o1)C)C(=O)Nc2ccccc2N3CCCCC3 HTS04347 Cc1c(snn1)C(=O)n2c(cc(n2)C(C)(C)C)C(C)(C)C SEW06681 c1cc(ccc1NC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)OC(F)(F)F HTS02562 CCOC(=O)c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CC(CC(C3)C)C KM10723 Cc1csc(c1NC(=O)CC2C(=O)NCCN2)C(=O)OC HTS01727 c1cc(cc(c1)S(=O)(=O)NCCSCc2c(cccc2Cl)F)C(F)(F)F HTS01728 Cc1ccc(cc1)C2C3COc4ccccc4C3=Nc5ccccc5S2 JFD02628 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)c2c(onc2c3ccccc3Cl)C HTS00026 CCn1c2ccc(cc2c3c1C(=O)CCC3)C(=O)OCC RJC04064 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccc(nc4C)C(F)(F)F HTS04238 Cc1cc(c(o1)C)C(=O)NC(C)c2ccccc2 HTS04343 c1ccc2c(c1)C(=O)N(C2=O)CCCOc3ccc(cc3)Cl HTS00295 Cc1ccc2c(c1)CCCN2CC(=O)Nc3ccc(cc3)C(=O)C HTS01705 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCC(CC4)C(=O)O SB02067 CCOC(=O)c1ccc2c(c1)c(cc(n2)c3ccccc3)O RH02104 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)NCc3cccs3 HTS02143 Cc1c(snn1)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04030 COc1ccc(cc1)c2ccnc(n2)c3cccs3 HTS01649 c1cc2c(cc1CN3CCN(CC3)C(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)OCO2 HTS03719 c1ccc(c(c1)C(F)(F)F)n2c(nnc2SCc3c(cccc3Cl)F)O HTS02456 c1cc(c(c(c1)Cl)OCc2nc(on2)CSc3nncn3c4ccc(cc4)C(F)(F)F)Cl HTS00213 c1ccc(c(c1)NC(=O)CSCC(=O)O)N2CCCCC2 HTS00138 Cn1c(nnc1SCC(=O)c2ccc(s2)Cl)CSc3ccnc4c3ccc(c4)Cl HTS00157 CC(CC=C)(c1ccccc1)NC2CCCCC2.Cl RJC04066 c1cc(sc1)CCN2CC(CC2=O)C(=O)O SEW06677 Cc1cc(c(c(c1)C)n2c(nnn2)SC3Cc4ccccc4C3=O)C HTS01988 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)c3cccnc3 HTS01646 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)O SP01351 Cc1ccc(cc1)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03711 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)N HTS02144 c1ccc(cc1)NC(=O)NCCSCc2c(cccc2Cl)F HTS01725 c1ccc(c(c1)C(F)(F)F)n2c(nnc2SCC(=O)c3ccc(cc3)F)O HTS02454 Cn1c(ccc1S(=O)(=O)N(CCO)CCO)C(=O)OC HTS01746 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(c(c2)F)Cl HTS00047 COc1ccc(cc1OC)C(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O HTS00206 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2ccc3c(c2)CCO3)/N HTS00480 Cc1nc(cn1CC(=O)c2ccc(cc2)OC)[N+](=O)[O-] RH02129 c1ccc(cc1)c2cc3c(s2)c(ncn3)N4CCSCC4 HTS00603 CC(=O)c1c(cc(s1)c2ccc(cc2)C(C)(C)C)NC(=O)C GK03541 c1cc(ccc1C(=O)CO)F HTS02459 Cn1c(ccc1S(=O)(=O)N(Cc2ccccc2)Cc3ccccc3)C(=O)O HTS01757 Cn1c(ccc1S(=O)(=O)N2CCCCCC2)C(=O)O HTS01761 Cc1ccsc1CNC(=O)c2cnn(c2C)c3ccc(cc3)OC HTS04293 Cc1nc(cs1)C(=O)NC2(C(=O)c3ccccc3C2=O)O HTS01974 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC(=O)c5ccc(cc5)OC HTS02045 Cc1c(cc(o1)S(=O)(=O)N(C)C)C(=O)O SP01364 COc1cc(cc(c1OC)OC)C(CC(=O)Nc2cc(c(cc2C(=O)OC)OC)OC)CC(=O)O HTS00612 c1ccc(cc1)CCN2CCN(CC2)S(=O)(=O)c3cccs3 HTS01829 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)O SPB08408 Cc1c(c(c(o1)C)S(=O)(=O)NCCSCc2c(cccc2Cl)F)C(=O)OC HTS01731 CSc1cccc(c1)NC(=O)CN2CCCCC2 HTS01902 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NS(=O)(=O)c3cn(cn3)C HTS01045 COc1ccc(cc1)c2c(sc(c2c3ccc(cc3)OC)C(=O)NC4(C(=O)c5ccccc5C4=O)O)C#N HTS01973 c1ccc(cc1)CCN2CCN(CC2)S(=O)(=O)c3cc(sc3Cl)Cl HTS02011 c1ccc(cc1)CCN2CCN(CC2)C(=O)Nc3ccc(cc3)F HTS02015 c1ccc(cc1)Nc2nc(cs2)c3ccc(s3)Cl HTS00002 Cc1c(sc(n1)c2ccc(cc2)Cl)c3ccnc(n3)SCc4ccccc4 HTS00006 c1cc2c(c(c1)S(=O)(=O)Nc3ccc(nc3)Oc4ccc(cc4C5CCCCC5)Cl)non2 HTS01792 COCCOc1cc2c(cc1OCCOC)nc[nH]c2=O GK03533 c1ccc(cc1)C(=O)Nc2c(ccs2)C#N HTS00442 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NC(=O)c3ccccc3 HTS01626 Cc1ccc2c(c1)CCCN2CC(=O)N(c3ccccc3)C4CCCCC4 HTS01707 c1ccc(cc1)NC(=O)CN2CCN(CC2)CCCc3c[nH]c4c3cc(cc4)F.C(=C/C(=O)O)\C(=O)O HTS01693 Cn1c(ccc1S(=O)(=O)N(CCO)Cc2ccccc2)C(=O)OC HTS01749 c1cc2c(cc1C(=O)N)OCO2 CC00048 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3cc(nn3c4cc(cc(c4)C(F)(F)F)C(F)(F)F)c5ccco5 SP01048 CCC1CSc2n1c(=O)c3c(n2)ccs3 GK03799 c1cc(oc1)C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F SPB08439 CC(C)c1ccc(cc1)NC(=O)CSc2nnnn2c3ccc(cc3)N(C)C HTS01660 COc1ccccc1NC(=O)N2CCN(CC2)CCc3ccccc3 HTS02014 c1ccc(cc1)CCN2CCCN(CC2)C(=O)c3ccccc3C(F)(F)F HTS01814 Cc1ccc2cc(ccc2n1)NC(=O)c3c(nccn3)C(=O)O HTS02188 COc1cc(ccc1NC(=O)c2c(nccn2)C(=O)O)C(=O)O HTS02189 c1ccc2c(c1)nc(s2)CC(=O)NC(=O)N HTS02060 Cc1cc(ccc1NC(=O)CCC(=O)O)C(C)(C)C HTS02065 c1ccn(c1)c2cc(ccc2N3CCN(CC3)C(=O)c4cc(oc4C(F)(F)F)c5ccc(cc5)Cl)[N+](=O)[O-] HTS01301 Cc1ccc(cc1)S(=O)(=O)CCSc2nnc(n2C)c3ccco3 HTS02853 Cc1nc(cn1CCCOc2ccc(cc2)Cl)[N+](=O)[O-] HTS00293 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC(=O)c5ccccc5 HTS02043 Cc1ccc(cc1)C(=O)NCCN2CCNC2=O HTS02477 CC(C)(C)c1ccc(s1)C(=O)O/N=C/2\C(NN(C(=S)S2)C)c3ccc(cc3)Cl MBE00222 COc1ccc(cc1)C2C(=C(OC3=C2C(=O)CC(C3)c4ccccc4)N)C#N S14800 CCN(CC)C(=S)Oc1ccc(c(c1)[N+](=O)[O-])C RDR00873 CN(C)c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3ccc(cc3)C(F)(F)F HTS01661 c1cc(ccc1C#N)N2CCN(CC2)C(=O)c3cc(oc3C(F)(F)F)c4ccc(cc4)Cl HTS01296 Cc1c(snn1)C(=O)NCc2ccc3c(c2)OCO3 HTS01673 COc1ccc(cc1)c2ccc(=O)[nH]n2 HTS01513 c1cc2c(nc1)n(c(=O)o2)CCS(=O)(=O)c3ccc(cc3)F HTS04461 CCc1ccccc1Cn2c3c(cccn3)oc2=O HTS04463 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCc5ccc(cc5F)Cl HTS02053 CCOC(=O)N1CCC2(CC1)c3c(c4ccccc4[nH]3)CCN2 HTS01686 Cc1ccc(cc1)S(=O)(=O)Nc2cc(sc2C(=O)N)c3ccc(cc3)C(C)(C)C GK03557 c1cc(ccc1N2C(=O)CCC2=O)S(=O)(=O)NCCN3CCNC3=O HTS02489 Cn1c(nnc1SCC(=O)c2cc(c(s2)Cl)Cl)c3ccco3 HTS02854 c1cc(oc1C(=O)O)Br AC10702 Cc1c(c(nc(n1)c2ccccc2)SCc3c(cccc3Cl)F)C#N HTS02498 Cc1ccc(cc1)C(Cn2cc(nc2C)[N+](=O)[O-])O HTS01863 c1cnc(nc1)SCCS(=O)(=O)c2ccc(cc2)F HTS04458 c1ccn2c(c1)nc3c(c2=O)cc(c(=N)n3Cc4ccco4)C(=O)N RJC04057 CC(C)Cn1c(=N)c(cc2c1nc3ccccn3c2=O)C#N RJC04058 c1ccc(cc1)Cn2c(=N)c(cc3c2nc4ccccn4c3=O)C(=O)N RJC04060 c1cc(ccc1NC(=O)c2c(nccn2)C(=O)O)S(=O)(=O)N3CCOCC3 HTS02190 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC(=O)C(C)(C)C HTS02055 Cc1ccc(cc1C)n2c(cc(n2)c3ccc(cc3)OC(F)(F)F)NS(=O)(=O)c4ccc(s4)c5cc(on5)C(F)(F)F SP01022 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(cc3Cl)C(F)(F)F)C(=O)OC HTS02617 Cn1c2c(cn1)c(ncn2)N/N=C/c3ccc(cc3)C#N GK03546 Cn1c2c(cn1)c(ncn2)N/N=C/c3ccc(cc3)Cl GK03547 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(sc2C(=O)C)c3ccc(cc3)C(C)(C)C GK03548 c1ccc(cc1)CCN2CCCN(CC2)S(=O)(=O)c3cccc4c3nccc4 HTS01230 c1ccc(cc1)CCN2CCCN(CC2)S(=O)(=O)c3cccc4c3non4 HTS01801 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2ccc(cc2)F HTS04369 Cc1c(c(n(n1)C)Cl)S(=O)(=O)Nc2ccc(cc2)Oc3ccc(cc3)F HTS00102 Cc1c(cn(n1)C)NC(=O)Nc2ccc(cc2)F HTS03837 Cc1cc(n(n1)C)NC(=O)C2CCN(CC2)C(=O)OCc3ccccc3 HTS04331 c1cc2c(cc1S(=O)(=O)NCCN3CCNC3=O)CCO2 HTS02791 c1ccc2c(c1)c(=O)c3c([nH]2)CCCC3 HTS00447 c1cc(sc1)c2ccnc(n2)SCC(=O)Nc3ccc(cc3)OC(F)(F)F HTS04566 CCOC(=O)c1cnc(nc1N)SCC(=O)c2cc(c(s2)Cl)Cl HTS02120 c1ccc(cc1)c2cc(c3c(c(sc3n2)C#N)N)C(F)(F)F SB02082 c1ccc2c(c1)CC3C2=Nc4ccccc4SC3c5ccc(cc5)C(F)(F)F S15517 COc1ccccc1NC(=S)N/N=C/c2ccccc2O RJF00962 CCNC(=S)NCC1CC1 RJF01245 Cc1c2c(c(sc2nc(n1)c3ccccc3)C(=O)c4ccc(cc4)Cl)N HTS02506 CCOC(=O)c1cc(c(cc1NS(=O)(=O)c2cccc3c2non3)OCCOC)OCCOC HTS00094 c1cc(ccc1c2cc(n(n2)c3ccc(cc3)F)NC(=O)Nc4ccc(cc4)OC(F)(F)F)Cl SP01038 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2ccc(cc2F)F HTS04370 Cc1c(cc(o1)C(C)(C)C)C(=O)NCCSCc2c(cccc2Cl)F HTS04651 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2ccccc2OC HTS04657 C1CN(CCC1C(=O)N)C(=O)CCC(=O)O PD00750 Cc1csc2c1c(ncn2)OC HTS02117 c1ccc(cc1)c2nc(sn2)Sc3ccccc3 HTS02529 c1ccc(cc1)c2nc(sn2)NC3Cc4ccccc4C3 HTS02581 c1ccn(c1)C2CCN(CC2)S(=O)(=O)c3cccc(c3)C(F)(F)F HTS00592 CC(c1ccccc1)NC(=S)N RDR00827 Cc1csc(c1NS(=O)(=O)c2cc(cc(c2)Cl)Cl)C(=O)OC HTS01022 COc1ccc(cc1)c2[nH]c(=O)n(n2)CCC#N NH00373 CCOC(=O)c1ccccc1CSC(=N)N.Cl PD00621 CC(C)c1ccc(cc1)C2C3COc4ccccc4C3=Nc5ccccc5S2 JFD02629 Cc1ccccc1C2C3CSc4ccccc4C3=Nc5ccccc5S2 JFD02632 c1ccc(cc1)c2cc(on2)C(=O)CSc3nccc(n3)c4cccs4 HTS04408 c1cnc(nc1)SCC(=O)Nc2ccc(c(c2)Cl)F HTS04456 c1cc(cnc1)/C=N/NC(=S)Nc2ccc(cc2)F RDR00907 CCS(=O)(=O)c1ccc(c(c1)NC(=O)Nc2ccccc2)O HTS04074 Cc1cccc(c1)C(=O)NCCSCc2ccc(cc2Cl)Cl SEW06686 c1ccc(c(c1)c2[nH]nnn2)F AW01202 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)N GK03406 c1cc(ccc1CSc2ccc(cc2C(F)(F)F)[N+](=O)[O-])Cl RJF01692 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)S(=O)(=O)c4cccs4 HTS00113 c1cc(cnc1)c2nc(cs2)c3ccc(s3)Cl HTS00031 Cc1cc(c(o1)C)C(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F HTS04336 Cc1cc(c(o1)C)C(=O)Nc2cc(on2)C(C)(C)C HTS04337 CCCc1cc(nn1c2ccccc2)C(=O)Nc3ccc(cc3)N(CC)CC HTS04532 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)O SP01432 Cc1c(cc(cc1Cl)F)S(=O)(=O)N TL01004 CCS(=O)(=O)c1ccc(c(c1)NC(=O)Nc2c(cc(cc2Br)C(C)C)Br)O HTS04078 CC(C(=O)NNC(=S)Nc1ccccc1F)n2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF01889 CCCCc1ccc(c(c1)C)NC(=O)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS00013 c1cc2c(cc1NC(=O)CN3CCN(CC3)c4ccc(cn4)[N+](=O)[O-])OCO2 HTS00015 c1ccc2c(c1)C3=Nc4ccccc4SC(C3CS2)c5ccc(cc5)F JFD02636 c1ccc(cc1)C(CN(CCN2CCNC2=O)CC(c3ccccc3)O)O HTS02812 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)N(Cc3ccccc3)Cc4cccs4 HTS02290 c1ccc2c(c1)ccc(c2c3c4ccccc4ccc3C(=O)O)C(=O)O HTS01514 CC(C)(C)OC(=O)NC1CCN(CC1)C(=O)CSCC(=O)O PD00757 COCc1cc(nc(n1)SCC(=O)c2ccc(cc2)c3ccccc3)O HTS02436 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)CCS(=O)(=O)c3ccc(cc3Cl)Cl HTS02445 Cc1ccc2c(c1)CCCN2C(C)C(=O)N3CCN(CC3)c4ccccc4OC HTS02136 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)Nc3ccccc3 HTS02232 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)Nc3ccc(cc3)F HTS02233 c1cc(c(c(c1)Cl)CN2CCN(CC2)C(=O)CSCC(=O)O)F HTS01677 c1cc(c(c(c1)Cl)CN2CCN(CC2)CC(COc3ccc(cc3)F)O)F HTS01922 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCC2CCN(CC2)C(=O)OC(C)(C)C HTS02342 c1cc2c(cc1Cl)sc(n2)N3CCCN(CC3)C(=O)CSCC(=O)O HTS01893 Cc1c(snn1)C(=O)NCCSCc2ccc(cc2Cl)Cl SEW06691 COc1ccc(cc1OC2CCCC2)/C=C/3\C(=O)OC(=N3)c4ccccc4 PD00761 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)Nc3ccc(cc3)C(C)C)C HTS01983 Cc1cc(c(o1)C)C(=O)Nc2ccc(cc2)F HTS04341 c1ccc(cc1)CN2CCC(CC2)Nc3ccccc3NS(=O)(=O)c4ccc(cc4)F HTS01905 CCOC(=O)c1c(n(nn1)c2cccc(c2)C#C)C HTS00892 c1ccc(cc1)C(=O)Nc2cc(ccc2N3CCc4ccccc4C3)C(F)(F)F HTS01782 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=O)c4cccs4)C(F)(F)F HTS01783 c1cc2c(cc1Cl)sc(n2)N3CCCN(CC3)C(=O)c4c(nccn4)C(=O)O HTS02169 c1cc(c(cc1C(F)(F)F)NC(=O)c2c(nccn2)C(=O)O)N3CCCC3 HTS02183 CCn1c2ccc(cc2c3c1C(=O)CCC3)OCC(C)C RJC04062 Cn1c(nnc1Sc2nc3ccc(cc3s2)Cl)c4ccc(cc4Cl)Cl HTS03449 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)N(C)c3ccccc3 HTS02137 c1cc(ccc1c2ccc(=O)n(n2)CCC#N)F HTS02139 Cc1c(c(no1)c2ccccc2)N3C(=O)CCN(C3=O)Cc4ccccc4 HTS06109 c1ccc(cc1)CN2CCC(=O)N(C2=O)c3ccc4c(c3)CCO4 HTS06111 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CSC[C@H]4C(=O)O SB02066 c1ccc2c(c1)-c3ccccc3C2COC(=O)N4CCCC[C@@H]4C(=O)O SB02069 Cc1cc(c(o1)C)C(=O)Nc2ccc(cc2F)F HTS04345 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)NCc3ccccn3 HTS03712 Cn1c2cccc(c2c(n1)NS(=O)(=O)c3cccc4c3non4)OC HTS03830 Cc1cc(n2c(n1)c(c(n2)C(F)(F)F)c3ccc(cc3)OC)C HTS03480 Cc1ccc(c(c1)C)n2c(nnn2)SCC(=O)C(C)(C)C HTS02080 Cc1ccc(c(c1)C)n2c(nnn2)SCC(=O)c3ccc(cc3)OC HTS02082 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)Nc2ccccc2 HTS02037 c1ccc(c(c1)C(=O)NN2CC(=O)N(CC2=O)c3cc(cc(c3)Cl)Cl)Br HTS02093 CCCc1c(cnn1c2ccccc2)C(=O)NCc3ccc(c(c3)OC)OC HTS03796 c1ccn(c1)C2CCN(CC2)C(=O)CSCC(=O)O HTS00579 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)c3ccco3 HTS04266 CCCCc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)NS(=O)(=O)C)C HTS04592 CCOC(=O)C1CCN(CC1)c2ccccc2CN3CCC(CC3)c4ccccc4OC HTS03468 c1ccn(c1)c2cc(c(cc2Cl)NC(=O)c3c(nccn3)C(=O)O)Cl HTS02184 c1ccn(c1)c2ccc(cc2)S(=O)(=O)N HTS04119 CCOC(=O)c1c2c(sc1NC(=O)CN3CCNCC3)CCCC2 HTS01897 Cc1ccsc1CNS(=O)(=O)c2ccccc2 HTS04015 Cc1ccsc1CNC(=O)c2ccccc2 HTS04019 c1ccc(cc1)CN2CCN(CC2)Cc3c[nH]c4c3cccc4 HTS04090 COc1ccc2c(c1)CCCN2Cc3ccc(o3)c4ccsc4C(=O)OC HTS04085 c1cc(ccc1c2nc(on2)CSCC(=O)O)Cl HTS00894 c1cc2c(cc1NC(=O)c3c(nccn3)C(=O)O)OCO2 HTS02181 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)CSCC(=O)O HTS01713 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc4c(c3)OCCO4 HTS01870 Cc1c(cc(o1)S(=O)(=O)N(C)C)C(=O)Nc2ccc(cc2)F HTS00481 CCCCNC(=O)c1cc(oc1C)S(=O)(=O)N(C)C HTS00482 CC(C)(CC(=O)Nc1cc(c(cc1C(=O)OC)OC)OC)CC(=O)O HTS00613 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS04656 c1ccc2c(c1)nc(s2)O AC40197 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)c3ccc4c(c3)OCCO4 HTS02148 c1cc2c(cc1N3C(=O)c4c(nccn4)C3=O)OCO2 HTS02182 c1ccc(cc1)OCCN2CCCN(CC2)C(=O)Nc3ccc(cc3F)F HTS00888 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)c2ccc(cc2F)F HTS04129 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)c2c(cccc2Cl)F HTS04130 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=O)c4ccccc4F)C(F)(F)F HTS01786 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=O)C4CCC4)C(F)(F)F HTS01788 c1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)NCc3cccs3 HTS01797 Cc1ccc(c(c1)C)n2c(nnn2)SCC(=O)c3ccccc3 HTS02079 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)NC(=O)Nc3ccc(cc3)Cl HTS01918 CCc1ccc(cc1)C(=O)NNc2ccc(cc2)S(=O)(=O)N HTS04480 c1cc2c(cc1C(=O)NCc3cc(cc4c3OCOC4)F)non2 HTS03230 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3c(nns3)C)C HTS04142 Cc1c(snn1)C(=O)Nc2ccc3c(c2)OCCO3 HTS04146 Cc1ccsc1CNC(=O)c2c(cccc2Cl)F HTS04020 Cc1ccsc1CNC(=O)c2c(ccs2)Cl HTS04291 CCNC(=O)c1c(onc1c2ccccc2)C HTS01706 c1cc2c(cc1C(=O)O)OCCO2 CC01301 c1cc2c(cc1C(=O)O)OCO2 CC01601 c1ccc(cc1)CCN2CCN(CC2)S(=O)(=O)c3cccc4c3non4 HTS01825 c1ccc(c(c1)C(F)(F)F)n2c(=O)n(c(=O)s2)CC3CC3 HTS01834 Cc1c(cnn1c2ccc(cc2)F)C(=O)O CC00080 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)NC3CCN(CC3)Cc4ccccc4 HTS02288 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)C(=O)Nc3ccc4c(c3)OCO4 HTS00395 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2coc(c2C(=O)OC)C HTS00872 Cc1ccnc(c1)n2c(ccc2C)C HTS00297 Cc1c(c(on1)C)NC(=O)NCC2CCN(CC2)S(=O)(=O)c3ccccc3 HTS02367 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3c[nH]nc3c4cccs4)C(=O)OC HTS04322 c1cc2c(cc1CNC(=O)CN3CCC(CC3)C(=O)N)OCO2 HTS04249 Cc1cc(nn1c2ccccc2)C(=O)NC3CCN(CC3)Cc4c(cccc4Cl)F HTS02406 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)c3ccc4c(c3)OCCCO4 HTS02149 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCN(CC4)Cc5c(cccc5Cl)F AW01191 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)c2ccc(cc2)F HTS02021 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)NNC(=O)c3ccc(cc3)Cl HTS01569 c1cc(cc(c1)S(=O)(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F)C(F)(F)F HTS00179 c1ccn(c1)C2CCN(CC2)S(=O)(=O)c3cccc4c3nccc4 HTS00593 CCCCCc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CCc3ccccc3 HTS01830 c1cc(oc1)c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)NC(=O)Nc4ccc(cc4)OC(F)(F)F SP01043 CC(C)(C)c1c(c(n(n1)C)C(C)(C)C)[N+](=O)[O-] SEW06666 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)Nc3ccc(cc3)F HTS02228 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)Nc3ccc(cc3)OC HTS02230 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccccc2c3ccccc3 HTS04381 c1cc(sc1)C(=O)NCCCN2CCN(CC2)c3nccc(n3)C(F)(F)F AW01225 c1cnc(nc1C(F)(F)F)N2CCN(CC2)CCCNC(=O)CCC(=O)O AW01227 c1cc(sc1)C(=O)NCCSCc2ccc(cc2Cl)Cl SEW06685 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCSCc3ccc(cc3Cl)Cl SEW06687 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)Cc3ccncc3 PD00765 c1ccc(c(c1)C(=O)Nc2ccc3c(c2)OCCO3)F HTS01881 CCCCCc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2N3CCOCC3)C(=O)OCC HTS02740 Cc1cc(c(nc1)NS(=O)(=O)c2ccc(cc2)F)Br HTS00127 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)OC(F)(F)F)c3ccco3 HTS02855 Cc1cn(c2c1cccc2)CCC(=O)Nc3ccccc3N4CCOCC4 HTS02294 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)N3CCN(CC3)c4ccccc4OC HTS02292 c1ccc(c(c1)/C=N/NC(=S)Nc2cccc(c2)Cl)O RJF00959 c1ccnc(c1)CCN(CCC#N)C(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F JP00909 c1ccc(cc1)c2csc(n2)NC(=O)c3ccco3 NH00363 Cc1cn(c2c1cccc2)CCC(=O)Nc3ccc(cc3)N4CCCCC4 HTS02295 Cc1ccc(cc1)S(=O)(=O)NCc2c(ccs2)C HTS04014 Cc1ccsc1CNS(=O)(=O)c2cccc3c2non3 HTS04016 c1ccc2c(c1)C(=O)N(C2=O)Cc3ccc(o3)C(=O)Nc4ccc(c(c4)C(F)(F)F)Br HTS01944 CN1CCN(CC1)c2ccc(cc2)NC(=O)c3c(nccn3)C(=O)O HTS02186 CCOC(=O)C1C(CC(=CC1=O)c2cccs2)c3ccc(c(c3Cl)OC)OC HTS00617 c1ccc2c(c1)c(c(c(=O)o2)CC(=O)c3ccc(cc3)[N+](=O)[O-])O HTS00209 CN1CCN(CC1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Cl HTS00071 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)CN3CCCCC3 HTS01899 Cc1ccc(cc1)Sc2c(cnc3c2c(nn3C)C)C(=O)O HTS01916 Cc1c(cc(o1)S(=O)(=O)N(C)C)C(=O)Nc2ccc(cc2)Cl HTS02223 Cn1cc(nc1)S(=O)(=O)Nc2ccccc2SCc3c(cccc3Cl)F HTS02195 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCC2CCN(CC2)S(=O)(=O)c3ccccc3 HTS02365 CCNC(=S)Nc1ccc(cc1)S(=O)(=O)Nc2cc(on2)C RJF01500 Cc1nc(cn1CCc2nc(on2)c3ccc(cc3)OC(F)(F)F)[N+](=O)[O-] HTS01917 Cc1nc(cn1CCc2nc(on2)c3ccsc3)[N+](=O)[O-] HTS02231 C1CN(CCC1C(=O)N)C(=O)/C=C/C(=O)O PD00754 COc1cc(c(cc1OC)NS(=O)(=O)c2ccsc2C(=O)OC)C(=O)OC HTS00107 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)S(=O)(=O)c4cccc(c4)C#N HTS00111 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)Nc3ccccc3 HTS02416 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)Nc3ccc(cc3)F HTS02422 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)N CC00094 c1cc(c(cc1C(F)(F)F)NC(=O)Nc2cc(ccc2F)F)N3CCOCC3 HTS02560 CC(C)(C)c1ccccc1NC(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS02517 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)NNc3c(cncc3Cl)Cl HTS03687 Cc1c(nc(s1)NC(=O)c2cccs2)CC(=O)OC HTS00252 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2cccc(c2)c3cnco3 HTS00154 COc1ccc2c(c1)cc([nH]2)C(=O)NCCSCc3ccc(cc3)F HTS00334 CCS(=O)(=O)c1ccc(c(c1)NC(=O)Nc2ccc(cc2)C(C)(C)C)O HTS04411 CC(C)(C)c1cc(c(s1)C(=O)OC)NC(=O)c2c(nccn2)C(=O)O HTS04415 Cc1ccsc1CNC(=O)Nc2ccc(cc2)C(F)(F)F HTS04008 c1ccc(c(c1)NS(=O)(=O)c2cccs2)SCc3c(cccc3Cl)F HTS02196 CC(C)(CC(=O)NC1CCN(CC1)Cc2c(cccc2Cl)F)CC(=O)O HTS02410 c1ccc(cc1)NC(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS02508 COC(=O)CNC(=O)c1ccncc1Br SPB08355 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)Cc2ccccc2F HTS00016 c1cc(nc(c1NC(=O)COCC(=O)O)N2CCOCC2)N3CCOCC3 HTS02193 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F HTS00044 Cc1c(cc(o1)S(=O)(=O)N2CCCCC2)C(=O)Nc3ccccc3 HTS00396 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2ccc3c(c2)OCCO3 HTS02028 Cc1ccsc1CNC(=O)c2ccc(cc2)Cl HTS04018 Cc1ccsc1CNC(=O)c2c(onc2c3ccccc3)C HTS04292 Cc1ccsc1Cn2c(ccc2C)C HTS04300 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)c3c(nccn3)C(=O)O)F HTS02411 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(cc3Cl)N(C)C)C(=O)OC HTS02616 COC(=O)c1cc(cn1c2ccc(cc2)Cl)/C=C(\C#N)/C(=O)OC SEW06673 COc1ccc2c(c1)c3c([nH]2)C(=O)NCC3 RJC04061 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)CSCC(=O)O)F HTS02408 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)COCC(=O)O)F HTS02409 CC(C)(C)OC(=O)NC1(CC1)C(=O)O SB02070 c1ccc2c(c1)-c3ccccc3C2COC(=O)NC4(CC4)C(=O)O SB02071 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2cccc(c2)C(F)(F)F HTS02032 Cc1ccccc1NC(=O)NCC2CCN(CC2)C(=O)OC(C)(C)C HTS02343 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)Nc3ccc(cc3)F HTS02417 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(c(nn2C)C(F)(F)F)c3ccc(cc3)F HTS02418 c1cc(c(c(c1)Cl)CN2CCN(CC2)CCCNC(=O)c3ccc(c(c3)Cl)Cl)F AW01208 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCC3CCN(CC3)C(=O)OC(C)(C)C HTS02023 CC(=O)c1ccc(cc1)OCC(=O)O SP01476 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)NCC3CCN(CC3)C(=O)OC(C)(C)C HTS02031 CCCc1c(cnn1c2ccccc2)C(=O)N(c3cc(ccn3)C)C(=O)c4cnn(c4CCC)c5ccccc5 HTS03539 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)Nc3ccc(cc3)OC(F)(F)F)F HTS02210 c1cc(sc1)S(=O)(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS00178 Cc1cc(ccc1NC(=O)COCC(=O)O)C(C)(C)C HTS02063 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)c3ccco3 HTS00346 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)c3ccco3 HTS00347 CCCc1c(cnn1c2ccccc2)C(=O)N3CCN(CC3)c4ccccc4OC HTS03788 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)CC(COc5ccc(c(c5)Cl)Cl)O AW01213 Cn1c2ccccc2c(n1)NC(=O)Cn3ccc(n3)C(F)(F)F HTS02215 c1ccc2c(c1)C[C@H](NC2)CO SPB08426 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)c3ccccc3C(=O)O HTS01718 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3cc(nn3c4ccccc4)c5ccccc5 HTS03559 c1cc(cnc1)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl HTS01318 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3Cl)C(F)(F)F HTS02737 COc1cc(c(cc1OC)NC(=O)C2CCC2C(=O)O)C(=O)OC HTS00614 CC(=O)Nc1cccc(c1)n2nc(nn2)SCc3cc(cc4c3OCOC4)Cl HTS02155 CCCCc1ccc(cc1)NC(=O)Nc2cc(nn2C)C HTS04325 c1cc(ccc1C(=O)Nc2ccc3c(c2)OCCO3)F HTS01867 Cn1c(nnc1SCC(=O)O)c2ccc3c(c2)cccn3 KM10672 Cn1c(nnc1SCCS(=O)(=O)c2ccc(cc2Cl)Cl)c3ccco3 HTS02852 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4ccc(cc4)[N+](=O)[O-] HTS02374 CCn1c(cc(n1)C)C(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F HTS00881 COc1ccc(cc1O)C2Nc3ccccc3C(=O)N2 HTS02006 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)c2c(noc2C)C HTS04132 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2cccc3c2nccc3 HTS02026 c1ccc(cc1)NC(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F HTS02211 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)c3ccco3 HTS00344 Cc1ccc2c(c1)CCCN2CC(=O)Nc3ccccc3 HTS02132 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(c(nn2C)C(F)(F)F)c3cccc(c3)C(F)(F)F HTS02424 c1cc(ccc1c2nc(on2)c3ccc4c(c3)CCO4)F HTS02105 CN(c1cnc2ccccc2n1)NC(=O)c3ccncc3Cl SEW06680 Cc1ccc(cc1)C(=O)Nc2c(nn(c2C(C)(C)C)C)C(C)(C)C SEW06684 COC(=O)/C=C/C(=O)Nc1ccccc1 PD00766 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2cc(sc2Cl)Cl HTS02029 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2ccc(s2)c3cc(n(n3)C)C(F)(F)F HTS02030 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS00910 CCOC(=O)/C(=C/Nc1cc(ccc1Cl)Cl)/C#N HTS00298 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)c2ccsc2 HTS04135 c1ccc(c(c1)C(=O)O)SCCS(=O)(=O)c2ccc(cc2Cl)Cl HTS02260 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCCN2CCCN(CC2)C(=O)OC(C)(C)C AW01216 c1ccc(cc1)CN2CCN(CC2)CCCNC(=O)c3cccs3 AW01218 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)C(C[N+](=O)[O-])c4ccc(cc4C)Cl PD00760 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2cccc3c2non3 HTS02027 COC(=O)c1c(cc(s1)c2cccs2)N3C(=O)C=CC3=O HTS01044 CC(C)(CC(=O)N1CCCN(CC1)c2nc3ccc(cc3s2)Cl)CC(=O)O HTS01895 COc1ccc(cc1OC)S(=O)(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O HTS00211 Cc1c(cc(o1)S(=O)(=O)N(Cc2ccc(cc2)OC)Cc3cccn3C)C(=O)OC HTS00086 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)Nc3ccccc3 HTS02133 CCCCCc1ccc(cc1)S(=O)(=O)Nc2ccsc2C(=O)OC HTS02247 CCCCCc1ccc(cc1)S(=O)(=O)Nc2nc(cs2)CC(=O)OCC HTS02249 CC(C)(C)c1cc(n(n1)c2ccc(cc2)N3C(=O)COCC3=O)C(C)(C)C SEW06665 c1c(cc(c2c1COCO2)CO)F CC01909 c1ccc(cc1)NNC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl HTS01884 c1cc2c(cc1F)c(c[nH]2)CCCN3CCN(CC3)c4nc5cc(ccc5s4)Cl HTS01699 c1cc(c(c(c1)Cl)CSCCNC(=O)Nc2cc(cc(c2)Cl)Cl)F HTS01723 CC(C)(C)c1ccc(cc1)SCC(=O)NCc2ccc3c(c2)OCO3 HTS04245 COc1ccc(cc1)SCC(=O)NCc2ccc3c(c2)OCO3 HTS04246 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2ccccc2c3ccccc3 HTS04383 c1ccc(cc1)c2ccccc2NC(=O)c3c(nccn3)C(=O)O HTS04384 c1ccc(cc1)c2ccccc2NC(=O)CCCC(=O)O HTS04385 c1cc(ccc1NC(=O)c2c(nccn2)C(=O)O)N3CCOCC3 HTS02187 c1ccn(c1)c2cc(c(cc2Cl)N3C(=O)c4c(nccn4)C3=O)Cl HTS02462 c1cc(c(cc1C(=O)NCCSCc2ccc(cc2Cl)Cl)Cl)Cl SEW06688 c1ccc(cc1)c2nc(sn2)NCCCN3CCN(CC3)Cc4c(cccc4Cl)F AW01199 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)NCCCN2CCN(CC2)Cc3c(cccc3Cl)F AW01207 Cc1c(c(no1)c2ccccc2)N TL01028 c1cc(c(c(c1)Cl)CN2CCN(CC2)CCCNS(=O)(=O)c3cc(ccc3Cl)Cl)F AW01209 c1ccnc(c1)CNC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl HTS01874 c1cc2c(cc1NC(=O)C3CC3)OCCO2 HTS01878 Cc1cn(c2c1cccc2)CCC(=O)Nc3ccc(cc3)N4CCOCC4 HTS02293 Cc1cc(ccc1NS(=O)(=O)c2ccc3c(c2)OCCO3)F HTS02352 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)CNS(=O)(=O)c3cccc4c3non4 HTS02369 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)CNS(=O)(=O)c3cccs3 HTS02495 Cc1c(cc(o1)S(=O)(=O)N(C)C)C(=O)Nc2ccccc2 HTS00483 Cc1cc(c(nc1)NS(=O)(=O)c2ccccc2)Br HTS00128 CN(C)c1ccc(cc1)n2c(nnn2)SCc3c(cccc3Cl)F HTS00695 CN(C)c1ccc(cc1)n2c(nnn2)SCC(=O)Nc3ccc(cc3)OC(F)(F)F HTS02546 CC(C)(C)C(=O)CSc1nnc(n1c2ccccc2C(F)(F)F)O HTS02453 CC1=C(CC(C(C1)C(=O)Nc2ccsc2C(=O)OC)C(=O)O)C PD00753 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)Nc3ccc(cc3)Cl HTS02227 c1ccc2c(c1)CCC3C2=Nc4ccccc4SC3c5ccc(cc5)F JFD02625 c1ccc(c(c1)C(=O)O)SCCS(=O)(=O)c2cccc(c2)C(F)(F)F HTS02259 COc1ccccc1NC(=O)Nc2ccccc2OC HTS00879 CCOC(=O)N1CCN(CC1)S(=O)(=O)c2ccc(cc2)C(F)(F)F HTS00046 Cc1c(c(nc(n1)c2ccccn2)SCC(=O)c3ccccc3)Cl HTS02083 Cc1ccc(c(c1)C)n2c(nnn2)SCC(=O)N3CCOCC3 HTS02081 CC1CCN(CC1)c2nc(ns2)c3ccccc3 HTS02582 c1ccc2c(c1)c(=O)c(co2)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)Cl HTS00150 COC(=O)c1cscc1S(=O)(=O)N2CCN(CC2)c3coc4ccccc4c3=O HTS00151 Cc1cc(c(o1)C(F)(F)F)C(=O)Nc2nc(c(s2)C)CC(=O)OC HTS00251 c1cc(ccc1C(=O)CN2CCN(CC2)CCCc3c[nH]c4c3cc(cc4)F)F HTS01701 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)c3ccccc3 HTS02140 CCOC(=O)c1ccc2c(c1)c(c([nH]2)C(=O)OCC)CCC(=O)O SEW06662 Cn1c(nnc1SCC(=O)c2ccc(cc2)F)c3ccco3 HTS02460 c1ccn(c1)c2ccsc2NC(=O)NCc3ccco3 HTS04258 CC(C)(C)c1ccc(cc1)NC(=O)Nc2c(ccs2)n3cccc3 HTS04259 c1cc(c(cc1c2csc(n2)NC(=O)Nc3ccc(cc3F)F)F)F HTS02511 Cc1nc(cn1CC(c2ccc3c(c2)OCCCO3)O)[N+](=O)[O-] HTS00299 c1cc(cc(c1)NC(=O)NCCSCc2c(cccc2Cl)F)C(F)(F)F HTS01726 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)C(=O)Nc3ccsc3C(=O)OC HTS02221 Cc1c(cc(o1)S(=O)(=O)N(C)C)C(=O)Nc2ccsc2C(=O)OC HTS02224 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4cn(c(n4)C)C HTS02371 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4ccc(s4)c5ccccn5 HTS02376 Cn1c(ccc1S(=O)(=O)NNC(=O)c2cn3cc(cc(c3n2)Cl)C(F)(F)F)C(=O)OC HTS01560 c1ccc2c(c1)CCC3C2=Nc4ccccc4SC3c5ccc(cc5)Cl JFD02626 c1ccc2c(c1)c(on2)C(=O)O PD00830 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)N3CCCCC3 HTS02641 Cc1c(c(nc(n1)c2ccccn2)SCC(=O)N3CCOCC3)Cl HTS02085 CC(C)(C)c1ccccc1NC(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F HTS02217 CCCCCc1ccc(cc1)S(=O)(=O)NCC2CCN(CC2)C(=O)OC(C)(C)C HTS02034 COc1ccc(cc1)NC(=O)CC2C(=O)NCCN2 HTS01733 c1cc2c(cc1S(=O)(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F)OCCO2 HTS02350 c1cc(ccc1NS(=O)(=O)c2ccc3c(c2)OCCO3)F HTS02351 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)CNC(=O)Nc3ccc(cc3)F HTS02364 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4ccc(c(c4)Cl)NC(=O)C HTS02160 Cc1cc(=O)c2ccccc2o1 JFD02612 c1ccc2c(c1)cc(o2)c3cc(=O)c4ccccc4o3 JFD02614 Cc1ccc(cc1)C2C3CSc4ccccc4C3=Nc5ccccc5S2 JFD02633 c1ccc2c(c1)CCN(C2)C(=O)c3c(nccn3)C(=O)O HTS02168 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4ccccc4 HTS04391 Cc1c(cc(o1)S(=O)(=O)N2CCOCC2)c3nc(no3)c4ccc(cc4)C(F)(F)F HTS02226 c1cc(ccc1n2c(c(cn2)C(=O)N3CCN(CC3)c4c5c(ccs5)ncn4)C(F)(F)F)Cl HTS00100 CCn1c2ccc(cc2c3c1C(=O)CCC3)OCc4ccccc4 RJC04063 CN(c1nc(cs1)c2ccc(s2)Cl)C(=O)c3ccc(cc3)F HTS00027 CC1(CN(C1=O)c2ccsc2C(=O)OC)C HTS02229 Cc1ccc(cc1)S(=O)(=O)CCN2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F HTS02441 c1cc(c(cc1Cl)Cl)S(=O)(=O)CCN2CCN=C(C=C2)C(F)(F)F HTS02442 Cc1cc(no1)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS02241 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4cc5ccccc5s4 HTS01768 Cc1cc(no1)C(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F HTS02405 c1ccc2c(c1)C(=O)C(C2=O)(NC(=O)c3ccc(cc3)c4csnn4)O HTS01964 Cc1cc(c(o1)C)C(=O)Nc2c3c(cccc3OC)n(n2)C HTS03813 COc1ccc(cc1)Oc2ccc(cc2N3C(=O)c4c(nccn4)C3=O)C(F)(F)F HTS04056 Cc1cc(c(o1)C(F)(F)F)NC(=O)NC2CCN(CC2)Cc3ccccc3 HTS04296 c1ccc(cc1)CN2CCN(CC2)CCCNC(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F AW01215 CCCc1cnc(nc1)N2CCCN(CC2)C(=O)OC(C)(C)C AW01228 COc1ccc(cc1NC(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F)Cl HTS02219 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)Oc4cccc(c4C#N)Cl HTS02642 Cc1cc(ccc1NS(=O)(=O)c2ccc(cc2)Oc3cccc(c3C#N)Cl)C(C)(C)C HTS02644 Cn1cc(nc1)S(=O)(=O)N(Cc2ccccc2)Cc3cccs3 HTS02207 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=O)c4ccc(cc4)F)C(F)(F)F HTS01785 c1cc2c(cc1Cl)sc(n2)N3CCCN(CC3)C(=O)COCC(=O)O HTS01892 c1ccc(cc1)CCC(=O)NN2CC(=O)N(CC2=O)c3cc(cc(c3)Cl)Cl HTS02091 Cc1cc(nc(c1C#N)SCC(c2cccc(c2)[N+](=O)[O-])O)C HTS02095 Cc1c(ccc(n1)C(F)(F)F)C(=O)NN2CCOCC2 HTS03359 c1cc(ccc1C(F)(F)F)NC(=O)Nc2ccc(cc2)C(F)(F)F HTS00880 c1ccc(cc1)CN(Cc2cccs2)C(=O)COCC(=O)O HTS02203 c1ccc2c(c1)CCN(C2)c3ccc(cc3NC(=O)c4ccc(cc4)C(F)(F)F)C(F)(F)F HTS01787 c1ccc2c(c1)CCN(C2)c3ccc(cc3NS(=O)(=O)c4cccc5c4non5)C(F)(F)F HTS01790 Cc1ccc(cc1)S(=O)(=O)CCSc2nnc(n2c3ccccc3C(F)(F)F)O HTS04172 c1c(cnc(c1Cl)N2CCC(CC2)N3C(=O)CC4(C3=O)CCCC4)C(F)(F)F AW01222 c1ccc2cc(ccc2c1)c3csc4c3c(ncn4)N5CCc6ccccc6C5 AW01224 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCCN2CCN(CC2)c3nccc(n3)C(F)(F)F AW01226 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NC(=O)c3ccco3 HTS00345 c1ccc2c(c1)c(c(s2)C(=O)NNc3c(cccc3Cl)Cl)Cl HTS06164 CCCc1cnc(nc1)N2CCN(CC2)C(=O)c3ccccc3 HTS05869 Cc1ccsc1CNC(=O)c2ccccc2C(=O)O HTS04004 c1ccn(c1)c2ccsc2NC(=O)NCC3CC3 HTS04260 c1cc(sc1)c2ccnc(n2)SCC(=O)c3ccc(cc3)F HTS04398 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)Nc2ccc(cc2F)F HTS02038 Cc1ccc(cc1)S(=O)(=O)CCSc2nc(cc(n2)O)COC HTS02276 COCc1cc(nc(n1)SCC(=O)c2ccccc2)O HTS02431 CCc1ccccc1CSc2c(c(cc(n2)C)C)C#N HTS02096 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)C HTS02158 Cc1ccc2c(c1)n(c(=O)o2)Cc3ccc(cc3)F HTS04442 c1ccc(cc1)NC(=O)Nc2cccc(c2)C(=O)O HTS03989 c1ccc(cc1)C(=O)N2CC(=O)N(CC2=O)C(=O)c3ccccc3 HTS00878 CC(C)c1ccc(cc1)NC(=O)CSCc2csc3c2cccc3 HTS05551 c1ccc(cc1)N2C(=O)c3c(nccn3)C2=O HTS03749 Cc1ccccc1C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS04093 CC(C)c1ccc(cc1)NNC(=O)c2cc3ccccc3s2 HTS03876 Cc1ccc(cc1NC(=O)CCn2cc(c3c2cccc3)C)F HTS01438 c1cc2c(cc1NC(=O)CSCC(=O)O)C(=O)OC2 HTS04479 CC1(c2ccccc2N3C1(NC(=O)C3)/C=C/C=C/c4ccc(cc4)N(C)C)C BTB15229 C1CC1c2nnc(s2)NC(=O)C3CCC3C(=O)O HTS03440 c1cc(sc1c2ccno2)S(=O)(=O)N3CCN(CC3)c4ccncc4 HTS05768 CC1(CCc2cc(ccc2O1)CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)C HTS05408 c1cc2c(cc1CN3CCN(CC3)C(=O)c4c(ccs4)Br)OCO2 HTS03259 c1cc2c(cc1CNCC(=O)NCc3ccc4c(c3)OCO4)OCO2 HTS04248 Cc1cc(n2c(n1)c(c(n2)C(F)(F)F)c3ccccc3)C HTS03479 c1cc(ccc1C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3)Cl HTS04092 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)C(=O)NC3CCCCC3 HTS03612 c1ccc2c(c1)CC(C2)NCc3nc(no3)c4cccs4 HTS03625 c1cc(nc(c1NC(=O)/C=C/C(=O)O)N2CCOCC2)N3CCOCC3 HTS02194 Cc1cc(no1)C(=O)Nc2c3ccccc3n(n2)C HTS02209 c1cc(ccc1NC(=O)COCC(=O)O)S(=O)(=O)N HTS04060 c1cc(ccc1NC(=O)CCCC(=O)O)S(=O)(=O)N HTS04064 CCc1ccnc(c1)NS(=O)(=O)c2ccc(c(c2)OC)OC HTS05399 c1cc(oc1)C=C(C(=O)N)C(=O)N HTS02002 c1c(cc(c2c1COCO2)CNC(=O)C3CC3)F HTS03232 c1ccc2c(c1)C(=O)N(C2=O)c3ccccc3N4CCOCC4 HTS06773 c1ccc(c(c1)N2CCOCC2)N3C(=O)CSCC3=O HTS06775 Cc1ccc(cc1Cl)NNC(=O)c2ccno2 HTS03643 c1cc(cc(c1)NC(=O)c2cccs2)C(=O)O HTS04233 c1cc2c(cc1Cl)c(cs2)CNC(=O)CCC(=O)O HTS03893 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2cccc3c2cccc3 HTS04371 Cc1cc(cc(c1)NC(=O)Nc2cc(nn2C)C(C)(C)C)C HTS04373 CCCCc1ccc(cc1)NC(=O)Nc2cc(nn2C)C(C)(C)C HTS04653 Cc1nc(cn1CC(c2ccc(cc2)c3ccccc3)O)[N+](=O)[O-] HTS01864 c1cc2c(cc1c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)CCO2 HTS02103 c1cc(c(c(c1)Cl)/C=N/O)F SPB08294 Cc1c(c(on1)C)C(=O)NNc2c(cncc2Cl)Cl HTS03080 CCOc1ccccc1N2CCN(CC2)Cc3ccccc3N4CCC(CC4)C(=O)OCC HTS04098 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)N3CCOCC3 HTS06776 c1ccc(c(c1)NS(=O)(=O)c2ccc3c(c2)CCO3)Sc4nc5ccc(cc5s4)Cl HTS03299 COc1ccc(cc1)C(=O)Nc2ccccc2Sc3nc4ccc(cc4s3)Cl HTS03931 c1ccc2c(c1)cc(s2)C(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F HTS02166 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)c3cccnc3 HTS01645 CCCCCc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)NS(=O)(=O)C)C HTS04139 CCc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)NS(=O)(=O)C)C HTS04140 Cc1cc(c(o1)C)C(=O)NCCSCc2ccc(cc2)[N+](=O)[O-] HTS04333 Cc1cc(c(o1)C)C(=O)NC2Cc3ccccc3C2 HTS04335 Cc1cc(c(o1)C)C(=O)NCc2ccc3c(c2)OCO3 HTS04338 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC(=O)c5ccc(cc5)F HTS02044 c1ccc(cc1)CN2CCN(CC2)CCCNS(=O)(=O)c3cccc(c3Cl)Cl AW01221 c1ccc2cc(ccc2c1)c3csc4c3c(ncn4)N5CCOCC5 AW01223 Cc1c(sc(n1)C(=O)NCc2cc(cc3c2OCOC3)F)c4ccc5c(c4)CCO5 HTS03228 c1cnoc1C(=O)NCc2cc(cc3c2OCOC3)F HTS03233 c1cnc(c(n1)C(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl)C(=O)O HTS04449 c1ccc(cc1)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS02234 Cn1c(nnc1Sc2nc3ccc(cc3s2)Cl)Cc4ccsc4 HTS03450 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccc(cc3)C(C)C HTS03887 c1ccc(c(c1)C(=O)NCc2csc3c2cc(cc3)Cl)C(=O)O HTS03894 CC(=O)Nc1ccc(cc1)Oc2nc(ns2)c3ccccc3 HTS02100 c1cc(ccc1C(=O)NCCSCc2ccc(cc2Cl)Cl)Cl SEW06689 c1cc(c(c(c1)F)C(=O)NCCSCc2ccc(cc2Cl)Cl)F SEW06690 Cc1nc(cn1CC(=O)c2ccc(cc2)F)[N+](=O)[O-] HTS00296 CN(C)c1ccc(cc1)n2c(nnn2)SCc3cc(cc(c3)F)F HTS00694 Cc1cc(n(n1)C)NC(=O)Nc2ccc(cc2F)F HTS03839 COc1ccccc1c2nnc(n2c3ccccc3)Sc4nc5ccc(cc5s4)Cl HTS04021 c1cc(ccc1NS(=O)(=O)c2ccc3c(c2)CCO3)Cl HTS02235 Cc1csc(c1NS(=O)(=O)c2ccc3c(c2)CCO3)C(=O)OC HTS02240 Cc1ccnc(c1)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS02243 CCOC(=O)c1cnc(nc1N)SCc2ccc(cc2)Cl HTS02123 c1cc(sc1)S(=O)(=O)Cc2nc(cs2)c3ccc(s3)Cl.Br HTS00032 Cc1c(snn1)c2nc(cs2)c3ccc(s3)Cl.Br HTS00034 CN(c1nc(cs1)c2ccc(s2)Cl)C(=O)C3CCCCC3 HTS00244 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)C#N HTS06243 CCCc1ccc(cc1)C(=O)NNc2ccc(cc2)S(=O)(=O)N HTS04481 CC1c2cc(c(cc2CCN1C(=O)Nc3ccc4c(c3)OCCO4)OC)OC HTS05930 Cc1cccc(c1)Cn2c3cc(ccc3oc2=O)C HTS04443 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)CNC(=O)Nc3ccc(cc3F)F HTS02368 COc1ccc(cc1)Oc2nc(ns2)c3ccccc3 HTS02524 Cc1ccc(cc1)N/C=C/2\C(=O)N(C(S2(=O)=O)c3cccnc3)c4ccc(cc4F)F S13395 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc(s3)S(=O)(=O)c4ccccc4 HTS06073 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3cn(cn3)C HTS06074 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2cn(cn2)C HTS02035 Cc1c2c(c(sc2nc(n1)c3ccccc3)C(=O)c4ccc(cc4)F)N HTS02501 Cc1c2c(c(sc2nc(n1)c3ccccc3)C(=O)c4cc5ccccc5o4)N HTS02502 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)Nc2cc(ccc2OC)Cl HTS00058 c1ccc2c(c1)ccc(n2)NC(=O)Nc3ccc(cc3)F HTS06271 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)Nc2ccc(cc2)C#N HTS05201 COc1ccc(cc1)Oc2ccc(cc2NC(=O)CC(CC(=O)O)c3ccccc3)C(F)(F)F HTS06054 CCCc1cnc(nc1)N2CCN(CC2)CC(=O)N(c3ccccc3)C4CCCCC4.C(=C/C(=O)O)\C(=O)O HTS03942 c1ccnc(c1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS03955 CN(c1ccc(cc1C(=O)c2ccccc2)Cl)C(=O)c3cccs3 HTS04261 CCCc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)NS(=O)(=O)C)C HTS04591 CC(=O)Nc1ccc(cc1)NC(=O)CC(CC(=O)O)c2ccccc2 HTS06051 CCCc1cnc(nc1)N2CCN(CC2)C(=O)c3c(c4ccccc4s3)Cl HTS05873 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3Cl)NC(=O)C HTS06242 c1ccc2c(c1)ccc(n2)NC(=O)Nc3ccccc3F HTS06272 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3c(noc3C)C)C HTS04144 CCCc1cnc(nc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)C(=O)C HTS03300 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=O)c3c(nccn3)C(=O)O)O HTS02185 c1cc2c(ccnc2cc1Cl)N3CCNCC3 KM10724 CC(c1ccco1)NCc2ccccc2 RJC04067 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)C4CC(=O)N(C4=O)c5ccccc5 PD00758 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)NCc3ccncc3)Cl HTS01876 c1cc(sc1)C(=O)Nc2ccc3c(c2)OCCO3 HTS01879 c1cc(ccc1C(=O)Nc2ccc3c(c2)OCCO3)C(F)(F)F HTS01880 c1cc(cnc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS03956 Cc1ccsc1CNC(=O)CC(C)(C)CC(=O)O HTS04007 c1cc2c(nc1)sc(n2)SCC(=O)O HTS02159 Cc1c(cn(n1)C)NC(=O)Nc2cc(ccc2OC)Cl HTS03838 Cn1c2cccc(c2c(n1)NC(=O)CCC(=O)O)OC HTS03832 Cc1ccc(cc1)NC(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS03460 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)Nc2cc(cc(c2)Cl)Cl HTS02036 COc1cc(c(cn1)C(=O)NC2(C(=O)c3ccccc3C2=O)O)C(F)(F)F HTS01956 CCCc1cnc(nc1)N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCCO4 HTS03941 C[C@H](c1ccccc1)NC(=O)C HTS06398 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C#N HTS05197 Cc1cc(c(cc1NC(=O)c2ccccc2)OC)NC(=O)CC(CC(=O)O)c3ccccc3 HTS06057 CN(c1ccc(cc1C(=O)c2ccccc2)Cl)C(=O)c3ccc(cc3)Cl HTS03150 CCCc1cnc(nc1)N2CCN(CC2)c3nc4ccc(cc4s3)Cl HTS03947 CCc1[nH]c(c(n1)C)/C=C\2/c3ccccc3NC2=O HTS05063 c1cc2c(cc1CN3CCN(CC3)C(=O)CCCC(=O)O)OCO2 HTS03707 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 HTS03708 CCOC(=O)c1c2c(sc1NC(=O)NS(=O)(=O)c3ccc(cc3)C)CN(CC2)C HTS02983 c1cc(sc1)C(=O)NN2CC(=O)N(CC2=O)c3cc(cc(c3)Cl)Cl HTS02089 c1ccc2c(c1)C(=O)NC(N2)c3ccc(cc3)OC(F)(F)F HTS02004 c1ccnc(c1)c2ccc(s2)C(=O)NCc3cc(cc4c3OCOC4)F HTS03229 CCCCCc1ccc(cc1)S(=O)(=O)Nc2ccc(c(c2)C(=O)OCC)N3CCCCC3 HTS02678 Cn1c(nnc1Sc2nc3ccc(cc3s2)Cl)c4cccs4 HTS03446 c1cc(sc1)c2cc(nn2c3ccc(cc3)NC(=O)c4cccs4)C(F)(F)F HTS04032 c1cc2c(cc1CN3CCN(CC3)C(=O)COCC(=O)O)OCO2 HTS03703 c1cc2c(cc1CN3CCN(CC3)C(=O)c4c(nccn4)C(=O)O)OCO2 HTS03705 Cc1c(c(nc(n1)c2ccccn2)SCC(=O)c3ccc(cc3)F)Cl HTS02084 c1ccc(c(c1)CNC(=O)c2ccccc2C(=O)O)OC(F)(F)F HTS03896 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3cccc4c3non4 HTS06072 c1ccc(cc1)CCC(=O)NNc2ccc(cc2F)F HTS06151 CCc1ccc(cc1)C(=O)NNc2ccc(cc2F)F HTS06152 Cc1cc(no1)C(=O)NNc2ccc(cc2F)F HTS06154 c1cc(c(c(c1)Cl)Cl)NC(=O)CSc2nccc(n2)c3cccs3 HTS04575 CCc1ccnc(c1)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS04559 CCc1ccnc(c1)NC(=O)c2ccccc2 HTS04803 c1cc2c(cc1C(=O)N3CCC(CC3)C(=O)O)OCO2 HTS07097 c1c(cc(c2c1COCO2)C(=O)N3CCC(CC3)C(=O)O)F HTS07098 c1ccc(cc1)CN2C(=O)c3ccccc3NS2(=O)=O HTS03690 c1ccnc(c1)N2CCN(CC2)CCS(=O)(=O)c3ccc(cc3Cl)Cl HTS02443 c1cc(sc1)C(=O)NNc2c(cncc2Cl)Cl HTS03082 Cc1ccsc1C2C3=C(CC(CC3=O)(C)C)NC(=C2C(=O)OC)C HTS04692 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)c3cccnc3 HTS01643 c1ccc(c(c1)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)C(=O)O HTS03706 Cc1ccsc1CNC(=O)CSCC(=O)O HTS04003 Cc1ccsc1CNC(=O)CCC(=O)O HTS04005 Cc1cc(c(c(c1)C)n2c(nnn2)SCC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C HTS01986 CC(C)(C)C(=O)Nc1c(c(nn1C)C(F)(F)F)c2ccc(cc2)OC HTS00349 Cc1ccc(cc1NC(=O)Nc2cc(nn2C)C(C)(C)C)F HTS04655 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccncc3)Cl HTS01319 CC(C)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)c3cc(sc3C(F)(F)F)C(=O)OC HTS03716 c1ccc(cc1)C(CN2CCN(CC2)Cc3ccc4c(c3)OCO4)O HTS04120 c1cc(sc1)C(=O)NNc2cc(ccc2Cl)Cl HTS03067 c1ccc(cc1)n2c(c(cn2)C(=O)NC3(C(=O)c4ccccc4C3=O)O)C(F)(F)F HTS01859 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NC(=O)c3ccc(c(c3)OC)OC HTS02282 c1cc(cnc1)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS03458 c1cc2c(cc1NC(=O)c3ccno3)OCCO2 HTS04147 Cc1c(c(on1)C)C(=O)Nc2ccc3c(c2)OCCO3 HTS04148 c1cc2c(cc1C(=O)Nc3ccc4c(c3)OCCO4)non2 HTS04150 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NC(=O)c3cccnc3 HTS01644 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)NCCSCc3cccc(c3)C(F)(F)F HTS02286 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)c3ccc(c(c3)OC)OC HTS02281 COc1cc(c(cc1OC)NS(=O)(=O)C)C(=O)OC HTS01823 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)c3ccc(c(c3)OC)OC HTS02283 c1ccc2c(c1)cc(s2)C(=O)N3CCCN(CC3)c4nc5ccc(cc5s4)Cl HTS02163 c1cc2c(c(c1)S(=O)(=O)NC3CCN(CC3)Cc4c(cccc4Cl)F)non2 HTS02220 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)c3ccc(cc3)OC HTS02151 c1ccc(cc1)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04033 Cc1c(cnn1c2ccc(cc2)OC)C(=O)Nc3ccc(cc3)F HTS04306 c1cc(sc1)C(=O)NNc2ccc(cc2F)F HTS06156 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccc(cc3F)F HTS06160 Cn1c(ccc1S(=O)(=O)N(Cc2ccccn2)Cc3ccccn3)C(=O)O HTS01756 Cn1c(ccc1S(=O)(=O)NCc2ccco2)C(=O)O HTS01758 c1ccc(cc1)NC(=O)NCC2CCN(CC2)S(=O)(=O)c3ccccc3 HTS02366 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)c2ccc(cc2F)F HTS02022 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)c2cccs2 HTS02024 Cn1c2cccc(c2c(n1)NC(=O)CSCC(=O)O)OC HTS03834 Cn1c2cccc(c2c(n1)NC(=O)c3c(nccn3)C(=O)O)OC HTS03835 Cc1cc(n(n1)C)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS04324 c1ccc2c(c1)-c3c(cccc3C(=O)NC4(C(=O)c5ccccc5C4=O)O)C2=O HTS01959 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)NCCCN2CCN(CC2)Cc3ccccc3 AW01219 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc(s3)c4ccno4 HTS06075 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)Oc2ccccc2N3CCCCC3 HTS06190 c1ccc2c(c1)c(c(s2)C(=O)Oc3ccccc3N4CCCCC4)Cl HTS06192 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4)C HTS04043 c1cc(cc(c1)NC(=O)c2ccco2)C(=O)O HTS04235 COc1ccc(cc1OC)C(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F HTS02407 Cc1ccc2c(c1)n(c(=O)o2)CC(=O)N3CCOCC3 HTS04444 Cc1ccc2c(c1)n(c(=O)o2)CC(=O)C(C)(C)C HTS04445 CCCc1cnc(nc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)F HTS03944 c1cc(ccc1N2C(=O)c3c(nccn3)C2=O)S(=O)(=O)N4CCOCC4 HTS02468 Cc1ccc(cc1)S(=O)(=O)NCCN2CCNC2=O HTS02479 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCCN3CCNC3=O HTS02483 c1cc(nc(c1NC(=O)CSCC(=O)O)N2CCOCC2)N3CCOCC3 HTS02192 c1ccc(cc1)CN2CCN(CC2)CCNC(=O)c3c(nccn3)C(=O)O HTS03745 Cn1c2cccc(c2c(n1)NS(=O)(=O)c3cc(sc3Cl)Cl)OC HTS03828 c1ccc2c(c1)CCC3C2=Nc4ccccc4SC3c5ccc(cc5)[N+](=O)[O-] HTS00891 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccc(cc3F)F HTS06159 c1cc(c(c(c1)Cl)C(=O)NNc2ccc(cc2)Cl)F HTS05650 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNc3ccc(cc3)OC(F)(F)F HTS05644 COc1ccc(cc1)SCCC(=O)NNS(=O)(=O)c2cccc(c2)Cl HTS05852 CCCc1ccc(cc1)C(=O)NNc2ccc(cc2)OC HTS04500 COc1ccc(cc1)NNC(=O)c2cccs2 HTS04742 CCOC(=O)c1cccc(c1)NC(=O)Nc2ccc3c(c2)C(=O)OC3 HTS03391 CCCCCc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)C(=O)OC3 HTS03395 c1ccc(cc1)C(CN2CCC(CC2)C(=O)N)(c3ccccc3)O HTS05466 COc1ccc(cc1OC)S(=O)(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl HTS05002 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc3ccccc3n2 HTS05968 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NS(=O)(=O)c4c(noc4C)C HTS04586 c1ccc(c(c1)C(=O)Nc2ccc(c(c2)C(F)(F)F)Br)C(=O)O HTS01934 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4ccc5c(c4)OCCO5 HTS02353 c1ccc(c(c1)N2CCCCC2)OC(=O)c3c(ccs3)Cl HTS06194 c1ccc(cc1)NC(=O)Nc2ccc3ccccc3n2 HTS05970 c1cc2cccnc2c(c1)S(=O)(=O)Nc3ccc4c(c3)C(=O)OC4 HTS03397 CCc1ccc(cc1)C(=O)NNc2ccccc2C(F)(F)F HTS03403 CCS(=O)(=O)c1ccc(c(c1)NC(=O)COCC(=O)O)O HTS04068 CCS(=O)(=O)c1ccc(c(c1)NC(=O)c2ccccc2C(=O)O)O HTS04069 c1ccc(cc1)CN2CCN(CC2)CCNC(=O)Nc3cc(cc(c3)Cl)Cl HTS03184 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3c(c4cc(ccc4s3)Cl)C HTS05879 CC1c2cc(c(cc2CCN1C(=O)Nc3ccccc3)OC)OC HTS05929 CC1c2cc(c(cc2CCN1C(=O)Nc3ccc(cc3)OC(F)(F)F)OC)OC HTS05932 Cc1nc(cs1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)OC(F)(F)F HTS03128 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS02242 Cc1cc(no1)NS(=O)(=O)c2ccc3c(c2)OCCO3 HTS02349 c1cc(sc1)c2ccnc(n2)SCC(=O)Nc3ccc(cc3)Oc4ccc(cc4Cl)Cl HTS04567 Cc1c(c(on1)C)NC(=O)NCCN2CCN(CC2)Cc3ccccc3 HTS03187 Cc1c(csc1C(=O)NC2CCN(CC2)Cc3ccccc3)S(=O)(=O)c4ccc(cc4)Cl HTS03170 Cn1cc(nc1)S(=O)(=O)N2CCN(CC2)c3ccccn3 HTS06598 Cc1ccc(cc1)S(=O)(=O)CCN2CCN=C(C=C2)C(F)(F)F HTS02438 c1ccc(cc1)c2nc(sn2)Oc3ccc(cc3)Cl HTS02522 CC(C)(CC(=O)Nc1ccc(cc1)S(=O)(=O)N)CC(=O)O HTS04058 c1cc(ccc1NC(=O)CSCC(=O)O)S(=O)(=O)N HTS04061 CC(=O)Nc1c(c(nn1C)C(F)(F)F)c2ccc(cc2)Br HTS00340 CCCc1cnc(nc1)N2CCN(CC2)C(=O)c3cc(on3)C HTS05872 c1ccc(cc1)Oc2c(cccn2)C(=O)NN(c3ccc(cc3)OC(F)(F)F)C(=O)c4cccnc4Oc5ccccc5 HTS05658 Cc1c(snn1)C(=O)NNc2c(cncc2Cl)Cl HTS03081 Cc1csc(c1c2nc3ccccc3s2)NC(=O)Nc4ccc(cc4)F HTS04621 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3c(cccn3)C#N HTS05325 COC(=O)c1cscc1NC(=O)CC(CC(=O)O)c2ccccc2 HTS06052 c1cc(c(c(c1)Cl)NNC(=O)c2ccc(cc2F)F)Cl HTS06162 CCCc1cnc(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)F HTS05870 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)F)CN(CC2)C HTS02984 CCOC(=O)c1ccc(c(c1)NC(=O)CCCC(=O)O)N2CCOCC2 HTS03063 c1cc(cc(c1)Cl)NC(=O)CSc2nccc(n2)c3cccs3 HTS04569 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSc4nccc(n4)c5cccs5)C(F)(F)F HTS04573 c1cc(c(cc1Cl)NNC(=O)c2ccno2)Cl HTS03068 Cc1c(c(no1)c2ccccc2)C(=O)NNc3cc(ccc3Cl)Cl HTS03070 Cc1ccc(c(c1)C)NNC(=O)c2ccno2 HTS05344 CCCc1c(cnn1c2ccccc2)C(=O)NNc3ccccc3OC HTS05545 COc1ccccc1NNC(=O)C2CCCCC2 HTS05546 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NCCCOc3cccc(c3)NC(=O)C HTS02707 COC(=O)C1=C(CSC1)Nc2ccccc2NS(=O)(=O)c3ccc(cc3)OC(F)(F)F HTS04270 COC(=O)C1=C(CSC1)Nc2ccccc2NS(=O)(=O)c3ccc(cc3Cl)C(F)(F)F HTS04271 c1ccc(c(c1)C(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl)C(=O)O HTS04549 c1cc(c(nc1)NC(=O)CCC(=O)O)OCc2ccc(c(c2)Cl)Cl HTS04553 CCc1ccnc(c1)NC(=O)Nc2cccc3c2cccc3 HTS04556 CCc1ccc(cc1)C(=O)NNc2c(cncc2Cl)Cl HTS03078 c1ccc(cc1)C(CNC(=O)c2ccccc2)O HTS05981 CCc1ccnc(c1)NS(=O)(=O)c2ccc(cc2)C HTS05390 c1ccc(c(c1)NC(=O)N2CCN(CC2)c3c(cccn3)C#N)F HTS04985 Cc1nc(cs1)c2ccc(cc2)NC(=O)CC(C)(C)CC(=O)O HTS03132 c1c(c(c(cn1)Cl)NNC(=O)C2CCC2)Cl HTS03084 c1cc(sc1)c2ccnc(n2)SCC(=O)Nc3ccc(c(c3)Cl)F HTS04570 c1cc(sc1)c2ccnc(n2)SCC(=O)Nc3ccc(cc3)Cl HTS04571 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)F)N3CCOCC3 HTS07055 c1ccc(c(c1)NC(=O)c2ccc(cc2)OC(F)(F)F)N3CCOCC3 HTS07058 Cc1c(cnn1c2ccccc2)C(=O)N3CCC(CC3)c4ccccc4OC HTS02987 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(c(c3)O)OC)C(=O)OC HTS04688 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3c[nH]nc3c4ccccc4)C(=O)OC HTS04689 Cc1c(cnn1c2ccc(cc2)OC)C(=O)O CC00105 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)OC SP01428 c1ccc2c(c1)cc(o2)C(=O)Cc3c(c4ccccc4oc3=O)O PD00832 CC(=O)Nc1c(c(nn1C)C(F)(F)F)c2cccc(c2)C(F)(F)F HTS00342 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3c[nH]nc3c4ccc(cc4)OC)C(=O)OC HTS04687 CCOC(=O)c1c2c(sc1NC(=O)Nc3cc(ccc3Cl)OC)CN(CC2)C HTS02980 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3cscc3c4ccccc4)C HTS07048 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccccc3)C HTS07049 c1ccc(c(c1)NC(=O)c2ccco2)N3CCOCC3 HTS07063 COc1ccc(cc1OC)C(=O)Nc2ccccc2N3CCOCC3 HTS07062 c1ccc(cc1)NC(=O)N2CCN(CC2)c3c(cccn3)C#N HTS04984 COc1ccc(cc1)Oc2ccc(cc2NC(=O)Nc3csc4c3cccc4)C(F)(F)F HTS07207 Cc1ccc(n1c2ccc(cc2)C3(CCSc4c3cccc4)O)C HTS01633 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccccc3F)C HTS07231 CCCc1ccc(cc1)C(=O)NNc2c(cncc2Cl)Cl HTS03079 c1cc(ccc1c2cc(c(=O)[nH]n2)Cc3ccncc3)F HTS03957 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2)SCc3cccc(c3F)Cl HTS04658 CC(C)c1cc(c(c(c1)Br)NC(=O)NCCN2CCN(CC2)c3nccc(n3)C(F)(F)F)Br HTS03012 COc1ccc(cc1)OCC(CNC(=O)Nc2ccc(cc2)OCc3ccccc3)O HTS05281 CCc1ccnc(c1)NC(=O)c2ccc(nc2C)C(F)(F)F HTS04806 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl HTS05000 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)c2c(nns2)C HTS04133 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS04601 CCOC(=O)C1CCCN(C1)S(=O)(=O)c2ccc3c(c2)CCO3 HTS06912 c1cc(sc1)C(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 HTS06955 c1ccc2c(c1)CCN(C2)C(=O)c3ccc(cc3)Cl HTS07008 c1c(c(sc1Cl)Cl)S(=O)(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 HTS07125 c1cc(sc1)c2cc(nn2c3ccc(cc3)NC(=O)COCC(=O)O)C(F)(F)F HTS04050 c1ccc(c(c1)C(=O)Nc2cc(ccc2F)C(F)(F)F)C(=O)Nc3cc(ccc3F)C(F)(F)F HTS04281 c1ccc(c(c1)N2CCOCC2)OC(=O)C3=Cc4cc(ccc4OC3)Cl HTS06449 c1ccc(cc1)COc2ccc(cc2)NC(=O)NNc3c(cccn3)C#N HTS04945 c1ccc2c(c1)c(cs2)CSCC(=O)Nc3ccc(c(c3)Cl)F HTS05340 c1ccc(c(c1)C(=O)O)S(=O)(=O)Nc2cccnc2 HTS05521 CCc1ccnc(c1)NS(=O)(=O)c2ccc(cc2)NC(=O)C HTS05389 Cc1c(snn1)C(=O)NCc2cc(cc3c2OCOC3)F HTS03234 Cc1c(c(on1)C)C(=O)NCc2cc(cc3c2OCOC3)F HTS03235 CCCc1cnc(nc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)C(C)C HTS03945 c1ccc(c(c1)NC(=O)Nc2cccc(c2)Cl)N3CCOCC3 HTS06778 CC(=O)c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc4c(c3)OCCO4 HTS06811 c1ccc2c(c1)cc([nH]2)C(=O)O CC12801 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cccs3 HTS04572 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04034 c1cc2c(c(c1)S(=O)(=O)Nc3ccc(cc3)n4c(cc(n4)C(F)(F)F)c5cccs5)non2 HTS04042 c1ccc(cc1)NC(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04045 Cc1c(c(no1)c2ccccc2)C(=O)NNc3cc(cc(c3)Cl)Cl HTS06459 CC(C)(C)c1ccc(cc1)NNC(=O)c2c(cccc2Cl)F HTS06465 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 HTS07124 CCCc1cnc(nc1)N2CCN(CC2)c3ncc(cn3)CCC HTS03946 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cc(nn4Cc5ccccc5)C(C)(C)C HTS04578 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cccnc4Oc5ccc(cc5)Cl HTS04579 c1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F HTS03996 c1ccc(cc1)Oc2cccc(c2CNC(=O)Nc3ccc(cc3)F)Cl HTS04313 Cc1csc(c1c2nc3ccccc3s2)NC(=O)Nc4ccc(cc4)C(C)(C)C HTS04622 c1cc(ccc1C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3)OC(F)(F)F HTS03456 c1cc(sc1)c2ccc(cc2)C(=O)O CC12001 Cc1ccc(cc1)S(=O)(=O)Nc2c(n(n(c2=O)c3ccccc3)C)C HTS06071 CC(C)(C)c1ccc(cc1)C(=O)NNc2ccc(cc2F)F HTS06153 CCCc1cnc(nc1)N2CCN(CC2)C(=S)NC HTS03954 Cn1c(nnc1Sc2nc3ccc(cc3s2)Cl)c4ccc5c(c4)cccn5 HTS03448 Cc1c(snn1)C(=O)Nc2ccccc2N3CCOCC3 HTS07069 Cn1cc(nc1)S(=O)(=O)Oc2ccccc2N3CCCCC3 HTS06187 c1ccc(c(c1)N2CCCCC2)OC(=O)C3CCN(CC3)c4nccc(n4)C(F)(F)F HTS06195 c1ccc2c(c1)ccc(n2)NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS05967 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3cscc3C#Cc4ccccc4)C(=O)OC HTS04349 CC(C)(C)c1ccc(cc1)NC(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F HTS04631 CC(C)(CC(=O)N1CCN(CC1)c2ccccn2)CC(=O)O HTS06068 c1cc(ccc1NC(=O)COc2c3ccc(cc3ncn2)Cl)OC(F)(F)F HTS06417 c1cc(c(cc1F)F)NNC(=O)C2CCC2 HTS06158 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)CCCC(=O)O HTS04274 c1ccc2c(c1)cc(s2)C(=O)N3CCC(CC3)(c4ccc(cc4)Cl)O HTS01769 c1cc(ccc1NS(=O)(=O)c2ccc3c(c2)CCO3)F HTS02236 COc1ccc(cc1)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS02237 Cc1nnc(n1c2ccc3c(c2)OCCO3)Sc4nc5ccc(cc5s4)Cl HTS04022 c1cc(sc1)c2cc(nn2c3ccc(cc3)NC(=O)c4ccno4)C(F)(F)F HTS04029 c1cc(sc1)c2cc(nn2c3ccc(cc3)NC(=O)c4ccc(cc4)F)C(F)(F)F HTS04031 CS(=O)(=O)Nc1ccc2c(c1)OCCO2 HTS06023 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)S(=O)(=O)c4ccsc4C(=O)OC)[N+](=O)[O-])C HTS06025 c1cc(sc1)c2ccnc(n2)SCC(=O)c3cc(no3)c4ccc(c(c4)Cl)Cl HTS04565 Cc1cccc(c1C(=O)O)NC(=O)C2CCCCC2 HTS05563 c1cc(oc1C(=O)NCCN2CCCCC2)Oc3cc(cc(c3)Cl)Cl HTS02330 c1cc(cc(c1)NC(=O)C2=Cc3cc(ccc3OC2)Cl)C(=O)O HTS04973 c1cc(ccc1C(=O)O)NCC(=O)NCc2ccc3c(c2)OCO3 HTS05485 c1cc(sc1)c2ccnc(n2)SCC(=O)c3ccc(s3)CC(=O)O HTS04568 COC(=O)c1cscc1N2C(=O)c3c(nccn3)C2=O HTS04055 COC(=O)c1c(ccs1)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS02239 Cn1cc(nc1)S(=O)(=O)NC2CCN(CC2)Cc3c(cccc3Cl)F HTS02401 c1ccc(cc1)S(=O)(=O)N2CCC(CC2)CNS(=O)(=O)c3cccc(c3)C(F)(F)F HTS02494 c1cc(ccc1NC(=O)CC2(CCCC2)CC(=O)O)S(=O)(=O)N HTS04062 Cc1c(csc1C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3)S(=O)(=O)c4ccc(cc4)Cl HTS03172 Cc1ccc(cc1)NC2=NCC(S2)COc3ccc(cc3)OC HTS05977 c1cc(ccc1NNC(=O)c2c(ccs2)Cl)Cl HTS05648 c1ccnc(c1)N2CCN(CC2)C(=O)CCC(=O)O HTS06069 c1cc(c(c(c1)Cl)CN2CCC(CC2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F)F HTS02402 c1cc(c(cc1F)F)C(=O)NNc2c(cncc2Cl)Cl HTS03073 c1csc(c1Cl)C(=O)NNc2c(cncc2Cl)Cl HTS03074 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F)C HTS06049 c1cc(sc1)c2ccnc(n2)SCc3ccc4c(c3)non4 HTS04577 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)Nc2ccc(cc2)F HTS02341 c1ccc(c(c1)NS(=O)(=O)c2cccc3c2non3)SCc4cccc(c4F)Cl HTS02199 c1ccc(c(c1)NS(=O)(=O)c2cc(sc2Cl)Cl)SCc3cccc(c3F)Cl HTS02200 c1ccc2c(c1)c(c(s2)C(=O)NNc3ccc(cc3)Cl)Cl HTS05649 CCc1ccnc(c1)NC(=O)Nc2c(cc(cc2Br)C(C)C)Br HTS04558 Cc1cccc(c1)NNC(=O)c2cccs2 HTS05358 Cc1cccc(c1)NNC(=O)C2CCC2 HTS05360 Cc1cc(ccc1Cl)C(=O)CSc2nccc(n2)c3cccs3 HTS04564 Cc1c(c(nc(n1)SCC(=O)Nc2ccccc2)O)CC(=O)OC HTS03952 c1cc(ccc1NC(=O)c2c(nccn2)C(=O)O)S(=O)(=O)N HTS04053 c1cc2c(cc1NC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl)OCCO2 HTS04151 CCOC(=O)C1CCN(CC1)c2ccccc2CN3CCN(CC3)Cc4ccccc4 HTS04097 c1cc(c(c(c1)Cl)NNC(=O)c2c(ccs2)Cl)Cl HTS06163 COc1cc(c(cc1OC)NC(=O)c2c(nccn2)C(=O)O)C(=O)OC HTS04418 Cc1csc(c1c2nc3ccccc3s2)NC(=O)c4ccccc4C(=O)O HTS04624 c1ccc(c(c1)C(=O)NNc2c(cccn2)C#N)C(=O)O HTS04940 CCc1ccnc(c1)NC(=O)c2cccs2 HTS04560 c1cc2c(cc1NS(=O)(=O)c3cc(sc3)c4cc(on4)C(F)(F)F)OCCO2 HTS04149 Cc1cccc(c1)NNC(=O)c2ccccc2 HTS05363 c1ccc(c(c1)NC(=O)N2CCCN(CC2)c3c(cccn3)C#N)F HTS05326 Cc1ccc(cc1C)NNC(=O)c2c(ccs2)Cl HTS05365 Cc1ccc(cc1C)NNC(=O)c2c(c3ccccc3s2)Cl HTS05366 Cc1cc(c(o1)C)C(=O)N2CCC(CC2)C(=O)O HTS07096 C1CCN(CC1)C2(CCN(CC2)C(=O)CSCC(=O)O)C(=O)N HTS07117 c1cc(cc(c1)S(=O)(=O)N)NC(=O)C2CCCCC2 HTS06218 c1ccc(c(c1)C(=O)Nc2ccc(cc2)S(=O)(=O)N)C(=O)O HTS04059 Cc1cccc(n1)C2C3=C(CC(CC3=O)(C)C)NC(=C2C(=O)OC)C HTS04691 Cn1c(nnc1SCC(=O)N(c2ccccc2)C3CCCCC3)c4ccc5ccccc5c4 HTS04506 Cc1c(ccc(n1)C(F)(F)F)C(=O)Oc2ccccc2N3CCCCC3 HTS05622 Cc1c(snn1)C(=O)Oc2ccccc2N3CCCCC3 HTS05623 c1cc(c(cc1Cl)NNC(=O)C2CCC2)Cl HTS03069 Cc1ccc(c(c1)C)NNC(=O)CCc2ccccc2 HTS05038 Cc1cccc(c1)NNC(=O)c2c(cccc2Cl)F HTS05352 c1cc(ccc1C#N)NC(=O)CC2(CCCC2)CC(=O)O HTS05125 Cc1cc(c(o1)C)C(=O)NCCNS(=O)(=O)c2ccc(cc2)Cl HTS04104 Cc1ccc(cc1C)NNC(=O)CCc2ccccc2 HTS05368 Cc1c(c(no1)c2ccccc2)C(=O)NNc3c(cncc3Cl)Cl HTS03085 Cc1c(csc1C(=O)NCCSCc2ccc(cc2)[N+](=O)[O-])S(=O)(=O)c3ccc(cc3)Cl HTS03171 COc1ccc(cc1)OCC(CNC(=O)c2c(c3ccccc3s2)Cl)O HTS05092 COc1ccc(cc1)OCC(CNC(=O)c2ccc(cc2)OC(F)(F)F)O HTS05093 COc1cc(c(cn1)C(=O)NCc2ccc(cc2Cl)Cl)C(F)(F)F RF04358 CC(C)(C)c1ccc(cc1)NC(=O)Oc2ccccc2N3CCOCC3 HTS05640 c1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)Cc4ccc5c(c4)OCO5 HTS05671 Cc1cccc(c1)NNC(=O)CCc2ccccc2 HTS05353 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3cccc(c3)S(=O)(=O)N HTS06219 c1ccc(cc1)COc2ccc(cc2)NC(=O)Oc3ccccc3N4CCCCC4 HTS05638 CCc1ccc(cc1)C(=O)NNc2ccc(c(c2)C)C HTS05522 Cc1ccc(cc1C)NNC(=O)c2ccc(cc2)C(C)(C)C HTS05523 Cc1ccc(cc1C)NNC(=O)c2cc(on2)C HTS05524 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc4c(c3)C(=O)OC4 HTS03088 c1ccc(c(c1)C(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl)C(=O)O HTS05257 Cn1cc(c(cc1=O)C(F)(F)F)C(=O)N(C)c2ccc(c(c2)Cl)Cl RF04781 c1ccc(cc1)Oc2cc(c(cn2)c3ncc(o3)c4ccc(cc4)Cl)C(F)(F)F RF04799 c1cc(ccc1c2cnc(o2)c3cnc(cc3C(F)(F)F)Oc4ccc(cc4)Cl)Cl RF04800 CCS(=O)(=O)c1ccc(c(c1)NC(=O)CC(C)(C)CC(=O)O)O HTS04066 CCS(=O)(=O)c1ccc(c(c1)NC(=O)CC2(CCCC2)CC(=O)O)O HTS04071 CCN(CC)c1ccc(cc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS03958 c1ccc(c(c1)C(=O)NNc2ccc(cc2)S(=O)(=O)N)C(=O)O HTS04424 Cc1cc(cc(c1)NC(=O)Oc2ccccc2N3CCCCC3)C HTS06183 CC1(CCc2cc(ccc2O1)CN3CCC(CC3)c4ccccc4OC)C HTS05403 c1ccc(cc1)NCN2C(=O)C3=C(C2=O)CCCC3 HTS05600 CC(C)(CC(=O)Nc1cccc(c1)C(=O)O)CC(=O)O HTS04979 c1c(c(c(cn1)Cl)N2CCC(CC2)C(=O)N)Cl HTS04183 Cc1cc(no1)NC(=O)c2cc(oc2C)C(C)(C)C HTS04662 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3 HTS04674 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2)C(F)(F)F HTS04675 Cn1cc(nc1)S(=O)(=O)Nc2ccc3c(c2)C(=O)OC3 HTS03393 Cn1c(ccc1S(=O)(=O)Nc2ccc3c(c2)C(=O)OC3)C(=O)OC HTS03396 c1ccc(c(c1)C(F)(F)F)NNC(=O)c2ccc(cc2F)F HTS03398 c1ccc(cc1)CC(=O)Nc2cccc(c2)C(=O)O HTS04970 Cc1c(snn1)C(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl HTS05268 COc1cccc(c1C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl)OC RF04813 COc1cccc(c1)C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl RF04832 CC1(OCCO1)C2(OCCO2)C RF04844 c1ccc(c(c1)c2nn(c(=O)o2)c3c(cccn3)C(F)(F)F)Cl RF04894 c1ccc2c(c1)/C(=C/c3c[nH]c4c3cc(cc4)[N+](=O)[O-])/C(=O)N2 HTS05065 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)Nc3ccc4c(c3)OCCO4 HTS03216 Cn1c2cccc(c2c(n1)NC(=O)c3ccc(cc3)Cl)N(C)C HTS06728 Cc1c(cc(o1)C(C)(C)C)C(=O)NCc2ccc(c(c2)OC)OC HTS04669 c1ccc(cc1)C(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 HTS06957 c1cc(oc1)C(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 HTS06958 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2F)F HTS04671 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)C HTS05877 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3cccs3 HTS05878 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(cc3)F HTS06600 COc1ccccc1C(=O)NNc2ccc(cn2)C(F)(F)F RF04855 c1cc(c(c(c1)F)C(=O)NNc2c(cccn2)C(F)(F)F)F RF04876 c1cc(c(cc1Cl)Cl)c2c[nH]nc2C(=O)NN RF05002 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS06793 Cn1c2cccc(c2c(n1)NC(=O)c3ccc(cc3)F)N(C)C HTS06729 CCOC(=O)C1CCCN(C1)S(=O)(=O)c2c(noc2C)C HTS05781 CCOC(=O)C1CCCN(C1)S(=O)(=O)c2ccc(n2C)C(=O)OC HTS05783 c1ccc(cc1)NC(=O)Nc2ccc3c(c2)OCCO3 HTS06001 CC(C)C(=O)NNc1c(cccn1)C(F)(F)F RF04899 Cn1cc(nc1)S(=O)(=O)Nc2c3c(cccc3N(C)C)n(n2)C HTS06740 c1cc(ccc1c2cn3c(n2)SCC3)NC(=O)C4CC4 HTS06791 Cc1c(snn1)C(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS06792 CC(C)C(=O)NNc1cc(ccn1)C(F)(F)F RF04961 COc1ccc(cc1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccccc3 HTS05044 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccccc2N3CCOCC3 HTS06777 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2)C(C)C HTS04672 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2)F HTS04676 COc1ccc(cc1)OCC(CNC(=O)c2cccnc2Oc3ccc(cc3)Cl)O HTS05089 Cc1cnc(c(n1)C)NC(=O)c2c(nccn2)C(=O)O HTS03726 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OCC(=O)Nc3ccc4c(c3)OCCO4 HTS06815 Cc1cc(cc(c1CNC(=O)C(C)C)Cl)Cl RF05048 CCSc1c(c(ccn1)C(F)(F)F)C(=O)NCc2ccc(cc2Cl)Cl RF05077 Cc1ccc(cc1)NC(=O)N(CCC#N)Cc2ccccc2 HTS05335 CCOc1ccccc1N2CCN(CC2)Cc3c[nH]nc3c4ccc(cc4)F HTS05427 CC(=O)c1ccc(cc1)NC(=O)CSc2nnc(n2C)c3ccc4ccccc4c3 HTS04507 COc1ccc(cc1)SCCc2nnc(n2C3CC3)SCC(=O)Nc4ccccc4 HTS04508 CC(C)N1CCC(=O)N(C1=O)c2ccccc2 HTS06118 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3cc(ccc3Cl)Cl HTS03071 c1cc(c(cc1Cl)NNC(=O)c2c(ccs2)Br)Cl HTS03072 c1ccc2c(c1)c(c[nH]2)CN3CCN(CC3)c4ccccn4 HTS06140 c1cc(cc(c1)Cl)C2=NC(=O)C(S2)CC(=O)O HTS04922 c1ccc2c(c1)CCNC2CC(=O)O HTS07006 Cc1cccc(n1)NC(=O)c2cccs2 HTS07031 Cc1cccc(n1)NC(=O)c2ccco2 HTS07032 CCOC(=O)N1CCC(CC1)NC(=O)c2ccccc2C(=O)O HTS05189 Cc1cccc2c1c(=O)oc(n2)c3cccnc3Oc4ccccc4 HTS05572 COc1ccc(c(c1)NC(=O)Nc2ccccc2N3CCOCC3)Cl HTS06779 Cc1cc(c(o1)C)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS04095 CCc1ccnc(c1)NC(=O)c2c(nns2)C HTS04807 c1cc2c(cc1NC(=O)Nc3ccc4c(c3)OCCO4)OCCO2 HTS06003 c1cc(ccc1NC(=O)Nc2ccc3c(c2)OCCO3)OC(F)(F)F HTS06005 Cc1c(cnn1c2ccc(cc2)OC)C(=O)N3CCOCC3 HTS06082 CCC(C)(C)C1CCc2c(sc(c2C#N)N)C1 HTS05438 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)F)c3ccc4ccccc4c3 HTS04509 Cc1c(c(no1)c2ccccc2)C(=O)NCc3c(cccc3Cl)Sc4ccc(cc4)Cl HTS05270 CCS(=O)(=O)c1ccc(c(c1)NC(=O)CSCC(=O)O)O HTS04070 Cc1ccsc1CNC(=O)Nc2cc(oc2C(F)(F)F)C HTS04295 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)Nc4c(cc(cc4Br)C(C)C)Br HTS03112 c1c(c(sc1Cl)Cl)C(=O)Nc2nnc(s2)C3CC3 HTS03421 c1cc(c(nc1)NNC(=O)CCC(=O)O)C#N HTS04939 COc1ccc(cc1)OCC(CNC(=O)c2ccccc2)O HTS05079 Cc1ccc(cc1)C(=O)NCC(COc2ccc(cc2)OC)O HTS05080 Cc1cccc2c1c(=O)oc(n2)c3ccccc3 HTS05574 Cc1cccc2c1c(=O)oc(n2)c3cc4ccccc4s3 HTS05573 CCOC(=O)c1c(cccc1NC(=O)c2cccs2)C HTS05576 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2c(c(nn2C)C(F)(F)F)c3ccccc3 HTS04794 c1ccc(cc1)C(CC(=O)O)CC(=O)Oc2ccccc2N3CCCCC3 HTS05617 CCOC(=O)c1cc(ccc1N2CCCCC2)NS(=O)(=O)c3cccc4c3non4 HTS04639 CCS(=O)(=O)c1ccc(c(c1)NC(=O)CCCC(=O)O)O HTS04067 Cc1ccc(cc1)S(=O)(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl HTS05261 CC(C)(C)c1ccc(cc1)NC(=O)N(CCC#N)CCc2ccccn2 HTS06106 c1ccc2c(c1)cc(s2)C(=O)NNc3c(cncc3Cl)Cl HTS03075 Cc1nc(cn1CC(c2ccc3c(c2)OCO3)O)[N+](=O)[O-] HTS02333 Cc1cnc(cn1)C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS02398 Cc1c(cnn1c2ccc(cc2)OC)C(=O)N3CCN(CC3)Cc4ccccc4 HTS06085 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2cc(c(cc2C(=O)OC)OC)OC HTS04673 Cc1c(cnn1c2ccc(cc2)OC)C(=O)NCc3ccc4c(c3)OCO4 HTS04305 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccc(cc3)S(=O)(=O)N HTS04488 c1cc(oc1)C(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS06788 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4c(c(cs4)S(=O)(=O)c5ccc(cc5)Cl)C HTS04582 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)C4CCC4 HTS04584 c1ccc(c(c1)C(=O)O)SCC(=O)NCc2ccc3c(c2)OCO3 HTS05470 Cc1ccc2c(c1)oc(=O)n2CC(=O)c3ccccc3 HTS04192 Cc1ccc(cc1Cl)NC(=O)N2CCN(CC2)c3c(cccn3)C#N HTS04988 c1ccc(c(c1)C(F)(F)F)NNC(=O)c2c(ccs2)Cl HTS03399 Cc1nc(cs1)c2ccc(cc2)NC(=O)COCC(=O)O HTS03131 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])NC(=O)c3ccc(cc3)F HTS04898 c1cc(ccc1n2ccc(=O)c(n2)c3ccnc(n3)N)Cl HTS03670 CCOC(=O)C1CCN(CC1)C(=O)c2c(nc(s2)c3ccc4c(c3)CCO4)C HTS06690 Cc1cc(n(n1)C)NC(=O)Nc2ccccc2OC HTS04326 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4c(onc4c5ccccc5)C HTS04580 c1ccc(cc1)CCC(=O)NNc2c(cncc2Cl)Cl HTS03077 Cc1ccc(cc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS04502 Cc1ccc(cc1Cl)NC(=O)Nc2cccc(n2)C HTS07027 Cc1c(cc(o1)C(C)(C)C)C(=O)NCc2ccc3c(c2)OCO3 HTS04677 CN(c1ccc(cc1C(=O)c2ccccc2)Cl)C(=O)c3ccccc3C(F)(F)F HTS04290 c1cc(ccc1F)S(=O)(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl HTS05003 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)Nc2cccc3c2cccc3 HTS04604 Cc1c(csc1C(=O)N2CCC(CC2)c3ccccc3OC)S(=O)(=O)c4ccc(cc4)Cl HTS03173 Cc1c(csc1C(=O)N2CCC(CC2)C(=O)c3ccc(cc3)F)S(=O)(=O)c4ccc(cc4)Cl HTS03174 c1ccc2c(c1)c(c[nH]2)CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl HTS04862 COc1ccc2c(c1)CCCN2Cc3c[nH]c4c3cccc4 HTS04864 Cc1cccc(n1)NC(=O)c2ccccc2 HTS07033 c1cc(ccc1c2nc(on2)C(=O)NNC(=O)c3ccc(cc3)Cl)OC(F)(F)F SPB03265 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cc(on4)C HTS04585 Cc1ccc(cc1)S(=O)(=O)CCSc2nccc(n2)c3cccs3 HTS04958 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OCC(=O)Nc3ccc(cc3)F HTS06813 Cc1ccc(cc1C)NNC(=O)c2cccs2 HTS05526 Cc1cc(c(o1)C(F)(F)F)C(=O)N2CCC(CC2)C(=O)O HTS07095 c1ccc(cc1)C(=O)NCC(COc2ccc(cc2)[N+](=O)[O-])O HTS07139 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)N3CCCN(CC3)c4c(cncc4Cl)Cl HTS04998 CCOc1ccccc1NC(=O)N2CCCN(CC2)c3c(cccn3)C#N HTS05331 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3c(nccn3)C(=O)O)C HTS07040 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)CCCC(=O)O)C HTS07043 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)c4ccc(cc4)F HTS05801 CCc1ccccc1NNC(=O)c2ccccc2 HTS04763 CCOC(=O)CS(=O)(=O)c1ccc(cn1)C(F)(F)F BTB07932 CC(C)(C)c1cc(n(n1)C)C(=O)NN2CCOCC2 HTS03357 CC1(CC2=C(C(C(=C(N2)N)C#N)c3ccco3)C(=O)C1)C HTS05054 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSc4ccc(cc4)F)C(F)(F)F HTS05062 CN(C)c1ccc(cc1)N2C(=O)CC(CC2=O)c3ccccc3 HTS07057 Cc1cc(cc(c1)N2C(=O)CCN(C2=O)Cc3ccccc3)C HTS05903 CSc1c(c(n[nH]1)c2ccc(cc2)Cl)SC(=O)c3c(cccc3F)F RF05142 CCN(c1ccc(cc1Cl)Cl)C(=O)c2cnccc2C(F)(F)F RF03981 COc1ccc(cc1)OCC(CNC(=O)Nc2ccc(cc2)OC(F)(F)F)O HTS05099 COc1ccc(cc1)OCC(CNC(=O)Nc2ccccc2)O HTS05282 Cc1ccc(cc1)C(=O)Nc2ccc3ccccc3n2 HTS05483 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)Nc3ccccc3N4CCOCC4 HTS07071 c1ccc(c(c1)NS(=O)(=O)c2cccs2)N3CCOCC3 HTS07074 CC(C)(C)c1csc(n1)c2ccc(cc2)Cc3cc(n[nH]c3=O)c4ccc(cc4)F HTS03959 c1ccc(c(c1)C(F)(F)F)NC(=O)CSc2nccc(n2)c3cccs3 HTS04574 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)S(=O)(=O)C)[N+](=O)[O-])C HTS06026 c1cc(ccc1NNC(=O)c2ccc(cc2F)F)F HTS04764 c1ccc(cc1)C(CNC(=O)CC2(CCCC2)CC(=O)O)O HTS05973 c1ccc(cc1)C(CNC(=O)c2ccccc2C(=O)O)O HTS05974 COc1ccc(cc1)OCC(CNS(=O)(=O)c2cccs2)O HTS05707 COc1ccccc1CC(=O)Nc2ccc3ccccc3n2 HTS06287 c1ccc(c(c1)C(=O)c2cc(ccc2NC(=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)Cl)Cl HTS05714 Cc1c(snn1)C(=O)NNC(=O)c2cccc3c2cccc3 HTS07093 Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc4ccccc4n3 HTS06289 c1ccc(c(c1)NS(=O)(=O)c2ccc3c(c2)OCC3)N4CCOCC4 HTS07075 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2N3CCOCC3 HTS07077 C#CC1CCCCC1NC(=O)Nc2cnccc2C(F)(F)F RF04024 c1cc(c(nc1)N2CCOCC2)NC(=O)c3cccs3 HTS03349 COc1ccc(cc1OC)C(=O)Nc2cccnc2N3CCOCC3 HTS03353 c1cc(ccc1NC(=O)COc2c3ccc(cc3ncn2)Cl)Cl HTS06414 Cc1c(snn1)C(=O)NNc2ccc(cc2)F HTS05012 CC(C)(C)c1ccc(cc1)NC(=O)NNc2c(cccn2)C#N HTS04942 CC(C)(C)c1ccc(cc1)NC(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl HTS05255 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccc(cc3)N(C)C HTS04526 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccccc3 HTS04527 c1ccc2c(c1)cc(o2)C(=O)CSc3nccc(n3)c4cccs4 HTS04576 CCN(CC)c1ccc(cc1)NC(=O)c2ccccc2C(=O)O HTS03920 c1cc2c(c(c1)S(=O)(=O)N3CCCN(CC3)c4nccc(n4)C(F)(F)F)non2 HTS03997 c1cc(ccc1NC(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F)F HTS04000 c1ccc(cc1)C(CC(=O)Nc2ccc3ccccc3n2)CC(=O)O HTS06058 c1cc(cc(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)C(=O)O HTS04975 c1ccc(c(c1)N2CCCCC2)OS(=O)(=O)c3ccc(s3)c4ccccn4 HTS05712 CCc1ccnc(c1)NC(=O)Nc2cc(cc(c2)C)C HTS04811 COC(=O)c1c(=O)ccn(n1)c2ccc(cc2)F SPB04004 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccn[nH]3 SPB04969 c1ccc(cc1)COC(=O)N2c3ccccc3CC2CO CC13409 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)c4ccncc4 HTS05767 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccncc3)C(=O)O HTS05769 c1ccc(c(c1)NS(=O)(=O)c2cc(sc2Cl)Cl)N3CCOCC3 HTS07078 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)Nc2ccccc2N3CCOCC3 HTS07080 c1cc(cc(c1)NC(=O)COc2c3ccc(cc3ncn2)Cl)C(F)(F)F HTS06415 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccccn3 HTS06596 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3cccc4c3non4 HTS06597 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)CC#N HTS04740 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)CC#N)C HTS05104 c1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl HTS05672 CC(C)(C)c1cc(no1)C(=O)NN SPB03153 CC(C)(C)c1ccc(cc1)C(=O)NNc2ccc(cc2)C(C)(C)C HTS06468 Cc1cc(no1)C(=O)NNc2ccc(cc2)C(C)(C)C HTS06469 Cc1cc(cc(c1)NC(=O)NCC(c2ccccc2)O)C HTS05725 CCCCNC(=O)Nc1cc(nn1C)C(C)(C)C HTS04374 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OCC(=O)Nc3cccc(c3)C#N HTS06814 Cc1cccc(n1)NC(=O)c2ccc(cc2)Cl HTS07034 c1cc(sc1)c2nc(cs2)CO CC11509 c1cc(sc1)c2ccnc(n2)SCCS(=O)(=O)c3ccc(cc3Cl)Cl HTS04960 CCc1ccnc(c1)NS(=O)(=O)c2ccc3c(c2)OCCCO3 HTS05586 c1ccc(cc1)OCc2ccc(cc2)NC(=O)Nc3cccc(c3)C(=O)O HTS04977 Cn1cc(nc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)F HTS05814 Cc1c(c(n(n1)C)c2nc(no2)c3ccc(cc3)C(F)(F)F)[N+](=O)[O-] SPB01800 c1ccc(c(c1)N2CCCCC2)OC(=O)c3ccco3 HTS05620 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)C(=O)N(C)C)[N+](=O)[O-])C HTS04916 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)CC3(CCCC3)CC(=O)O)C HTS07042 Cc1ccc(cc1)S(=O)(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F HTS03995 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCCN(CC3)c4nccc(n4)C(F)(F)F HTS03999 c1ccc(cc1)CN(CCC#N)C(=O)c2ccc(cc2)Cl HTS06378 Cc1ccc(cc1Cl)NC(=O)Oc2ccccc2N3CCOCC3 HTS06432 Cc1c(c(n[nH]1)C)c2ccccc2C(=O)O CC15701 c1ccc(c(c1)C(=O)NNC(=O)c2ccc(cc2)OC(F)(F)F)Cl SPB03441 COC(=O)c1cnn(c1/C=N/O)c2ccccc2 SPB05287 Cc1ccc(cc1)NC(=O)c2c(n3c(s2)nc(n3)c4ccc(cc4)Cl)C SPB05411 CCOC(=O)NNC(=S)Nc1cccc(c1)Cl SPB00519 CS(=O)(=O)Nc1ccc(cc1)c2cn3c(n2)SCC3 HTS05745 COc1ccc(cc1)NNC(=O)C2CCC2 HTS04745 Cc1c2cc(ccc2sc1S(=O)(=O)NNC(=O)CCSc3ccc(cc3)OC)Cl HTS05876 Cc1cccc(n1)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS07025 CCCc1cnc(nc1)N2CCN(CC2)C(=O)c3c(onc3c4ccccc4)C HTS05871 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4ccc5c(c4)CCO5 HTS03019 c1ccc2c(c1)cnn(c2=O)CCOC(=O)Nc3ccc(cc3)OC(F)(F)F HTS03341 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)C(=O)c4c(nns4)C)[N+](=O)[O-])C HTS04920 CCc1ccnc(c1)NC(=O)NS(=O)(=O)c2ccc(cc2)C HTS04555 Cc1cc(c(o1)C)C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3 HTS04344 CC(C)(C)c1ccc(cc1)NC(=O)NCc2c(cccc2Cl)Oc3ccccc3 HTS04314 CC(C)(C)c1ccc(cc1)NC(=O)Nc2cccc(c2)C(=O)O HTS04974 CC(C)(C)c1ccc(cc1)C(=O)OCCN(C)c2nc3cc(ccc3s2)Cl TG00096 CCCCNc1nc2cccnc2s1 TG00182 CC(C)Nc1nc2cccnc2s1 TG00183 c1ccc(c(c1)N2CCOCC2)OC(=O)Nc3ccc(cc3)F HTS06433 c1ccc(c(c1)N2CCOCC2)OC(=O)c3cccnc3Sc4ccc(cc4)Cl HTS06448 CCOC(=O)c1c(csc1N)c2ccc(cc2)Br CC00243 CC1c2cnc(nc2-c3cc(ccc3S1)Cl)n4cccc4 HTS05748 c1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS05742 c1cc(ccc1c2cn3c(n2)SCC3)NC(=O)c4ccc(cc4)F HTS05743 CC1=C(C(C2=C(N1)CCCC2=O)c3ccccc3N4CCOCC4)C(=O)OC HTS03819 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3Cl)N(C)C)C(=O)OC HTS03840 Cc1ccc(cc1C)NNC(=O)c2c(onc2c3c(cccc3Cl)F)C HTS05530 c1cc(sc1)c2cc(nn2c3ccc(cc3)F)C(F)(F)F HTS05939 COc1ccc(cc1OC2CCCC2)NC(=O)Nc3ccc4c(c3)OCCO4 HTS06002 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3c[nH]cn3)C(=O)OC HTS04681 Cc1c(snn1)C(=O)NNc2ccc(cc2)OC HTS04741 Cn1c(nnc1SCC(=O)Nc2ccc3c(c2)OCCO3)c4ccc5ccccc5c4 HTS04503 Cn1c(nnc1Sc2nc3ccc(cc3s2)Cl)c4ccc5ccccc5c4 HTS04504 COc1ccc(cc1)NNC(=O)c2ccccc2 HTS04748 COC(=O)c1cnc(cc1C(F)(F)F)Oc2ccc(cc2)NC(=O)NC(=O)c3c(cccc3Cl)F RF04745 COc1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS05744 c1cc2c(cc1NC(=O)Nc3ccc(cc3Cl)Cl)OCCO2 HTS06004 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc3c(c2)OCCO3 HTS06006 Cc1ccc(cc1NC(=O)Nc2cc(nn2C)C)F HTS04327 Cc1cc(n(n1)C)NC(=O)c2cc(oc2C)C HTS04334 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)NCc3ccc4c(c3)OCO4 HTS04682 c1c(cc(cc1Cl)Cl)OCc2nc(cs2)C(=O)NN SPB02120 c1cc2c(cc1Cl)c(cs2)CNC(=O)CSCC(=O)O HTS03892 CCCc1c(cnn1c2ccccc2)C(=O)NNc3ccc(cc3)C HTS05540 Cc1nc(cn1CC(c2ccc3c(c2)OCCO3)O)[N+](=O)[O-] HTS02332 CCCCc1ccc(cc1)NC(=O)NCCN2CCNC2=O HTS02807 c1ccc2c(c1)c(c[nH]2)CN3CCN(CC3)c4ccc(cc4)F HTS06141 CCc1ccc(cc1)C(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl HTS05269 COc1cc(cc(c1)OC)C(=O)O AC11546 c1cc(ccc1NNC(=O)c2c(nccn2)C(=O)O)S(=O)(=O)N HTS04420 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)COCC(=O)O HTS03113 c1cc(cc(c1)Cl)NC(=O)Nc2nc(no2)c3ccc(cc3)OC(F)(F)F SPB03290 COc1ccc(cc1)NC(=S)NNC(=O)c2ccc(cc2)OC(F)(F)F SPB03790 COC(=O)c1ccc(c(c1)CSc2ccccn2)O SPB04387 c1ccc(cc1)n2c3cnn(c(=O)c3cn2)c4ccccc4 SPB05288 Cc1cccc(c1)NNC(=O)c2c(nns2)C HTS05357 c1cc(c(nc1)NNC(=O)c2c(nccn2)C(=O)O)C#N HTS04937 COc1ccc(cc1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3)F HTS02425 Cn1cc(nc1)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS04169 Cc1cc(c(o1)C(F)(F)F)NC(=O)Nc2ccc3c(c2)OCCO3 HTS06007 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccc(cc3)S(=O)(=O)N HTS04487 Cc1cc(no1)c2c(c(no2)C)C(=O)O/N=C(/c3cccc(c3)C(F)(F)F)\N SPB03267 COc1ccc(cc1OC2CCCC2)NC(=O)Nc3nnc(s3)C4CC4 HTS03428 Cc1c(c(no1)c2ccccc2)C(=O)Nc3nnc(s3)C4CC4 HTS03423 c1ccc(c(c1)NC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F)N4CCOCC4 HTS07061 c1ccc2c(c1)c(c[nH]2)CN3CCN(CC3)c4cc(ccn4)C(F)(F)F HTS06143 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccc(n2)C HTS07026 c1ccc2c(c1)cccc2NC(=O)Nc3ccccc3N4CCOCC4 HTS07054 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NS(=O)(=O)C HTS00352 c1ccc(c(c1)C(=O)NCCN2CCNC2=O)NC(=O)Nc3ccc(cc3F)F HTS06736 c1ccc(cc1)c2cnc(o2)c3cnccc3C(F)(F)F RF04092 Cc1cccc(c1)NNC(=O)c2ccc(cc2F)F HTS05349 c1ccc(c(c1)N2CCCCC2)OS(=O)(=O)c3cccc4c3non4 HTS05625 c1ccc(c(c1)NC(=O)Cn2c3c(cccn3)oc2=O)Oc4ccc(cc4Cl)Cl HTS04469 c1cc(ccc1n2ccc(=O)c(n2)c3ccnc(n3)N)F HTS03669 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccccc3N4CCOCC4)Cl HTS07059 c1ccc(cc1)C(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F HTS04634 c1cnc(nc1C(F)(F)F)N2CCCN(CC2)C(=O)c3c(ccs3)Cl HTS04635 CN(C)c1ccc(cc1)C(=O)Nc2ccccc2N3CCOCC3 HTS07060 c1ccc2c(c1)c(c[nH]2)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS04861 CCOC(=O)c1cc(ccc1N2CCCCC2)NS(=O)(=O)c3ccccc3 HTS04638 COc1ccc(cc1)OCC(CNS(=O)(=O)c2ccccc2)O HTS05290 CC(C)(CC(=O)Nc1ccc2ccccc2n1)CC(=O)O HTS05611 c1ccc(c(c1)C(F)(F)F)NC(=O)c2c(nccn2)C(=O)O HTS03314 Cc1c2c(nc(nc2sc1C(=O)c3ccccc3)c4ccc(cc4)Cl)C SPB05343 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3c(cccc3Cl)Cl HTS06175 Cc1ccc(cc1NC(=O)C2CCCCC2)S(=O)(=O)N(C)C HTS06216 c1ccc2c(c1)cccc2NC(=O)NNc3c(cccn3)C#N HTS04943 Cc1ccc(cc1NC(=O)c2cccnc2Sc3ccccc3)S(=O)(=O)N(C)C HTS06220 c1cc(sc1)S(=O)(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 HTS07121 c1ccc(cc1)C(=O)Nc2ccc(cc2)C#N HTS05127 c1cc(sc1)C(=O)Nc2ccc(cc2)C#N HTS05128 c1cc(oc1)C(=O)Nc2ccc(cc2)C#N HTS05129 Cc1c(c(no1)c2ccccc2)C(=O)NCC(COc3ccc(cc3)OC)O HTS05091 c1ccc(cc1)C(=O)NCCN2CCN(CC2)c3nccc(n3)C(F)(F)F HTS03016 CCN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)OCC RF04306 CC(=O)Nc1ccc(cc1)c2cn3c(n2)SCC3 HTS06790 c1cc(ccc1c2cn3c(n2)SCC3)NC(=O)c4ccc5c(c4)non5 HTS06794 c1ccc2c(c1)CCCC2NC(=O)CCCC(=O)O HTS05598 c1ccc2c(c1)cccc2NC(=O)N3CCCN(CC3)c4c(cncc4Cl)Cl HTS04997 c1ccc(cc1)C(CNC(=O)Nc2ccccc2)O HTS05723 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3cccnc3 HTS04522 Cc1ccc(cc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)C HTS04524 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2c(noc2C)C HTS07104 c1ccc2c(c1)ccc(n2)NC(=O)C3CCN(CC3)c4nccc(n4)C(F)(F)F HTS06294 Cc1c(csc1C(=O)NCC(COc2ccc(cc2)OC)O)S(=O)(=O)c3ccc(cc3)Cl HTS05085 COc1ccc(cc1)OCC(CNC(=O)c2c(ccs2)Cl)O HTS05094 CN(C)c1ccc(cc1)C(=O)NCC(COc2ccc(cc2)OC)O HTS05095 Cc1[nH]cc(n1)/C=C\2/c3ccccc3NC2=O HTS05067 CCN(Cc1cc(cc(c1)Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04318 COc1cc(c(cn1)C(=O)NCc2cccc(c2)Cl)C(F)(F)F RF04332 COc1cccc(c1)CNC(=O)c2cnc(cc2C(F)(F)F)OC RF04342 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl HTS04993 CCc1ccc(cc1)C(=O)NNc2cccc(c2)C HTS05354 Cc1ccc(cc1C)NNC(=O)c2c(onc2c3ccccc3)C HTS05529 CCCc1ccc(cc1)C(=O)NNc2cccc(c2)C HTS05355 c1cc2c(cc1S(=O)(=O)N3CCC(CC3)(C(=O)N)N4CCCCC4)OCC2 HTS07122 Cc1c(c(on1)C)S(=O)(=O)N2CCC(CC2)(C(=O)N)N3CCCCC3 HTS07123 c1ccc(cc1)Sc2c(cccn2)C(=O)Nc3cccc(c3)S(=O)(=O)N HTS06222 c1cc(ccc1N2CCN(CC2)C(=O)CSCC(=O)O)F HTS05796 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NCc3cc(cc4c3OCOC4)F HTS04161 COc1cc(ccc1CN2CCN(CC2)Cc3ccc4c(c3)OCO4)OCc5ccccc5 HTS05157 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc4ccccc4n3 HTS06279 c1ccc(c(c1)NC(=O)NNc2c(cccn2)C#N)F HTS04944 Cc1cc(cc(c1)NC(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl)C HTS04991 Cc1c(cccc1Cl)NC(=O)Nc2cc(nn2C)C(C)(C)C HTS04376 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS06787 Cc1ccc(cc1C)C(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS06789 Cc1c(cc(o1)C(C)(C)C)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 HTS04661 Cc1ccc(cc1NC(=O)c2cc(nn2Cc3ccccc3)C(C)(C)C)S(=O)(=O)N(C)C HTS06224 Cc1ccc(cc1NC(=O)c2c(onc2c3c(cccc3Cl)F)C)S(=O)(=O)N(C)C HTS06227 Cc1c(c2ccccc2[nH]1)/C=C\3/c4ccccc4NC3=O HTS05069 c1ccc2c(c1)c(c(s2)C(=O)NNc3ccc(cc3)F)Cl HTS04766 Cc1c(cnn1c2ccc(cc2)OC)C(=O)NCc3c(cccc3Cl)Sc4ccc(cc4)Cl HTS05267 c1ccc(cc1)CN2CCN(CC2)Cc3c[nH]nc3c4ccccc4 HTS05674 c1ccc(cc1)CN(CCC#N)C(=O)c2ccccc2 HTS06377 c1ccc(cc1)C(CNC(=O)Nc2cccc(c2)C(F)(F)F)O HTS05726 c1cc2c(cc1c3nc(cs3)C(=O)N4CCC(CC4)C(=O)O)CCO2 HTS06678 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(s3)c4cccs4)C(=O)OC HTS04323 CCOC(=O)N1CCC(CC1)NC(=O)c2c(nccn2)C(=O)O HTS05190 c1cc(cc(c1)NC(=O)CCCC(=O)O)C(=O)O HTS05072 c1ccc(c(c1)C(=O)Nc2cccc(c2)C(=O)O)C(=O)O HTS05074 c1ccc(c(c1)N2CCCCC2)OC(=O)CC3(CCCC3)CC(=O)O HTS05618 Cc1ccc(cc1C)NNC(=O)c2c(nns2)C HTS05525 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)C#N)C HTS05117 c1ccc(c(c1)C(=O)NCCN2CCNC2=O)NC(=O)Nc3ccc(cc3)C(F)(F)F HTS06743 c1ccc(cc1)Oc2ccccc2NC(=O)CN3CCC(CC3)C(=O)O HTS07141 Cc1c(snn1)C(=O)NNc2ccc(cc2)C(C)(C)C HTS06470 CCOC(=O)c1c2csc(c2c(=O)n(n1)c3ccc(cc3)OC)N HTS01528 c1ccc(cc1)Oc2ccc(o2)C(=O)O HTS06019 c1ccc(c(c1)NC(=O)N(CCC#N)CCc2ccccn2)Cl HTS06105 c1ccc2c(c1)c(c[nH]2)CN3CCN(CC3)Cc4ccc5c(c4)OCO5 HTS06142 CCc1ccnc(c1)NC(=O)CCCC(=O)O HTS04821 c1ccc(c(c1)C(=O)Nc2ccccc2SCCS(=O)(=O)c3ccc(cc3)Cl)C(=O)O HTS05792 Cc1ccc(cc1C)NNC(=O)c2ccc(cc2F)F HTS05364 Cc1ccc(cc1C)NNC(=O)c2c(cccc2Cl)F HTS05367 Cc1ccccc1NCN2C(=O)C3=C(C2=O)CCCC3 HTS05603 Cn1c(ccc1S(=O)(=O)N)C(=O)OC SP01482 c1ccc(c(c1)/C=N/c2ccccc2O)O CD03500 CCOC(=O)c1cnn(c1C(F)(F)F)c2cc(cc(c2)Cl)Cl SP01469 CCOC(=O)c1cnn(c1C(C)C)c2cc(cc(c2)Cl)Cl SP01470 Cc1ccc(cc1)C(CSc2nnc(n2C)c3ccc4ccccc4c3)O HTS06252 COc1ccc(cc1)SCCC(=O)NCc2ccncc2 HTS06254 c1ccc2c(c1)ccc(n2)NC(=O)c3ccccc3Cl HTS06283 c1ccc2c(c1)ccc(n2)NC(=O)C3CCCCC3 HTS06284 c1cc(cnc1)CCC(=O)O HTS01877 c1ccc(cc1)CNC(=O)CCn2c(=O)ccc(n2)c3ccc(cc3)F HTS02389 c1ccc2c(c1)CCCC2NS(=O)(=O)c3cccs3 HTS05610 Cc1c(cc(o1)C(C)(C)C)C(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O HTS04877 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS04884 Cc1ccc(cc1Cl)NC(=O)Nc2ccccc2C(=O)NCC3CC3 HTS04888 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)N3CCOCC3 HTS07066 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccccc2N3CCOCC3 HTS07068 c1cc(ccc1N2CCN(CC2)C(=O)CCCC(=O)O)F HTS05800 c1ccc(c(c1)NS(=O)(=O)c2ccc(c(c2)Cl)F)N3CCOCC3 HTS07201 CC(C)(C)c1ccc(cc1)NNC(=O)c2cccs2 HTS06471 Cc1c(sc(n1)c2ccccc2)C(=O)Oc3ccccc3N4CCOCC4 HTS06511 Cc1c(csc1C(=O)NN(c2ccc(cc2)OC(F)(F)F)C(=O)c3c(c(cs3)S(=O)(=O)c4ccc(cc4)Cl)C)S(=O)(=O)c5ccc(cc5)Cl HTS05659 c1ccc(cc1)c2c(c[nH]n2)CN3CCC(CC3)(c4ccc(cc4)Cl)O HTS05680 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)Nc3cc(cc(c3)Cl)Cl HTS05131 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)Nc3c(cc(cc3Cl)Cl)Cl HTS05135 CCc1ccc(cc1)NCN2C(=O)C3=C(C2=O)CCCC3 HTS05604 c1ccc2c(c1)CCCC2NC(=O)c3cccs3 HTS05605 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3c(onc3c4ccccc4)C)C HTS07047 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ccc(cc3)F)C(=O)O HTS05797 CC(C)(CC(=O)N1CCN(CC1)c2ccc(cc2)F)CC(=O)O HTS05799 Cc1ccc2nc(cn2c1)c3ccc4c(c3)OCCO4 HTS07134 c1cc(ccc1C(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F)Cl HTS04633 c1ccc2cc(ccc2c1)NC(=O)Nc3ccccc3C(=O)NCC4CC4 HTS05138 Cc1cc(=O)oc2c1ccc(c2)NS(=O)(=O)c3ccc(cc3)F HTS06545 c1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)C(=O)O CC03101 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3ccccc3N4CCOCC4 HTS07070 CCOC(=O)C1CCN(CC1)C(=O)c2cc(nn2Cc3ccc(cc3Cl)Cl)C(C)(C)C HTS07084 CCOC(=O)C1CCN(CC1)C(=O)c2cccnc2Oc3ccccc3 HTS07090 Cc1c(c2ccccc2[nH]1)CN3CCN(CC3)c4ccc(cc4)F HTS06500 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2)S(=O)(=O)N)CC(=O)O HTS06059 c1ccc2c(c1)ccc(n2)NC(=O)c3ccc(cc3)Cl HTS06277 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3)F)C HTS07050 c1ccc(cc1)C(=O)Nc2ccccc2N3CCOCC3 HTS07065 c1ccc(cc1)S(=O)(=O)Nc2ccccc2N3CCOCC3 HTS07073 Cc1c(c(on1)C)S(=O)(=O)Nc2ccccc2N3CCOCC3 HTS07076 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3cccc(c3)Cl)C HTS07234 Cc1c(sc(n1)c2cnccn2)C(=O)Nc3ccc(cc3)N4CCOCC4 HTS05750 CN(C(=O)CN1CCN(CC1)C(=O)CCSc2ccc(cc2)OC)c3ccccc3.C(=C/C(=O)O)\C(=O)O.C(=C/C(=O)O)\C(=O)O HTS06267 c1ccc2c(c1)ccc(n2)NC(=O)c3cc(sc3Cl)Cl HTS06278 CN1CCN(CC1)Cc2c[nH]nc2c3ccc(cc3)F HTS05414 CC(C)(C)c1ccc(cc1)NC(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl HTS04992 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCCN(CC3)c4c(cncc4Cl)Cl HTS04996 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)C#N HTS05113 c1cc(ccc1C#N)NC(=O)Nc2ccc(cc2)OC(F)(F)F HTS05115 c1ccc(cc1)CN(CCC#N)C(=O)c2cccs2 HTS06383 Cc1cc(cc(c1)NC(=O)Oc2ccccc2N3CCOCC3)C HTS06430 CCc1ccccc1NNC(=O)c2c(ccs2)Cl HTS04750 CCc1ccccc1NNC(=O)c2c(cccc2Cl)F HTS04752 CCc1ccccc1NNC(=O)c2c(nns2)C HTS04757 CCCc1c(cnn1c2ccccc2)C(=O)NCc3cc(cc4c3OCOC4)F HTS04152 c1cc(ccc1c2cc([nH]n2)C(F)(F)F)Cl HTS03200 Cn1cc(nc1)S(=O)(=O)Nc2ccccc2N3CCOCC3 HTS07079 CCOC(=O)C1CCN(CC1)C(=O)c2cc(ccc2Oc3ccc(cc3)OC)[N+](=O)[O-] HTS07091 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc(cc3)C#N HTS05110 c1ccc(cc1)Oc2c(c(ccn2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F RF05097 c1cc2c(cc1C3=NC(=O)C(S3)CC(=O)O)OCO2 HTS04926 CC(C)(CC(=O)NNc1c(cccn1)C#N)CC(=O)O HTS04934 c1cc(ccc1F)S(=O)(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F HTS03993 Cc1cc(=O)oc2c1ccc(c2)NC(=O)CC(CC(=O)O)c3ccccc3 HTS07016 c1cc(cc(c1)[N+](=O)[O-])C2=NNC(C2)(C(F)(F)F)O HTS03201 CCCc1ccc(cc1)C(=O)NNc2ccccc2C(F)(F)F HTS03404 COc1ccc(cc1)c2c(nn3c2[nH]c(cc3=O)C(F)(F)F)C(F)(F)F HTS01629 Cc1c(c(c(o1)C)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3)C(=O)OC HTS04103 Cc1nc(cn1C)S(=O)(=O)NCc2cc(cc3c2OCOC3)F HTS03239 c1ccc(cc1)NC(=O)Oc2ccccc2N3CCOCC3 HTS06431 c1ccc(c(c1)N2CCOCC2)OC(=O)Nc3cccc(c3)C(F)(F)F HTS06434 c1ccnc(c1)c2ccc(s2)C(=O)NC3CCS(=O)(=O)C3 HTS03272 c1ccc(cc1)NC(=O)CN2CCN(CC2)c3nc4cc(ccc4s3)Cl HTS03274 Cc1cc(cc(c1)NC(=O)Nc2nnc(s2)C3CC3)C HTS03430 Cc1ccccc1/N=N/c2c(c(c(nc2C)S)C#N)C SPB06735 Cc1c(c(nc(n1)c2ccccc2)S)C(=O)C SPB05363 COc1cc(c(cc1OC)NC(=O)CC(CC(=O)O)c2ccccc2)C(=O)O HTS06312 Cn1c(ccn1)NC(=O)c2c(nccn2)C(=O)O HTS06313 c1ccc(c(c1)C(F)(F)F)NNC(=O)c2c(ccs2)Br HTS03412 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)NCCSCc3ccc(cc3)F HTS02287 Cc1cn(c2c1cccc2)CCC(=O)NC3Cc4ccccc4C3 HTS02298 c1ccc2c(c1)c(cs2)c3csc(n3)c4ccc(s4)c5ccno5 HTS02300 c1ccnc(c1)c2ccc(s2)C(=O)Nc3ccc4c(c3)OCCO4 HTS03214 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl)C(=O)OC HTS05001 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)Nc2ccc(c(c2)Cl)C HTS04602 c1ccc(cc1)CNc2nc3cccnc3s2 TG00184 c1cc(sc1)c2nc(on2)CCC(=O)O HTS03592 Cc1ccc(cc1Cl)NC(=O)Nc2ccc3c(c2)C(=O)OC3 HTS03089 COc1ccc(cc1)OCC(CNC(=O)C2CCC2)O HTS05087 c1cc(ccc1CC#N)NC(=O)COCC(=O)O HTS04728 CC1c2cc(c(cc2CCN1C(=O)c3ccno3)OC)OC HTS04856 Cn1cnc(c1Sc2ccccc2C(=O)O)[N+](=O)[O-] HTS03326 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccccc3C(F)(F)F HTS03410 c1cc(c(cc1F)F)C(=O)NNc2cc(ccc2Cl)Cl HTS02731 c1cc2c(cc1S(=O)(=O)NC3CCS(=O)(=O)C3)CCO2 HTS02838 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)NC2CCS(=O)(=O)C2 HTS02842 CCN(c1ccc(cc1Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04389 c1ccc(cc1)Sc2cc(c(cn2)C(=O)Nc3ccc(cc3Cl)Cl)C(F)(F)F RF04397 COC(=O)c1c(ccs1)S(=O)(=O)NC2CCS(=O)(=O)C2 HTS02841 COc1ccc(cc1)OCC(CNC(=O)C2=Cc3cc(ccc3OC2)Cl)O HTS05084 Cc1cc(no1)C(=O)NCC(COc2ccc(cc2)OC)O HTS05088 Cc1nc(cs1)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)Oc4cccc(c4C#N)Cl HTS03126 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4)C(=O)O HTS01759 c1ccc(c(c1)C(=O)NCCN2CCNC2=O)N HTS05752 CCS(=O)(=O)c1ccc(c(c1)NC(=O)Nc2ccc(c(c2)Cl)C)O HTS04412 c1cc(ccc1NNC(=O)CC2(CCCC2)CC(=O)O)S(=O)(=O)N HTS04426 COc1ccc(cc1)NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS06341 c1cc(sc1)CN(CCC#N)C(=O)c2cccs2 HTS06388 CC1c2cc(c(cc2CCN1C(=O)c3c(nccn3)C(=O)O)OC)OC HTS06400 c1cc(c(cc1[N+](=O)[O-])C#N)NCC#N HTS03224 c1cnc(nc1C(F)(F)F)N2CCC(CC2)C(=O)NC3CCS(=O)(=O)C3 HTS02847 c1ccc(cc1)c2c(c[nH]n2)CN3CCc4ccccc4C3 HTS05683 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3nccc(n3)C(F)(F)F HTS04632 c1cc(cc(c1)NC(=O)c2c(nccn2)C(=O)O)C(=O)O HTS05075 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)c3c(cncc3Cl)Cl HTS04994 Cc1ccc2c(c1)CCCN2C(=O)c3c(c(cs3)S(=O)(=O)c4ccc(cc4)Cl)C HTS03175 CCOC(=O)C1=C(NC(=O)NC1C)C(C)c2ccccc2 HTS03204 CCOC(=O)C1=C(Oc2c(cc(cc2Cl)Cl)C1C(C#N)C(=O)OCC)N HTS02704 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)CC(C)(C)CC(=O)O HTS02685 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccc(o3)c4ccc(cc4)OC(F)(F)F HTS05855 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc(cc3)CC#N HTS04736 Cc1ccc(cc1Cl)NC(=O)Nc2ccc(cc2)CC#N HTS05101 COc1ccc(cc1)Oc2cccc(c2CNC(=O)Nc3ccccc3)Cl HTS05278 c1cc2c(cc1CNC(=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)OCO2 HTS05629 c1ccc(cc1)NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS05846 CC1c2cc(c(cc2CCN1C(=O)CCC(=O)O)OC)OC HTS05934 Cc1cc(n(n1)C)NC(=O)CC2(CCCC2)CC(=O)O HTS04712 CCCCc1ccc(cc1)NC(=O)Nc2ccccc2C(=O)NCC3CC3 HTS05139 CCN(c1cccc(c1C)C)C(=O)c2cnccc2C(F)(F)F RF04410 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)CSCC(=O)O HTS02700 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2ccc(cc2)Oc3cccc(c3C#N)Cl HTS02718 CC1c2cc(c(cc2CCN1C(=O)c3ccc(cc3)F)OC)OC HTS05913 Cc1c(c(no1)c2ccccc2)NC(=O)N(CCC(=O)O)Cc3ccccc3 HTS05891 CC1c2cc(c(cc2CCN1C(=O)c3cccs3)OC)OC HTS05915 c1cc2c(cc1C(=O)NCc3ccsc3)CCO2 HTS03025 Cc1ccc(cc1Cl)NC(=O)Oc2ccccc2N3CCCCC3 HTS06185 Cc1c(c(on1)C)C(=O)NNc2ccccc2C(F)(F)F HTS03405 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NC3CCS(=O)(=O)C3 HTS02845 CCOc1ccccc1N2CCN(CC2)Cc3c[nH]nc3c4ccccc4 HTS05681 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccc(s3)c4cccs4 HTS05854 c1cc(ncc1C(F)(F)F)N2CCN(CC2)C(=O)CSCC(=O)O HTS05884 Cc1ccc(cc1)NC(=O)N(CCC(=O)O)Cc2ccccc2 HTS05898 Cc1cccc(c1)Oc2c(c(ccn2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F RF05099 Cc1cc(c(nc1)NC(=O)Nc2ccc(cc2)OCc3ccccc3)Br HTS03487 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(CCC#N)Cc2ccccc2 HTS05908 CC(C)N1CCC(=O)N(C1=O)c2ccc3c(c2)CCO3 HTS06361 CC(C)N1CCC(=O)N(C1=O)c2ccc(cc2)C(C)(C)C HTS06363 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(=O)NCc4ccc5c(c4)OCO5 HTS05630 CCc1ccc(cc1)C(=O)NNc2ccccc2CC HTS04754 CCc1ccc(cc1)S(=O)(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl HTS04598 COc1ccccc1C2CCN(CC2)Cc3cccc(c3)C(=O)N4CCC(CC4)O HTS04081 c1cc2cccnc2c(c1)S(=O)(=O)NCc3csc4c3cc(cc4)Cl HTS03898 c1ccc(cc1)C(CNC(=O)Nc2ccc3c(c2)CCO3)O HTS05729 CCc1ccn2cc(nc2c1)c3ccc(c(c3)C)Cl HTS05396 CCc1ccn2cc(nc2c1)c3ccc(cc3)C HTS05397 CSc1c(c(sn1)SC)C(=O)NCc2ccc3c(c2)OCO3 HTS03580 c1cc(oc1)CNC(=O)c2ccc3c(c2)CCO3 HTS03024 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3cc(cc4c3OCOC4)F HTS02316 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)CC#N)F HTS05103 CCOc1ccccc1NC(=O)Nc2ccc(cc2)CC#N HTS05105 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccccn3 HTS04521 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)Nc3ccc(cc3)F HTS05810 Cc1ccc(cc1)c2cn3cccnc3n2 HTS04841 CC1c2cc(c(cc2CCN1C(=O)Nc3ccc(cc3)C(C)(C)C)OC)OC HTS05935 c1ccc(c(c1)C(=O)NCCN2CCNC2=O)NC(=O)Nc3ccc(cc3Cl)Cl HTS06742 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)C#N)F HTS05116 c1cc(ccc1CNC(=O)CCCO)F HTS03319 Cc1nc(c(o1)C(F)(F)F)/C(=N/OC(=O)c2ccccc2)/N RF04259 CC(C)(C#Cc1cncnc1)OC(=O)NC RF04260 c1ccc2c(c1)/C(=C/c3c[nH]nc3c4cccs4)/C(=O)N2 HTS05070 CCc1ccn2cc(nc2c1)c3cc(no3)c4ccccc4 HTS05585 CCc1ccnc(c1)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS05588 c1cc(ccc1N2C(=O)CC3(C2=O)CCCC3)[N+](=O)[O-] AW01217 c1ccn(c1)CCCNC(=O)c2c(cccc2F)F CD03933 Cc1cccc(c1)N(C(=O)c2c(c3ccccc3s2)Cl)NC(=O)c4c(c5ccccc5s4)Cl HTS05657 c1cc(ccc1C#N)NC(=O)C2CCC2 HTS05130 Cc1c(c(no1)c2ccccc2)CN3CCCCC3 HTS04316 Cc1cc(cc(c1)NC(=O)NCC(COc2ccc(cc2)OC)O)C HTS05284 c1ccc(c(c1)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4)C(=O)O HTS04831 c1ccc(cc1)CN2Cc3c([nH]c4cc(nn4c3=O)c5ccco5)C2=O HTS06827 COc1ccc(cc1)Oc2cccc(c2CNC(=O)CCCC(=O)O)Cl HTS05277 CN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04307 CCN(Cc1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)OCC RF04313 c1cc(c(c(c1)Cl)CNC(=O)Nc2ccc(cc2)F)Sc3ccc(cc3)Cl HTS05252 c1ccc(cc1)C(=O)NC2CCCc3c2cccc3 HTS05606 c1cc(ccc1c2cn3c(n2)SCC3)NS(=O)(=O)c4ccc(cc4)Cl HTS06796 c1ccc(cc1)C(CNC(=O)c2cccs2)O HTS05978 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCC(c2ccccc2)O HTS05979 c1ccc(cc1)S(=O)(=O)Oc2ccccc2N3CCCCC3 HTS05626 CCOC(=O)N1CCC(CC1)NC(=O)Nc2cc(oc2C(F)(F)F)C HTS05184 c1ccc2c(c1)ccc(n2)C(=O)O CC04401 CCOC(=O)C1CCN(CC1)C(=O)c2cc(n(n2)C(C)(C)C)C HTS07083 c1ccc(cc1)NC(=O)Nc2ccc(cc2)CC#N HTS04733 c1ccc2c(c1)cccc2NC(=O)Nc3ccc(cc3)CC#N HTS04735 CC(C)c1cc(c(c(c1)Br)NC(=O)Nc2ccc(cc2)CC#N)Br HTS04737 CCCCCc1ccc(cc1)S(=O)(=O)Nc2ccccc2C(=O)NCC3CC3 HTS05146 COc1ccccc1N2CCN(CC2)Cc3c[nH]nc3c4ccccc4 HTS05679 Cc1ccc2nc(cn2c1)c3ccc(s3)c4ccccn4 HTS07136 c1cc(oc1)c2cc3[nH]c4c(c(=O)n3n2)CN(C4=O)C5CCCCC5 HTS06829 Cc1c2ccccc2sc1CN3CCc4cc(c(cc4C3C)OC)OC HTS06961 c1ccc(c(c1)c2nnc(o2)c3cnc(cc3C(F)(F)F)Oc4ccc(cc4)Cl)Cl RF04793 COC(=O)NNc1c(cc(cn1)C(F)(F)F)Cl RF04955 c1cc(ccc1N2C(=O)CC3(C2=O)CCCC3)I AW01125 c1ccc(c(c1)C(=O)N)NC(=O)c2ccoc2 RH02133 COc1ccccc1C2CCN(CC2)Cc3c[nH]nc3c4ccccc4 HTS05676 CCc1ccc(cc1)C(=O)NNc2ccccc2F HTS05024 c1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS05677 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccc(c(c2)Cl)NC(=O)C HTS05761 Cc1cccc(c1)NNC(=O)c2c(onc2c3ccccc3)C HTS05361 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccccc3C(=O)NCC4CC4)Cl HTS05147 CCOc1ccc2c(c1)sc(n2)NC(=O)c3cc4ccccc4s3 HTS02165 c1ccc2c(c1)CCCC2NC(=O)C3=Cc4cc(ccc4OC3)Cl HTS05609 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(cc2)NC(=O)C HTS07100 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccccc2 HTS07101 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04040 c1cc(sc1)c2cc(nn2c3ccc(cc3)NS(=O)(=O)c4ccc(cc4)F)C(F)(F)F HTS04041 CC(C)(CC(=O)Nc1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)CC(=O)O HTS04047 COc1ccccc1NC(=O)Nc2ccc(cc2)CC#N HTS04739 Cc1cc(no1)C(=O)N(CCC#N)Cc2ccccc2 HTS06381 c1cc(sc1)CN(CCC#N)C(=O)c2ccc(cc2)Cl HTS06386 CC(C)c1cc(c(c(c1)Br)NC(=O)Nc2ccc(cc2)C#N)Br HTS05111 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C#N HTS05196 CS(=O)(=O)c1ccc(cc1)C(=O)Nc2ccccc2 TG00185 COC(=O)c1cnc(cc1C(F)(F)F)Oc2ccc(cc2)NC(=O)NC(=O)c3c(cccc3F)F RF04743 CN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)O RF04771 c1ccc(cc1)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS02309 CC(C)c1nn(c(=O)o1)c2cc(ccn2)C(F)(F)F RF04970 COc1c(c(ccn1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl RF05070 CCSc1c(c(ccn1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl RF05079 CCCc1ccc(cc1)C(=O)NNc2ccccc2F HTS05025 c1ccc(c(c1)NNC(=O)C2CCC2)F HTS05030 COc1ccc(cc1)c2c(nn3c2[nH]c(cc3=O)c4cccc(c4)[N+](=O)[O-])C(F)(F)F HTS01632 Cc1nc(cn1CC(=O)c2ccc(cc2)OC(F)(F)F)[N+](=O)[O-] HTS04158 CCOC(=O)Cc1csc(n1)NC(=O)c2c(nccn2)C(=O)O HTS04429 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)C#N HTS05108 Cc1c2ccccc2sc1CN3CCC(CC3)c4ccccc4OC HTS06963 Cc1cc(=O)oc2c1ccc(c2)NC(=O)CSCC(=O)O HTS07010 CCOC(=O)c1cc2c(s1)n3ccsc3n2 SPB05855 c1cc(nc(c1)C(F)(F)F)C(=O)NN SPB06723 Cc1c(c(nc(c1/N=N/c2ccccc2)C)S)C#N SPB06734 CCNc1nc2cccnc2s1 TG00181 CN(c1ccc(c(c1)Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)O RF04776 CNC(=S)NNC(=O)c1cnccc1C(F)(F)F SPB05999 c1cc(ccc1NC(=S)NNC(=O)c2cnccc2C(F)(F)F)Cl SPB06000 c1ccnc(c1)CNC(=O)c2cccc(n2)C(F)(F)F SPB06494 CNC(=S)NNC(=O)Cn1ccc(cc1=O)C(F)(F)F SPB06510 c1cc(c(nc1)N2CCCN(CC2)C(=O)Nc3cccs3)C#N HTS05332 CCCCCc1ccc(cc1)S(=O)(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl HTS04597 c1ccc(cc1)CN2CCOC(C2)C(=O)O.Cl CC12401 c1cc2c(cc1CN3CCS(=O)(=O)CC3)OCO2 HTS06440 COc1ccc(cc1)OCC(CN2CCS(=O)(=O)CC2)O HTS06443 Cn1cc(nc1)S(=O)(=O)Nc2ccc(cc2)C#N HTS05205 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc3c(c2)CCO3 HTS07105 Cc1c(nn(n1)c2ccccc2)C(=O)NC3CCS(=O)(=O)C3 HTS02849 CCOC(=O)C1CCN(CC1)c2ccccc2CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl HTS04099 COc1ccc(cc1)Oc2cccc(c2CNC(=O)Nc3ccc(cc3)OCc4ccccc4)Cl HTS05280 Cn1cnc(c1NCCN2CCNC2=O)[N+](=O)[O-] HTS03366 c1ccc(cc1)CN2CCC(CC2)NCC(=O)Nc3ccc(cc3C(=O)c4ccccc4Cl)Cl HTS05294 c1ccc(cc1)CN(CCC#N)C(=O)Nc2ccccc2 HTS05333 Cc1cc([nH]n1)NC(=O)CCCO HTS03583 c1ccc(c(c1)N2CCOCC2)OS(=O)(=O)c3cc(sc3Cl)Cl HTS06517 c1ccc(c(c1)N2CCOCC2)OS(=O)(=O)c3cccc(c3)Cl HTS06522 c1cc(c2nc(cn2c1)c3ccc(cc3)F)OCc4ccc(c(c4)Cl)Cl HTS06527 Cc1cc(=O)oc2c1ccc(c2)NC(=O)c3c(nccn3)C(=O)O HTS07012 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc3c(c2)OCCO3 HTS07106 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)c3ccccn3 HTS07107 Cc1c(cnn1c2ccc(cc2)OC)C(=O)N3CCN(CC3)c4ccccn4 HTS07143 Cn1cc(c(cc1=O)C(F)(F)F)C(=O)N(C)c2ccc(cc2)Cl RF04777 CC(C)(C)c1ccc(cc1)NC(=O)N2CCN(CC2)CCN3CCOCC3 HTS05178 Cc1c2ccccc2sc1CN3CCN(CC3)c4ccccn4 HTS06509 Cc1ccc(cc1Cl)C(=O)C(C)Sc2nnc(n2C)c3ccc4ccccc4c3 HTS04516 CS(=O)(=O)c1ccc(cc1)C(=O)Nc2ccccc2Cl TG00186 CC(C)c1ccc(cc1)Nc2nc3cccnc3s2 TG00189 c1cc(ccc1CC#N)OC(=O)c2cnccc2C(F)(F)F RF04712 c1cc(cc(c1)NC(=O)CSCC(=O)O)C(=O)O HTS04980 c1cc(cc(c1)NC(=O)COCC(=O)O)C(=O)O HTS05071 c1cc(ccc1C2=NC(=O)C(S2)CC(=O)O)Oc3ccc(cn3)C(F)(F)F HTS04925 Cc1c(c(no1)c2ccccc2)C(=O)Oc3ccccc3N4CCOCC4 HTS06447 c1ccc2c(c1)cccc2NC(=O)N3CCN(CC3)c4c(cccn4)C#N HTS04989 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)c4c(cccn4)C#N HTS04990 Cc1c2ccccc2sc1C3C4=C(CC(CC4=O)(C)C)NC(=C3C(=O)OC)C HTS04693 CC(=O)c1ccc(cc1)NC(=O)CN2CCN(CC2)c3nc4cc(ccc4s3)Cl HTS03277 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)Nc4csc5c4cccc5 HTS07213 c1ccc2c(c1)c(cs2)NC(=O)N3CCC(CC3)C(=O)N HTS12331 c1ccc2c(c1)cc(s2)C(=O)NNc3ccccc3C(F)(F)F HTS03400 c1cc(ccc1c2c(c[nH]n2)CN3CCC(CC3)C(=O)c4ccc(cc4)F)F HTS05428 c1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4ccccn4 HTS05429 Cc1cc(n(n1)C)NC(=O)c2c(nccn2)C(=O)O HTS04436 Cc1ccc(cc1)c2cn3cccc(c3n2)OCc4ccc(c(c4)Cl)Cl HTS06530 c1ccc(cc1)N(C2CCCCC2)C(=O)CN3CCN(CC3)c4nc5cc(ccc5s4)Cl HTS03276 c1cc(ccc1NC(=O)NCCN2CCNC2=O)OC(F)(F)F HTS02819 CC(C)(C)c1ccccc1NC(=O)NCCN2CCNC2=O HTS02820 COc1ccc(cc1NC(=O)NCCN2CCNC2=O)Cl HTS03361 CC(C)(C)OC(=O)C(C)(C)ONC(=O)Nc1ccc(cc1Cl)Cl RF04769 c1cc(ccc1NC(=O)N2CCN(CC2)CCN3CCOCC3)F HTS05179 c1ccc(c(c1)C(F)(F)F)NC(=O)COCC(=O)O HTS03310 CC(C)(C)c1cc(n(n1)C)C(=O)NCC(COc2ccc(cc2)OC)O HTS05083 Cc1ccc2nc(cn2c1)c3ccc(s3)c4ccccc4 HTS07271 c1cc(ccc1c2cnco2)C(=O)O CC14501 Cc1c(cc(o1)C(C)(C)C)C(=O)NC2Cc3ccccc3C2 HTS04380 c1ccc(c(c1)CC(=O)Nc2nnc(s2)C3CC3)F HTS02730 CCCNC(=O)NCCN1CCNC1=O HTS03363 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)Nc3ccccc3 HTS05808 c1ccc(c(c1)C(F)(F)F)NNC(=O)c2c(cccc2Cl)F HTS03401 c1ccc(cc1)CCC(=O)NNc2ccccc2C(F)(F)F HTS03402 Cc1cc(n(n1)C)N2C(=O)CC(CC2=O)(C)C HTS04715 c1cc(ccc1C#N)NC(=O)c2c(nccn2)C(=O)O HTS04723 Cc1cc(n(n1)C)NC(=O)CCC(=O)O HTS04713 CCCCc1ccc(cc1)S(=O)(=O)NC2CCS(=O)(=O)C2 HTS02844 CSc1cccc(c1)NC(=O)NCCN2CCNC2=O HTS03362 CCOC(=O)c1cc(ccc1N2CCCCC2)n3c(ccc3C)C HTS02680 c1ccc2c(c1)C(=O)N(C2=O)Cc3ccc(o3)/C=C\4/c5ccccc5NC4=O HTS05823 CCCc1c(cnn1c2ccccc2)C(=O)NC3Cc4ccccc4C3 HTS03520 Cc1cccc(n1)NC(=O)Nc2cccs2 HTS07030 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccncc3 HTS04523 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccc(cc3)F HTS04525 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3cccs3 HTS04528 c1ccc(c(c1)NC(=O)Nc2cccs2)N3CCOCC3 HTS07053 CCOC(=O)C1CCN(CC1)C(=O)c2cccnc2Oc3ccc(cc3)Cl HTS07092 Cc1c(cc(o1)C(C)(C)C)C(=O)Nc2ccc(cc2)N3CCOCC3 HTS04659 c1ccc(cc1)C(CNC(=O)Nc2ccc(cc2)F)O HTS05724 Cc1cc(c(o1)C(F)(F)F)NC(=O)NCC(c2ccccc2)O HTS05728 c1ccc2c(c1)/C(=C/c3c[nH]nc3c4ccc(cc4)F)/C(=O)N2 HTS05822 Cc1cc(c(nc1)NS(=O)(=O)c2cccc3c2non3)Br HTS03488 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cccc(c3)S(=O)(=O)N HTS06223 Cc1cc(c(nc1)NS(=O)(=O)c2cn(cn2)C)Br HTS03484 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)Nc3ccc(cc3)C(C)(C)C HTS05809 c1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS04091 c1ccc(cc1)C(CNC(=O)Nc2cccs2)O HTS05730 c1cc(ccc1NC(=O)N2CCN(CC2)c3ccncc3)F HTS05765 c1cc2c(c(c1)S(=O)(=O)Nc3ccc4c(c3)C(=O)OC4)non2 HTS04220 CCCc1c(cnn1c2ccccc2)C(=O)NCc3csc4c3cc(cc4)Cl HTS04226 COc1ccc(cc1)NNC(=O)c2c(c3ccccc3s2)Cl HTS04496 c1ccc(cc1)c2c(c[nH]n2)/C=C\3/c4ccccc4NC3=O HTS05824 CCCCCc1ccc(cc1)S(=O)(=O)Nc2c(cc(cn2)C)Br HTS02696 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2cccnc2N3CCOCC3 HTS03351 Cn1c(nnc1SCC(c2ccc(cc2)F)O)c3ccc4ccccc4c3 HTS06251 COc1ccc(cc1)SCCc2nnc(o2)c3ccccc3 HTS06253 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccccc3C(F)(F)F HTS03411 COc1ccc(cc1)OCC(CNC(=O)c2cccs2)O HTS05077 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCC(COc2ccc(cc2)OC)O HTS05081 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3ccc4c(c3)OCCO4 HTS03213 Cn1cc(nc1)S(=O)(=O)NCCN2CCNC2=O HTS02796 Cc1ccc(cc1NC(=O)C2CCC2)S(=O)(=O)N(C)C HTS06226 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCNC(=O)C3CC(=O)Nc4ccc(cc4)F HTS05834 COc1ccc(cc1)Oc2cccc(c2CNC(=O)c3ccccc3C(=O)O)Cl HTS05275 CC(C)(CC(=O)NCc1c(cccc1Cl)Oc2ccccc2)CC(=O)O HTS02399 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3ccc4c(c3)OCO4 HTS02888 c1ccc2c(c1)CC(C2)NC(=O)CSCC(=O)O HTS02892 c1cc2c(cc1NC(=O)Nc3ccc4c(c3)CCO4)CCO2 HTS02959 c1ccc(c(c1)NC(=O)CCCC(=O)O)SCCS(=O)(=O)c2ccc(cc2)Cl HTS05795 c1ccc(cc1)C(CNC(=O)c2ccco2)O HTS05980 COc1cc(ccc1CN2CCN(CC2)Cc3ccccc3)OCc4ccccc4 HTS04873 CCc1ccc(cc1)C(=O)NNc2cc(cc(c2)Cl)Cl HTS06452 Cc1cccc(c1C(=O)O)NC(=O)C2CCC2 HTS05562 Cc1cccc(c1C(=O)O)NC(=O)c2cccnc2Oc3ccccc3 HTS05566 c1cc(oc1C(=O)NCc2cc(cc3c2OCOC3)F)Oc4cc(cc(c4)Cl)Cl HTS02315 c1cc(c(c(c1)Oc2ccc(cc2)S(=O)(=O)NC3CCS(=O)(=O)C3)Cl)C#N HTS02843 COC(=O)c1c(ccs1)S(=O)(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS06797 CCc1ccnc(c1)NS(=O)(=O)c2ccc(cc2)C#N HTS05392 CCc1ccn2cc(nc2c1)Nc3ccccc3Cl HTS05583 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccccc3C(=O)NCCCN4CCOCC4 HTS05833 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccccc3c4[nH]c5ccccc5n4 HTS05835 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccccc2C(=O)NCC3CC3 HTS04886 COc1ccc(cc1)OCC(CNC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F)O HTS05096 CC(C)(CC(=O)NCc1c(cccc1Cl)Oc2ccc(cc2)OC)CC(=O)O HTS05276 c1cc(c(c(c1)Cl)NNC(=O)C2CCC2)Cl HTS06173 c1ccc(cc1)OCc2ccc(cc2)NC(=O)Oc3ccccc3N4CCOCC4 HTS05703 c1cc(c(nc1)N2CCCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F)C#N HTS05328 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)NCc3cc(cc4c3OCOC4)F)Cl HTS02317 c1ccc(cc1)CN2Cc3c([nH]c4cc(nn4c3=O)c5ccccc5)C2=O HTS06823 c1ccc2c(c1)CCCC2NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS05592 CC(C)(CC(=O)NCc1c(cccc1Cl)Sc2ccc(cc2)Cl)CC(=O)O HTS05259 Cn1cc(nc1)S(=O)(=O)NCC2CCN(CC2)S(=O)(=O)c3ccccc3 HTS02497 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CN4CCN(CC4)c5ccc(cn5)C(F)(F)F HTS02378 CC(=O)Nc1cccc(c1)n2nc(nn2)SCc3ccccc3 HTS02379 CC(C)(C)c1ccc(cc1)CSc2ncc(c(n2)N)C(=O)OC HTS02129 CCc1ccccc1NNC(=O)c2c(onc2c3ccccc3)C HTS04761 CCc1ccccc1NNC(=O)c2c(onc2c3c(cccc3Cl)F)C HTS04762 CCc1[nH]c(cn1)/C=C\2/c3ccccc3NC2=O HTS05056 Cn1c(nnc1SCC(=O)c2ccc(cc2)F)c3ccc4ccccc4c3 HTS04515 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNc3cc(ccc3Cl)C(F)(F)F HTS05549 CCCc1c(cnn1c2ccccc2)C(=O)NNc3cc(ccc3Cl)C(F)(F)F HTS05550 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N(CCC#N)Cc3cccs3 HTS06375 c1ccc(cc1)c2[nH]cc(n2)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS06125 COc1ccccc1N2CCN(CC2)Cc3c[nH]c(n3)c4ccccc4 HTS06126 c1ccc(cc1)S(=O)(=O)N(CCC#N)Cc2cccs2 HTS06370 c1cc(ccc1c2ccc(=O)n(n2)CCC(=O)O)F HTS02385 c1ccc(cc1)C(=O)NC2CCN(CC2)CC(=O)Nc3ccccc3 HTS02388 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)NC3CCS(=O)(=O)C3)Cl HTS02390 Cc1c(cnn1c2ccc(cc2)OC)C(=O)N3CCN(CC3)C HTS06081 Cc1cc(n(n1)C)NC(=O)CSCC(=O)O HTS04711 c1cc(ccc1CC#N)NC(=O)CCC(=O)O HTS04731 CC(C)(CC(=O)Nc1ccc(cc1)C#N)CC(=O)O HTS05119 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3cc(cc(c3)Cl)Cl HTS06460 Cc1c(cnn1c2ccc(cc2)F)C(=O)NCc3ccc4c(c3)OCO4 HTS06782 c1ccc(c(c1)C(=O)NCC2CC2)NS(=O)(=O)c3cc(c(c(c3)Cl)Oc4ccc(cc4Cl)[N+](=O)[O-])Cl HTS05144 Cc1nc(cn1C)S(=O)(=O)Nc2ccccc2C(=O)NCC3CC3 HTS05148 c1ccc2c(c1)/C(=C/c3c(nc4n3ccs4)Sc5ccc(cc5)Cl)/C(=O)N2 HTS04703 Cc1c(cnn1c2ccc(cc2)F)C(=O)Nc3ccc(cc3)OC HTS06784 Cc1c(c(on1)C)S(=O)(=O)Nc2ccccc2SCCS(=O)(=O)c3ccc(cc3)Cl HTS06080 c1ccc(cc1)c2nc(cs2)C(=O)O CC18301 c1ccc(cc1)COC(=O)N2c3ccccc3CC2C(=O)O CC13401 CCOC(=O)c1cc(ccc1N2CCCCC2)n3cccc3 HTS02679 CCOC(=O)c1c(n(c(c1/C=C\2/c3ccccc3NC2=O)C)Cc4cccs4)C HTS04706 c1cc(sc1)c2cc(nn2c3ccc(cc3)Cl)C(F)(F)F HTS05936 Cc1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3 HTS05937 CC(C)(C)c1ccc(cc1)NNC(=O)c2c(c3ccccc3s2)Cl HTS06464 c1ccc2c(c1)C(=O)N(C(N2)c3ccccn3)CCCN4CCOCC4 HTS04789 c1cc(ccc1CN2CCS(=O)(=O)CC2)NC(=O)c3ccc(cc3)F HTS04105 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)c3ccc(cc3)OC HTS04110 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccc(c2)S(=O)(=O)N HTS05233 Cc1ccc(cc1NC(=O)c2cc(on2)C)S(=O)(=O)N(C)C HTS05242 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl HTS02709 COc1ccc(cc1)OCC(CNC(=S)Nc2ccccc2)O HTS04965 COc1ccc(cc1)OCC(CNC(=O)c2ccccc2C(=O)O)O HTS04967 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)c3cc(n(n3)C)C(F)(F)F HTS07358 c1cc(ccc1C#N)NC(=O)CSCC(=O)O HTS05122 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSc4nc5ccccc5s4)C(F)(F)F HTS04710 COc1ccc(cc1)c2ccnc(n2)SCC(=O)N3CCc4c5ccccc5[nH]c4C3C(F)(F)F HTS05042 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSC4=NCCS4)C(F)(F)F HTS05060 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)Nc3ccc(cc3F)F HTS01415 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)OC)NC(=O)Nc3ccc(cc3F)F HTS01416 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)c3ccc(cc3)F HTS04109 Cn1c(nnc1SCC(=O)c2ccc3c(c2)OCCO3)c4ccc5ccccc5c4 HTS04513 Cn1c(nnc1SCC(=O)c2ccc3c(c2)OCCCO3)c4ccc5ccccc5c4 HTS04514 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS05746 Cn1c(nnc1SCC(=O)NNC(=O)c2cccc3c2cccc3)c4ccco4 HTS04853 Cn1c(nnc1SCC(=O)N(c2ccccc2)C3CCCCC3)c4ccco4 HTS04854 Cc1nc(cn1C)S(=O)(=O)N2CCC(CC2)NC(=O)c3ccccc3 HTS02383 COc1ccc(cc1)NNC(=O)c2c(cccc2Cl)F HTS04497 CCc1ccc(cc1)C(=O)NNc2ccc(cc2)OC HTS04499 Cc1c2ccccc2sc1CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS06962 c1ccc(cc1)CCC(=O)NNc2ccccc2F HTS05023 C/C(=N\Nc1c(cc(cc1[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])/c2cc(cc(c2O)Cl)Cl CD03812 Cc1c(cnn1c2ccc(cc2)F)C(=O)NC3Cc4ccccc4C3 HTS02628 Cc1c(cnn1c2ccc(cc2)F)C(=O)N3CCC(CC3)c4ccccc4OC HTS02629 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)NCc2cc(cc3c2OCOC3)F HTS04160 Cc1cc(=O)oc2c1ccc(c2)NC(=O)CCC(=O)O HTS07013 CCc1ccnc(c1)NS(=O)(=O)c2ccc3c(c2)OCCO3 HTS05589 Cc1ccc(cc1NC(=O)c2ccc(cc2)C(C)(C)C)S(=O)(=O)N(C)C HTS06212 c1ccc2c(c1)OCC(O2)C(=O)Nc3cccc(c3)S(=O)(=O)N HTS06215 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCCN(CC3)c4c(cccn4)C#N HTS05330 Cc1cccc(c1C(=O)O)NC(=O)c2c(nns2)C HTS05560 Cc1cccc(c1C(=O)O)NC(=O)c2ccc(s2)c3ccccc3 HTS05561 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CN4CCC(CC4)NC(=O)c5ccccc5 HTS02380 CC(C)(C)c1cc2[nH]c3c(c(=O)n2n1)CN(C3=O)C4CCCCC4 HTS06828 c1ccc2c(c1)CC(C2)NC(=O)Nc3csc4c3cccc4 HTS07216 c1ccc(cc1)CN2CCC(CC2)NC(=O)Nc3csc4c3cccc4 HTS07217 CCCc1ccc(cc1)C(=O)NNc2ccccc2CC HTS04755 CCc1ccccc1NNC(=O)c2cc(on2)C HTS04756 CCc1ccccc1NNC(=O)c2cccs2 HTS04758 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3ccc4ccccc4c3 HTS04505 Cc1cc(=O)[nH]c2n1nc(c2)c3ccccc3 HTS05432 Cc1c(cnn1c2ccc(cc2)F)C(=O)N(Cc3ccccc3)Cc4cccnc4 HTS02631 c1cc(sc1)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS04094 CCc1ccccc1NNC(=O)c2ccc(cc2F)F HTS04749 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccc(cc3)C(C)(C)C HTS06475 c1ccc2c(c1)c(c(s2)C(=O)NNc3cc(cc(c3)Cl)Cl)Cl HTS06179 Cc1c(cnn1c2ccc(cc2)F)C(=O)NCCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F HTS05759 Cc1ccc(cc1Cl)NC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nc(cc(n3)C)C HTS07238 CC(C)(C)c1cc(n(n1)C)C(=O)NCc2cc(cc3c2OCOC3)F HTS04154 c1ccc(cc1)c2nc(nn2c3ccccc3)C(=O)O HTS05434 c1ccc(cc1)c2nc(nn2c3ccccc3)C(=O)Nc4ccccc4 HTS05435 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)C#N)Cl HTS05192 c1ccc(cc1)CN(CCC#N)S(=O)(=O)c2cccs2 HTS06366 Cc1c(snn1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F HTS07110 c1ccnc(c1)N2CCN(CC2)C(=O)c3cccs3 HTS07142 CN(C)c1ccc(cc1)NC(=O)Nc2csc3c2cccc3 HTS07210 c1ccc(cc1)Oc2ccc(cc2)NC(=O)Nc3csc4c3cccc4 HTS07211 CCOC(=O)N1CCC(CC1)NC(=O)Nc2ccc3c(c2)CCO3 HTS05185 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nc(cc(n3)C)C)C HTS07240 c1ccc(cc1)c2ccc(s2)c3cn4cccc(c4n3)OCc5ccc(c(c5)Cl)Cl HTS07267 c1cc(c(cc1c2csc(n2)NC(=O)Nc3ccc(cc3Cl)Cl)F)F HTS02510 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])N2CCN(CC2)CCO AW01274 Cc1cc(no1)C(=O)N(CCC#N)Cc2cccs2 HTS06387 c1ccc2c(c1)c(c(s2)C(=O)NC3CCS(=O)(=O)C3)Cl HTS02848 Cc1c(sc(n1)c2ccc3c(c2)CCO3)C(=O)NC4CCS(=O)(=O)C4 HTS03271 c1ccc2c(c1)c(c(s2)C(=O)NCc3cc(cc4c3OCOC4)F)Cl HTS04155 c1cc(ccc1S(=O)(=O)NCCNC(=O)C2=Cc3cc(ccc3OC2)Cl)Cl AW01269 c1cc(cc(c1)S(=O)(=O)N)N(S(=O)(=O)c2cc(sc2Cl)Cl)S(=O)(=O)c3cc(sc3Cl)Cl HTS07174 c1cnccc1CCCOC(=O)c2c(nccn2)C(=O)O HTS06325 Cc1ccc(cc1C)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS06348 Cc1ccc2nc(cn2c1)c3ccc(cc3)Cl HTS07280 Cc1ccc2nc(cn2c1)c3c(c4ccccc4s3)C HTS07281 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccccc3 HTS07291 c1cc2c(cc1CNC(=O)CCCO)OCO2 HTS02947 Cc1c(cc(o1)S(=O)(=O)Nc2c3c(cccc3F)n(n2)C)C(=O)OC HTS00090 c1ccc(c(c1)N2CCOCC2)OS(=O)(=O)c3cccc4c3non4 HTS06519 Cc1c(c(on1)C)S(=O)(=O)Oc2ccccc2N3CCOCC3 HTS06521 C1CCNC(=O)C(C1)NC(=O)COCC(=O)O HTS06538 c1ccc(cc1)CN(CCC#N)S(=O)(=O)c2ccc3c(c2)CCO3 HTS06368 CCOc1ccccc1N2CCN(CC2)Cc3c[nH]c(n3)c4ccccc4 HTS06136 CCOC(=O)c1cnc(nc1N)SCc2cccc(c2)C(F)(F)F HTS02125 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3cccnc3Oc4ccccc4 HTS02396 c1ccc(cc1)Oc2ccccc2NC(=O)CCC(=O)O HTS06089 c1ccc(cc1)Oc2ccccc2NC(=O)CCCC(=O)O HTS06090 CC(C)c1cc(c(c(c1)Br)NC(=O)NCCN2CCNC2=O)Br HTS03365 CCOC(=O)c1ccc(cc1)NC(=S)NCCN2CCNC2=O HTS03381 C1CC1NC(=S)NCCN2CCNC2=O HTS03382 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F HTS07351 c1cc(cc(c1)C(F)(F)F)CSc2ncc(c(n2)N)C(=O)O HTS02690 Cc1cnc(c(n1)C)NC(=O)c2cc(sc2Cl)Cl HTS03425 c1ccc(c(c1)N2CCOCC2)OC(=O)c3ccco3 HTS06435 c1ccc(cc1)C(=O)Oc2ccccc2N3CCOCC3 HTS06436 Cc1ccc(cc1)C(=O)Oc2ccccc2N3CCOCC3 HTS06439 c1cc2c(cc1NC(=O)Nc3nnc(s3)C4CC4)OCCO2 HTS03429 Cn1c(ccn1)NC(=O)CCCC(=O)O HTS06315 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccccc3C(=O)NCCCN4CCOCC4)Cl HTS06331 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)c3ccccc3C(=O)O HTS04272 CCc1ccc(cc1)C(=O)N(C)c2ccc(cc2C(=O)c3ccccc3)Cl HTS04289 Cc1cc(n(n1)C)NC(=O)CC(C)(C)CC(=O)O HTS04437 CC1c2cc(c(cc2CCN1C(=O)CC(C)(C)CC(=O)O)OC)OC HTS06399 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(s3)C#Cc4ccccc4)C(=O)OC HTS02633 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(o3)CN4C(=O)c5ccccc5C4=O)C#N HTS02637 CC1c2cc(c(cc2CCN1C(=O)CCCC(=O)O)OC)OC HTS06401 Cc1ccc(cc1)S(=O)(=O)OCC(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS02901 CC(C)n1c2ccc(cc2nc1Sc3c(ncn3C)[N+](=O)[O-])Cl HTS02663 Cc1ccc(cc1NC(=O)c2c(onc2c3ccccc3)C)S(=O)(=O)N(C)C HTS06230 Cc1ccc(cc1)S(=O)(=O)CCSc2n[nH]c(=O)n2c3ccc(cc3)OCc4ccccc4 HTS02873 CCOC(=O)c1cn(nc1N)C(=O)CCSc2ccc(cc2)OC HTS06244 c1ccc(cc1)NC(=O)N(CCC#N)CCc2ccccn2 HTS06102 Cn1cc(c(n1)c2cccc(c2)NC(=O)CSCC(=O)O)Br HTS02653 CC(C)(CC(=O)Nc1cccc(c1)c2c(cn(n2)C)Br)CC(=O)O HTS02659 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3ccccn3 HTS02319 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3cccnc3 HTS02320 CCOC(=O)C1=C(Oc2c(cc(cc2C1C(C#N)C(=O)OCC)Cl)C)N HTS02706 c1cc(ccc1C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F)Cl HTS06349 COc1ccc(cc1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3)OCc4ccccc4 HTS06351 c1cc(cnc1)NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS02323 CCc1[nH]c(c(n1)C)CN2CCN(CC2)c3ccc(cc3)F HTS06145 CC1c2cc(c(cc2CCN1C(=O)Nc3ccc(c(c3)OC4CCCC4)OC)OC)OC HTS05931 c1cc(cc(c1)S(=O)(=O)N)NC(=O)C2CCC2 HTS06228 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)N3CCCN(CC3)c4nc5ccc(cc5s4)Cl HTS02650 c1cc(sc1)C(=O)N2CCCN(CC2)C(=O)c3c(nccn3)C(=O)O HTS02813 c1cc(ccc1NC(=O)N2CCN(CC2)c3ccc(cc3)F)F HTS05805 Cc1c(cc(o1)S(=O)(=O)Nc2c3ccccc3n(n2)C)C(=O)OC HTS00088 CC(C)(C)c1ccc(cc1)NNC(=O)C2CCC2 HTS06473 Cc1cc(n(n1)C)NC(=O)COCC(=O)O HTS04439 Cc1cc(n(n1)C)NC(=O)c2ccccc2C(=O)O HTS04440 c1cc(c(c(c1)Cl)C(=O)NNc2ccc(cc2)F)F HTS04767 c1ccc(cc1)CCC(=O)NNc2ccc(cc2)F HTS04768 Cc1c(snn1)C(=O)Nc2c3c(cccc3OC)n(n2)C HTS02618 Cc1c(cnn1c2ccc(cc2)F)C(=O)Nc3ccc(c(c3)Cl)N4CCOCC4 HTS02623 c1ccc(cc1)CCC(=O)Nc2cccc(c2)S(=O)(=O)N HTS06233 CCOC(=O)C1=C(NC(=O)NC1c2c(nn(c2Cl)C)C)C HTS02772 CCOC(=O)C1=C(NC(=O)NC1c2ccc(s2)C#Cc3ccccc3)C HTS02773 c1ccc2c(c1)ccc(n2)NC(=O)c3ccc4c(c3)OCC4 HTS06290 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc4ccccc4n3 HTS06291 Cn1cc(c(n1)c2cccc(c2)NC(=O)c3c(nccn3)C(=O)O)Br HTS02655 c1cc(sc1)S(=O)(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS02518 Cn1cc(nc1)S(=O)(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F HTS02566 Cc1ccc(cc1Cl)NC(=O)NCCSCc2ccc(o2)CN(C)C HTS02911 c1ccc2c(c1)CC(C2)NC(=O)COCC(=O)O HTS02889 c1ccc2c(c1)CC(C2)NC(=O)/C=C/C(=O)O HTS02893 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCCS(=O)(=O)c4cccc(c4)C(F)(F)F HTS02876 CCc1ccc(cc1)C(=O)NNc2ccc(cc2)F HTS04769 Cc1ccc(cc1NC(=O)c2ccc(cc2F)F)S(=O)(=O)N(C)C HTS06232 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)Cc4ccncc4 HTS06235 c1ccc(cc1)C2Nc3ccccc3C(=O)N2 HTS02955 CCOc1cc(ccc1O)C2Nc3ccccc3C(=O)N2 HTS02965 COc1ccc(cc1)C2Nc3ccccc3C(=O)N2 HTS02966 c1ccc2c(c1)ccc(n2)NC(=O)c3c(cccc3Cl)Cl HTS06285 Cc1cc(cc(c1)NC(=O)Nc2ccccc2C(=O)NCC3CC3)C HTS04887 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccccc3C(=O)NCC4CC4 HTS05136 c1ccc2c(c1)c(cs2)CSCCS(=O)(=O)c3ccc(cc3Cl)Cl HTS05339 CCc1ccnc(c1)NS(=O)(=O)c2ccc(c(c2)Cl)C HTS05393 COc1ccc(cc1)Oc2cccc(c2CNC(=O)CCC(=O)O)Cl HTS05274 c1ccc(c(c1)NNC(=O)c2c(ccs2)Cl)F HTS05020 c1ccc(cc1)c2[nH]cc(n2)CN3CCN(CC3)c4ccc(cc4)F HTS06130 Cc1nc(cn1C)S(=O)(=O)NC2CCS(=O)(=O)C2 HTS02391 c1ccc(cc1)CN2CCN(CC2)Cc3c[nH]c(n3)c4ccccc4 HTS06133 Cc1c(c(on1)C)NC(=O)N2CCN(CC2)Cc3ccccc3 HTS02784 CC(C)(C)c1ccc(cc1)NC(=O)/C=C/C(=O)O HTS00520 Cn1c(c(cn1)Br)c2cccc(c2)NC(=O)COCC(=O)O HTS00874 CN(C)Cc1ccc(o1)CSCCNC(=O)Nc2ccc(cc2)F HTS02914 c1ccc(cc1)CC(c2ccccc2)NC(=S)NCc3ccc(cc3)F HTS00516 Cc1c(c(no1)c2ccccc2)C(=O)NCCCOc3ccc(cc3)NC(=O)C HTS02708 Cc1cc(no1)C(=O)NNc2ccc(cc2)F HTS05011 c1cc(ccc1NNC(=O)C2CCC2)F HTS05015 c1cc(ccc1S(=O)(=O)Nc2ccc(cc2Cl)C(F)(F)F)Cl HTS02733 c1cc(oc1C(=O)Nc2ccncc2)Oc3cc(cc(c3)Cl)Cl HTS02324 Cc1cnc(cn1)C(=O)Nc2[nH]nnn2 HTS02386 c1ccc(c(c1)NNC(=O)c2ccc(cc2F)F)F HTS05019 c1cc2c(c(c1)S(=O)(=O)NCc3csc4c3cc(cc4)Cl)non2 HTS04206 Cc1cc(=O)oc2c1ccc(c2)NS(=O)(=O)c3ccccc3 HTS06544 CCCCN1Cc2c([nH]c3cc(nn3c2=O)c4ccccc4)C1=O HTS06822 CCc1ccn2cc(nc2c1)c3ccc(s3)c4ccccn4 HTS05582 CC(=O)Nc1ccc(cc1)S(=O)(=O)Oc2ccccc2N3CCCCC3 HTS05627 Cn1c(ccc1S(=O)(=O)N(C)C)C(=O)OC SP01481 CN(Cc1cc(cc(c1)Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04317 c1cc(ccc1NNC(=O)C2CCCCC2)OC(F)(F)F HTS05646 c1cc(ccc1NNC(=O)c2ccc(cc2F)F)Cl HTS05647 Cc1c2cc(ccc2sc1S(=O)(=O)NNC(=O)c3c(nc4n3cccc4)C)Cl HTS04512 c1ccc(cc1)NC(=O)Nc2ccccc2C(=O)NCC3CC3 HTS04880 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)Nc3ccc(cc3F)F HTS04881 COc1ccc(cc1NC(=O)Nc2ccccc2C(=O)NCC3CC3)Cl HTS04882 COc1ccc(cc1)OCC(CNC(=O)Nc2ccc(cc2)F)O HTS05286 c1cc(c(c(c1)Cl)C(=O)NNc2c(cccc2Cl)Cl)F HTS06165 CCc1ccc(cc1)C(=O)NNc2c(cccc2Cl)Cl HTS06167 c1cc(c(c(c1)Cl)NNC(=O)c2cccs2)Cl HTS06171 c1cc(c(c(c1)Cl)NNC(=O)c2ccno2)Cl HTS06172 CCCCN1Cc2c([nH]c3cc(nn3c2=O)c4ccco4)C1=O HTS06826 c1c(cc(cc1Cl)Cl)NNC(=O)C2CCC2 HTS06458 COc1ccccc1C(=O)NNc2c(cc(cn2)C(F)(F)F)Cl RF04854 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)Nc2cccc(c2)F)C)C CD03697 Cc1c(ccc(n1)C(F)(F)F)C(=O)NC2CCCc3c2cccc3 HTS05608 Cc1c(snn1)C(=O)NNc2ccccc2F HTS05027 COc1ccc(cc1)OCC(CNS(=O)(=O)c2cccc(c2)Cl)O HTS05704 CN(C)Cc1ccc(o1)CSCCNC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS02756 CCOC(=O)c1c(n(c(c1/C=C\2/c3ccccc3NC2=O)C)c4ccccc4)C HTS04707 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)c3ccccc3 HTS04108 CC1(CCc2cc(ccc2O1)CN3CCN(CC3)c4ccc(cc4)F)C HTS05406 CC1(CCc2cc(ccc2O1)CN3CCN(CC3)Cc4ccc5c(c4)OCO5)C HTS05407 c1cc2cc[nH]c2c(c1)C(=O)NN SB02108 c1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)CO CC03109 c1cc(c(nc1)N2CCN(CC2)C(=O)c3cccs3)C#N HTS05005 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)CNC(=O)c3ccc(cc3)Cl HTS07359 CCOC(=O)C1CCCN(C1)C(=O)S(=O)(=O)c2ccc(s2)c3csc(n3)C HTS06902 CC(C)(C)c1ccc(cc1)NC(=O)NC2CCCc3c2cccc3 HTS05591 c1cc(cc(c1)S(=O)(=O)N)NC(=O)c2ccno2 HTS05232 Cc1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)/C=C\4/c5ccccc5NC4=O HTS05064 Cc1cn(c2c1cccc2)CCC(=O)NC3CCN(CC3)Cc4ccccc4 HTS01095 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cccnc2 HTS10987 c1ccc2c(c1)-c3nc4ccccc4n3C(N2)c5ccccn5 HTS04773 c1cc(sc1)C(=O)NNc2ccc(cc2)S(=O)(=O)N HTS04484 COc1cccc(c1)C(=O)NNc2c(cccn2)C(F)(F)F RF04873 COc1cccc(c1)c2nn(c(=O)o2)c3c(cccn3)C(F)(F)F RF04883 Cc1c(c(on1)C)S(=O)(=O)NCC(COc2ccc(cc2)OC)O HTS05705 COc1ccc(cc1)OCC(CNS(=O)(=O)c2ccc(s2)c3ccccn3)O HTS05706 c1ccc(c(c1)NNC(=O)c2cccs2)F HTS05028 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccccc3F HTS05032 CCc1[nH]c(c(n1)C)CN2CCN(CC2)c3cc(ccn3)C(F)(F)F HTS06483 Cc1csc(c1c2nc3ccccc3s2)NC(=O)COCC(=O)O HTS04626 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCC(CC3)NC(=O)c4ccccc4 HTS02384 Cc1ccc(c(c1)C)NNC(=O)c2c(ccs2)Cl HTS05035 Cc1c(snn1)C(=O)Nc2cccc(c2)S(=O)(=O)N HTS05231 Cc1c(c(n2c(n1)c(c(n2)C(F)(F)F)c3ccc(cc3)OC)C)c4ccccc4 HTS04790 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04027 CC(C)(C)OC(=O)NCCCNC(=S)Nc1ccc2c(c1)OCCO2 AW01298 c1ccc2c(c1)ccc(n2)CO CC04409 CCOC(=O)C1CCN(CC1)C(=O)c2cnn(c2C)c3ccc(cc3)OC HTS06083 Cc1c(cnn1c2ccc(cc2)OC)C(=O)N3CCCCC3 HTS06084 c1ccc2c(c1)CCCC2NC(=O)Nc3ccccc3F HTS05593 c1ccc(cc1)COc2ccc(cc2)NC(=O)NC3CCCc4c3cccc4 HTS05594 CCOC(=O)Cc1c(nn(c1O)c2ccccc2)C HTS02381 CC(=O)c1ccc(cc1)NC(=O)CN2CCC(CC2)NC(=O)c3ccccc3 HTS02382 COc1ccc(cc1)Oc2cccc(c2CNC(=O)CSCC(=O)O)Cl HTS05273 CCCCN1Cc2c([nH]c3cc(nn3c2=O)C(C)(C)C)C1=O HTS06824 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NCc3cc(cc4c3OCOC4)F HTS04153 c1ccn(c1)S(=O)(=O)c2cccc(c2)C(F)(F)F CD03851 Cc1cc(no1)C(=O)NNc2ccccc2F HTS05026 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)C#N)Sc3nc4ccc(cc4s3)Cl HTS03939 c1ccc2c(c1)/C(=C/c3c[nH]cn3)/C(=O)N2 HTS05058 c1ccc(cc1)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS05043 c1ccc(cc1)c2[nH]cc(n2)/C=C\3/c4ccccc4NC3=O HTS05057 c1ccc(cc1)CN(CCC#N)C(=O)Nc2ccc(cc2)F HTS05334 COc1ccccc1C2CCN(CC2)Cc3ccc(cc3OC)OCc4ccccc4 HTS04872 Cn1ccnc1SCC(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F HTS05041 c1ccc2c(c1)c(cs2)NC(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS07218 CC1c2cc(c(cc2CCN1C(=O)CSCC(=O)O)OC)OC HTS06403 c1cc(ccc1n2c(c(cn2)C(=O)NCc3ccc4c(c3)OCO4)C(F)(F)F)[N+](=O)[O-] HTS02886 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS02509 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccccc3F HTS05031 c1ccc(cc1)C(=O)NNc2ccccc2F HTS05033 Cc1c(c(on1)C)S(=O)(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F HTS02570 Cc1cc(nn1c2ccccc2)C(=O)Nc3cc(ccc3N4CCOCC4)C(F)(F)F HTS02575 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2)CC#N)CC(=O)O HTS06060 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cccc3c2non3 HTS07109 Cc1ccc(cc1NC(=O)Nc2cccs2)S(=O)(=O)N(C)C HTS05519 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3)C(C)(C)C)C HTS07233 CC(C)c1ccc(cc1)NC(=O)CSc2nc3cc(ccc3n2C(C)C)Cl HTS03001 CC(C)c1ccc(cc1)NC(=O)CSc2nc3cc(c(cc3c(=O)n2c4ccccc4)OC)OC HTS02535 CC1c2cc(c(cc2CCN1C(=O)c3ccccc3c4ccccc4C(=O)O)OC)OC HTS06402 Cc1ccccc1NC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nc(cc(n3)C)C HTS07239 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)c2ccccc2C(=O)O AW01101 Cc1c(sc2c1c(nc(n2)c3ccccc3OC)C)C#N SPB05358 c1ccc(cc1)CN2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F HTS02783 CC(C)(C)c1ccc(cc1)NNC(=O)c2ccccc2 HTS06476 CCc1[nH]c(c(n1)C)CN2CCN(CC2)c3ccc(cn3)C(F)(F)F HTS06481 Cc1ccc(cc1)c2csc3c2c(ncn3)NCCN4CCNC4=O HTS03371 COC(=O)c1c(ccs1)NC(=S)NCCN2CCNC2=O HTS03383 Cc1cc(cc(c1)NC(=O)N(CCC#N)Cc2ccccc2)C HTS05336 COc1ccccc1N2CCN(CC2)Cc3c[nH]nc3c4ccc(cc4)F HTS05425 c1ccc(c(c1)N2CCOCC2)OS(=O)(=O)c3cccs3 HTS06523 Cn1cc(nc1)S(=O)(=O)Oc2ccccc2N3CCOCC3 HTS06525 COC(=O)c1ccc(o1)S(=O)(=O)Oc2ccccc2N3CCOCC3 HTS06526 c1ccc(c(c1)C(=O)NC2CCCCNC2=O)C(=O)O HTS06534 c1cc(oc1)C(=O)c2coc3c2cc(cc3)O HTS05433 Cc1c(c(c(cn1)CN2CCSCC2)CO)O HTS01523 Cc1cc(=O)oc2c1ccc(c2)NS(=O)(=O)c3cccs3 HTS06546 Cc1cc(=O)oc2c1ccc(c2)NS(=O)(=O)c3cccc4c3non4 HTS06548 CC(C)(CC(=O)Nc1ccnn1C)CC(=O)O HTS06314 Cn1c(ccn1)NC(=O)COCC(=O)O HTS06316 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(cc3)OCCCN4C(=O)c5ccccc5C4=O)C(=O)OC HTS02626 c1ccc(cc1)CCC(=O)NNc2c(cccc2Cl)Cl HTS06166 c1ccc(c(c1)C(=O)NCCCN2CCOCC2)NC(=O)c3ccc(cc3F)F HTS06332 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)CCCC(=O)O HTS03114 Cc1ccc(c(c1)C)c2cn3cc(ccc3n2)C HTS07273 Cc1c(c2ccccc2[nH]1)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS06503 Cc1c(c2ccccc2[nH]1)CN3CCC(CC3)c4ccccc4OC HTS06504 c1ccc(c(c1)NNC(=O)c2c(cccc2Cl)F)F HTS05022 c1cc(sc1)C(=O)NNc2ccc(cc2)F HTS05013 Cn1c(ccn1)NC(=O)CSCC(=O)O HTS06317 Cn1c(ccn1)NC(=O)CCC(=O)O HTS06318 c1ccc(cc1)C(=O)NNc2ccc(cc2)F HTS05018 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccc(cc3)F HTS05017 c1ccc(cc1)c2[nH]cc(n2)CN3CCN(CC3)c4ccccn4 HTS06129 Cc1cccc2c1c(=O)oc(n2)c3c(nns3)C HTS05570 CC(C)(C)c1ccc(cc1)NC(=O)Oc2ccccc2N3CCCCC3 HTS05635 C1CCNC(=O)C(C1)NC(=O)CCCC(=O)O HTS06536 CC(C)(CC(=O)NC1CCCCNC1=O)CC(=O)O HTS06537 c1ccc(cc1)CN(CCC#N)C(=O)c2c(nccn2)C(=O)O HTS06542 COc1cc(c(cn1)C(=O)NCc2cc(ccc2Cl)Cl)C(F)(F)F RF04359 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)c3cccc(c3)C(F)(F)F HTS04268 COc1ccc(cc1OC)Cc2nnc(n2c3ccc(cc3)F)SCC(=O)N4CCOCC4 HTS06563 c1ccc(c(c1)C(=O)Nc2ccc(cc2)C#N)C(=O)O HTS05123 c1cc(ccc1C#N)NC(=O)c2ccc(cc2)OC(F)(F)F HTS05191 c1cc(ccc1NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3)F)F HTS06339 CC(C)(C)c1ccc(cc1)C(=O)NNc2c(cccc2Cl)Cl HTS06168 Cc1c(snn1)C(=O)NNc2c(cccc2Cl)Cl HTS06170 c1ccc(cc1)C(=O)NNc2c(cccc2Cl)Cl HTS06176 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)CNC(=O)c4ccccc4 HTS06241 c1cc2c(c(c1)S(=O)(=O)NCc3cc(cc4c3OCOC4)F)non2 HTS02314 Cn1cnc(c1N2CCOCC2)[N+](=O)[O-] HTS02946 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)Nc3ccc(cc3)OCc4ccccc4 HTS02689 CC1(CCc2cc(ccc2O1)CN3CCN(CC3)Cc4ccccc4)C HTS05401 Cc1cc(no1)NC(=O)c2ccccc2C(=O)Nc3cc(on3)C HTS05162 Cc1cc(n(n1)C)N2C(=O)CCC2=O HTS04720 CC(C)NC(=O)CSc1nnc(n1c2ccc(cc2)F)Cc3ccc(c(c3)OC)OC HTS06560 c1cc(ccc1CC#N)NC(=O)Nc2ccc(cc2)OC(F)(F)F HTS05102 CC(C)(C)C(=O)CSc1nnc(n1c2ccc(cc2)F)Cc3ccc(c(c3)OC)OC HTS06561 c1cc(ccc1C(F)(F)F)NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS06340 CC(C)(C)c1ccc(cc1)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS06346 Cc1c(c(no1)c2ccccc2)C(=O)NNc3c(cccc3Cl)Cl HTS06174 c1ccc2c(c1)ccc(n2)NC(=O)C3=Cc4cc(ccc4OC3)Cl HTS06282 Cc1ccc2c(c1)CCCN2Cc3ccc(cc3OC)OCc4ccccc4 HTS04871 c1cc(ccc1c2ccnc(n2)c3ccc(s3)Br)C(=O)N HTS01647 COc1ccc(cc1)OCC(CNC(=O)c2c(nccn2)C(=O)O)O HTS04428 COc1cc(c(cn1)C(=O)NCc2ccc(c(c2)Cl)Cl)C(F)(F)F RF04361 CC1CCN(CC1)CC(=O)Nc2ccc(cc2C(=O)c3ccccc3Cl)Cl HTS05718 COc1ccc(cc1)C(=O)NC2CCS(=O)(=O)C2 HTS02826 CCOC(=O)c1cc(ccc1N2CCCCC2)N3C(=O)c4ccccc4C3=O HTS02694 c1cc(sc1)CN(CCC#N)S(=O)(=O)c2cccs2 HTS06372 Cc1cccc(c1C(=O)O)NC(=O)c2ccccc2 HTS05568 Cc1cccc(c1C(=O)O)NC(=O)c2ccco2 HTS05569 C1CN(CCC12OCCO2)C(=O)CSCC(=O)O HTS05886 Cc1cc(cc(c1)NC(=O)N(CCC(=O)O)Cc2ccccc2)C HTS05889 Cc1ccc(n1c2ccc(c(c2)[N+](=O)[O-])N3CCOCC3)C HTS01890 Cc1csc(c1c2nc3ccccc3s2)NC(=O)CCCC(=O)O HTS04628 CC1(CCc2cc(ccc2O1)CN3CCN(CC3)c4ccccn4)C HTS05405 c1cc(ccc1c2c(c[nH]n2)CN3CCN(CC3)c4ccc(cc4)F)F HTS05411 c1ccc(cc1)C(=O)NNc2ccc(cc2)S(=O)(=O)N HTS04489 COc1ccccc1C2CCN(CC2)Cc3c[nH]nc3c4ccc(cc4)F HTS05418 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNc3cccc(c3)Cl HTS05534 c1ccc(cc1)CN2CCN(CC2)C(=O)Nc3ccccc3 HTS02779 COc1ccc(cc1NC(=O)N2CCN(CC2)Cc3ccccc3)Cl HTS02781 c1cc(ccc1C#N)NC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F HTS05194 c1cc(ccc1C#N)NS(=O)(=O)c2cc(sc2Cl)Cl HTS05195 c1cc(ccc1C#N)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS05200 Cc1ccsc1CNC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS04009 COc1ccccc1n2c(coc2=O)c3ccc(cc3)F HTS02869 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccc(cc3)C(C)(C)C HTS06474 CC(C)N1CCC(=O)N(C1=O)c2ccccc2Cl HTS06362 Cc1ccc(cc1Cl)c2c(sc(n2)NS(=O)(=O)c3cccc4c3non4)C HTS01888 c1ccc(cc1)S(=O)(=O)NC2CCCc3c2cccc3 HTS05942 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccccc2C(=O)NCC3CC3 HTS05132 Cc1c(snn1)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS05737 c1ccc(c(c1)C(=O)NCC2CC2)NS(=O)(=O)c3ccc(cc3)Oc4cccc(c4C#N)Cl HTS05140 c1ccc(cc1)c2c(nn3c2[nH]c(cc3=O)c4cccc(c4)[N+](=O)[O-])C(F)(F)F HTS02998 COC(=O)c1c(ccs1)c2ccc(o2)CN3CCN(CC3)c4ccccc4 HTS02999 CCCCc1ccc(cc1)NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccsc3C(=O)OC HTS07301 c1cc(ccc1F)S(=O)(=O)N2CCC3(CC2)OCCO3 HTS07000 c1ccc(cc1)c2c(nn3c2[nH]c(cc3=O)C(F)(F)F)C(F)(F)F HTS02997 c1ccc2c(c1)ccc(n2)NC(=O)c3c(c4ccccc4s3)Cl HTS06281 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)CSc4nc5ccccc5o4)C(F)(F)F HTS04704 Cc1c(c(c([nH]1)C)C(=O)OC)/C=C\2/c3ccccc3NC2=O HTS04705 Cc1c(c(nc(n1)c2ccccc2)SCc3ccc(cc3Cl)Cl)C#N HTS02503 c1cc(ccc1NNC(=O)C2CCC2)S(=O)(=O)N HTS04486 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2cccc(c2)[N+](=O)[O-] HTS05421 CC1=C(C(C2=C(N1)CC(CC2=O)c3ccc(cc3)F)c4c[nH]nc4c5ccc(cc5)F)C(=O)OC HTS05050 Cn1c(nnc1SCC(=O)c2ccc(cc2)OC)c3ccc4ccccc4c3 HTS04517 Cn1c(nnc1SCC(=O)c2ccc(cc2)C#N)c3ccc4ccccc4c3 HTS04520 Cc1ccc(cc1NS(=O)(=O)c2ccc(s2)c3csc(n3)C)S(=O)(=O)N(C)C HTS06645 c1ccc2cc(ccc2c1)NC(=O)NCc3ccc4c(c3)OCO4 HTS03098 COc1cc(cc(c1O)Br)c2[nH]c3ccccc3c(=O)n2 HTS03316 Cc1ccc(cc1)S(=O)(=O)NCc2csc(n2)c3cccs3 HTS06308 CC1=C(C(C2=C(N1)CCCC2=O)c3c[nH]c4c3cccc4)C(=O)OC HTS02624 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nc(cc(n3)C)C HTS07253 Cc1ccc(cc1Cl)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nc(cc(n3)C)C HTS07256 c1ccc(c(c1)NC(=O)CCC(=O)O)N2CCOCC2 HTS06759 COc1ccccc1N2CCN(CC2)Cc3c[nH]c4c3cccc4 HTS04868 c1cc(ccc1OCC(CN2CCN(CC2)Cc3ccc4c(c3)OCO4)O)F HTS04123 CCOC(=O)c1ccc(c(c1)NS(=O)(=O)c2cc(c(s2)Cl)Br)N3CCOCC3 HTS02741 COC(=O)Cc1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccc(cc3)Br HTS01640 CCOC(=O)C1CCN(CC1)C(=O)c2c(cccc2Cl)F HTS06480 CCc1ccc(cc1)C(=O)N2CCN(CC2)c3ccc(cc3)F HTS06064 c1cc(cc(c1)NC(=O)N(CCC#N)Cc2cccs2)C(F)(F)F HTS06091 Cc1ccc(c(c1)C)NNC(=O)c2cc(on2)C HTS05341 Cc1ccc(c(c1)C)NNC(=O)c2cccs2 HTS05343 c1cnoc1C(=O)NNc2c(cncc2Cl)Cl HTS03083 c1ccc2c(c1)-c3nc4ccccc4n3C(N2)c5ccc(o5)c6cccc(c6)S(=O)(=O)N HTS04781 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])NC(=O)c3c(noc3C)C HTS04902 CC(C)(CC(=O)Nc1ccccc1N2CCOCC2)CC(=O)O HTS06758 Cc1cccc(n1)NC(=O)Nc2cccc(c2)Cl HTS07023 Cc1ccc(cc1)S(=O)(=O)NCC(c2ccccc2)O HTS05989 Cc1c(snn1)C(=O)N2CCN(CC2)c3ccc(cc3)F HTS06063 c1cc(sc1)CN(CCC#N)C(=O)Nc2ccc3c(c2)CCO3 HTS06093 CC(=O)Nc1ccc(cn1)NC(=O)c2ccccc2C(=O)O HTS06709 CC(=O)Nc1ccc(cn1)NC(=O)c2c(nccn2)C(=O)O HTS06711 c1ccnc(c1)CCN(CCC#N)C(=O)Nc2ccc(cc2)F HTS06103 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2ccc(cc2)OC HTS02712 c1cc(c(cc1C(F)(F)F)Cl)NS(=O)(=O)c2ccc(s2)Br HTS02735 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3F)F HTS07292 Cc1c(cnn1c2ccc(cc2)OC)C(=O)N3CCN(CC3)c4ccc(cc4)F HTS06062 Cc1cc(cc(c1)NC(=O)N(CCC#N)Cc2cccs2)C HTS06095 CC(C)N(CCC#N)C(=O)Nc1ccccc1 HTS06096 CC(C)N(CCC#N)C(=O)Nc1ccc(cc1)F HTS06097 COc1ccc(cc1)OCC(CNC(=O)Nc2cccc3c2cccc3)O HTS05288 CC(C)(CC(=O)N1CCCN(CC1)c2c(cncc2Cl)Cl)CC(=O)O HTS04446 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)c3c(nccn3)C(=O)O HTS04796 c1ccc(cc1)CN(CCC#N)C(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F HTS06384 Cc1ccc2c(c1)n(c(=O)o2)CC/C(=N/OC(=O)c3ccccc3)/N HTS07391 Cc1ccc2c(c1)n(c(=O)o2)CCc3nc(on3)c4ccccc4 HTS07395 Cc1ccc(n1c2ccc(cc2)C3(CCSc4c3cc(cc4)F)O)C HTS01634 Cc1nc(cs1)c2ccc(s2)CO CC18209 c1cc(ncc1C(=O)O)N2CCOCC2 CC17501 Cc1cc(cc(c1)NC(=O)Nc2cccc(c2)C(=O)O)C HTS04978 CC(C)(C)c1ccc(cc1)NC(=O)NCC(COc2ccc(cc2)OC)O HTS05098 Cc1ccc(c(c1)C)NNC(=O)c2c(c3ccccc3s2)Cl HTS05036 Cc1ccc(cc1C)NNC(=O)C2CCC2 HTS05528 Cc1ccc(cc1C)NNC(=O)c2ccccc2 HTS05531 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 HTS07360 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)S(=O)(=O)c3ccccc3 HTS07361 Cc1ccc(cc1NC(=O)Nc2c(onc2c3ccccc3)C)S(=O)(=O)N(C)C HTS05518 Cc1cc(=O)oc2c1ccc(c2)NC(=O)CC3(CCCC3)CC(=O)O HTS07015 CN(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS05739 Cc1ccc(cc1)S(=O)(=O)CCSc2ncccn2 HTS04459 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccc(cc3Cl)C(F)(F)F HTS06574 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCN(CC3)CC(=O)N(C)c4ccccc4 HTS06831 CCOC(=O)C1=C(C(=O)N(C1)Cc2ccco2)O HTS06834 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCc3c(cccc3Cl)Oc4ccccc4 HTS04312 Cc1c(c2ccccc2[nH]1)CN3CCN(CC3)c4ccccn4 HTS06499 c1ccnc(c1)c2ccc(s2)C(=O)Nc3ccc(cc3)n4c(cc(n4)C(F)(F)F)c5cccs5 HTS04028 Cn1cc(nc1)S(=O)(=O)Nc2ccccc2NC3=C(CSC3)C(=O)OC HTS04264 c1cc(c(nc1)NNC(=O)CC2(CCCC2)CC(=O)O)C#N HTS04938 c1ccc(cc1)C(=O)N2CCN(CC2)c3c(cccn3)C#N HTS05004 Cc1cc(no1)C(=O)N2CCN(CC2)c3c(cccn3)C#N HTS05008 CN1CCN(CC1)CC(=O)Nc2ccc(cc2Cl)C(F)(F)F HTS06571 Cc1ccsc1C2C3=C(CCCC3=O)NC(=C2C(=O)OC)C HTS02635 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)C#N HTS05198 c1ccc(cc1)CN(CCC#N)S(=O)(=O)c2ccccc2 HTS06364 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)CC(CC(=O)O)c3ccccc3)C HTS07045 CCOC(=O)c1cnc(nc1N)SCC(=O)Nc2ccc(cc2)[N+](=O)[O-] HTS02122 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)c4ccccn4 HTS07146 Cc1ccc(cc1C)NNC(=O)c2ccno2 HTS05527 c1ccc2c(c1)OCC(O2)C(=O)N3CCN(CC3)CC(=O)Nc4ccc5c(c4)OCCO5 HTS06264 c1cc(cc(c1)C(F)(F)F)CSCC(=O)NCc2ccc3c(c2)OCO3 HTS05462 c1ccc2c(c1)ccc(n2)NS(=O)(=O)c3ccc(cc3)C#N HTS06605 CCOC(=O)C1CCN(CC1)C(=O)c2c(onc2c3c(cccc3Cl)F)C HTS06670 CCOC(=O)C1CCN(CC1)C(=O)c2ccccc2 HTS06671 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2c(cccc2Cl)Oc3ccc(cc3)OC HTS05279 Cc1ccc(cc1NS(=O)(=O)c2cccc(c2)Cl)S(=O)(=O)N(C)C HTS05492 Cc1c(csc1C(=O)NNc2cccc(c2)Cl)S(=O)(=O)c3ccc(cc3)Cl HTS05532 c1ccc(cc1)Oc2c(cccn2)C(=O)NNc3cccc(c3)Cl HTS05533 Cc1ccc(cc1NC(=O)c2cccs2)S(=O)(=O)N(C)C HTS04619 Cc1ccc2c(c1)n(c(=O)o2)CCC#N HTS06551 c1cc(ccc1C(=O)NCc2ccc3c(c2)OCO3)OC(F)(F)F HTS03597 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)COCC(=O)O HTS04797 CC1c2cc(c(cc2CCN1C(=O)c3ccc(s3)c4ccccn4)OC)OC HTS04858 c1ccc2c(c1)c(c[nH]2)CCCC(=O)O SB02058 c1cc(c(c(c1)Cl)CNC(=O)CSCC(=O)O)Sc2ccc(cc2)Cl HTS05256 c1cc(c(c(c1)Cl)CNC(=O)CCCC(=O)O)Sc2ccc(cc2)Cl HTS05260 c1cc(c(nc1)N2CCC(CC2)C(=O)N)C#N HTS06616 CCOC(=O)C1CCN(CC1)C(=O)c2c(nns2)C HTS06665 CCOC(=O)C1CCN(CC1)C(=O)c2cccs2 HTS06666 c1ccc2c(c1)ccc(n2)NC(=O)Nc3cccs3 HTS06273 c1ccc(cc1)CN(CCC#N)S(=O)(=O)c2ccc(s2)c3ccccn3 HTS06369 c1cc(sc1)CN(CCC#N)S(=O)(=O)c2ccc(cc2)F HTS06371 c1cc(sc1)CN(CCC#N)S(=O)(=O)c2ccc3c(c2)CCO3 HTS06374 c1ccc(cc1)NC(=O)Nc2csc3c2cccc3 HTS07209 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3)OCc4ccccc4)C HTS07236 Cn1c(cc(n1)C2CC2)NC(=O)Nc3csc4c3cccc4 HTS07212 c1ccc2c(c1)c(cs2)NC(=O)NCc3ccc4c(c3)OCO4 HTS07214 c1cc(sc1c2ccno2)S(=O)(=O)N3CCN(CC3)CCN4CCOCC4 HTS05172 COc1cc(cc(c1OC)OC)C2CC(=O)N(C(=O)C2)c3cc(c(cc3C(=O)OC)OC)OC HTS00618 c1ccc2cc(ccc2c1)S(=O)(=O)Nc3ccc(cc3)C#N HTS05204 CC(C)n1c2ccc(cc2nc1SCc3c(cccc3Cl)F)Cl HTS02669 CSc1nnc(s1)NCC2CC2 HTS00513 Cc1ccc(cc1NC(=O)Nc2ccc(cc2)C(C)(C)C)S(=O)(=O)N(C)C HTS05221 c1cc(c(cc1C(F)(F)F)NNC(=O)C2CCCCC2)Cl HTS05641 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)COCC(=O)O HTS02683 Cc1ccc(cc1)SCc2ccc(cc2)C(=O)Nc3ccsc3C(=O)O HTS02246 c1ccc2c(c1)c(c(s2)C(=O)Nc3cccc(c3)S(=O)(=O)N)Cl HTS05499 Cc1cc(c(o1)C(F)(F)F)NC(=O)Nc2cccc(c2)S(=O)(=O)N HTS05503 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)CSCC(=O)O HTS05816 c1cc2c(c3c1nc4c(n3)CCCC4)non2 HTS06945 CCc1ccc(cc1)C(=O)NNc2ccc(cc2C)C HTS05039 CCCc1ccc(cc1)C(=O)NNc2ccc(cc2C)C HTS05040 CC(=O)Nc1ccc(cc1)C(=O)CSc2nnc(n2c3ccccc3C(F)(F)F)O HTS02455 C1CCNC(=O)C(C1)NC(=O)CSCC(=O)O HTS06539 c1ccc(cc1)c2[nH]cc(n2)CN3CCN(CC3)c4cc(ccn4)C(F)(F)F HTS06127 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)C(=O)c4cc(nn4C)C(C)(C)C)[N+](=O)[O-])C HTS04919 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)CCC(=O)O HTS02681 c1cc2c(cc1CNC(=O)C3CCN(CC3)c4nccc(n4)C(F)(F)F)OCO2 HTS02887 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3ccncc3 HTS02321 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)Nc3ccc(cc3)F HTS02686 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccc4c(c3)OCCO4 HTS06873 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)NCCCN3CCOCC3 HTS05836 c1ccc2c(c1)c(c[nH]2)C(=O)O CC12701 COc1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3 HTS05938 CCOC(=O)C1CCCN(C1)C(=O)c2ccc(cc2Cl)Cl HTS05777 c1ccc(c(c1)NS(=O)(=O)c2cccc3c2non3)SCCS(=O)(=O)c4ccc(cc4)Cl HTS06077 c1ccc2c(c1)CCCC2NC(=O)CSCC(=O)O HTS05599 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3cc(sc3)Cl)C HTS07254 c1ccc(cc1)C(=O)N2CCC3(CC2)OCCO3 HTS06994 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N3CCC4(CC3)OCCO4 HTS07004 Cc1cccc(n1)NC(=O)Nc2ccc(cc2)OC(F)(F)F HTS07021 c1ccc(c(c1)C(=O)Nc2ccc(cc2)CC#N)C(=O)Nc3ccc(cc3)CC#N HTS05164 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N HTS05511 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCC(c2ccccc2)OC(=O)NS(=O)(=O)c3ccc(cc3)C HTS06533 c1ccc(cc1)S(=O)(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F HTS02572 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2ccc(s2)N(C)C(=O)c3ccc(cc3)Cl HTS02720 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)Nc3ccc(c(c3)Cl)C HTS02687 CCCc1cnc(nc1)Oc2c3ccc(cc3ncn2)Cl HTS05851 COc1cccc(c1)C(=O)N2CCC3(CC2)OCCO3 HTS06995 Cc1c(ccc(n1)C(F)(F)F)C(=O)N2CCC3(CC2)OCCO3 HTS06998 c1ccc(cc1)S(=O)(=O)N2CCC3(CC2)OCCO3 HTS06999 Cc1ccc(c(c1)C)NNC(=O)c2c(onc2c3ccccc3)C HTS05346 Cc1ccc(c(c1)C)NNC(=O)c2ccccc2 HTS05348 Cc1ccc(c(c1)C)NNC(=O)c2c(cccc2Cl)F HTS05037 Cc1ccc(cc1)S(=O)(=O)CCSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4 HTS02877 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(c(c3)[N+](=O)[O-])N4CCOCC4)C(=O)OC HTS02627 COc1cc(c(cc1OC)NCC(=O)Nc2ccc(cc2C(=O)c3ccccc3Cl)Cl)C(=O)OC HTS05295 CCOC(=O)C1CCN(CC1)CC(=O)Nc2ccc(cc2C(=O)c3ccccc3Cl)Cl HTS05296 c1ccc(c(c1)NC(=O)c2c(nccn2)C(=O)O)N3CCOCC3 HTS06761 Cc1cc(cc(c1)NC(=O)Nc2ccccc2N3CCOCC3)C HTS06770 Cc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2C)S(=O)(=O)N(C)C HTS06642 c1ccc(cc1)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N HTS06643 Cc1cc(no1)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS05738 CC(C)(C)c1ccc(cc1)C(=O)Nc2cccc(c2)S(=O)(=O)N HTS06214 c1cc(c(cc1C(F)(F)F)Cl)NS(=O)(=O)c2cc(c(s2)Cl)Br HTS02734 CC(=O)Nc1cccc(c1)OCCCNC(=O)c2ccc(cc2)F HTS02711 Cn1c(nnc1SCC(=O)Nc2ccccc2)c3ccco3 HTS04832 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS02339 CS(=O)(=O)CS(=O)(=O)Nc1ccc2c(c1)OCCO2 HTS02340 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])N HTS03219 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)CCc4ccncc4 HTS05515 Cc1ccc(cc1NC(=O)c2cccnc2Oc3ccccc3)S(=O)(=O)N(C)C HTS06217 Cc1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccccc3 HTS02996 COc1ccc(cc1OC)C(=O)NCc2csc(n2)c3cccs3 HTS06309 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3ccc4c(c3)OCC4)Cl HTS04644 Cc1ccc2nc(cn2c1)c3ccc(cc3)c4ccccc4 HTS07287 c1ccc(cc1)CN2CCN(CC2)C(=O)Nc3cc(cc(c3)Cl)Cl HTS02787 Cc1cc(cc(n1)O)C(=O)O MO00027 c1cc(c(cc1F)F)C(=O)NNc2cc(cc(c2)Cl)Cl HTS06177 COc1ccccc1C2CCN(CC2)Cc3ccc(o3)c4ccsc4C(=O)OC HTS03000 Cc1c(snn1)C(=O)NNc2cc(ccc2Cl)Cl HTS02936 c1ccc(cc1)c2ccnc3n2nc(c3)c4ccccc4 HTS01529 c1ccc(cc1)n2c(=O)c3c(csc3N)c(n2)C(=O)NN HTS01525 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc3c(c2)C(=O)OC3 HTS03090 Cc1ccc(cc1)S(=O)(=O)NCc2c(cccc2Cl)Oc3ccccc3 HTS04649 Cc1c2cc(ccc2sc1C(=O)CSc3nccc(n3)c4cccs4)Cl HTS04563 c1cc(cc(c1)NC(=O)CC2(CCCC2)CC(=O)O)C(=O)O HTS05073 Cc1cc(c(nc1)NC(=O)c2c(cccc2Cl)F)Br HTS03492 c1ccc(cc1)NC(=O)C2=C(CCCC2)C(=O)O HTS06204 c1ccc(cc1)C(CNC2CCCCNC2=O)O HTS06424 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cccc(c3)S(=O)(=O)N HTS05243 Cc1c(c(no1)c2ccccc2)NC(=O)NCc3csc(n3)c4cccs4 HTS06310 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccc(cc3)Cl HTS05664 COc1cc(ccc1CN2CCN(CC2)c3ccccn3)OCc4ccccc4 HTS05155 COc1cc(ccc1CN2CCN(CC2)c3ccc(cc3)F)OCc4ccccc4 HTS05156 c1cc(c(cc1C(F)(F)F)Cl)NC(=O)CN2CCOCC2 HTS06572 c1cc(c(cc1C(F)(F)F)Cl)NC(=O)CN2CCCCC2 HTS06575 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2Oc3ccccc3 HTS06576 c1cc2c(cc1N)nsn2 CC09214 COc1ccc(cc1)c2ccnc(n2)c3ccncc3 HTS01648 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)c3ccc(c(c3)OC)OC HTS02284 c1ccc(cc1)c2nc(cs2)CO CC18309 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccc(cc3F)F HTS07302 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cccs2 HTS07357 c1cc(c(nc1)N2CCN(CC2)C(=O)c3ccco3)C#N HTS05006 COc1cccc(c1)C(=O)N2CCN(CC2)c3c(cccn3)C#N HTS05010 CN(c1cc(c(cc1C(=O)OC)OC)OC)S(=O)(=O)C HTS03197 CCOC(=O)C1CCN(CC1)Cc2c[nH]c3c2cccc3 HTS04679 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)S(=O)(=O)c3ccsc3 HTS03615 COc1ccc(cc1NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccsc3C(=O)OC)Cl HTS07299 CC(=O)Nc1ccc(cn1)NC(=O)c2ccco2 HTS06714 CC(=O)Nc1ccc(cn1)NC(=O)c2ccccc2 HTS06715 Cc1ccc(c(c1)C)NNC(=O)c2ccc(cc2F)F HTS05034 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NC3CCCCNC3=O HTS06702 Cc1c(snn1)C(=O)NC2CCCCNC2=O HTS06696 c1cc(cc(c1)NC(=O)c2ccno2)C(=O)O HTS04972 CC(=O)Nc1cccc(c1)OCCCNC(=O)C2CCC2 HTS02710 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)c3cccnc3 HTS04774 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3cccc(c3)S(=O)(=O)N HTS05226 Cc1c(c2ccccc2[nH]1)CN3CCc4ccccc4C3 HTS06488 Cc1ccc2nc(cn2c1)c3ccc(cc3)C#N HTS07290 c1ccnc(c1)N2CCN(CC2)Cc3c[nH]nc3c4ccc(cc4)F HTS05410 c1cc(ccc1c2c(c[nH]n2)CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)F HTS05413 c1cc2c(cc1C(=O)O)nccn2 CC11701 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(cc3Cl)N(C)C)C#N HTS02636 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCc3c(cccc3Cl)Sc4ccc(cc4)Cl HTS05251 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl HTS05254 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3)OC(F)(F)F)C HTS07232 COc1cc(ccc1CN2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)OCc4ccccc4 HTS05153 Cc1c(c(n2c(n1)c(c(n2)C(F)(F)F)c3ccc(cc3)Br)C)c4ccccc4 HTS04791 Cc1c(c(n2c(n1)c(c(n2)C(F)(F)F)c3ccccc3)C)c4ccccc4 HTS04792 c1cnc2nc(cn2c1)c3ccc(cc3)OC(F)(F)F HTS04844 Cc1ccc(cc1NC(=O)NCC(COc2ccc(cc2)OC)O)F HTS05287 c1cc(ccc1c2c(c[nH]n2)CN3CCN(CC3)c4cc(ccn4)C(F)(F)F)F HTS05424 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3c[nH]nc3c4ccc(cc4)F)C(=O)OC HTS04686 COc1ccc(cc1OC2CCCC2)/C=C\3/c4ccccc4NC3=O HTS04708 CC(C)c1cc(c(c(c1)Br)NC(=O)Nc2ccc3ccccc3n2)Br HTS05966 CCOC(=O)c1cc(ccc1N2CCCCC2)NS(=O)(=O)c3ccc(cc3)F HTS04637 c1ccc(cc1)Oc2cccc(c2CNS(=O)(=O)c3ccccc3)Cl HTS04646 CSc1c(c(sn1)SC)C(=O)NN2CCOCC2 HTS03358 Cn1c(ccc1S(=O)(=O)NN2CCOCC2)C(=O)OC HTS03663 Cc1cc(c2cc([nH]c2c1)C(=O)N(C)C3CCN(CC3)C)C HTS06801 c1cc(cc(c1)S(=O)(=O)N)NC(=O)Nc2ccc(cc2)OC(F)(F)F HTS05227 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)c5ccccc5)C1=O HTS06839 COc1ccc(cc1)c2c(c[nH]n2)CN3CCC(CC3)c4ccccc4OC HTS05691 Cc1c(cnn1c2ccc(cc2)F)C(=O)Nc3ccccc3 HTS05758 CCCCc1[nH]cc(n1)/C=C\2/c3ccccc3NC2=O HTS05055 Cc1ccc(cc1)C(=O)CSc2nnc(n2C)c3ccc4ccccc4c3 HTS04519 CCOC(=O)C1=C(Oc2c(cc(cc2Br)Cl)C1C(C#N)C(=O)OCC)N HTS02702 c1ccc(c(c1)N2CCOCC2)OS(=O)(=O)c3ccc(s3)c4ccccn4 HTS06520 c1ccc(cc1)c2[nH]cc(n2)CN3CCC(CC3)C(=O)c4ccc(cc4)F HTS06137 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc4ccccc4n3 HTS06274 Cc1cc(c2cc([nH]c2c1)C(=O)NCCNc3ccc(cn3)C(F)(F)F)C HTS06803 c1ccc(cc1)C(=O)Nc2cccc(c2)S(=O)(=O)N HTS05229 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)Cc5ccccc5)C1=O HTS06836 CC(C)(CC(=O)Nc1ccccc1Oc2ccccc2)CC(=O)O HTS06088 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])NC(=O)c3c(nns3)C HTS04903 Cc1c(sc(n1)c2cnccn2)C(=O)NCc3ccncc3 HTS05751 Cc1c(sc(n1)c2cnccn2)C(=O)Nc3ccccc3 HTS05755 c1ccc(cc1)Oc2cccc(c2CNS(=O)(=O)c3cccc4c3non4)Cl HTS04648 c1ccc(cc1)Oc2ccccc2NC(=O)CSCC(=O)O HTS06086 c1ccc(cc1)CSC(=S)NC(=O)c2ccc(cc2)C(F)(F)F SPB01636 COc1ccc(cc1)c2c(c[nH]n2)CN3CCC(CC3)(c4ccc(cc4)Cl)O HTS05695 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)c5ccc(cc5)OC)C1=O HTS06840 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)CC(C)(C)CC(=O)O HTS05818 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])NC(=O)c3ccno3 HTS04900 c1ccc(cc1)NC(=O)CN2CCN(CC2)C(=O)C3COc4ccccc4O3 HTS06262 c1ccc2c(c1)OCC(O2)C(=O)N3CCN(CC3)CC(=O)Nc4ccc(cc4)F HTS06265 Cc1c(snn1)C(=O)N2CCN(CC2)c3ccccn3 HTS07144 CC(C)(C)NC(=O)Nc1c(c(nn1C)C(F)(F)F)c2ccc(cc2)OC HTS01420 CCOc1ccccc1NC(=O)Nc2ccc(cc2)S(=O)(=O)Nc3nc(cc(n3)C)C HTS07242 c1cc(c2nc(cn2c1)c3ccc(cc3)Cl)OCc4ccc(c(c4)Cl)Cl HTS07276 Cc1ccc2nc(cn2c1)c3ccc(cc3)OC HTS07278 c1cc(ccc1CN2CCS(=O)(=O)CC2)NC(=O)c3ccc(cc3)Cl HTS05732 c1cc(ccc1N2CCN(CC2)S(=O)(=O)c3ccc4c(c3)CCO4)F HTS05812 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc4c(c3)OCCO4 HTS06874 CCOC(=O)C1CCN(CC1)C(=O)c2c(onc2c3ccccc3)C HTS06669 c1cc2c(cc1CNC(=O)CSCC(=O)O)OCO2 HTS02884 Cc1ccc(cc1NS(=O)(=O)c2cc(sc2Cl)Cl)S(=O)(=O)N(C)C HTS05491 COc1ccc(cc1OC)Cc2nnc(n2c3ccc(cc3)F)SCC4CC4 HTS06558 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CN4CCN(CC4)c5ccc(cn5)[N+](=O)[O-] HTS02377 Cc1ccc(cc1)COc2c3ccc(cc3ncn2)Cl HTS06405 Cc1c(c(no1)c2ccccc2)C(=O)NCc3c(cccc3Cl)Oc4ccccc4 HTS04645 c1ccc(cc1)C(=O)NC2CCCCNC2=O HTS06694 Cc1c(ccc(n1)C(F)(F)F)C(=O)NC2CCCCNC2=O HTS06695 Cc1ccc2c(c1)n(c(=O)o2)CCc3nc(on3)c4cc(on4)C HTS07397 COC(=O)c1c(ccs1)OCc2ccc(cc2)Cl HTS02746 CCCc1ccc(cc1)C(=O)NN2CC(=O)N(CC2=O)c3cc(cc(c3)Cl)Cl HTS02090 c1ccc2c(c1)nc(n2CCC#N)S HTS00511 CCCc1c(cnn1c2ccccc2)C(=O)NNc3cccc(c3)Cl HTS05535 Cc1ccc(cc1)NNC(=O)c2cc(nn2Cc3ccccc3)C(C)(C)C HTS05539 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)N(Cc3ccccc3)Cc4cccnc4 HTS02291 c1cc(ccc1C(=O)Nc2ccc(cc2Cl)C(F)(F)F)F HTS02736 c1cnc(nc1C(F)(F)F)N2CCN(CC2)CCNC(=O)NC3CCCCC3 HTS03008 CCOC(=O)c1cc(ccc1N2CCCCC2)NC(=O)Nc3ccc(cc3)C(F)(F)F HTS02688 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(c4ccccc4)(c5ccccc5)O HTS05465 Cn1cc(c(n1)c2cccc(c2)NC(=O)CCCC(=O)O)Br HTS02651 Cc1ccc2c(c1)CCCN2C(=O)c3cnn(c3C)c4ccc(cc4)F HTS02622 CC(C)(C)c1ccc(cc1)NC(=O)c2ccc(cc2)N3C(=O)CSCC3=O HTS00518 COc1ccccc1NC(=O)Nc2ccccc2C(=O)NCCCN3CCOCC3 HTS05838 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCc3csc4c3cccc4 HTS00514 COc1ccccc1NNC(=O)c2cccnc2Oc3ccccc3 HTS05543 c1ccc(cc1)Oc2c(cccn2)C(=O)NNc3cc(ccc3Cl)C(F)(F)F HTS05548 c1cc(sc1)CN(CCC#N)C(=O)CSCC(=O)O HTS06541 c1cc2c(cc1n3c(=O)[nH]nc3SCCS(=O)(=O)c4ccc(cc4Cl)Cl)OCCO2 HTS02878 c1cc(ccc1F)S(=O)(=O)CCSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4 HTS02879 COc1ccc(cc1)OCC(CNC(=S)Nc2ccc3c(c2)OCO3)O HTS06939 Cc1cccc(n1)NC(=O)Nc2ccc(cc2)F HTS06629 CCOC(=O)c1cc(nc(c1C#N)N2CCC(CC2)C(=O)N)C HTS06625 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)F)c3ccco3 HTS04833 c1cc2c(cc1CO)non2 CC09709 c1ccc(cc1)c2cc(=O)n3c([nH]2)c(c(n3)C(F)(F)F)c4ccccc4 HTS02993 CCCc1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccccc3 HTS02995 Cc1ccc(cc1)NNC(=O)C2CCCCC2 HTS05541 Cc1c(cc(o1)S(=O)(=O)NCC2CN(CN(C2)Cc3ccccc3)Cc4ccccc4)C(=O)OC HTS02114 COc1ccccc1C2CCN(CC2)c3nc(ns3)c4ccccc4 HTS02586 CC(C)(CC(=O)NC1Cc2ccccc2C1)CC(=O)O HTS02891 c1ccc(cc1)CN2CCN(CC2)Cc3c[nH]nc3c4ccc(cc4)F HTS05415 c1ccc2c(c1)CCCC2NC(=O)C3=C(SCCS3)C(=O)O HTS05596 c1ccc(cc1)CN2CCN(CC2)C(=O)Nc3ccc(cc3)F HTS02785 c1cc(cc(c1)Cl)NNC(=O)C2CCCCC2 HTS05536 Cc1ccc(cc1)NNC(=O)c2c(c(cs2)S(=O)(=O)c3ccc(cc3)Cl)C HTS05537 Cc1ccc(cc1)NNC(=O)c2cccnc2Oc3ccccc3 HTS05538 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)NC3Cc4ccccc4C3 HTS03161 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(s3)C#Cc4ccccc4)C#N HTS03163 CC1=C(C(C2=C(N1)CCCC2=O)c3c[nH]nc3c4cccs4)C#N HTS03164 c1ccc2c(c1)cc(s2)C(=O)Nc3ccc4c(c3)C(=O)OC4 HTS02929 CCCc1ccc(cc1)C(=O)NNc2cc(ccc2Cl)Cl HTS02933 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)C#N HTS05206 c1cc(ccc1NC(=O)CCCC(=O)O)n2ccc(n2)C(F)(F)F HTS05207 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3)C(F)(F)F HTS03527 CC1=C(C(C2=C(N1)CCCC2=O)c3c[nH]cn3)C#N HTS03168 c1cc(c(c(c1)Cl)CNS(=O)(=O)c2ccc3c(c2)CCO3)Sc4ccc(cc4)Cl HTS05262 Cc1cc2c(cc1C)nc3c(n2)CCCC3 HTS06944 c1cc(sc1)C(=O)N2CCC3(CC2)OCCO3 HTS06996 Cn1cc(nc1)S(=O)(=O)Nc2ccccc2Oc3ccccc3 HTS06579 Cc1cc(c2cc([nH]c2c1)C(=O)N3CCC(CC3)C(=O)c4ccc(cc4)F)C HTS06809 c1ccc(cc1)C(CNS(=O)(=O)c2ccccc2)O HTS05987 COc1ccccc1NC(=O)Nc2ccccc2N3CCOCC3 HTS06769 c1ccnc(c1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)c4ccno4 HTS06599 Cn1cc(c(n1)C(F)(F)F)S(=O)(=O)Nc2ccccc2N3CCOCC3 HTS07221 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3cccnc3Oc4c5ccc(cc5ncn4)Cl HTS07330 CC1=C(C(C2=C(N1)CCCC2=O)c3c[nH]c4c3cccc4)C#N HTS03166 Cc1c2ccccc2sc1C3C(=C(NC4=C3C(=O)CCC4)C)C#N HTS03157 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(cc3Cl)C(F)(F)F)C#N HTS03158 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc4c(c3)CCO4 HTS03023 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(on3)C HTS03526 c1cc(ccc1C#N)NS(=O)(=O)c2ccc(cc2)F HTS05202 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F)CC(=O)O HTS05210 c1cnc(nc1C(F)(F)F)N2CCCN(CC2)C(=O)COCC(=O)O HTS03510 c1ccc2c(c1)CC(C2)NC(=O)CCC(=O)O HTS02890 c1ccc2c(c1)CC(C2)NC(=O)c3ccccc3C(=O)O HTS02894 c1ccnc(c1)N2CCN(CC2)C(=O)Nc3ccc(cc3)F HTS06585 Cn1c2cccc(c2c(n1)NC(=O)c3cc4ccccc4s3)OC HTS02619 c1ccc(c(c1)NC(=O)CCCC(=O)O)N2CCOCC2 HTS06754 c1ccc(c(c1)NC(=O)CSCC(=O)O)N2CCOCC2 HTS06756 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3ccc(cc3)OC(F)(F)F)Cl HTS04642 Cc1cc(no1)C(=O)NNc2cc(ccc2Cl)Cl HTS02934 CN(C)c1ccc(cc1)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)OC HTS06722 Cc1ccc(cc1)CSCC(=O)NCc2ccc3c(c2)OCO3 HTS05467 c1cc(ccc1OC(F)(F)F)SCC(=O)NCc2ccc3c(c2)OCO3 HTS05471 c1cc2c(c(c1)S(=O)(=O)NCc3c(cccc3Cl)Sc4ccc(cc4)Cl)non2 HTS05263 c1ccc(c(c1)C(=O)Nc2ccccc2N3CCOCC3)C(=O)O HTS06760 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)C(=O)C3COc4ccccc4O3 HTS03609 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N HTS06639 Cc1cccc(n1)NC(=O)Nc2ccc(cc2)C(C)(C)C HTS07022 COC(=O)c1c(ccs1)NC(=S)Nc2ccccc2N3CCOCC3 HTS07230 c1ccnc(c1)CCN(CCC#N)S(=O)(=O)c2ccc3c(c2)CCO3 HTS06376 Cc1ccc(cc1)C(=O)NC2CCCCNC2=O HTS06697 Cc1c(c(on1)C)S(=O)(=O)N(CCC#N)Cc2ccccc2 HTS06367 c1cc2c(cc1NC(=O)c3ccc(cc3F)F)C(=O)OC2 HTS02939 c1cc2c(cc1NC(=O)c3ccno3)C(=O)OC2 HTS02940 Cc1ccc(cc1C)C(=O)Nc2cc(ccc2C)S(=O)(=O)N(C)C HTS06633 c1ccc(cc1)C(=O)NCc2c(cccc2Cl)Oc3ccccc3 HTS04643 Cc1c(csc1C(=O)N(Cc2ccccc2)Cc3cccnc3)S(=O)(=O)c4ccc(cc4)Cl HTS03179 Cc1c(csc1C(=O)Nc2ccc3c(c2)COCO3)S(=O)(=O)c4ccc(cc4)Cl HTS03180 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc4c(c3)CCO4)C#N HTS03545 c1ccc(c(c1)C(F)(F)F)NC(=O)CCCC(=O)O HTS03309 Cc1c(cnn1c2ccc(cc2)F)C(=O)NCCSCc3c(cccc3Cl)F HTS02620 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)C#N)C HTS07255 c1ccc2c(c1)cccc2NC(=O)NCc3ccco3 HTS03040 c1cc(oc1)CNC(=O)Nc2ccc(cc2)OC(F)(F)F HTS03042 c1ccc(cc1)Oc2cccc(c2CNS(=O)(=O)c3ccc4c(c3)CCO4)Cl HTS04647 c1ccc2c(c1)c(cs2)CSCC(=O)NCc3ccc4c(c3)OCO4 HTS05472 Cc1ccc(c(c1)C)NNC(=O)c2c(nns2)C HTS05342 CC(C)(C)c1ccc(cc1)COc2c3ccc(cc3ncn2)Cl HTS06407 c1ccc2c(c1)ccc(n2)NC(=O)c3cccs3 HTS05480 c1cc(c(c(c1)Cl)C(=O)NNc2cc(cc(c2)Cl)Cl)F HTS06180 CC(C)(C)c1ccc(cc1)C(=O)NNc2cc(cc(c2)Cl)Cl HTS06453 c1cc(sc1)C(=O)NNc2cc(cc(c2)Cl)Cl HTS06456 Cc1ccc(cc1NC(=O)Nc2cc(oc2C(F)(F)F)C)S(=O)(=O)N(C)C HTS05502 c1cc(ccc1CC#N)N2C(=O)CCC2=O HTS05213 Cc1cc(n(n1)C)NC(=O)CC(CC(=O)O)c2ccccc2 HTS06304 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3cn(cn3)C HTS05880 Cc1ccc(cc1NC(=O)Nc2ccc(cc2)OCc3ccccc3)S(=O)(=O)N(C)C HTS05222 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc3ccccc3n2 HTS05476 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3ccccc3n2 HTS05477 CCCc1c(cnn1c2ccccc2)C(=O)NCc3ccc4c(c3)OCO4 HTS03594 c1ccc(cc1)COC(=O)N2CCC(CC2)NC(=O)Nc3ccccc3N4CCOCC4 HTS06766 Cc1ccc(cc1NC(=O)c2c(ccs2)Cl)S(=O)(=O)N(C)C HTS05496 COc1ccc(cc1)SCCC(=O)NNS(=O)(=O)c2ccc(s2)c3ccccn3 HTS05874 Cc1cnc(cn1)C(=O)NCc2c(cccc2Cl)Oc3ccccc3 HTS02397 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccc3ccccc3n2 HTS05484 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)C4=Cc5cc(ccc5OC4)Cl HTS04581 CSc1c(cccn1)C(=O)Nc2ccc3c(c2)C(=O)OC3 HTS02927 CC(c1ccccc1)n2c(nnc2SCCS(=O)(=O)c3ccc(cc3)F)O HTS08008 Cc1c(csc1C(=O)NNc2cc(ccc2Cl)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl HTS05547 Cn1c(nnc1SCC(c2ccccc2)O)c3ccc4ccccc4c3 HTS06248 CC(C)(C)c1ccc(cc1)C(=O)NNc2ccc(cc2)Cl HTS05653 Cc1c(n2ccccc2n1)C(=O)NNS(=O)(=O)c3ccc(s3)c4ccccn4 HTS05866 COc1ccc(cc1OC)Cc2nnc(n2c3ccc(cc3)F)SCC(=O)c4ccccc4 HTS06562 Cc1ccc(cc1NC(=O)Nc2cc(cc(c2)C)C)S(=O)(=O)N(C)C HTS05240 CCCc1ccc(cc1)C(=O)Nc2cc(ccc2C)S(=O)(=O)N(C)C HTS05241 c1cc2c(cc1NC(=O)c3c(ccs3)Cl)C(=O)OC2 HTS02928 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)C(=O)c4ccccc4)[N+](=O)[O-])C.CO HTS04913 CCc1ccc(cc1)C(=O)NNc2ccc(cc2)Cl HTS05652 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)C(=O)c4cccs4)[N+](=O)[O-])C HTS04915 Cc1c(snn1)C(=O)NNc2ccc(cc2)Cl HTS05655 COc1ccc(cc1)NC(=O)CC(CC(=O)O)c2ccccc2 HTS06036 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2)Oc3ccccc3)CC(=O)O HTS06037 CCOC(=O)Cc1csc(n1)NC(=O)Nc2cccc(c2)OC HTS08076 Cc1ccc(cc1)C(=O)COc2c3ccc(cc3ncn2)Cl HTS07335 Cc1ccc(cc1)C(=O)CN(Cc2ccccc2)c3ccccc3 HTS07697 c1cc2c(cc1c3cc(nc(n3)N)C(F)(F)F)CCCC2 HTS03196 CCCc1c(cnn1c2ccccc2)C(=O)NCCSCc3c(cccc3Cl)F HTS03519 Cc1cc(no1)C(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F HTS02574 c1ccc(cc1)CCC(=O)Nc2ccc3c(c2)C(=O)OC3 HTS02931 c1cc2c(cc1CNC(=O)NC3CCCCC3)OCO2 HTS03097 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)c3csc(n3)C HTS03121 Cc1c2ccccc2sc1CN3CCC(CC3)N4CCCCC4 HTS06972 Cc1cc(c2cc([nH]c2c1)C(=O)NC3CCN(CC3)Cc4ccccc4)C HTS06802 Cc1cc(c2cc([nH]c2c1)C(=O)Nc3ccccc3SCc4cccc(c4F)Cl)C HTS06805 c1ccc(cc1)C(CC(=O)N2CCN(CC2)c3ncccn3)CC(=O)O HTS05215 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCCN3CCNC3=O HTS02810 COc1cc2c(cc1OC)nc(n(c2=O)c3ccccc3)SCC(=O)Nc4ccc(c(c4)Cl)F HTS02534 CC1c2cc(c(cc2CCN1C(=O)c3ccc(cc3)OC)OC)OC HTS05912 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cn(cn2)C HTS07108 Cc1ccc2c(c1)n(c(=O)o2)CC/C(=N/OC(=O)c3cc(on3)C)/N HTS07393 COC(=O)c1ccc(o1)Oc2c3c(csc3ncn2)c4ccccc4 HTS00521 c1cc(oc1)CSCC(=O)NCc2ccc3c(c2)OCO3 HTS05310 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2)N3CCOCC3)CC(=O)O HTS06032 CN(C)c1ccc(cc1)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS06350 CC(C)N(CCC#N)C(=O)Nc1ccccc1Cl HTS06100 Cc1nc(cs1)c2ccc(cc2)NC(=O)c3cccs3 HTS03123 CC(C)n1c2ccc(cc2nc1SCC(=O)Nc3ccccc3Cl)Cl HTS03002 c1ccc(cc1)CN(CCC#N)C(=O)Nc2cccc(c2)C(F)(F)F HTS05904 Cc1c2ccccc2sc1CN3CCc4ccccc4C3 HTS06971 Cc1c(cc(o1)C(C)(C)C)C(=O)NC2CCN(CC2)Cc3ccccc3 HTS04652 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)Nc5ccc(cc5)F)C1=O HTS06838 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3)N4CCOCC4 HTS03536 Cc1cc(=O)oc2c1ccc(c2)NS(=O)(=O)c3ccc(s3)c4ccccn4 HTS06549 c1ccc(cc1)C(CC(=O)Nc2ccccc2)CC(=O)O HTS05220 CCc1ccc(cc1)C(=O)N2CCN(CC2)c3ccccn3 HTS07145 Cc1ccc(cc1NC(=O)Nc2ccccc2)S(=O)(=O)N(C)C HTS05224 c1ccc(cc1)C(CNS(=O)(=O)c2cc(sc2Cl)Cl)O HTS05986 c1ccc(cc1)NC(=O)Nc2ccccc2N3CCOCC3 HTS06768 Cc1c(c(no1)c2ccccc2)NC(=O)N(CCC#N)C(C)C HTS06098 Cc1nc(cs1)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl HTS03122 Cc1nc(cs1)c2ccc(cc2)NC(=O)c3ccco3 HTS03125 Cn1c(nnc1SCC(=O)Nc2ccc3c(c2)OCCO3)c4ccco4 HTS04835 c1ccc(cc1)C(CC(=O)N2CCN(CC2)C(=O)c3ccco3)CC(=O)O HTS05214 COc1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4ccc(cc4)F HTS05685 COc1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl HTS05687 Cn1cc(nc1)S(=O)(=O)NNC(=O)CCSc2ccc(cc2)OC HTS05860 Cc1cc(no1)C(=O)N2CCc3cc(c(cc3C2C)OC)OC HTS04855 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2cn(c(n2)C)C HTS07364 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)N3CCN(CC3)c4ccccc4 HTS06655 Cc1c(c(on1)C)S(=O)(=O)N2CCC(CC2)C(=O)N HTS05951 CCc1ccc(cc1)C(=O)Nc2ccccc2Oc3ccccc3 HTS07150 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccccc3Oc4ccccc4 HTS07151 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3ccc4c(c3)OCCO4 HTS06876 COc1ccc(cc1)OCCNC(=O)CCCO HTS03584 c1ccc2c(c1)cc(o2)C(=O)CSc3c(cccn3)C(=O)O HTS02069 COCc1cc(nc(n1)SCC(=O)c2cc3ccccc3o2)O HTS02435 Cc1ccc(cc1NC(=O)c2c(c3ccccc3s2)Cl)S(=O)(=O)N(C)C HTS05497 c1cc(cc(c1)S(=O)(=O)N)NC(=O)c2c(ccs2)Cl HTS05498 c1cnc2nc(cn2c1)c3ccc(cc3)C#N HTS04843 c1ccc2c(c1)C(=O)N(C2=O)Cc3csc(n3)c4cccs4 HTS03377 c1cc(ccc1NC(=O)COCC(=O)O)n2ccc(n2)C(F)(F)F HTS05208 c1cc(ccc1NC(=O)CCC(=O)O)n2ccc(n2)C(F)(F)F HTS05211 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccccc3C(F)(F)F)C HTS07245 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3cccc(c3C)Cl)C HTS07246 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccccc3N4CCOCC4 HTS06780 c1cc(c(nc1)N2CCOCC2)NC(=O)c3ccco3 HTS03350 CCc1ccc(cc1)S(=O)(=O)NCC(COc2ccc(cc2)OC)O HTS05293 c1cc(ccc1CSCC(=O)NCc2ccc3c(c2)OCO3)Cl HTS05309 c1cc(c(c(c1)Cl)CNC(=O)Nc2ccc(cc2)C(F)(F)F)Sc3ccc(cc3)Cl HTS05253 Cc1cccc(n1)NC(=O)Nc2ccccc2 HTS06628 COc1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4ccccc4OC HTS05694 CCOc1ccccc1N2CCN(CC2)Cc3c[nH]nc3c4ccc(cc4)OC HTS05697 COc1ccc(cc1)c2c(c[nH]n2)CN3CCC(CC3)C(=O)c4ccc(cc4)F HTS05698 CC1CCCN(C1)S(=O)(=O)c2ccc(cc2)c3cc(sc3C(F)(F)F)C(=O)OC HTS06657 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NC(=O)c3ccco3 HTS04775 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCC(c2ccccc2)O HTS05988 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3ccccc3N4CCOCC4 HTS06765 c1ccc2c(c1)c(cs2)NC(=O)Nc3ccccc3N4CCOCC4 HTS06771 COc1ccc(cc1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3)C(F)(F)F HTS06356 c1ccc(cc1)CN(CCC#N)S(=O)(=O)c2ccc(cc2)F HTS06365 c1ccc(cc1)CN(CCC#N)C(=O)CSCC(=O)O HTS06390 c1ccc(cc1)CCC(=O)NNc2cc(cc(c2)Cl)Cl HTS06451 c1cc2nc3ccsc3c(=O)n2cc1C(=O)O HTS06946 c1cc2nc3ccsc3c(=O)n2cc1C(=O)N HTS06948 COc1ccc(cc1)OCC(CNC(=S)Nc2ccc3c(c2)OCCO3)O HTS07111 c1ccc(c(c1)C(=O)NCCN2CCNC2=O)NC(=O)Nc3ccc(cc3)F HTS06735 Cc1cccc(n1)NC(=O)Nc2ccccc2F HTS06630 c1ccc(cc1)C2CC(=O)N(C(=O)C2)c3ccc(cc3)N4CCOCC4 HTS07056 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)Nc3ccccc3N4CCOCC4 HTS07202 COc1ccc(cc1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccc(cc3)Cl HTS06723 c1ccc(c(c1)NC(=O)CC2(CCCC2)CC(=O)O)N3CCOCC3 HTS06763 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)c3c(nccn3)C(=O)O HTS05820 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3ccc(cc3)OCc4ccccc4 HTS05856 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)F)C HTS07251 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cccs3)C HTS07035 COc1ccc(cc1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccc(cc3)F HTS06358 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc4c(c3)CCC(O4)(C)C)C#N HTS03546 CC(C)(C)c1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccccc3 HTS02994 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3)OC)OC)C HTS07257 c1cc(sc1)NC(=O)Nc2ccc3c(c2)OCCO3 HTS06008 COc1ccc(cc1)SCCc2nnc(n2C3CC3)SCC(=O)Nc4ccc(cc4)F HTS06247 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(c(c3)Cl)N4CCOCC4 HTS03518 c1cc(oc1)C(=O)NCc2ccc3c(c2)OCO3 HTS03588 CCCc1ccc(cc1)C(=O)NCc2ccc3c(c2)OCO3 HTS03589 c1ccc(cc1)NC(=O)Nc2cccc(c2)S(=O)(=O)N HTS05228 Cc1c(csc1C(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)S(=O)(=O)c4ccc(cc4)Cl HTS03541 c1cc2c(cc1Cl)ncnc2Oc3ccc(cn3)[N+](=O)[O-] HTS06409 c1cc2c(cc1C(=O)COc3c4ccc(cc4ncn3)Cl)OCCO2 HTS07333 c1cc2c(cc1C(=O)COc3c4ccc(cc4ncn3)Cl)OCCCO2 HTS07334 c1cc2c(c(c1)S(=O)(=O)N3CCC4(CC3)OCCO4)non2 HTS07003 CCOC(=O)C1CCCN(C1)C(=O)c2ccc(c(c2)OC)OC HTS06909 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)c5ccc(cc5)C#N)C1=O HTS07742 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccco3)C HTS07036 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc(cc3)Cl)C HTS07038 Cc1ccc(cc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)S(=O)(=O)N(C)C HTS05223 c1cc(cc(c1)S(=O)(=O)N)NC(=O)c2cccs2 HTS05230 c1cc(sc1)C(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F HTS02576 c1ccc2c(c1)c(=O)nc([nH]2)c3ccc(cc3)O HTS02970 Cc1c(c(c(o1)C)S(=O)(=O)NC(c2ccccc2)c3ccccc3)C(=O)OC HTS01165 CC(=O)c1ccc(cc1)NC(=O)CSc2nnc(n2C)c3ccco3 HTS04834 COc1ccc(cc1)OCC(CNC(=O)Nc2ccc(cc2F)F)O HTS05285 CCc1cc2c(cc1C(=O)Cn3cc(nc3C)[N+](=O)[O-])C(CCC2(C)C)(C)C HTS04163 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Nc3ccc4c(c3)OCCO4 HTS04167 c1ccc(cc1)Oc2ccccc2NS(=O)(=O)c3ccc(s3)c4ccno4 HTS06578 CCc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2C)S(=O)(=O)N(C)C HTS05505 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)OC HTS06354 Cc1c(snn1)C(=O)Nc2ccc3c(c2)C(=O)OC3 HTS02938 c1ccc(c(c1)NC(=O)Nc2cccc(c2)S(=O)(=O)N)F HTS05234 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(c(c3)OC)OCc4ccccc4)C#N HTS03544 CCOC(=O)C1CCN(CC1)CC(=O)Nc2ccc(cc2Cl)C(F)(F)F HTS06573 c1cc(ccc1C(=O)NCc2ccc(s2)S(=O)(=O)Nc3ccc4c(c3)OCCO4)Cl HTS04166 c1cnc2nc(cn2c1)c3ccc(cc3)F HTS04838 c1cc(oc1)CNC(=O)NC2CCCCC2 HTS03039 c1cc(c(c(c1)Cl)C(=O)Nc2ccc3c(c2)C(=O)OC3)F HTS02930 c1cc(c(cc1Cl)NNC(=O)c2c(ccs2)Cl)Cl HTS02918 c1cc2c(cc1NC(=O)COCC(=O)O)C(=O)OC2 HTS02922 CNc1nnc(s1)c2ccco2 HTS04836 c1cc(ccc1CC#N)NC(=O)CC2(CCCC2)CC(=O)O HTS04732 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)CC#N HTS04734 c1ccc(cc1)C2CC(=O)N(C(=O)C2)c3ccccc3 HTS06034 CC1c2cc(c(cc2CCN1S(=O)(=O)c3cn(cn3)C)OC)OC HTS05918 c1ccnc(c1)N2CCN(CC2)C(=O)CCCC(=O)O HTS06070 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)c4ccccn4 HTS06581 Cc1c(c(on1)C)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N HTS05510 Cc1cc(cc(c1)NC(=O)N2CCN(CC2)Cc3ccncc3)C HTS06234 Cc1ccc(cc1NC(=O)Nc2cccc(c2)C(F)(F)F)S(=O)(=O)N(C)C HTS06239 c1cc(ccc1NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3F)F)F HTS06342 Cc1ccc(cc1NS(=O)(=O)c2ccc(s2)c3ccno3)S(=O)(=O)N(C)C HTS05493 Cc1ccc(cc1C)C(=O)Nc2cccc(c2)S(=O)(=O)N HTS06635 c1cc(c(c(c1)Cl)C(=O)NNc2ccc(cc2F)F)F HTS05670 c1ccc(cc1)NC(=O)Nc2ccccc2C(=O)NCCCN3CCOCC3 HTS05841 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccc(cc3F)F)N(C)C HTS05850 c1ccc2c(c1)ccc(n2)NS(=O)(=O)c3cccs3 HTS05473 c1cnc2nc(cn2c1)c3ccc4c(c3)OCCO4 HTS04839 c1cc(ccc1c2c(c[nH]n2)CN3CCN(CC3)Cc4ccc5c(c4)OCO5)F HTS05412 CCOC(=O)c1cc(nc(c1C#N)N2CCCCC2)C HTS06622 c1cc(cc(c1)NC(=O)Nc2cccc(c2)S(=O)(=O)N)C(F)(F)F HTS06240 Cc1cc(cc(c1)NC(=O)Nc2cccc(c2)S(=O)(=O)N)C HTS05236 Cc1ccc(c(c1)C)NNC(=O)c2c(onc2c3c(cccc3Cl)F)C HTS05347 c1cc2c(cc1NS(=O)(=O)c3ccc(s3)c4ccno4)OCCO2 HTS04168 Cc1c(snn1)C(=O)Nc2ccccc2Oc3ccccc3 HTS07149 CC1c2cc(c(cc2CCN1S(=O)(=O)c3ccc(cc3)F)OC)OC HTS05923 c1ccc2c(c1)ccc(n2)NS(=O)(=O)c3ccccc3Cl HTS06609 c1ccc2c(c1)ccc(n2)NS(=O)(=O)c3ccc4c(c3)CCO4 HTS06611 c1cc2c(cc(=O)oc2cc1O)CSc3nnc(n3C4CC4)O HTS08007 c1ccc(cc1)S(=O)(=O)n2c3ccccc3cc2C(=O)O CC03301 COc1c(csc1Cl)C(=O)Nc2nnc(s2)C3CC3 HTS08161 Cc1ccn2c(c1)nc(c2C(=O)NNC(=O)c3ccccc3)C HTS07425 C=CCn1c(nnc1SCC(=O)N/N=C/c2ccc(cc2)[N+](=O)[O-])c3ccccc3 HTS07428 Cc1ccc(cc1)S(=O)(=O)N2CCc3cc(c(cc3C2C)OC)OC HTS05917 c1cc2c(cc1c3cc(nc(n3)N)C(F)(F)F)OCCCO2 HTS03195 c1ccc2c(c1)nc(s2)CO CC06009 c1ccc(cc1)S(=O)(=O)Nc2ccc3ccccc3n2 HTS05475 CCc1ccnc(c1)NC(=O)Nc2ccccc2C HTS04810 c1cc(cc(c1)S(=O)(=O)N)NC(=O)c2c(cccc2Cl)F HTS05244 c1cc(cc(c1)S(=O)(=O)N)NC(=O)c2ccc(cc2F)F HTS05245 Cc1ccc(cc1)C(=O)Nc2cccc(c2)C(=O)O HTS04971 CCc1ccnc(c1)NC(=O)Nc2ccc(c(c2)Cl)C HTS04808 c1ccc2c(c1)CC(C2)n3c(nnc3SCCS(=O)(=O)c4ccc(cc4)F)O HTS08312 Cn1c(cc(n1)C2CC2)NC(=O)CC(CC(=O)O)c3ccccc3 HTS06043 Cc1cc(no1)C(=O)NNc2ccc(cc2)Cl HTS05654 c1ccc(cc1)C(CC(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)CC(=O)O HTS06033 Cc1cnc(c(n1)C)N(C(=O)c2c(onc2c3ccccc3)C)C(=O)c4c(onc4c5ccccc5)C HTS03427 CCc1ccc(cc1)C(=O)N2CCC(CC2)C(=O)OCC HTS06662 c1ccc(cc1)S(=O)(=O)NC2CCCCNC2=O HTS06698 c1cc(sc1)S(=O)(=O)NC2CCCCNC2=O HTS06699 c1cc2c(cc1S(=O)(=O)NC3CCCCNC3=O)CCO2 HTS06700 Cc1ccc(cc1NS(=O)(=O)c2cc(c(o2)C)C(=O)OC)S(=O)(=O)N(C)C HTS06650 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3ccc(cc3)n4ccc(n4)C(F)(F)F HTS06045 c1ccc(cc1)NC(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F HTS06047 c1ccc2c(c1)c(cs2)CSCc3cccc(c3)C(=O)N HTS07409 CCOc1ccccc1NC(=O)Nc2cccc(c2)S(=O)(=O)N HTS05235 c1cc(c(c(c1)Cl)CSCC(=O)NCc2ccc3c(c2)OCO3)F HTS05461 CC(C)(CC(=O)NCCN1CCNC1=O)CC(=O)O HTS02470 c1ccc(c(c1)C(=O)NCCN2CCNC2=O)C(=O)O HTS02472 CCOC(=O)c1c(c2ccccc2[nH]1)N HTS03676 COc1ccc(c(c1OC)Cl)C2CC(=Nc3ccccc3S2)c4cccs4 HTS00616 Cc1cccc2c1c(=O)oc(n2)c3ccco3 HTS05575 Cc1c(c(on1)C)S(=O)(=O)Nc2ccccc2C(=O)OC HTS05959 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C3CC3)O HTS08319 COc1c(csc1Cl)C(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS06924 CN(C)c1ccc(cc1)NC(=O)CC(CC(=O)O)c2ccccc2 HTS06035 Cc1ccc2cc(ccc2n1)NC(=O)CC(CC(=O)O)c3ccccc3 HTS06044 c1csc(c1Cl)C(=O)NNc2cc(cc(c2)Cl)Cl HTS06178 c1cc(sc1)c2cc(nn2c3ccc(cc3)NC(=O)Nc4ccc(cc4)F)C(F)(F)F HTS04044 c1ccc(cc1)SCC(CN2CCN(CC2)Cc3ccc4c(c3)OCO4)O HTS04124 Cc1ccc(cc1NC(=O)c2ccccc2)S(=O)(=O)N(C)C HTS04618 Cc1ccc(cc1)S(=O)(=O)NC(=O)OCCn2c(=O)c3ccccc3cn2 HTS03338 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS03241 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)N3CCCC3 HTS03243 c1cc2c(cc1CN3CCN(CC3)C(=O)c4ccc(cc4F)F)OCO2 HTS03249 c1ccc2c(c1)CCN(C2)C(=O)c3cccs3 HTS07009 c1ccc(cc1)CN(CCC#N)C(=O)Nc2ccc3c(c2)CCO3 HTS05907 c1cc(sc1)CN(CCC#N)C(=O)Nc2ccc(cc2)F HTS05910 c1ccc(cc1)C(CNS(=O)(=O)c2ccc(s2)c3ccccn3)O HTS05992 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)c4ccc(cc4)F HTS06065 COc1ccccc1OCC(CNCc2ccc3c(c2)OCO3)O HTS02908 Cc1nc(cn1C)S(=O)(=O)NNC(=O)CCSc2ccc(cc2)OC HTS05861 Cc1c(n2ccccc2n1)C(=O)NNS(=O)(=O)C HTS05863 c1cc(ccc1C#N)C(COc2c3ccc(cc3ncn2)Cl)O HTS07349 Cc1c(n2ccccc2n1)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl HTS05862 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)Nc3cscc3C(=O)OC HTS07177 c1ccc(cc1)Oc2ccccc2NC(=O)c3c(ccs3)Cl HTS07147 Cc1ccc2c(c1)n(c(=O)o2)CCc3nc(on3)c4ccc(nc4C)C(F)(F)F HTS07396 CCc1ccc(cc1)S(=O)(=O)NCC(c2ccccc2)O HTS05990 Cc1c(c(n(n1)C)C)C(=O)O CC14701 Cc1c(sc(n1)c2cnccn2)C(=O)N3CCN(CC3)C HTS05757 Cc1c(cnn1c2ccc(cc2)F)C(=O)NCc3ccncc3 HTS05760 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])NC(=O)Nc3ccc(cc3)F HTS06010 c1ccc(cc1)c2cc(on2)c3cn4cccnc4n3 HTS04845 Cc1ccc(cc1)C(=O)NCC(c2ccccc2)O HTS05982 c1ccc(cc1)C(CNC(=O)C2CCC2)O HTS05984 c1cc(ccc1C(=O)COc2c3ccc(cc3ncn2)Cl)F HTS07332 c1ccc(c(c1)C(=O)c2cc(ccc2NC(=O)CN3CCC(CC3)C(=O)N)Cl)Cl HTS04395 COc1ccc(cc1)OCC(CNS(=O)(=O)c2cc(sc2Cl)Cl)O HTS05289 c1ccc2cc(ccc2c1)c3c(c4ccccc4[nH]3)/C=C\5/c6ccccc6NC5=O HTS05068 c1cc(c(c(c1)Cl)CNC(=O)CCC(=O)O)Sc2ccc(cc2)Cl HTS05258 Cc1c(c2c(cc1Br)nc3c(n2)CCCC3)C HTS06931 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(c(c2)Cl)NC(=O)C HTS07362 Cc1c(c(no1)c2ccccc2)C(=O)N3CCc4cc(c(cc4C3C)OC)OC HTS05911 Cc1c(nn(n1)c2ccccc2)C(=O)N3CCc4cc(c(cc4C3C)OC)OC HTS05916 CCOC(=O)C1CCN(CC1)C(=O)c2cc3c(cc(cc3[nH]2)C)C HTS06806 CC1c2cc(c(cc2CCN1C(=O)c3ccccc3)OC)OC HTS05914 Cc1c(c(on1)C)S(=O)(=O)N2CCN(CC2)c3ccccn3 HTS05949 c1cc(ccc1C(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl)F HTS06419 c1cc(c(nc1)Oc2c3ccc(cc3ncn2)Cl)NC(=O)c4cccs4 HTS07328 CC(C)N(CCC#N)C(=O)Nc1ccc2c(c1)CCO2 HTS06099 CC(C)N(CCC#N)C(=O)Nc1ccc(cc1)C(C)(C)C HTS06101 Cc1ccc(cc1)S(=O)(=O)NCC(COc2ccc(cc2)OC)O HTS05292 Cc1c(c(on1)C)C(=O)N2CCc3cc(c(cc3C2C)OC)OC HTS04860 c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccn3 HTS06583 CC(C)(CC(=O)NCc1ccc2c(c1)OCO2)CC(=O)O HTS02883 Cc1cccc2c1nc3c(n2)CCCC3 HTS06933 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCC(COc2ccc(cc2)OC)O HTS05291 Cc1ccc2c(c1)n(c(=O)o2)Cc3cccc(c3)C(=O)N HTS07410 Cc1cc(=O)n2c(n1CC(=O)NNC(=S)Nc3ccc(cc3Cl)Cl)ncn2 HTS07535 Cn1cc(nc1)S(=O)(=O)Nc2ccccc2SCCS(=O)(=O)c3ccc(cc3)Cl HTS06079 c1ccc(cc1)/C=C/C2(CC(=O)N(C2=O)C3CCCCC3)Nc4ccc(cc4)S(=O)(=O)N5CCCC5 HTS07413 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc4c(c3)OCCO4 HTS04896 c1ccc(c(c1)NC(=O)c2ccco2)OCc3ccc(c(c3)Cl)Cl HTS04545 COCc1cc(nc(n1)SC2CC(=O)N(C2=O)c3ccc(cc3)N4CCOCC4)O HTS02273 c1cc(ccc1C(=O)COc2c3ccc(cc3ncn2)Cl)OC(F)(F)F HTS07338 Cc1c(cnn1c2ccc(cc2)OC)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS07940 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2 HTS08223 CCOC(=O)C1CCN(CC1)C(=O)Nc2ccc(c(c2)Cl)C HTS07373 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccccc3O)Cl HTS02675 c1ccc(cc1)c2csc(n2)c3ccc(s3)c4ccccn4 HTS03053 c1ccnc(c1)c2ccc(s2)c3nc(cs3)c4ccc(cc4)F HTS03055 Cn1cc(nc1)S(=O)(=O)Nc2ccccc2C(=O)NCC3CC3 HTS05142 c1ccc2c(c1)-c3nc4ccccc4n3C(N2)c5ccc(o5)c6ccc(cc6)S(=O)(=O)N HTS04782 CCOC(=O)c1cc(=O)c2ccc(cc2o1)OCC(=O)Nc3ccccc3 HTS06261 COc1ccccc1NC(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F HTS06048 COc1ccc(cc1OC)Cc2nnc(n2c3ccc(cc3)F)SCc4ccc(cc4)C(=O)N HTS06557 CCOC(=O)C1CCN(CC1)C(=O)Nc2cccc(c2)Cl HTS07369 c1ccc2c(c1)CCCC2NS(=O)(=O)c3cccc4c3non4 HTS05941 Cc1cc(sc1C(=O)NCC(c2ccccc2)O)S(=O)(=O)c3ccc(cc3)Cl HTS05983 Cc1c(c(on1)C)S(=O)(=O)Nc2ccccc2Oc3ccccc3 HTS06580 C1CC1n2c(nnc2S)O HTS07408 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)Nc5ccccc5)C1=O HTS07748 c1cc(c(nc1)N2CCN(CC2)C(=O)COCC(=O)O)C#N HTS04948 c1ccc2c(c1)c(cs2)CSCCS(=O)(=O)c3ccc(cc3)F HTS05338 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5ccc6c(c5)nsn6 HTS08252 c1cc(c(cc1F)F)C(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS07976 c1cc(c(c(c1)Cl)C(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl)F HTS07979 c1ccc(cc1)NC(=S)NNC(=O)c2cnn(c2N)c3ccccc3 HTS07439 COc1ccc(cc1)c2csc(n2)c3ccc(s3)c4ccccn4 HTS03332 Cn1cnc(c1N2CCC(CC2)C(=O)N)[N+](=O)[O-] HTS03118 CC(=O)c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)F HTS06269 CCOC(=O)C1CCCN(C1)C(=O)c2csc(n2)c3ccc4c(c3)CCO4 HTS06901 c1ccc(c(c1)NC(=S)Nc2ccc3c(c2)OCCO3)N4CCOCC4 HTS07831 CC(C)(CC(=O)N1CCN(CC1)c2c(cccn2)C#N)CC(=O)O HTS04947 c1cc2cccnc2c(c1)S(=O)(=O)NCCN3CCNC3=O HTS02792 c1ccc2c(c1)-c3nc4ccccc4n3C(N2)c5ccc(o5)c6ccc(cc6)OC(F)(F)F HTS04783 c1ccc(cc1)Oc2ccccc2NS(=O)(=O)c3cccc4c3non4 HTS06577 c1cc(sc1)S(=O)(=O)N2CCC3(CC2)OCCO3 HTS07001 c1cc2c(cc1S(=O)(=O)N3CCC4(CC3)OCCO4)CCO2 HTS07002 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3nc(cs3)c4ccc(c(c4)F)F HTS06930 Cc1ccc2c(c1)n(c(=O)o2)CCC(=O)O HTS07018 CCOC(=O)C1CCCN(C1)S(=O)(=O)c2ccc(c(c2)Cl)F HTS06911 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)c3c(cccc3Cl)F HTS07305 CN(C)c1ccc(cc1)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccsc3C(=O)OC HTS07310 c1ccc(cc1)NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS07311 c1cc(c(cc1c2csc(n2)NC(=O)COCC(=O)O)F)F HTS07864 CCOC(=O)C1CCN(CC1)C(=O)Nc2cccc(c2)OC HTS07921 CC(=O)c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)CNC(=O)c4ccccc4 HTS07754 CCOC(=O)C1CCN(CC1)C(=O)Nc2ccccc2 HTS07370 CCOC(=O)C1CCN(CC1)C(=O)Nc2cccc(c2)C(F)(F)F HTS07371 c1ccc(cc1)COc2ccc(cc2)/C=N/NC(=O)c3c(c4c(c(nnc4s3)c5ccccc5)c6ccccc6)N HTS07467 Cc1c(c(on1)C)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)C(=O)C HTS07755 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc4c(c3)OCCO4)Cl HTS04893 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)Nc5ccc6c(c5)OCCO6)C1=O HTS07746 c1ccc(cc1)c2nnc(o2)C(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS08011 c1ccc(cc1)c2nnc(o2)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 HTS08012 Cc1c(cnc(n1)c2ccccc2)C(=O)O CC20201 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Nc3cccc(c3)S(=O)(=O)N HTS06229 c1ccc(cc1)c2cc(on2)c3csc(n3)N HTS07723 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)CC3(CCCC3)CC(=O)O)C(F)(F)F HTS08393 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)CCCC(=O)O)C(F)(F)F HTS08394 Cc1ccsc1C2C(=C(NC3=C2C(=O)CCC3)C)C#N HTS03155 c1ccc(cc1)c2c3c4c(c(=O)n(c(=O)[nH]4)c5cccc(c5)Cl)sc3nnc2c6ccccc6 HTS07474 c1ccc(cc1)c2c3c4c(c(=O)n(c(=O)[nH]4)c5ccc(cc5)Cl)sc3nnc2c6ccccc6 HTS07475 Cc1c(csc1C(=O)Nc2ccc3c(c2)C(=O)OC3)S(=O)(=O)c4ccc(cc4)Cl HTS03061 Cn1c(nnc1SCC=C)c2c(c3c(c(nnc3s2)c4ccccc4)c5ccccc5)N HTS07483 Cc1cccc(c1C(=O)O)NC(=O)c2cccs2 HTS05315 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)Nc5cccc(c5)C#N)C1=O HTS07747 CCOC(=O)C1=C(NC(=O)NC1c2ccc(o2)CN3C(=O)c4ccccc4C3=O)C HTS03203 c1cc(sc1)NC(=O)NCC(COc2ccc(cc2)[N+](=O)[O-])O HTS08014 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccccc3)N(C)C HTS05842 Cc1cc2nccc(n2n1)c3cccnc3 HTS08461 Cc1cc2ncc(c(n2n1)c3cccs3)/N=N/c4ccccc4 HTS08464 Cn1c(nnc1SCc2ccc(cc2)F)CSc3nnc(n3CC=C)c4ccccc4 HTS07461 c1ccc(cc1)n2c3c(cn2)c(ncn3)N/N=C/c4ccc5c(c4)OCO5 HTS07606 COc1ccccc1NC(=O)N2CCN(CC2)Cc3ccccc3 HTS02782 C=CCn1c(nnc1SCc2ccc(cc2)Cl)c3c(c4c(c(nnc4s3)c5ccccc5)c6ccccc6)N HTS07484 CCOC(=O)C1CCN(CC1)C(=O)c2cc(nn2Cc3ccccc3)C(C)(C)C HTS06685 c1cc(c(cc1F)F)C(=O)N2CCC(CC2)C(=O)O HTS06687 Cn1c(=O)c2c3c(sc2nc1SCC(=O)c4ccc(cc4)Br)CCCC3 HTS07644 COc1ccc(c(c1)C(=O)/C(=N/O)/C#N)Br CD05305 Cc1ccc(cc1NC(=O)c2ccccc2C(=O)O)S(=O)(=O)N(C)C HTS07903 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccccc3OC)N(C)C HTS05844 c1cc2c(cc1n3c(nnc3SCc4cc(=O)oc5c4ccc(c5)O)O)OCCO2 HTS07996 c1cc(oc1)C(=O)NC2CCCCNC2=O HTS06693 c1cc(sc1)C(=O)NNc2ccc(cc2)Cl HTS05656 c1cc(ccc1NNC(=O)C2CCC2)Cl HTS05663 c1ccc(cc1)CN2CCN(CC2)CCNC(=O)Nc3ccc(cc3)OCc4ccccc4 HTS03191 c1ccc(cc1)c2c3c4c(c(=O)[nH]cn4)sc3nnc2c5ccccc5 HTS07487 Cc1cc(cc(c1)NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl)C HTS07972 c1ccc(cc1)n2c(nnc2SCC(=O)c3ccc4c(c3)OCCO4)O HTS07992 Cc1c(snn1)C(=O)NNS(=O)(=O)c2ccc(cc2)Cl HTS07764 Cc1cc(c(c(c1)C)n2c(nnc2SCc3cc(=O)oc4c3ccc(c4)O)O)C HTS08003 c1ccc2c(c1)CC(C2)n3c(nnc3SCc4cc(=O)oc5c4ccc(c5)O)O HTS08006 CCc1ccn2cc(nc2c1)c3ccc(cc3)F HTS05394 c1ccc(c(c1)C(=O)NCC2CC2)NS(=O)(=O)c3cc(sc3Cl)Cl HTS05141 Cn1cnc(c1Sc2nnc(n2c3ccccc3C(F)(F)F)O)[N+](=O)[O-] HTS03323 Cn1cnc(c1SCc2csc3c2cccc3)[N+](=O)[O-] HTS03324 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)Sc5c(ncn5C)[N+](=O)[O-] HTS03328 CC1CCc2c(sc3c2c(=O)n(c(n3)SCC(=O)c4ccccc4)CC=C)C1 HTS07645 CC1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4cccc(c4)Cl)C1 HTS07651 CC(C)N(Cc1ccccc1)C(=O)Nc2ccc(cc2)C(F)(F)F HTS07904 CN(C1CCCCC1)S(=O)(=O)c2ccc(s2)S(=O)(=O)c3ccccc3 HTS07910 COc1ccc(cc1)Oc2ccc(cc2NC(=O)c3c(nccn3)C(=O)O)C(F)(F)F HTS03727 c1ccc(cc1)NC(=O)CSc2nnc(n2c3ccc4c(c3)OCCO4)O HTS08001 c1cc(ccc1C(F)(F)F)OC(CN2CCN(CC2)Cc3ccc4c(c3)OCO4)O HTS04125 c1ccc2c(c1)c(=O)nc([nH]2)c3ccncc3 HTS02968 COc1cc(ccc1OCc2ccccc2)C3Nc4ccccc4C(=O)N3 HTS02963 Cc1c(cnn1c2ccc(cc2)OC)C(=O)Nc3ccccc3Oc4ccccc4 HTS07148 Cn1cnc(c1NCc2ccc3c(c2)OCO3)[N+](=O)[O-] HTS03302 Cc1cc(c2cc([nH]c2c1)C(=O)N3CCC(CC3)N4CCCCC4)C HTS06808 Cc1c2ccccc2sc1C3C4=C(CCCC4=O)NC(=C3C(=O)OC)C HTS02634 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccc(cc3)OCc4ccccc4)OC HTS03824 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc(cc3)n4cccn4 HTS07813 c1cc(c(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)n4cccn4)C(F)(F)F HTS07815 c1cc2c(cc1C(=O)Nc3nnc(s3)C4CC4)OCO2 HTS07887 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)c3ccccc3 HTS07913 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccccc3Cl)C HTS07259 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccc(cc3)F HTS07309 c1ccc(cc1)C(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS07861 c1cc(sc1)c2nc(cs2)C(=O)O CC11501 Cc1c(cccc1Cl)NC(=O)Nc2cc(on2)C(C)(C)C HTS07320 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc(cc3)N4CCCCC4 HTS06980 c1ccc2c(c1)nc3c(n2)CCCC3 HTS08198 c1cc(cnc1)NC(=O)Nc2ccc(cc2)OC(F)(F)F HTS03051 CC(C)(C)c1ccc(cc1)c2[nH]c3ccccc3c(=O)n2 HTS03315 c1cc(c(nc1)N2CCN(CC2)C(=O)CSCC(=O)O)C#N HTS04949 Cn1c(ccc1S(=O)(=O)NCCN2CCNC2=O)C(=O)OC HTS02486 c1cc(c(c(c1)Cl)C(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O)F CD05403 c1cc(cc(c1)Cl)NC(=O)Nc2ccc(cc2)N3CCCCC3 HTS06981 CCOC(=O)C1CCN(CC1)C(=O)Nc2cc(ccc2C)F HTS07925 Cc1c(nn(n1)c2ccccc2)c3nnc(o3)c4ccc(cc4)C(F)(F)F HTS08258 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS07941 Cc1c(cnn1c2ccc(cc2)F)C(=O)N(C)C3CCN(CC3)C HTS06785 Cc1nc(cn1C)S(=O)(=O)NCCCOc2cccc(c2)NC(=O)C HTS02713 C=CCn1c(nnc1SCC(=O)NNC(=O)Nc2cccc(c2)Cl)c3ccccc3 HTS07524 Cc1nc2c3c(c(nnc3sc2c(=O)n1N(C(=O)C)C(=O)C)c4ccccc4)c5ccccc5 HTS07497 c1ccc2c(c1)N(c3ccccc3S2)Cc4n[nH]c(=S)n4c5ccc(cc5)Cl HTS07499 c1ccc(cc1)CCC(=O)NNc2cc(ccc2Cl)Cl HTS02921 CCOC(=O)c1ccc(c(c1)NC(=O)c2c(nccn2)C(=O)O)N3CCOCC3 HTS03066 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)N(c4ccccc4)C5CCCCC5 HTS06257 Cc1c(sc(n1)c2ccc3c(c2)CCO3)C(=O)NNC(=O)c4cccc5c4cccc5 HTS07376 COCCOC(=O)c1c(nccn1)C(=O)Nc2cc(ccc2Oc3ccc(cc3)OC)C(F)(F)F HTS04063 COc1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS05692 CC1(CC(=O)N(C(=O)C1)c2cccc(c2)c3c(cn(n3)C)Br)C HTS03005 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2cccc3c2non3 HTS02715 CCC(C)(C)C1CCc2c(sc(c2C#N)NC(=O)c3c(nns3)C)C1 HTS06881 Cc1c2c([nH]n1)OC(=C(C2c3ccccc3)C#N)N HTS07489 CCC(C)(C)C1CCc2c(sc(c2C#N)NC(=O)c3ccno3)C1 HTS06882 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3c(nccn3)C(=O)O)Cl HTS02400 c1cc(sc1)c2cc(nn2c3ccc(cc3)[N+](=O)[O-])C(F)(F)F HTS02726 CC(C)(C)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccccn3 HTS06584 c1ccc(cc1)COC(=O)N2c3ccccc3CC2C(=O)N4CCN(CC4)C5c6ccccc6-c7c5cccc7 HTS08259 c1c(c(sc1Cl)Cl)S(=O)(=O)NCCN2CCNC2=O HTS02487 COc1ccc(cc1OC)S(=O)(=O)NCCN2CCNC2=O HTS02488 COc1ccc(cc1)c2csc(n2)c3ccc4c(c3)OCO4 HTS03336 c1cc2c(cc1c3csc(n3)c4ccc5c(c4)OCO5)OCCO2 HTS03337 c1ccc2c(c1)cccc2NC(=O)OCCn3c(=O)c4ccccc4cn3 HTS03339 Cc1c(sc(n1)c2ccccc2)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS07939 Cc1cccc2c1c(=O)oc(n2)c3cccs3 HTS05553 COc1cc2c(cc1OC)nc(oc2=O)c3cccs3 HTS05554 c1ccc(cc1)c2ccc(cc2)C3=Nn4c(nnc4SC3)c5ccncc5 HTS07530 Cn1cnc(c1NC2Cc3ccccc3C2)[N+](=O)[O-] HTS03119 CS/C(=N\c1ccccc1)/C(C#N)c2[nH]c3ccccc3n2 HTS07506 c1ccc(cc1)/C=N/NC(=O)CN2c3ccccc3Sc4c2cccc4 HTS07508 c1ccc(cc1)c2csc(n2)c3ccc4c(c3)OCO4 HTS03054 c1cc2c(cc1C#N)nc3c(n2)CCCC3 HTS06943 Cc1ccc(cc1NS(=O)(=O)c2ccc(cc2)NC(=O)C)S(=O)(=O)N(C)C HTS06637 Cc1c(c(no1)NC(=O)c2c(nccn2)C(=O)O)Br HTS07725 c1ccc(cc1)C(CC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)CC(=O)O HTS05216 Cc1ccc(cc1NS(=O)(=O)c2ccccc2)S(=O)(=O)N(C)C HTS06641 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3cccc(c3)S(=O)(=O)N HTS06647 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)N3CCN(CC3)Cc4ccccc4 HTS06659 Cc1cccc(n1)NC(=O)Nc2ccc(s2)c3ccccc3 HTS06627 Cc1cc(c(o1)C(F)(F)F)NC(=O)N(CCC#N)Cc2ccccc2 HTS05906 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)F HTS05811 c1cc2c(c(c1)S(=O)(=O)N3CCN(CC3)c4ccc(cc4)F)non2 HTS05813 Cc1c(c(=O)n(n1C)c2ccccc2)NC(=O)CCCC(=O)O HTS05819 CCOC(=O)C1=C(OC(=C(C12c3ccccc3NC2=O)C(=O)OCC)N)c4ccccc4 HTS07527 c1cc(ccc1C(=O)Nc2cc(ccc2N3CCOCC3)C(F)(F)F)OC(F)(F)F HTS02577 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)NNC(=S)Nc4ccc(cc4)Cl HTS07504 C=CCSc1nnc(n1c2ccc(cc2Cl)Cl)CN3c4ccccc4Sc5c3cccc5 HTS07505 c1ccc(cc1)C(CC(=O)N2CCOCC2)CC(=O)O HTS06039 c1cc(c(cc1F)F)NC(=O)NCCN2CCNC2=O HTS02806 c1cc(sc1)c2cc(cnc2)C(=O)O CC11601 CCCCCc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS06987 Cc1ccc(cc1NC(=O)Nc2ccccc2F)S(=O)(=O)N(C)C HTS05238 CCc1ccnc(c1)NS(=O)(=O)c2ccccc2 HTS05388 CCCc1c(cnn1c2ccccc2)C(=O)Nc3c4c(cccc4OC)n(n3)C HTS03516 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)NC3CCN(CC3)Cc4c(cccc4Cl)F HTS03151 Cn1cnc(c1N2CCN(CC2)c3ccc(cn3)C(F)(F)F)[N+](=O)[O-] HTS03120 c1ccc(cc1)/C=N/NC(=O)c2c(c3c(cc(nc3o2)c4ccc(cc4)Cl)c5ccccc5)N HTS07538 c1ccc(cc1)Sc2c(cccn2)C(=O)Nc3ccc4c(c3)OCCO4 HTS04894 c1cc(ccc1Cc2cc(n[nH]c2=O)c3ccc(cc3)F)F HTS04501 c1ccc(cc1)c2nnc(o2)C(=O)Nc3ccccc3 HTS07738 c1ccc(cc1)c2nnc(o2)C(=O)NC3Cc4ccccc4C3 HTS07740 CCOC(=O)C1CCN(CC1)C(=O)C2Cc3ccccc3N2C(=O)OCc4ccccc4 HTS06681 c1ccc(c(c1)NS(=O)(=O)c2cccc3c2non3)N4CCOCC4 HTS07203 c1cc(ccc1C#N)N2C(=O)C3=C(C2=O)SCCS3 HTS07223 c1cc(sc1)C(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl HTS07323 c1ccc(c(c1)NC(=O)COCC(=O)O)N2CCOCC2 HTS06755 Cc1ccc2nc(cn2c1)c3cccc(c3)C#N HTS07691 Cc1ccc(cc1)C(=O)CN(Cc2ccccc2)Cc3ccccc3 HTS07695 c1cc(ccc1NC(=O)Nc2ccc3c(c2)CCO3)n4ccc(n4)C(F)(F)F HTS06046 c1cc(cc(c1)Cl)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS05495 CCOC(=O)C1CCN(CC1)c2ccccc2C3Nc4ccccc4-c5n3c6ccccc6n5 HTS04787 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc4c(c3)OCCO4)Cl HTS04170 CC(=O)c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F HTS07752 c1ccc2c(c1)c(c(s2)C(=O)NNc3ccc(cc3F)F)Cl HTS05669 CCOC(=O)C1CCN(CC1)C(=O)Nc2ccc(cc2)OCc3ccccc3 HTS07368 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)c5cc(no5)c6ccccc6)C1=O HTS07745 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)N/N=C/c5ccc(cc5)Cl)N HTS07468 c1ccc(c(c1)NNC(=O)c2ccno2)F HTS05029 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)N)N HTS07476 CC(=O)c1c(c2c(c(nnc2s1)c3ccccc3)c4ccccc4)N HTS07477 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3)Cl)NC(=O)C)C HTS07772 Cc1cc(c2cc([nH]c2c1)C(=O)N3CCC(CC3)Cc4ccccc4)C HTS07801 CCOC(=O)C1CCN(CC1)C(=O)Nc2ccc(cc2)C(C)(C)C HTS07923 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCc3ccco3 HTS03041 Cc1c(cnn1c2ccc(cc2)F)C(=O)NC3CCN(CC3)Cc4ccccc4 HTS06786 CCOC(=O)C1CCCN(C1)C(=O)S(=O)(=O)c2ccc(s2)c3ccccn3 HTS06903 CC(C)(C)c1ccc(cc1)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)OC HTS06360 Cc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N HTS06644 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)N/N=C/c4cccs4 HTS07511 c1cc(c(cc1c2csc(n2)NC(=O)CSCC(=O)O)F)F HTS07862 Cc1ccc(cc1C)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS05733 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccc(cc3)OCc4ccccc4)N(C)C HTS05843 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)Nc3ccc4c(c3)OCCO4 HTS06020 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)S(=O)(=O)c4cn(cn4)C)[N+](=O)[O-])C HTS06024 c1ccc(cc1)n2c(c(cn2)C(=O)N/N=C/c3ccc4c(c3)OCO4)N HTS07445 c1ccc(cc1)n2c3c(cn2)c(=O)n(nn3)/N=C/c4ccc(cc4)Cl HTS07448 C=CCn1c(nnc1SCc2n[nH]c(=S)o2)c3ccccc3 HTS07463 c1ccc(c(c1)NC(=O)COc2c3ccc(cc3ncn2)Cl)Cl HTS06412 CC(C)c1ccc(cc1)NC(=O)COc2c3ccc(cc3ncn2)Cl HTS06413 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccccc3Oc4ccccc4 HTS06586 c1ccc(c(c1)C#N)NC(=O)c2c(c3ccccc3s2)Cl HTS08138 c1ccc(cc1)/C=C/C2(CC(=O)N(C2=O)C3CCCCC3)Nc4ccc(cc4)S(=O)(=O)N5CCOCC5 HTS07412 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS05734 c1cc(oc1)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS05735 c1cc(ccc1CN2CCS(=O)(=O)CC2)NC(=O)c3ccc(cc3)C(F)(F)F HTS05736 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccc(cc3Cl)Cl)N(C)C HTS05845 Cn1c2cccc(c2c(n1)NC(=O)c3cc(sc3Cl)Cl)N(C)C HTS06732 c1cnccc1CN2CCN(CC2)C(=O)c3c(nccn3)C(=O)O HTS05513 Cc1ccc(cc1)S(=O)(=O)NC(=O)NC2CCCc3c2cccc3 HTS05590 Cc1cc(cc(c1)NC(=O)NCC(COc2ccc(cc2)[N+](=O)[O-])O)C HTS08018 c1ccc(cc1)/C=C/C2(CC(=O)N(C2=O)C3CCCCC3)Nc4ccc(cc4)[N+](=O)[O-] HTS07411 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)c3ccc(cc3)C(F)(F)F)C(F)(F)F HTS08387 Cc1nc2c(c(n1)Sc3nnc(n3C)c4ccccc4)sc(=S)n2c5ccccc5 HTS07564 C=CCn1c2c(c(ncn2)Sc3[nH]c4ccccc4n3)sc1=S HTS07565 Cc1c(c(on1)C)C(=O)NNc2cc(ccc2Cl)Cl HTS02935 Cc1c(c(on1)C)C(=O)Nc2ccc3c(c2)C(=O)OC3 HTS02937 CC1(CCc2cc(ccc2O1)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)C HTS05404 c1ccc(cc1)CCC(=O)N2CCC(CC2)C(=O)O HTS06688 C1CC(C1)C(=O)N2CCC(CC2)C(=O)O HTS06689 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3cc(sc3Cl)Cl)C HTS07780 CC(=O)c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccccc3 HTS06268 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)F)N3CCCCC3 HTS08401 CC(C)(C)c1ccc(cc1)NC(=O)N(C)C2CCCCC2 HTS08342 CCOC(=O)c1c(n(c(=S)s1)c2ccccc2)N HTS07567 Cc1ccn2c(c1)nc(c2C(=O)N/N=C/c3cccc(c3)OC)C HTS07418 Cc1ccn2c(c1)nc(c2C(=O)NNC(=S)NC)C HTS07421 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccccc3)CCCC2 HTS07423 c1cc(c(cc1F)F)NNC(=O)c2c(ccs2)Cl HTS05668 CCOC(=O)c1ccc(c(c1)NC(=O)COCC(=O)O)N2CCOCC2 HTS03062 c1ccc(c(c1)NC(=O)Nc2cccc(c2)C(=O)O)F HTS04976 Cc1cc(c(c(c1)C)SCC(=O)NCc2ccc3c(c2)OCO3)C HTS05468 c1ccc(cc1)c2c3c4c(c(=O)n(cn4)Cc5ccc(cc5)Cl)sc3nnc2c6ccccc6 HTS07488 Cc1c(snn1)C(=O)NNS(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 HTS07769 c1cc2c(cc1S(=O)(=O)NNc3c(cncc3Cl)Cl)OCC2 HTS03686 COCCOC(=O)c1c(nccn1)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS03724 COc1ccc(cc1)C(=O)c2coc3c2cc(c4c3cccc4)O HTS06867 c1ccc(cc1)n2c3c(cn2)c(ncn3)N/N=C/c4ccc(cc4)Cl HTS07605 C=CCn1c(c(sc1=S)C(=O)N/N=C/c2cccs2)N HTS07573 C=CCn1c(c(sc1=S)C(=O)N/N=C/c2ccc(cc2Cl)Cl)N HTS07574 CC1c2cc(c(cc2CCN1S(=O)(=O)c3ccccc3)OC)OC HTS05922 c1ccc(c(c1)C(=O)Nc2cccc(c2)S(=O)(=O)N)C(=O)O HTS07902 c1ccc(cc1)NC(=O)C2=C(SCCS2)C(=O)O HTS06327 CC(=O)Nc1ccc(cc1)NC(=O)c2c(nccn2)C(=O)O HTS03735 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccc(cc2)F HTS08077 CCOC(=O)Cc1csc(n1)NC(=O)Nc2cc(ccc2OC)Cl HTS08082 Cc1c(c(n2c3ccccc3nc2c1C#N)N4CCOCC4)CCN5CCOCC5 HTS07566 Cn1c(c(sc1=S)C(=O)N/N=C/c2ccccc2)N HTS07572 Cc1c2cc(ccc2sc1S(=O)(=O)N3CCc4cc(c(cc4C3C)OC)OC)Cl HTS05919 CC1c2cc(c(cc2CCN1S(=O)(=O)c3ccc(s3)c4ccccn4)OC)OC HTS05920 C=CCn1c(n[nH]c1=S)c2cnn(c2N)c3ccccc3 HTS07434 Cc1nc(cn1C)S(=O)(=O)N2CCc3cc(c(cc3C2C)OC)OC HTS05921 CCc1ccc(cc1)C(=O)Nc2cccc(c2)S(=O)(=O)N HTS05246 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3c(nccn3)C(=O)O HTS03728 COC(=O)c1cscc1NC(=O)c2c(nccn2)C(=O)O HTS03736 c1cc(ccc1C(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl)Cl HTS07980 c1cc(c(cc1F)F)C(=O)NNc2ccc(cc2F)F HTS05667 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)c3c(c4ccccc4s3)Cl HTS07304 CCOC(=O)c1ccc(c(c1)NC(=O)c2ccccc2C(=O)O)N3CCOCC3 HTS03065 CC1c2cc(c(cc2CCN1C(=O)Nc3ccc(cc3)F)OC)OC HTS05927 Cc1cc(cc(c1)NC(=O)N2CCc3cc(c(cc3C2C)OC)OC)C HTS05928 COc1ccc2c(c1)nc3c(n2)CCCC3 HTS05995 c1ccc(cc1)CN2CCc3c(c4c(=O)[nH]cnc4s3)C2 HTS03591 CCOC(=O)Cc1csc(n1)NC(=O)Nc2cccc(c2)Cl HTS08083 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)NNC(=O)Nc4ccc(c(c4)Cl)Cl HTS07514 c1cc2c(cc1CNC(=O)c3ccsc3)OCO2 HTS03581 c1ccc2c(c1)OCC(O2)C(=O)NCc3ccc4c(c3)OCO4 HTS03578 Cn1cc(c(n1)c2cccc(c2)N3C(=O)CCCC3=O)Br HTS03006 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3)C(F)(F)F HTS07295 c1ccc(c(c1)NS(=O)(=O)c2ccc(s2)c3ccccn3)N4CCOCC4 HTS07219 c1cc(cc(c1)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N)C(F)(F)F HTS05506 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3cccnc3 HTS03050 CC(C)c1cc(c(c(c1)Br)NC(=O)Nc2cccnc2)Br HTS03052 COc1cc(ccc1CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)OCc4ccccc4 HTS05150 c1cc(ccc1OC(F)(F)F)S(=O)(=O)NCCN2CCNC2=O HTS02478 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)NCCN3CCNC3=O HTS02485 c1cc(c(c(c1)Cl)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)F HTS03250 CCc1ccn2cc(nc2c1)c3ccc4c(c3)OCO4 HTS05964 c1cc2c(cc1F)nc3c(n2)CCCC3 HTS05996 c1cc(ccc1NC(=O)Nc2cc(cc(c2)Cl)Cl)S(=O)(=O)N HTS07180 c1c(c(c(cn1)Cl)NNC(=O)COCC(=O)O)Cl HTS03678 c1ccc(cc1)N/C(=N\NC(=O)CN2c3ccccc3Sc4c2cccc4)/SCC(=O)c5ccc(cc5)Cl HTS07515 Cc1c(ccc(n1)C(F)(F)F)C(=O)Oc2ccccc2N3CCOCC3 HTS03575 CSc1c(c(sn1)SC)C(=O)Oc2ccccc2N3CCOCC3 HTS03576 CC(C)c1cc(c(c(c1)Br)NC(=O)NCc2ccco2)Br HTS03043 c1cc2c(c(c1)S(=O)(=O)NCCN3CCNC3=O)non2 HTS02799 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCc3ccc4c(c3)OCO4 HTS03099 C1CN(C(=O)N1)CCNC(=O)COCC(=O)O HTS02474 c1ccc(cc1)C(=O)COc2c3ccc(cc3ncn2)Cl HTS07336 COc1ccc(cc1)C(=O)COc2c3ccc(cc3ncn2)Cl HTS07337 CC(C)n1c2ccc(cc2nc1SCC(=O)c3ccc(cc3)F)Cl HTS02661 c1cc(sc1)C(=O)NCCN2CCN(CC2)c3nccc(n3)C(F)(F)F HTS03013 c1ccc2c(c1)cccc2NC(=O)Nc3cccnc3 HTS03049 CCOC(=O)C1=C(OC(=C(C12c3ccccc3NC2=O)C(=O)OCC)N)C HTS07525 c1cc(ccc1C2=Nn3c(nnc3SC2)c4ccncc4)[N+](=O)[O-] HTS07531 c1ccc(cc1)c2ccc(cc2)NC(=O)CC(CC(=O)O)c3ccccc3 HTS06038 c1cc2c(cc1NC(=O)CCCC(=O)O)C(=O)OC2 HTS02923 CC(C)(C)c1ccc(cc1)C(=O)N2CCC(CC2)C(=O)O HTS07926 CN1CCN(CC1)C(=O)c2c(nccn2)C(=O)O HTS01067 Cn1cnc(c1N2CCN(CC2)C(c3ccccc3)c4ccccc4)[N+](=O)[O-] HTS03117 Cc1c(c(on1)C)S(=O)(=O)NCc2cc(cc3c2OCOC3)F HTS03240 c1cc(ccc1CC#N)NC(=O)CSCC(=O)O HTS04729 c1ccc(c(c1)C(=O)Nc2ccc(cc2)CC#N)C(=O)O HTS04730 c1c2c(cc(c1Cl)Cl)nc3c(n2)CCCC3 HTS06932 c1cc(c(cc1S(=O)(=O)NCCN2CCNC2=O)Cl)F HTS02793 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NCCN2CCNC2=O)C(F)(F)F HTS02797 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)NCCN3CCNC3=O HTS02804 c1ccc(cc1)NC(=O)N(CCC#N)Cc2cccs2 HTS05909 c1ccc(cc1)C2=CS/C(=C(/C#N)\c3[nH]c4ccccc4n3)/N2c5ccccc5 HTS07516 c1ccc(cc1)C2=Nn3c(nnc3SC2)c4ccncc4 HTS07528 c1cc(ccc1C2=Nn3c(nnc3SC2)c4ccncc4)Cl HTS07529 c1ccc(cc1)COc2ccc(cc2)NC(=O)OCCn3c(=O)c4ccccc4cn3 HTS03340 Cn1c(cc(n1)c2ccc(cc2)Cl)NS(=O)(=O)c3ccc(cc3)F HTS08068 Cn1c(nnc1Sc2c3c(nc4n2ncn4)CCC3)c5ccccc5 HTS07592 c1ccc(cc1)c2nnc(n2c3ccccc3)Sc4c5c(nc6n4ncn6)CCC5 HTS07594 c1ccc(cc1)n2c3c(cn2)c(ncn3)N4CCOCC4 HTS07599 CCOC(=O)c1c2c(sc1N)CCC2C(=O)OCC HTS07583 c1ccc(cc1)NC(=O)Nc2ccccc2Oc3ccccc3 HTS06590 CN1CCN(CC1)CC(=O)Nc2ccccc2Oc3ccccc3 HTS06591 c1ccc(c(c1)C#N)NC(=O)C2CCCCC2 HTS08133 Cc1c(snn1)C(=O)Oc2ccc(cc2)OC CD05442 CCOC(=O)c1cnn(c1NC(=O)c2c(nccn2)C(=O)O)C HTS03733 CC(C)[C@@H](C(=O)O)NC(=O)c1c(nccn1)C(=O)O HTS03738 CCOC(=O)C1CCN(CC1)CC(=O)c2ccc(cc2)C HTS07930 CCOC(=O)N1CCc2c(sc(c2C(=O)c3ccc(cc3)OC)NC(=O)Cc4ccccc4)C1 HTS08127 Cc1[nH]c(=O)c2c(n1)n(c(=S)s2)c3ccccc3 HTS07576 c1ccc(cc1)C2=CC(n3c(ncn3)N2)c4cn(nc4c5ccc(cc5)Cl)c6ccccc6 HTS07577 CC1=C(C(n2c(=O)/c(=C\c3ccc(cc3)Cl)/sc2=N1)c4ccc(cc4)OC)C(=O)OC HTS07580 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C(C)c3ccccc3)O HTS08314 c1cc(ccc1C#N)C(=O)COc2c3ccc(cc3ncn2)Cl HTS07339 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5ccc6c(c5)OCO6 HTS07943 Cc1ccc(cc1NC(=O)Nc2cc(on2)C(C)(C)C)F HTS07954 c1ccc(cc1)CN2CCN(CC2)C(=O)Nc3ccc(cc3F)F HTS02780 Cc1nc(cn1C)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS04102 c1cc(ccc1c2csc(n2)c3ccc4c(c3)OCO4)F HTS03056 c1ccnc(c1)c2ccc(s2)c3nc(cs3)c4ccc5c(c4)OCCO5 HTS03333 Cc1c(snn1)c2nnc(n2C3CC3)SCC(=O)Nc4ccc(cc4)F HTS08126 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5ccno5 HTS08253 c1ccc(cc1)Oc2ccccc2NC(=O)CN3CCCCC3 HTS06595 Cc1c2c(c(c(=O)[nH]c2n(n1)c3ccccc3)C#N)c4ccc(cc4)Cl HTS07622 CCOC(=O)C1CCN(CC1)C(=O)c2c(nn(n2)c3ccccc3)C HTS06676 CCOC(=O)C1CCN(CC1)C(=O)c2cc(cnc2)c3cccs3 HTS06683 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2c3ccc4c(c3)OCCO4)O HTS08000 c1cc(oc1)Cn2c(nnc2SCc3cc(=O)oc4c3ccc(c4)O)O HTS08005 Cc1cc(cc(c1)Sc2c(ncn2C)[N+](=O)[O-])C HTS03863 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5cc(cnc5)c6cccs6 HTS08255 c1ccc(cc1)n2c3c(cn2)c(ncn3)Nc4ccc(cc4)Cl HTS07596 CCOC(=O)C1CCN(CC1)C(=O)c2cc(nn2C(C)(C)C)C HTS07082 Cc1c(snn1)C(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08251 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5csc(n5)c6ccc7c(c6)CCO7 HTS08262 Cc1c(nn(n1)c2ccccc2)c3nnc(o3)c4cccc5c4cccc5 HTS08256 Cc1c(snn1)c2nnc(o2)c3ccc(cc3)C(F)(F)F HTS08257 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2c(c3cc(ccc3s2)Cl)C HTS07365 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc(s2)c3ccno3 HTS07366 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS06988 c1ccc(c(c1)C(=O)NCC2CC2)NS(=O)(=O)c3cccc4c3non4 HTS05143 CC1=C(C(C2=C(N1)CC(CC2=O)c3ccco3)c4ccco4)C(=O)OC HTS04696 CC1=C(C(C2=C(N1)CC(CC2=O)c3ccc(cc3)F)c4ccc5c(c4)CCC(O5)(C)C)C(=O)OC HTS05045 CC(=O)c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(s3)S(=O)(=O)c4ccccc4 HTS07753 c1ccc(cc1)CN2CCN(CC2)CCNC(=O)Nc3ccc(cc3)F HTS03183 c1cc(ccc1NC(=O)c2cc(cc(c2)Cl)Cl)S(=O)(=O)N HTS08349 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccccc2C#N HTS08146 CC(C)(C)C(=O)CSc1[nH]c2cc(c(cc2n1)Cl)Cl HTS08205 Cc1cc(n(n1)c2ccccc2)NC(=O)c3cccc(c3)[N+](=O)[O-] HTS07632 Cc1cc(n(n1)c2ccccc2)NC(=O)c3ccc(cc3)Cl HTS07633 CCOC(=O)Cn1cnc2c(c1=O)nnn2Cc3ccc(cc3)Cl HTS07634 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccccc4 HTS04240 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cc(nn4C)C(C)(C)C HTS04241 CCOC(=O)COc1c(c(cc(n1)c2ccccc2)c3ccccc3)C#N HTS07545 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccc(cc3)Cl)c4ccccc4)N HTS07547 Cc1cc(nc2c1c(c(o2)C(=O)c3ccc(cc3)Cl)N)c4ccccc4 HTS07548 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2Cl)Cl)C(=O)Nc3nnc(s3)C4CC4 HTS08166 COc1cccc(c1)/C=N/NC(=O)c2cnn(c2N)c3ccccc3 HTS07443 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)NNC(=S)Nc5ccc(cc5)Cl)N HTS07471 Cc1ccc(cc1)n2c(=O)c3c(c4c(c(nnc4s3)c5ccccc5)c6ccccc6)[nH]c2=O HTS07473 CCc1ccnc(c1)NS(=O)(=O)c2cccs2 HTS05386 CN(C1CCCCC1)S(=O)(=O)c2ccccc2 HTS08356 c1cc(c(c(c1)Cl)C(=O)Nc2ccc(cc2)N3CCCCC3)F HTS08410 CN1CCN(CC1)Cc2nc(no2)/C=C/c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04864 Cc1cc(c2cc([nH]c2c1)C(=O)N(Cc3ccccc3)Cc4ccccn4)C HTS07810 c1ccc(cc1)C(=O)N(Cc2cccnc2)Cc3ccc(cc3Cl)Cl HTS07399 c1cc(cnc1)CN(Cc2ccc(cc2Cl)Cl)C(=O)c3cccs3 HTS07401 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)N3CCCCC3 HTS06979 c1ccc(cc1)c2c3c(nc(c2C#N)N)CCCC3 HTS07556 Cc1c(c(=O)n2c3ccccc3[nH]c2c1C#N)CCO HTS07558 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(cc3)N4CCCCC4)Cl HTS08403 c1cc(ccc1C(=O)Nc2ccc(cc2)N3CCCCC3)F HTS08406 Cc1cc(no1)C(=O)Nc2ccc(cc2)N3CCCCC3 HTS08409 c1ccc(cc1)n2c(c(cn2)C(=O)N/N=C/c3ccc(cc3)Cl)N HTS07446 COc1cccc(c1)/C=N/n2cnc3c(c2=O)cnn3c4ccccc4 HTS07450 Cc1c(sc(n1)c2cnccn2)C(=O)N3CCc4cc(c(cc4C3C)OC)OC HTS07812 C=CCn1c(nnc1SCC(=O)NNC(=S)Nc2ccccc2)c3ccccc3 HTS07457 c1cc(c(c(c1)Cl)C(=O)NNc2cc(ccc2Cl)Cl)F HTS02920 CC(C)(CC(=O)Nc1ccc2c(c1)C(=O)OC2)CC(=O)O HTS02924 CCc1ccc(cc1)C(=O)NNc2cc(ccc2Cl)Cl HTS02932 CCOC(=O)C1CCN(CC1)C(=O)c2c(c(cs2)S(=O)(=O)c3ccc(cc3)Cl)C HTS06684 Cc1ccc(cc1)S(=O)(=O)CCSCc2csc3c2cccc3 HTS05337 COc1ccc(c(c1)S(=O)(=O)c2ccc(cc2)Br)OC CD05141 c1ccc(cc1)n2c3c(cn2)c(=O)n(cn3)/N=C/c4ccc(cc4)Cl HTS07453 c1ccc(cc1)n2c3c(cn2)c(=O)n(cn3)/N=C/c4ccc(cc4)[N+](=O)[O-] HTS07454 Cc1cc(c2cc([nH]c2c1)C(=O)NCCSCc3c(cccc3Cl)F)C HTS07811 c1cc(ccc1C(F)(F)F)NC(=O)Nc2ccc(cc2)S(=O)(=O)N HTS07181 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)Nc3csc4c3cccc4 HTS07208 c1cc(sc1)c2ccc(s2)C(=O)O CC14601 c1cc(cc(c1)Cl)NC(=S)Nc2c(cc(cc2F)Br)F CD05074 c1c(cc(c(c1F)NC(=S)N2CCOCC2)F)Br CD05075 COc1ccc(c(c1)S(=O)(=O)c2ccc(cc2)[N+](=O)[O-])OC CD05143 CCc1cccc(c1NC(=O)N(C)C2CCCCC2)C HTS08343 CN(C1CCCCC1)C(=O)Nc2ccc(cc2)OC(F)(F)F HTS08347 Cc1c(c(c(o1)C)S(=O)(=O)Nc2c(c(nn2C)C(F)(F)F)c3ccccc3)C(=O)OC HTS04778 CCc1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)N HTS08348 c1cc(c(cc1Cl)Cl)n2c(=O)c3c4c(sc3[nH]c2=S)CCCC4 HTS07641 CCOC(=O)C(C(=O)C)Sc1nc2c(c3c(s2)CCCC3)c(=O)n1C HTS07642 c1cc2c(c(c1)F)c(=O)[nH][nH]2 HTS01520 CCC1(c2ccccc2NC(O1)c3ccc(cc3)[N+](=O)[O-])c4ccccc4 HTS01521 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)OC(=O)c4c(onc4c5ccccc5)C HTS08501 Cc1ccc2c(c1)n(c(=O)o2)CC/C(=N/OC(=O)c3cccs3)/N HTS07394 Cc1c2c(c(s1)N)c(=O)n(nc2C(=O)OC)c3ccccc3 HTS08471 Cc1c(snn1)C(=O)NNS(=O)(=O)c2cccs2 HTS07765 COC(=O)C1C(=CC(=NN1c2ccccc2)C(=O)c3cccs3)C(=O)OC HTS06862 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)n3cccc3)C HTS07789 C=CCn1c(nnc1SCc2nnc(n2c3ccccc3)SCC(=O)c4ccc(cc4)Cl)c5ccccc5 HTS07462 c1ccc(cc1)CN2CCN(CC2)Cc3cccc(c3)C(=O)N4CCC(CC4)O HTS04083 Cc1c2c([nH]n1)OC(=C(C2c3cccnc3)C#N)N HTS07496 C=CCn1c(n[nH]c1=S)CN2c3ccccc3Sc4c2cccc4 HTS07498 c1ccc2c(c1)N(c3ccccc3S2)Cc4n[nH]c(=S)n4c5ccc(cc5Cl)Cl HTS07500 Cc1c(c(no1)c2ccccc2)C(=O)NCCN(C)C HTS08218 Cc1c(c(no1)c2ccccc2)C(=O)NCCN3CCOCC3 HTS08220 CC(=O)Nc1cc(nn(c1=O)c2ccccc2)C(=O)c3ccc(cc3)Cl HTS08473 COC(=O)C1C(=CC(=NN1c2ccccc2)C(=O)c3ccccc3)C(=O)OC HTS08474 CCc1c2c([nH]n1)OC(=C(C2c3ccccc3)C#N)N HTS08476 Cc1cc2ncc(c(n2n1)c3cccs3)/N=N/c4ccc(cc4)Cl HTS06863 Cc1c(c(c(o1)C)S(=O)(=O)N(C)C2CCCCC2)C(=O)OC HTS08357 CN(C1CCCCC1)S(=O)(=O)c2ccc(o2)C(=O)OC HTS08358 Cc1c(cc(o1)S(=O)(=O)N(C)C2CCCCC2)C(=O)OC HTS08359 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)Nc3ccccc3N4CCOCC4)C(F)(F)F HTS07222 CC1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4cccc(c4)C(F)(F)F)C1 HTS07654 CCOC(=O)c1c2c(sc1NC(=O)Nc3cccc(c3)Cl)CC(CC2)C HTS07657 CSc1ccc(cc1NC(=S)Nc2ccccc2)C(F)(F)F CD05851 c1ccc2c(c1)c(=O)n(c(n2)C(=O)N3CCCC3)N CD05864 CN(C1CCCCC1)C(=O)Nc2ccccc2 HTS07906 CN(C1CCCCC1)C(=O)Nc2cc(cc(c2)Cl)Cl HTS07907 Cc1ccc(cc1)C(=O)C/C(=C\C(=C/2\C(=O)N=C(S2)N3CCOCC3)\c4ccc(cc4)C)/c5ccc(cc5)Cl HTS05456 Cc1ccc(cc1)n2c(nnn2)c3cnc4cc(ccc4c3N)Cl HTS05458 Cc1ccc(cc1)n2c(nnn2)c3cnc4ccc(cc4c3c5ccccc5)Cl HTS05460 c1ccc2c(c1)[nH]c(n2)Sc3c4c(nc5n3ncn5)CCC4 HTS07595 c1ccc(cc1)n2c3c(cn2)c(ncn3)Nc4cccc(c4)C(F)(F)F HTS07597 Cc1cc(no1)C(=O)Nc2c(c(nn2C)C(F)(F)F)c3ccccc3 HTS04776 CN(C)C(=S)SCC(=O)c1ccc(cc1)Cl CD06384 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)N/N=C/c4ccc(cc4Cl)Cl HTS07509 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC#N HTS07512 CC1CCc2c(sc3c2c(ncn3)S)C1 HTS07677 Cc1ccc2c(c1)n(c(=O)o2)CCc3nc(on3)c4cccs4 HTS07398 Cc1cc(cc(c1)NC(=O)Nc2ccccc2N3CCCCC3)C HTS08446 Cc1c(snn1)C(=O)Nc2ccccc2N3CCCCC3 HTS08451 CS/C(=C(/C#N)\C(=O)c1ccco1)/Nc2ccc(cc2)F CD05268 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCC=CC3 CD05282 COC(=O)C1C(=CC(=NN1c2ccccc2)C(=O)c3ccc(cc3)Cl)C(=O)OC HTS06866 CCOC(=O)CN(C)S(=O)(=O)c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)OC HTS07171 c1ccc(c(c1)NC(=S)Nc2ccc(cc2)OC(F)(F)F)N3CCOCC3 HTS07229 c1ccc(cc1)c2c(cn(n2)c3ccccc3)NC(=O)Nc4ccc(cc4F)F HTS03561 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)Nc3cc(oc3C(F)(F)F)C)C HTS06896 c1cc(c(nc1)Oc2c3ccc(cc3ncn2)Cl)NC(=O)c4ccc(cc4)F HTS07327 Cc1c(c(no1)c2c(cccc2Cl)Cl)CSC(=S)N(C)C CD06374 Cc1c(c(c(c(c1C)C)CSC(=S)N(C)C)C)C CD06380 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc(cc2)NC(=O)C HTS07190 Cc1c(c(on1)C)S(=O)(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08271 c1ccc(cc1)n2c3c(cn2)c(ncn3)N4CCN(CC4)c5ccccc5 HTS07600 CC1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4ccc(c(c4)Cl)Cl)C1 HTS07653 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccccc3)CC(CC2)C HTS07655 Cc1cc(c(c(c1)C)n2c(nnc2SCCS(=O)(=O)c3ccc(cc3)F)O)C HTS08009 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(on3)C(C)(C)C HTS03793 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3cc(cnc3)c4cccs4)C HTS06893 CC1=C(C(C2=C(N1)CC(CC2=O)c3ccc(cc3)F)c4ccc(cc4Cl)N(C)C)C(=O)OC HTS03551 COCCOc1ccc(cc1)NC(=O)c2ccc(c(c2)Cl)Cl CD05908 COCCOc1ccccc1NC(=O)c2cc(c(c(c2)OC)OC)OC CD05909 CC(C)N(Cc1ccccc1)C(=O)c2c(cccc2Cl)F HTS07187 c1ccc(cc1)Cn2c3c(c(=O)n(cn3)CC(=O)c4ccc(cc4)Br)nn2 HTS07636 c1cc(ccc1C(=O)O)n2cncn2 CC18601 c1ccc(cc1)C(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS07312 c1ccc(c(c1)C#N)NS(=O)(=O)c2cccs2 HTS08141 c1ccc(c(c1)C#N)NS(=O)(=O)c2ccc(cc2)C(F)(F)F HTS08143 COc1cccc(c1)C(=O)NCCN2CCN(CC2)c3nccc(n3)C(F)(F)F HTS03017 Cc1cc(c2cc([nH]c2c1)C(=O)NCCSCc3ccco3)C HTS07807 CCOC(=O)c1c(n(c(=S)s1)c2ccccc2)NC(=O)C HTS07568 c1cc(c(cc1Cl)Cl)/C=N/NC(=O)CC#N HTS07569 CN(C)C(=S)Nc1c(cc(cc1F)F)F CD05581 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)C(=O)CSCC(=O)O HTS03495 c1ccc(cc1)n2c3c(cn2)c(=N)n(cn3)/N=C/c4ccc(cc4)Cl HTS07542 Cc1ccc(cc1)n2c(=O)c3c(c4c(cc(nc4o3)c5ccccc5)c6ccccc6)[nH]c2=O HTS07543 Cc1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)N HTS08360 c1cc(ccc1NC(=O)c2ccc3c(c2)OCO3)S(=O)(=O)N HTS08361 CCOC(=O)c1cnn(c1N)C(=O)c2c(nns2)C HTS08113 c1ccc2c(c1)c(c(s2)C(=O)N3CCNC(=O)C3CC(=O)Nc4cc(ccc4Cl)Cl)Cl HTS07978 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)Cl)CC(CC2)C HTS07658 CCOC(=O)c1c2c(sc1NC(=O)Nc3cccc(c3)C(F)(F)F)CC(CC2)C HTS07659 CCOC(=O)Cn1cnc2c(c1=O)c3c(s2)CCCC3 HTS07663 Cc1c(csc1C(=O)Nc2nnc(s2)C3CC3)S(=O)(=O)c4ccc(cc4)Cl HTS07890 c1c(cc(c(c1F)NC(=S)N2CCOCC2)F)F CD05577 c1cnc(c(n1)C(=O)NNc2c(cncc2Cl)Cl)C(=O)O HTS03680 CCOC(=O)C1CCN(CC1)CC(=O)c2ccc(cc2)OC HTS07931 Cc1cc(nc2c1c(c(o2)C(=O)N/N=C/c3ccc(c(c3)OC)O)N)c4ccccc4 HTS07539 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4ccccc4)N HTS07546 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS08261 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5ccc(o5)Oc6cc(cc(c6)Cl)Cl HTS08263 c1cnn(c1)c2ccc(cc2)C(=O)NCCN3CCOCC3 HTS07818 CC(C)c1cc(c(c(c1)Br)NC(=O)OCCn2c(=O)c3ccccc3cn2)Br HTS03342 CC1=C(C(n2c(=O)/c(=C\c3ccc4c(c3)OCO4)/sc2=N1)c5ccccc5)C(=O)OC HTS07579 CCOC(=O)c1c(c2c(=O)n(c(=S)n(c2s1)c3ccccc3)c4ccccc4)OC(=O)c5ccco5 HTS07581 C=CCn1c(nnc1SCC(=O)N/N=C/c2cn(nc2c3ccccc3)c4ccccc4)c5ccccc5 HTS07582 c1cc(cnc1)n2c(nnc2SCc3cc(=O)oc4c3ccc(c4)O)O HTS08004 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(cc3)NC(=O)C)C HTS07252 c1ccc(cc1)C2Nc3ccccc3C(=O)N2CCN4CCNC4=O HTS06749 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccccc3 HTS06750 c1ccc2c(c1)nc3n2c(c4c(c3C#N)CCC4)Nc5ccc(cc5)Cl HTS07560 Cc1ccc(cc1C)C(=O)Nc2ccc(cc2)N3CCCCC3 HTS08405 c1ccc(cc1)C(=O)Nc2ccc(cc2)N3CCCCC3 HTS08407 CC(C)N(Cc1ccccc1)C(=O)Nc2ccc(cc2)C(C)(C)C HTS07920 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)N/N=C/c5ccc6c(c5)OCO6)N HTS07466 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C3Cc4ccccc4C3)O HTS08318 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2Cc3ccco3)O HTS08317 C1CCC(CC1)C(=O)N2CCC(CC2)C(=O)O HTS07929 C=CCNC(=S)NNC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4ccccc4)N HTS07549 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)Nc5ccc(cc5)C(C)(C)C)C1=O HTS07749 Cc1cc(n2c3ccccc3nc2c1C#N)N4CCCCC4 HTS07554 c1cc(c(cc1c2csc(n2)N)Cl)Cl HTS07720 c1cc(c(cc1S(=O)(=O)NCCN2CCNC2=O)C(=O)O)O HTS02794 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)NCCN3CCNC3=O HTS02798 C=CCn1c(nnc1SCc2nnc(o2)SCC(=O)c3ccc(cc3)Cl)c4ccccc4 HTS07464 c1ccc(cc1)/C=N/NC(=O)c2c(c3c(c(nnc3s2)c4ccccc4)c5ccccc5)N HTS07465 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(s3)c4cccs4)C#N HTS03162 COc1ccc(cc1OC2CCCC2)NC(=O)N3CCC(CC3)C(=O)O HTS07950 c1cc(sc1)c2ccn3cnnc3n2 HTS08469 Cc1c2c(c(s1)N)c(=O)n(nc2C(=O)OC)c3ccc(cc3)OC HTS08470 c1ccc(c(c1)C(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F)C(=O)O HTS08390 CCc1cccc(c1NC(=O)N(Cc2ccccc2)C(C)C)C HTS08341 CC(C)N(Cc1ccccc1)C(=O)Nc2ccc(cc2)OC(F)(F)F HTS08345 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)N/N=C/c5ccc(cc5Cl)Cl)N HTS07469 Cc1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C(=N/OC(=O)c3ccc(cc3)Cl)/C CD05203 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)c5n[nH]c(=S)n5c6ccccc6)N HTS07482 c1ccc(cc1)S(=O)(=O)n2c3ccccc3cc2CO CC03309 CCN(c1cccc2c1cccc2)C(=O)c3ccccc3 HTS08195 CCOC(=O)C1CCCc2c1c(c(s2)N)C#N HTS07584 Cc1ccccc1NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS07974 CCOC(=O)c1c2c(sc1N)CCCC2C(=O)OCC HTS07585 c1ccc(cc1)N2CCN(CC2)c3c4c(nc5n3ncn5)CCC4 HTS07587 c1ccc(cc1)C(=O)Nc2c(cc(cc2Br)Br)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS01518 CC(=O)N(c1ccc(cn1)NS(=O)(=O)c2ccccc2)S(=O)(=O)c3ccccc3 HTS07703 C=CCn1c2c(c(ncn2)N/N=C/c3ccco3)sc1=S HTS07563 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2c3cccnc3)O HTS08316 CCOC(=O)C1CCN(CC1)C(=O)Nc2c(onc2c3ccccc3)C HTS07372 c1ccc(cc1)n2c(c(cn2)C(=O)NNC(=S)Nc3ccc(cc3)Cl)N HTS07440 c1ccc(cc1)/C=N/NC(=O)c2cnn(c2N)c3ccccc3 HTS07442 CCOC(=O)C1CCN(CC1)c2ccccc2C3C4=C(CCCC4=O)NC(=C3C(=O)OCC)C HTS03154 CC(=O)c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3cccc(c3)C#N HTS06270 CC(C)(C)c1ccccc1NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)F HTS06347 CCC1(c2ccccc2NC(O1)c3cc(cc(c3O)Cl)Cl)c4ccccc4 HTS01522 Cc1c(sc(n1)c2cnccn2)C(=O)N(Cc3ccccc3)Cc4cccs4 HTS05756 Cc1ccn2c(c1)nc(c2C(=O)N/N=C/c3ccc(cc3)OCc4ccccc4)C HTS07419 Cc1c(n2ccccc2n1)C(=O)N/N=C/c3ccccc3Cl HTS07420 CN1CCc2c(sc(c2C#N)N)C1 HTS07422 c1ccc(cc1)c2c3c4c(c(ncn4)SCc5ccc(cc5)Cl)sc3nnc2c6ccccc6 HTS07485 Cc1c2c([nH]n1)OC(=C(C23CCCCC3)C#N)N HTS07486 c1cc(oc1)Cn2c(nnc2SCCS(=O)(=O)c3ccc(cc3)F)O HTS08311 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccc(cc2)OC(F)(F)F HTS08080 CC(=O)N(c1ccc(cn1)NS(=O)(=O)c2ccc3c(c2)CCO3)S(=O)(=O)c4ccc5c(c4)CCO5 HTS07705 Cc1cc(c(nc1)NS(=O)(=O)c2ccc(cc2)Cl)Br HTS00129 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)C)CN(CC2)C HTS02981 Cc1cc(c2cc([nH]c2c1)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F)C HTS06807 Cc1c(n2ccccc2n1)C(=O)NNC(=O)Nc3ccccc3 HTS07416 Cc1c(n2ccccc2n1)C(=O)N/N=C/c3ccccc3 HTS07417 c1ccc(cc1)COc2ccc(cc2)/C=N/n3cnc4c(c3=O)cnn4c5ccccc5 HTS07451 Cn1c(nnc1SCC(=O)NNC(=S)NCC=C)c2ccccc2 HTS07455 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)c5ccc(cc5)Cl)N HTS07479 C=CCn1c(n[nH]c1=S)c2c(c3c(c(nnc3s2)c4ccccc4)c5ccccc5)N HTS07480 Cc1cc(c(o1)C(F)(F)F)NC(=O)Nc2ccccc2Oc3ccccc3 HTS06588 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3ccccc3Oc4ccccc4 HTS06589 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)COc3ccc(cc3Cl)Cl)C HTS06880 Cc1c2ccccc2sc1CN3CCN(CC3)Cc4ccccc4 HTS06964 Cn1c(nnc1SCC(=O)N/N=C/c2ccc3c(c2)OCO3)c4ccccc4 HTS07426 CC(=O)CSc1nnc(n1c2ccccc2)c3ccccc3 HTS07432 c1ccc(cc1)n2c(c(cn2)c3n[nH]c(=S)n3c4ccc(cc4Cl)Cl)N HTS07435 c1ccc(cc1)c2ccc(cc2)C3=CS/C(=C(/C#N)\c4[nH]c5ccccc5n4)/N3c6ccccc6 HTS07519 CCOC(=O)c1c(c(c(s1)Nc2ccccc2)c3[nH]c4ccccc4n3)N HTS07520 Cc1c(c(no1)c2ccccc2)C(=O)NC3CCCCC3NC(=O)c4c(onc4c5ccccc5)C HTS08211 CCCc1c(cnn1c2ccccc2)C(=O)Nc3nc(c(s3)C)c4ccc(c(c4)Cl)C HTS06879 Cn1c(nnc1SCC(=O)N/N=C/c2ccc(cc2)OCc3ccccc3)c4ccccc4 HTS07427 Cn1c(nnc1SCC(=O)NN)c2ccccc2 HTS07430 C=CCn1c(nnc1SCC(=O)NN)c2ccccc2 HTS07431 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)NNC(=O)Nc4ccc(cc4)Cl HTS07513 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)CCCC(=O)O HTS08515 CNC(=S)NNC(=O)c1cnn(c1N)c2ccccc2 HTS07436 CN(C1CCCCC1)S(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 HTS07909 CN(C1CCCCC1)S(=O)(=O)c2ccc(s2)c3ccccn3 HTS07911 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccccc3NC(=O)c4c(onc4c5ccccc5)C HTS08213 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(ccc3N4CCCC4)C(F)(F)F HTS08216 c1nc(c2c3c(sc2n1)CCCC3)S HTS07678 c1cc(ccc1NC(=O)Nc2ccc(cc2F)F)N3CCCCC3 HTS06974 C=CCNC(=S)NNC(=O)c1cnn(c1N)c2ccccc2 HTS07437 CC(C)N(Cc1ccccc1)C(=O)Nc2cc(cc(c2)Cl)Cl HTS07905 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCNC(=O)C3CC(=O)Nc4cc(ccc4Cl)Cl HTS07965 c1cnn(c1)c2ccc(cc2)C(=O)Nc3ccc(cc3)N4CCOCC4 HTS07814 CC1=C(C(C2=C(N1)CC(CC2=O)c3ccco3)c4ccc5c(c4)OCO5)C(=O)OC HTS04695 CC1=C(C(C2=C(N1)CC(CC2=O)c3ccco3)c4ccc5c(c4)CCO5)C(=O)OC HTS04698 CS/C(=C(/C#N)\C(=O)c1cccs1)/Nc2cccc(c2Cl)Cl CD05239 c1cc(ccc1CO)n2cncn2 CC18609 CC(C)(CC(=O)N1CCN(CC1)c2nc3cc(ccc3s2)Cl)CC(=O)O HTS03283 Cn1cnc(c1Sc2cccc(c2)C(F)(F)F)[N+](=O)[O-] HTS03860 COc1cc(ccc1O)C2c3c(c4ccccc4oc3=O)OC(=C2C#N)N HTS07628 c1cc2c(cc1CNS(=O)(=O)c3cc(sc3Cl)Cl)OCO2 HTS03964 Cc1c(c(no1)c2ccccc2)C(=O)CN3CCN(CC3)c4nc5cc(ccc5s4)Cl HTS03292 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)NS(=O)(=O)C HTS04777 CCOc1ccccc1NC(=O)Nc2cc(ccc2C)S(=O)(=O)N(C)C HTS05239 c1ccc(cc1)/N=C(/C(C#N)c2[nH]c3ccccc3n2)\SCc4ccc(cc4)Cl HTS07507 c1ccc(cc1)c2nnc(n2c3ccccc3)Sc4c5c6c(sc5ncn4)CCCC6 HTS07679 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCC(=O)c3ccccc3 HTS01519 Cc1cc(c2cc([nH]c2c1)C(=O)N3CCc4ccccc4C3)C HTS07808 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3)N4CCOCC4 HTS03569 Cc1cc(c2cc([nH]c2c1)C(=O)N3CCc4cc(c(cc4C3C)OC)OC)C HTS07809 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3cccnc3Oc4ccccc4)C HTS06891 c1cnn(c1)c2ccc(cc2)C(=O)NCc3ccncc3 HTS07816 c1ccc2c(c1)CCN(C2)C(=O)c3ccc(cc3)n4cccn4 HTS07817 c1ccc(c(c1)C#N)NC(=O)CCCC(=O)O HTS07790 Cc1c(c(on1)C)S(=O)(=O)NC2Cc3ccccc3C2 HTS05950 c1ccc(c(c1)N2CCOCC2)OC(=O)c3cccs3 HTS03574 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCc2ccc3c(c2)OCO3 HTS03579 Cc1ccc(cc1C)OCC(CN2CCN(CC2)Cc3ccc4c(c3)OCO4)O HTS04127 c1cc(sc1)c2nc(cs2)C(=O)Nc3ccc4c(c3)OCCO4 HTS06888 c1cc(sc1)c2cc(cnc2)C(=O)Nc3ccc4c(c3)OCCO4 HTS06889 c1ccnc(c1)c2nc(on2)CCC(=O)NCc3ccc4c(c3)OCO4 HTS07819 CC(C)N(Cc1ccccc1)C(=O)c2ccc(cc2F)F HTS07188 Cc1cc(ccc1NNC(=O)c2c(cccc2Cl)F)Cl HTS03651 Cc1cc(n(n1)c2ccccc2)NC(=O)Nc3ccc(cc3)Cl HTS07630 c1cc(ccc1NC(=O)c2ccc(cc2Cl)Cl)N3CCCCC3 HTS08413 c1cc(ccc1NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)N3CCCCC3 HTS08415 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)NC(=O)c3ccccc3O)C HTS08230 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=O)Nc3ccc(cc3F)F)O HTS08232 c1ccc(cc1)C(=O)Nc2ccc(cc2)NC(=O)c3ccccc3O HTS08236 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=O)c3ccc(cc3F)F)O HTS08239 COc1ccc(cc1NC(=O)Nc2ccc(cc2)N3CCCCC3)Cl HTS06975 c1cc(ccc1NC(=O)Nc2ccc(cc2)OC(F)(F)F)N3CCCCC3 HTS06977 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3csc(n3)c4cccs4)C HTS06892 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)Nc3c(onc3c4ccccc4)C)C HTS06895 c1ccc2c(c1)c(cc3c2occ3C(=O)c4ccc(cc4)Cl)O HTS08467 c1ccc(cc1)CN(Cc2ccccc2)c3c4c(nc5n3ncn5)CCC4 HTS07589 CCCc1ccc(cc1)C(=O)NNc2ccc(cc2C)Cl HTS03654 Cc1cc(ccc1NNC(=O)c2c(nns2)C)Cl HTS03656 Cc1cc(ccc1NNC(=O)C2CCC2)Cl HTS03659 CC1CCc2c(sc3c2c(=O)[nH]cn3)C1 HTS07660 CC(C)(C)c1cc(no1)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS07313 CC(C)(C)c1cc(no1)NC(=O)Nc2ccccc2 HTS07314 COc1cccc(c1)C(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F HTS08385 c1ccc(cc1)C(CC(=O)O)CC(=O)Oc2ccccc2N3CCOCC3 HTS06428 c1cc(cc(c1)[N+](=O)[O-])c2csc(n2)c3ccc4c(c3)OCO4 HTS03335 CC(=O)Nc1cccc(c1)OCCCNS(=O)(=O)c2cccc(c2)Cl HTS02714 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=O)Nc3ccc(cc3)F)O HTS07970 Cc1c(snn1)C(=O)NNC(=O)C2CCCCC2 HTS08110 CCc1cc(c(s1)N)C(=O)c2ccc(cc2)OC HTS08114 Cc1cc(c(o1)C(F)(F)F)NC(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl HTS08293 Cc1c(cn(n1)c2ccccc2)/C=N/Nc3c4cnn(c4ncn3)c5ccccc5 HTS07607 c1cc(c(nc1)N2CCN(CC2)C(=O)c3ccc(s3)c4cccs4)C(F)(F)F HTS08523 CCCc1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc4c(c3)CCO4 HTS03297 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCc2ccc3c(c2)OCO3 HTS03969 Cc1ccc(cc1Cl)NC(=O)Nc2ccccc2N3CCCCC3 HTS08444 Cc1ccccc1NC(=O)Nc2ccccc2N3CCCCC3 HTS08445 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccccc3Cl HTS08632 c1cc(oc1C(=O)N2CCC(CC2)C(=O)N)Oc3cc(cc(c3)Cl)Cl HTS08733 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08769 Cc1c(c(on1)C)S(=O)(=O)NNC(=O)c2c(nns2)C HTS07767 Cc1cc2nccc(n2n1)c3ccc(cc3)Cl HTS06864 Cc1cccc(c1C)C(=O)N(Cc2ccccc2)C(C)C HTS07895 CN(C1CCCCC1)C(=O)c2ccc(cc2)OC(F)(F)F HTS07897 c1cc2c(cc1Cl)ncnc2Oc3ccc(cn3)NC(=O)COCC(=O)O HTS08301 Cc1ccc2c(c1)n(c(=O)o2)CCC(=O)Nc3ccccc3N4CCCCC4 HTS07983 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3c(cccc3Cl)Cl)\N4CCCC4 CD06035 Cc1csc(c1c2nc3ccccc3s2)NC(=O)CSCC(=O)O HTS03494 Cc1ccccc1NC(=O)Nc2cc3ccccc3s2 HTS03761 CCOC(=O)CS/C(=N\c1ccccc1)/c2c(onc2c3c(cccc3Cl)Cl)C CD06242 c1ccc(cc1)CN2CCN(CC2)CC(=O)Nc3ccccc3Oc4ccccc4 HTS06594 CCOC(=O)C1=C(Oc2c3ccccc3oc(=O)c2C1c4ccccc4Cl)N HTS07617 CCOC(=O)C1=C(Oc2c3ccccc3oc(=O)c2C1c4ccc(cc4)[N+](=O)[O-])N HTS07619 Cc1cc(n(n1)c2ccccc2)NC(=O)Nc3cccc(c3)C(F)(F)F HTS07631 CCOC(=O)C1CCN(CC1)C(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS06686 CCOC(=O)Cc1csc(n1)NC(=O)Nc2cccs2 HTS08072 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccccc2 HTS08073 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3c4ccc5c(c4)OCCO5)O HTS07999 c1ccc(c(c1)N2CCOCC2)OC(=O)c3c(ccs3)Br HTS03600 Cc1c(snn1)c2nnc(o2)c3cccc4c3cccc4 HTS07932 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN(C)c3ccc(cc3[N+](=O)[O-])C(F)(F)F CD06996 CC1CN(CC(O1)C)c2ccc(cc2C(=O)O)NC(=O)c3ccco3 CD07017 CC(C)(C)c1cc(no1)NC(=O)Nc2ccccc2OC(F)(F)F HTS07953 CCOc1ccccc1NC(=O)Nc2cccc(c2)C(=O)O HTS03987 Cc1c(c(c(c(c1C)C)/C=N/OC(=O)c2c(onc2c3c(cccc3Cl)Cl)C)C)C CD06103 CCOC(=O)C1CCN(CC1)C(=O)Nc2ccc(cc2F)F HTS07922 CCOC(=O)C1CCN(CC1)C(=O)Nc2ccc(cc2)F HTS07924 C(C(=O)Nc1nnc(s1)C(F)(F)F)OCC(=O)O HTS08615 c1ccc2c(c1)c(c[nH]2)CCNC(=O)/C(=C/c3c(cccc3Cl)Cl)/C#N CD06579 c1cc(ccc1C2CCCCC2)NC(=O)CN3CCN(CC3)c4nc5cc(ccc5s4)Cl HTS03278 c1cc(ccc1NC(=O)C2CCCCC2)S(=O)(=O)N HTS07182 CN(c1cccc(c1C#N)F)NC(=O)c2ccccc2Cl CD07022 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nnc(s3)NC(=O)Nc4c(onc4c5c(cccc5Cl)Cl)C CD05828 Cc1c(csc1C(=O)Nc2ccc3c(c2)OCCO3)S(=O)(=O)c4ccc(cc4)Cl HTS06890 C=CCn1cnc2c(c1=O)nnn2Cc3ccc(cc3)F HTS07637 c1ccc(c(c1)Cn2c3c(c(=O)n(cn3)Cc4ccc(cc4)[N+](=O)[O-])nn2)Cl HTS07638 c1ccc(cc1)C(=O)C2C(N=C(N2)N)c3ccc(cc3)Cl HTS07933 c1ccc(cc1)c2cc(nc3c2c(c(o3)C(=O)N/N=C/c4ccc(cc4)Cl)N)c5ccccc5 HTS07540 c1ccc(cc1)c2cc(nc3c2c(c(o3)C(=O)N/N=C/c4cccs4)N)c5ccccc5 HTS07541 CC(c1ccccc1)n2c(nnc2S)O HTS07403 c1ccc(cc1)SCC(=O)NCc2ccc3c(c2)OCO3 HTS04243 CCN(CC)C(=S)Oc1ccc(cc1C(=O)Nc2ccc(cc2F)F)Br CD07070 CCN(CC)C(=S)Oc1ccc(cc1C(=O)Nc2ccc(c(c2)Cl)F)Br CD07074 c1ccc(c(c1)NC(=O)c2ccco2)N3CCCCC3 HTS08449 CN(C)c1ccc(cc1)NC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05893 Cc1c(cnn1c2ccc(cc2)F)C(=O)Nc3ccc(cc3)F HTS06783 c1ccc(cc1)NC(=O)CSc2nnc(n2C3CC3)O HTS08647 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccccc3OC)OC HTS03826 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccc(cc3Cl)Cl)OC HTS03827 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccccc2 HTS07191 c1ccc(c(c1)c2ccccc2C(=O)O)C(=O)NCCN3CCNC3=O HTS03375 C1CN(C(=O)N1)CCN2CCS(=O)(=O)CC2 HTS03386 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N(Cc3ccccc3)C(C)C HTS07197 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccccc3N4CCCCC4 HTS08454 c1ccc(c(c1)NC(=O)C2CCCCC2)N3CCCCC3 HTS08455 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)NS(=O)(=O)c3ccc(cc3)Cl HTS07826 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc(cc3)NC(=O)c4ccccc4O HTS07969 c1cc(ccc1NS(=O)(=O)c2cc(cc(c2)Cl)Cl)N3CCCCC3 HTS06990 Cc1ccc(cc1C)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccsc3C(=O)OC HTS07307 c1cc(ccc1F)SCC(=O)NCc2ccc3c(c2)OCO3 HTS04244 CC1=C(C(C2=C(N1)CCCC2=O)c3c[nH]nc3)C(=O)OC HTS03554 c1ccc(cc1)c2cc(n3c4ccccc4nc3c2C#N)Nc5ccc(cc5)Cl HTS07555 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)N3CCCCC3 HTS08411 c1cc(oc1C(=O)N2CCCCC2)Oc3cc(cc(c3)Cl)Cl HTS08460 c1cc(cnc1)CNC(=O)c2ccc(s2)c3cccs3 HTS08525 c1cc([nH]c1)CN2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F HTS08528 CN(C)c1ccc(cc1)CN2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F HTS07829 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)NC(=O)c3ccccc3O HTS07968 CC(C)(C)C1=C(C(C(=C(O1)NC(=O)NC(=O)c2c(cccc2Cl)F)C#N)c3cccs3)C#N CD06692 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)Nc3ccccc3 HTS08507 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(nc2)Oc3ccc(cc3)C(C)(C)C HTS08510 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)Nc3ccc(cc3)F HTS08511 c1ccc2c(c1)c(c[nH]2)CN3CCc4c(ccs4)C3c5ccc(cc5)OC(F)(F)F HTS08529 Cc1c(snn1)C(=O)NNC(=O)c2ccc(cc2)F HTS08109 c1ccc(cc1)CN2CCc3c(sc(c3C(=O)c4ccc(cc4)Cl)N)C2 HTS08120 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)Nc3ccc(cc3)N4CCCCC4 HTS06984 Cc1c2c([nH]n1)OC(=C(C2c3ccccc3Cl)C#N)N HTS07492 c1ccc(cc1)c2cc(=O)n3c4ccccc4[nH]c3c2C#N HTS07559 Cc1c2c(n3c4ccccc4nc3c1C#N)SCC2 HTS07562 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccc(cn2)C(F)(F)F HTS08584 c1cc(ncc1C(F)(F)F)NC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F HTS08585 Cc1c(snn1)C(=O)NNC(=O)c2ccc(cc2)OC HTS08111 COc1ccc(cc1)C(=O)c2c3c(sc2N)CN(CC3)Cc4ccccc4 HTS08115 CCOC(=O)N1CCc2c(sc(c2C(=O)c3ccc(cc3)OC)N)C1 HTS08118 c1cc(c(c(c1)F)C#N)N(Cc2cccnc2)C(=S)Nc3ccc(c(c3)Cl)Cl CD05668 CN(CC(=O)O)c1ncc(c(n1)c2ccccc2Cl)c3nnnn3c4ccccc4 HTS06856 CS(=O)(=O)Cc1cc(cc2c1OCOC2)Cl CD06096 c1ccc(c(c1)CN2CCCC2)c3nc(no3)/C=C\c4cc(cc(c4)C(F)(F)F)C(F)(F)F CD06183 Cn1c(nnc1SCC(=O)NNC(=S)NCc2ccccc2)c3ccccc3 HTS07456 c1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)NNC(=S)Nc4ccccc4 HTS07458 Cc1ccccc1CNc2ccc(cc2)S(=O)(=O)Nc3nc(cc(n3)C)C HTS07787 c1ccc(cc1)NC(=O)Nc2ccc(cc2)S(=O)(=O)N HTS07176 Cc1c2c([nH]n1)OC(=C(C2c3ccc(cc3Cl)Cl)C#N)N HTS07494 Cc1c2c([nH]n1)OC(=C(C2c3ccc(cc3)[N+](=O)[O-])C#N)N HTS07495 c1ccc(cc1)CNC(=S)NNC(=O)CN2c3ccccc3Sc4c2cccc4 HTS07502 c1cc(cc(c1)c2nc(no2)/C=C\c3cc(cc(c3)C(F)(F)F)C(F)(F)F)CN4CCCC4 CD06189 c1ccc(cc1)n2c3c(cn2)c(ncn3)Sc4nnc(n4c5ccccc5)c6ccc(cc6)Cl HTS07614 CCOC(=O)C1=C(Oc2c3ccccc3oc(=O)c2C1c4ccc(cc4)OC)N HTS07616 CCOC(=O)C1=C(Oc2c3ccccc3oc(=O)c2C1c4ccc(cc4)Cl)N HTS07618 CC1CCc2c(sc3c2c(=O)n(c(n3)SCC(=O)C)c4ccccc4)C1 HTS07647 CN1CCc2c(sc(c2C(=O)c3ccc(cc3)Cl)N)C1 HTS08121 CCOC(=O)CSc1c2c3c(sc2ncn1)CC(CC3)C HTS07676 CC(=O)CSc1c2c3c(sc2ncn1)CCCC3 HTS07680 c1ccc(cc1)Sc2c3c4c(sc3ncn2)CCCC4 HTS07681 Cc1c(ccc(n1)C(F)(F)F)C(=O)NNc2c(cncc2Cl)Cl HTS03684 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3)OC HTS03537 c1cc(c(cc1Cl)Cl)NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS07973 Cc1cccc(c1)NC(=O)Nc2ccc(cc2)S(=O)(=O)N HTS07179 CCc1c(nnc2n1nc(c2)C)C(=O)OC HTS08468 Cc1ccc(cc1)n2c(nnn2)c3c[nH]c4c3ccc(c4)Cl HTS06844 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)Nc3nnc(s3)C4CC4)Cl HTS03438 COc1ccc(cc1)C(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS03445 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(C)N CD06972 Cc1c2c(c(c(=O)[nH]c2n(n1)c3ccccc3)C#N)c4ccc(cc4)OC HTS07621 Cc1c2c(c(c(=O)[nH]c2n(n1)c3ccccc3)C#N)c4cccs4 HTS07624 CCCCc1ccc(cc1)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03691 Cc1c(snn1)C(=O)NCCc2c[nH]c3c2cccc3 CD06524 c1ccc(cc1)CN(Cc2ccccc2)c3c4cnn(c4ncn3)c5ccccc5 HTS07598 c1ccc(cc1)NC(=S)NNC(=O)CN2c3ccccc3Sc4c2cccc4 HTS07503 CC1CCc2c(sc3c2c(=O)n(cn3)CC(=O)N/N=C/c4ccc(cc4)Cl)C1 HTS07671 c1ccc(cc1)NC(=O)Nc2ccc(cc2)NC(=O)c3ccccc3O HTS07967 Cc1ccc(cc1NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl)F HTS07971 c1cc2c(cc1C(=O)CN3CCN(CC3)c4nc5cc(ccc5s4)Cl)OCCO2 HTS03288 c1cc2c(cc1C(=O)CN3CCN(CC3)c4nc5cc(ccc5s4)Cl)OCCCO2 HTS03289 c1cc(ccc1NC(=O)Nc2nnc(s2)C3CC3)F HTS03436 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN(C)c3ccc(cn3)[N+](=O)[O-] CD06969 CCc1ccc(cc1)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03269 CN1CCC(CC1)N(C)C(=O)c2cc3cc(ccc3[nH]2)OC HTS03466 c1ccc(c(c1)C(F)(F)F)n2c(nnc2SCCS(=O)(=O)c3ccc(cc3)F)O HTS04171 Cc1cc(c(nc1)NC(=O)c2ccc(cc2)Cl)Br HTS03506 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cccc(c4)Cl HTS04242 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3cccc(c3)Cl HTS08634 c1ccc(c(c1)C(=O)Nc2ccc(cn2)C(F)(F)F)C(=O)O HTS08593 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)S(=O)(=O)c5ccc(s5)CNC(=O)c6ccc(cc6)Cl HTS08770 c1cc(oc1C(=O)Nc2nnc(s2)C3CC3)Oc4cc(cc(c4)Cl)Cl HTS08749 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)CSCC(=O)O)C(F)(F)F HTS08395 CC(=O)N(c1ccc(cn1)NS(=O)(=O)c2cccs2)S(=O)(=O)c3cccs3 HTS07704 CCCc1c(cnn1c2ccccc2)C(=O)N(Cc3ccccc3)Cc4cccs4 HTS03522 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)S(=O)(=O)c3ccc(cc3)C(F)(F)F HTS03617 Cc1c(csc1C(=O)N(C)c2nnc(s2)C(F)(F)F)S(=O)(=O)c3ccc(cc3)Cl HTS03176 c1cc(cc(c1)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)C(F)(F)F HTS03263 Cc1ccc(cc1)n2c(nnn2)c3cnn(c3C(F)(F)F)c4cccc(c4)F HTS05452 c1cc(cc(c1)F)n2c(c(cn2)c3nnnn3c4ccc(cc4)Cl)C(F)(F)F HTS05453 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)S(=O)(=O)c5cccc6c5nsn6 HTS08276 CCOC(=O)CSc1c2cnn(c2ncn1)c3ccccc3 HTS07611 c1ccc(cc1)n2c3c(cn2)c(ncn3)N/N=C/c4ccco4 HTS07602 c1ccc(cc1)n2c3c(cn2)c(ncn3)N/N=C/c4cccs4 HTS07603 c1cc(ccc1C(=O)Cn2cnc3c(c2=O)c4c(s3)CCCC4)Br HTS07662 CCCc1c(cnn1c2ccccc2)C(=O)NCCCn3ccnc3 HTS03538 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3F)F HTS03784 CCCc1c(cnn1c2ccccc2)C(=O)NCc3ccncc3 HTS03792 Cc1c(snn1)C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05353 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)ONC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD05392 c1ccc2c(c1)cccc2NC(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 HTS03698 Cc1ccc(cc1)C2=NN=C(C=C(C2)c3ccc(cc3)Cl)c4ccc(cc4)C HTS05455 Cc1ccc(cc1)n2nnnc2/C=C/N(CCN(/C=C/c3n(nnn3)c4ccc(cc4)C)C)C HTS05440 c1ccc(cc1)S(=O)(=O)NCc2ccc3c(c2)OCO3 HTS03968 c1cc2cccnc2c(c1)S(=O)(=O)NCc3ccc4c(c3)OCO4 HTS03975 CN(C)c1ccc(cc1)/C=C(/C#N)\C(=O)O CD05531 CC1=NCCN1CCNC(=O)Nc2ccc(cc2)C(C)(C)C HTS08021 CN1CCN(CC1)C(=O)CCc2nc(no2)c3ccccn3 HTS07821 c1ccc(cc1)S(=O)(=O)Nc2nnc(s2)C3CC3 HTS08185 c1ccnc(c1)c2ccc(s2)C(=O)CN3CCN(CC3)c4nc5cc(ccc5s4)Cl HTS03291 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS08278 c1cc(ccc1NC(=O)c2ccc(cc2Cl)F)N3CCCCC3 HTS08416 CCOC(=O)CC(=O)c1ccc(cc1)[N+](=O)[O-] BTB10449 Cc1c(c(no1)c2ccccc2)C(=O)NNC(=O)c3nc(no3)c4cccs4 HTS08322 c1cc2c(cc1NC(=O)c3c(nccn3)C(=O)O)C(=O)OC2 HTS02926 c1ccc(cc1)S(=O)(=O)Nc2ccccc2C#N HTS08144 Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc(cc3)S(=O)(=O)N HTS08362 c1cc(sc1)c2nc(on2)CN3CCC(CC3)C(=O)N HTS03627 c1c(c(sc1Cl)S(=O)(=O)NN2CCOCC2)Br HTS03662 c1ccc(cc1)NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS08731 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS08294 COc1ccc(cc1OC2CCCC2)NC(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS08296 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc(s3)c4cccs4 HTS08521 c1cc(sc1)c2ccc(s2)C(=O)N3CCC(CC3)C(=O)c4ccc(cc4)F HTS08522 CN(C)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)c3csnn3 HTS08630 c1ccc(c(c1)C(=O)Nc2ccc(cc2)N3CCCCC3)Cl HTS08412 CCc1ccc(cc1)C(=O)NNc2ccc(c(c2)Cl)C HTS03638 Cc1c(c(on1)C)S(=O)(=O)N(C)C2CCCCC2 HTS08354 c1cc(ccc1NC(=O)c2ccc(cc2F)F)S(=O)(=O)N HTS08363 Cc1ccc2c(c1)n(c(=O)o2)CCC(=O)NNC(=O)c3nc(no3)c4cccs4 HTS08323 c1ccnc(c1)c2nc(on2)CCC(=O)NCc3ccc(cc3)F HTS08530 c1cc(ccc1NC(=O)c2ccc(cc2F)F)N3CCCCC3 HTS08404 Cc1ccc(cc1C)C(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS07977 c1ccc(cc1)Oc2c(cccn2)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS07936 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc4c(c3)cc[nH]4 HTS08309 CN(C1CCCCC1)S(=O)(=O)c2ccc3ccccc3c2 HTS08353 c1cc(c(c(c1)F)C#N)NCc2ccc(cc2)Cl CD05690 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cn(nc2c3ccccc3)c4ccccc4 HTS03560 CC1CN(CCN1C(=O)c2csc(n2)c3cccs3)Cc4ccccc4.C(=C/C(=O)O)\C(=O)O HTS07763 c1cc(nc(c1)NCCN2CCNC2=O)C#N HTS03376 c1cc2c(cc1Cl)nc(s2)N3CCN(CC3)C(=O)CSCC(=O)O HTS03285 Cc1ccc2c(c1)n(c(=O)o2)CCC(=O)Nc3ccc(cc3)N4CCOCC4 HTS07982 c1cc(ccc1NS(=O)(=O)c2cc(sc2Cl)Cl)N3CCCCC3 HTS06986 CCC1c2c(c3ccccc3oc2=O)OC(=C1C#N)N HTS07626 COc1ccc(cc1)c2c(nnn2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C#N CD05276 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)N/N=C/c5cccnc5)N HTS07470 c1cc(c(c(c1)Cl)CSc2[nH]c3cc(c(cc3n2)Cl)Cl)F HTS08201 Cc1ccc(cc1Cl)NNC(=O)c2c(onc2c3c(cccc3Cl)F)C HTS03646 Cc1cc(ccc1NNC(=O)c2c(onc2c3c(cccc3Cl)F)C)Cl HTS03871 CN(C1CCCCC1)C(=O)c2ccccc2 HTS07898 Cc1cccc(c1C)C(=O)N(C)C2CCCCC2 HTS07899 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2ccc(cc2)S(=O)(=O)N HTS08368 CCCc1cnc(nc1)N2CCN(CC2)C(=O)c3ccc(cc3)OC HTS03296 COCCOc1ccccc1NC(=O)c2ccc(c(c2)Cl)Cl CD05896 COCCOc1ccc(cc1)NC(=O)c2ccc(cc2)Cl CD05911 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)NNc2c(cncc2Cl)Cl HTS03688 CCc1c(c(=O)n(nc1C(=O)OC)c2ccc(cc2)OC)C#N HTS08465 Cc1cc2ncc(c(n2n1)c3ccc(cc3)Cl)/N=N/c4ccccc4 HTS08466 C/C(=C\C#N)/NC(=O)c1c(nccn1)C(=O)O HTS03387 CCOc1ccc(cc1)NC(=O)c2c(nccn2)C(=O)O HTS03390 c1ccc(c(c1)NC(=O)c2cc(sc2Cl)Cl)N3CCCCC3 HTS08453 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)NNC(=S)Nc5ccc(cc5Cl)Cl)N HTS07472 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)c5ccccc5)N HTS07478 c1ccc(cc1)n2c3c(cn2)c(ncn3)S HTS07609 C=CCSc1c2cnn(c2ncn1)c3ccccc3 HTS07610 c1cc(ccc1CSc2[nH]c3cc(c(cc3n2)Cl)Cl)Cl HTS08203 CCCCCCCNC(=O)c1c(onc1c2c(cccc2Cl)Cl)C CD06798 c1ccc(cc1)c2cc(n(n2)CCC#N)NC(=O)NC(=O)c3c(cccc3Cl)F CD06926 c1cc(ccc1C(=O)Nc2ccc(cc2)N3CCCCC3)Cl HTS08414 COCCOC(=O)c1c(nccn1)C(=O)Nc2ccc3c(c2)OCO3 HTS03722 CCc1ccc(cc1)C(=O)N(Cc2ccccc2)C(C)C HTS07194 CC(C)N(Cc1ccccc1)C(=O)c2cccs2 HTS07196 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc3c(c2)CCO3 HTS07198 c1cnc(nc1C(F)(F)F)N2CCC(CC2)C(=O)N AW01249 Cc1c(c(on1)C)S(=O)(=O)Nc2cccc(c2)CO HTS08046 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(nc3)NC(=O)C HTS06718 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccccc3N HTS08212 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3c(nccn3)C(=O)O HTS03741 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS08270 c1ccc(cc1)n2c3c(cn2)c(ncn3)SCc4ccc(cc4)F HTS07612 Cn1c(nnc1Sc2c3cnn(c3ncn2)c4ccccc4)c5ccccc5 HTS07613 c1ccc(cc1)N\2C(=CS/C2=C(/C#N)\c3[nH]c4ccccc4n3)c5ccc(cc5)Br HTS07518 c1cc(sc1)c2nc(cs2)CN3CCSCC3 HTS07162 Cn1c(cc(n1)c2ccc(cc2)Cl)NC(=O)CSCC(=O)O HTS08048 CC(CO)(CO)NC(=S)Nc1ccc(c(c1)Cl)F CD06979 Cn1cc(nc1)S(=O)(=O)NCc2ccc3c(c2)OCO3 HTS03965 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3)S(=O)(=O)Nc4nc(cc(n4)C)C HTS07781 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc(s2)c3ccccn3 HTS07199 c1cc(sc1)/C=N/NC(=O)Cn2cnc3c(c2=O)c4c(s3)CCCC4 HTS07667 CC1CCc2c(sc3c2c(=O)n(cn3)CC(=O)N/N=C/c4ccco4)C1 HTS07668 CC1CCc2c(sc3c2c(=O)n(cn3)CC(=O)N/N=C/c4cccnc4)C1 HTS07669 Cc1ccc(cc1)C(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F HTS08398 COc1ccc(cc1OC)C(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F HTS08400 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS08279 c1cc(ccc1NC(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl)OC(F)(F)F HTS08290 Cc1cc(ccc1NNC(=O)c2cccs2)Cl HTS03657 Cc1cc(ccc1NNC(=O)c2c(onc2c3ccccc3)C)Cl HTS03660 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)c4ccc(cc4)[N+](=O)[O-] HTS07627 Cc1ccc(cc1)NC(=O)NNC(=O)CSc2nnc(n2CC=C)c3ccccc3 HTS07523 CCOC(=O)C1=C(OC(=C(C12c3ccccc3NC2=O)C(=O)C)C)N HTS07526 Cc1cc(n(n1)c2cc(nc3n2ncn3)c4ccccc4)C HTS07533 CC1CCc2c(sc3c2c(=O)n(cn3)CC(=O)N/N=C/c4ccc(cc4Cl)Cl)C1 HTS07672 Cc1c2c(c(c(=O)[nH]c2n(n1)c3ccccc3)C#N)c4ccccc4 HTS07620 Cn1c(=O)c2c3c(sc2nc1SCc4ccc(cc4)[N+](=O)[O-])CCCC3 HTS07643 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)C#N)N3CCCCC3 HTS08153 Cc1ccc(cc1Cl)S(=O)(=O)Nc2ccccc2N3CCCCC3 HTS08154 Cc1c(c(no1)c2ccccc2)N3C(=O)CCN(C3=O)C(C)C HTS06120 Cc1ccc2c(c1)n(c(=O)o2)CC/C(=N/OC(=O)c3ccc(nc3C)C(F)(F)F)/N HTS07392 Cc1cc(c(c(c1)C)n2c(nnc2SCC(=O)Nc3ccc(cc3)C(C)C)O)C HTS08315 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)F)N3CCCCC3 HTS08432 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3cccc(c3)OC HTS08496 c1ccn(c1)c2nnc(s2)C(C(C(F)(F)F)(F)F)(F)F CD05832 Cc1c(c(no1)c2cccc(c2)[N+](=O)[O-])C(=O)ONC(=O)c3ccccc3 CD05841 CS/C(=N/c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/N2CCCC2 CD06200 c1cc(ccc1c2csc(n2)N3CCCN(CC3)c4nc(cs4)c5ccc(cc5)Cl)Cl HTS06849 Cc1cccc(c1NC(=O)c2ccc(cc2)Cl)C(C)C CD06342 CC1CCc2c(sc3c2c(=O)n(c(n3)SCC(=O)N)c4ccccc4)C1 HTS07648 CC1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4ccccc4)C1 HTS07649 c1ccc(cc1)n2c(nnn2)c3cnn(c3C(F)(F)F)c4ccccc4Cl HTS05454 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3cccn3CCc4ccccn4 HTS01622 CC(C)(C)c1ccc(cc1)NC(=O)Nc2nnc(s2)C3CC3 HTS08175 CCc1ccc(c(c1)NC(=O)Nc2nnc(s2)C3CC3)C HTS08179 CC1CCc2c(sc3c2c(=O)n(cn3)CC(=O)N/N=C/c4ccc(c(c4)OC)O)C1 HTS07674 Cc1c(c(c(o1)C)S(=O)(=O)Nc2ccc(cc2)C(C)C)C(=O)OC HTS01168 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(C)c3nnc(s3)C(F)(F)F HTS06015 CC1CCc2c(sc3c2c(=O)n(c(n3)SC)c4ccccc4)C1 HTS07646 Cc1c(n2ccccc2n1)C(=O)N/N=C/c3ccc(cc3)[N+](=O)[O-] HTS08975 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)Nc3ccc(cn3)C(F)(F)F HTS08587 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccc(c(c3)Cl)F HTS08631 COc1ccc(cc1OC)CCNC(=O)c2nc3ccccc3c(=O)n2NC(=O)Nc4c(cccc4Cl)Cl CD07618 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccc(cc3)OCc4ccccc4 HTS07296 c1ccc2c(c1)cc(s2)C(=O)NNc3cc(ccc3Cl)Cl HTS02919 CCCc1ccc(cc1)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03270 Cn1c(ccc1S(=O)(=O)NCc2csc3c2cc(cc3)Cl)C(=O)OC HTS03897 c1cc2c(cc1S(=O)(=O)NCc3csc4c3cc(cc4)Cl)CCO2 HTS04201 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)NCc3csc4c3cc(cc4)Cl)C#N HTS03900 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(nc2)N3CCN(CC3)C(=O)OC(C)(C)C HTS07827 Cc1c(c(n(n1)C(=O)c2ccc(cc2)Cl)C)Br CD07237 CC(C)c1ccc(cc1)NC(=O)CN2C(=O)c3ccccc3S2(=O)=O HTS08635 c1ccc(cc1)NC(=O)CSc2nnc(n2C3Cc4ccccc4C3)O HTS08646 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccccc3N4CCCCC4)Cl HTS08458 c1cc(sc1)NC(=O)Nc2nnc(s2)C3CC3 HTS08180 c1ccc(cc1)C(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F HTS08388 c1cc(cc(c1)S(=O)(=O)N)NC(=O)Nc2cccs2 HTS06211 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccc(cc3F)F HTS08633 Cc1c2cc(ccc2sc1C(=O)CSc3nnc(n3C(C)c4ccccc4)O)Cl HTS08650 CC(c1ccccc1)n2c(nnc2SCC(=O)c3ccc(cc3)F)O HTS08653 CC(C)(C)c1cc(n(n1)C)C(=O)NNc2c(cncc2Cl)Cl HTS03682 CCN(c1cccc2c1cccc2)C(=O)c3cccc(c3)OC HTS08619 CCN(c1cccc2c1cccc2)C(=O)c3cccs3 HTS08620 Cc1c(snn1)C(=O)NC(C)(C)C#C CD05414 Cc1c(nns1)C(=O)NC(=S)Nc2ccccc2 CD05430 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(o3)c4ccc(cc4)OC(F)(F)F)C#N HTS03820 Cc1c(c(on1)C)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03255 Cc1cc(no1)C(=O)Nc2ccc3c(c2)cc[nH]3 HTS08308 c1ccnc(c1)CN2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F HTS07830 Cc1cc(n(n1)c2c3cnn(c3ncn2)c4ccccc4)C HTS07601 c1ccc(cc1)n2c3c(cn2)c(ncn3)N/N=C/c4cccnc4 HTS07604 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 HTS07912 c1cc2c(cc1CN3CCN(CC3)S(=O)(=O)c4ccc(c(c4)Cl)F)OCO2 HTS03261 Cc1cccc(c1N2C(=O)C3CC=CC(C3C2=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)C CD06008 Cn1cnc(c1Sc2ccccc2)[N+](=O)[O-] HTS03861 c1ccc(cc1)n2c(nnc2SCC(=O)N3CCOCC3)O HTS07991 CCOC(=O)C1=C(Oc2c3ccccc3oc(=O)c2C1c4ccccc4)N HTS07615 c1ccc(cc1)Oc2ccccc2NC(=O)CN3CCOCC3 HTS06592 CCOC(=O)/C(=C/c1cn(nc1c2ccc(cc2)Cl)c3ccccc3)/C#N HTS07629 c1cc(cc(c1)NS(=O)(=O)c2cccs2)CO HTS08047 c1cc2c(c(c1)S(=O)(=O)Nc3nnc(s3)C4CC4)non2 HTS02722 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)NNc3ccc(cc3)S(=O)(=O)N HTS03564 CCCCc1ccc(c(c1)C)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03697 c1cc(ccc1C(F)(F)F)S(=O)(=O)NCc2csc3c2cc(cc3)Cl HTS04209 COc1ccc(c(c1)S(=O)(=O)NCc2csc3c2cc(cc3)Cl)OC HTS04210 c1ccc(c(c1)NC(=O)c2ccc(cc2)F)Sc3nc4ccc(cc4s3)Cl HTS03932 Cn1c(nnc1SCC(=O)NNC(=S)Nc2ccccc2)c3ccccc3 HTS08986 c1ccc(cc1)CNC(=S)NNC(=O)c2c(c3c(c(nnc3s2)c4ccccc4)c5ccccc5)N HTS08993 c1cc(sc1)c2ccnc(n2)SCC(=O)c3ccc4c(c3)OCCCO4 HTS04407 c1ccc2c(c1)cc(s2)NC(=O)Nc3ccc4c(c3)OCCCO4 HTS03766 c1cc(ccc1C(=O)N2CCN(CC2)C(=O)CSCC(=O)O)Cl HTS08060 Cn1cc(nc1)S(=O)(=O)Nc2cc(nn2C)c3ccc(cc3)Cl HTS08066 COC(=O)c1c(nccn1)C(=O)Nc2ccccc2N3CCOCC3 HTS07228 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)F)N3CCCCC3 HTS08438 c1ccc(c(c1)NC(=O)Nc2cccc(c2)Cl)N3CCCCC3 HTS08441 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F HTS08494 c1ccc2c(c1)CC(C2)n3c(nnc3S)O HTS07407 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2ccc(cc2)C(F)(F)F HTS08096 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3F)F HTS03566 Cc1cc(cc(c1)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)C HTS03700 Cc1ccc(cc1)C(=O)Nc2ccccc2Sc3nc4ccc(cc4s3)Cl HTS03933 CN(C)C(=O)Oc1nnc(n1C2CC2)SCC(=O)c3ccc4c(c3)OCCO4 HTS08656 c1ccc2c(c1)c(c[nH]2)CCNC(=O)/C(=C/c3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)/C#N CD06581 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)S(=O)(=O)c5ccc(s5)c6cc(on6)C(F)(F)F HTS08771 Cc1c2c([nH]n1)OC(=C(C23c4ccccc4NC3=O)C#N)N HTS06870 c1ccc2c(c1)c3cc[nH]c(=O)c3c(=O)[nH]2 HTS08462 COc1ccc(cc1)c2c(nn3c2[nH]c(cc3=O)CC(=O)OC)C(F)(F)F HTS01631 c1cc(cc(c1)C(F)(F)F)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS03455 Cc1c(nns1)C(=O)Nc2c(nn(c2C(C)(C)C)C)C(C)(C)C HTS03461 c1cc(c(c(c1)Cl)C(=O)Nc2ccc(cc2)S(=O)(=O)N)F HTS08369 CCN(CC)c1ccc(cc1)NC(=O)Nc2cccc3c2cccc3 HTS03916 CC(=O)c1ccc(c(c1)CS/C(=C(/C#N)\C(=O)N)/NCCCOC)OC CD06586 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3cccs3 HTS08497 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(c(cc3C(=O)OC)OC)OC HTS03535 CC(C)(C)c1ccc(cc1)NC(=O)NCC(COc2ccc(cc2)[N+](=O)[O-])O HTS08016 Cc1c(nn(n1)c2ccccc2)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS08260 CCc1ccc(cc1)C(=O)NNc2ccc(cc2C)Cl HTS03653 Cc1cc(ccc1NNC(=O)c2c(noc2C)C)Cl HTS03655 CN(CCc1ccccn1)C(=O)Nc2cccc(c2)Cl HTS08267 c1ccc(cc1)c2c(sc(n2)Nc3ccccc3)C(=O)c4ccccc4 HTS08326 c1ccc(c(c1)C(=O)Nc2ccc3c(c2)C(=O)OC3)C(=O)O HTS02925 CC(=O)Nc1ccc(cc1)NC(=O)CCC(=O)O HTS08561 CC(=O)Nc1ccc(cc1)NC(=O)CCCC(=O)O HTS08564 CC(=O)Nc1ccc(cc1)NC(=O)CC(C)(C)CC(=O)O HTS08565 c1ccnc(c1)c2ccc(s2)C(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS07325 c1cc2c(cc1C(COC3=NCNc4c3ccc(c4)Cl)O)OCCO2 HTS08303 CC(C)(C)c1c(c(n(n1)C)C(C)(C)C)NC(=O)c2ccc(cc2)OC HTS03465 c1ccc(cc1)NC(=O)CSc2nnc(n2c3cccnc3)O HTS08644 c1ccc2c(c1)C3(C(=C(OC4=C3C(=O)CCC4)N)C#N)C(=O)N2 HTS08463 c1ccc(cc1)c2cc(on2)C(=O)CN3CCN(CC3)c4nc5cc(ccc5s4)Cl HTS03293 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc3ccccc3c2 HTS07192 Cc1c(c(on1)C)S(=O)(=O)N(Cc2ccccc2)C(C)C HTS07193 c1cc(sc1)S(=O)(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl HTS08281 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS08284 c1ccc(cc1)NC(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl HTS08287 CC(=O)Nc1ccc(cc1)NC(=O)CC2(CCCC2)CC(=O)O HTS08566 CC(=O)Nc1ccc(cc1)NC(=O)Nc2cccs2 HTS08569 CCc1ccc(cc1)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03253 CC(C)(C)c1cc(n(n1)C)C(=O)N2CCCN(CC2)c3ncc(c(n3)C(F)(F)F)C(=O)OC HTS03608 Cc1c(snn1)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03256 c1cc(ccc1NC(=O)CN2CCN(CC2)c3nc4cc(ccc4s3)Cl)OC(F)(F)F HTS03279 C[C@@H](C(=O)N1CCN(CC1)c2ccccc2OC)N3CCN(CC3)c4nc5cc(ccc5s4)Cl HTS03281 CC(C)(C)c1ccc(cc1)NC(=O)CSc2[nH]c3cc(c(cc3n2)Cl)Cl HTS08892 c1cnn(c1)c2ccc(cc2)CO CC18409 c1cc2c(cc1C(COC3=NCNc4c3ccc(c4)Cl)O)OCCCO2 HTS08304 Cc1ccc(cc1)C(COC2=NCNc3c2ccc(c3)Cl)O HTS08305 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)NC(=O)C)C HTS08571 CC(=O)Nc1ccc(cc1)NC(=O)Nc2ccccc2OC(F)(F)F HTS08576 CC1SCC(=NOC(=O)c2ccc(cc2)Cl)CS1 CD10006 Cc1ccc(cc1Cl)NNC(=O)CCc2ccccc2 HTS03637 c1ccc(cc1)Oc2cccc(c2CNC(=O)CSCC(=O)O)Cl HTS04309 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(ccc3N4CCOCC4)C(F)(F)F HTS03781 CCN(CC)c1ccc(cc1)NC(=O)c2ccco2 HTS03928 Cc1c(snn1)C(=O)N(Cc2ccccc2)C(C)C HTS07195 Cc1ccccc1C(=O)Nc2ccc(nc2)Oc3ccc(cc3)C(C)(C)C HTS08500 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3ccco3 HTS08502 Cc1c(c(ncn1)OCC(=O)Nc2ccc3c(c2)OCCO3)CC(=O)OC HTS07760 Cn1c(cc(n1)c2ccc(cc2)Cl)NC(=O)c3ccccc3C(=O)O HTS08049 c1cc(ncc1C(F)(F)F)NC(=O)CSCC(=O)O HTS08592 CCCc1c(cnn1c2ccccc2)C(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 HTS03530 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3)C(C)C HTS03540 Cc1cc(c(o1)C(F)(F)F)NC(=O)Nc2ccsc2C(=O)OC HTS04299 CC1=NCCN1CCNC(=O)Nc2cccc(c2)OC HTS08020 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(nc2)N(C(=O)C)S(=O)(=O)c3c(noc3C)C HTS07707 Cc1nc(cn1C)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)C(=O)C HTS07756 c1ccn(c1)c2nnc(s2)C3CC3 HTS08190 c1cc(ccc1F)S(=O)(=O)CCSc2nnc(n2C3CC3)O HTS08313 CC(C)(C)c1cc(no1)NS(=O)(=O)c2ccc(cc2)C#N HTS08225 Cc1ccc(n1c2ccsc2C(=O)NN)C CD08752 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(C)c3ccc(cc3)Cl CD07013 CC(=O)CCc1ccc(c(c1)OC)OC(=O)c2ccc(cc2)C(C)(C)C CD07221 CC(=O)CCc1ccc(c(c1)OC)OC(=O)c2c(cccc2Cl)F CD07234 Cc1ccc(c(c1)C)NS(=O)(=O)c2c(nn(c2Cl)C)C CD10235 CC1=NCCN1CCNC(=O)Nc2ccc(cc2)F HTS08022 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(s3)c4cccs4)C(=O)OC HTS03555 CCc1cc(c(s1)NC(=O)COc2ccccc2)C(=O)c3ccc(cc3)OC HTS08677 Cc1c(c(no1)c2ccccc2)C(=O)NCCN3CCNC3=O HTS08371 CN(C)CCCNS(=O)(=O)c1ccc(cc1)Cl CD05608 CN(C)CCCNS(=O)(=O)c1cc(c(cc1Cl)Cl)Cl CD05610 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)CC3(CCCC3)CC(=O)O HTS08514 c1ccc(cc1)NC(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F HTS08491 Cc1c(c(n(n1)C(=O)c2ccc(cc2)[N+](=O)[O-])C)Br CD07251 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(c(c3)OC)OCc4ccccc4)C(=O)OC HTS03557 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)S(=O)(=O)c3cccc4c3non4 HTS03616 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCc3csc4c3cc(cc4)Cl HTS04214 c1ccc2c(c1)cccc2NC(=O)NCc3csc4c3cc(cc4)Cl HTS04218 Cc1c(cc2c(c1n3cccc3)C(CC2(C)C)(C)C)N4CCCC4 CD03912 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD07034 Cc1ccc(cc1)n2c(nnn2)c3cnn(c3c4ccccc4C)c5ccc(c(c5)Cl)Cl HTS05451 CCN(CC)C(=S)Oc1ccc(cc1C(=O)Nc2cc(cc(c2)Cl)Cl)Br CD07066 CC1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)CC=C)C1 HTS07639 CC1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)Cc4ccccc4)C1 HTS07640 Cc1ccc(cc1)n2c(=O)c3c4c(sc3[nH]c2=O)CC(CC4)C HTS07650 CN(C)C(=S)SCc1nc(no1)c2ccc(cc2)Cl CD06383 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)C HTS08380 Cc1c(c(no1)c2ccccc2)C(=O)N3CCCN(CC3)C(=O)c4c(onc4c5ccccc5)C HTS08384 Cc1c(snn1)C(=O)Nc2ccccc2C#N HTS07798 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(s3)c4cc(n(n4)C)C(F)(F)F)C HTS07771 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)ONC(=O)c3ccco3 CD05764 CC1SCC(CS1)NC(=O)c2ccc(cc2)Cl CD10274 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)Cl)N3CCCCC3 HTS08157 c1ccc(cc1)NC(=O)c2c(nccn2)C(=O)O HTS03747 c1cc2c(cc1NC(=O)c3c(nccn3)C(=O)O)OCCCO2 HTS03748 CCCCCc1ccc(cc1)S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 HTS03264 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)N(CCC#N)Cc3ccco3 HTS03268 Cc1c(snn1)c2nnc(n2C3CC3)SCC(=O)c4ccc(cc4)C#N HTS08683 Cc1ccc(cc1)c2ccn(c(=S)n2)c3cc(ccc3OC)C(F)(F)F HTS05444 Cc1cc(c(o1)C)C(=O)Nc2ccc(nc2)Oc3ccc(cc3)C(C)(C)C HTS08503 Cc1ccc(cc1)C(=O)Nc2ccc(nc2)Oc3ccc(cc3)C(C)(C)C HTS08504 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)Nc3cccc(c3)OC HTS08509 CSCCNC(=O)c1ccccc1N CD07085 CCN(CC)C(=O)Oc1ccc(cc1C(=O)Nc2ccc(c(c2)Cl)F)Br CD07076 c1cc2c(cc1CNS(=O)(=O)c3ccc(c(c3)Cl)F)OCO2 HTS03870 c1ccc(c(c1)n2c(noc2=O)c3cccnc3)F RF05156 COc1ccc(cc1)c2noc(=O)n2c3cccnc3 RF05168 CC1CCc2c(sc3c2c(ncn3)Sc4ccccc4)C1 HTS07682 c1ccc(cc1)CNc2ncc(s2)C(=O)O MO00042 Cc1cc(nc2c1cccc2)O AC12157 c1cc2c(cc1CNC(=O)c3c(ccs3)Br)OCO2 HTS03596 c1ccc(cc1)CN2CCN(CC2)CCNC(=O)Nc3ccc4ccccc4c3 HTS03190 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)CC(C)(C)CC(=O)O HTS08517 Cc1c2c(cccc2F)n(n1)C(=O)c3ccccc3Cl CD07205 Cc1ccc(cc1Cl)S(=O)(=O)Nc2ccccc2C#N HTS08150 COc1ccccc1NC(=O)Nc2ccc(cc2)NC(=O)c3ccccc3O HTS08231 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)Cc4nc(no4)c5cccs5 HTS03623 Cc1c2cc(ccc2sc1S(=O)(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6)Cl HTS08762 c1ccc(cc1)S(=O)(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08766 CN(/C=C/c1n(nnn1)c2ccccc2)CCN(/C=C/c3n(nnn3)c4ccccc4)C HTS05439 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)COCC(=O)O HTS08513 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)CSCC(=O)O HTS08516 CC(C)(C)c1cc(n(n1)c2ccccc2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl CD06941 Cc1ccccc1Nc2ncnc(n2)N RJF00601 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS08285 CC(=O)Nc1ccc(cc1)NC(=O)CSCC(=O)O HTS08568 CC(=O)Nc1ccc(cc1)NC(=O)Nc2ccc(cc2)C(C)(C)C HTS08572 c1cc(cc(c1)NC(=O)CSc2nccc(n2)c3cccs3)C(F)(F)F HTS04403 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=N)N3CCCC3 CD07790 c1cc(c(c(c1)Cl)CSCCNC(=O)Nc2c(cccc2Cl)Cl)F CD07811 c1cc2c(cc1CN3CCN(CC3)S(=O)(=O)c4ccc(cc4F)F)OCO2 HTS03694 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc4c(c3)OCC4)C(=O)OC HTS03556 CC(C)(C)c1c(c(n(n1)C)C(C)(C)C)NC(=O)c2c(ccs2)Cl HTS03463 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)N(C)C3CCN(CC3)C HTS03467 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS08286 CCc1cc(c(s1)NC(=O)CN2CCN(CC2)C(=O)OCC)C(=O)c3ccc(cc3)OC HTS08690 C=CCn1c(=N)c2c3c(sc2nc1SCc4ccc(cc4)Cl)CCCC3 HTS08974 COc1cccc(c1)/C=N/NC(=O)CSc2nnc(n2CC=C)c3ccccc3 HTS08979 Cc1cc(=O)n2c3ccccc3[nH]c2c1C#N HTS09052 C=CCn1c(c(sc1=S)C(=O)N)N HTS09055 CCN(CC)c1c2c(nc(n1)C)n(c(=S)s2)c3ccccc3 HTS09057 c1ccc(cc1)n2c3c(cn2)c(=N)n(cn3)NC(=S)Nc4ccc(cc4Cl)Cl HTS09038 c1cc(sc1)C(=O)Nc2cc(cc(c2)NC(=O)c3cccs3)C(F)(F)F CD10955 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5cc(cc6c5OCOC6)F HTS07944 Cc1c(c(no1)c2ccccc2)NC(=O)N(C)CCc3ccccn3 HTS08268 Cc1c(sc(n1)Nc2ccccc2)C(=O)c3ccccc3 HTS08327 c1ccc(c(c1)C(F)(F)F)NC(=S)NNC(=O)C2CC2 RJF00619 c1ccnc(c1)CCNC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF00945 Cc1ccc(cc1)S(=O)(=O)CC(=O)N(c2ccc(cc2)F)C(C(=O)c3ccc(cc3)Cl)C(=O)NC4CCCCC4 HTS08971 c1ccc(cc1)/N=C\2/C3=C(CCCC3)/C(=N/C4CCCCC4)/S2 HTS08972 Cc1ccn2c(c1)nc(c2C(=O)O)C HTS08973 Cc1cc(nc(n1)c2ccc(cc2)Cl)O RJF00199 CNC(=S)NNC(=O)CSc1nnc(n1CC=C)c2ccccc2 HTS08985 COc1ccc(cc1)NS(=O)(=O)c2ccc(cc2)Oc3c(cccc3C#N)C#N CD10985 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)Oc3ccc(cc3)[N+](=O)[O-])C#N CD11032 COc1ccc(cc1)OS(=O)(=O)c2ccc(cc2)Oc3c(cccc3C#N)C#N CD11033 CCN(CC)c1ccc(cc1)NS(=O)(=O)c2cccs2 HTS03911 CCN(c1cccc2c1cccc2)C(=O)c3ccc(cc3)C(F)(F)F HTS08621 Cc1c(cnn1c2ccccc2)C(=O)N(Cc3ccccc3)C(C)C HTS07892 CCCCOc1ccc(cc1)NC(=O)C MO00821 Cc1c(c(nc(n1)c2ccc(cc2)Cl)O)CC=C RJF00222 c1cc(cc(c1)F)OC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS08756 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3nnc(s3)C4CC4 HTS08173 c1cc(sc1)c2nc(on2)CN3CCOCC3 HTS03628 COc1cc(cc(c1)NC(=O)c2ccc(cc2)C(F)(F)F)C(F)(F)F CD11052 COc1cc(cc(c1)NC(=O)OC)C(F)(F)F CD11053 CN(C)C(=O)c1c2ccccc2c(=O)n(n1)c3ccc(cc3)Cl CD11077 CN(C)C(=O)Oc1nnc(n1c2ccccc2)SCCS(=O)(=O)c3ccc(cc3)F HTS08657 c1cc(ccc1N)n2cncn2 CC18614 COc1ccc(cc1NC(=O)Nc2ccccc2N3CCCCC3)Cl HTS08442 c1cc(oc1)Cn2c(nnc2S)O HTS07406 Cc1ccc(cc1Cl)NNC(=O)c2c(nns2)C HTS03641 Cc1ccc(cc1Cl)NNC(=O)c2cccs2 HTS03642 Cc1ccc(cc1Cl)NNC(=O)c2c(onc2c3ccccc3)C HTS03645 CCOC(=O)Cc1csc(n1)N2C(=O)CC(CC2=O)c3ccccc3 HTS08098 Cc1c(snn1)c2nnc(o2)C3CCCCC3 HTS08123 c1cc(ccc1C(F)(F)F)S(=O)(=O)Nc2ccc3c(c2)C(=O)OC3 HTS04221 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)NCc3csc4c3cc(cc4)Cl HTS04224 Cc1c(c(no1)c2ccccc2)C(=O)NCc3csc4c3cc(cc4)Cl HTS04225 CCN(CC)c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)F HTS03913 CCN(CC)c1ccc(cc1)NC(=O)Nc2ccccc2 HTS03915 Cc1c(cnn1c2ccccc2)C(=O)N(C)C3CCCCC3 HTS07896 CC(c1ccccc1)n2c(nnc2SCC(=O)Nc3ccccc3)O HTS08642 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2S(=O)(=O)c3ccccc3C#N HTS07963 c1cc(ccc1c2ccnc3n2cnn3)Cl HTS08472 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc4c(c3)OCO4)C#N HTS03816 CC1=C(C(C2=C(N1)CCCC2=O)c3ccccc3N4CCOCC4)C#N HTS03818 Cc1c(snn1)C(=O)NCc2csc3c2cc(cc3)Cl HTS04229 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NCc3csc4c3cc(cc4)Cl HTS04473 c1ccc(cc1)CCC(=O)NNc2ccc(cc2)S(=O)(=O)N HTS04478 CC(C)c1ccc(cc1)NNC(=O)c2ccc(cc2F)F HTS03874 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN(C)c3cccc(c3C#N)F CD06833 c1ccc(c(c1)NS(=O)(=O)c2cccs2)N3CCCCC3 HTS08158 c1c(cc(cc1Br)Br)CN2CCSCC2 CD08470 c1ccnc(c1)c2ncc(c(n2)C(F)(F)F)c3nnnn3c4ccc(cc4)Cl HTS06852 c1ccc(c(c1)NC(=O)CN2CCC(CC2)C(=O)N)N3CCOCC3 HTS07836 CN(C1CCCCC1)S(=O)(=O)c2cccs2 HTS07908 Cc1c(c(on1)C)C(=O)NNc2ccc(cc2)C(C)C HTS03881 CC(C)c1ccc(cc1)NNC(=O)c2cccs2 HTS03883 CN(CCc1ccccn1)C(=O)Nc2ccc(cc2)F HTS08781 COC(=O)c1c(ccs1)NC(=O)CC2C(=O)NCCN2S(=O)(=O)c3cccs3 HTS07964 C(C(=O)Nc1nnc(s1)C(F)(F)F)SCC(=O)O HTS08618 Cn1c2cccc(c2c(n1)NC(=O)Nc3ccc(cc3F)F)OC HTS03823 Cc1cc2nccc(n2n1)c3cccs3 HTS06868 Cn1c(ccc1S(=O)(=O)NNc2c(cncc2Cl)Cl)C(=O)OC HTS03689 COc1ccc(cc1OC)CCNC(=O)c2c(nccn2)C(=O)O HTS03731 CC(C)c1ccc(cc1)NC(=O)CSc2[nH]c3cc(c(cc3n2)Cl)Cl HTS08887 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)N3C(=O)C4=C(C3=O)SCCS4)C HTS08140 c1ccc2c(c1)cccc2NC(=O)NCCN3CCNC3=O HTS02809 CCN(CC)C(=S)Oc1ccc(cc1C(=O)NCCc2ccncc2)Br CD07088 COc1ccc(cc1NC(=O)Nc2nnc(s2)C3CC3)Cl HTS08176 Cc1ccc(cc1NC(=O)Nc2nnc(s2)C3CC3)F HTS08177 C1CC1c2nnc(s2)NC(=O)COCC(=O)O HTS08183 Cc1c(snn1)C(=O)NNS(=O)(=O)C HTS07766 Cc1ccc(cc1)C(=O)C/C(=C\C(=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])\c3ccc(cc3)C)/c4ccccc4 HTS06857 c1ccc2cc(ccc2c1)n3c(nnn3)c4c[nH]c5c4cc(cc5)Cl HTS06845 c1cc(cc(c1)NC(=O)CSc2[nH]c3cc(c(cc3n2)Cl)Cl)C(F)(F)F HTS08894 Cc1ccc(cc1)n2c(nnn2)/C=C/Nc3cc(ccc3OC)C(F)(F)F HTS06846 COc1ccc(cc1)n2c(nnn2)/C=C/Nc3cc(ccc3OC)C(F)(F)F HTS06847 CC(=O)Nc1ccc(cc1)NC(=O)Nc2ccccc2 HTS08570 CC(=O)CCc1ccc(c(c1)OC)OC(=O)c2ccc(cc2Cl)Cl CD07219 CCOC(=O)c1cnc(s1)NCc2ccccc2 MO00029 Cc1c(c(no1)c2ccccc2)C(=O)NCCNC(=O)c3c(onc3c4ccccc4)C HTS08215 c1ccc(c(c1)Cn2cnc3c(c2=O)c4c(s3)CCCC4)Cl HTS07664 CC1CCc2c(sc3c2c(=O)n(cn3)CC=C)C1 HTS07665 CC(C)(CC(=O)NNc1c(cncc1Cl)Cl)CC(=O)O HTS03677 COc1ccc(cc1)OCCNC(=O)c2c(nccn2)C(=O)O HTS03730 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)S(=O)(=O)c5ccc6c(c5)CCO6 HTS08272 c1ccc(cc1)c2c3ccccc3ncc2c4nnnn4c5ccc(cc5)Cl HTS05457 c1cc(sc1)C(=O)Nc2nnc(s2)C3CC3 HTS08162 c1cc(ccc1c2c(cno2)c3nnnn3c4ccc(cc4)Cl)C(F)(F)F HTS05449 Cc1cc(c(o1)C(F)(F)F)NC(=O)Nc2ccc(cc2)F HTS04298 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3c4ccccc4)O HTS07993 Cc1c(c(no1)c2ccccc2)C(=O)N3CCNCC3 HTS11379 c1ccnc(c1)CCN(CCC#N)C(=O)Nc2ccc3c(c2)CCO3 HTS06107 c1ccc2c(c1)CCC(=C2)N3CCN(CC3)c4ccccc4Cl HTS06842 Cc1ccc(cc1)n2c(nnn2)c3c[nH]c4c3cc(c(c4)Cl)F HTS06843 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)Oc3ccc(cc3OC)CCC(=O)C CD07220 c1ccc(cc1)S(=O)(=O)Nc2ccccc2N3CCCCC3 HTS08431 c1cc(c(c(c1)Cl)CSc2nccn2c3ccc(cc3Cl)Cl)Cl CD09910 CC(C)(C)c1ccc(cc1)Sc2c(ncn2C)[N+](=O)[O-] HTS03865 c1ccc(cc1)Oc2cccc(c2CNC(=O)Nc3ccc(cc3)C(F)(F)F)Cl HTS04311 c1cc(cc(c1)[N+](=O)[O-])NC(=O)CSc2nccc(n2)c3cccs3 HTS04405 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(cc(c3)OC)OC HTS03782 CN(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)S(=O)(=O)N3CCOCC3 HTS03457 CC1CCc2c(sc3c2c(=O)n(cn3)CC(=O)C)C1 HTS07666 CCOC(=O)C(C(=O)C)Sc1c2c3c(sc2ncn1)CCCC3 HTS07675 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)S(=O)(=O)c5ccc(s5)c6ccccn6 HTS08273 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6)C(F)(F)F HTS08277 c1cc2c(cc1Cl)ncnc2Oc3ccc(cn3)NC(=O)/C=C/C(=O)O HTS08297 Cc1ccccc1c2c(cno2)c3nnnn3c4ccccc4 HTS05450 c1ccc(cc1)NC(=O)NC2CCSC2 CD10095 CCCCNC(=O)OC(CSCc1c(cccc1Cl)F)CSCc2c(cccc2Cl)F CD09354 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc4c(c3)CCC(O4)(C)C)C(=O)OC HTS03558 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)NCc3ccc4c(c3)OCO4 HTS03567 CCCc1c(cnn1c2ccccc2)C(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS03786 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cccc(c3)SCc4cccc(c4F)Cl HTS03787 c1ccc(cc1)n2c(nnn2)c3cnoc3c4ccc(cc4)Cl HTS05445 CSc1cccc(c1)Nc2nc(c(s2)/N=C/c3cc(cc(c3O)Cl)Cl)c4ccccc4 CD03953 CN(c1c(cccc1Cl)[N+](=O)[O-])/N=C/c2cc(cc(c2O)Cl)Cl CD07004 CN(C)/C=N/NC(=O)c1cccnc1 CD09223 COc1ccc(cc1)n2ccc(nc2=S)c3ccccc3 HTS05441 c1ccc(cc1)c2ccn(c(=S)n2)c3ccc(cc3)OC(F)(F)F HTS05442 c1c(cc(cc1Cl)Cl)N/C=N/c2cc(cc(c2)Cl)Cl CD07507 c1cc(c(cc1F)F)N/C=N/c2ccc(cc2F)F CD07508 CC(C)(C)c1c(c(n(n1)C)C(C)(C)C)NC(=O)c2c(c3ccccc3s2)Cl HTS03462 CCCc1c(cnn1c2ccccc2)C(=O)Nc3nc[nH]n3 HTS03791 c1cc(cc(c1)S(=O)(=O)NCc2ccc3c(c2)OCO3)C(F)(F)F HTS03961 c1cc(ccc1/C=N/NC(=O)Cn2cnc3c(c2=O)c4c(s3)CCCC4)[N+](=O)[O-] HTS07673 c1cc(cc2c1cc(cc2S(=O)(=O)O)S(=O)(=O)O)O HTS01517 c1ccc(c(c1)NS(=O)(=O)c2cccc3c2non3)N4CCCCC4 HTS08159 c1cc(ccc1C(F)(F)F)NC(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl HTS08291 Cc1cc(c(c(c1)C)n2c(nnc2SCC(=O)N3CCOCC3)O)C HTS08331 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccccc2N3CCCCC3 HTS08440 CN(C)/C=C(\C#N)/C(=O)c1ccc(cc1)OC CD07553 c1cc(cc(c1)OC(=O)c2ccc(cc2)CSC(=S)NCCc3ccc(cc3)Cl)N4CCOCC4 CD09612 c1ccc2c(c1)cccc2NC(=O)Nc3cccc(c3)C(=O)O HTS03988 COc1ccc(cc1)Oc2ccc(cc2C(=O)Nc3ccc(cc3)S(=O)(=O)N)[N+](=O)[O-] HTS08370 CC(=O)Nc1cccc(c1)OCCCNC(=O)CCc2nc(no2)c3ccccn3 HTS08531 Cc1ccc(cc1)C(=O)CSc2nnc(n2C3CC3)c4c(nns4)C HTS08682 c1cc2c(cc1CN3CCN(CC3)S(=O)(=O)c4cc(cc(c4)Cl)Cl)OCO2 HTS03262 Cc1ccc(cc1)n2c(nnn2)c3cnoc3c4cccc(c4)F HTS05446 c1ccc(cc1)C(=O)Nc2cccc(c2)COC(=O)c3ccccc3 HTS07154 CC(c1[nH]c2ccccc2n1)OS(=O)(=O)c3cc(sc3Cl)Cl CD09587 c1ccc(cc1)CN2CCN(CC2)CC(=O)N3CCN(CC3)c4ccccn4 HTS08704 Cc1ccc(n1c2cc(n[nH]2)c3ccccc3)C HTS08712 CC(=O)Nc1ccc(cc1)NC(=O)Nc2cccc(c2Cl)Cl HTS08575 CCOC(=O)C1CCN(CC1)Cc2csc(n2)c3cccs3 HTS07160 Cc1nc(cs1)c2cccc(c2)C(=O)O CC19401 c1cc2cc(ccc2nc1)Cl AC31488 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN(C)c3cccc(c3C#N)F CD06968 CCc1cc(c(s1)NC(=O)c2ccc(cc2)F)C(=O)c3ccc(cc3)OC HTS08693 c1ccc(cc1)NS(=O)(=O)c2ccc(cc2)c3csnn3 HTS08626 c1cc(n(c1)CCC#N)CN2CCOCC2 HTS08536 CC(=O)Nc1ccc(cc1)NC(=O)COCC(=O)O HTS08567 COc1ccc(cn1)NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS08737 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)Nc3ccc(cc3)Cl)C#N CD10984 c1cc(cc(c1)NC(=O)c2c(ccs2)Cl)COC(=O)c3c(ccs3)Cl HTS07155 CC(=O)c1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3cccc4c3non4 HTS07757 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2cc(nn2c3ccccc3)C(C)(C)C)C)C CD06957 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN(C)c3cccc(c3C#N)Cl CD06967 CC1SCC(CS1)NC(=O)c2ccccc2Cl CD10275 CC(=O)Nc1ccc(cc1)NC(=O)Nc2cccc(c2)Cl HTS08577 c1cc(oc1C(=O)NCC2CC2)Oc3cc(cc(c3)Cl)Cl HTS08738 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl HTS08742 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)c3ccc4c(c3)CCO4)C(F)(F)F HTS08399 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2N3CCCCC3 HTS08434 c1ccc2c(c1)cc(s2)NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS03769 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccco4 HTS04239 CCOC(=O)Cc1csc(n1)NC(=O)CCC(=O)O HTS08084 c1ccnc(c1)N2CCN(CC2)C(=O)CN3CCOCC3 HTS08702 c1ccc(cc1)c2cc([nH]n2)NC(=O)c3ccccc3C(=O)O HTS08708 Cc1cc(c(o1)C)C(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS07942 CC(C)(C)c1c(c(n(n1)C)C(C)(C)C)NC(=O)c2cccs2 HTS03452 c1ccc(cc1)c2c(sc(n2)Nc3ccccc3)C(=O)c4ccc(cc4)F HTS08328 c1ccc(c(c1)/C=N/N=C\2/N(C(=O)CS2)c3cc(ccc3Cl)C(F)(F)F)Cl RJF00960 c1cc2c(cc1Cl)c(cs2)CNC(=O)COCC(=O)O HTS03891 Cc1ccc2cc(ccc2n1)OC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl HTS08751 CCOC(=O)c1cnn(c1N)C(=S)N HTS08984 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3ccc(cc3)n4c(cc(n4)C(F)(F)F)c5cccs5 HTS04035 Cc1cc(c(o1)C(F)(F)F)NC(=O)NCCNc2c(cccn2)C(F)(F)F HTS04297 Cc1c(cnn1c2ccccc2)C(=O)Nc3ccccc3SCc4cccc(c4F)Cl HTS02986 CN(CCc1ccccn1)C(=O)c2cccnc2Oc3ccccc3 HTS07946 Cn1cc(c(n1)c2cccc(c2)NC(=O)/C=C/C(=O)O)Br HTS02657 CCN(c1cccc2c1cccc2)C(=O)c3ccc4c(c3)CCO4 HTS08623 Cc1c(snn1)C(=O)Nc2ccccc2SCc3cccc(c3)C(F)(F)F CD05447 CC(c1ccccc1)n2c(nnc2SCc3nc(no3)c4ccc(cc4)C(C)(C)C)O HTS08651 Cc1cc(no1)C(=O)Nc2ccccc2N3CCCCC3 HTS08452 Cc1cc(ccc1NNC(=O)c2c(ccs2)Cl)Cl HTS03649 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2C3CC3)OC(=O)N(C)C HTS08662 c1ccc(cc1)c2nc(nn2c3ccccc3)C(=O)N4CCCCC4 HTS08475 Cc1c(c(no1)c2ccccc2)C(=O)Cn3cc(nc3C)[N+](=O)[O-] HTS04908 c1ccc2c(c1)cccc2C(=O)NNC(=O)c3ccc4c(c3)nsn4 HTS08787 c1cc(c(c(c1)F)C(=O)NC(=O)C(=O)Nc2ccc(cc2F)Cl)F RF04048 c1cc(sc1)CNC(=S)Nc2ccc(c(c2)Cl)F RJF00372 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=O)C2CC2 DFP00249 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 HTS03258 c1ccc2c(c1)cccc2NC(=O)Nc3ccc4c(c3)C(=O)OC4 HTS03392 c1cc(cc(c1)[N+](=O)[O-])/C=N/NC(=O)CC#N CD04223 CC1CCC(C(C1)NC(=S)Nc2cccc(c2)F)C(C)C CD04293 c1ccc(cc1)n2c3c(cn2)c(=N)n(cn3)/N=C/c4ccc(cc4Cl)Cl HTS09039 CCc1cc(c(s1)NC(=O)CSc2nnc(n2C)c3cccs3)C(=O)c4ccc(cc4)OC HTS08673 Cn1c(nnc1SCC(=O)Nc2ccc3c(c2)OCCO3)Cc4ccsc4 HTS08676 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS06420 c1ccc2c(c1)nc(s2)S(=O)(=O)/C(=C/Nc3ccc(cc3)F)/C#N KM01292 CN1C(=O)C(=Cc2ccccc2Cl)C(=O)N(C1=O)C HTS09000 c1cc(ccc1c2cnc(o2)c3cnccc3C(F)(F)F)Cl RF04072 c1cc(ccc1c2nc(no2)c3cnccc3C(F)(F)F)[N+](=O)[O-] RF04186 c1cc(cc(c1)Cl)c2cnc(o2)c3cnccc3C(F)(F)F RF04243 c1ccc(cc1)NC(=S)C(C#N)c2[nH]c3ccccc3n2 HTS09008 COc1ccc(c(n1)Nc2ccc3c(c2)C(=O)OC3)[N+](=O)[O-] HTS03631 Cc1ccc(cc1Cl)NNC(=O)c2ccc(cc2F)F HTS03633 Cc1cc(cc(c1F)C)S(=O)(=O)NC(=N)c2ccccn2 CD08329 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccccc2N3CCCCC3 HTS08443 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)Nc3cccs3)C(F)(F)F HTS08492 Cc1cc(ccc1NNC(=O)c2cc3ccccc3s2)Cl HTS03650 Cc1cc(ccc1NNC(=O)CCc2ccccc2)Cl HTS03652 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)Nc3nnc(s3)C4CC4 HTS08163 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCc4ccc(cc4)Cl HTS09011 c1ccc2c(c1)/C(=N/Nc3nc(cs3)c4ccc(cc4)Cl)/C(=O)N2 HTS09016 c1ccc2c(c1)/C(=N/Nc3nc(cs3)c4ccc(cc4)Br)/C(=O)N2 HTS09017 Cc1nc(c(o1)C(F)(F)F)c2nc(on2)c3ccccc3 RF04262 COc1cc(c(cn1)C(=O)NCc2ccc(cc2)Cl)C(F)(F)F RF04308 CN(Cc1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04309 c1c(cc(cc1C(F)(F)F)N2C(=O)CCC2=O)C(F)(F)F FV00047 c1ccn(c1)c2ccc(cc2NC(=S)Nc3cc(ccc3Cl)C(F)(F)F)C(F)(F)F CD04456 c1cc(ccc1C(COC2=NCNc3c2ccc(c3)Cl)O)F HTS08302 CC1C/C(=N\N=C\c2cc(cc(c2O)Cl)Cl)/c3c1cccc3 JPV00071 CSc1cccc(c1)NC(=O)C(=O)NCc2ccco2 JPV00076 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=O)C(=O)Nc2cccc(c2)SC JPV00081 c1cc(cc(c1)NC(=O)Nc2nnc(s2)C3CC3)C(F)(F)F HTS08178 c1cc(ccc1C(=S)N)S(=O)(=O)N2CCOCC2 CD10813 Cc1cc(=O)n2c([nH]1)ncn2 HTS09027 c1ccc(cc1)c2cc(=O)n3c(n2CC(=O)N/N=C/c4ccc5c(c4)OCO5)ncn3 HTS09029 C=CCNC(=S)NNC(=O)Cn1c(cc(=O)n2c1ncn2)c3ccccc3 HTS09032 CCOc1cc(c(cn1)C(=O)N(C)Cc2ccc(cc2)Cl)C(F)(F)F RF04312 Cc1c(c(no1)NC(=O)CSCC(=O)O)Br HTS07729 c1ccc2c(c1)cc(s2)NC(=O)NCc3cccs3 HTS03776 c1ccc2c(c1)cc(s2)NC(=O)Nc3ccc(cc3F)F HTS03779 c1cc(ccc1c2csnn2)OCC(CN3CCC(CC3)C(=O)N)O HTS03851 c1cc(ccc1C(=O)CN2CCN(CC2)c3nc4cc(ccc4s3)Cl)OC(F)(F)F HTS03294 COc1cc(c(cc1OC)NC(=O)CSCC(=O)O)C(=O)O HTS02698 c1cc(cc(c1)C(F)(F)F)/C(=C/c2ccc(s2)[N+](=O)[O-])/C#N CD04227 Cc1cc(nc2c1c(c(o2)C(=O)N/N=C/c3ccc(cc3Cl)Cl)N)c4ccccc4 HTS09036 c1cc(oc1C(=O)Nc2cc(cc(c2)NC(=O)c3ccc(o3)[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD10961 Cc1cc(n2c3ccccc3nc2c1C#N)N HTS09042 Cc1cc([nH]c(=O)c1C#N)c2ccccc2 HTS09043 Cc1cc(nc2c1c3c(o2)c(ncn3)SCC(=O)c4ccc(cc4)c5ccccc5)c6ccccc6 HTS09044 CN1CCN(CC1)c2c3c(nc4n2ncn4)CCC3 HTS09068 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)N3CCC(CC3)O HTS02643 C1CC1c2nnc(s2)NC(=O)CSCC(=O)O HTS08181 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)c3cccs3)C(F)(F)F HTS08386 CN(C1CCCCC1)C(=O)c2c(cccc2Cl)F HTS07918 CCOC(=O)C1CCN(CC1)C(=O)Nc2cc(cc(c2)Cl)Cl HTS07380 c1cc(c(c(c1)F)C(=O)Nc2cc(cc(c2)NC(=O)c3c(cccc3F)F)C(F)(F)F)F CD10962 c1ccc(cc1)S(=O)(=O)NCCC2CC2(Cl)Cl CD10994 Cc1cc(nc2c1c(c(o2)C(=O)NNC(=S)NC)N)c3ccccc3 HTS09045 c1ccc2c(c1)[nH]c3n2c(=O)c4c(c3C#N)CCCC4 HTS09049 C=CCn1c2c(c(ncn2)C(C#N)C#N)sc1=S HTS09056 c1ccc(c(c1)C(F)(F)F)NNC(=O)c2ccno2 HTS03408 c1ccc(c(c1)C(F)(F)F)NNC(=O)C2CCC2 HTS03409 Cc1ccc(cc1)S(=O)(=O)Nc2cc(nn2C)c3ccc(cc3)Cl HTS08063 c1ccc(cc1)C(=O)CN2CCN(CC2)c3nc4cc(ccc4s3)Cl HTS03286 Cn1cnc(c1Sc2nccc(n2)c3cccs3)[N+](=O)[O-] HTS03864 c1cc(cc(c1)N2CCN(CC2)/C=C/c3nnnn3c4ccc(cc4)Cl)C(F)(F)F HTS06851 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)S(=O)(=O)N HTS08351 C=CCNC(=O)O/N=C/c1cc(sc1)[N+](=O)[O-] DFP00104 c1cc(ccc1c2cn3c(n2)scn3)[N+](=O)[O-] DP00621 c1ccc(cc1)Oc2c(cccn2)C(=O)NCc3ccc4c(c3)OCO4 HTS03595 c1ccc(cc1)Oc2c(cccn2)C(=O)Oc3ccccc3N4CCOCC4 HTS03599 CC1SCC(=NOC(=O)c2ccccc2Cl)CS1 CD10013 c1cc(c(cc1Cl)Cl)N/C(=N\O)/c2cnccc2C(F)(F)F RF05225 c1ccc2c(c1)c(nn(c2=O)c3ccc(cc3)[N+](=O)[O-])c4ccc(cc4)F DP00624 Cc1c(c(no1)c2ccccc2)C(=O)Nc3c(nn(c3C(C)(C)C)C)C(C)(C)C HTS03454 CSc1cccc(c1)NC(=S)NCCNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03711 Cc1cc(no1)C(=O)Nc2ccc(cc2)S(=O)(=O)N HTS08367 c1cc(ccc1c2c(cno2)c3nnnn3c4ccc(cc4)Cl)F HTS05448 c1cc(c(cc1F)F)NC(=O)C23CC4CC(C2)CC(C4)C3 CD08930 c1cc(ccc1CCNC(=O)C23CC4CC(C2)CC(C4)C3)Cl CD08936 CC1(COC(OC1)C2CCNCC2)C.C(=O)(C(=O)O)O MO00374 Cc1ccc(cc1)c2ccn(c(=S)n2)c3ccc(c(c3)Cl)C HTS05443 CN1C(=O)C(=Cc2ccc(cc2Cl)Cl)C(=O)N(C1=O)C HTS09002 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)c4cc(cc(c4)Cl)Cl DP00682 c1ccc(cc1)Cn2c(=O)c3ccccc3c(n2)c4ccccc4 DP00711 Cc1ccc(cc1Cl)NNC(=O)c2c(cccc2Cl)F HTS03636 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(o3)CN4C(=O)c5ccccc5C4=O)C(=O)OC HTS02625 CCOC(=O)c1c2cc(c(c(c2c(=O)n(n1)c3ccccc3)N)C#N)c4ccccc4 HTS08485 CC(=O)NCCc1c(cccc1Cl)F CD07767 c1cc(cc(c1)N/C(=N\O)/c2cnccc2C(F)(F)F)C(F)(F)F RF05226 Cc1c(c(n(n1)C)Cl)S(=O)(=O)Nc2ccc(cc2)Br CD10238 CCc1cc(c(s1)NC(=O)COc2ccc(cc2)Cl)C(=O)c3ccc(cc3)OC HTS08679 CC(C)(CC(=O)Nc1cc(n[nH]1)c2ccccc2)CC(=O)O HTS08709 c1ccc2c(c1)CC(C2)NC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl HTS08732 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3ccc4c(c3)CCO4 HTS08505 CCN(CC)C(=O)Oc1ccc(cc1C(=O)Nc2cc(cc(c2)Cl)Cl)Br CD07064 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc(c(c2)C(F)(F)F)S(=O)(=O)Cc3ccc(cc3)Cl)Cl RJF01700 Cc1cc(no1)C(=O)Nc2cccc(c2)COC(=O)c3cc(on3)C HTS07156 COC(=O)c1ccc(c(c1)NC(=O)Nc2ccc(cc2)F)C(=O)OC HTS07169 c1ccc(cc1)c2ccc(cc2)c3csc(n3)N/N=C\4/c5ccccc5NC4=O HTS09018 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)N)C1=O HTS07744 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(=O)N/N=C/c3ccccn3 HC00114 COc1cc(cc(c1)OC)Nc2ncnc(n2)N RJF00682 CCN(c1c(cccc1C)C)C(=O)c2c(ccnc2OC)C(F)(F)F RF04611 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OS(=O)(=O)c4ccc(cc4)Cl RJF01549 CC(C)c1ccc(cc1)NNC(=O)CCc2ccccc2 HTS03878 CCc1cccc(c1NC(=S)NCCCC(=O)O)CC RJF01729 CCc1cccc(c1NC2=NCCC(=O)S2)C RJF01737 Cc1ccc(cc1)C(=O)N(Cc2ccccc2)C(C)C HTS07186 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)c5ccc(cc5)F)C1=O HTS07743 c1ccc(cc1)c2cc(=O)n3c([nH]2)ncn3 HTS09028 Cc1cc(ccc1NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl)C(C)(C)C HTS08735 Cc1ccc(cc1)n2c(nnn2)c3cnoc3c4cc(cc(c4)F)F HTS05447 CC(C)(C)c1cc(no1)NC(=O)Nc2ccc(cc2Cl)Cl HTS07315 CS(=O)(=O)N1CCN(CC1)C2c3ccccc3-c4c2cccc4 HTS08767 COC(=O)c1c(ccs1)S(=O)(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08768 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3ccc(c(c3)OC)OC HTS08506 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)Nc3cccs3 HTS08508 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)NN3CCOCC3 HTS03360 c1cc(c(c(c1)F)C(=O)NC(=O)Nc2ccc(c(c2)Cl)S(=O)(=O)Cc3ccc(cc3)Cl)F RJF01705 CN(CCc1ccccn1)C(=O)c2ccccc2C(=O)O HTS09182 c1nc2[nH]c3c(c(=O)n2n1)CCCC3 HTS09072 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccc4c(c3)cc[nH]4 HTS08914 Cc1c(c2ccccc2o1)CC(=O)NNC(=S)Nc3cccc(c3)C(F)(F)F FV00183 Cn1c(cc(n1)C(F)(F)F)C(=O)Nc2cc(cc(c2)Cl)Cl RF04322 CC(c1ccccc1)n2c(nnc2SCc3cc(=O)oc4c3ccc(c4)O)O HTS08002 Cc1cc(c(c(c1)C)n2c(nnc2SCC(=O)Nc3ccccc3)O)C HTS08643 Cc1c(snn1)c2nnc(n2C3CC3)SCC(=O)N(c4ccccc4)C5CCCCC5 HTS08129 COc1c(c(ccn1)C(F)(F)F)C(=O)NC(=O)Nc2ccccc2 RF04650 Cc1c(cc(o1)C(C)(C)C)C(=O)NCc2csc3c2cc(cc3)Cl HTS04471 c1ccc(cc1)c2ccc(cc2)C(=O)c3c(c4c(cc(nc4o3)c5ccccc5)c6cn(nc6c7ccccc7)c8ccccc8)N HTS09064 c1nc2[nH]c3c(c(=O)n2n1)CCC3 HTS09070 CCO.CCOC(=O)N1CCc2c(sc(c2C(=O)c3ccc(cc3)OC)NC(=O)COc4ccc(cc4Cl)Cl)C1 HTS08125 CN(CCc1ccccn1)C(=O)c2cccnc2Oc3ccc(cc3)Cl HTS07948 c1cc(ccc1NC(=S)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl RJF00941 Cc1cc(no1)NC(=S)NCCc2ccccc2 RJF00944 c1cc(cc(c1)Cl)n2c(nnc2SCc3c(cccc3Cl)Cl)C4CC4 RJF00642 CCCc1cc(=O)oc2c1ccc(c2)OS(=O)(=O)c3ccc(cc3)Cl RJF01539 CCCc1cc(nc(n1)c2cccc(c2)C)OC(=O)N(C)C RJF01567 CCCc1cc(nc(n1)NC(=N)Nc2cccc(c2)C(F)(F)F)O RJF01624 CCOC(=O)c1cc2cc(ccc2n1C(=O)c3ccccc3C(=O)O)OCc4ccccc4 HTS08636 CCOC(=O)/C(=C/c1ccco1)/C#N HTS09076 Cc1c2c(c(c(=O)[nH]c2n(n1)c3ccccc3)C#N)c4cccnc4 HTS09077 c1ccc2c(c1)CC(C2)n3c(nnc3SCC(=O)N4CCOCC4)O HTS08334 c1cc2n(c1)-c3ccc(cc3NC2c4cc(cc(c4O)Cl)Cl)C(F)(F)F CD04132 C/C(=N\Oc1nc(ns1)c2ccccc2)/c3cccs3 HTS02602 COc1cccc(c1)N/N=C(\C#N)/C(=O)N HTS09024 Cc1cc(=O)n2c(n1CC(=O)N/N=C/c3ccc(cc3)[N+](=O)[O-])ncn2 HTS09031 CCOC(=O)Cn1cnc2c(c1=O)nnn2Cc3ccc(cc3)F HTS09084 C=CCn1c(nnc1Sc2c3c4c(sc3ncn2)CCCC4)c5ccccc5 HTS09097 c1ccc(cc1)n2c3c(cn2)c(=N)n(cn3)/N=C/c4ccc(cc4)[N+](=O)[O-] HTS09040 Cn1c(nnc1SCc2n[nH]c(=S)n2CC=C)c3ccccc3 HTS08987 Cc1c2c([nH]n1)OC(=C(C2c3cccs3)C#N)N HTS08998 c1ccc(c(c1)N2CCCCC2)OC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl HTS08759 c1nc2[nH]c3c(c(=S)n2n1)CCC3 HTS09071 COc1ccc(cc1)S(=O)(=O)N2CCCC2c3cccs3 CD10416 Cc1ccc(cc1Cl)NC(=O)NCc2csc3c2cc(cc3)Cl HTS04215 c1ccc(cc1)NC(=O)NCc2csc3c2cc(cc3)Cl HTS04217 c1ccc2cc(ccc2c1)CC(=O)Nc3ccc(c(c3)C(F)(F)F)Br HTS03598 CC(c1ccccc1)n2c(nnc2SCC(=O)N3CCOCC3)O HTS08330 c1cc(cnc1)n2c(nnc2SCC(=O)N3CCOCC3)O HTS08332 c1cc(sc1C2OCCO2)[N+](=O)[O-] CD07527 COc1ccc(cc1)/C=N/N=C\2/N(C(=O)CS2)c3cc(ccc3Cl)C(F)(F)F RJF00963 c1cc2c(cc1Cl)c(cs2)CNC(=O)c3c(nccn3)C(=O)O HTS03895 CCCS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/Nc2ccccc2Cl KM00999 c1cc(cc(c1)C(F)(F)F)C(C#N)c2cccc(c2)C(F)(F)F CD10689 Cc1c(snn1)c2nnc(n2C3CC3)SCC(=O)c4ccccc4 HTS08680 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)Nc3cc4ccccc4s3 HTS03845 CN(C)c1c(cc(cn1)[N+](=O)[O-])C(F)(F)F RF05249 CCc1cc(c(s1)NC(=O)CN2CCN(CC2)C)C(=O)c3ccc(cc3)OC HTS08688 COc1cccc(c1O)/C=N/c2ccccc2Nc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03734 c1ccnc(c1)CCNC(=S)Nc2ccc(c(c2)Cl)F RJF00374 Cc1cc(ccc1NC(=S)N(CCO)N)Cl DP01642 CC(C)(C)c1ccc(cc1)/N=C\2/N(C(=O)CS2)Cc3cccs3 RJF00412 Cc1cc(ccc1NNC(=O)c2ccno2)Cl HTS03658 CCCc1ccc(cc1)C(=O)NNc2ccc(cc2)C(C)C HTS03880 Cc1c(snn1)C(=O)NNc2ccc(cc2)C(C)C HTS03882 Cc1nc(c2c(n1)n(c(=S)s2)c3ccccc3)N/N=C/c4ccc(cc4)[N+](=O)[O-] HTS09053 COc1ccc-2c(c1)NC(c3n2ccc3)c4ccc(cc4)F HTS08245 CN1C(=O)C(=Cc2cccc(c2)OC)C(=O)N(C1=O)C HTS08999 c1ccc(cc1)NNC(=O)Nc2cc(sc2Cl)Cl CD10325 c1cc(ccc1SC/C(=N/O)/NC(=O)N)Cl CD11095 c1ccc(cc1)c2nc(no2)c3ccc(cc3)S(=O)(=O)N4CCOCC4 CD10844 CCc1cc(c(s1)NC(=O)CN2CCCC2)C(=O)c3ccc(cc3)OC HTS08686 CCc1cc(c(s1)NC(=O)CN2CCOCC2)C(=O)c3ccc(cc3)OC HTS08687 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC3=NC(ON3c4ccccc4)(C)C CD06701 CC(=O)c1ccccc1OC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD08737 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2)C(F)(F)F)N3CCCCC3 HTS08160 c1ccc2c(c1)cccc2NC(=O)Nc3nnc(s3)C4CC4 HTS08172 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3C)F HTS03533 CNC(=S)NNC(=O)c1c(c2c(c(nnc2s1)c3ccccc3)c4ccccc4)N HTS08991 C=CCNC(=S)NNC(=O)c1c(c2c(c(nnc2s1)c3ccccc3)c4ccccc4)N HTS08992 c1ccc(cc1)C(=O)N2CCOc3c2cccc3 MGH00075 c1cc(c(c(c1)Cl)Oc2c(cc(cn2)N)C(F)(F)F)Cl RF05255 c1ccc(cc1)Sc2ccc(cn2)[N+](=O)[O-] RF05305 Cc1c(c(no1)c2ccccc2)C(=O)n3cccc3 CD03857 Cc1c(c(no1)c2ccccc2Cl)NC(=O)OC(C)c3cccnc3 CD03880 CC(C)(C)c1ccc(cc1)NC(=S)NCCc2ccccn2 RJF00416 CC(C)(C)c1ccc(cc1)/N=C\2/N(C(=O)CS2)CCc3ccccn3 RJF00424 Cc1c(c(c(c(c1C)C)CSc2ccccc2NS(=O)(=O)c3cccc(c3)C(F)(F)F)C)C JP00433 Cc1ccc(cc1)S(=O)(=O)NC(=O)N(C)CCc2ccccn2 HTS08777 CC(C)(CC(=O)N1CCCc2c1cccc2)CC(=O)O HTS08884 Cc1c(c(no1)c2ccccc2Cl)C(=O)Oc3ccc(cc3)I JP00920 C=CCS/C(=N\c1ccccc1)/C(C#N)c2[nH]c3ccccc3n2 HTS09005 CCOC(=O)c1cc(nc(c1C#N)O)c2ccccc2 RF01078 c1cc(sc1/C(=N/OC(=O)C2CC2)/N)[N+](=O)[O-] RF01781 CCN(c1ccc(cc1)Cl)C(=O)c2cnccc2C(F)(F)F RF03970 c1cc(oc1)CNC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS08734 Cc1ccc2cc(ccc2n1)NC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl HTS08746 c1cc(ccc1NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl)N4CCOCC4 HTS08747 COc1cccc(c1)NC(=O)Nc2nnc(s2)C3CC3 HTS08174 Cc1cccc(c1NC(=O)Nc2ccc(cc2)NC(=O)c3ccccc3O)Cl HTS08233 Cc1c(sc(n1)Nc2ccccc2)C(=O)c3ccc(cc3)F HTS08329 Cc1ccc(cc1)S(=O)(=O)CCSc2nnc(n2c3ccccc3)O HTS07988 c1ccc(cc1)n2c(nnn2)c3cnc(nc3c4cccc(c4)C(F)(F)F)c5ccccn5 HTS06853 COc1ccc(cc1)n2c(nnn2)c3cnc(nc3C(F)(F)F)N HTS06854 c1cc(ccc1n2c(nnn2)c3cnc(nc3C(F)(F)F)N)F HTS06855 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N(C)C3CCCCC3 HTS07916 CN(C1CCCCC1)C(=O)c2cc(cc(c2)Cl)Cl HTS07917 c1ccc2c(c1)N(CCO2)C(=O)c3ccc(cc3)Cl MGH00079 c1cc(c(c(c1C(=O)N)OCC(F)(F)F)C#N)OCC(F)(F)F MWP01167 c1c(cc(c(c1[N+](=O)[O-])NC2CCSC2)[N+](=O)[O-])C(F)(F)F CD10419 Cc1cc(cc(n1)NNC(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F CD10507 Cc1cc(nc(n1)c2ccc(cc2)Cl)OC(=O)N(C)C RJF00202 CC(=O)Cn1cnc2c(c1=O)nnn2Cc3ccccc3Cl HTS09085 CCCCC#Cc1ccc(cc1)C2C(=C(NC(=O)N2)C)C(=O)OCC HTS02774 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)C4CCCCC4 JP00921 c1cc(cc(c1)Cl)C(=O)Oc2ccc(cc2)C3CCCCC3 JP00924 c1ccc(cc1)NC(=O)CSc2[nH]c3cc(c(cc3n2)Cl)Cl HTS08890 c1cc(ccc1C(=O)Nc2ccc3c(c2)cc[nH]3)F HTS08911 CCCCCCCCCCCC(=O)Nc1ccc(cc1)OC RG00113 CC(C)c1ccc(cc1)NNC(=O)c2c(cccc2Cl)F HTS03877 CCN(CC)c1ccc(cc1)NC(=O)c2ccc(cc2)Cl HTS03930 COc1ccc(cc1)Oc2ccc(cc2C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6)[N+](=O)[O-] HTS07937 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)NC(C)(C)C#Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C CD04564 c1cc(ccc1/C(=N/OC(=O)c2ccc(cc2)Cl)/N)S(=O)(=O)N3CCOCC3 CD10831 c1cc(ccc1C(=O)NC(=O)Nc2ccc(cc2)Cl)S(=O)(=O)N3CCOCC3 CD10835 c1cc(ccc1C(=O)NC(=O)N2CCOCC2)S(=O)(=O)N3CCOCC3 CD10838 Cc1[nH]c(=O)c2c(n1)n(c(=S)s2)CC=C HTS09061 C=CCNC(=S)NNC(=O)CN1c2ccccc2Sc3c1cccc3 HTS09004 CSc1nc2c(c3ccccc3[nH]2)nn1 HTS09009 c1cc(cnc1)n2c(nnc2SCC(=O)c3ccc4c(c3)OCCO4)O HTS08338 c1ccc(cc1)CN2CCN(CC2)CCNC(=O)Nc3ccccc3 HTS03185 Cc1c(c(on1)C)c2nc(no2)CSc3nnc(n3C(C)c4ccccc4)O HTS08652 c1cc(ccc1C#N)S(=O)(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS08224 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)ON=C3CSC(SC3)C CD09974 CC1SCC(=NOC(=O)c2ccc(cc2)OC)CS1 CD10012 c1cc(cc(c1)S(=O)(=O)Nc2cc(cc(c2)NS(=O)(=O)c3cccc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F CD10911 Cc1cc(ccc1NC(=S)Nc2ccc(cc2)S(=O)(=O)Nc3cc(on3)C)Cl RJF01491 c1ccc(c(c1)C(F)(F)F)NC(=S)Nc2ccc(cc2)S(=O)(=O)NC34CC5CC(C3)CC(C5)C4 RJF01493 C#CCOC(=O)Nc1cc(c(nc1)Oc2c(cccc2Cl)Cl)C(F)(F)F RF05259 CN1C(=O)C(=Cc2ccc(cc2)Cl)C(=O)N(C1=O)C HTS09001 CC(C)(C)c1c(c(n(n1)C)C(C)(C)C)NC(=O)c2ccc(cc2)F HTS03451 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NC(=O)Nc3c(onc3c4ccccc4Cl)C CD03867 c1cc(sc1)C(=O)Nc2ccc3c(c2)cc[nH]3 HTS08306 COc1ccccc1c2nn(c(=O)o2)c3cccc(n3)C(F)(F)F RF05182 Cn1c(cc(n1)C(=O)OC)O CD11878 CCNC(=O)NC(=O)c1cc(sc1)[N+](=O)[O-] DFP00089 c1ccc(cc1)CN(CC(=O)c2ccc(cc2)c3ccccc3)c4ccccc4 HTS08033 c1ccc(cc1)C2Nc3ccccc3C(=O)N2CCCN4CCOCC4 HTS06748 Cc1ccc(cc1Cl)NNC(=O)c2c(ccs2)Cl HTS03634 Cc1ccc(cc1Cl)NNC(=O)c2cc3ccccc3s2 HTS03635 Cc1ccc(cc1Cl)NNC(=O)c2c(ccs2)Br HTS03647 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)S(=O)(=O)c3ccccc3 HTS03618 c1ccc2c(c1)C(=O)N(C(N2)c3cccs3)CCN4CCNC4=O HTS08235 CC1CC(=O)Nc2ccccc2N1C(=O)Nc3ccccc3 HTS08250 c1cc(cc(c1)OS(=O)(=O)c2ccc(cc2)Cl)N3CCOCC3 CD09586 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)/C=N/Nc4c5cnn(c5ncn4)c6ccccc6 HTS09073 C=CCSc1nc2c(c3ccccc3[nH]2)nn1 HTS09010 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC(=O)c4ccc(cc4)Cl HTS09012 Cc1ccc(cc1)NC(=O)NNC(=O)CN2c3ccccc3Sc4c2cccc4 HTS09013 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)NNC(=O)Nc4cccc(c4)Cl HTS09014 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OS(=O)(=O)C RJF01548 C=C1COC(=O)N1c2ccccc2[N+](=O)[O-] RF05449 CN(C)c1ccncc1C(=O)Nc2cc(cc(c2)Cl)Cl RF05517 c1ccc2c(c1)N(C(O2)c3ccc(c(c3)Cl)Cl)S(=O)(=O)c4cc(ccc4Cl)Cl DP01194 CSC1=NCCCN1C(=O)c2ccccc2I DP01349 c1ccc(cc1)Cn2c3c(c(=O)[nH]cn3)nn2 HTS09090 CC(C)(C)c1cs/c(=N\c2ccc(cc2Cl)Cl)/o1 RJF00544 Cn1c(c(sc1=S)C(=O)N/N=C/c2ccc(c(c2)OC)O)N HTS09060 Cc1ccc(cc1Cl)NC(=N)NC(=N)N RJF01060 Cc1ccc(cc1Cl)c2nc(cc(n2)OC(=O)N(C)C)C RJF01077 CCCNC(=S)Nc1ccc(cc1F)F RJF01206 Cc1ccccc1N/C(=N\O)/c2cccnc2 RF05150 c1ccc(c(c1)C(F)(F)F)n2c(noc2=O)c3cccnc3 RF05161 c1ccc(cc1)NC(=O)C(=O)NC(=O)c2c(cccc2Cl)Cl RF03648 c1cc2c(ccc(c2nc1)NC(=O)Nc3ccc(cc3)Cl)Br RF03671 c1ccc(cc1)Cn2c(n[nH]c2=S)c3c(c4c(cc(nc4o3)c5ccc(cc5)Cl)c6ccccc6)N HTS09047 CCCc1ccc(cc1)C(=O)NNc2ccc(c(c2)Cl)C HTS03639 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccc(cc2)C(C)(C)C HTS08075 CN(C)c1ccc(cc1)/C=N/NC2=NCCN2 DP01512 CC(C)(C)c1cc(no1)NC(=O)Nc2ccc(cc2F)F HTS07316 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(on2)C(C)(C)C HTS07955 CCOC(=O)C1=C(NC(=O)NC1c2ccc(s2)c3cccs3)C HTS03202 c1cc(ccc1CS(=O)(=O)Cc2ccc(cc2Cl)[N+](=O)[O-])Cl RF03618 Cc1nc(c(o1)C(F)(F)F)C(=O)NCC(=O)c2ccccc2 RF04224 CN(CCc1ccccn1)C(=O)Nc2ccccc2.Cl HTS08773 c1cc(ccc1CSc2c3c4c(sc3ncn2)CCCC4)F HTS09096 C=CCNc1c2c3c(sc2nc(n1)SCc4ccc(cc4)Cl)CCCC3 HTS08976 Cc1c(cn(n1)c2ccccc2)c3cc(nc4c3c(c(o4)C(=O)c5ccccc5)N)c6ccc(cc6)Cl HTS09063 CC1=C(C(n2c(=O)/c(=C\c3cccnc3)/sc2=N1)c4ccc(cc4)OC)C(=O)OC HTS09065 COc1cc(c(cn1)C(=O)NCc2cc(cc(c2)Cl)Cl)C(F)(F)F RF04316 CC(=O)CSc1nnc(n1c2ccccc2)CSc3nnc(n3CC=C)c4ccccc4 HTS08989 c1ccc2c(c1)c(=O)n(c(n2)S)c3c(cccc3Cl)Cl RJF01464 CC1=NN(C(=O)C1CC(=C)C)S(=O)(=O)c2ccc(cc2)Cl RJF01225 c1cc(cc(c1)[N+](=O)[O-])C(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl RJF01376 CC1=CC(N=C(N1c2ccc(cc2F)F)SCc3ccc(cc3Cl)Cl)(C)C RJF01394 Cc1c(c(n(n1)C)C(=O)O/N=C(/c2ccc(cc2)C(F)(F)F)\N)[N+](=O)[O-] SPB01659 c1cc(cnc1)c2c3c(nc(c2C#N)N)CCCC3 HTS09050 c1cc2c(cc1C(=O)Nc3ccc4c(c3)cc[nH]4)non2 HTS08916 c1cc(cc(c1)C(F)(F)F)/C(=N/OC(=O)c2cc(sc2)[N+](=O)[O-])/N SEW02734 Cc1ccn2c(c1)nc(c2C(=O)NNC(=O)C)C HTS08978 Cc1c(c(on1)C)S(=O)(=O)N2CCC3(CC2)OCCO3 HTS07005 CCOC(=O)Cc1csc(n1)N2C(=O)c3ccccc3C2=O HTS08962 CC(C)(C)c1csc(n1)Sc2ccc(cn2)[N+](=O)[O-] CD08407 CC(C)(C)c1cs/c(=N\c2cc(cc(c2)Cl)Cl)/o1 RJF00565 c1ccc(cc1)COc2ccc(cc2)/C=N/n3c(=O)c4cnn(c4nn3)c5ccccc5 HTS08982 CC(C)(C)NC(=S)Nc1ccc(c(c1)Cl)F RJF01231 c1ccc(c(c1)/C=N/NC(=S)NCC2CC2)Cl RJF01273 c1cc2c(cc1NC(=O)COc3ccc(cc3Cl)Cl)OCCO2 HTS08791 CN(CCc1ccccn1)S(=O)(=O)c2cccc(c2)Cl.Cl HTS09194 c1ccc(cc1)C(CN2CCOCC2)O HTS08840 Cc1c(c(no1)c2ccccc2)C(=O)N(C)CCc3ccccn3 HTS09189 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/n4c(n[nH]c4=S)c5ccncc5 HTS09928 c1cc(ccc1S(=O)(=O)Cc2cc(sc2Cl)Cl)Cl CD11588 c1c(csc1[N+](=O)[O-])C(=O)NC(=S)N2CCCCC2 DFP00150 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)c5n[nH]c(=S)n5c6ccc(cc6)Cl)N HTS08996 COc1ccc(c(c1)S(=O)(=O)Nc2ccc3c(c2)C(=O)OC3)OC HTS04222 c1ccc(cc1)N/N=C(\C#N)/C(=O)N HTS09023 c1cc2c(cc1Cl)c(cs2)CNC(=O)c3ccno3 HTS04230 Cc1c(cccc1Cl)NC(=S)N(C)/N=C/c2cc(c(c(c2)OC)OC)OC DP01656 c1cc2c(cc1Cl)c(cs2)CNS(=O)(=O)c3cc(sc3Cl)Cl HTS04207 c1cc(sc1)S(=O)(=O)NCc2csc3c2cc(cc3)Cl HTS04208 CCCc1cnc(nc1)N2CCN(CC2)CC(=O)Nc3ccccc3 HTS03940 c1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)NN HTS08981 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2c3ccccc3)OC(=O)N(C)C HTS08661 c1ccnc(c1)/C(=N/OC(=O)c2cc(sc2)[N+](=O)[O-])/N SEW02736 c1ccc2c(c1)cccc2c3nnc(o3)c4cc(cnc4)c5cccs5 HTS08784 Cc1c(sc(n1)c2ccccc2)C(=O)NNC(=O)c3cccc4c3cccc4 HTS08785 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)NNC(=S)Nc5ccccc5)N HTS08994 c1ccc(cc1)c2nnc(n2c3ccccc3)SCC(=O)N/N=C/c4ccc(cc4Cl)Cl HTS08980 CN(C)c1cc(oc(=O)c1Cl)c2cccc(c2)[N+](=O)[O-] CD11158 CS(=O)(=O)CS(=O)(=O)Oc1ccc(c(c1)Cl)Cl CD11200 c1ccc2c(c1)cc(s2)NC(=O)N3CCC(CC3)C(=O)N HTS03842 c1ccc2c(c1)cc(s2)NC(=O)N3CCN(CC3)Cc4c(cccc4Cl)F HTS03843 C=CCn1c(nnc1SCc2n[nH]c(=S)n2c3ccccc3)c4ccccc4 HTS08988 c1cc(c(c(c1)Cl)CCNC(=O)NC(=O)Cc2c(cccc2Cl)F)F CD08243 c1ccc(cc1)S(=O)(=O)NCc2csc3c2cc(cc3)Cl HTS04202 Cn1cc(nc1)S(=O)(=O)NCc2csc3c2cc(cc3)Cl HTS04205 Cc1cc(n(n1)c2ccccc2)NC(=O)Nc3ccccc3 HTS09082 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)Nc3ccccc3)C HTS06897 Cc1cccc(c1NC(=O)Nc2ccc(cc2)N3CCCCC3)Cl HTS08420 CCc1cccc(c1NC(=O)Nc2ccc(cc2)N3CCCCC3)C HTS08422 COC(=O)c1c(ccs1)NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS08744 COC(=O)c1ccccc1NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS08745 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccccc3 HTS08249 c1cc(cc(c1)Sc2c3c(ccs3)nc(n2)C(F)(F)F)C(F)(F)F SEW02806 CCN(c1cccc2c1cccc2)S(=O)(=O)c3ccc(cc3)F HTS10681 CN(C)NC(=O)NC(=O)c1ccc(o1)[N+](=O)[O-] SPB00927 C/C(=C(/C(=O)c1c(cccc1F)F)\C(=O)OC)/NC SPB00936 c1cc(ccc1/C=N/NC(=O)Cn2c3c(c(=O)n4c2ncn4)CCC3)[N+](=O)[O-] HTS09960 CCCc1c(c(nc(n1)SCC(=O)c2ccccc2Cl)O)C RJF01922 CCN(Cc1ccc(cc1OC)OC)C(=O)c2cnc(cc2C(F)(F)F)OC RF04480 CC(C)(C)c1ccc(cc1)c2nc(on2)CSc3nnc(n3Cc4ccco4)O HTS09149 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CCC(=O)O HTS09160 c1ccc(cc1)Oc2ccc(cc2)NC(=O)CCCC(=O)O HTS09154 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)N/N=C/c4cccs4)C#N HTS09894 Cc1nc2c(c(=O)n1/N=C/c3ccc(cc3Cl)Cl)sc(=S)n2CC=C HTS09900 Cc1nc(c(o1)C(F)(F)F)C(=O)NNC(=O)c2ccccc2Cl RF04206 COc1ccc(cc1)N(Cc2ccccn2)C(=O)c3ccc(cc3)F HTS10583 CCN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04302 c1cc(ccc1/C=N/NC(=O)Cn2c3c(c(=O)n4c2ncn4)CCC3)Cl HTS09961 c1ccc(c(c1)C(F)(F)F)NC(=S)NNS(=O)(=O)c2ccc(cc2)Cl SPB00991 c1ccc(cc1)c2csc(n2)N/N=C\3/c4ccccc4NC3=O HTS09015 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)NCc3csc4c3cc(cc4)Cl)Cl HTS04472 c1cc(ccc1NNC(=O)c2ccc(cc2F)F)S(=O)(=O)N HTS04474 CNc1ccccc1C(=O)N/N=C/c2ccc3c(c2)OCO3 DP01751 c1cc(cc(c1)Cl)C(=O)Nc2ccc(c(c2)Cl)N3CCOCC3 DP01814 CCN(CC)c1ccc(cc1)NC(=O)c2cccs2 HTS03924 CCN(CC)c1ccc(cc1)NC(=O)Nc2c(cc(cc2Br)C(C)C)Br HTS03918 CCN(CC)c1ccc(cc1)NC(=O)c2ccccc2 HTS03925 c1ccc2c(c1)CC(C2)n3c(nnc3SCC(=O)c4ccc5c(c4)OCCO5)OC(=O)c6cccs6 HTS08664 c1ccc2c(c1)c(c(s2)C(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl)Cl HTS07321 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc3c(c2)cc[nH]3 HTS08923 Cc1[nH]c(=O)c2c(n1)Oc3c4ccccc4oc(=O)c3C2c5ccc(cc5)[N+](=O)[O-] HTS09877 CCN(Cc1cccc(c1)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04335 COc1cc(c(cn1)C(=O)NCc2cccc(c2Cl)Cl)C(F)(F)F RF04357 CCN(Cc1cccc(c1Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04363 c1ccc(cc1)c2c(cn(n2)c3ccccc3)C=C(C#N)C#N HTS09081 c1ccc2c(c1)nc3n2c(c4c(c3C#N)CCC4)N5CCCCC5 HTS09908 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)O/N=C(/c3cccc(c3)C(F)(F)F)\N SEW02870 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)O/N=C(/c3ccc(cc3Cl)Cl)\N SEW02872 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3cccs3 HTS08852 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3cccc(c3Cl)Cl HTS08859 CC1CCc2c(sc(c2C#N)NC(=O)c3ccco3)C1 HTS09931 c1ccc(cc1)CC2(CC2)NC(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04296 C#Cc1cccc(c1)n2c(=O)c3ccccc3[nH]c2=S FV00062 c1cc(ccc1S(=O)(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl)Cl HTS07350 c1cc(ccc1NC(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl)F HTS08288 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3ccc(nc3)Oc4c5ccc(cc5ncn4)Cl HTS08289 CC(C)(CC(=O)Nc1cc(nn1C)c2ccc(cc2)Cl)CC(=O)O HTS08050 Cc1ccc(cc1)C(=O)NNC(=O)c2cc(c(s2)C(F)(F)F)c3ccccc3 SEW02917 c1c(cc(c2c1COCO2)CSCCO)[N+](=O)[O-] SEW03618 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc4c(c3)cc[nH]4)Cl HTS08925 CCOC(=O)CS/C(=N\c1ccccc1)/C(C#N)c2[nH]c3ccccc3n2 HTS10015 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F HTS03614 c1ccc(cc1)n2c(nnc2SCC(=O)N)c3ccco3 HTS09933 c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)F)c4ccco4 HTS09934 CN1C(=O)C(=Cc2cn(nc2c3ccc(cc3)[N+](=O)[O-])c4ccccc4)C(=O)N(C1=O)C HTS09935 Cc1ccc(c(c1)C)n2c(n[nH]c2=S)CC#N HR00191 c1ccc(cc1)Sc2cc(c(cn2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F RF04419 c1cc(ccc1NC(=O)c2cnc(cc2C(F)(F)F)NC3CCCCC3)Cl RF04432 COc1cc(cc(c1OC)OC)C(=O)ON=C2C3CC4CC(C3)CC2C4 JP00899 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)Nc3ccc(c(c3)OC4CCCC4)OC)C HTS06898 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)Nc3ccc(cc3)OCc4ccccc4)C HTS06899 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2cc(nn2C)c3ccc(cc3)Cl HTS08056 c1ccc(cc1)NC(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08790 c1ccc(cc1)c2c(n3c(n2)SCC3)/C=N/O SEW03639 c1ccc(cc1)COc2ccc(cc2)/C=N/n3cnc4c5c(c(nnc5sc4c3=O)c6ccccc6)c7ccccc7 HTS10014 CC1CCc2c(sc(c2C#N)NC(=O)c3cccs3)C1 HTS09932 c1ccc2c(c1)CC(C2)n3c(nnc3SCC(=O)c4ccc5c(c4)OCCO5)O HTS08340 c1cc(sc1)CNC(=O)c2ccc(cc2)F HTS08417 c1ccc(cc1)NC(=S)N2CCC(CC2)C3CCN(CC3)C(=S)Nc4ccccc4 CD04746 C/C(=N\OC(=O)c1c(cccc1F)F)/c2c(cccc2F)F CD04785 c1ccc2c(c1)nc(c(n2)C(F)(F)F)C(=O)N/N=C/c3ccc(cc3)C(F)(F)F HC00115 COc1ccccc1NC(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS02513 Cn1c(cc(n1)c2ccc(cc2)Cl)NC(=O)Nc3ccccc3 HTS08058 COc1ccc(c(c1)NC(=O)C(=O)NCc2ccccc2)OC JPV00087 Cc1ccc(c(c1)C)C(C)NC(=O)C(=O)Nc2cccc(c2)C(F)(F)F JPV00095 Cc1c(c(n(n1)C)C)NC(=O)Nc2ccccc2 CD09917 Cc1cc(n2c3ccccc3nc2c1C#N)N4CCOCC4 HTS10018 CCOC(=O)CSc1c(c(=O)n(c(=S)n1c2ccccc2)c3ccccc3)C(=O)OCC HTS10019 Cc1cc(no1)CN2C(=O)c3ccccc3S2(=O)=O HTS10028 c1cc(cc(c1)NC(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl)C(F)(F)F HTS08295 c1cc2c(cc1Cl)ncnc2Oc3ccc(cn3)NC(=O)CCCC(=O)O HTS08298 c1cc(ccc1S(=O)(=O)CCC#N)Cl SEW00730 c1cc(cc(c1)NC(=S)N2CCC(CC2)CC3CCN(CC3)C(=S)Nc4cccc(c4)C(F)(F)F)C(F)(F)F JP00980 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NNC(=O)c3ccco3 RJF02081 Cc1ccccc1C(=O)O/N=C(/CCSc2ccc(cc2)Cl)\N SEW00741 c1cc(c(c(c1)Cl)Cl)NC(=O)Nc2ccc(cc2)N3CCCCC3 HTS08418 CN(C)C(=O)Oc1nnc(n1C2CC2)SCCS(=O)(=O)c3ccc(cc3)F HTS08660 Cc1nc(cn1C)S(=O)(=O)N(C)C2CCCCC2 HTS08355 Cn1c(cc(n1)c2ccc(cc2)Cl)NS(=O)(=O)c3cccc4c3non4 HTS08065 c1ccc2c(c1)C(=O)N(C(N2)c3cccs3)CCCN4CCOCC4 HTS08234 c1ccc(c(c1)CO)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl JPV00042 c1ccc(c(c1)n2ccnc2SCc3c(cccc3Cl)Cl)Cl CD09959 c1cc(ccc1/C=C/C(=O)c2ccc(o2)c3ccc(cc3F)F)Cl CD10939 CCNC(=S)NNC(=O)CN1c2ccccc2Sc3c1cccc3 HTS09850 CC(=O)Nc1cc(nn(c1=O)c2ccc(cc2)Cl)C(=O)c3cccs3 HTS08477 CCc1c(c(=O)n(nc1C(=O)OC)c2ccc(cc2)C)C#N HTS08478 CCOC(=O)c1c2csc(c2c(=O)n(n1)c3ccccc3)NC(=O)C HTS08479 Cc1ccc(cc1C)NC(=S)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F JP00983 c1cc(cc(c1)Cl)C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F JP00984 c1cc(ncc1N)OCC(F)(F)F RF05263 COc1ccc(s1)/C=C(\C#N)/S(=O)(=O)c2ccccc2Cl KM01149 c1c(cc(cc1C(F)(F)F)N/C=C(\C#N)/S(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F KM01260 C=CC(=O)NCc1ccc(cc1)c2csnn2 SEW00916 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)c3ccncc3 HTS09852 CC1CCc2c(sc3c2c(ncn3)SCC(=O)N/N=C/c4ccc5c(c4)OCO5)C1 HTS09856 CCCc1c(cnn1c2ccccc2)C(=O)N3CCC(CC3)c4ccccc4OC HTS03524 Cc1ccc(cc1Cl)NNC(=O)C2CCC2 HTS03644 c1cc(c(cc1[N+](=O)[O-])C(=O)NNC(=O)CC#N)N DP01081 CN(C)c1ccc(cc1)C(=O)NNC(=O)c2cc(ccc2N)Cl DP01069 c1cc(oc1)C(=O)NNC(=O)c2cc(ccc2N)Cl DP01087 C1CSCCN1C(=O)C23CC4CC(C2)CC(C4)C3 CD08935 Cc1c(c(n[nH]1)C)Cc2c(cccc2Cl)Cl CD08959 c1c(c([nH]n1)/C(=N/O)/N)Cl RF05327 C#CCOC(=O)Nc1ccccc1[N+](=O)[O-] RF05443 c1cc(c(c(c1)Cl)Oc2ccc(cn2)NC(=O)CSCC(=O)O)Cl HTS11136 c1cncc2c1C(=O)N(C2=O)CO HTS09588 COc1ccc(cc1NC(=O)N2CCN(CC2)c3ncccn3)Cl HTS10749 c1ccc(cc1)c2c3c4c(c(=O)n(c(=O)[nH]4)c5ccc(c(c5)Cl)Cl)sc3nnc2c6ccccc6 HTS08995 c1ccc(cc1)c2c3c4c(c(=O)n(cn4)/N=C/c5ccc(cc5)[N+](=O)[O-])sc3nnc2c6ccccc6 HTS08997 COc1ccc(cc1)C(=O)CSc2nnc(n2c3cccnc3)O HTS09139 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)Oc3ccccc3 HTS09153 c1ccc(cc1)S(=O)(=O)/C(=N/Nc2ccc(cc2)F)/C#N KM01277 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)NNC(=S)Nc4ccc(c(c4)Cl)Cl)C#N HTS09975 c1ccc(cc1)C2=CC(n3c(=O)/c(=C/c4ccc(cc4)Cl)/sc3=N2)c5cn(nc5c6ccc(cc6)Cl)c7ccccc7 HTS09978 CSc1c(c(c(s1)C(=O)O)c2ccccc2Cl)C#N KM02566 c1cc2c(cc1OC(F)(F)F)cc([nH]2)C(=O)NN KM09295 CN(C)c1ccc(cc1)NC(=O)Nc2ccccc2F HTS10996 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)Nc3ccc(cc3)N4CCCCC4 HTS09305 c1cc(ccc1N2CCN(CC2)C(=O)c3cc4cc(ccc4[nH]3)Cl)F HTS09329 COc1cc(cc(c1OC)OC)C(=O)Nn2c(=O)c3ccccc3nc2S DP01151 CCOC(=O)Cc1csc(n1)NC(=O)CCCC(=O)O HTS08087 C#Cc1cccc(c1)NC(=O)NC(=O)Cc2c(cccc2Cl)F CD07963 c1ccc(cc1)NC(=O)N2CCC(C(=C2)C(=O)N)C(F)(F)F RF04553 c1ccc(c(c1)/C=N/N=C\2/N(C(=O)CS2)c3cccc(c3)F)OC(=O)C4CC4 RJF01022 Cc1ccc(n1C)CNC(=O)Nc2ccccc2 HTS10872 c1cc(c(c(c1)Cl)CSc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)F SPB00412 CC(C)Oc1cccc(c1)NC(=O)c2cnccc2C(F)(F)F RF03967 Cc1cc(ccc1NC(=S)N(C)N)Cl DP01655 CN(C)c1ccc(cc1)/C=N/Nc2cccc(c2)C(F)(F)F DP01636 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=O)Cn3c(=O)c(c(c(n3)c4ccccc4)c5ccccc5)C#N HTS09984 CCNc1nc2c(s1)cc(cc2Cl)Cl RF04018 c1cc(ccc1C(=O)NNC(=O)c2cnccc2C(F)(F)F)Cl RF04051 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2ccccc2 HTS08090 CCO.CCOC(=O)N1CCc2c(sc(c2C(=O)c3ccc(cc3)Cl)N)C1 HTS08122 CCC(C)Sc1cc(c(cn1)C(=O)Nc2ccc(cc2)Cl)C(F)(F)F RF04416 CCSc1c(c(ccn1)C(F)(F)F)C(=O)Nc2c(cccc2C)C RF04607 c1ccc2c(c1)CC(C2)NCC(=O)Nc3ccccc3N4CCOCC4 HTS07835 CCOC(=O)Cc1csc(n1)NC(=O)Nc2cccc3c2cccc3 HTS08078 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS08081 Cn1cc(c(n1)/C=N/Nc2ccccc2)Br RF04136 Cn1cc(c(n1)/C=N/Nc2cc(cc(c2)Cl)Cl)Br RF04138 c1ccc(cc1)c2csc(n2)NC(=O)c3ccc(c(c3)Cl)F RJF00483 Cc1nc(c(o1)C(F)(F)F)/C(=N/O)/N RF04256 Cc1nc(c(o1)C(F)(F)F)/C(=N/OC(=O)c2cccc(c2)Cl)/N RF04264 Cc1cc(=O)n2c(n1CC(=O)NNC(=S)Nc3ccc(cc3)Cl)ncn2 HTS09033 c1ccc(c(c1)/C=N/NC(=S)Nc2cc(ccc2Cl)C(F)(F)F)Cl RJF00950 CC1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)c4ccccc4)C1 HTS09087 CCOC(=O)CSc1c2c3c(sc2ncn1)CCCC3 HTS09095 CC1CCc2c(sc3c2c(ncn3)SCc4ccc(cc4)[N+](=O)[O-])C1 HTS09094 c1cc(cc(c1)Cl)C(=O)NNC(=O)c2cnccc2C(F)(F)F RF04085 CCN(c1ccc(cc1Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)NC RF04474 Cc1cc(cnc1O)I RF04498 c1cc(cc(c1)F)NC(=S)NCCNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03712 c1cc(cc(c1)C(F)(F)F)C(=O)NCCNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03726 COc1c(c(ccn1)C(F)(F)F)C(=O)NC(=O)Nc2c(cccc2F)F RF04719 Cc1cccc(c1NC(=O)NC(=O)c2c(ccnc2OC)C(F)(F)F)C RF04722 Cc1c(snn1)c2nnc(n2C3CC3)SCC(=O)Nc4ccc5c(c4)OCCO5 HTS08130 CCc1cc(c(s1)NC(=O)CSc2nnc(n2C3CC3)c4c(nns4)C)C(=O)c5ccc(cc5)OC HTS08671 c1cc(ccc1NNC(=O)c2c(ccs2)Cl)S(=O)(=O)N HTS04475 c1cc(ccc1/C=N/Nc2c3c4c(sc3ncn2)CCCC4)Cl HTS09853 c1c2cc(c(=O)oc2c(cc1Cl)Br)C(=O)O HTS11322 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccsc3 HTS10689 c1cc(cnc1)C(=O)NNC(=S)N SPB00551 CCOC(=O)c1c2c(sc1NC(=S)NCc3ccccc3)CC(CC2)C HTS09955 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)NNC(=S)Nc3cc(ccc3Cl)Cl RJF01961 COc1cccc(c1)CNC(=O)c2cc3cc(ccc3[nH]2)Cl HTS09320 Cc1cc(c(o1)C)C(=O)Nc2cc(sc2)c3ccc(cc3)Cl HTS09395 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)c3c(nccn3)C(=O)O HTS09398 Cc1c(c(on1)C)C(=O)Nc2nc3ccc(cc3s2)Cl HTS08909 Cc1ccc(c(c1)C)NC(=O)NC(=O)c2cnccc2C(F)(F)F RF04502 c1ccc(cc1)/C(=N/O)/Nc2cccc(c2)Cl RF05112 c1cc(c(c(c1)Cl)/C(=N/OC(=O)c2cc(cc(c2)Cl)Cl)/N)Cl SPB00375 Cc1[nH]c(=O)c2c(n1)Oc3c4ccccc4oc(=O)c3C2c5cccc(c5)OC HTS09879 Cc1cc(ccc1Br)NC(=S)NNC(=O)c2cccc(c2)[N+](=O)[O-] SEW00920 c1cc(cc(c1)[N+](=O)[O-])C(=O)NNC(=S)Nc2ccc(cc2)F SEW00921 CSc1c(c(sn1)SC)C(=O)NC(=O)OCc2ccccc2 SEW00964 Cc1c2c(c3c(c(oc3nc2n(n1)c4ccccc4)C(=O)c5ccc(cc5)Br)N)c6cccnc6 HTS09080 c1ccc(c(c1)/C=N/c2ccccc2Nc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])O CD03732 CN1C(=O)C(=Cc2ccc(cc2)[N+](=O)[O-])C(=O)N(C1=O)C HTS09003 CC(CO)(CO)NC(=S)NC1CC1 RJF00390 c1ccc(cc1)c2cc(nc3c2c4c(o3)c(=O)n(cn4)/N=C/c5ccc(cc5)Cl)c6ccccc6 HTS09037 c1cc(c(c(c1)Cl)C(=O)NNc2ccc(cc2)S(=O)(=O)N)F HTS04477 c1cc(oc1)Cn2c(nnc2SCC(=O)N3CCOCC3)O HTS08333 COc1ccc(cc1)C2c3cccn3-c4ccc(cc4N2)OC HTS08244 CSc1nnc(n1Cc2ccccc2)c3c(c4c(cc(nc4o3)c5ccc(cc5)Cl)c6ccccc6)N HTS09048 Cc1ncc(c(n1)c2ccccc2)C(=O)O CC20101 c1cc2c(cc1Cl)C(CCS2)O SEW01955 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccsc2)C(=O)OC SEW02066 c1cc(cc(c1)C(F)(F)F)/C(=N/OC(=O)c2cccc(c2)Cl)/N SEW02402 Cc1ccc(cc1Cl)NC(=O)N(C)CCc2ccccn2.Cl HTS08269 c1ccc(cc1)C(=O)CN2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS09210 CCOC(=O)c1cnn(c1NC(=O)Nc2cccc(c2)Cl)c3ccccc3 HTS09925 CCSc1c(c(ccn1)C(F)(F)F)C(=O)Nc2ccc(cc2Cl)Cl RF04602 CC(=O)NNc1ccc(cn1)C(F)(F)F RF04810 CCN(CC)CC(=O)N1c2ccccc2Sc3c1cccc3 HTS09939 c1ccc2c(c1)cccc2NC(=O)OCc3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F HTS10520 CCOC(=O)/C(=C/c1cccnc1)/C#N HTS09881 c1ccc(cc1)n2c3c(cn2)c(=O)n(cn3)CC(=O)c4ccc(cc4)Cl HTS09882 CC1=C(C(NC(=S)N1)c2ccc(cc2)OC)C(=O)OC HTS09891 COc1c(c(ccn1)C(F)(F)F)C(=O)NC(=O)Nc2c(cccc2Cl)Cl RF04723 Cc1c(cnn1c2ccccc2)CO CC15509 COC(=O)c1cc(ccc1S(=O)(=O)Cc2ccc(cc2)Cl)NC(=O)NC(=O)c3c(cccc3Cl)Cl RJF01698 c1cc(sc1)C(=O)Oc2nnc(n2C3CC3)SCC(=O)c4ccc5c(c4)OCCO5 HTS08665 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)c4ccco4 HTS09078 CCc1cc(c(s1)NC(=O)CN2CCCCC2)C(=O)c3ccc(cc3)OC HTS08678 c1cc(sc1)S(=O)(=O)Nc2ccc3c(c2)cc[nH]3 HTS08921 Cn1cc(nc1)S(=O)(=O)Nc2ccc3c(c2)cc[nH]3 HTS08924 CC(=O)Nc1ccc(cc1)NC(=O)c2ccccc2C(=O)O HTS08562 C/C(=N\NC(=S)NCc1ccco1)/c2cc(cc(c2O)Cl)Cl CD03805 CC1CN(CC(O1)C)c2ccc(cc2)NC(=S)NCc3ccco3 RJF00394 COc1ccc(cc1OC)CCNC(=S)Nc2c(cc(cc2Br)F)Br RJF00409 CC(C)(C)c1ccc(cc1)NC(=S)NCCc2ccncc2 RJF00417 c1c(cc(c(c1Br)NC(=S)NN)Br)F RJF00419 CC(C)(C)c1ccc(cc1)NC(=S)NCc2cccnc2 RJF00420 c1cc(sc1)/C=N/NC(=O)CC#N HTS09059 CC(C)c1ccc(cc1)NNC(=O)c2ccno2 HTS03884 CC(C)c1ccc(cc1)NNC(=O)C2CCC2 HTS03885 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccc(cc3)C(C)C HTS03886 CC1CC(c2c1nc3ccccc3c2c4ccccc4)(C)C HR00182 Cc1ccc(c(c1)Cl)NC(=S)Nc2ccccc2Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F JP00474 c1cc(c(c(c1)Cl)C(=O)NC(=O)Nc2ccc(c(c2)C(F)(F)F)S(=O)(=O)Cc3ccc(cc3)Cl)Cl RJF01701 c1cc(sc1)CCNC(=O)C2CC2 SEW01028 c1cc(ccc1SCc2ccsc2C#N)Cl SEW01660 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=O)c2ccccc2N DP01074 CC(=O)Nc1ccc(cc1)NC(=O)Nc2cccc(c2)OC HTS08573 CC(=O)Nc1ccc(cc1)NC(=O)Nc2cc(ccc2OC)Cl HTS08578 c1ccc(cc1)c2cc([nH]n2)NC(=O)CSCC(=O)O HTS08707 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=O)c2cc(ccc2N)Cl DP01079 c1ccc(cc1)CN2CCc3c(sc4c3c(=O)n(c(=S)[nH]4)c5ccccc5)C2 HTS09944 COc1ccc(cc1)/C=N/Nc2c3c4c(sc3ncn2)CCCC4 HTS09946 c1cc(sc1)/C=N/Nc2c3c4c(sc3ncn2)CCCC4 HTS09948 CSc1cccc(c1)NC(=O)C(=O)NCc2ccccc2 JPV00077 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)Nc2ccc(cc2)C(F)(F)F HTS11104 COc1c(csc1Cl)C(=O)O/N=C/c2c(cccc2Cl)Cl KM00601 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=S)NC(=O)C=C RJF01749 Cc1c(snn1)c2nnc(n2C3CC3)SCC(=O)c4ccc5c(c4)OCO5 HTS08681 CCc1cc(c(s1)NC(=O)CN2CCN(CC2)c3ccccc3)C(=O)c4ccc(cc4)OC HTS08689 c1csc2c1sc(c2)C(=O)NN SEW02081 CC(C)(C)C(=O)NNC(=O)c1cc2c(s1)ccs2 SEW02172 c1ccc(cc1)c2c3ccccc3c(=O)n(n2)c4ccc(c(c4)Cl)Cl DP00666 c1cc(oc1)C(=O)NNC(=O)c2cc(ccc2N)[N+](=O)[O-] DP01089 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)c2cc(ccc2N)Cl DP01097 COc1cc(cc(c1OC)OC)C(=O)NNC(=O)c2cc(ccc2N)[N+](=O)[O-] DP01099 CCc1cc(c(s1)NC(=O)CSc2nnc(n2C)c3ccc4ccccc4c3)C(=O)c5ccc(cc5)OC HTS08672 CC1CCc2c(sc3c2c(=O)n(c(n3)SCc4ccc(cc4)F)CC=C)C1 HTS09088 c1cc2c(cc1C(=O)CSc3[nH]c4cc(c(cc4n3)Cl)Cl)OCO2 HTS08886 c1ccc(c(c1)NC(=O)CSc2[nH]c3cc(c(cc3n2)Cl)Cl)Cl HTS08888 c1ccc(cc1)C(=O)CSc2[nH]c3cc(c(cc3n2)Cl)Cl HTS08889 Cc1cc(cc(c1)OC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl)C HTS08750 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)/C(=N/O)/N SEW02529 c1cc(sc1)c2ccc(s2)C(=O)O/N=C(/c3ccc(cc3)C(F)(F)F)\N SEW02611 c1cc(cc(c1)C(F)(F)F)/C(=N/OC(=O)c2ccc(s2)c3cccs3)/N SEW02612 c1ccc2c(c1)ncn2C3CC(=O)N(C3=O)c4ccc(cc4)F DP01244 CN1CNC(=NC1)SCc2cccc(c2)C#N.Br DP01301 Cc1c2c(n(n1)c3ccccc3)NC4=C(C2c5ccc(cc5)Cl)C(=O)CC(C4)(C)C HTS09954 Cc1cc(n(n1)c2ccccc2)NC(=O)c3ccc(cc3)F HTS09956 Cc1c2c(c3c(c(oc3nc2n(n1)c4ccccc4)C(=O)c5ccc(cc5)Cl)N)c6ccc(cc6)Cl HTS09959 c1ccc(cc1)c2nc(cs2)CSc3nnc(n3Cc4ccco4)c5ccc(cc5)C(F)(F)F HTS11111 CC(C)(C)c1cc2ncc(c(n2n1)N)C#N KM00649 CC(C)(C)c1ccc(cc1)c2csc(n2)N SPB00134 CCN/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Br KM00759 CNC(=O)Nc1ccc(cc1)C2SCCS2 KM00784 CC(C)(C)OC(=O)N1CCc2c(sc(c2C(=O)c3ccc(cc3)OC)N)C1 HTS08691 c1cc(ccc1C2SCCS2)OC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl HTS08754 Cc1c(sc(n1)c2ccc3c(c2)CCO3)c4nnc(o4)c5cccc6c5cccc6 HTS08783 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=S)N HTS09987 c1ccc(cc1)c2c3c(nc(c2C#N)/N=C/N4CCCCC4)CCCC3 HTS09990 c1ccc(cc1)NC(=O)CSc2nnc(n2Cc3ccco3)O HTS08645 CSC1=NCCN1C(=O)c2ccc(c(c2)Cl)Cl DP01344 c1ccc(c(c1)Cn2c3c(c(=O)[nH]cn3)nn2)Cl HTS09092 CN1CCc2c(sc(c2C#N)NC(=S)Nc3ccccc3)C1 HTS08977 c1cc(ccc1NC(=O)Nc2nc(cs2)c3ccc(c(c3)F)F)F HTS02512 c1cc(oc1)Cn2c(nnc2SCC(=O)c3ccc4c(c3)OCCO4)O HTS08339 c1cc2c(cc1Cl)ncnc2Oc3ccc(cn3)NC(=O)CCC(=O)O HTS08300 COc1ccc(cc1)C(=O)Nc2ccc3c(c2)cc[nH]3 HTS08912 c1ccc(cc1)Sc2c(cccn2)C(=O)Nc3ccc4c(c3)cc[nH]4 HTS08913 CCOC(=O)Cc1csc(n1)NC(=O)Nc2cc(cc(c2)C)C HTS08074 Cc1c(sc(=S)n1CCc2ccc(cc2)Cl)C(=O)/C=C/N(C)C CD09870 c1ccc(c(c1)C(=O)NC(=O)C(=O)Nc2ccc(cc2)Cl)Cl RF03989 CCOc1cccc(c1)NC(=O)c2cnccc2C(F)(F)F RF04001 c1ccc2c(c1)nc(s2)NC(=O)c3cnccc3C(F)(F)F RF04002 c1ccc(cc1)c2cc(n3c(n2)ncn3)N/N=C/c4ccc5c(c4)OCO5 HTS09995 c1nc2c(c3c(s2)CCC3)c(=N)n1N HTS09997 Cc1c2c(c3cc(cc(c3n1)OC)OC)N(CC2)c4cccc(c4)C(F)(F)F HTS10005 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N/N=C/c3cc(cc(c3O)Cl)Cl SPB00149 c1c(cc(c(c1Br)O)Br)/C=N/Nc2c(cncc2Cl)Cl SPB00302 c1cc(c(c(c1)Cl)/C(=N/OC(=O)COc2ccc(cc2Cl)Cl)/N)Cl SPB00367 c1ccc(cc1)c2cc(nc3c2c(c(o3)C(=O)NN)N)c4ccccc4 HTS09993 CN(Cc1ccccc1Cl)C(=O)c2cnccc2C(F)(F)F RF04006 CN(c1nc2cc(ccc2s1)Cl)C(=O)c3cnccc3C(F)(F)F RF04019 CCN(c1nc2cc(ccc2s1)Cl)C(=O)c3cnccc3C(F)(F)F RF04020 CCOC(=O)CS/C(=N/NC(=O)c1c(nc2n1ccc(c2)C)C)/NC HTS10009 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCCS(=O)(=O)c4ccc(cc4Cl)Cl HTS02874 c1cc(ccc1C(=O)NCCN2CCNC2=O)OC(F)(F)F HTS02480 CCOC(=O)c1c2csc(c2c(=O)n(n1)c3ccc(cc3)OC)NC(=O)C HTS08480 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC3CCSC3 CD10068 Cc1ccc(n1c2ccccc2C3C=NNC3=O)C CD10081 CC(C)OC(=O)Nc1cnccc1C(F)(F)F RF04030 C#CCOC(=O)Nc1cnccc1C(F)(F)F RF04031 C1CCN(CC1)CC(=O)NNC(=O)Cn2nc(nn2)N3CCCC3 RJF01898 CCCCCCCC1C(=NN(C1=O)C(=O)c2ccc(cc2)Cl)C RJF01902 c1cc(ccc1c2csc(n2)NC(=O)c3ccc(c(c3)Cl)F)Cl RJF00484 CC1CCc2c(sc3c2c(ncn3)SCC(=O)c4ccc(cc4)Br)C1 HTS10010 Cc1nc(c(o1)C(F)(F)F)c2nnc(o2)c3ccc(cc3)Cl RF04211 Cc1nc(c(o1)C(F)(F)F)c2nnc(o2)c3ccccc3 RF04217 c1cc(sc1)CNC(=S)Nc2c(cc(cc2Br)F)Br RJF00410 c1c(cc(c(c1F)NC(=S)NN)Br)F RJF00432 Cc1c2c(c(s1)NC(=O)C)c(=O)n(nc2C(=O)OC)c3ccccc3 HTS08481 CCOC(=O)c1c2ccc(c(c2c(=O)n(n1)c3ccccc3)N)C#N HTS08483 c1cc(sc1)c2c3c(nc(c2C#N)O)CCCC3 HTS09051 C=CCn1c2c(c(ncn2)N/N=C/c3ccc(cc3)Cl)sc1=S HTS09054 Cc1nc(c(o1)C(F)(F)F)c2ncc(o2)c3ccccc3 RF04226 Cc1nc(c(o1)C(F)(F)F)c2nc(on2)c3cccc(c3)Cl RF04267 Cc1nc(c(o1)C(F)(F)F)c2nc(on2)c3ccc(cc3)Cl RF04268 CCN(CC)C(=O)Oc1c(c(nc(n1)SCC(=O)C(C)(C)C)C)CC=C RJF00450 COc1cccc2c1c(no2)N MO00345 CCN(CC)C(=O)Oc1c(c(nc(n1)SCC(=O)C(C)(C)C)C)Cc2ccc(cc2)C RJF00455 c1cc(ccc1Nc2ncnc(n2)N)Cl RJF00584 c1ccc(c(c1)NC(=S)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl)F RJF02021 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)Nc3ccc(cc3)C(F)(F)F)C HTS08793 COc1cccc(c1c2nn(c(=O)o2)c3c(cc(cn3)C(F)(F)F)Cl)OC RF04820 CCOc1cc(c(cn1)C(=O)NCc2ccc(cc2)Cl)C(F)(F)F RF04311 CNc1nc2c(s1)cc(cc2Cl)Cl RF04017 c1ccc(cc1)C(=O)NNC(=O)c2cnccc2C(F)(F)F RF04063 C=CCn1c2c(c(ncn2)N(Cc3ccccc3)Cc4ccccc4)sc1=S HTS09058 c1ccc(c(c1)C(=O)NC(=O)c2cccs2)O HTS08897 c1ccc(c(c1)C(=O)NC(=O)c2ccc(cc2)F)O HTS08900 Cc1c(c(on1)C)C(=O)N2CCCCC2c3ccccn3 HTS08904 CN(Cc1ccccc1Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04328 CCOC(=O)C1CCc2c1c(c(s2)N)C#N HTS09067 CCOc1cc(c(cn1)C(=O)N(C)Cc2c(cccc2OC)OC)C(F)(F)F RF05408 c1ccc(cc1)c2cc(sc2C(F)(F)F)/C=N/Nc3cccc(c3)C(F)(F)F SEW03699 Cc1c(c(n(n1)C)C(=O)O/N=C(/c2ccc(o2)[N+](=O)[O-])\N)[N+](=O)[O-] SPB01660 c1cc(ccc1n2ccnc2)[N+](=O)[O-] RF03768 Cc1cc(no1)NC(=O)C(=O)NC(=O)c2c(cccc2Cl)Cl RF03652 Cn1cc(c(n1)/C=N/Nc2ccccn2)Br RF04139 Cc1c2c(c(c(nc2n(n1)c3ccccc3)OCC(=O)c4ccc(cc4)Br)C#N)c5cccnc5 HTS09079 Cn1cnc2c(c1=O)nnn2Cc3ccc(cc3)Cl HTS09083 Cc1c(c(no1)c2ccccc2)NC(=O)N(Cc3ccccc3)C(C)C HTS08838 C=CCNC(=S)NNC(=O)c1c(c2c(cc(nc2o1)c3ccc(cc3)Cl)c4ccccc4)N HTS09046 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccccc3OC(F)(F)F HTS08861 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3cccc4c3non4 HTS08864 c1ccc(c(c1)c2nn(c(=O)o2)c3cc(ccn3)C(F)(F)F)Cl RF04915 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F RJF01098 COCCOc1c(cc(cn1)[N+](=O)[O-])C(F)(F)F RF05248 c1cc(c(c(c1)Cl)C(=O)NC(=O)C(=O)Nc2ccc(cc2F)F)F RF03682 c1cc2c(cc(c(c2nc1)N)Cl)Cl RF03784 Cn1c(=O)c2c3c(sc2[nH]c1=S)CCCC3 HTS09086 Cc1nc(c(o1)C(F)(F)F)C(=O)NNC(=O)c2cccc(c2)Cl RF04207 CC1CCc2c(sc3c2c(=O)n(c(n3)SCC=C)Cc4ccccc4)C1 HTS09089 Cn1c(nnc1SCC(=O)N/N=C/c2cn(nc2c3ccc(cc3)Cl)c4ccccc4)c5ccccc5 HTS09066 CC(C)(C#C)NC(=S)NC1CC2CC1C=C2 HR00071 c1cc(c(c(c1)Cl)Oc2ccc(cn2)NC(=O)CCC(=O)O)Cl HTS11132 c1cc(c(c(c1)Cl)Oc2ccc(cn2)NC(=O)c3c(nccn3)C(=O)O)Cl HTS11134 COC(=O)c1cnc(nc1C(F)(F)F)N2CCCN(CC2)C(=O)Nc3ccc(cc3)OCc4ccccc4 HTS03613 CN1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)c4ccccc4)C1 HTS09945 CN1C(=O)C(=Cc2cn(nc2c3ccccc3)c4ccccc4)C(=O)N(C1=O)C HTS10328 Cc1ccc(cc1)NC(=O)N2CCCn3c2nnc3SCc4ccc(cc4)F HTS09884 CC(CC(=O)Nc1ccc(cc1)Cl)C(Cl)(Cl)Cl SEW00886 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)c3ccccc3C(=O)O HTS09400 CS/C(=N\c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/N2CCCCC2.I CD06256 c1cc(cc(c1)S(=O)(=O)N)NC(=O)C2CC(=O)N(C2)Cc3ccco3 HTS09688 Cc1cc(n(n1)C)C(=O)Nc2cc(sc2C(=O)OC)c3ccc(cc3)Cl HTS09403 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N/N=C/c3ccccn3 SPB00148 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Nc3ccc(cn3)C(F)(F)F HTS07881 c1ccc(cc1)Oc2ccc(cc2)NC(=O)c3c(c4ccccc4s3)Cl HTS09162 CN(C)c1ccc(c(c1)Cl)/C=C\2/C(=NOC2=O)c3cccs3 RF01001 Cc1c(c(on1)C)c2nc(no2)CS(=O)(=O)Cc3ccc(cc3)Cl SEW00847 c1cc(cnc1)/C=N/NC(=O)Cn2c3c(c(=O)n4c2ncn4)CCC3 HTS09962 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C(=N/OC(=O)c2cc(sc2)[N+](=O)[O-])/N SEW02735 c1cc(ncc1C(F)(F)F)NC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl HTS08591 CC(C)(C)c1ccc(cc1)Oc2c(c(ncn2)Oc3ccc(cc3)C(C)(C)C)Br SPB00025 CC(C)(C)c1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)ONC(=O)Cc3ccccc3 SPB00353 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3ccc4c(c3)cc[nH]4 HTS08917 COC(=O)c1c(n(nn1)c2cc(cc(c2)Cl)Cl)O SEW00016 c1ccc(cc1)n2c(=O)c3c(c(sc3n(c2=S)c4ccccc4)C#N)OC(=O)c5cccs5 HTS09889 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)c4cccnc4 HTS09875 c1ccc2c(c1)[nH]c(n2)Sc3c4c(c(c5n3c6ccccc6n5)C#N)CCCC4 HTS09909 c1cc(ccc1C(=O)NNC(=O)c2ccc3c(c2)nccn3)C(F)(F)F HTS09186 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)F)S SPB00608 COCCCNC(=O)c1nc2ccccc2c(=O)n1NC(=O)C(Cl)(Cl)Cl CD02926 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc(o2)C(=O)OC HTS08822 Cc1c(c(on1)C)c2nc(no2)CSc3nnc(n3c4cccnc4)O HTS09136 Cc1cc(no1)C(=O)Nc2ccc(cc2)Oc3ccccc3 HTS09163 c1cc(cnc1)n2c(nnc2SCC(=O)c3ccc(cc3)C#N)O HTS09140 c1cc(sc1)/C=N/NC(=O)Cn2c3c(c(=O)n4c2ncn4)CCC3 HTS09963 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(c(c3)Cl)Cl)CCC2C(=O)OCC HTS09970 CCOC(=O)c1c2c(sc1NC(=O)Nc3cccc(c3)Cl)CCC2C(=O)OCC HTS09971 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)NNC(=O)c3cccc(c3)C(F)(F)F SEW02932 CCOC(=O)c1cc2c(nccn2c1)C SEW03497 CN(C)/N=C(/c1ccc(cc1)Cl)\N.I DP01518 COc1ccc(cc1NC(=O)Nc2ccc(cn2)C(F)(F)F)Cl HTS08601 Cc1ccc(cc1Cl)NC(=O)Nc2ccc(cn2)C(F)(F)F HTS08604 c1ccc(cc1)c2cc(on2)C(=O)CSc3nnc(n3c4cccnc4)O HTS09133 c1ccc(cc1)Oc2ccc(cc2)NC(=O)c3ccccc3C(=O)O HTS09158 c1ccc(c(c1)n2cccc2)N3CCCCC3 HTS09161 Cc1c2cc(ccc2sc1C(=O)CSc3nnc(n3c4cccnc4)O)Cl HTS09134 CN(Cc1ccc(c(c1)Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04372 CC(=O)Cn1nc(nn1)c2ccc(cc2)C(F)(F)F SEW00318 c1cc(oc1/C(=N/OC(=O)c2csnn2)/N)[N+](=O)[O-] SEW00656 c1ccc(c(c1)NC(=S)Nc2ccc(cc2)c3csnn3)Cl SEW00801 C=CCn1c(nnc1Sc2c3c(c(c4n2c5ccccc5n4)C#N)CCCC3)c6ccccc6 HTS09911 COc1ccc2cc(ccc2c1)C(=O)O TL00772 Cc1c(c(nc(n1)c2ccccn2)N(C)c3ccccc3)Cl SEW02976 c1ccc(cc1)c2ccc(s2)NC(=O)Nc3ccc(cn3)C(F)(F)F HTS08597 c1cc(sc1)NC(=O)Nc2ccc(cn2)C(F)(F)F HTS08598 COc1cccc(c1)NC(=O)Nc2ccc(cn2)C(F)(F)F HTS08599 COc1ccc(c(c1)CNC(=O)c2cnc(cc2C(F)(F)F)OC)OC RF04464 c1ccc(c(c1)C(F)(F)F)n2c(nnn2)c3ccc(cc3)Cl RF04540 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)NNC(=S)Nc4ccccc4)C#N HTS09976 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)Nc2ccccc2 HTS11129 Cc1c(cn(n1)c2ccccc2)C3C=C(N=C4N3C(=O)CS4)c5ccc(cc5)Cl HTS09981 c1ccc(c(c1)C(=O)Oc2ccc(cc2)I)I JP00927 CCN(c1c(cccc1C)C)C(=O)c2c(ccnc2SCC)C(F)(F)F RF04612 c1cc(ccc1C(=O)O/N=C(/C2(CC2)c3ccc(cc3Cl)Cl)\N)OC(F)(F)F SEW03875 Cc1cc(n2c3ccccc3nc2c1C#N)/N=C\N(C)C HTS10017 c1cc(ccc1NC(=O)COCC(=O)O)OC(F)F HTS09560 c1ccc(cc1)NC(=O)Nc2ccc(cc2)OC(F)F HTS09570 c1ccc2c(c1)cccc2c3nnc(o3)c4ccc5c(c4)nccn5 HTS09760 Cc1cccc(c1C)N(C)C(=O)c2cnccc2C(F)(F)F RF04409 COc1cc(cc(c1OC)OC)C(=O)Nc2ccccc2Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F JP00458 c1ccc(c(c1)NC(=O)c2ccc(cc2)Cl)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F JP00459 CC(=O)Nc1ccc(cc1)OC(=O)c2cccc(c2)Cl JP00934 c1cc(c(cc1Cl)Cl)NC(=O)c2cnc(cc2C(F)(F)F)NC3CCCCC3 RF04433 c1ccc(cc1)c2cc(c3c(c(sc3n2)C(=O)O)N)C(F)(F)F SB02115 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3c(c(cs3)S(=O)(=O)c4ccc(cc4)Cl)C)C HTS06894 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)N3CCCCC3)OC(F)(F)F HTS08421 COC(=O)c1c(c2c(s1)cc(s2)[N+](=O)[O-])NC(=O)C(F)(F)F SEW03214 Cc1c(c(c(c(c1C)C)CS/C(=N/c2ccc(cc2)C(C)C)/N3CCOCC3)C)C JP00554 Cc1ccsc1C(=S)N SEW03532 CC(C)(C)C(=O)Nc1c(cccc1Cl)OC(F)(F)F SEW03573 c1ccc(cc1)c2c(n3c(n2)SCC3)C#N SEW03643 CCc1cc(c(s1)NC(=O)c2ccc(cc2)OC)C(=O)c3ccc(cc3)OC HTS08696 c1cc(sc1)S(=O)(=O)NCc2ccc(cc2)N3CCOCC3 HTS09730 Cc1cccc(c1NC(=O)c2c(ccnc2OC)C(F)(F)F)C RF04606 Cc1nc(c(o1)C(F)(F)F)C(=O)Nc2cccc(c2Cl)Cl RF04637 COC(=O)C1Cc2c3ccccc3[nH]c2C(N1)c4ccccc4 HTS11285 COc1ccccc1NC(=O)Nc2c(ccs2)c3nc4ccccc4s3 HTS10888 Cc1cccc(n1)NC(=S)Nc2cc(c(cc2OC)Cl)OC CD02076 c1cc(ccc1Cn2c3c(c(=O)[nH]cn3)nn2)Cl HTS09093 CCn1c(n[nH]c1=S)CN2c3ccccc3Sc4c2cccc4 HTS09849 c1ccc(cc1)c2c(sc(n2)Nc3ccc4c(c3)OCCO4)C(=O)c5ccccc5 HTS09625 CC(C)NC(=O)NNC(=O)Cn1nc(nn1)c2cccc(c2Cl)Cl RJF02072 CSc1cccc(c1)NC(=S)N2CCC(CC2)CC3CCN(CC3)C(=S)Nc4cccc(c4)SC JP00976 c1cc(c(c(c1)Cl)Oc2ccc(cn2)NC(=O)c3ccc4c(c3)CCO4)Cl HTS09447 Cc1ccc(cc1)S(=O)(=O)N2CCC(CC2)CC3CCN(CC3)S(=O)(=O)c4ccc(cc4)C JP00993 c1ccc(cc1)c2cc([nH]n2)NC(=O)CCCC(=O)O HTS08711 COc1ccccc1NC(=O)OCC#C RF05440 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3)I JP00922 c1ccc(c(c1)n2c(noc2=O)c3cnccc3C(F)(F)F)Cl RF05229 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N(Cc2ccccc2)Cc3ccc(c(c3)OC)OC CD02036 c1ccc(c(c1)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])[N+](=O)[O-])Cl CD02062 COc1cc(cc(c1OC)OC)C(=O)NCc2ccc(cc2)C#N SEW04454 CCOC(=O)c1cn2c(n1)ccc(n2)N3CCCC3 HTS10955 c1ccc2c(c1)nc(s2)c3ccsc3NC(=O)Nc4ccc(cc4F)F HTS11221 c1ccc(cc1)c2c3c4c(c(=O)n(cn4)/N=C/c5ccc(cc5Cl)Cl)sc3nnc2c6ccccc6 HTS10011 c1cc(ccc1C2CCC(CC2)C(=O)NN)Cl MO00405 Cc1c2c(c(s1)NC(=O)C)c(=O)n(nc2C(=O)OC)c3ccc(cc3)OC HTS08482 c1cc(ccc1S(=O)Cc2ccsc2C#N)Cl SEW01663 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc(cc2)C(=O)c3ccc4c(c3)CCC4 JPV00057 CC(C)(C)c1ccc(cc1)c2nc(on2)CSc3nnc(n3c4cccnc4)O HTS09135 CCS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/Nc2cccc(c2)C(F)(F)F KM00998 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/N2CCSCC2 KM01006 CCCCCCCCCCCC(=O)Nc1nccs1 RG00115 c1cnn(c1)c2ccc(cc2)C(=O)O CC18401 c1cnn(c1)c2ccc(cc2)N CC18414 Cc1c(c(c(c(c1C)C)C(=O)c2c(c(c(c(c2Cl)Cl)Cl)Cl)C(=O)NCCc3ccc(c(c3)OC)OC)C)C CD02141 Cc1c(c(c(c(c1C)C)C(=O)c2c(c(c(c(c2Cl)Cl)Cl)Cl)C(=O)NCc3cccnc3)C)C CD02155 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc3c(c2)OCCO3 HTS09630 c1cc(sc1)S(=O)(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS09662 CCc1cccc(c1N(C)C(=O)c2cnccc2C(F)(F)F)CC RF04406 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3ccc4c(c3)nsn4)C HTS11106 c1cc(c(c(c1)Cl)Oc2ccc(cn2)NC(=O)COCC(=O)O)Cl HTS11133 Cc1c(c(c(c(c1C)C)/C=N/NC(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C)C)C SPB00146 Cc1c(c(n(n1)C)NC(=O)OCC#C)[N+](=O)[O-] SPB01688 Cc1nc(c(o1)C(F)(F)F)/C(=N/OC(=O)c2ccccc2Cl)/N RF04263 CC(C(=O)Nc1cc(cc(c1)Cl)Cl)O RF04925 COC(=O)c1cnc(cc1C(F)(F)F)Oc2c(cc(cc2Cl)N)Cl RF04740 c1ccc(cc1)COc2ccc(cc2)NC(=O)OCc3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F HTS10518 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)N/N=C/c4ccc(cc4)Cl HTS09007 c1ccc2c(c1)CC(C2)n3c(nnc3SCC(=O)c4ccc5c(c4)OCCO5)OCC(=O)c6ccc(cc6)F HTS09122 Cc1c2c(c(c(nc2n(n1)c3ccccc3)OCC(=O)c4ccc(cc4)Cl)C#N)c5ccc(cc5)Cl HTS09964 Cc1[nH]c(=O)c2c(n1)Oc3c4ccccc4oc(=O)c3C2c5ccc(cc5)OC HTS09966 CS/C(=C(/C#N)\S(=O)(=O)c1ccc(cc1)Cl)/NCC=C KM01290 CC(=O)NNC(=S)Nc1cccc(c1)F KM01323 c1cc(cnc1)/C=N/Nc2c3c(nc4n2ncn4)CCC3 HTS09968 COc1ccc(cc1)/C=N/NC(=O)CSc2c3c4c(sc3ncn2)CCCC4 HTS09855 COc1cccc(c1)CC(=O)c2ccc(cc2)C#N MO00229 CN(C)C(=O)Oc1nnc(n1C2Cc3ccccc3C2)SCCS(=O)(=O)c4ccc(cc4)F HTS08659 c1cc(ccc1N)S(=O)(=O)Nc2ccc(cc2C(F)(F)F)Cl RJF02118 c1ccc2c(c1)-c3cccn3C(N2)c4ccc(cc4)N5CCOCC5 HTS11093 c1ccc2c(c1)-c3cccn3C(N2)c4ccc(o4)CN5C(=O)c6ccccc6C5=O HTS11094 Cc1cc(nc2c1c3c(o2)c(=O)n(cn3)/N=C/c4ccc(cc4Cl)Cl)c5ccccc5 HTS09919 Cc1ccc(n1C)CNC(=O)Nc2ccc(cc2)C(C)(C)C HTS10871 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccc(cc2)C HTS10600 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccc(cc2)C#N HTS10601 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)S(=O)(=O)c5ccc(cc5)c6cnco6 HTS10651 C#CCSc1nnc(n1c2ccccc2)O SPB00800 CCOC(=O)COc1ccc2c(cc(=O)oc2c1)C(F)(F)F RJF01900 CCCCCCCC1C(=NN(C1=O)S(=O)(=O)c2ccccc2Cl)C RJF01901 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3cc4cc(ccc4[nH]3)Cl HTS09319 c1cc(ccc1c2c(nc([nH]2)c3ccc(cc3)Cl)c4ccc(cc4)Cl)Cl DP01606 Cc1c2c(n(n1)c3ccccc3)OC(=C(C2c4ccc(cc4Cl)Cl)C#N)N HTS09020 COc1cc(cc(c1OC)OC)NC(=N)NC(=N)N RJF00882 c1cc(ccc1NC(=O)CCN2CCOCC2)S(=O)(=O)Nc3cc(cc(c3)Cl)Cl RJF00855 CCOC(=O)c1c(=O)n(c(=S)n(c1SC)c2ccccc2)c3ccccc3 HTS09980 CSc1nc(nc(n1)NC(=O)NS(=O)(=O)c2ccccc2Cl)C3CC3 RF02947 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)N/N=C/c4cn(nc4c5ccc(cc5)Cl)c6ccccc6)C#N HTS09982 Cc1nc(c(o1)C(F)(F)F)/C(=N/OC(=O)c2ccc(cc2)Cl)/N RF04265 c1cc2c(cc1/C=N/Nc3c4c5c(sc4ncn3)CCCC5)OCO2 HTS09947 c1cnc(nc1)N2CCN(CC2)C(=O)CCCC(=O)O HTS10166 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2nc(no2)c3c(cccc3Cl)Cl)Cl SPB00339 CCOC(=O)c1c2c(sc1N)CC(CC2)C HTS09864 Cc1cc(n(n1)c2ccccc2)NC(=O)c3ccccc3 HTS09865 Cc1cc(n(n1)c2ccccc2)NC(=O)Nc3ccc(c(c3)Cl)Cl HTS09866 CCOC(=O)/C(=C/c1cn(nc1c2ccccc2)c3ccccc3)/C#N HTS09867 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)NN)C#N HTS09920 CCOC(=O)C(C(=O)C)Sc1nnc(n1CC=C)c2cnn(c2N)c3ccccc3 HTS09924 CC1=C(C(n2c(=O)/c(=C\c3ccc(cc3)OC)/sc2=N1)c4ccc(cc4)OC)C(=O)OC HTS09896 c1ccc2c(c1)CC(C2)n3c(nnc3SCCS(=O)(=O)c4ccc(cc4)F)OC(=O)c5cccs5 HTS08667 C#CCSc1ccccc1C2=NCCCN2.Br CD05713 CC(C)(C)c1ccc(cc1)NC(=O)c2ccsc2 HTS10690 CC(C)(C)c1ccc(cc1)Oc2ccc(cc2[N+](=O)[O-])/C(=N/O)/N SPB00971 CNc1ccccc1C(=O)N/N=C/c2ccc(cc2)N(C)C DP01748 COC(=O)C1=C(n2c(=O)/c(=C/c3ccc(cc3)Cl)/sc2=C(C1c4ccc(cc4)Cl)C#N)N FV00095 Cn1c(cc(n1)C(F)(F)F)C(=O)O RF04315 Cn1c(cc(n1)C(F)(F)F)C(=O)Nc2ccc(cc2)Cl RF04321 COc1cccc(c1OC)CNC(=O)c2cnc(cc2C(F)(F)F)OC RF04457 COc1ccc(cc1)/C=N/NC(=S)Nc2cc(ccc2Cl)C(F)(F)F RJF00954 c1ccc(cc1)/C=N/N=C\2/N(C(=O)CS2)c3cc(ccc3Cl)C(F)(F)F RJF00964 COc1cccc(c1)C2c3c(c4ccccc4oc3=O)OC(=C2C#N)N HTS09872 Cn1cc(nc1)S(=O)(=O)N(Cc2ccccc2)Cc3ccccc3N4CCC(CC4)C(=O)O HTS10562 Cc1ccc(cc1Cl)NC(=O)Nc2cc(nn2C)c3ccccc3 HTS10593 Cc1ccc(n1C)CNC(=O)Nc2ccc(cc2)F HTS10870 CCCCCc1ccc(cc1)C(=O)NNC(=S)N SPB01038 C/C(=C(/C(=O)c1ccccc1F)\C(=O)OC)/NC SPB00965 c1cc(oc1)CN2CC(CC2=O)C(=O)Nc3ccc(c(c3)Cl)N4CCOCC4 HTS09690 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5ccc(s5)c6cccs6 HTS09778 Cc1c(sc(n1)c2cnccn2)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS09780 Cc1c2ccccc2sc1c3ccnn3C(=O)NC MWP00407 c1cc(sc1)C(=O)Oc2nnc(n2C3CC3)SCCS(=O)(=O)c4ccc(cc4)F HTS08668 C=CCn1c2c(c(ncn2)N3CCN(CC3)c4ccccc4)sc1=S HTS09902 c1ccc2c(c1)cccc2NS(=O)(=O)c3ccc(cc3)C(F)(F)F HTS09167 Cc1ccc(cc1)S(=O)(=O)Nc2cccc3c2cccc3 HTS09171 c1ccc2c(c1)CC(C2)NC(=O)c3ccc4c(c3)OCCCO4 HTS09174 COc1ccccc1C(=O)O/N=C(/c2cccc(c2)C(F)(F)F)\N SEW02403 c1cc(ccc1NC(=O)c2cc3c(s2)ccs3)Cl SEW02435 CCN(CC)C(=O)c1cc2c(s1)ccs2 SEW02437 c1cc(ccc1CNC(=O)c2ccc(cc2)Cl)C#N CD02727 CCOC(=O)CSc1nnc(n1N)c2cccs2 HTS09926 Cc1c(cn(n1)c2ccccc2)/C=N/n3c(n[nH]c3=S)c4cccs4 HTS09927 c1ccc(cc1)Oc2c(c(ncn2)Oc3ccccc3)Br SPB00024 Cc1ccc(n1c2c(cccn2)Oc3cnn(c(=O)c3Cl)Cc4ccccc4)C HTS10415 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)N/N=C/c3c(cccc3Cl)Cl RJF01971 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)N/N=C/c3ccc(cc3)Cl RJF01979 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)c4ccccc4Cl HTS09873 CN(Cc1c(cccc1OC)OC)C(=O)c2cnc(cc2C(F)(F)F)OCc3ccccc3 RF05416 c1cc(c(c(c1)Cl)/C=N/OC(=O)Nc2nc(no2)c3c(cccc3Cl)Cl)Cl SPB00389 Cc1c(c(c(c(c1C)C)CSC(=Nc2cc(ccc2Cl)Cl)N3CCOCC3)C)C SJC00271 c1ccc(cc1)C(=O)NC(=C(C#N)C#N)Nc2ccccc2Cl TL00031 Cc1c(cn(n1)c2ccccc2)C=C(C#N)C#N HTS09869 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)/C=C/C(=O)O HTS09399 CCC(C)(C)C1CCc2c(sc(c2C#N)NC(=O)c3ccccc3C(=O)O)C1 HTS06887 CCCc1cc(=O)oc2c1ccc(c2)OC(C)C(=O)N/N=C/c3c(cccc3Cl)F RJF01983 c1ccc(c(c1)/C=N/NC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl)Cl RJF02013 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3cc(sc3C(=O)OC)c4ccc(cc4)Cl HTS09406 C=CCn1c2c(c(ncn2)Sc3nnc(n3c4ccccc4)c5ccccc5)sc1=S HTS09988 Cc1nc2c(c(n1)Sc3[nH]cnn3)sc(=S)n2c4ccccc4 HTS09989 Cn1c2ccccc2n3c1c(c(cc3=O)c4ccccc4)C#N HTS09991 CC1CCc2c(sc(c2C#N)NC(=O)c3cccc(c3)[N+](=O)[O-])C1 HTS09930 c1ccnc(c1)c2ccc(s2)c3nc(cs3)c4ccc5c(c4)OCCCO5 HTS03334 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)CSCC(=O)O HTS09401 Cc1c(csc1C(=O)Nc2cc(sc2C(=O)OC)c3ccc(cc3)Cl)S(=O)(=O)c4ccc(cc4)Cl HTS09404 CN(C)NC(=O)Cn1nc(nn1)c2cc(cc(c2)Cl)Cl RJF02007 C=CCSc1nnc2n1CCCN2C(=O)Nc3cccc(c3)Cl HTS09885 CSc1cccc(c1)NC(=O)C(=O)NCCc2ccccn2 JPV00078 CC(C)(C)c1ccc(cc1)CSc2nnc(n2C)c3ccc(cc3)C(C)(C)C SPB00605 c1ccc2c(c1)c(c(s2)c3nnc(o3)c4ccccc4C(F)(F)F)Cl HTS08719 c1ccc2c(c1)CCCN2C(=O)CSCC(=O)O HTS10631 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)Nc3ccc(cc3)F)C HTS08792 CN(C1CCCCC1)C(=O)Nc2cccc(c2)C(F)(F)F HTS08837 CC1CC(=O)Nc2ccccc2N1C(=O)Nc3ccc(cc3)F HTS08857 c1cc(ccc1c2nnc(o2)c3cnc(cc3C(F)(F)F)Oc4ccc(cc4)Cl)Cl RF04798 Cn1c(=O)c2c(n(c1=O)C)OC(=C(C2c3ccccc3)C#N)N HTS09999 CCCc1cnc(nc1)N2CCN(CC2)C(=O)Nc3cc(oc3C(F)(F)F)C HTS09259 Cc1c(snn1)c2nnc(n2N)S HTS09260 Cc1c(snn1)c2nnc3n2N=C(CS3)c4ccc(cc4)C#N.Br HTS09262 Cn1ccnc1SCC(=O)N2c3ccccc3Sc4c2cccc4 HTS09940 Cn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])c3ccncc3 HTS09942 Cc1cc(n(n1)c2c3c4c(sc3ncn2)CCCC4)C HTS09943 Cc1nnc2n1cnc3c2c4c(s3)CCCC4 HTS09950 COc1ccc(c(c1)NC(=O)C(=O)NCc2ccco2)OC JPV00088 CC1CC(CC(C1)(C)C)NC(=O)C(=O)Nc2cc(ccc2OC)OC JPV00090 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)Nc2cccc(c2)Cl HTS11103 CN(C)c1ccc(cc1)C(=O)Nc2ccc(nc2)Oc3c(cccc3Cl)Cl HTS11131 COc1c(csc1Br)C(=O)NNC(=O)c2ccccc2Cl KM00639 COC(=O)c1ccccc1NC(=O)c2ccc3c(c2)OCCCO3 HTS09176 Cc1c(sc(n1)c2ccccc2)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F HTS09183 c1cc(ccc1C(=O)NNC(=O)c2ccc3c(c2)OCO3)C(F)(F)F HTS09184 c1ccc(cc1)CNC(=O)c2cc3c(s2)ccs3 SEW02438 CC(c1ccccc1)NC(=O)c2cc3c(s2)ccs3 SEW02439 Cc1c(snn1)C(=O)N2CCN(CC2)C(=O)C3COc4ccccc4O3 HTS08796 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)C(=O)C3COc4ccccc4O3 HTS08798 Cc1c(sc(n1)c2ccccc2)c3nnc(o3)c4cccc5c4cccc5 HTS09757 c1ccc(c(c1)C(=O)NC(=O)c2ccc(cc2)C(F)(F)F)O HTS08898 COc1cccc(c1)C(=O)NC(=O)c2ccccc2O HTS08899 c1ccc2c(c1)cccc2c3nnc(o3)c4ccc5c(c4)OCO5 HTS09758 c1ccc(cc1)Oc2c(c(ccn2)C(F)(F)F)C(=O)Nc3ccc(cc3)Cl RF05102 C/C(=N\O)/C(C)(C)Nc1cccc(c1)Cl HTS10433 CCSc1cc(c(cn1)C(=O)N(C)Cc2c(cccc2OC)OC)C(F)(F)F RF05413 Cc1c(c(c(o1)C)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)C(=O)OC HTS11045 c1ccc(cc1)n2c(c(cn2)C(=O)NN)N HTS10000 Cc1c2c(c3cc(cc(c3n1)OC)OC)CN(C2)C(=O)Nc4ccccc4 HTS10003 Cc1c2c(c3cc(ccc3n1)Cl)N(CC2)c4cccc(c4)OC HTS10004 Cc1cc(c(c(c1)C)n2c(nnc2SCc3nc4ccccc4s3)O)C HTS09609 Cc1ccc(n1C)CNS(=O)(=O)c2ccc(cc2)C(F)(F)F HTS10877 c1cc(ccc1Oc2c3c4c(sc3ncn2)CCCC4)Cl HTS09951 CC1(CC2=C(C(c3c([nH]c(=S)[nH]c3=O)N2)c4ccccc4)C(=O)C1)C HTS09953 Cc1c(c(no1)c2c(cccc2Cl)Cl)COC(=O)Nc3ccc(cc3)Cl SPB00097 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)N3CCCCC3)C HTS08419 c1cc(c(cc1Cl)Cl)/C(=N/O)/C#N SPB00235 CN(c1ccccc1)C(=O)c2cc3c(s2)ccs3 SEW02440 c1ccc(cc1)c2cc(nc3c2c(c(o3)C(=O)NN)N)c4ccc(cc4)Cl HTS09992 c1ccc2c(c1)nc3n2c(c(s3)C#N)/N=C/c4cccs4 HTS09994 c1ccc(cc1)c2cc(n3c(n2)ncn3)N/N=C/c4ccc(cc4Cl)Cl HTS09996 COC(=O)c1ccc(o1)CSCCN.Cl HTS09264 COC(=O)c1ccc(cc1)c2cn3cccnc3n2 HTS09265 c1ccc(c(c1)C(=O)NC(=O)C2CCCCC2)O HTS10037 CN(Cc1cccc(c1)Cl)C(=O)c2cnc(cc2C(F)(F)F)OC RF04334 Cc1cccc(c1C)NC(=O)c2cnc(cc2C(F)(F)F)SC RF04390 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)OC(F)F HTS10054 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS11051 CC(C)(C)NC(=O)N1CCCN(CC1)c2ccc(cn2)C(F)(F)F HTS11052 c1ccc2c(c1)CC(C2)N3CC(CC3=O)C(=O)O HTS10895 Cc1cc(nn1C)C(=O)NNC(=S)Nc2cccc(c2)C(F)(F)F SPB00747 c1cc(c(cc1C(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-])Cl)Cl SPB01372 C=CCNC(=S)Nc1c(c2c(s1)CCCC2)C#N HTS10006 COc1ccc(cc1)/C=C/C(=O)Nc2ccccc2C(Cc3ccccc3)(c4ccccc4)O CD01953 c1ccc(cc1)CC(c2ccccc2)(c3ccccc3NC(=S)Nc4cc(ccc4Cl)Cl)O CD01955 CCOC(=O)c1c(n[nH]c1Nc2ccc(cc2C)Br)C SJC00427 c1cc(cc(c1)C(F)(F)F)CS(=O)CC(=O)NN CD03707 c1cc(ccc1CN2CCS(=O)(=O)CC2)NS(=O)(=O)c3ccc(cc3)Cl HTS09663 C1CC1CNC(=S)NNC(=O)C2CC2 RJF01759 Cc1ccc(cc1)/C=N/Nc2ccc(cc2)[N+](=O)[O-] SPB00276 Cc1c(c(c(c(c1C)C)CS/C(=N/c2cc(c(cc2OC)Cl)OC)/N3CCOCC3)C)C JP00553 CCc1cc(c(s1)NC(=O)CC(C)(C)CC(=O)O)C(=O)c2ccc(cc2)OC HTS09247 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(cc3)N HTS09660 Cc1ccc(n1C)CNC(=O)Nc2cccc(c2C)Cl HTS10882 c1ccc2c(c1)nc(s2)c3ccsc3NC(=O)Nc4ccc(cc4)F HTS10885 c1ccc(cc1)NC(=O)Nc2c(ccs2)c3nc4ccccc4s3 HTS10886 c1ccc(c(c1)C#N)NC(=O)c2ccco2 HTS08136 CSc1cc(c(cn1)C(=O)Nc2ccc(cc2)Cl)C(F)(F)F RF04412 CCN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)SCC RF04436 c1ccc(cc1)C(C[N+](=O)[O-])c2c[nH]c3c2cccc3 SEW04392 Cc1c(sc2n1nc(n2)C(F)(F)F)c3ccnc(n3)S SPB05647 CNC(=S)NNC(=O)c1ccc(cn1)C(F)(F)F SPB06119 c1cc(ccc1CSc2[nH]nc(n2)NC(=O)COCC(=O)O)Cl HTS10711 c1ccc(cc1)c2cc(nc\3c2CCC/C3=C(\c4cccs4)/Oc5ccc(cc5)Cl)c6ccccc6 TL00051 c1c(cc(nc1OCC(F)(F)F)OCC(F)(F)F)C(=O)NN RF04935 Cc1c(n2ccccc2n1)C(=O)N/N=C/c3cn(nc3c4ccc(cc4)[N+](=O)[O-])c5ccccc5 HTS09937 CN1CCN(CC1)CC(=O)N2c3ccccc3Sc4c2cccc4 HTS09938 c1cc(oc1)C(=O)N(c2ccc(c(c2)Cl)F)C3=NCCC(=O)S3 RJF01786 c1ccc(cc1)c2nc(no2)CO RF02995 COc1cc(cc(c1O)Br)C2Nc3ccccc3C(=O)N2 HTS02957 CCCc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)OC(=O)N(CC)CC)C RJF01931 CCOC(=O)CS/C(=N/NC(=O)c1c(nc2n1ccc(c2)C)C)/NCc3ccccc3 HTS10007 CCOC(=O)CS/C(=N/NC(=O)c1c(nc2n1ccc(c2)C)C)/NCC=C HTS10008 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(cc2)OC HTS09629 CC(C)(C)c1ccc(cc1)NC(=S)NNC(=O)c2ccccc2Cl SPB00778 CCOC(=O)C1=C(OC(=C(C1c2ccc(cc2)N3CCOCC3)C#N)N)C MO00269 c1cc(ccc1C(=O)CNC(=O)CCC(=O)O)F HTS10074 Cc1cc(n(n1)C)C(=O)Nc2ccc(nc2)Oc3c(cccc3Cl)Cl HTS09449 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2ccccc2C(C)C SJC00437 CS(=O)(=O)N(Cc1ccccc1)Cc2ccccc2N3CCC(CC3)C(=O)O HTS10561 CC1CCc2c(sc3c2c(ncn3)SCC(=O)N/N=C/c4ccco4)C1 HTS09949 c1cc(c(cc1F)F)NC(=O)NC(=O)c2ccc(o2)[N+](=O)[O-] SPB00924 c1cc(ccc1CC(=O)c2ccc(cc2)Cl)C(=O)N MO00235 c1cnc(nc1)N2CCN(CC2)C(=O)CCC(=O)O HTS10167 c1cnc(nc1)N2CCN(CC2)C(=O)CSCC(=O)O HTS10170 COc1ccc(cc1)Oc2ccc(cc2C(=O)Nc3ccc4c(c3)OCCO4)[N+](=O)[O-] HTS10411 Cc1c(c(n(n1)c2ccccc2)C)c3nnc(o3)C(F)(F)F SEW04238 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)N/N=C/c3ccccc3Cl RJF01968 CCCc1cc(=O)oc2c1ccc(c2)OC(C)C(=O)N/N=C/c3c(cccc3Cl)Cl RJF01982 c1cc(ccc1Nc2ncnc(n2)N)F RJF00582 c1ccc(cc1)CC(c2ccccc2)(c3ccccc3N)O CD01948 CC(C(=O)NNC(=S)NCC1CC1)n2nc(nn2)N3CCOCC3 RJF01835 c1ccnc(c1)CNC(=O)C2CCC(CC2)c3ccc(cc3)Cl HTS10095 c1cc(ccc1c2csnn2)NC(=S)Nc3ccc(cc3)Cl SEW00802 Cn1c(nnc1SCC(=O)c2ccccc2)C(F)(F)F SPB04139 Cc1ccc(c(c1)C)N/C(=N/O)/c2cnccc2C(F)(F)F RF05224 c1ccc(cc1)Sc2c(cc(cn2)[N+](=O)[O-])C(F)(F)F RF05309 Cc1cccc2n1cc(n2)c3ccc(cc3)[N+](=O)[O-] SJC00435 c1cc(ccc1C(=O)NNC(=O)c2ccc3c(c2)nsn3)C(F)(F)F HTS09185 c1ccc(cc1)Oc2c3c4c(sc3ncn2)CCCC4 HTS09952 c1ccc(cc1)C2=Nc3ccccc3N=C(C2)c4ccccc4 HTS10693 c1ccc(cc1)C2=Nc3cc(cc(c3N=C(C2)c4ccccc4)Cl)C(F)(F)F HTS10696 C=CCSc1[nH]c(nn1)c2cccnc2 SPB00561 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCc3ccc(cc3)Cl SPB00598 CCc1cc(c(s1)NC(=O)c2ccc(cc2)C(F)(F)F)C(=O)c3ccc(cc3)OC HTS08697 c1cc(ccc1c2nc(on2)CSc3ccc(cc3)Cl)Cl CD02834 Cc1c(c(no1)c2ccccc2)c3nnc(o3)c4ccccc4C(F)(F)F HTS08716 Cc1cc(cc(c1)NC(=O)N2c3ccccc3NC(=O)CC2C)C HTS08854 Cc1cc(cc(c1)NC(=O)N2CCNC(=O)C2CC(=O)Nc3cccc(c3)C(=O)OC)C HTS08858 c1ccc2c(c1)[nH]c(n2)SC(C#N)C#N HTS09034 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2cccs2 HTS10555 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccccc3Cl RJF01044 c1cc(ccc1Oc2c(c(ccn2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F)Cl RF05098 c1cc(cc(c1)Oc2c(c(ccn2)C(F)(F)F)C(=O)Nc3ccc(cc3F)F)C(F)(F)F RF05101 CCCCCCCCCCCC(=O)Nc1c(cccc1C)C RG00116 Cc1ccc(n1C)CNC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS10869 Cc1cc(nn1c2ccc(cc2)[N+](=O)[O-])C(=O)NN SPB00803 Cn1c(nnc1SCC(=O)NNC(=S)Nc2ccccc2)c3ccncc3 HTS09941 Cc1cc(nn1C)C(=O)NNC(=S)N SPB00817 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccc(cc3)OC(F)(F)F HTS09634 CCc1cc(c(s1)NC(=O)c2c(nccn2)C(=O)O)C(=O)c3ccc(cc3)OC HTS09246 Cc1ccc(cc1)C(=O)CN2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS09764 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)C(F)(F)F HTS08865 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccccc3)CC(CC2)C HTS09862 CCOC(=O)c1c2c(sc1NC(=S)NC)CCCC2 HTS09863 Cc1c2c(c(c(nc2n(n1)c3ccccc3)OCC(=O)c4ccccc4)C#N)c5ccc(cc5)[N+](=O)[O-] HTS09870 c1ccc(c(c1)/N=C\c2cc(cc(c2O)Cl)Cl)SCc3nc(no3)c4ccc(cc4)Cl CD03146 Cc1c(c(no1)c2ccccc2)C(=O)N/N=C/c3ccc4ccccc4c3 CD03165 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)CC(=O)c5ccc(cc5)F HTS09763 CCc1cc(c(s1)NC(=O)Nc2ccc(cc2)F)C(=O)c3ccc(cc3)OC HTS09250 CC(C)N(Cc1ccccc1)C(=O)Nc2cccc(c2)C(F)(F)F HTS08839 CC1CC(=O)Nc2ccccc2N1C(=O)Nc3ccccc3OC(F)(F)F HTS08856 Cc1c(c(no1)c2ccccc2)C(=O)N/N=C/c3ccc(c(c3)OC)O CD03125 COc1ccc(cc1OC)CNC(=O)c2cnc(cc2C(F)(F)F)OC RF04468 CCCNC(=O)NC(=O)c1cnccc1C(F)(F)F RF04470 Cc1[nH]c(=O)c2c(n1)Oc3c4ccccc4oc(=O)c3C2c5ccc(cc5)Cl HTS09965 c1cc(sc1)/C=N/Nc2c3c(nc4n2ncn4)CCC3 HTS09969 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)NNC(=O)Nc4cccc(c4)C(F)(F)F)C#N HTS09972 CCc1cc(c(s1)NC(=O)COCC(=O)O)C(=O)c2ccc(cc2)OC HTS09241 CCc1cc(c(s1)NC(=O)CCC(=O)O)C(=O)c2ccc(cc2)OC HTS09245 COc1ccc(cc1)C(=O)CSc2nnc(n2Cc3ccco3)O HTS09451 CCn1c(nnc1SCc2ccc(cc2)Cl)CN3c4ccccc4Sc5c3cccc5 HTS10336 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)c3ccc(cc3F)F HTS08867 CN(C)c1ccc(cc1)C2Nc3ccccc3C(=O)N2CCN4CCNC4=O HTS08875 CCC1c2c(c3ccccc3oc2=O)Oc4c1c(=O)[nH]c(n4)C HTS09880 CCOC(=O)Cn1cnc2c(c1=O)cnn2c3ccccc3 HTS09883 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03263 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03306 c1ccnc(c1)/C=C(\C#N)/c2cccc(c2)C(F)(F)F CD03359 c1cc(oc1)Cn2c(nnc2SCc3nc(no3)COc4ccc(cc4)[N+](=O)[O-])O HTS09453 c1ccc(c(c1)NC(=O)CSc2nnc(n2Cc3ccco3)O)Cl HTS09455 CC1CC(=O)Nc2ccccc2N1C(=O)Nc3ccccc3OC HTS08878 CC1CC(=O)Nc2ccccc2N1C(=O)Nc3ccc(cc3F)F HTS08879 CCN(c1ccc(cc1Cl)Cl)C(=O)c2cnc(cc2C(F)(F)F)NC(C)C RF04475 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/NC(=S)N HTS09986 c1cc2cc(ccc2nc1)C(=O)NN KM10250 c1ccc2c(c1)CCCN2C(=O)c3ccccc3C(=O)O HTS10628 Cc1c(c(no1)c2ccccc2)CSc3nnc(n3Cc4ccco4)O HTS09462 c1cc(c(cc1Br)OC(F)(F)F)NCN2C(=O)CCC2=O TL00644 CC(=O)Nc1ccc(cc1)NS(=O)(=O)c2ccc(s2)S(=O)(=O)c3ccccc3 HTS08945 CC(=O)Nc1ccc(cc1)NC(=O)c2ccccc2 HTS08949 CC(=O)Nc1ccc(cc1)NC(=O)c2ccco2 HTS08950 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3ccc(cc3)NC(=O)C HTS08954 c1ccc(c(c1)C(=O)NC(=C(C#N)C#N)Nc2ccc(cc2)Cl)Cl TL00098 CC(C)(C)C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F TL00156 CC1=C(C(NC(=S)N1)c2cccc(c2)OC)C(=O)OC HTS09892 Cc1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)c4ccc(cc4)Cl)N)c5cn(nc5c6ccccc6)c7ccccc7 HTS09899 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2SCCS(=O)(=O)c3ccc(cc3)Cl HTS06076 CN1CCN(CC1)C(=O)c2ccc(s2)c3cccs3 HTS08524 c1cc(ccc1C(=O)CSc2nnc(n2C3CC3)O)F HTS09141 c1ccc(cc1)c2cc(on2)C(=O)CSc3nnc(n3C4CC4)O HTS09142 COc1cccc(c1C(=O)NC(=O)Nc2ccc(cc2)Oc3cc(c(cn3)C(=O)OC)C(F)(F)F)OC RF04749 c1ccc(cc1)Oc2cc(c(cn2)c3nnc(o3)c4ccccc4Cl)C(F)(F)F RF04792 CC(C)(C)CC(=O)O/N=C(/C1(CC1)c2ccc(cc2Cl)Cl)\N SEW03878 c1cc(c(cc1C(=O)O)F)C(=O)O RDR03446 Cc1ccc(n1C)CNC(=O)Nc2ccccc2OC HTS10878 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3c(ccs3)c4nc5ccccc5s4 HTS11222 CCCSc1c(cccn1)C(=O)Nc2c(noc2C)C HTS11159 Cn1c2c(c(=O)n(cn2)/N=C/c3ccc(c(c3)OC)O)sc1=S HTS09901 Cc1cc(nc2c1c3c(o2)c(=O)n(cn3)Cc4ccc(cc4)Cl)c5ccccc5 HTS09916 c1ccc2c(c1)nc(s2)CN3CCc4c(ccs4)C3c5ccc(cc5)OC(F)(F)F HTS08550 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)C(=O)C4COc5ccccc5O4 HTS08797 c1cc(c(cc1NC(=O)C2=NNC(=O)CC2)Cl)N3CCOCC3 HTS09711 c1ccc2c(c1)C(=O)N(S2(=O)=O)Cc3ccc4c(c3)nsn4 HTS10026 c1cc(c(cc1Cl)Cl)C(c2c([nH]c(=S)[nH]c2=O)N)c3c([nH]c(=S)[nH]c3=O)N HTS10493 CCOC(=O)c1c2c(sc1NC(=S)NCC=C)CC(CC2)C HTS10495 CCOC(=O)C(C(=O)C)Sc1nnc(n1CC=C)c2ccncc2 HTS10496 c1ccc2c(c1)OCC(O2)C(=O)N3CCN(CC3)C(=O)Nc4ccc(cc4)F HTS08800 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)C(=O)C4COc5ccccc5O4 HTS08801 CC(C)c1ccc(cc1)NC(=O)C2=NNC(=O)CC2 HTS09710 c1ccc2c(c1)C(=O)N(S2(=O)=O)Cc3ccc4c(c3)non4 HTS10027 Cc1cc(n(n1)c2ccc(cc2)N)C SEW04169 COC(=O)CC1(N(C(=O)c2cc(ccc2O1)Br)c3cccc(c3Cl)Cl)C(=O)OC SJC00384 Cc1ccc(cc1)c2nc(c(c(n2)S)C(=O)C)C SPB05391 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)COc3ccc(cc3Cl)Cl HTS08968 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4cccc5c4non5 HTS09506 CS(=O)(=O)c1ccc(cc1)C2=Nn3c(nnc3SC2)c4cccs4 HTS09255 Cc1ccc(n1C)CNS(=O)(=O)c2cccs2 HTS10875 c1ccc(c(c1)C(=O)NC(=O)c2ccccc2Cl)O HTS10036 c1cc(oc1)CN2CC(CC2=O)C(=O)Nc3ccc(nc3)N4CCOCC4 HTS11016 c1cc(c(c(c1)F)C#N)N/N=C(/C(=O)c2cccs2)\C(=O)C(F)(F)F CD05787 Cc1ccc(cc1NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)F HTS11053 Cc1ccc(n1C)CNC(=O)Nc2cc(ccc2OC)Cl HTS10880 Cc1c(c(no1)c2ccccc2Cl)C(=O)N(CCC#N)CCC#N CD02234 COc1cc(cc(c1OC)OC)C(=O)NC(=S)Nc2nc(cs2)c3ccc(cc3)F CD02476 CCOC(=O)c1c(n[nH]c1Nc2cccc(c2Cl)Cl)C SJC00425 COC(=O)NNc1c(cccn1)C(F)(F)F RF04964 CC(=O)NNc1cccc(n1)C(F)(F)F RF05180 CC(C)(CC(=O)Nc1ccc(cc1)OC)Sc2ccc(cc2)Cl HTS09665 CCN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)Oc3ccccc3 RF04440 CN(C)/C(=N\O)/c1c(cccc1Cl)Cl SPB00102 c1ccc2c(c1)-c3cccn3C(N2)c4ccc5c(c4)CCO5 HTS11088 c1ccc2c(c1)-c3cccn3C(N2)c4ccc5c(c4)OCCO5 HTS11089 c1cc(cc(c1)[N+](=O)[O-])/C=N/Nc2ccc(cc2)[N+](=O)[O-] SPB00279 c1c(cc(cc1Cl)Cl)OCc2nc(cs2)CSc3[nH]c(nn3)C(F)(F)F SPB01818 c1cc(cc(c1)Cl)NC(=C(C#N)C#N)N TL00091 CCN(C(Cc1ccccc1)c2ccc(cc2)OC)C(=O)c3c(onc3c4c(cccc4Cl)Cl)C CD01987 Cc1c(c(c(c(c1C)C)C(=O)/C(=N/OCc2cccc(c2)C#N)/c3ccccc3)C)C CD02480 Cc1cc(c(c(c1)C)/N=C\2/NC3(CCCCC3)C(=C)S2)C BTB15254 c1cc2c(cc1CCC(=O)O)CCO2 HTS10422 c1cc(sc1)C(=O)O/N=C(/C2(CC2)c3ccc(cc3Cl)Cl)\N SEW03876 Cn1c(cc(n1)c2ccc(cc2)Cl)NC(=O)Nc3ccc(cc3)OCc4ccccc4 HTS08055 Cc1cccc(c1NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(C)C CD06453 c1cc(ccc1S(=O)(=O)NNC(=S)Nc2ccc(c(c2)Cl)Cl)Cl SPB00990 Cc1nc(nc(n1)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)N RF02945 CCOC(=O)C1=C(N2CCCN=C2S1)C.Cl HTS10973 CCOC(=O)c1c(n(cn1)Cc2ccccc2)N HTS10974 c1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3ccco3 HTS10310 CCOc1ccc(cc1)/C=N/NC(=O)c2ccccc2n3cccc3 CD02576 COC(=O)c1c(cc(s1)[N+](=O)[O-])N GK01860 c1cc(cc(c1)F)NC2=NCCCC(=O)S2 RJF01764 Cc1c(cnn1c2ccccc2)C(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS09779 COC(=O)CNC(=O)C1CCC(CC1)c2ccc(cc2)Cl HTS10092 Cc1cc(no1)C(=O)NNC(=O)c2ccc(cc2)Cl SPB02784 c1cc2c(cc1c3nnc(o3)N)nsn2 HTS10723 C1CNc2nnc(n2C1)S HTS09887 CC1=C(C(NC(=S)N1)c2cccs2)C(=O)OC HTS09890 Cc1cc(nc(n1)NC(=O)C(=O)NC(=O)c2c(cccc2Cl)F)C RF03635 Cc1c(nnn1c2cc(ccc2Cl)C(F)(F)F)/C(=N/O)/C BTB15255 c1ccc(c(c1)C#N)NS(=O)(=O)c2ccc(cc2)Cl HTS08152 c1ccc2c(c1)c(cs2)C(=O)CSc3nnc(n3Cc4ccco4)O HTS09472 CCn1c(cc(n1)C)/C(=N/O)/N SPB01881 Cc1c(c(nc(n1)SCC(=O)c2ccc(cc2)OC)O)Oc3ccc(cc3)Cl SPB04142 c1ccn(c1)Cc2c(ccs2)COc3ccc(cc3)Cl SEW02523 c1cc(ccc1CNCC(CO/N=C/C2=C(c3cc(ccc3OC2)Cl)Cl)O)C(F)(F)F SEW03010 c1cc2c(cc1Cl)C(=C(CO2)/C=N/OCC(CN3CCOCC3)O)Cl.Cl SEW03014 CC(=O)Nc1c(cc(cc1F)F)[N+](=O)[O-] SPB00771 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccco3)Sc4ccc(cn4)[N+](=O)[O-] SPB00789 c1cc(ccc1S(=O)(=O)CC/C(=N/O)/N)Cl SEW00732 Cc1ccnc(n1)NC(=O)Nc2ccccc2 HTS09740 c1cc(oc1C(=O)NCc2ccncc2)Oc3cc(cc(c3)Cl)Cl HTS08739 Cc1ccc(cc1)C2=CC(N3C(=O)CSC3=N2)c4cn(nc4c5ccccc5)c6ccccc6 HTS09893 c1ccc(c(c1)NC(=O)CSc2nnc(n2c3cccnc3)O)Cl HTS09138 c1cc(ccc1N)n2ccnc2 RF03777 c1ccc(cc1)COc2ccc(cn2)[N+](=O)[O-] RF05222 Cc1cc(nc(c1C#N)SCc2ccc(cc2)F)C HTS10313 Cc1ccc(cc1Cl)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS08427 c1cc(ccc1NC(=S)NC(=O)c2cc(sc2)[N+](=O)[O-])Cl DFP00132 COc1ccccc1NC(=O)N2CCN(CC2)c3ncccn3 HTS10744 c1cnc(nc1)N2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F HTS10746 Cc1c(c(no1)c2ccccc2)NC(=O)ON(Cc3cccc(c3)C(F)(F)F)Cc4cccc(c4)C(F)(F)F CD05726 CC(c1ccccc1)n2c(nnc2SCC(=O)c3ccc(cc3)OC)O HTS09479 Cc1ccc(cc1Cl)NC(=O)O/N=C/c2c(nn(c2C)C(C)(C)C)C CD07459 c1ccc(c(c1)C2=NCCCN2S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)SCc4c(cccc4Cl)F CD07476 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS08429 c1ccc(cc1)CN2c3ccccc3/C(=N/c4ccccc4)/C2=O HTS10315 c1ccc2c(c1)/C(=N/c3ccc(cc3)Cl)/C(=O)N2 HTS10316 Cc1ccc(cc1)/N=C\2/c3ccccc3NC2=O HTS10317 COC(=O)c1ccc2c(c1)nc[nH]2 MO00298 c1ccc2c(c1)c(c(s2)C(=O)N3CCN(CC3)C(=O)c4ccco4)Cl HTS09512 c1cc(oc1)C(=O)n2ccc(n2)c3cccs3 HTS09514 c1cc(cnc1)CNC(=O)C2CCC(CC2)c3ccc(cc3)Cl HTS10093 c1ccc(c(c1)C(=O)N2CCN(CC2)c3ncccn3)C(=O)O HTS10168 CC1CCc2c(sc3c2c(ncn3)N4CCN(CC4)c5ccccc5)C1 HTS09859 C=CCn1c2c(c(ncn2)Sc3nnc(n3CC=C)c4ccccc4)sc1=S HTS09905 C=CCNC(=S)NC(=O)c1cc(sc1)[N+](=O)[O-] DFP00146 c1ccc(cc1)CSc2nc3cc(ccc3s2)Cl EN00191 Cc1c2cc(ccc2sc1S(=O)(=O)Nc3ccc(cc3)N4CCCCC4)Cl HTS08428 CCNc1c2c3c(sc2nc(n1)SCC(=O)c4ccccc4)CC(CC3)C HTS10318 CCNc1c2c3c(sc2nc(n1)SCC(=O)C)CC(CC3)C HTS10319 c1cnc(nc1)N2CCN(CC2)C(=O)c3c(nccn3)C(=O)O HTS10169 Cc1ccc(cc1Cl)S(=O)(=O)Nc2cc(nn2C)c3ccccc3 HTS10216 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)Nc3ccc4c(c3)OCCO4 HTS10412 c1cc2c(cc1Br)/C(=N/N=C/c3ccncc3)/C(=O)N2 HR00132 Cc1c2c(n3c4ccccc4nc3c1C#N)N(CC2)c5cccc(c5)OC HTS09906 CN1CCN(CC1)c2c3c(c(c4n2c5ccccc5n4)C#N)CCC3 HTS09907 c1cc(ccc1C(=O)COc2nnc(n2C3CC3)SCCS(=O)(=O)c4ccc(cc4)F)F HTS09126 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3cn(nc3c4ccccc4)c5ccccc5)N)C HTS10282 c1ccc2c(c1)c(cc3c2oc(=O)s3)OC(=O)c4ccccc4I JP00893 c1ccc(c(c1)C(=O)Oc2ccc(cc2)C3CCCCC3)I JP00928 COc1ccc(cc1)NC(=S)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl RJF02024 c1ccc2c(c1)cccc2C(=O)NNC(=O)c3ccc4c(c3)nccn4 HTS08788 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNC(=O)c3cccc4c3cccc4 HTS08789 c1ccc(c(c1)c2nnc(o2)c3c(ccs3)Cl)C(F)(F)F HTS08718 Cc1c(c(c(o1)C)S(=O)(=O)N(Cc2ccccc2)C(C)C)C(=O)OC HTS08821 CC1CCc2c(sc3c2c(nc(n3)SC(C)C)NCc4ccccc4)C1 HTS10323 CC1CCc2c(sc(c2C#N)NC(=O)CN3CCOCC3)C1 HTS10330 c1cc(ccc1C(=O)O/N=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)Cl KM01225 c1ccc(cc1)NC(=O)Nc2ccc(cn2)C(F)(F)F HTS08602 c1cc2c(cc1Cl)sc(n2)NC(=O)C3CCCCC3 HTS10700 c1cc(ncc1C(F)(F)F)NC(=O)Nc2cc(cc(c2)Cl)Cl HTS08605 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(cn2)C(F)(F)F HTS08606 CN(C)c1ccc(cc1)C(=O)NNC(=O)C2CCC2 CD01943 CC1(C2CCC(C2)C1(C)NC(=S)N/N=C/c3cc(cc(c3O)Cl)Cl)C CD01961 Cc1c(c(c(c(c1C)C)C(=O)/C=N/N)C)C CD02395 Cc1cc(c(o1)C)C(=O)Nc2ccc3c(c2)OCCO3 HTS10414 Cc1c2cc(ccc2sc1C(=O)CSc3nnc(n3Cc4ccco4)O)Cl HTS09148 Cc1cc(nc2c1c(c(s2)C(=O)NNC(=S)NCc3ccccc3)N)C HTS10284 Cc1c2cc(c(nc2n(n1)c3ccccc3)N)C(=O)N HTS09915 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)CC(=O)c4ccccc4)C HTS10289 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)Cc4ccc(cc4)[N+](=O)[O-])C HTS10290 Cc1cccc(c1C(=O)O)NC(=O)c2ccno2 HTS05564 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)Nc3cccs3 HTS09380 Cc1ccc(cc1)C(=O)Nc2nc3ccc(cc3s2)Cl HTS10704 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Nc3nc([nH]n3)SCc4ccc(cc4)Cl HTS10722 Cc1cc2c(cccc2NC(=O)CCCC(=O)O)nn1 HTS09556 CC(C)(CC(=O)Nc1ccc(cc1)OC(F)F)CC(=O)O HTS09559 CN(C)c1ccc(cc1)C2Nc3ccccc3C(=O)N2CCCN4CCOCC4 HTS08874 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)NC(=O)C HTS08956 CC1CC(=O)Nc2ccccc2N1C(=O)c3ccccc3 HTS08851 CC1CC(=O)Nc2ccccc2N1C(=O)Nc3cccc(c3Cl)Cl HTS08855 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3cn(cn3)C HTS08862 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)c2c(c3ccccc3s2)Cl HTS10671 CCN(C(Cc1ccccc1)c2ccc(cc2)OC)C(=O)c3c(c4ccccc4s3)Cl CD02001 CCN(c1cccc2c1cccc2)S(=O)(=O)c3ccccc3 HTS10559 c1cnc(nc1)N2CCN(CC2)C(=O)COCC(=O)O HTS10741 Cc1cc(cc(c1)NC(=O)N2CCN(CC2)c3ncccn3)C HTS10745 c1ccc(c(c1)C(=O)O/N=C(/c2ccc(cc2)[N+](=O)[O-])\N)F BTB04196 Cc1c(c(on1)C)c2nc(no2)CSc3nnc(n3Cc4ccco4)O HTS09150 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2nc(cs2)c3ccc(cc3)c4ccccc4 CD03846 COc1cccc(c1C(=O)O/N=C(/c2ccc(cc2)Cl)\N)OC CD04004 Cc1c(snn1)C(=O)Nc2ccc(cc2)Oc3ccccc3 HTS09164 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)Cc4ccccc4Cl)C HTS10291 Cc1cc(nc2c1c(c(s2)C(=O)NN)N)C HTS10298 Cc1cc(nc2c1c(c(s2)C(=O)c3ccc(cc3)c4ccccc4)N)C HTS10297 Cn1c(cc(n1)c2ccccc2)NC(=O)Nc3ccccc3F HTS10591 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2c(noc2C)C HTS10602 c1cc(ccc1NC(=O)CCCC(=O)O)OC(F)F HTS09561 c1cc(ccc1CCNC(=O)c2ccc(cc2)F)Cl BTB04893 c1cc(ccc1CCNS(=O)(=O)c2ccc(cc2)Cl)Cl BTB04895 c1ccc2c(c1)cc(s2)C(=O)NCCc3ccc(cc3)Cl BTB04898 c1ccc(cc1)c2c(sc(n2)Nc3ccc(cc3)F)C(=O)c4ccccc4 HTS09624 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(cc2)F HTS09628 COc1ccc(cc1)C(=O)CN2C(=O)c3ccccc3S2(=O)=O HTS10033 c1ccc(cc1)C(=O)Nc2nc3ccc(cc3s2)Cl HTS08906 c1cc(sc1)C(=O)Nc2nc3ccc(cc3s2)Cl HTS08908 COc1cc(c(cn1)C(=O)NCc2ccccc2Cl)C(F)(F)F RF04326 c1ccc2c(c1)C(=O)N(S2(=O)=O)Cc3ccc(cc3)c4csnn4 HTS10035 c1cc(c(c(c1)F)c2noc(=O)n2c3ccc(cc3)C(F)(F)F)F RF05133 c1ccc(c(c1)N/C(=N/O)/c2cccnc2)F RF05151 c1cc(ncc1C(F)(F)F)N2CCCN(CC2)C(=O)CSCC(=O)O HTS10859 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F HTS11043 CN(Cc1c(cccc1OC)OC)C(=O)c2cnc(cc2C(F)(F)F)Oc3ccccc3 RF05415 CCN(c1cccc2c1cccc2)S(=O)(=O)c3ccc4c(c3)OCC4 HTS10558 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccc(c(c2)OC)OC HTS10603 Cc1c(c(no1)c2c(cccc2Cl)Cl)CSC(=S)SC(C)(C)C CD07738 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)c3ccco3 HTS09511 CCOC(=O)C1CCN(CC1)c2ccccc2CN(Cc3ccccc3)S(=O)(=O)c4ccc(cc4)Cl HTS09671 Cc1c(cc(o1)c2ccccc2)C(=O)NCc3ccncc3 HTS09674 CCOC(=O)COc1c(c(cc(n1)c2ccc(cc2)C)c3ccco3)C#N HTS10299 CCOC(=O)COc1c(c(cc(n1)c2cccs2)c3ccco3)C#N HTS10304 Cc1ccc(cc1NC(=O)N2CCCN(CC2)C(=O)OC(C)(C)C)F HTS11283 Cc1ccc(n1C)CNS(=O)(=O)c2c(noc2C)C HTS10873 Cc1ccc(n1C)CNC(=O)Nc2cccc(c2)Cl HTS10881 c1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3cccs3 HTS10306 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccc(s2)Cl HTS10607 Cc1c(cnn1c2ccccc2)S(=O)(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS10652 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN(C)C(=S)SCc3c(cccc3Cl)F CD07773 c1cc(oc1)CN2CC(CC2=O)C(=O)NCc3ccc(cc3)F HTS09661 Cc1c(c(on1)C)C(=O)n2ccc(n2)c3cccs3 HTS09517 c1ccc(cc1)C(=O)Cc2ccc(cc2)Oc3ccccc3 MO00241 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc3c(c2)OCO3 HTS10112 Cc1cccc(c1NC(=O)c2cnc(cc2C(F)(F)F)SC)C RF04391 CSc1cc(c(cn1)C(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F RF04392 Cc1cccc(c1NC(=O)c2cnc(cc2C(F)(F)F)Sc3ccccc3)C RF04396 CSc1c(c(sn1)SC)CO SEW00194 Cc1cc(c(cc1Cl)C)SCc2csc(n2)COc3ccc(cc3)OC SPB01816 CC(C)S(=O)(=O)c1csc(c1N)C(=O)Nc2ccc(cc2)F HTS11056 CC(C)(C)c1ccc(cc1)c2nnc(s2)NC(=O)C(Cl)(Cl)Cl SPB00178 c1ccc2c(c1)ccc(n2)C3Nc4ccccc4-c5n3ccc5 HTS11090 Cc1c(c(n(n1)C)NC(=O)NNc2cc(cc(c2)Cl)Cl)[N+](=O)[O-] SPB01682 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3c4c([nH]n3)CCCC4 CD07756 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CCC(=O)c4ccccc4 HTS09215 c1ccc(cc1)Oc2cccc(c2)CC(=O)c3cccc(c3)C#N MO00233 c1cc(cc(c1)C(=O)N)CC(=O)c2ccc(cc2)Cl MO00236 c1csc(c1Br)C(=O)NNc2c(cncc2Cl)Cl HTS03087 Cc1ccc(cc1Cl)NC(=O)N2CCCN(CC2)C(=O)OC(C)(C)C HTS11287 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)C(=O)OC(C)(C)C HTS11288 Cc1cc(c2nncn2n1)OCc3nnc(o3)c4ccc5ccccc5c4 HTS08814 CCCSc1c(cccn1)C(=O)Nc2cccc3c2non3 HTS11341 c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3ccco3 HTS09230 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)c3cccs3 HTS09231 c1cc(sc1)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS08424 c1ccc(c(c1)F)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS08425 COC(=O)CSc1cc(c(cn1)C(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F RF04443 CCN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)NC(C)C RF04446 COC(=O)c1ccc(o1)CSc2nnc(n2Cc3ccco3)c4ccc(cc4)C(F)(F)F HTS11110 COC(=O)CC1(N(C(=O)c2cc(ccc2O1)Br)c3cc(c(cc3Cl)Cl)Cl)C(=O)OC SJC00382 c1cc(ccc1C(=O)O/N=C(/CCSc2ccc(cc2)Cl)\N)Cl SEW00742 Cc1cccc(c1NNC(=O)Nc2c(c(nn2C)C)[N+](=O)[O-])Cl SPB01684 c1ccn(c1)c2nc3cccnc3s2 TG00155 c1ccc(cc1)C2=CC(=C3CCCC(=C3N2c4ccc(cc4)Cl)C(=O)Nc5ccc(cc5)Cl)c6ccccc6 TL00044 Cc1cc(no1)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F SPB02785 c1cc(oc1)C(=O)N2CCN(CC2)C(=O)c3ccc(cc3)C(F)(F)F HTS09232 Cc1c(c(on1)C)C(=O)N2CCN(CC2)C(=O)c3ccco3 HTS09234 CCc1ccccc1CSc2nnc(n2Cc3ccco3)O HTS09452 Cc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3ccco3 HTS10309 CC1N=C(N2N1C(=NC2C)SCC#N)SCC#N CD03247 Cc1c(sc(n1)c2ccsc2)C(=O)C SEW04002 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2cn(cn2)C HTS11116 Cc1cc(n2c(n1)nc(n2)SCC#N)C SPB00987 c1cc(c(cc1[N+](=O)[O-])Cl)NC(=O)c2cnccc2C(F)(F)F SPB05537 Cc1cc(nc(c1C#N)SCc2ccc(cc2)[N+](=O)[O-])C HTS10311 c1ccc(cc1)c2nc(cs2)CSc3nnc(n3Cc4ccco4)O HTS09457 c1ccc2c(c1)nc(s2)CSc3nnc(n3Cc4ccco4)O HTS09458 Cc1cc(nc(c1C#N)SCc2ccccc2Cl)C HTS10312 c1c(c(c(cn1)Cl)C(=O)N)Cl BTB15253 c1cc(cc(c1)C#N)CSC(=N)N.Br CD02200 c1ccn(c1)c2c(c(cc(c2Br)C(F)(F)F)C(F)(F)F)Br CD03331 c1cc(ccc1C2CCC(CC2)C(=O)NCc3ccncc3)Cl HTS10094 c1nc(c2c3c(sc2n1)CCCC3)N4CCOCC4 HTS09858 c1cc(cnc1)/C=N/NC(=O)CSc2c3c4c(sc3ncn2)CCCC4 HTS09857 COC(=O)CC1(N(C(=O)c2cc(ccc2O1)Br)c3ccc(cc3Cl)Br)C(=O)OC SJC00383 Cc1cc(nc(c1[N+](=O)[O-])N)C TL00650 CCOC(=O)Cn1cnc2c3c(cc(nc3oc2c1=O)c4ccccc4)c5ccccc5 HTS09917 Cc1cc(nc2c1c(c(o2)C(=O)NN)N)c3ccccc3 HTS09918 c1ccc(cc1)S(=O)(=O)Nc2cccc3c2cccc3 HTS09168 c1ccc2c(c1)cccc2NS(=O)(=O)c3ccc(cc3)F HTS09169 c1ccc2c(c1)cccc2NS(=O)(=O)c3ccc(cc3)C#N HTS09172 c1ccc2c(c1)nc(s2)c3ccsc3NC(=O)Nc4ccc(cc4)OC(F)(F)F HTS10883 CCNc1c2c3c(sc2nc(n1)SCc4ccc(cc4)F)CC(CC3)C HTS10320 CC(C)(CO)NC(=S)NCc1ccco1 SJC00357 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN(C)C(=S)SC CD07776 CCC(C)Sc1c(c(cs1)c2ccc(cc2)Cl)C#N KM02813 CNC(=O)Nc1nc2cccnc2s1 TG00193 c1ccc(cc1)C2=CC(=C3CCCC(=C3N2c4ccc(cc4)Cl)C(=S)Nc5ccc(cc5)Cl)c6ccccc6 TL00046 c1ccc(cc1)NC(=C(C#N)C#N)N TL00087 CCc1c(nc2ccccc2n1)CC CD07481 c1c(cc(cc1C(F)(F)F)NC(=O)/C=C/C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD07698 CC1CCc2c(sc3c2c(nc(n3)SCc4ccc(cc4)Cl)NCc5ccccc5)C1 HTS10322 CC1CCc2c(sc3c2c(nc(n3)SC)NCc4ccccc4)C1 HTS10324 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)C=C(C#N)C#N HTS09868 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)C=C4C(=O)N(C(=O)N(C4=O)C)C HTS10327 Cc1c(sc(n1)c2cccc(c2Cl)Cl)C(=O)N/N=C/N(C)C SPB01130 C=CS(=O)(=O)c1ccc(cc1[N+](=O)[O-])C(F)(F)F KM03341 CCOc1c2c3c(sc2ncn1)CCCC3 HTS09860 CC1(CC2=C(C(c3c([nH]c(=S)[nH]c3=O)N2)c4ccc(cc4)Cl)C(=O)C1)C HTS09861 c1c(cc(cc1Cl)Cl)NC(=O)/C=C/C(=O)Nc2cc(cc(c2)Cl)Cl CD07705 c1cc(sc1)c2cc(nc(c2)c3cccs3)c4cccs4 CD07718 CCNc1c2c3c(sc2nc(n1)SCC(=O)OCC)CC(CC3)C HTS10321 Cc1c(c(n(n1)C)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] EN00279 Cc1c(c(c(cn1)CSC(=S)N2CCSCC2)CO)O CD08204 CC(c1ccccc1)n2c(nnc2SCC(=O)c3csc4c3cccc4)O HTS09601 COc1cccc(c1)NC(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS09203 CC(=O)CSc1nnc(n1CC=C)c2c(c3c(cc(nc3o2)c4ccccc4)c5ccco5)N HTS10277 CC(=O)/C(=C(/c1ccccc1Cl)\N)/C(=O)OC CD06918 CN(C)/C=C\1/c2ccccc2NC1=O CD07564 c1cc(cc(c1)Cl)C(=O)NC2CCSC2 CD10353 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])NC2CCSC2 CD10418 c1cc(ccc1S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)Cc3cc(cc(c3)NS(=O)(=O)c4ccc(cc4)Cl)C(F)(F)F)Cl CD10712 CC1=C(C(n2c(=O)/c(=C\c3cccs3)/sc2=N1)c4ccccc4)C(=O)OC HTS09897 CC(=O)Nc1c(c2c(s1)CN(CC2)C(=O)OC(C)(C)C)C(=O)c3ccc(cc3)OC HTS09248 CCOC(=O)c1cnn(c1N)C(=O)c2ccc(cc2)C(F)(F)F HTS09762 Cc1nc2c(c(n1)N3CCOCC3)sc(=S)n2c4ccccc4 HTS09904 c1ccc(cc1)Oc2ccc(cc2)NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS09152 c1ccc(c(c1)/C=N/NC(=S)NC2CC3CC2C4C3CC=C4)O CD03151 c1ccc(cc1)n2c3c(cn2)c(ncn3)N/N=C/c4ccc(cc4)[N+](=O)[O-] HTS09967 Cc1cc(n(n1)c2ccccc2C#N)C CD07945 c1ccc2c(c1)N(c3ccccc3S2)C(=O)CN4CCCCC4 HTS10346 c1cc(cc(c1)NC(=O)/C=N/O)C(F)(F)F CD03059 Cc1c(c(no1)c2ccccc2)C(=O)N/N=C/c3cc(ccc3O)Br CD03135 Cn1c(nnc1SCC(=O)N2c3ccccc3Sc4c2cccc4)c5ccc(cc5)Cl HTS10355 CSc1[nH]c2ccsc2c(=O)n1 GK00277 C/C(=N\NC(=O)N)/c1ccccc1Cl CD06413 CCOC(=S)SCc1nc(no1)c2ccc(cc2)Cl CD06442 COc1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)c4ccc(cc4Cl)Cl)c5ccc(cc5)[N+](=O)[O-])c6ccccc6 HTS09108 COc1ccc(cc1OC)CC2c3cc(c(cc3CCN2/N=N/c4cccc(c4)F)OC)OC BW00086 CC(C)(C)C(=O)Nc1ccncc1C(=O)O MO00291 c1ccc(cc1)CN(CCCC#N)Cc2ccccc2 BTB15243 c1ccc(cc1)Cn2c(nnc2SCC(=O)N3c4ccccc4Sc5c3cccc5)c6ccncc6 HTS10352 C=CCn1c(nnc1SCC(=O)N2c3ccccc3Sc4c2cccc4)c5ccccc5 HTS10354 CCOC(=O)c1nn(c2n1c(=O)cc(n2)Nc3ccc(cc3)C)c4ccccc4 HTS09102 Cc1c(nnn1c2cccc(c2C#N)Cl)c3ccccc3 CD08444 c1c(cc(cc1C(F)(F)F)NC(=O)C23CC4CC(C2)CC(C4)C3)C(F)(F)F CD08933 Cc1ccn2c(c1)nc(c2C(=O)NN)C HTS09844 COc1ccc(cc1)C2c3c(c4ccccc4oc3=O)OC(=C2C#N)N HTS09871 c1ccc(cc1)C2c3c(c4ccccc4oc3=O)OC(=C2C#N)N HTS09874 COc1ccc(cc1)/C=N/n2cnc3c(c2=O)sc(=S)n3c4ccccc4 HTS09847 COc1cccc(c1O)/C=N/NC(=S)Nc2cc(c(cc2OC)Cl)OC CD03230 c1cc(c(cc1C#N)[N+](=O)[O-])Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F CD08019 Cc1cccc(c1NS(=O)(=O)c2c(c(c(c(c2C)C)C)C)C)C(C)(C)C CD06474 c1cc(c(cc1NC(=O)c2cc(ccc2O)Br)Cl)F CD06845 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NN(C)c3cccc(c3C#N)Cl CD06832 c1cc(ccc1n2c(c(c(n2)c3ccc(cc3Cl)Cl)C#N)N)[N+](=O)[O-] HTS09113 CCOC(=O)C1=NN(C2(C1c3ccc(cc3)Cl)C(=O)c4ccccc4C2=O)c5ccccc5 HTS09115 c1ccc(cc1)c2ccc(cc2)c3csc(n3)NC(=N)N.Br CD01618 c1ccc(cc1)c2cnn3c2ncc4c3-c5ccccc5C4=O HTS09275 COc1ccc(c(c1)[N+](=O)[O-])n2cccc2 CD03450 c1cc(c(c(c1)Cl)CSC2=NCCN2)F.Br CD05341 C[C@H](c1ccccc1)N2[C@H]3CCC(=O)C[C@@H]3CCC2=O BTB15250 Cc1c(c(=O)n2c3ccccc3[nH]c2c1C#N)/C=N/N4C(=O)CNC4=S HTS10261 CCOc1ccc(cc1)C2C3=C(CC(CC3=O)(C)C)OC4=C2C(=O)CC(C4)(C)C CD03408 c1ccc(cc1)COc2cnc(nc2O)N BTB15242 CSc1ncc(c(n1)O)OCc2ccccc2 BTB15240 Cc1c(c(c(c(c1C)C)CSc2nnc(n2C)CC#N)C)C CD02581 Cc1cc(c(c(c1)C)NC(=O)NC(=O)c2c(c(cc(c2OC)Cl)[N+](=O)[O-])OC)C BTB07720 c1cc(ccc1C#N)N2CCC(CC2)C(=O)NN MO00066 Cc1c(n2ccsc2n1)C(=O)O MO00015 Cc1cn[nH]c1NC=C2C(=O)c3ccccc3C2=O HTS09278 CN(C(=S)SC)NC(=O)Nc1cccc(c1)C(F)(F)F CD07778 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C/c3ccc(cc3Cl)Cl)Cc4ccc(cc4Cl)Cl HTS11165 Cc1ccc(cc1Cl)NC(=S)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03439 CC(=O)c1ccccc1OC(=O)c2c(cccc2Cl)F CD08731 C/C(=N\O)/C(C)(C)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F HTS10427 C/C(=N\O)/C(C)(C)Nc1cccc(c1)Br HTS10430 C/C(=N\O)/C(C)(C)Nc1ccc(cc1)Cl HTS10432 CC(=O)OCC(=O)C1(CCC2C1(CC(C3C2CCC4=CC(=O)C=CC34C)O)C)O TL00535 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)NN HTS09923 c1ccc(c(c1)/C=N/NC(=O)CSc2c3c4c(sc3ncn2)CCCC4)Cl HTS09848 c1ccc(c(c1)NC(=S)Nc2ccc(c(c2)Cl)Cl)SCC(=O)Nc3ccc(c(c3)Cl)Cl CD03499 CCOC(=O)C1CCN(CC1)c2ccc(cc2)C#N MO00017 c1cc2c(cc1C(=O)O)CCCN2 MO00019 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C/c3cccc(c3)O)Cc4ccccc4Br HTS11199 CN(C(=S)SC)NC(=O)Nc1cccc(c1)Cl CD07779 Cc1ccc-2c(c1)NC(c3n2ccc3)c4cccc(c4)[N+](=O)[O-] CD03481 c1cc(cc(c1)C(F)(F)F)/C(=C/c2cccnc2)/C#N CD03602 c1cc(c(c(c1)Cl)C(=C(C#N)C#N)O)Cl CD09114 c1cc(sc1)C(=O)CC2=NCCS2 CD09782 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)Cc5csc(n5)c6ccc(cc6)Cl HTS10662 CCOC(=O)c1cn2c(n1)ccc(n2)N3CCCCC3 HTS10968 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)Nc5cccc(c5)Cl HTS09197 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4cccs4 HTS09721 Cc1ccc(cc1)C(=O)CN2C(=O)c3ccccc3S2(=O)=O HTS10032 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC3CC3 HTS10034 c1ccc(cc1)COC(=O)N2CCC(CC2)NC(=O)Nc3ccc(cc3)OC(F)F HTS10052 Cc1nc(cs1)CSc2nnc(n2Cc3ccco3)c4ccc(cc4)C(F)(F)F HTS11113 CCc1cccc(c1NS(=O)(=O)c2ccc(cc2)C)C(C)CC CD06404 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2cccc(c2)C(F)(F)F HTS11115 c1cc(oc1)c2cc([nH]c(=O)c2C#N)c3cccs3 HTS10307 c1cc(sc1)c2nnc3n2N=C(CS3)c4ccc5c(c4)OCO5.Br HTS09252 CC(C)(C)c1csc(n1)Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD08389 c1ccc(cc1)CNC(=O)CSCCS(=O)(=O)c2ccc(cc2)Cl KM01697 c1cc(ccc1CSC/C(=N\O)/NC(=O)N)Cl CD11209 C/C(=N\O)/C(C)(C)Nc1ccc(cc1)F HTS10437 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C\c3ccc(cc3)N(C)C)C/C=C\c4ccccc4 HTS11164 Cc1cc(c(cc1Cl)C)SCSc2cc(cc(c2)C(F)(F)F)C(F)(F)F EN00254 c1cc(ccc1CSc2[nH]nc(n2)NS(=O)(=O)c3ccc(cc3)F)Cl HTS10718 Cc1ccc(cc1Cl)NC(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS09200 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)Nc5cc(cc(c5)Cl)Cl HTS09202 c1ccc(cc1)c2cc(on2)C3=Nn4c(nnc4SC3)c5cccs5.Br HTS09253 c1ccc(cc1)c2c(n(nn2)c3ccc(cc3F)F)CSc4nnc(s4)N CD08690 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3ccc(cc3)OC(F)F HTS10053 CC(=O)/C(=C(/c1c(cccc1Cl)Cl)\N)/C#N CD06883 CC(C)(C)c1ccc(cc1)c2nnc(o2)CS(=O)(=O)c3ccc(cc3)Cl SPB01811 Cc1ccc(cc1)C(=O)NC(=O)c2ccccc2O HTS10043 c1ccc2c(c1)c(c(s2)C(=O)NC(=O)c3ccccc3O)Cl HTS10046 CCc1ccc(cc1)C(=O)NC(=O)c2ccccc2O HTS10050 c1ccc(cc1)S(=O)(=O)CCSCC(=O)Sc2cccc(c2)Cl KM01731 CC(C)(C)c1ccc(cc1)C(=O)N(C(C)(C)C)OC(=O)c2ccc(cc2Cl)Cl CD08626 CC(=O)NC(=O)c1c(cccc1F)F CD08639 Cc1c(c(no1)c2c(cccc2Cl)Cl)N3C(N(OC3=O)c4ccc(c(c4)Cl)Cl)c5ccccc5Cl CD06803 c1cc(sc1)c2nnc(o2)SCC(=O)c3ccc(cc3)Br HTS10360 c1cc(ccc1CSc2nnc(o2)c3ccncc3)[N+](=O)[O-] HTS10361 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)Oc3ccc4ccccc4c3)Cc5c(cccc5Cl)Cl HTS11166 c1ccc(c(c1)NC(=O)c2ccc(s2)c3ccccn3)Cl KM02485 COc1ccc(cc1OC)NC(=O)c2ccccc2C(=O)O HTS09622 c1ccc2c(c1)ccc(n2)/C=N/Nc3nc4c(ncnc4n3[C@@H]5[C@H]([C@H]([C@@H](O5)CO)O)O)N HTS09837 CC(=NOC(=O)c1csc(n1)Cc2c(cccc2Cl)Cl)C SPB02099 CC1CCc2c(sc3c2c(nc(n3)SCC(=O)N)NCc4ccccc4)C1 HTS10325 c1cc(ccc1C(=O)C2CC2C(=O)c3ccc(cc3)F)F CD08800 Cc1cccc2c1N(CCC2)C(=O)c3c(onc3c4ccccc4)C HTS09533 c1cc(sc1)c2ccc(cn2)C(F)(F)F SEW04044 COc1ccc(cc1)C(=O)c2c(nc(s2)Nc3ccccc3)c4ccccc4 HTS09465 c1ccc(cc1)c2c(sc(n2)Nc3ccccc3)C(=O)c4ccc5c(c4)OCCO5 HTS09466 c1cc(cnc1)n2c(nnc2SCC(=O)c3ccc(cc3)N4CCOCC4)O HTS09469 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNC(=O)c3c(cccc3Cl)Cl CD07189 Cc1ccccc1C(=O)Cc2ccc(cc2)C(=O)N MO00238 COc1ccc(cc1OC)NC(=O)COCC(=O)O HTS09618 COc1ccc(cc1OC)NC(=O)CSCC(=O)O HTS09619 c1c(cc(c(c1[N+](=O)[O-])NC2CCCCNC2=O)[N+](=O)[O-])C(F)(F)F CD10136 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NC(=O)c3c(cccc3Cl)Cl CD10140 c1cc(ccc1C(=O)NCc2ccc(s2)S(=O)(=O)Nc3ccc(cc3)N4CCCCC4)Cl HTS09302 c1ccc(cc1)n2cc(c(n2)c3cccs3)/C=N/NC(=O)c4cccs4 HTS10366 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=O)c3cccs3 HTS10367 CCOC(=O)c1nn(c2n1c(=O)cc(n2)Nc3ccc(cc3)Cl)c4ccccc4 HTS09099 CCOC(=O)c1nn(c2n1c(=O)cc(n2)N)c3ccccc3 HTS09100 c1cc(ccc1C(=O)ONC(=O)CS(=O)(=O)c2ccc(cc2)Cl)Cl KM02124 c1ccc2c(c1)nc(o2)SCC#N KM01287 CC(C)c1cccc2c1OC(C(=S)N2CC(=O)O)C(C)C KM06746 CCOC(=O)C(Cc1cc(c(c(c1)[N+](=O)[O-])O)[N+](=O)[O-])NC(=O)C KM08331 c1coc2c1/C(=N\O)/CCC2 MWP00893 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)NC(=S)N3CCc4c3cccc4 KM09956 CC1CCc2c(sc(c2C#N)NC(=O)CN3CCN(CC3)C)C1 HTS10331 Cc1cccc(c1NC(=O)c2c(ccnc2NC)C(F)(F)F)C RF04608 Cc1c(sc(n1)Nc2ccccc2)C(=O)c3ccc(cc3)OC HTS09474 c1cc2c(cc1C(=O)N3CCOCC3)OCCCO2 HTS09482 c1ccc(cc1)/C=C/C=N/NC(=S)NC2CC3CC2C4C3CC=C4 HR00151 Cc1cccc(c1)C(=O)Nc2c(c3c(s2)CCCC3)C(=O)N HR00224 c1ccc-2c(c1)NC(c3n2ccc3)c4cccs4 HR00248 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2csc(n2)Cc3c(cccc3Cl)Cl)/N SPB02105 Cc1c(sc(n1)Cc2c(cccc2Cl)Cl)C(=O)NN SPB02170 CC(C)(C)C(=O)Nc1c(cccn1)C(=O)O MO00352 CCCN(Cc1ccco1)S(=O)(=O)c2ccc(c(c2)OC)OC KM09248 CCOC(=O)c1nn(c2n1c(=O)c(c(n2)Nc3ccccc3)C(=O)C)c4ccccc4 HTS09101 COCCCNC(=S)N/N=C/c1ccc(cc1O)O CD03150 COc1cccc(c1O)/C=N/NC(=S)NC2CC3CC2C4C3CC=C4 CD03152 CCCCC#Cc1ccc(o1)c2nnc(n2C)S KM09626 c1cc(cc(c1)N)c2ncon2.Cl SEW01229 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)ON(Cc3c(cccc3Cl)F)Cc4c(cccc4Cl)F CD07780 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)c2ccc(cc2)Cl CD03099 COc1ccc(cc1OC)CCNC(=S)Nc2cccc(c2)Cl CD03740 c1ccc(cc1)c2ccc(cc2)C(=O)CSc3nnc(o3)c4ccncc4 HTS10359 c1cc2c(cc1N/N=C(/C#N)\C(=O)N3CCCC3)OCO2 CD01903 c1ccc(cc1)c2nnc(n2c3ccccc3)Sc4c5c(c(c6n4c7ccccc7n6)C#N)CCC5 HTS09910 c1ccc(cc1)c2cc(n3c4ccccc4nc3c2C#N)SCc5ccc(cc5)Cl HTS09913 CCOC(=O)c1c(n(nn1)Cc2ccccc2Cl)N HTS10286 c1ccc(c(c1)Cn2c(c(nn2)C(=O)N)N)Cl HTS10287 Cn1c(nnc1SCc2ccccc2Cl)c3c(c4c(cc(nc4o3)c5ccccc5)c6ccco6)N HTS10288 Cc1ccc(cc1)S(=O)(=O)OC2COc3cc4c(cc3OC2)OCO4 BTB15230 CCN(c1ccc(cc1)Cl)C(=O)c2cnc(cc2C(F)(F)F)SC RF04434 Cc1ccc(c(c1)[N+](=O)[O-])n2cccc2 CD03440 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2cc(cc(c2)OC)C(F)(F)F CD03178 c1cc(ccc1Sc2cc(c(cc2C(F)(F)F)[N+](=O)[O-])Sc3ccc(cc3)Cl)Cl CD04380 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NCCCN)C(F)(F)F CD04330 CCOC(=S)SCc1c(onc1c2c(cccc2Cl)Cl)C CD06441 c1ccc(cc1)C2(Oc3cc(oc(=O)c3C(=O)O2)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)c5ccccc5 CD03188 c1cc(c(c(c1)Cl)CN(Cc2c(cccc2Cl)F)OC(=O)C3CC3)F CD07795 c1c(cc(cc1C(F)(F)F)NCCC(=O)N)C(F)(F)F CD04252 Cc1cc(cc(c1F)C)S(=O)(=O)c2ccc(c(c2)Cl)Cl CD05612 c1cc(cc(c1)Cl)N2CC(CC2=O)C(=O)O CD05924 CC(=O)Nc1ccc(cc1)OCCCNC(=O)C2=NNC(=O)CC2 HTS10247 c1ccc2c(c1)-n3cccc3C(N2C(=O)C(F)(F)F)(C(F)(F)F)O CD03430 c1ccc(cc1)/C=C/C(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD03834 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)C)C HTS10295 Cc1cc(nc2c1c(c(s2)C(=O)c3ccccc3)N)C HTS10296 c1cc(c(c(c1)Cl)CN(Cc2c(cccc2Cl)F)OC(=O)c3ccc(cc3)Cl)F CD07794 Cc1c(c(c(c(c1C)C)CSc2cccc(c2)N)C)C CD02183 Cc1ccc2c(c1)c(cc(=O)o2)CN3CCOCC3 CD04586 c1cc(sc1)/C=C/C(=O)Nc2ccc(c(c2)C(=O)O)N3CCCC3 CD05905 c1cc(sc1)/C=N/OCc2ccc(cc2)Cl CD02586 Cc1cc(c-2c(c1)CC(c3c2nc([nH]3)c4ccc(cc4Cl)Cl)(C)C)C CD02716 CC1(C2CCC(C2)C1(C)NC(=S)N/N=C/c3ccc(cc3O)O)C CD03217 c1ccc(cc1)C2=NN(C(=C3C(=O)c4ccccc4C3=O)C2c5cccs5)c6ccccc6 HTS09120 c1cc(ncc1[N+](=O)[O-])OCC(F)(F)F RF05261 CS(=O)(=O)c1ncc(cn1)OCc2ccccc2 BTB15239 c1cc(ccc1CCC(=O)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])O CD03569 c1ccc(c(c1)/C=N/c2nc(cs2)c3ccccc3Cl)O CD03583 c1cc(c(cc1Br)/C=N/Nc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])O CD03586 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3c(onc3c4c(cccc4Cl)Cl)C CD06075 CC1CN(CC(O1)C)CCCNC(=O)Nc2ccc(cc2)Cl CD06538 COc1cccc(c1O)/C=N/O CD02674 Cc1c(cccc1Cl)NC(=S)NNC(=O)CC#N CD02842 c1ccc(cc1)c2cc(on2)C(=O)CSc3nnc(n3Cc4ccco4)O HTS09147 c1ccc(cc1)C(=O)NC(=S)Nc2ccccc2 CD03873 c1ccc2c(c1)cccc2NS(=O)(=O)c3cccs3 HTS09165 c1ccc2c(c1)cccc2NS(=O)(=O)c3cccc4c3non4 HTS09166 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)Nc2ccc(cc2)OC(F)(F)F HTS11130 Cn1c2c(nc1Oc3ccc(cc3Br)Br)n(c(=O)n(c2=O)Cc4ccc(cc4)Br)C HTS11202 CCOC(=O)COc1c(c(cc(n1)c2ccc(cc2)Cl)c3ccco3)C#N HTS10300 CCOC(=O)COc1c(c(cc(n1)c2ccccc2)c3cccs3)C#N HTS10301 CCOC(=O)COc1c(c(cc(n1)c2ccccc2)c3ccco3)C#N HTS10303 CN(C)CCCNC(=O)c1cc(ccc1O)Br CD06877 c1ccc(c(c1)NC(=O)c2cccc(c2)Cl)SCc3cc(cc4c3OCOC4)Cl CD03412 Cc1cc(c(c(=O)o1)/C(=N/Nc2ccccc2)/C)O CD10303 Cc1ccc(cc1)OCCC#N SEW04413 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)CSCC(=O)O HTS09771 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Cl)Sc3ccc(cc3Cl)Cl HTS10476 c1ccc(c(c1)/C=N/NC(=S)NC2CC3CC2C=C3)O CD03013 Cc1ccc(n1C)CNC(=O)Nc2ccc(cc2F)F HTS10868 COc1ccc(cc1NC(=O)Nc2c(ccs2)c3nc4ccccc4s3)Cl HTS10889 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)Nc2cccc(c2)OC HTS11282 c1ccc(c(c1)/C=N\c2ccccc2SCc3csc(n3)c4ccc(cc4)Cl)O CD03539 COc1cc(cc(c1OC)OC)C(=O)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03567 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cccc2F)F)OC)Cl)Cl BTB07690 c1cc(cc(c1)[N+](=O)[O-])/C=C(\C#N)/c2cccc(c2)C(F)(F)F CD03606 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N3CCCC3c4ccc(cc4)F CD08255 CC1(C2CCC(C2)C1(C)NC(=S)N/N=C/C=C/c3ccccc3)C CD01962 CCN(C(Cc1ccccc1)c2ccc(cc2)OC)C(=O)c3c(onc3c4ccccc4Cl)C CD01979 COC(CNC(=O)C(=O)Nc1nnc(s1)C(F)(F)F)OC CD11670 c1ccc(cc1)C(CC(=O)c2ccc(cc2)F)Sc3ccc(cc3Cl)Cl HTS10477 c1cc(sc1)S(=O)(=O)Nc2nc([nH]n2)SCc3ccc(cc3)Cl HTS10719 c1cc(ccc1CN2CCS(=O)(=O)CC2)C(=O)O HTS08540 c1cc2c(cc1C(=O)N3CCCCC3)OCCCO2 HTS09180 COC(=O)c1c(ccs1)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS09301 COCCCNC(=S)N/N=C/c1cc(cc(c1O)Br)Br CD03211 c1ccc(cc1)c2cc3c(s2)c(ncn3)Sc4ccccc4NC(=O)CSCC(=O)O HTS03498 c1cc(cnc1)n2c(nnc2S)c3ccc(cc3)C(F)(F)F HTS11298 COc1ccc2cc(c(=O)oc2c1)C(=O)O HTS11321 Cc1c(c(nc(n1)c2ccc(cc2)Cl)S)C(=O)C SPB05327 c1cc(c(cc1NC(=S)NCCNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])Cl)Cl CD03709 c1ccc2c(c1)c(=O)n(c(n2)C(=O)NCc3cccnc3)N CD02828 c1cc(ccc1CO)n2ccnc2 CC18509 c1ccc(cc1)c2c(nco2)CO CC10209 Cc1cc(c(c(=O)o1)/C(=N/Nc2c(cc(cc2Cl)Cl)Cl)/C)O CD10299 Cn1cc(nc1)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS08423 c1cc(ccc1C(=O)O)n2ccnc2 CC18501 Cn1c2c(nc1Sc3ccccc3N)n(c(=O)n(c2=O)C)C HTS09819 c1ccc(cc1)[C@H]2[C@@H](N(NC2=O)C(=O)Nc3ccc(cc3)Br)c4ccccc4 BTB15231 c1ccc(cc1)NC(=O)N2CCN(CC2)c3ncccn3 HTS10743 c1ccc2c(c1)c(cc(n2)O)CSC(=S)N3CCSCC3 CD08206 C/C(=N\O)/c1cc(cc(c1O)Cl)Cl CD03801 c1ccn(c1)c2cccc(c2)c3nc(on3)C(=O)NN SPB01493 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)NN3CCOCC3)Cl SPB01172 c1ccc(c(c1)C2Nc3ccccc3C(=O)N2CCCN4CCOCC4)C(=O)O HTS10256 CC(=O)Cc1nc(sn1)Nc2ccc(cc2)Cl SEW04143 CC(=O)c1ccccc1OC(=O)c2cc(cc(c2)Cl)Cl CD08740 c1ccc(cc1)NC(=N)SCc2ccc(cc2)C#N.Br CD00408 c1c(c(c(c(n1)O)[N+](=O)[O-])O)C(=O)O SPB07356 CNc1nc2cccnc2s1 TG00180 Cc1c(c(no1)c2ccccc2)C(=O)Oc3ccc(cc3OC)CCC(=O)C CD07230 c1ccc(cc1)S(=O)(=O)Nc2nc([nH]n2)SCc3ccc(cc3)Cl HTS10717 Cc1c(cccc1Cl)NC(=S)Nc2cc(ccc2n3cccc3)OC CD03468 CCCCNC(=O)NNC(=O)c1cc(on1)C SPB01198 Cc1cc(no1)n2nc(nn2)CC(=O)C CD09268 Cn1c(cc(n1)c2ccccc2)NC(=O)c3ccccc3C(=O)O HTS10207 C[C@@H](c1ccccc1)N2[C@H]3CCC(=O)C[C@@H]3CCC2=O BTB15247 Cc1ccc(cc1)n2c(nnn2)c3c[nH]c4c3cc(cc4)C HTS10403 COc1ccc(cc1N/C=C/c2nnnn2c3ccc(cc3)F)C(F)(F)F HTS10406 c1cc(sc1)c2ccn(n2)C(=O)c3ccc(cc3)C(F)(F)F HTS09515 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC(C)C(OC)OC CD08279 CCOC(=O)NNC(=S)Nc1ccc(c(c1)Cl)Cl SPB01176 c1c(cc(cc1Cl)Cl)C/C(=N/O)/N SPB01241 c1ccc(c(c1)NC(=S)Nc2cc(ccc2Cl)Cl)SCc3nc(no3)c4ccc(cc4)Cl CD03172 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/NC(=O)CN4c5ccccc5Sc6c4cccc6 HTS10338 c1cc(c(c(c1)Cl)OCc2cc(no2)C(=O)NN)Cl SPB01363 c1ccc(c(c1)C(c2c([nH]c(=S)[nH]c2=O)N)c3c([nH]c(=S)[nH]c3=O)N)Cl HTS09842 Cc1c(c(=O)n2c3ccccc3[nH]c2c1C#N)/C=N/NC(=S)N HTS09843 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)NCc3ccco3)C#N HTS11257 Cc1cc(no1)NC(=O)c2ccc(cc2)C(F)(F)F SPB03063 Cc1cc(cc(c1N2CCOCC2)C)[N+](=O)[O-] CD08282 CCOC(=O)C(c1ccccc1)C(c2ccccn2)Nc3ccc(cc3)F CD03624 c1ccc(c(c1)C(=O)O)Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03735 c1ccc2c(c1)N(c3ccccc3S2)C(=O)c4cccc(c4)[N+](=O)[O-] HTS10342 c1ccc2c(c1)N(c3ccccc3S2)C(=O)CN4CCOCC4 HTS10345 Cc1c(cn(n1)S(=O)(=O)c2ccc(cc2)Cl)c3ccccc3 CD09353 CCCCNC(=O)Nc1cc(cc(c1)Cl)Cl CD12019 CSC1=NCCCN1S(=O)(=O)c2cc(c(cc2Cl)Cl)Cl DP01328 Cc1ccc(cc1)Oc2c(cccn2)C(=O)n3ccc(n3)c4cccs4 HTS09527 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)n3ccc(n3)c4cccs4 HTS09532 C#Cc1cccc(c1)/N=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD07886 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)[N+](=O)[O-])/C=N/NC(=O)CN4c5ccccc5Sc6c4cccc6 HTS10341 c1ccc2c(c1)N(c3ccccc3S2)C(=O)CSc4nnc(o4)c5ccncc5 HTS10349 c1cc(cnc1)/C=N/n2c(n[nH]c2=S)c3ccncc3 HTS09845 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4ccc(cc4)OC)C HTS10278 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4ccc(c(c4)OC)O)C HTS10279 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4ccccc4Cl)C HTS10280 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)Nc4cc(cc(c4)C)C HTS09488 Cc1c(nn(n1)c2ccccc2)CO CC16209 CCOC(=O)/C(=N\Nc1ccccc1Cl)/C(=O)CSc2ccc(cc2)Cl SPB04016 COc1ccc(cc1)OC/C(=N/O)/N SPB04281 c1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)C(=O)Nc4ccccc4)c5ccccc5)c6ccccc6 HTS09285 CNC(=O)OCCSCCS(=O)(=O)c1ccc(cc1)Cl KM01840 C/C(=N\O)/C(C)(C)Nc1ccccc1 HTS10439 Cc1c2c(cc(s2)C(C)(C)C)sc1C(=O)NCc3ccccc3 GK01922 Cc1nc(cs1)c2cccc(c2)N CC19414 Cn1c(nnc1SC)c2ccc(s2)Br KM02912 c1ccc(c(c1)n2c(nnn2)c3cnccc3C(F)(F)F)Cl RF04522 c1ccc(c(c1)n2c(nnn2)c3cnccc3C(F)(F)F)F RF04524 Cc1cc(n2c(n1)nc(n2)SCC(=O)Nc3ccc(cc3)C(C)C)C SPB02422 CCOC(=O)C1=NN(C2(S1)N(C(=O)/C(=C\c3ccc(cc3)C)/S2)c4ccccc4)c5ccccc5 HTS09284 Cc1c(c(on1)C)c2nc(no2)CSc3nnc(n3C4CC4)O HTS09145 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cccc3c2cccc3 HTS09170 Cc1c(sc(n1)c2ccc(cc2)Cl)C(=O)NN SPB01248 Cc1c(cc2c(c1NC(=O)c3c(cccc3OC)OC)C(CC2(C)C)(C)C)N4CCCC4 CD03940 c1ccc(cc1)NC(=S)Nc2nccs2 CD04340 Cc1c(c(no1)c2ccccc2Cl)NC(=O)OCc3c(cccc3OC)OC CD04768 CC(=N)NS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F CD06839 CCc1cccc(c1NC(=O)Nc2ccccc2)C(C)C CD06435 CCc1cccc(c1NC(=O)c2cccs2)C(C)CC CD06436 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)N/N=C/c4ccc(cc4Cl)Cl KM09831 CN1CCCCC(C1=O)c2cccc(c2c3cccc(c3)OC)OC BTB15237 Cc1c(c(nn1c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3Cl)Cl)C(=O)Nc4ccccc4 HTS09110 c1ccc(cc1)c2c(c(nn2c3ccc(cc3)[N+](=O)[O-])c4ccc(cc4Cl)Cl)C(=O)c5ccccc5 HTS09111 CCOC(=O)c1c(nn(c1c2ccccc2)c3ccc(cc3)[N+](=O)[O-])c4ccc(cc4Cl)Cl HTS09112 COc1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)c4ccccc4)c5ccccc5)c6ccccc6 HTS09287 c1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)c4ccccc4)c5ccccc5)c6ccccc6 HTS09288 c1ccc(cc1)NC(=O)c2ccc3c(c2)OCCCO3 HTS09173 c1cc(oc1)CNC(=O)c2ccc3c(c2)OCCCO3 HTS09178 COCCOc1ccc(cc1)NC(=O)c2cc(c(c(c2)OC)OC)OC CD05910 CN(Cc1ccccc1)C(=O)Nc2ccccc2 CD06448 CSc1c(c(cs1)c2ccc(cc2)Cl)CNC(=O)Nc3ccccc3 KM02140 c1ccc(c(c1)C(=O)NC2CCSC2)NC(=O)c3ccc(cc3)[N+](=O)[O-] CD10411 c1ccc(c(c1)NC(=O)NC(=O)c2cccc(c2)CS(=O)(=O)c3ccc(cc3)Cl)Cl KM02352 Cc1c(c(no1)c2ccccc2)NC(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS09199 COc1ccc(cc1OC)NC(=O)CC2(CCCC2)CC(=O)O HTS09623 Cc1cc(nc2c1c(c(s2)C(=O)NNC(=S)NC)N)C HTS10372 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/n4cnc5c6c(cc(nc6sc5c4=O)C)C HTS10373 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)Nc5ccc(cc5F)F HTS09204 Cc1c(c(no1)c2ccccc2Cl)C(=O)NN(C)C CD01647 COc1ccc(c(c1)C(=O)c2ccc(cc2)Cl)OC CD02511 c1c(cc(c(c1[N+](=O)[O-])NNC(=O)/C=C/C(=O)O)[N+](=O)[O-])C(F)(F)F CD03431 CCOC(=O)C1=NN(C2(S1)N(C(=O)/C(=C\c3ccccc3)/S2)c4ccccc4)c5ccc(cc5)Cl HTS09118 CCN(CC)CC(=O)Nc1c(c2c(s1)CC(CC2)C)C#N HTS10333 c1ccc(cc1)Cn2c(c(nn2)C(=O)N)N HTS10374 CC(C)(C)OC(=O)N1CCc2c(sc(c2C(=O)c3ccc(cc3)OC)NC(=O)CCC(=O)O)C1 HTS09249 CC1CCc2c(sc(c2C#N)NC(=O)CN3CCCCC3)C1 HTS10334 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=O)CN3c4ccccc4Sc5c3cccc5 HTS10339 CC(=O)/C(=C\Nc1cc(cc(c1)Cl)Cl)/C(=O)C(F)(F)F KM02443 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)Nc4ccccc4 HTS09485 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)Nc4cccs4 HTS09489 Cc1cc(nc2n1nc(c2Br)c3ccc(cc3)C(C)(C)C)C(F)(F)F KM02455 CCOC(=O)c1cnn(c1N)C(=O)Cc2cccc(c2)OC HTS11290 CCn1c(nnc1SCc2ccc(cc2)[N+](=O)[O-])CN3c4ccccc4Sc5c3cccc5 HTS10335 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)/C=N/NC(=O)CN4c5ccccc5Sc6c4cccc6 HTS10337 CN(C)c1ccc(cc1)C(=O)Cc2ccccc2 MO00225 CN(C)c1ccc(cc1)C(=O)Cc2ccccc2Cl MO00226 Cc1c(snn1)C(=O)NCc2ccc(cc2)N3CCOCC3 HTS09729 c1cc(ccc1C(=O)O)n2ccc(n2)C(F)(F)F MO00070 c1cc(ccc1NC(=O)c2ccc3c(c2)nccn3)S(=O)(=O)N HTS08966 Cc1cc(nc2c1c(c(s2)C(=O)NNC(=S)NCC=C)N)C HTS10283 CCOC(=O)c1c(n(nn1)Cc2ccccc2)N HTS10285 CC(=O)C1=NN(C2(S1)N(C(=O)/C(=C\c3ccc(cc3)OC)/S2)c4ccccc4)c5ccccc5 HTS09279 Cc1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)C(=O)c4cccs4)c5ccccc5)c6ccccc6 HTS09281 c1cc(c(c(c1)Cl)CN(Cc2c(cccc2Cl)F)OC(=O)c3cccs3)F CD07747 c1ccc(cc1)n2cc(c(n2)c3cccs3)/C=N/NC(=O)CN4c5ccccc5Sc6c4cccc6 HTS10340 c1ccc(cc1)OCC(=O)N2c3ccccc3Sc4c2cccc4 HTS10343 c1ccc(cc1)N2CCN(CC2)CC(=O)N3c4ccccc4Sc5c3cccc5 HTS10344 Cc1cc2c(cccc2NC(=O)Nc3ccc(cc3)C(F)(F)F)nn1 HTS09565 Cc1cc2c(cccc2NC(=O)Nc3ccc(cc3)F)nn1 HTS09567 c1cc(ccc1C(=O)CN2C(=O)CCC2=O)OC(F)F HTS10065 CC(=O)Nc1ccc(cc1)c2[nH]c(=O)c3ccccc3n2 HTS10513 c1ccc(cc1)C(=O)n2ccc(n2)c3cccs3 HTS09513 c1ccc(cc1)C2=NOC(C2)Cn3cc(c(=O)n(c3=O)CC4CC(=NO4)c5ccccc5)F HTS09783 c1nc(c2c(n1)n(c(n2)N3CCCCC3)[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09785 c1cc(c(c(c1)Cl)/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N)Cl HTS09790 c1ccc(cc1)C(CC(=O)c2ccc(cc2)Br)Sc3ccc(cc3Cl)Cl HTS10475 CS(=N/C=C(\C#N)/S(=O)(=O)C)(=O)c1ccsc1 KM05868 Cc1ccc(cc1)CC(=O)c2cccnc2 MO00230 c1ccc(cc1)C(=O)Cc2cccc(c2)C(=O)N MO00240 c1ccc2c(c1)nc(s2)SCC(=O)N3c4ccccc4Sc5c3cccc5 HTS10347 c1ccc2c(c1)[nH]c(n2)SCC(=O)N3c4ccccc4Sc5c3cccc5 HTS10350 c1ccc2c(c1)nc(o2)SCC(=O)N3c4ccccc4Sc5c3cccc5 HTS10351 Cc1cc2c(cccc2NC(=O)CSCC(=O)O)nn1 HTS09552 c1cc(ccc1NC(=O)CSCC(=O)O)OC(F)F HTS09557 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)Cc4ccc(cc4)F)C HTS10292 c1ccc(cc1)c2cc(c(c(n2)OCC#N)C#N)c3ccco3 HTS10302 c1ccc(cc1)/C=C/C(=O)OCC2CCCN3C2CCCC3 HTS11200 C=CCn1c(nnc1SCC(=O)N2c3ccccc3Sc4c2cccc4)c5ccco5 HTS10353 c1ccc(cc1)n2c(nnc2SCC(=O)N3c4ccccc4Sc5c3cccc5)c6ccco6 HTS10356 CCOC(=O)c1c(c2c(c(sc2s1)C(=O)OCC)N)C(C)(C)C KM03475 c1ccc2c(c1)c(c(s2)C(=O)n3ccc(n3)c4cccs4)Cl HTS09522 Cc1cc(c(o1)C)C(=O)n2ccc(n2)c3cccs3 HTS09530 c1ccc2c(c1)c-3ccc(oc3c2C(=O)C(F)(F)F)c4ccc(cc4)Cl HTS10379 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)NN3CCOCC3)Cl SPB02098 c1cc(ccc1C(=O)O/N=C(/COc2ccc3c(c2)non3)\N)Cl KM07275 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)C KM07350 CC(C)(C)c1ccc(cc1)C2=NNC(=NN2)SCC(=O)c3ccccc3 HTS06860 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(sc3C(=O)OC)c4ccc(cc4)Cl HTS09394 CN(C)/C=N/c1nc(n(n1)CCC#N)SC CD10155 c1ccc(c(c1)CSc2[nH]c(cn2)c3ccc(cc3)Cl)Cl SPB01533 c1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)C(=O)c4cccs4)c5ccccc5)c6ccccc6 HTS09280 CN(C)c1cc(oc(=O)c1Cl)c2ccc(c(c2)Cl)Cl CD11125 CC(C)(C)c1cc(c(s1)C(=O)OC)NC(=O)NC(=O)c2ccccc2Cl GK00738 c1cc(cnc1)NC(=O)CCCC(=O)Nc2cccnc2 CD07599 CC(C)(C)c1nnc(n1C)S CD07622 c1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3ccc(cc3)Cl)N KM09684 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(Cc3c(cccc3Cl)Cl)Cc4c(cccc4Cl)Cl CD06837 Cc1ccc(cc1)C2C(=NN(C23C(=O)c4ccccc4C3=O)c5ccccc5)c6ccccc6 HTS09114 CC(C)(C)c1ccc(cc1)C2=NNC(=NN2)SC HTS06858 CC(C)(C)c1ccc(cc1)C2=NNC(=NN2)SCC=C HTS06859 c1ccc2c(c1)CC(C2)NC(=O)CC3C(=O)NCCN3 HTS08247 CC(C)(C)c1ccc(cc1)c2nnc(n2C)SCC(=O)c3ccc4ccccc4c3 SPB00604 c1ccc-2c(c1)NC(c3n2ccc3)c4ccc5c(c4)nsn5 HTS11091 c1ccc(cc1)C2(C(=O)c3ccccc3C2=O)N4CCN(CC4)c5ccccn5 HTS11161 CC1SCC(=NOCc2ccccc2)CS1 CD10162 CN(C)C(=O)CS(=O)(=O)c1ccc(cc1)Cl KM01686 CCC/C(=N/Nc1nc2c(n1C)c(=O)n(c(=O)n2C)Cc3ccccc3Cl)/C HTS11163 Cn1c2c(nc1NCCO)n(c(=O)n(c2=O)Cc3ccccc3)C HTS09814 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC3CC(=NO3)c4ccccc4 HTS09835 Cc1c(cnn1c2ccccc2)S(=O)(=O)N3CCCc4c3cccc4 HTS10624 c1ccc(c(c1)C(F)(F)F)NC(=O)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl SPB01164 CC1SCC(CS1)NC(=O)Nc2ccc(cc2)Cl CD10170 Cc1c(nc2nnc(n2n1)S)O SPB01530 C#CCSc1[nH]c(nn1)c2ccc(cc2)C(F)(F)F SPB01429 Cn1c2c(nc1Oc3ccc(cc3)OCc4ccccc4)n(c(=O)n(c2=O)Cc5ccc(c(c5)Cl)Cl)C HTS09808 c1cc(oc1)c2ccnc(n2)S MWP00518 Cn1c(nnc1S)c2csc(n2)c3cccnc3 MWP00427 c1ccc2c(c1)cccc2c3nnc(n3Cc4ccco4)S HTS11303 CC1CN(CC(O1)C)c2ccc3nnc(n3n2)c4ccc(cc4)C(F)(F)F HTS10498 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NC3CSC(SC3)C CD10182 CC1CCc2c(sc3c2c(nc(=S)[nH]3)NCc4ccccc4)C1 HTS10368 c1ccc(cc1)N2C(=O)CSC23N(N=C(S3)c4cccs4)c5ccccc5 HTS08488 Cc1cc2nnc(c(n2n1)C)C#N KM01310 Cn1ccc(n1)c2cccc(c2)[N+](=O)[O-] KM01914 CC(C)S(=O)(=O)c1csc(c1n2cccc2)C(=O)NN KM02211 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4ccc(c(c4)OC)OC HTS09723 CCOC(=O)/C(=N\Nc1ccccc1Cl)/C(=O)CSc2c(c(cc(n2)C)C)C#N SPB03980 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)OCc3ccccc3Cl)Cc4ccc(cc4)Cl HTS09806 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)Sc3ccccc3)Cc4ccc(cc4Cl)Cl HTS09809 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NC3CCCCC3)Cc4ccc(cc4)Br HTS09810 CCOC(=S)Nc1ccc(cc1)I NH00781 COc1cccc(c1)Cc2nnc(n2Cc3ccco3)S HTS11295 c1ccc(cc1)C2CCC(=O)C(C2=O)C(=O)c3ccc(cc3Cl)Cl KM05556 COc1ccccc1CC(=O)NC(=O)c2ccccc2O HTS10045 Cc1cc(c(cc1Cl)C)SCc2nc(no2)c3ccc(cc3)OC(F)(F)F SPB03043 c1ccc(cc1)S(=O)(=O)CCSCC(=O)Sc2ccc(cc2)Cl KM01726 CCOC(=O)c1c(c(n2c1-c3cc(c(cc3CC2)OC)OC)C)/N=N/c4ccc(cc4)C HTS09098 CCOC(=O)c1nn(c2n1c(=O)cc(n2)Nc3ccccc3)c4ccccc4 HTS09103 c1ccc(cc1)C2=CCN(CC2)CCCC(=O)O.Cl KM09821 CCOC(=O)c1c(nc(s1)c2ccccc2)OC(=O)c3ccc(cc3)C(F)(F)F SPB02743 c1ccc(cc1)CSc2nccc(n2)/C=N/O SPB04300 c1ccc(cc1)S(=O)(=O)c2csc(c2NC(=O)c3ccccc3Cl)Cl KM01810 Cc1ccc(cc1)S(=NC(=O)NC(=O)c2c(cccc2Cl)F)(=O)C KM02957 c1cc(oc1)CSc2cc(c(cn2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F RF04441 CCOC(=O)/C(=C/Nc1ccsc1C(=O)C)/C#N GK00030 Cc1c(sc(n1)CS(=O)(=O)c2ccccn2)C(=O)NN SPB02447 CC(=O)Nc1ccc(cc1)NCN2C(=O)c3ccccc3C2=O HTS08958 COc1cc2c(cc1OC)C3N(CC2)C(=NN3c4ccc(cc4)[N+](=O)[O-])c5ccc(cc5Cl)Cl HTS09106 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)ONC(=O)Cc3ccccc3 CD05774 Cc1c(c(no1)c2ccccc2)C(=O)N/N=C/c3cccs3 CD03166 c1cc(cnc1)/C=N/Nc2ccc(cc2[N+](=O)[O-])S(=O)(=O)NCc3ccco3 BLT00208 CSC(=C(C#N)c1nc2ccccc2s1)SC GK00582 COC(=O)c1cc(c(s1)C(=O)OC)O GK00695 c1ccc(cc1)C(=O)O/N=C(/c2cc[nH]n2)\N SPB02828 CN(C(=S)SCc1c(cccc1Cl)F)NC(=O)Nc2c(cccc2Cl)Cl CD07772 Cc1c(c(on1)C)CSc2nnc(n2Cc3ccco3)O HTS09463 c1cc(ccc1C(=O)CSc2nnc(n2C3CC3)O)N4CCOCC4 HTS09470 CN(C)c1ccc(cc1)C2c3cccn3-c4ccc(cc4N2)OC HTS08871 c1cc(c(c(c1)Cl)CSCCNC(=O)c2ccc3c(c2)nccn3)F HTS09578 Cc1cc2c(cccc2NC(=O)CC(C)(C)CC(=O)O)nn1 HTS09554 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)OC/C=C/c3ccccc3)Cc4ccc(c(c4)Cl)Cl HTS09838 c1cc(c(c(c1)Sc2ccc(cc2)Cl)CNC(=O)Nc3ccc(cc3)Cl)F CD11854 C#CCNC(=S)NC(=O)c1cc(sc1)[N+](=O)[O-] DFP00147 CC(C)CNC(=S)NC(=O)c1cc(sc1)[N+](=O)[O-] DFP00148 Cc1c(nn(n1)c2ccccc2)C(=O)N(C)c3nnc(s3)C(F)(F)F HTS08803 c1cc(ccc1C(=O)O/N=C(/c2cc[nH]n2)\N)Cl SPB02829 CN1c2ccccc2C(=O)C(=C(SC)SC)S1(=O)=O KM01627 CC(C)NC(=O)O/N=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl KM01736 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(s3)c4ccccn4 HTS09692 Cc1c(sc(n1)Nc2ccccc2)C(=O)c3ccc4c(c3)OCCO4 HTS09475 Cc1c(sc(n1)Nc2ccccc2)C(=O)c3ccc4c(c3)OCCCO4 HTS09476 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)Cl HTS09697 CC1CC(=O)Nc2ccccc2N1C(=O)c3ccc(cc3F)F HTS09701 COc1cc(ccc1O)/C=N/NC(=S)Nc2cc(c(cc2OC)Cl)OC CD03235 c1ccc2c(c1)c(c(s2)C(=O)NNc3ccccc3F)Cl HTS05021 c1ccc(cc1)C2=NN(C3(C2c4ccc(cc4)Cl)C(=O)c5ccccc5C3=O)c6ccccc6 HTS09116 c1ccc2cc(ccc2c1)c3nnc(o3)CO/N=C/c4cccc5c4OCO5 HTS08815 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F HTS09702 c1ccc(cc1)n2c(nnc2SCC(=O)N3c4ccccc4Sc5c3cccc5)c6cccs6 HTS10357 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3cccc(c3)Cl HTS09703 c1ccc(c(c1)CSc2nnc(o2)c3cccs3)Cl HTS10362 c1cc(c(c(c1)Cl)CSc2nc3cc(ccc3s2)Cl)F EN00190 C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/C=C/c2ccccc2 EN00224 Cn1c(nnc1SCC(=O)N2c3ccccc3Sc4c2cccc4)c5ccncc5 HTS10358 CC(C)(C)c1cc(no1)N/C=C/C(=O)c2ccc(cc2)Cl HTS09294 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)[N+](=O)[O-])/C=N/NC(=O)c4cccs4 HTS10363 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/NC(=O)c4cccs4 HTS10364 c1ccc(cc1)C(=O)c2cc(ccc2N/C=C/c3nnnn3c4ccc(cc4)Cl)Cl HTS09290 COc1cc(c(cc1Cl)OC)NC(=S)N/N=C/c2cc(cc(c2O)Br)Br CD03246 c1c(cc(cc1C(F)(F)F)NC(=S)NNC(=O)CC#N)C(F)(F)F CD03304 c1ccnc(c1)/C=N/Nc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03427 c1cc(c(c(c1)Cl)C#N)Oc2ccc(cc2)S(=O)(=O)Oc3ccc(cc3)F CD07111 C=CCc1cccc(c1O)C(=O)O HTS11162 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)c3cccs3 HTS08869 COc1ccc-2c(c1)NC(c3n2ccc3)c4ccccc4 HTS08873 CN(Cc1nnc(o1)c2ccc3ccccc3c2)c4nnc(s4)C(F)(F)F HTS08817 c1cc(cc(c1)Cl)c2c(cno2)c3nnnn3c4ccc(cc4)Cl HTS09291 c1cc(ccc1n2c(nnn2)c3cnoc3c4ccc(cc4F)F)Cl HTS09293 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/NC(=O)c4cccs4 HTS10365 CC(=O)C1=NN(C2(S1)N(C(=O)CS2)c3ccccc3)c4ccccc4 HTS08487 c1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4cccc(c4)Cl HTS09297 CCOC(=O)c1c(c(n2c1-c3cc(c(cc3CC2)OC)OC)c4cccs4)/N=N/c5ccc(cc5)C HTS08489 Cc1c(c(on1)c2ccccc2)C(=O)O CC20301 CN1CCN(CC1)c2ccc(cc2)C(=O)O CC18701 c1cc(cc(c1)C(=O)NN)COc2ccc(cc2)C3SCCS3 SPB01991 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3cc(on3)C)C HTS08819 Cc1ccc(cc1NC(=O)N2c3ccccc3NC(=O)CC2C)F HTS08877 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccsc3C(=O)OC HTS09693 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3cccc(c3)F HTS09696 c1ccc2c(c1)[nH]c(n2)SCn3c4ccccc4sc3=S HTS09300 CCOC(=O)c1c(c(n2c1-c3cc(c(cc3CC2)OC)OC)c4ccccc4)/N=N/c5ccccc5 HTS08490 c1ccc(cc1)c2c(c(nn2c3ccc(cc3)[N+](=O)[O-])c4ccc(cc4Cl)Cl)S(=O)(=O)c5ccccc5 HTS09104 c1ccc(cc1)C2C3(C(=NN2c4ccc(cc4)[N+](=O)[O-])c5ccc(cc5Cl)Cl)C(=O)c6ccccc6C3=O HTS09105 c1cc2c(cc1F)CC(C(=O)C2)C3=Cc4ccc(cc4CC3)F BTB15248 c1cc(sc1)c2c(cno2)c3nnnn3c4ccc(cc4)Cl HTS09292 CC(C)(CC(=O)N1CCN(CC1)c2ccccc2)Sc3ccc(cc3)Cl HTS09677 c1ccc(cc1)c2cc(sc2C(F)(F)F)c3cc([nH]n3)N SEW03390 c1cc(ncc1C(F)(F)F)N2CCCN(CC2)C(=O)CCCC(=O)O HTS11041 COC(=O)c1c(nc(s1)SC)N KM05084 c1cc(ccc1Cc2nc(on2)C(=O)NN)[N+](=O)[O-] SPB01581 c1cc(oc1)/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09794 c1cc(sc1)C2CC(=CC(=S)S2)N3CCCCC3 KM04230 c1c(nc2c(cnn2c1C(F)(F)F)C(=S)N)C(F)(F)F KM05243 Cn1c(nnc1S)Cn2cccc(c2=O)OC KM07212 c1ccc(c(c1)c2c(cn[nH]2)c3nnnn3c4ccc(cc4)Cl)Cl HTS09296 c1cc(ncc1C(F)(F)F)N2CCCN(CC2)C(=O)COCC(=O)O HTS10860 Cc1c(c(n(n1)C)NNS(=O)(=O)c2ccc(c(c2)Cl)Cl)[N+](=O)[O-] EN00285 Cc1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)c4ccc(cc4Cl)Cl)c5ccc(cc5)[N+](=O)[O-])c6ccccc6 HTS09109 c1cc(ccc1c2csc(n2)N3CCN(CC3)c4ccc(c(c4)Cl)Cl)Cl HTS10386 c1ccc(cc1)n2c(nnn2)c3cnc(nc3c4cc(cc(c4)F)F)c5ccccn5 HTS10388 c1ccc2c(c1)/C(=N/Nc3nc4c(ncnc4n3[C@@H]5[C@H]([C@H]([C@@H](O5)CO)O)O)N)/C(=O)N2 HTS09797 Cn1c2c(c(=O)n(c1=O)C)n(cn2)Cc3ccc(cc3)OC HTS09802 CCC(c1c(nc([nH]c1=O)SCc2ccc(cc2)[N+](=O)[O-])N)c3c(nc([nH]c3=O)SCc4ccc(cc4)[N+](=O)[O-])N HTS10370 c1ccc2c(c1)C(=O)C(=C3C=CNC=C3)C2=O HTS09829 c1ccc(cc1)C2=NOC(C2)COC(=O)c3ccc4ccccc4n3 HTS09830 c1c(cc(cc1Br)Br)CSc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00762 Cc1cc(=O)[nH]n1c2ccccc2C#N CD07944 c1ccc(cc1)c2cn[nH]c2NC=C3C(=O)c4ccccc4C3=O HTS09277 Cn1c2c(nc1N/N=C/c3ccccn3)n(c(=O)n(c2=O)C)C HTS09816 CCOC(=O)CC(=O)CSc1nccc(n1)c2cccnc2 MWP01041 Cc1ccc(cc1Cl)NC(=S)N2CCOC2c3cccnc3 NH00093 CCOC(=O)NC(=S)NCCc1c[nH]c2c1cccc2 NH00409 Cn1c2c(nc1N/N=C/c3ccncc3)n(c(=O)n(c2=O)Cc4ccccc4)C HTS09817 c1cc(ccc1C(=O)/C(=N/O)/C#N)Cl KM01411 c1cc2c(cc1C(=O)NCc3ccsc3)OCCCO2 HTS09725 CC(=O)/C(=C(\N=C\N(C)C)/SCc1c(cccc1Cl)Cl)/C#N CD09261 Cc1ccc(cn1)C(=O)/C=C/N(C)C CD11041 c1cc(ccc1SCc2cc(no2)C(=O)NN)Cl SPB01357 c1ccc2c(c1)C(=O)C(=Cc3cccs3)C2=O CD12035 c1ccc(cc1)C(=O)C2=NOC3(C2c4ccc(cc4)Cl)C(=O)c5ccccc5C3=O HTS09274 c1ccc(cc1)C2C(=NOC23C(=O)c4ccccc4C3=O)C(=O)c5cccs5 HTS09276 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N3CCCC3)Cc4ccc(c(c4)Cl)Cl HTS09811 CCN(CC)CCNc1nc2c(n1Cc3ccc(c(c3)Cl)Cl)c(=O)n(c(=O)n2C)C HTS09813 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)c3cc(sc3Cl)Cl HTS08868 c1cc(c(c(c1)Cl)/C=N/OC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl)F SPB01174 Cc1ccc(cc1)CN2CCS(=O)(=O)CC2 HTS11011 c1cc(cc(c1)/C(=N/OC(=O)c2cccs2)/N)COc3ccc(cc3)Cl KM01654 CNC(=S)Nc1cscc1S(=O)(=O)c2ccc(cc2)Cl KM01663 CCOC(=O)c1ccc(cc1)Oc2ccc(nn2)C CC21323 c1ccc(cc1)S(=O)(=O)c2csc(c2NC(=O)c3ccccc3Cl)Br KM01792 COc1ccc(cc1N/C=C/c2nnnn2c3ccc(cc3)Cl)C(F)(F)F HTS10407 c1ccc2c(c1)c(=O)n(c(n2)S)c3ccc(cc3)F RDR01284 COc1ccc(cc1N/C=C/c2nnnn2c3ccc4ccccc4c3)C(F)(F)F HTS10408 c1ccc(cc1)c2c3cc(ccc3ncc2c4nnnn4c5ccc(cc5)F)Cl HTS10471 c1ccc(cc1)CN2CCN(CC2)CCCNC(=O)c3ccc(cc3)C(F)(F)F HTS10448 CSc1[nH]c(cn1)c2ccc(cc2)Cl SPB01509 CC(C)(C)c1ccc(s1)C(=O)Nc2cc(cc(c2)Cl)Cl MBE00128 Cc1c(cccc1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3)C(=O)OC KM09982 CCOC(=O)c1cnn(c1N)C(=O)Cc2ccsc2 HTS11293 CCCc1ccc(cc1)C(=O)NC(=O)c2ccccc2O HTS10049 CCOC(=O)C1=C(OC(=C(C1c2ccccc2)C#N)N)C MO00202 Cn1c(cc(n1)c2ccccc2)NC(=O)c3cc(sc3Cl)Cl HTS10201 Cc1cc(no1)C(=O)Nc2ccc(cc2)Cl SPB03088 Cc1c(c(n(n1)C(=O)c2ccc(cc2)C(F)(F)F)C)Oc3ccc(cc3)Cl SPB03998 Cc1cc(no1)C(=O)NN2C3CSC2CS3 SPB04006 CC(=O)/C(=N/Nc1ccccc1Cl)/C(=O)c2ccccc2 SPB04007 c1cc(ccc1C(c2c([nH]c(=S)[nH]c2=O)N)c3c([nH]c(=S)[nH]c3=O)N)[N+](=O)[O-] HTS10494 Cc1c(cc2c(c1/N=C/c3cc(cc(c3O)Cl)Cl)C(CC2(C)C)(C)C)n4cccc4 CD03899 CSc1nnc(n1c2ccc(cc2Cl)Cl)CCCO CD10439 CC(C)(C)c1ccc(cc1)C(=O)CC(=O)N CD11784 c1ccc2c(c1)nc(s2)C/C(=N/O)/N GK00662 c1ccc(cc1)Oc2c(cccn2)C(=O)n3ccc(n3)c4cccs4 HTS09525 C=C(C(CCCCOc1ccc(cc1)Cl)O)C(=O)O BTB15249 c1ccc(cc1)S(=O)(=O)N(c2ccc(cc2)S(=O)(=O)N)S(=O)(=O)c3ccccc3 HTS10187 c1ccnc(c1)c2ccc(s2)C(=O)Nc3ccc(cc3)Cl KM02483 c1cc(ccc1S(=O)(=O)/C(=C/NN2CCCCC2)/C#N)Cl KM02640 Cc1ccc(cc1)S(=NC(=O)c2ccc(cc2)C(C)(C)C)(=O)C KM02795 c1cc(c(c(c1)Cl)Cn2cc(c(=O)[nH]c2=O)F)Cl HTS09781 CC(=O)Nc1ccc(cc1)NC(=O)Nc2ccc(cc2)F HTS08574 c1cc(c(cc1[N+](=O)[O-])Cn2ccnc2)N3CCCC3 HTS08811 CCOC(=O)c1cc(nc(c1C#N)S)C(C)(C)C RF01037 c1ccc(cc1)c2csc(n2)c3ccc(cc3)c4csnn4 HTS10087 Cc1cc(nn1c2cc(ccc2Cl)Cl)C(=O)ONC(=O)c3ccco3 RF01039 c1ccc(cc1)CSc2nc(cn2CC(=O)c3ccccc3)c4ccccc4 HTS10101 Cc1c(nc(s1)c2ccc(cc2)c3csnn3)c4ccccc4 HTS10089 CS(=O)(=O)c1ccc(cc1)c2csc(n2)c3ccc(cc3)c4csnn4 HTS10090 Cc1cc2c(cccc2NC(=O)Nc3ccc(cc3)C(C)(C)C)nn1 HTS09569 Cc1cc2c(cccc2NS(=O)(=O)c3ccc(cc3)F)nn1 HTS10063 c1ccc(c(c1)C(=O)NC(=O)c2ccoc2)O HTS10442 CC(C)(CC(=O)Nc1ccc(c(c1)OC)OC)CC(=O)O HTS09617 COc1cc(ccc1O)/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09787 c1ccc(cc1)CNC(=O)C2CC(=NO2)c3ccc(cc3)Cl HTS11436 Cn1c2c(nc1N3CCCC3)n(c(=O)n(c2=O)C)C HTS11439 c1cc(ccc1[N+](=O)[O-])OCC2CC(=NO2)c3ccc(cc3Cl)Cl HTS11447 CC(C)S(=O)(=O)c1csc(c1NC(=O)c2ccc(cc2)C(F)(F)F)C(=O)OC KM02050 c1cc(ccc1S(=O)(=O)CC(=O)NOC(=O)c2cc(cc(c2)Cl)Cl)Cl KM02130 c1cc(cc(c1)C(=O)NC(=O)Nc2cccc(c2)Cl)CS(=O)(=O)c3ccc(cc3)Cl KM02359 Cc1c(c(c(c(c1C)C)C(=O)C2CCN(CC2)C(=O)NC)C)C CD10721 CCN(Cc1cc(cc(c1)OC)OC)C(=O)c2c(ccnc2OC)C(F)(F)F RF04672 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccc4c(c3)nccn4 HTS08964 c1ccnc(c1)CCNC(=O)c2ccc3c(c2)nccn3 HTS09584 Cc1cc2c(cccc2NC(=O)Nc3ccccc3)nn1 HTS09568 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5ccccc5C(=O)O HTS09181 CC(=O)Nc1ccc(cc1)NS(=O)(=O)c2ccccc2 HTS08953 c1cc(c(c(c1)F)C#N)NC(=O)COCC(=O)O HTS09362 c1ccc(cc1)CN2CCN(CC2)c3c[nH]c(=O)[nH]c3=O HTS09782 CCOC(=O)c1cnc2c(c1Oc3ccccc3F)c(nn2C)C KM05103 CCOc1ccccc1/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09792 c1ccc(c(c1)COn2c3ccccc3nn2)COn4c5ccccc5nn4 HTS09833 c1ccc(cc1)Cn2cncc2CO HTS09270 Cc1c(c(no1)c2ccccc2)c3nnc(o3)Cc4cccc(c4)OC HTS11284 Cn1c(cc(n1)C2CC2)NC(=O)COc3ccc(cc3Cl)Cl HTS09571 Cc1ccc(cc1C)C(=O)Nc2ccc3c(c2)OCCO3 HTS11314 c1ccc(cc1)S(=O)(=O)Nc2ccc(cn2)C(F)(F)F HTS11348 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C(/c3ccc(s3)[N+](=O)[O-])\N RF02345 Cn1c(cc(n1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)C(F)(F)F HTS10211 c1cc(oc1)C(=O)Oc2ccc(cc2)/C=N/Nc3nc4c(ncnc4n3[C@@H]5[C@H]([C@H]([C@@H](O5)CO)O)O)N HTS09793 c1cc(sc1)/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09795 CN(CCN(C)c1nc(cs1)c2ccc(cc2)Cl)c3nc(cs3)c4ccc(cc4)Cl HTS10383 c1ccnc(c1)c2ccc(s2)SCc3ccc(cc3)Cl KM02368 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CC4(CCCC4)CC(=O)O HTS09493 CCOC(=O)c1cnn(c1N)C(=O)c2ccc(cc2)n3c(ccc3C)C HTS11291 c1ccc(cc1)c2ccc(s2)NC(=O)OCc3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F HTS10529 COCCNC(=O)c1cc2ccccc2oc1=O HTS11451 c1ccc(c(c1)/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N)OCc5ccc(cc5)[N+](=O)[O-] HTS11450 COc1ccc(cc1OC)NC(=O)c2c(nccn2)C(=O)O HTS09620 c1cc(sc1)c2nnn(n2)CC(=O)NN SPB02314 COc1ccc(cc1)c2c(snn2)N MO00323 Cn1c(cnc1SCc2ccc(cc2)Cl)c3ccc(cc3)Cl TG00112 Cc1cc(c(c(c1)C)n2c(nnc2SCc3nc(no3)COc4ccc(cc4)[N+](=O)[O-])O)C HTS09604 c1cc(ccc1C#N)Oc2c(cc(cn2)C(F)(F)F)Cl SPB02967 c1ccc(c(c1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl)Cl SPB02954 Cn1c(cc(n1)c2ccccc2)NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS10224 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)N3CCCCC3)C#N HTS11251 Cc1cc(nc(n1)Sc2ccccc2NC(=O)Nc3ccc(cc3)OC(F)(F)F)C(=O)OC SPB06399 c1ccc(cc1)N2CCN(CC2)c3nc(cs3)c4ccc(cc4)Cl HTS10385 COc1cccc(c1)C(=O)n2ccc(n2)c3cccs3 HTS09516 COc1ccc(cc1OC)C(=O)n2ccc(n2)c3cccs3 HTS09520 Cc1cc(c(c(c1)C)n2c(nnc2SCC(=O)c3ccc(cc3)C#N)O)C HTS09605 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)CCCC(=O)O HTS09767 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)COCC(=O)O HTS09769 COc1cccc(c1)Cc2nnc(n2c3ccc(cc3)Cl)S HTS11294 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(nn2C)c3ccccc3 HTS10221 c1cc(ccc1NS(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F)N4CCCCC4 HTS09304 Cc1ccc(cc1)c2ccc-3c4ccccc4c(c3o2)C(=O)C(F)(F)F HTS10378 CCc1ccc(cc1)C(=O)c2cnc3ccccc3c2c4ccccc4 HTS10390 COc1ccc(cc1)C(=O)c2cnc3ccccc3c2c4ccccc4 HTS10391 CCNc1c2c3c(sc2[nH]c(=S)n1)CC(CC3)C HTS10264 c1cc(sc1)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)[N+](=O)[O-] HTS10273 Cc1cc(no1)C(=O)NNC(=O)c2cccc(c2)C(F)(F)F SPB03155 Cc1c(c(no1)C(=O)NN)c2csc(n2)COc3ccc(cc3)Cl SPB04403 c1ccc2c(c1)C(=O)N(S2(=O)=O)CCS(=O)(=O)c3ccc(cc3Cl)Cl HTS09649 Cc1c(c(no1)C(=O)NN)c2csc(n2)COc3ccccc3 SPB04404 Cc1cc(no1)C(=O)Nc2ccc3c(c2)OCCO3 HTS11319 Cc1cc(no1)c2c(c(nn2c3ccccc3)C)C(=O)O SPB05093 c1ccn(c1)c2cccc(c2)c3nc(on3)C(=O)NNC(=O)C(Cl)(Cl)Cl SPB01598 c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccc(cc4)Cl KM09691 CS(=O)c1ccccc1n2c3c(c(=O)n(c2=O)Cc4ccccc4F)[nH]cn3 KM09733 c1ccc2c(c1)c(ccn2)/C=N/Nc3nc4c(ncnc4n3[C@@H]5[C@H]([C@H]([C@@H](O5)CO)O)O)N HTS09796 c1cc(c(c(c1)Cl)/C=N/OCc2c(cc(cn2)C(F)(F)F)Cl)Cl HC00036 Cc1cc(nc(n1)SCn2c3ccccc3sc2=S)C HTS10376 c1cc(ccc1COc2ccc(cc2Cl)C#N)C(F)(F)F SPB01996 Cc1ccc(cc1Cl)N/C=C\C(=O)c2ccc(c(c2)Cl)Cl HTS10393 COc1ccc(cc1)N2C(=O)C3C(C2=O)N(N=C3c4ccc(cc4Cl)Cl)c5ccc(cc5)[N+](=O)[O-] HTS09107 c1cc(ccc1c2csc(n2)N3CCN(CC3)c4ccc(cc4)F)Cl HTS10384 CCCc1c(cnn1c2ccccc2)C(=O)Nc3ccc(cc3)N4CCCCC4 HTS09311 C1CCCN(CC1)c2nc3c(=O)[nH]c(nc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09824 CN(C)/C=C/C(=O)c1csc(n1)c2ccc(cc2)C(F)(F)F SPB04599 COC(CNC(=O)Nc1ccccc1)OC SPB01567 CC(C)(C)c1cc(no1)N/C=C/c2nnnn2c3ccc(cc3)Br HTS10396 Cn1c2c(c(=O)n(c1=O)C)nc([nH]2)N3CCN(CC3)Cc4ccccc4 HTS09800 c1cc(ccc1C(=O)O/N=C(/c2c(c[nH]n2)Br)\N)Cl SPB02861 Cn1c(cc(n1)c2ccccc2)NC(=O)c3ccccc3 HTS09750 Cc1cc(no1)c2c(c(nn2c3ccc(c(c3)Cl)F)C)C(=O)OC SPB03296 Cc1cc2c(cccc2NS(=O)(=O)c3cn(cn3)C)nn1 HTS10061 c1ccc(cc1)CC2c3ccccc3NC2=O HTS10084 CCOC(=O)CNc1cc(ccc1C)S(=O)(=O)N(C)C HTS10649 CN1CCN(CC1)C(=O)c2ccc(cc2)C(=O)N3CCN(CC3)C HTS10639 Cc1c(c(nc(n1)c2csc(n2)C)O)Cl SPB03572 CN(C)C(=O)O/N=C(/c1ccc(cc1)OCc2ccccc2F)\N SPB01470 CN(C)/C=N/NC(=O)c1cc(c(c(c1)Cl)OCc2cccc(c2)Cl)Cl SPB01479 CN(C)/C=N/NC(=O)c1cc(c(c(c1)Cl)OCc2ccc(cc2)F)Cl SPB01480 Cc1ccc(cc1)/C(=C/C=C(C#N)C#N)/N2CCN(CC2)c3ccc(cc3)Cl HTS10399 Cc1ccc(cc1)/C(=C/C=C(C#N)C#N)/N2CCN(CC2)c3ccc(c(c3)Cl)Cl HTS10400 COc1ccc(cc1)c2c(nco2)C(=O)O MO00452 c1cc2c(cc1[N+](=O)[O-])S(=O)(=O)CC2SCC(=O)NN KM08289 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)c2cc(cnc2)C#Cc3ccccc3 KM08462 Cc1c(c(c(c(c1C)C)C(=O)c2c(onc2c3c(cccc3Cl)Cl)C)C)C CD08661 Cc1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)C(=O)Nc4ccccc4)c5ccccc5)c6ccccc6 HTS09283 CCOC(=O)C1=NN(C2(S1)N(C(=O)/C(=C\c3ccccc3)/S2)c4ccccc4)c5ccccc5 HTS09286 Cc1c(c(nn1c2ccccc2)C3C(C(=NN3c4ccccc4)c5ccccc5)c6ccccc6)C(=O)C HTS09272 c1ccc(cc1)n2cc(c(n2)/C=N/NC(=O)CSc3c4c5c(sc4ncn3)CCCC5)c6ccc(cc6)Cl HTS10369 CCOC(=O)c1cnn(c1N)C(=O)c2cccc3c2cccc3 HTS09777 Cc1c(c(no1)c2ccccc2)CN3C(=O)c4ccccc4S3(=O)=O HTS09659 CCOC(=O)/C(=C/C=C(/c1ccc(cc1)Cl)\N2CCOCC2)/C#N HTS10397 c1ccc(cc1)CSc2nc(cs2)c3ccc(cc3)Cl TG00047 c1cc(ccc1CSc2nc(cs2)c3ccc(cc3)Cl)Cl TG00048 c1cc2c(cc1Cl)c(c(s2)Cl)CC(=S)N MWP00305 Cc1c(cnn1c2ccccc2)C(=O)NNC(=O)Cc3cccc(c3)OC HTS10677 CCn1cnc2c1c(=O)[nH]c(n2)N HTS11456 CN(C)c1nc2c(ncnc2n1[C@@H]3[C@H]([C@H]([C@@H](O3)CO)O)O)N HTS11458 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N3CCC(CC3)C(=O)N)Cc4ccccc4Cl HTS11465 c1ccc2c(c1)C(C(=O)N2)C(C[N+](=O)[O-])c3ccccn3 HTS10085 c1cc(cc(c1)S(=O)(=O)N2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F)F HTS10239 CCOC(=O)N1CCC(CC1)NC(=O)c2c(nns2)C HTS10615 c1c(cc(cc1Cl)Cl)NC(=O)C23CC4CC(C2)CC(C4)C3 CD08934 c1ccc(c(c1)C(=O)NCC(=O)c2ccc(cc2)Cl)C(F)(F)F SPB01756 CCCCOc1nc2c(n1Cc3ccc(cc3)Br)c(=O)n(c(=O)n2C)C HTS09805 COc1ccc(cc1)OC(=O)Nc2csc(n2)Cc3ccsc3 MWP00462 Cc1c2cc(ccc2sc1c3ccnc(n3)NC(=O)c4ccc(cc4)Cl)Cl MWP00782 c1ccc(cc1)c2c(nco2)C(=O)Nc3ccc4c(c3)OCCO4 HTS11318 c1cc2c(cc1NC(=O)c3ccoc3)OCCO2 HTS11315 c1cc(c2c(c1)OCC2)c3nc(cs3)C(=O)Nc4ccc5c(c4)OCCO5 HTS11313 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccccc2 HTS10604 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2ccc(c(c2)Cl)C HTS10609 CCOC(=O)N1CCC(CC1)NC(=O)c2cc(on2)C HTS10614 COc1ccc(cc1)C2=NOC(C2)COC(=O)c3ccc(cc3)I HTS11467 Cc1c2c(cc(s2)C(C)(C)C)sc1C(=O)Nc3ccc(cc3)OC(F)(F)F GK01923 C/C(=N\O)/C(C)(C)NCCc1c[nH]c2c1cccc2 HTS10438 CC(=O)Nc1ccc(cc1)NC(=O)COc2ccc(cc2Cl)Cl HTS08970 CC(C)(C)c1ccc(cc1)NC(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS09205 Cc1cnc(c(c1OC)C)CO KM07183 C/N=C\1/N(C(=O)C(S1)CC(=O)O)C MO00336 Cc1ccccc1C(=O)Nc2nc([nH]n2)SCc3ccc(cc3)Cl HTS10137 c1cc(ccc1OC(F)(F)F)S(=O)(=O)NN SPB03408 c1ccc(cc1)NC(=S)N2CCCCC2c3cccnc3 HTS09801 c1cc(ccc1c2nnc(o2)c3ccc4c(c3)OCO4)C(F)(F)F HTS09773 CS(=N/C=C(\C#N)/C(=O)c1ccc(cc1)Cl)(=O)c2ccsc2 KM05876 CNC(=S)NNC(=O)CSCc1nc(cs1)c2ccccc2 KM05925 Cn1c2c(nc1N/N=C/c3ccc(cc3)OCC=C)n(c(=O)n(c2=O)C)C HTS09820 C/C(=C\C(=O)O)/C(=O)NNc1ccsc1C(=O)OC GK02693 CN(C)/N=C/c1ccc(cc1)[N+](=O)[O-] HC00001 Cc1ccc(cc1)S(=NC(=O)NC(=O)c2c(cccc2Cl)Cl)(=O)C KM02951 Cc1ccc(n1c2c(cccn2)OCc3nnc(o3)c4ccc5ccccc5c4)C HTS08816 Cc1c(sc(n1)c2ccc3c(c2)OCC3)C(=O)Nc4ccc(cc4)N5CCCCC5 HTS09310 COc1cccc(c1OCc2c(cccc2Cl)Cl)CC3CC(=NO3)c4ccccc4 HTS09822 Cc1cc(c(n1C2CC2)C)C(=O)O CC25301 Cc1[nH]cc(n1)S(=O)(=O)Nc2cc(nn2C)c3ccccc3 HTS10212 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)Nc4ccc(cc4)F HTS09486 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc3c(c2)CCO3 HTS10553 CCOC(=O)c1c(nc(s1)SC)N GK00772 Cn1c2c(c(=O)n3c1ncn3)CCCC2 HTS10497 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N3CCOCC3)Cc4cccc(c4)F HTS09812 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCCOCCO)Cc3c(cccc3Cl)Cl HTS09815 c1cc(oc1)Cn2c(nnc2S)c3ccc(cc3)C(F)(F)F HTS09752 c1ccc(c(c1)C(=O)NC(=O)c2ccc(cc2F)F)O HTS10464 c1ccc(cc1)NC(=O)NCC2CC2 HTS10469 Cc1cccc(c1)NC(=O)NCC2CC2 HTS10501 COc1ccc(cc1OC)c2nc(=O)c3ccccc3o2 HTS10551 Cn1c2c(nc1N/N=C\3/c4ccc(cc4NC3=O)Br)n(c(=O)n(c2=O)C)C HTS09839 Cc1cc(cc(c1)NC(=O)Nc2cc(nn2C)c3ccccc3)C HTS10226 Cc1cc(no1)C(=O)N(C)C2CCCCC2 HTS08832 Cc1cc(cc(c1)NC(=O)N(C)Cc2ccccc2)C HTS08844 c1[nH]c(=O)c2c(n1)n(cn2)COCCO HTS11460 CNc1nc2c(ncnc2n1[C@@H]3[C@H]([C@H]([C@@H](O3)CO)O)O)N HTS11461 c1ccc(cc1)N2CCN(CC2)c3nc4c(=O)[nH]c(nc4n3[C@@H]5[C@H]([C@H]([C@@H](O5)CO)O)O)N HTS09840 c1cc(cnc1)C2N(C(=O)CS2)CCN3C(SCC3=O)c4cccnc4 PD00257 Cn1c2c(c(=O)n(c1=O)C)n(cn2)Cc3nnc(o3)c4ccccc4 HTS11463 c1ccc2c(c1)ccc(n2)C(=O)OCc3ccc(cc3Cl)Cl HTS11464 c1ccc(c(c1)CC2CC(=NO2)c3ccc(cc3)Cl)OCc4c(cccc4Cl)Cl HTS11466 c1c(cc(cc1Cl)Cl)n2c(c(nn2)C#N)N RF01075 CNC(=O)Nc1ccc(cc1)C2CC2(Cl)Cl RF02121 COc1ccc(cc1)NC(=O)c2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS11020 CCOC(=O)c1nnc(o1)c2ccc(cc2)C(F)(F)F HTS11301 c1ccc(cc1)Oc2ccc(cn2)N CC19614 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C/c3ccc(cc3)O)Cc4c(cccc4Cl)Cl HTS11431 CC(=O)Nc1ccc(cc1)NS(=O)(=O)c2ccc(c(c2)Cl)F HTS08944 CC(=O)Nc1ccc(cc1)NS(=O)(=O)c2cc(sc2Cl)Cl HTS08955 c1cc(c(cc1S(=O)(=O)Nc2cc(cc(c2)NS(=O)(=O)c3ccc(c(c3)Cl)Cl)C(F)(F)F)Cl)Cl CD10923 c1ccc2c(c1)OCC(O2)CNC(=O)CSCC(=O)O HTS10159 c1ccc(c(c1)C2=NCCCN2S(=O)(=O)c3ccc(c(c3)Cl)Cl)SCc4c(cccc4Cl)F CD07470 c1ccc(c(c1)C(F)(F)F)NC(=O)N/C=C/c2ccsc2 GK00861 CC(C)(C)c1ccccc1NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS10531 c1cc(oc1)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)Cl HTS10272 C/C(=N\O)/C(C)(C)Nc1ccc(cc1)C(C)(C)C HTS11312 Cn1c2c(c(=O)[nH]c1=O)n(cn2)CCN(Cc3ccccc3)Cc4ccccc4 HTS09834 Cc1cc(=O)oc2c1ccc(c2)OCC3CC(=NO3)c4ccccc4 HTS11475 c1[nH]c(=O)c2c(n1)n(cn2)[C@@H]3C[C@H]([C@@H](O3)CO)O HTS11476 Cc1cc2c(cccc2NC(=O)COCC(=O)O)nn1 HTS09555 Cc1nc(cs1)c2ccnc(n2)S SPB03876 c1cc(ccc1C(=O)N2CCCCCC2)C(=O)N3CCCCCC3 HTS10641 c1ccc2c(c1)OCC(O2)CNC(=O)CCC(=O)O HTS10155 CC(=O)N1CCSC1C(=O)NN(C(=O)c2cc3ccccc3s2)C(=O)c4cc5ccccc5s4 HTS11309 Cn1c2c(nc1N3CCN(CC3)c4ccccn4)n(c(=O)n(c2=O)Cc5ccc(cc5)Cl)C HTS11443 Cn1c2c(nc1Oc3ccccc3Br)n(c(=O)n(c2=O)C)C HTS11446 Cc1c(snn1)c2nnc(n2C3CC3)S MO00089 CCn1cc(c(=O)c2c1ccc(c2)Cl)C(=O)Nc3ccc(cc3)C(F)(F)F DFP00357 c1ccc(cc1)CNC(=O)CN2C(=O)c3ccccc3S2(=O)=O HTS09540 CC(C)(C)c1ccc(cc1)NC(=O)Nc2cc(nn2C)c3ccccc3 HTS10225 c1cc(c(c(c1)C#N)Oc2ccc(cc2)S(=O)(=O)N3CCC(CC3)C(=O)N)C#N HTS11252 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N3CCCCCC3)Cc4ccccc4Cl HTS11441 c1cc(cnc1)/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09788 c1ccnc(c1)Oc2cccc3c2nccc3 HTS11444 CC(=O)N1CCSC1C(=O)NNC(=O)c2ccc3c(c2)OCO3 HTS11308 c1cc(oc1)Cn2c(nnc2SCC(=O)c3ccc(cc3)F)O HTS09146 c1ccc(c(c1)C(=O)Nc2ccc(cc2)OC(F)F)C(=O)O HTS09558 c1ccc2c(c1)cccc2c3nnc(n3c4cccnc4)S HTS11302 c1ccc(cc1)n2c(nnc2SCC(=O)N3c4ccccc4Sc5c3cccc5)c6ccncc6 HTS10266 Cc1cc(c(c(c1)C)n2c(nnc2SCC(=O)c3ccc(cc3)OC)O)C HTS09602 c1cc(ccc1/C=N/Nc2nc3c(s2)cc(cc3Cl)Cl)Cl RF02711 CC(C)(C)c1ccc(cc1)NC(=O)CN2C(=O)c3ccccc3S2(=O)=O HTS09641 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccccc3C(F)(F)F HTS09642 c1cc(cc(c1)Cl)n2cc(c(=O)c(n2)C(=O)NN)Sc3ccc(cc3)Cl SPB04059 Cn1c(cc(n1)c2ccccc2)NS(=O)(=O)c3ccccc3 HTS10222 c1c(cnc(c1C(F)(F)F)S)C(F)(F)F SPB04490 Cc1cc(nc(n1)c2csc(n2)C)NC SPB04569 CCOC(=O)c1c(sc(n1)C)C(=O)/C=C/N(C)C SPB04594 COc1ccc(cc1)n2c(nnn2)c3cnn(c3C(F)(F)F)c4cccc(c4)F HTS10381 c1ccc(cc1)c2c3c(nc4c2sc5c4c6c(s5)c(c7c(n6)CCC7)c8ccccc8)CCC3 HR00147 c1ccc(cc1)NC(=O)CN2C(=O)c3ccccc3S2(=O)=O HTS09632 c1cc(c(c(c1)Cl)Cc2nc(cs2)NC(=O)Nc3ccc(c(c3)Cl)Br)Cl SPB02021 c1ccc(cc1)c2c(sc(n2)Nc3ccc(cc3)F)C(=O)c4ccc(cc4)F HTS10132 CN(C)c1ccc(cc1)Nc2nc(c(s2)C(=O)c3ccc(cc3)F)c4ccccc4 HTS10135 c1cc(c(c(c1)F)C#N)NC(=O)CSCC(=O)O HTS09360 Cc1cc(no1)C(=O)Nc2ccc(cc2)F SPB03611 COC(=O)c1ccc(o1)Oc2ccc(cc2)C3SCCS3 HTS11401 c1ccc2c(c1)n(c(=S)s2)CSc3nccc(n3)C(F)(F)F HTS10377 COc1ccc(cc1)C2=NOC(C2)CN3C(=O)c4ccccc4S3(=O)=O HTS11448 Cc1c(nc(nc1O)C(F)(F)F)C SPB04772 CS(=NC(=O)c1cc2ccccc2o1)(=O)c3ccc(cc3)Cl KM05489 c1cc(ccc1c2cnc(o2)S)Cl SPB02670 Cc1cc(c(c(c1)C)n2c(nnc2SCC(=O)Nc3ccccc3Cl)O)C HTS09606 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccc(cc3C(=O)c4ccccc4Cl)Cl HTS09636 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccc(cc3)Cl HTS09638 Cn1c(cc(n1)c2ccccc2)NC(=O)CN3C(=O)c4ccccc4S3(=O)=O HTS09650 c1ccc(cc1)c2[nH]nc(n2)c3cccc(c3)Cl HTS11300 COC(=O)C1Cc2c3ccccc3[nH]c2C(N1)c4ccc(cc4)Cl HTS11304 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)S SPB05134 c1ccc(cc1)c2c3ccccc3ncc2C(=O)c4ccc(cc4)Cl HTS10392 CC(C)(C)c1cc(no1)N/C=C/c2nnnn2c3ccc(cc3)Cl HTS10394 CC(C)n1c2ccc(cc2nc1SCc3ccc(cc3)Cl)C(F)(F)F TG00032 c1ccc-2c(c1)NC(c3n2ccc3)c4ccc(cc4)Cl HR00249 COc1ccc(cc1OC)S(=O)(=O)NC2CCc3c2cccc3 KM09259 c1cc(c(cc1[N+](=O)[O-])Cl)CSc2ccc(cc2F)F SPB01603 Cc1cc(c2c(c(sc2n1)C#N)N)C(F)(F)F SB02114 c1c(nc2nc(nn2c1C(F)(F)F)S)C(F)(F)F SPB02095 c1cc(ccc1c2csc(n2)c3cnn4c3nc(cc4C(F)(F)F)C(F)(F)F)Cl KM05256 Cc1ccc(cc1)S(=O)(=O)Nc2cc(nn2C)c3ccccc3 HTS10215 c1cnc(nc1)Sc2c[nH]c(=S)nc2c3ccc(cc3)Cl SPB04189 CCOc1ncc(c(n1)c2cccc(c2)Cl)c3nnnn3c4ccc(cc4)C HTS10387 c1cc(ccc1c2c(cnc(n2)N)c3nnnn3c4ccc(cc4)Cl)F HTS10389 COc1cc(nc(n1)SC)OC SPB07200 c1cnc(cn1)c2nnc(s2)S SPB07295 CCOC(=O)/C(=C/C=C(/c1ccc(cc1)Cl)\N2CCSCC2)/C#N HTS10398 CC1CN(CC(O1)C)c2[nH]c3c(n2)c(=O)n(c(=O)n3C)C HTS09799 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C(=N/OC(=O)c3csc(n3)C)/N SPB02779 CNC(=O)NNC(=O)c1csc(n1)Cc2c3cc(ccc3sc2Cl)Cl MWP00310 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS09664 Cc1cc(no1)C(=O)Nc2cccc(c2)Cl SPB03089 c1ccc(cc1)C(=O)NNC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl SPB03105 CC1CC(=O)Nc2ccccc2N1C(=O)c3ccc(cc3)C(C)(C)C HTS09699 c1ccc(cc1)NC(=O)O/N=C(/c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3F)F)\N SPB01980 Cc1ccnc(n1)SCn2c3ccccc3sc2=S HTS09299 c1cnc(nc1)N2CCN(CC2)C(=O)CC3(CCCC3)CC(=O)O HTS10165 CC(C)N(Cc1ccccc1)C(=O)c2ccc3c(c2)nsn3 HTS08830 Cc1c(c(no1)c2ccccc2)NC(=O)N(C)C3CCCCC3 HTS08836 Cn1cc(nc1)S(=O)(=O)N(C)Cc2ccccc2 HTS08843 COc1cccc(c1)NC(=O)N2CCN(CC2)C(=O)C3CCCO3 HTS10767 c1cc(cc(c1)F)n2c(c(cn2)c3nnnn3c4ccc(cc4)F)C(F)(F)F HTS10380 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)n3ccc(n3)c4cccs4 HTS09531 CC(C)(C)c1ccc(cc1)C2=NNC(=NN2)SCC(=O)c3ccc(cc3)Cl HTS06861 CC(C)(C)C(=O)OCc1nc(cs1)c2ccc(c(c2)O)O HTS10114 Cc1cc(on1)c2ccccc2C(=O)NC3CCCCC3 HTS09826 Cn1c2c(nc1Oc3ccc4c(c3)OCO4)n(c(=O)n(c2=O)Cc5ccc(cc5)F)C HTS09807 c1cc(ccc1CSc2nccc(n2)/C=N/O)Cl SPB04299 Cc1c(c(on1)C)S(=O)(=O)N2CCN(CC2)C(=O)C3COc4ccccc4O3 HTS08799 c1ccc2c(c1)[nH]c(=O)c(n2)c3ccc(cc3)Cl HTS10976 c1c(cc(c2c1sc(n2)S)Cl)Cl SPB01267 Cc1ccccc1n2c(cc(=O)n(c2=O)Cc3ccccc3SC)N KM09769 Cc1ccccc1n2c(cc(=O)n(c2=O)Cc3ccccc3[N+](=O)[O-])N KM09867 c1cc(sc1)C(=O)N2CCN(CC2)CC(=O)N3CCCC3 HTS10777 CN(C(=S)SCc1c(cccc1Cl)F)/N=C/c2cc(cc(c2O)Cl)Cl CD07766 Cc1ccc(cc1F)NC(=O)C2=NNC(=O)CC2 HTS09714 CC1CC(=O)Nc2ccccc2N1C(=O)CN3CCN(CC3)c4ccccn4 HTS09720 CC1CC(=O)Nc2ccccc2N1C(=O)c3cc(sc3Cl)Cl HTS09700 Cc1nc(nc(n1)N/N=C/c2ccccn2)N RF02944 c1cc2c(cc1C(=O)Nc3ccc4c(c3)OCCO4)OCO2 HTS10419 CC(=O)Nc1ccc(cc1)OCc2ccc(o2)C(=O)OC HTS09263 Cc1ccc(cc1)N2C(=C3C(=O)c4ccccc4C3=O)SC(=N2)C(=O)c5cccs5 HTS09119 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COCc3ccccc3)OCc4ccccc4 HTS09803 Cc1ccc(cc1NC(=O)NCc2ccccc2)OC KM09926 COc1cc2c(cc1OC)C(=NCC2)c3cccc(c3)Cl MB00254 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)Nc3ccccc3 HTS08248 COC(=O)c1cccc(c1)NC(=O)CC2C(=O)NCCN2C(=O)c3c(c4ccccc4s3)Cl HTS08866 c1ccc(c(c1)CN2c3ccccc3Sc4c2cccc4)CN5c6ccccc6Sc7c5cccc7 HTS09832 Cc1c(c(n(n1)C)COC(=O)Nc2ccc(cc2)Cl)[N+](=O)[O-] SPB01736 Cc1c(snn1)C(=O)Nc2cc(nn2C)c3ccccc3 HTS09746 Cn1c(cc(n1)c2ccccc2)NC(=O)c3c(c4ccccc4s3)Cl HTS09748 Cc1cccc(c1)C(=O)/C=C\Nc2ccc(cn2)Cl HTS10401 CCc1ccc(cc1)C(=O)/C=C\Nc2ccc(cn2)Cl HTS10402 Cc1ccc2c(c1)c(c[nH]2)c3nnnn3c4ccc(cc4)OC HTS10404 CC(C)CNC(=O)c1cnn2c1nc(cc2C(F)(F)F)C(F)(F)F KM06152 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccc(cc3)N4CCCCC4 HTS09312 c1c(ccc(c1)c2scc(n2)C34C[C@H]5C[C@@H](C3)C[C@@H](C4)C5)c6nnsc6 HTS10088 c1cc(ccc1n2c3c(cc(cn3)C(F)(F)F)nc2S)Cl SPB04406 c1cc(cc(c1)C(=O)N)CS(=O)(=O)c2ccc(cc2)Cl KM02286 Cc1c2c(c(cnc2n(n1)C)NC(=O)Nc3ccc(cc3)C(F)(F)F)Cl KM02357 Cc1c2cc(sc2n(n1)C)C(=O)NN GK02347 c1ccnc(c1)c2ccc(s2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F KM02484 CCCc1c(cn(n1)C)C(=O)NCC(=O)OCC GK02183 Cc1cccc(c1NC(=O)N(Cc2ccccc2)C(=O)CC#N)C KM09937 Cn1c2c(nc1N/N=C/c3ccc(c(c3)OC)O)n(c(=O)n(c2=O)Cc4ccccc4)C HTS09818 c1cc(ccc1c2nnc(o2)c3ccc4c(c3)nsn4)C(F)(F)F HTS09774 CCOC(=O)c1c(c(on1)C)c2csc(n2)c3cccc(c3)Cl SPB03328 COc1ccc(cc1OC)N2C(=O)CSCC2=O HTS10123 COc1ccc(cc1OC2CCCC2)C(=O)NNS(=O)(=O)c3cccs3 HTS10096 COc1ccc(cc1OC2CCCC2)C(=O)NNS(=O)(=O)c3ccc(s3)CNC(=O)c4ccc(cc4)Cl HTS10099 c1ccc2c(c1)c3c([nH]2)C4(CCNCC4)NCC3 HTS09269 COc1cccc(c1)NC(=O)Nc2cc(sc2C(=O)OC)c3ccc(cc3)Cl HTS09385 c1cc(cc(c1)/C(=N/O)/N)CS(=O)(=O)c2cccs2 KM02378 Cc1cc(c(cc1NC(=O)c2ccccc2)OC)NC(=O)COc3ccc(cc3Cl)Cl HTS08969 Cc1ccc(cc1)NC(=O)NNC(=O)Cn2c(cc(=O)n3c2ncn3)C HTS09921 c1ccc(cc1)COc2ccc(cc2)/C=N/Nc3cc(nc4n3ncn4)c5ccccc5 HTS09922 CCc1cc(c(s1)NC(=O)CSCC(=O)O)C(=O)c2ccc(cc2)OC HTS09244 CC(C)(CC(=O)NC1CCN(CC1)Cc2ccccc2)Sc3ccc(cc3)Cl HTS09666 CC(C)(CC(=O)N1CCN(CC1)c2c(cccn2)C(F)(F)F)Sc3ccc(cc3)Cl HTS09667 c1ccc2c(c1)OCC(O2)CN3CCS(=O)(=O)CC3 HTS10161 c1ccc(c(c1)C(=O)NC(=O)c2ccc3c(c2)CCO3)O HTS10445 c1ccc(cc1)c2c(sc(n2)Nc3ccccc3)C(=O)c4ccc5c(c4)OCCCO5 HTS09467 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CCCC(=O)O HTS09492 c1cc(sc1C#N)c2ccnc(n2)S KM04307 c1ccc(c(c1)C(=O)/C(=C/Nc2ccc(cc2)Cl)/C#N)OC(F)(F)F KM04812 c1ccc2c(c1)C(=O)C(CS2)/C(=N/O)/N MBE00274 CS(=NC(=O)c1cnn2c1nc(cc2C(F)(F)F)C(F)(F)F)(=O)C KM05676 Cc1c(sc(n1)c2ccccc2)C(=O)NC(=O)c3ccccc3O HTS10441 Cn1cc(c(n1)C(F)(F)F)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F GK00789 CCOC(=O)c1cn(nc1C(F)(F)F)CC(=O)NN GK00851 COc1cc(c(cc1NC(=O)C(c2ccccc2)Sc3ccccc3N)Cl)OC RF00260 C/C(=N\OC(=O)Nc1cc(n(n1)c2ccccc2)C(C)(C)C)/C(C)(C)C RF01186 CN(C)/C=N/c1c(nnn1c2cc(cc(c2)Cl)Cl)C#N RF01216 CN/N=C/c1c(cc(cn1)C(F)(F)F)Cl HC00069 CSc1nc(n(n1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)NC(=O)C(F)(F)F JM00015 CN(C)C(=O)Oc1ccnc(n1)SCc2ccc(cc2Cl)Cl JM00430 c1ccnc(c1)/C=N/NC(=O)C(=O)Nc2cccc(c2)C(F)(F)F JPV00101 Cc1ccc2c(c1)c(cs2)CC(=O)OC MWP00143 CCc1cccc(c1NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)CC RF00386 c1nc(nn1[C@@H]2[C@H]([C@H]([C@@H](O2)CO)O)O)C(=O)N HTS11462 Cn1c(cc(n1)c2ccccc2)NS(=O)(=O)c3ccc(c(c3)OC)OC HTS10217 Cn1c(cc(n1)c2ccccc2)NC(=O)Nc3ccc(cc3)OCc4ccccc4 HTS10223 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4ccc(cc4)F HTS09510 CCCSc1c(cccn1)C(=O)Nc2cc(no2)C HTS11346 Cc1csc2c1ncnc2NCCc3ccc(cc3)Cl GK01670 Cc1c(cnc(n1)N2CCSCC2)S(=O)(=O)c3ccc(cc3)Cl KM01324 Cc1csc2c1c(c(s2)/C(=N/O)/C)C KM03912 C/C(=N\Nc1nc2c(n1C)c(=O)n(c(=O)n2C)Cc3ccc(cc3Cl)Cl)/c4ccccc4 HTS11433 c1ccc(cc1)OC(=O)Nc2csc(n2)Cc3ccsc3 MWP00461 CCOC(=O)COc1c(c(cc(n1)C)C)C#N RF00474 c1cc(c(c(c1)F)NC(=O)Cc2ccc(cc2)[N+](=O)[O-])F RF00481 COC(=S)SC/C(=N\O)/c1ccc(cc1)[N+](=O)[O-] RF00515 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/OC(=O)c3ccccc3 RF00573 c1cc(ccc1CC(=O)c2ccc(cc2)O)Cl RF01468 c1cc(cc(c1)[N+](=O)[O-])/C=N/N=C\2/NC(=O)CS2 RF01532 CC1C(=O)N/C(=N/N=C/c2cccc(c2)[N+](=O)[O-])/S1 RF01533 c1cc(sc1)C(=O)/C(=N/Nc2cc(ccc2Cl)C(F)(F)F)/C(=O)C(F)(F)F RF00198 c1cc(ccc1Cn2ccnc2C(=O)c3ccc(c(c3)Cl)Cl)Cl JM00138 CNC(=O)NNC(=O)c1ccc(cc1)Cl JM00240 CC(C)(C)CN/C(=C(/C#N)\N=C\c1cc(c(c(c1)Br)O)OC)/C#N KM00306 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C/c3ccccc3OC)Cc4ccccc4Cl HTS11220 CCOC(=O)COc1ccc(cc1)/C=N/Nc2nc3c(n2C)c(=O)n(c(=O)n3C)Cc4ccc(cc4Cl)Cl HTS11432 COc1ccc(c(c1)C(=O)Nc2ccc(cc2)F)Br RF00417 CC(=O)NNC(=O)c1csc(n1)Cc2c3cc(ccc3sc2Cl)Cl MWP00308 Cc1c2ccccc2sc1/C=N/O MWP00783 c1cc2c(cc1C(F)(F)F)Nc3c(c(=O)c3=O)N2 MWP00863 CCOc1c(c(=O)c1=O)Nc2cccc(c2)Cl MWP00938 COc1ccc(cc1OC)NC(=O)CCC(=O)O HTS09621 c1cc2c(cc1C(=O)Nc3ccc4c(c3)OCCO4)nccn2 HTS11320 c1cc2c(cc1C(=O)Nc3ccc4c(c3)OCCO4)nsn2 HTS11316 CCCSc1c(cccn1)C(=O)Nc2cc(sc2C(=O)C)C(C)(C)C HTS11344 CCC1(CCCCNC1=O)c2cccc(c2)OC HTS10499 c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccccc3 SPB02931 CC(C)CNC(=O)C1CC(=NO1)c2ccccc2 HTS11435 c1cc(cc(c1)C(F)(F)F)c2cc([nH]n2)N KM09235 Cc1c(cccc1S(=O)C)n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)OC)[nH]cn3 KM10370 Cc1c(cccc1SC)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM10238 Cc1ccc(cc1)NC(=O)c2c(c3c(s2)cc(s3)C(C)(C)C)C GK01921 Cc1cc(nc2c1c3c(s2)c(ncn3)SCc4ccc(cc4)F)C HTS11502 c1cc(cnc1)CNCc2ccc(cc2)Cl.Cl HTS11486 c1cc(ccc1CN2CCOCC2)S(=O)(=O)N3CCOCC3 HTS11098 CNc1c(c(ncn1)SCCO)[N+](=O)[O-] KM07791 c1ccc(cc1)C2=NOC(C2)COC(=O)c3ccc(cc3)Cl HTS11438 Cn1c2c(nc1N3CCCCCC3)n(c(=O)n(c2=O)C)C HTS11440 Cn1c2c(nc1NC3CCCC3)n(c(=O)n(c2=O)C)C HTS11442 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)NCCc5cccs5 HTS09209 c1ccc(cc1)C(=O)Nc2cccc(c2C#N)F HTS09358 Cc1c(sc(n1)COc2ccccc2Cl)c3ccnc(n3)S SPB02607 c1ccc(cc1)CN(Cc2ccccc2)CC(=O)N3c4ccccc4Sc5c3cccc5 HTS10267 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/NC(=O)CN4c5ccccc5Sc6c4cccc6 HTS10268 c1cc(ccc1C(=O)N2CCCC2)C(=O)N3CCCC3 HTS10638 c1ccc(cc1)C(=O)c2c(nn(n2)c3ccc(cc3)Cl)N HTS11205 Cc1cc(no1)NC(=O)c2ccc(cc2)Cl SPB03062 Cc1c(c(nc(n1)SCC(=O)c2ccc(c(c2)F)F)O)Oc3ccc(cc3)Cl SPB03984 c1cc(oc1/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N)[N+](=O)[O-] HTS11449 c1ccc2c(c1)cc(c(=O)o2)C(=O)NCc3ccco3 HTS11452 c1cc(c(cc1/C=N/NC(=N)N)Cl)Cl SPB06189 Cc1cc(sc1)C(=O)Nc2ccc(cc2Cl)Cl GK01998 CCOC(=O)N1CCC(CC1)NC(=O)CCCC(=O)O HTS10802 c1ccc(cc1)/C=c\2/c(=O)n3c(=NC(=CC3c4cn(nc4c5ccccc5)c6ccccc6)c7ccccc7)s2 HTS11490 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)c3ccc(cc3)F HTS09657 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3Cl)NC(=O)C HTS09691 CC(C)(C)c1ccc(cc1)NC(=O)Nc2cc(ccc2N3CCCC3)C(F)(F)F HTS09340 CC(C)CNc1nc2c(ncnc2n1[C@@H]3[C@H]([C@H]([C@@H](O3)CO)O)O)N HTS11216 CCOC(=O)c1cc(n(n1)c2ccc(cc2)[N+](=O)[O-])C JM00383 c1cnccc1n2c3cc(c(cc3[nH]c2=O)Cl)Cl HTS11481 c1cc(c(cc1Cl)N)Nc2ccncc2 HTS11483 c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4cccc(c4)N KM09359 COc1cc2c(cc1OC)C(=O)N(CC2)Cc3cccc(c3)Cl GK02022 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)c4ccc5c(c4)OCCCO5 HTS09502 Cc1c2cc(ccc2sc1CC(=O)NC)Cl MWP00254 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NS(=O)(=O)c4ccc(cc4)C(F)(F)F HTS09507 c1ccc(cc1)C(=O)CN2C(=O)c3ccccc3S2(=O)=O HTS09644 c1ccc2c(c1)C(=O)N(S2(=O)=O)Cc3csc(n3)c4ccc(cc4)Cl HTS09645 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)c4ccco4 HTS09504 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)c4ccc(nc4C)C(F)(F)F HTS09505 Cc1csc2c1ncnc2N3CCN(CC3)C(=O)NC(C)(C)C GK02684 COc1ccc(cc1OC)C(=O)NC(=O)c2ccccc2O HTS10460 COc1ccc(cc1)C(=O)CSc2nnc(n2C3Cc4ccccc4C3)O HTS09612 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)CC(=O)c5ccc6c(c5)OCCCO6 HTS10659 COc1ccc(cc1OC2CCCC2)C(=O)NNS(=O)(=O)c3ccc(s3)c4ccccn4 HTS10100 c1ccc(c(c1)NC(=O)C2=NNC(=O)CC2)N3CCOCC3 HTS10249 Cc1ccc2cc(ccc2n1)NC(=O)c3cc(oc3C)c4ccccc4 HTS10584 c1cc(cc(c1)C#N)Cn2cc(ccc2=O)C(F)(F)F SPB06648 CCOC(=O)c1cnc(cc1O)O SPB07340 CCOC(=O)c1cc2c(ccnc2O)nc1C(F)(F)F HC00057 COC(=O)c1cn(cc(c1=O)F)Cc2ccc(cc2)Cl HC00062 c1cc(ccc1C#N)S(=O)(=O)N2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F HTS10236 Cc1c(c(on1)C)c2nc(no2)CN3C(=O)c4ccccc4S3(=O)=O HTS09655 COC(=O)c1cccc(c1)NC(=O)C2=NNC(=O)CC2 HTS10250 c1cc(sc1)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS10425 c1cc(ccc1C2c3ccsc3CCN2Cc4ccc5c(c4)CCO5)OC(F)(F)F HTS08549 Cc1c(c(no1)c2ccccc2)C(=O)N(Cc3ccccc3)C(C)C HTS08829 CCc1ccccc1NC(=O)c2cnccc2C(F)(F)F RF04519 c1cc(ccc1C(F)(F)F)NC(=O)c2cnccc2C(F)(F)F RF04527 Cc1c(c(c(o1)C)S(=O)(=O)N2CCCc3c2cccc3)C(=O)OC HTS10180 c1ccc2c(c1)CCCN2S(=O)(=O)c3cccc4c3nsn4 HTS10181 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(nn3C)c4ccccc4 HTS10202 Cn1c(cc(n1)c2ccccc2)NC(=O)C3CCCCC3 HTS10204 c1cc(cc(c1)Cl)NC(=O)NCC2CC2 HTS10466 c1c(cc(cc1F)F)NC(=O)C2=NNC(=O)CC2 HTS10254 Cc1c(c(nc(n1)c2ccc(cc2Cl)Cl)S)C(=O)C SPB05362 CCN(CC)c1ccc(cc1)CN2CCN(CC2)Cc3ccccc3 HTS10571 Cn1c2c(c(=O)n(c1=O)C)n(cn2)Cc3cc(ccc3Cl)OC HTS11470 CCCCNC(=O)c1cc(cc(c1)OCc2ccccc2Cl)OCc3ccccc3Cl HTS11474 C1CCN(C1)c2nc3c(=O)[nH]c(nc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS11477 Cn1c2c(cc(s2)C(=O)Nc3ccc(cc3)C(F)(F)F)c(n1)C(F)(F)F GK02686 CC(=O)Nc1ccc(cc1N)C(C)(C)C RF01558 c1cc(c(cc1Cl)Cl)c2cc(on2)c3ccnc(n3)S SPB05088 Cc1ccc(cc1C)C(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10843 c1cc(ccc1CC#N)OC(=O)c2ccncc2 RF04709 CCN(c1ccc(cc1)Cl)C(=O)c2cccnc2OCC(F)(F)F RF04886 CC(C)(C)NC(=S)N/N=C/c1c(cccc1Cl)Cl RF01520 CC(C)(C)NC(=S)N/N=C/c1cccc(c1)[N+](=O)[O-] RF01529 Cc1ccc(c(c1)C)n2c(noc2=O)c3cnc(cc3C(F)(F)F)SC RF05246 CCOC(=O)c1csc(n1)NC(=O)CN2CCN(CC2)C HTS10109 CN(C)c1ccncc1C(=O)Nc2ccc(cc2F)F RF05521 COc1ccc(cc1)NCc2ccccn2 HTS10575 c1ccc(cc1)/C(=N/O)/Nc2ccc(c(c2)Cl)Cl RF05115 Cc1nccc(n1)c2cccc(c2)N/N=C(\C#N)/C(=O)c3cccc(c3)OC KM02508 c1ccn(c1)c2ccc(c(c2)C(=O)O)N3CCOCC3 HTS08546 c1ccc2c(c1)c(c[nH]2)CC(C(=O)O)NCc3ccc(cc3)[N+](=O)[O-] HTS11455 CCCc1cnc(nc1)N2CCN(CC2)C(=O)NS(=O)(=O)c3ccc(cc3)C HTS09257 CC(C)NC(=O)O/N=C(\C)/C=C/c1ccccc1 EN00226 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4cn(nc4c5ccccc5)c6ccccc6)C HTS10275 CC(=O)OC[C@@H]1[C@H](C[C@@H](O1)n2cc(c(=O)[nH]c2=O)Br)OC(=O)C HTS11478 Cc1csc(n1)SCC(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F TG00085 c1ccc(c(c1)C2CC(=O)c3ccccc3O2)Cl RG00009 CC(C)(C)c1ccc(c(c1)[N+](=O)[O-])NC(=O)c2ccc(cc2)Cl RF01716 c1cc(sc1)NC(=O)NCC2CC2 HTS10504 Cc1cc(cc(c1)NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C HTS10528 Cc1ccc(cc1Cl)NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS10530 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCC3CC3 HTS10505 c1ccc(cc1)Cn2c(nnc2SCc3ccccc3)c4c(c5c(cc(nc5o4)c6ccccc6)c7ccco7)N HTS10274 CC(=O)OC[C@H]1[C@@H]([C@@H]([C@H](O1)n2cnc3c2nc([nH]c3=O)N)OC(=O)C)OC(=O)C HTS11459 c1ccc(cc1)Nc2c(c(c(s2)C(=O)c3ccc(cc3)[N+](=O)[O-])N)c4[nH]c5ccccc5n4 HTS10016 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)Nc3cc(sc3)c4ccc(cc4)Cl HTS09393 c1ccc(c(c1)Cn2c3ccccc3nc2COc4ccc(cc4Cl)Cl)Cl HTS09825 Cc1cc(on1)c2ccccc2C(=O)Nc3ccccc3O HTS09827 Cc1cc(on1)c2ccccc2C(=O)NCCCOC HTS09828 Cc1ccc(cc1)S(=O)(=O)NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS10516 c1cc(ccc1NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)F HTS10532 c1ccc(cc1)NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS10533 Cc1cc(nc2c1c(c(s2)C(=O)NNC(=S)Nc3ccccc3)N)C HTS10276 c1cc(ccc1n2c(nnc2S)Cc3ccsc3)F HTS11296 Cc1c(=O)nc([nH]n1)SCC(=O)O CD09705 Cc1ccc(cc1)c2cnc(n2C)S TG00115 Cn1c(cnc1Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F)c3ccc(cc3)Cl TG00118 c1ccc(cc1)N/N=C/2\CCCC(=O)C2 BTB15241 CCOC(=O)c1cc(n(n1)c2cccc(c2C#N)F)C RF00741 c1cc(c(c(c1)F)C(=O)CSC(=S)N2CCCCC2)F RF02025 c1c(c(cc2c1OCO2)Br)/C=N/O RF01307 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3ccc(s3)[N+](=O)[O-])\N RF01776 c1cc(c(c(c1)Cl)/C=N/NC(=O)Cn2cc(c(=O)c(c2)Cl)Cl)Cl RF02073 COc1ccc(cc1NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl HTS10535 c1ccc(cc1)Cn2c(nnc2S)Cc3ccsc3 HTS11297 C/C(=N\O)/C(C)(C)Nc1ccc2c(c1)OCO2 HTS11311 Cc1c(=O)nc([nH]n1)N2CCCC2 CD09710 Cc1c(cn(n1)c2ccccc2)C=C3C(=O)N(C(=O)N(C3=O)C)C HTS10270 CC1CCc2c(sc3c2c(nc(n3)SCC(=O)c4ccc(cc4)Br)NCc5ccccc5)C1 HTS10271 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cccc(c3Cl)Cl RF00038 c1cc(c(c(c1)Cl)CSc2ccnc(n2)SCc3c(cccc3Cl)Cl)Cl HTS11469 c1ccc2c(c1)c3ccccc3n2Cc4ccc(cc4Cl)Cl HTS11471 CCCCNCCn1cnc2c1ncnc2N HTS11472 CCOC(=O)c1cc(nc(c1C#N)SC)C(C)(C)C RF01044 Cc1ccc(cc1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3)S(=O)C KM10257 Cc1ccc(cc1n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)OC)[nH]cn3)SC KM10354 CCOC(=O)/C(=C/c1cn(nc1c2cccs2)c3ccccc3)/C#N HTS11496 Cc1ccc(cc1)n2c(=O)c3cnn(c3[nH]c2=O)c4ccccc4 HTS11497 c1ccc(cc1)C(=O)c2cnn(n2)c3ccc(cc3)Cl HTS11203 c1ccc(cc1)N2C(C(=CC(=N2)C(=O)c3cccs3)C(=O)NN)C(=O)NN HTS10500 CN(C(=O)c1ccccc1Cl)/N=C/c2c(cc(cn2)C(F)(F)F)Cl HC00079 Cc1ccc(cc1n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)OC)[nH]cn3)S(=O)C KM10368 COc1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4SC KM10369 c1cc(ccc1S(=O)(=O)c2cscc2C(=O)O)Cl MO00552 COC(=O)Nc1ccc(cc1)SC(F)(F)F TL00415 Cc1csc(n1)SCC(=O)NNS(=O)(=O)c2ccc(cc2)Cl TG00081 c1cc2c(cco2)cc1C(=O)O CC07101 c1ccc2c(c1)cccc2c3nnc(o3)Nc4cccnc4 HTS11307 Cc1ccc2c(c1N)c(cc(n2)C(F)(F)F)OC KM08259 C/C(=N\Nc1nc2c(n1C)c(=O)n(c(=O)n2C)C)/Cc3ccccc3 HTS11434 c1ccc(cc1)Cn2c(=O)cc(n(c2=O)c3cccc(c3)[N+](=O)[O-])N KM09350 CNC(=S)NNC(=O)C1(CN2CCC1CC2)O MWP01210 CC(C)(C)c1ccc(s1)C(=O)Nc2ccc(cc2)F MBE00132 CCOC(=O)/C(=N\O)/C1=CSC2=NNC(N12)(C)C RF00714 CNC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F RF00766 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)c3ccc(c(c3)O)O HTS09643 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)N3CCOCC3 HTS09651 c1ccn(c1)c2ccc(cc2)CO CC25509 c1cc(c(cc1F)c2c(nc3n(c2=O)CCCC3)O)F KM10110 c1ccc(cc1)C2=NOC(C2)COC(=O)c3ccco3 HTS11437 c1cc(c(c(c1)Cl)/C=N/OC(=O)Nc2csc(n2)Cc3ccsc3)Cl MWP00463 Cc1ccccc1NC(=O)N(Cc2cccs2)C(=O)CC#N KM09690 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)C4c5ccccc5-c6c4cccc6 HTS09208 CS(=NC(=O)c1c(cc(cn1)C(F)(F)F)Cl)(=O)c2ccc(cn2)C(F)(F)F KM07555 Cn1c(nnc1SCC(=O)NNC(=O)c2ccc(cc2)C(F)(F)F)Cc3ccsc3 SPB02393 CCn1c(cc(n1)C)c2nnc(n2c3ccccc3)S SPB02500 CCOC(=O)C(=C/N=c/1\[nH]c(cs1)c2ccc(cc2)Cl)C(=O)OCC TG00086 c1cc2c(cc1C(=O)NCCN3CCNC3=O)nccn2 HTS09572 CCn1c(nnc1SCC(=O)c2ccc(cc2)Br)CN3c4ccccc4Sc5c3cccc5 HTS10269 Cc1ccccc1Cn2cc(c(=O)[nH]c2=O)C HTS11214 c1ccc(cc1)CCn2cnc3c2ncnc3N HTS11215 COC(=O)c1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4cccc(c4)SC KM10225 Cc1nc2ccc(cc2o1)NC(=O)NC(=O)c3c(cccc3F)OC MWP00034 c1ccc2c(c1)n(c(=O)n2Cc3ccc(cc3Cl)Cl)Cc4ccc(cc4Cl)Cl HTS11209 Cc1cc2c(cccc2NC(=O)c3ccccc3C(=O)O)nn1 HTS09553 Cc1c2c([nH]n1)OC(=C(C23CCN(CC3)Cc4ccccc4)C#N)N HTS11488 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccc4c(c3)OCCCO4 HTS09726 CC(C)c1ccc(cc1)NC(=O)CC2C(=O)NCCN2 HTS08853 c1ccc(cc1)COc2ccc(cc2)/C=N/Nc3nc4c(ncnc4n3[C@@H]5[C@H]([C@H]([C@@H](O5)CO)O)O)N HTS11217 c1ccc2c(c1)cccc2Cn3c(=O)c(cn(c3=O)C4CCCO4)F HTS11454 CCOC(=O)C1=C(N2CCN=C2S1)C.Cl HTS10971 c1nc(c2c(n1)n(c(n2)NN=C3C(=O)NC(=O)NC3=O)[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09798 COc1ccc(cc1)C(=O)CSc2nnc(n2c3ccccc3)O HTS09614 c1ccc2c(c1)c(cs2)C(=O)CSc3nnc(n3c4ccc5c(c4)OCCO5)O HTS09616 CC(C)(C)c1ccc(cc1)NC(=O)Nc2cc(sc2C(=O)OC)c3ccc(cc3)Cl HTS09386 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3cc(cc(c3)Cl)Cl HTS09639 c1cc(cnc1)CNCc2ccco2.Cl HTS11487 Cc1nc(cs1)c2nc(cc(n2)N(C)C)COC SPB04579 CN(C)/C=C/c1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC SPB04590 Cc1c(c(n(n1)CCC#N)C)Sc2ncccn2 SPB06151 c1cc(sc1)NC(=O)N2CCN(CC2)c3ncccn3 HTS10747 Cc1ccc(cc1)CN2CCc3cc(c(cc3C2=O)OC)OC GK02023 c1ccc(cc1)S(=O)(=O)NCC2COc3ccccc3O2 HTS10757 c1cc(ccc1NC(=O)c2cc3cc(ccc3[nH]2)Cl)F HTS09317 COc1ccc(cc1)Oc2ccc(cc2C(=O)N3CCCc4c3cccc4)[N+](=O)[O-] HTS10172 c1ccc2c(c1)CCCN2S(=O)(=O)c3ccc(cc3)n4cccn4 HTS10625 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(CN3CCOCC3)c4ccccc4 HTS10198 Cc1c(snn1)C(=O)NC(=O)c2ccccc2O HTS10456 Cn1cc(nc1)S(=O)(=O)NNC(=O)c2ccc(c(c2)OC3CCCC3)OC HTS10098 CCOC(=O)c1c(sc(n1)C)c2cc[nH]n2 SPB04600 Cc1nc(cs1)c2cc(no2)C(=O)O CC14001 Cc1cc(nc(n1)Sc2ccccc2N)C(=O)OC SPB06391 COc1cc2c(cc1OC)C(=O)N(CC2)Cc3ccc(cc3)F GK02020 c1ccc2c(c1)c(c(s2)C(=O)NCC3COc4ccccc4O3)Cl HTS10753 Cc1c(snn1)C(=O)NCC2COc3ccccc3O2 HTS10754 c1ccc2c(c1)OCC(O2)CNC(=O)c3ccco3 HTS10756 CC(=O)Nc1cccc(c1)OCCCN2CCS(=O)(=O)CC2 HTS08539 CC(C)(C)c1cc(n(n1)C)C(=O)N(C)c2nnc(s2)C(F)(F)F HTS08804 CC(=O)Nc1ccc(cc1)N(CN2C(=O)CCC2=O)CN3C(=O)CCC3=O HTS10162 Cc1c(cccc1Cl)NC(=O)C2=NNC(=O)CC2 HTS09713 Cc1cc(no1)NC(=O)CC2C(=O)N(CCN2)Cc3ccccc3 HTS09718 c1cc2c(c(c1)S(=O)(=O)Nc3ccc(cc3)OC(F)F)non2 HTS10056 Cn1cc(nc1)S(=O)(=O)Nc2ccc(cc2)OC(F)F HTS10057 CC(C)(C)c1cc(no1)C(=O)NNC(=O)c2ccc(cc2)Cl SPB03156 c1cc(cc(c1)NC(=O)NCC2CC2)C(F)(F)F HTS10470 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3cc(nn3C)C(C)(C)C)C HTS08820 Cc1cc(no1)c2nc(c(s2)C(=O)NNC(=S)NC)C SPB05305 c1cc2c(cc1C#N)nc([nH]2)C(C(c3[nH]c4ccc(cc4n3)C#N)O)O SPB07794 Cc1c(c(on1)C)S(=O)(=O)NCC2COc3ccccc3O2 HTS10759 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)C(=O)C4CCCO4 HTS10766 Cn1c2c(cc(s2)C(=O)O)c(n1)C(F)(F)F GK02655 Cc1csc2c1ncnc2N3CCN(CC3)C(=O)Nc4ccc(c(c4)Cl)Cl GK02683 CC(C)(CC(=O)Nc1ccc(cc1)F)Sc2ccc(cc2)Cl HTS09678 Cc1c(c(no1)c2c(cccc2Cl)F)c3nnc(o3)c4ccc(cc4)C(F)(F)F HTS09776 CS(=O)c1cccc(c1)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM09347 CSc1nc(nc(n1)NC(=O)NS(=O)(=O)c2ccccc2C(F)(F)F)C34CC5CC(C3)CC(C5)C4 RF02816 COc1nc(nc(n1)NC(=O)NS(=O)(=O)Oc2ccc(cc2Cl)Cl)C34CC5CC(C3)CC(C5)C4 RF02817 CSc1nc(nc(n1)NC(=O)NS(=O)(=O)Oc2ccc(cc2Cl)Cl)C34CC5CC(C3)CC(C5)C4 RF02818 c1ccc2c(c1)cccc2NC(=O)NCC3CC3 HTS10468 c1cc(ccc1NC(=O)C2=NNC(=O)CC2)F HTS10251 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)O SPB05409 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)c3ccc4c(c3)nsn4 HTS09402 CCCCc1c(nc(nc1O)O)COC GK02336 c1cc(ccc1NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)F HTS10835 Cc1c(sc(n1)c2ccccc2)c3nnc(o3)c4ccc(cc4)C(F)(F)F HTS09772 c1cc(ccc1c2nnc(o2)c3ccc4c(c3)nccn4)C(F)(F)F HTS09775 c1cc2c(cc1NC(=O)NCC3CC3)CCO2 HTS10503 c1cc(sc1)CN2C(=O)CNC2=S RF02885 Cc1cc(c(cc1Cl)C)S(=O)(=O)n2cc(c(n2)C)c3ccccc3 CD09351 COc1c(cc(c(c1NC(=S)Nc2ccc(cc2)F)OC)Cl)Cl RF00688 CCOC(=O)c1c(cc(nc1O)C)C RF00883 c1cc(sc1/C=N/O)[N+](=O)[O-] RF00893 c1cc(sc1S(=O)(=O)N2CCN(CC2)CC(=O)N3CCOCC3)Cl HTS10981 Cc1c(nn(n1)c2ccccc2)C(=O)N(C)CCc3ccccn3.Cl HTS09191 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3cc(ccc3N4CCCC4)C(F)(F)F HTS09337 CC(C)(C)c1ccc(c(c1)NC(=O)C(Cl)(Cl)Cl)NC(=O)CN2CCOCC2 RF01722 COc1ccc(cn1)NS(=O)(=O)c2ccc(s2)Cl HTS10813 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(nc2)OC HTS10818 COc1ccc(cn1)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS10819 c1cc(cc(c1)Cl)N2CCN(CC2)/C=C/c3nnnn3c4ccc(cc4)Cl HTS10410 c1ccc(cc1)c2c3cc(ccc3ncc2c4nnnn4c5ccc(cc5)Cl)Cl HTS10472 Cn1c(nnc1S)C2COc3ccccc3O2 KM07018 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)Nc5ccc(cc5)F HTS09206 c1ccc2c(c1)ccc3c2sc(c3)C(=O)O PD00013 c1ccc2c(c1)ccc3c2sc(c3)C(=O)Nc4ccc(cc4)Cl PD00021 COc1ccc2c(c1)c(cc(n2)c3ccc(cc3)F)C(=O)O PD00094 CSC1=N/C(=C\Nc2ccccc2Cl)/C(=O)N1Cc3cccc(c3)Cl RF03495 Cc1c(cccc1S(=O)C)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM10256 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc(s2)c3ccccn3 HTS10554 Cc1c(c(no1)c2cccc(c2)[N+](=O)[O-])C(=O)O/N=C(\C#N)/c3ccccc3 RF00889 c1ccc(c(c1)c2[nH]nc(n2)c3ccc4c(c3)CCO4)O HTS10550 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4ccc(cc4Cl)Cl)C HTS10375 COc1cccc(c1)C(=O)Nc2nc([nH]n2)SCc3ccc(cc3)Cl HTS10138 c1ccc(c(c1)C(=O)NCC2COc3ccccc3O2)C(=O)O HTS10156 CC(C)(CC(=O)Nc1cccnc1)Sc2ccc(cc2)Cl HTS09681 CCc1cccc(c1NC(=O)Nc2c(cccc2CC)CC)CC RF00385 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/O RF00371 CS/C(=C\C(=O)c1cccs1)/NCc2ccccc2 MGH00243 COc1c(cc(c(c1C(=O)NNc2cc(ccc2Cl)Cl)OC)Cl)Cl RF00634 c1ccc(cc1)C2(C(=O)c3ccccc3C2=O)Nc4ccc(c(c4)Cl)Cl HTS11213 COc1cccc(c1)NC(=O)N2CCCc3c2cccc3 HTS10194 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCCc4c3cccc4 HTS10193 CSc1nc(nc(n1)NC(=O)NS(=O)(=O)c2ccccc2Cl)c3ccncc3 RF02739 Cc1cc(no1)/N=C/c2cccnc2 RF03202 CCCCCNc1nc2c(n1C)c(=O)n(c(=O)n2C)Cc3cccc(c3)Br HTS11192 c1ccc(cc1)C(=O)O/N=C(/c2csc(n2)c3cccnc3)\N MWP01183 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COC(=O)c3ccco3)OC(=O)c4ccco4 HTS11210 COc1ccc(cc1)NC(=O)C2CC(=O)N(C2)Cc3ccc(cc3)F HTS10901 CCc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C/c3c(cccc3Cl)Cl RF01136 c1cc(ccc1COCC(=O)O)Br HTS11100 Cc1c(c(on1)c2ccco2)C(=O)NN JM00049 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)CC(=O)c5ccc6c(c5)OCO6 HTS10658 Cn1c(cc(n1)c2ccccc2)NC(=O)Nc3cccs3 HTS10230 CC(=O)Cn1cc(c(=O)c(c1)Cl)Cl RF03245 c1ccc(c(c1)CNC(=O)c2ccc3c(c2)snn3)Cl RF03278 c1ccc(cc1)NC(=S)Nc2ccc(cc2)C3CC3(Cl)Cl RF02127 Cc1nc(cs1)c2ccccc2 RF02932 CSc1cccc(c1)n2c3c(c(=O)n(c2=O)Cc4ccc(cc4)C(=O)O)[nH]cn3 KM10224 c1cc(ccc1CC(=O)Nc2cc(ccc2Cl)C(F)(F)F)[N+](=O)[O-] RF00482 c1cc(ccc1CC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] RF00484 CC1CCc2c(sc3c2c(ncn3)SCC(=O)N/N=C/c4ccc(cc4)Cl)C1 HTS11491 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)N3CCCc4c3cccc4 HTS10197 c1cc(cc(c1)N2C(=O)CCC2=O)C(=S)N JM00306 c1ccc2c(c1)nc(s2)c3cccnc3 HTS11482 c1cc(ccc1NC(=O)c2ccc3c(c2)non3)N4CCCCC4 HTS09309 Cc1c(c(no1)c2ccccc2)NC(=O)Nc3cccc(c3)S(=O)(=O)N HTS05520 CCCCCCCc1ccc(cc1)NC(=O)N(Cc2ccc(cc2)Cl)Cc3cccnc3 RF03314 c1ccc(cc1)n2c(nnc2S)c3cccc4c3cccc4 HTS10654 c1ccc(cc1)CNc2nc3c(=O)[nH]c(nc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS11169 c1cc(cnc1)CN(Cc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl RF03423 CC(C)(C)c1ccc(cc1)NC(=O)N(C)CCc2ccccn2 HTS08780 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)CCC(=O)O HTS09768 c1cc(oc1)Cn2c(nnc2SCc3cc(cc4c3OCOC4)Cl)c5ccc(cc5)C(F)(F)F HTS10657 COc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3cccnc3 HTS11499 CC(C)(C)/C=N/Nc1nc2c(s1)cc(cc2Cl)Cl RF02708 CCOC(=O)c1c(noc1c2ccco2)C JM00026 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F HTS10833 COc1ccccc1NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10834 c1cc(ccc1C(=O)CN2C(=O)CCC2=O)F HTS10067 c1ccc(cc1)Cn2c(n[nH]c2=S)c3c(c4c(cc(nc4o3)c5ccccc5)c6ccco6)N HTS11506 Cc1cc(nc2c1c(c(s2)c3n[nH]c(=S)n3Cc4ccccc4)N)C HTS11507 c1ccc(cc1)Cn2c3c(c(ncn3)N(Cc4ccccc4)Cc5ccccc5)nn2 HTS11508 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C/c3cc(c(c(c3)OC)OC)OC)Cc4ccc(cc4)Br HTS11179 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)Nc3ccc4c(c3)OCCO4 HTS10424 c1cc2c(cc1C(=O)N3CCN(CC3)CC(=O)N4CCCC4)CCO2 HTS10782 Cc1c(c(on1)c2ccccc2)CO CC20309 CC(=O)CSc1[nH]c(=O)c(c(n1)N)C(c2ccc(cc2)OC)c3c(nc([nH]c3=O)SCC(=O)C)N HTS11492 c1ccc(cc1)C(CN2CCN(CC2)C3c4ccccc4-c5c3cccc5)O HTS09751 CCOC(=O)c1csc(n1)NC(=O)CN2CCOCC2 HTS10108 c1ccc2c(c1)CCCN2C(=O)c3ccc4c(c3)nccn4 HTS10183 CC(=O)Nc1ccccc1OCC2CC(=NO2)c3ccccc3 HTS11485 c1cc2c(cc1CNC(=O)c3cc4cc(ccc4[nH]3)Cl)OCO2 HTS09315 c1cc(c(cc1F)F)NC(=O)/C=N/O RF01202 c1cc(sc1)NC(=O)Nc2cc(ccc2N3CCCC3)C(F)(F)F HTS09338 COc1cccc(c1)NC(=O)Nc2cc(ccc2N3CCCC3)C(F)(F)F HTS09339 Cc1cccc2c1N(CCC2)C(=O)Nc3ccc(cc3)OCc4ccccc4 HTS09416 Cn1c2c(nc1N/N=C/c3ccc(c(c3)OC)OC)n(c(=O)n(c2=O)Cc4ccccc4F)C HTS11180 c1cc([nH]c1)CN2CCN(CC2)c3c(cccn3)C(F)(F)F HTS10568 COc1ccc(cc1)NCc2ccc[nH]2 HTS10573 CCOC(=O)N1CCC(CC1)NC(=O)c2ccco2 HTS10610 Cc1cc(cc(c1)NC(=O)Nc2ccc(nc2)OC)C HTS10821 COc1ccc(cn1)NC(=O)Nc2cccs2 HTS10822 CCOc1ccccc1NC(=O)Nc2ccc(nc2)OC HTS10823 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)COCC(=O)O HTS09397 Cn1c(cc(n1)c2ccccc2)NC(=O)CCCC(=O)O HTS10205 c1ccnc(c1)c2ccc(s2)S(=O)(=O)Nc3ccc(cc3)N4CCCCC4 HTS09307 CC(C)(C)c1ccc(cc1)NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10836 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(cn2)C(F)(F)F HTS09348 c1cc(ccc1NS(=O)(=O)c2ccc(s2)c3ccno3)OC(F)F HTS10058 Cc1c(c(no1)c2ccc(cc2)F)C(=O)O MO00391 c1ccc2c(c1)CC(C2)n3c(nnc3SCC(=O)c4csc5c4cccc5)O HTS09613 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)OC(F)F HTS10055 c1cc(ccc1NS(=O)(=O)c2ccc(cc2)F)OC(F)F HTS10059 c1cc(ccc1C#N)c2cn3c(n2)SCC3 HTS10081 CCCNC(=C(C(=O)Nc1cccc(c1)Cl)C(=O)Nc2cccc(c2)Cl)c3ccc(cc3)OC HTS11484 c1c(cc(c(c1Br)O)Br)/C=N/NC(=S)N RF01546 CCOC(=O)N1CCC(CC1)NC(=O)Nc2ccc(c(c2)Cl)C HTS10807 c1cc(ccc1[N+](=O)[O-])OC(=O)CCCC(=O)Oc2ccc(cc2)[N+](=O)[O-] CD07647 Cc1c(c(n(n1)C(C)(C)C)C)C#N CD07672 CCOC(=O)N1CCC(CC1)NC(=O)c2ccc(cc2)C HTS10618 c1c(csc1[N+](=O)[O-])C(=O)NC(=S)NN2CCOCC2 DFP00153 CCCc1c(cnn1c2ccccc2)C(=O)NC3CCN(CC3)C(=O)OCC HTS10611 CCOC(=O)N1CCC(CC1)NC(=O)c2cccs2 HTS10612 c1cc(ccc1n2c(nnn2)c3cnccc3C(F)(F)F)Cl RF04515 Cc1c(c(no1)c2ccccc2)C(=O)N3CCCc4c3cccc4 HTS10173 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)c3cccnc3Oc4ccccc4 HTS09389 CC(C)(C)NC(=S)N/N=C/c1coc2c(c1=O)cc(cc2Cl)Cl RF01260 c1c(cc(c(c1/C=N/NC(=S)N)O)Cl)Cl RF01460 c1ccc(c(c1)C(=O)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl)O HTS10462 Cc1c(csc1C(=O)Nc2cc(ccc2N3CCCC3)C(F)(F)F)S(=O)(=O)c4ccc(cc4)Cl HTS09429 c1ccc2c(c1)cccc2NC(=O)Nc3cc(ccc3N4CCCC4)C(F)(F)F HTS09431 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2ccc(cc2)N(C)C HTS10997 c1cc(c(cc1C(F)(F)F)NC(=O)CSCC(=O)O)N2CCCC2 HTS09436 Cn1cc(cn1)S(=O)(=O)Nc2ccc(nc2)Oc3c(cccc3Cl)Cl HTS11139 c1cc(c(c(c1)Cl)CSc2nc3cc(ccc3s2)Cl)Cl EN00192 CN(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)OC(F)(F)F HTS10993 CN(C)c1ccc(cc1)NC(=O)Nc2cccc(c2)Cl HTS10995 Cc1cc(cc(c1)NC(=O)Nc2ccc(cc2)N(C)C)C HTS10998 c1cc(c(c(c1)Cl)/C=N/N=C\2/NC(=O)CS2)Cl RF01537 CC(C)(C)N/C(=N/N=C/c1cc(cc(c1O)Cl)Cl)/SC RF01539 COc1ccc(cc1OC)C(=O)N2CCCc3c2cccc3 HTS10185 c1ccc2c(c1)CCCN2C(=O)Nc3cc(cc(c3)Cl)Cl HTS10192 Cc1cc(c(c(c1)O)C(=O)CC(=O)c2ccccc2Cl)C RG00025 Cc1cc(nc(n1)Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])C RF00391 COc1ccc(cc1OC)C2=NOC(C2)COc3ccc(cc3)[N+](=O)[O-] HTS11208 Cc1cc(nc2c1c3c(o2)c(=O)[nH]cn3)c4ccccc4 HTS11489 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F HTS10845 c1cc(c(cc1F)F)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10847 CC(C)(C(=O)NN)Oc1ccc(cc1)Cl RDP00173 Cc1cc(cc(c1)NC(=O)Nc2cccnc2)C HTS10990 c1cc(ccc1c2csc(n2)Sc3nc4cc(ccc4s3)Cl)Cl TG00091 c1cc(c(c(c1)F)c2csc(n2)Nc3ccc(c(c3)Cl)Cl)F RF02030 c1ccc(cc1)C(Cc2cccnc2)(c3ccccc3)O RF01077 c1cc(cc(c1)Nc2nc(cs2)c3c(cccc3F)F)C(F)(F)F RF02031 CN(C)C(=O)Oc1ccnc(n1)SCc2c(cccc2Cl)Cl JM00426 CCOC(=O)Cn1c(c(c(n1)C)[N+](=O)[O-])C KM01045 c1cc(ccc1NC(=O)NNC(=O)Cn2cc(c(=O)c(c2)Cl)Cl)Cl RF02084 Cc1ccc(cc1)NC(=O)C2CC(=O)N(C2)CCc3ccc(cc3)Cl HTS10908 Cc1ccc2cc(ccc2n1)NC(=O)C3CC(=O)N(C3)CCc4ccc(cc4)Cl HTS10909 c1cc(ccc1C(=O)CNC(=O)CCC(=O)O)OC(F)F HTS10078 c1ccc(c(c1)C(=O)N)NCC(=O)c2ccc(cc2)F HTS10816 Cn1c2c(nc1N3CCCCC3)n(c(=O)n(c2=O)Cc4ccc(cc4Cl)Cl)C HTS11191 CSc1nc(cc(n1)O)C(=O)O RF03525 CC1=CCC(C(C1)C(=O)O)C(=O)N(Cc2cccnc2)Cc3ccc(cc3Cl)Cl RF03585 c1ccnc(c1)SCc2cccc(c2)/C(=N/OC(=O)c3ccc(c(c3)Cl)Cl)/N KM01531 CC(C)(C)S(=O)(=O)/C(=C/c1ccsc1)/C#N KM02137 c1cc(ncc1C(=O)N)C(=O)O RF03037 c1cc(ccc1/N=N/N2CCOCC2)Cl RF00305 Cn1c(cnc1SCc2c(cccc2Cl)Cl)c3ccc(cc3)Cl TG00113 Cc1cc(no1)c2nc(c(s2)C(=O)NN)C SPB04691 c1c(cc(c2c1c(cc(=O)[nH]2)C(=O)O)Cl)Cl RF00901 c1cc(c(cc1/C=N/NC(=O)Cn2cc(c(=O)c(c2)Cl)Cl)Cl)Cl RF02072 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nnc(n3c4ccccc4)c5ccc(cc5)Cl)C1 HTS11493 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/c2ccc(s2)[N+](=O)[O-])\N RF01782 c1cc(ccc1C2CC2(Cl)Cl)NC(=S)Nc3ccc(cc3Cl)Cl RF02128 CCOC(=O)C(C(=O)C)Sc1cc(nc2n1ncn2)c3ccccc3 HTS11494 Cc1ccc(cc1)C2Nc3ccccc3C(=O)N2CCCN4CCOCC4 HTS10233 Cc1ccc(cc1)C2Nc3ccccc3C(=O)N2CCN4CCNC4=O HTS10234 CSc1nc(nc(n1)NC(=O)NS(=O)(=O)Oc2ccc(cc2Cl)Cl)c3cccnc3 RF02795 c1ccc2c(c1)C(=O)N(S2(=O)=O)Cc3nc4ccccc4s3 HTS10024 c1cc(cc(c1)Cl)C(=O)OCCSc2c(cccn2)[N+](=O)[O-] BTB08937 Cn1c2ccccc2c3c1CCC(C3=O)Cn4ccnc4.Cl BTB15251 COc1cc(cc(c1OC)OC)CSC2=NCCN2.Cl CD02327 CS/C(=C\C(=O)c1cccs1)/NCc2ccco2 MGH00244 COc1ccc(cc1)NC(=O)C2CC(=O)N(C2)CCc3ccc(cc3)Cl HTS10906 c1cc(ccc1CCN2CC(CC2=O)C(=O)NCc3ccc4c(c3)OCO4)Cl HTS10907 Cn1c(cc(n1)c2ccccc2)NC(=O)c3cccs3 HTS09745 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C/C(=O)c3ccccc3 RF00885 CCOC(=O)/C(=C/c1cn(nc1c2ccco2)c3ccccc3)/C#N HTS11495 Cc1cc(nc2c1c3c(s2)c(ncn3)SCc4ccccc4Cl)C HTS11501 c1ccc(c(c1)/C=N/Nc2nc3c(s2)cc(cc3Cl)Cl)O RF02710 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3ccc(cc3)C(F)(F)F HTS09640 Cc1c(sc(n1)c2ccccc2)C(=O)N3CCCc4c3cccc4 HTS10174 c1ccc2c(c1)CCCN2C(=O)Nc3ccc(cc3)C(F)(F)F HTS10190 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3ccc4c(c3)nccn4)C HTS11107 Cc1c(cnn1c2ccccc2)S(=O)(=O)N3CCCN(CC3)C(=O)OC(C)(C)C HTS11117 CSC1=N/C(=C\Nc2ccc(cc2)Cl)/C(=O)N1Cc3ccccc3Cl RF03510 CSc1nc(cc(n1)O)C(=O)N RF03533 c1cc(cc(c1)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)F HTS10848 c1cc(ccc1C#N)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10849 Cc1ccc(cc1Cl)NC(=O)Nc2cccnc2 HTS10989 c1cc(cc(c1)Cl)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3 HTS09306 c1cc(ccc1NS(=O)(=O)c2ccc(s2)c3ccno3)N4CCCCC4 HTS09308 Cc1c(nn(n1)c2ccccc2)C(=O)N3CCCc4c3cccc4 HTS10177 Cc1cccc(c1NC(=O)C(c2ccccc2)Sc3c(c(cc(n3)C)C)C#N)Cl RF00242 c1cc(c(c(c1)F)C#N)NC(=O)c2c(nccn2)C(=O)O HTS09363 CCc1ccccc1CSc2nnc(n2C(C)c3ccccc3)O HTS09480 c1ccc2c(c1)C(=O)N(S2(=O)=O)CCS(=O)(=O)c3ccc(cc3)F HTS09652 COc1ccc(cc1)c2nc(no2)CN3C(=O)c4ccccc4S3(=O)=O HTS09656 c1cc2c(c(c1)S(=O)(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F)non2 HTS10852 Cc1c(c(on1)C)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10853 c1cnc2nc(cn2c1)c3ccc(cc3)C(=O)O HTS09268 COc1ccc(cc1)NC(=O)C2=NNC(=O)CC2 HTS09708 CC(=O)C1=NN(C2(S1)N(C(=O)/C(=C\c3ccccc3)/S2)c4ccccc4)c5ccc(cc5)Cl HTS10486 COC(=O)c1cc(ccc1OCS(=O)(=O)c2ccc(cc2)Cl)NC(=O)NC(=O)c3c(cccc3F)F RF03592 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F HTS10851 c1ccc(cc1)c2ccc(s2)NC(=O)NCc3ccc(cc3)C#N HTS10932 c1ccc(c(c1)C(F)(F)F)NC(=O)c2ccsc2 HTS10687 c1ccc2c(c1)CCCN2S(=O)(=O)c3ccc4c(c3)CCO4 HTS10182 c1ccc2c(c1)CCCN2C(=O)c3ccc(cc3F)F HTS10186 CCOC(=O)c1c(c(nc(c1[N+](=O)[O-])C(C)(C)C)O)C#N RF01047 c1cc(ccc1NC(=O)c2cc3cc(ccc3[nH]2)Cl)N4CCOCC4 HTS09316 COc1ccc(cc1)OCCNC(=O)c2ccc3c(c2)nccn3 HTS09575 c1ccc(cc1)Oc2cccc(c2CNC(=O)c3ccc4c(c3)nccn4)Cl HTS09577 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3c(cc(cc3Cl)Cl)Cl SPB00274 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)c3ccc4c(c3)OCCO4 HTS10021 Cc1cccc2c1N(CCC2)C(=O)Nc3ccc(cc3)OC HTS09418 c1cc(ccc1C(F)(F)F)S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10855 c1ccc2c(c1)OCC(O2)CNS(=O)(=O)c3ccc4c(c3)CCO4 HTS10758 c1ccc(cc1)COc2ccc(cc2)NC(=O)N3CCN(CC3)c4ncccn4 HTS10748 Cc1ccc(cc1Cl)NC(=O)NCc2ccc(cc2)C#N HTS10933 c1ccc2c(c1)OCC(O2)CNS(=O)(=O)c3cc(sc3Cl)Cl HTS10760 c1ccc(cc1)S(=O)(=O)c2ccc(s2)S(=O)(=O)NCC3COc4ccccc4O3 HTS10761 c1cc(ccc1CCNC(=O)c2ccc3c(c2)nccn3)Cl HTS09580 CCc1ccccc1CSc2nnc(n2c3c(cc(cc3C)C)C)O HTS09603 COC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)c3ccc4c(c3)CCO4 HTS09391 c1cc(cc(c1)Cl)S(=O)(=O)N(c2ccc(cc2)S(=O)(=O)N)S(=O)(=O)c3cccc(c3)Cl HTS10178 Cc1cc(n(n1)C)C(=O)Nc2cc(ccc2N3CCCC3)C(F)(F)F HTS09428 COc1nc(nc(n1)NC(=O)NS(=O)(=O)c2ccccc2C(F)(F)F)C34CC5CC(C3)CC(C5)C4 RF02815 Cc1cccc(c1C)C(=O)NC(=O)c2ccccc2O HTS10465 Cc1c(cc(o1)c2ccccc2)C(=O)NCc3ccc4c(c3)OCO4 HTS10586 CC(=O)Nc1ccc(cc1[N+](=O)[O-])C(C)(C)C RF01556 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)OC HTS10809 CCOC(=O)N1CCC(CC1)NC(=O)c2c(c3ccccc3s2)Cl HTS10619 c1ccc(cc1)NC(=O)NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F RF04511 c1ccc2c(c1)OCC(O2)CNS(=O)(=O)c3cccs3 HTS10762 c1ccc(cc1)Nc2nnc(o2)c3cccc4c3cccc4 HTS10656 c1ccc(cc1)C(CNCC2COc3ccccc3O2)O HTS10160 CCOC(=O)NC(=S)Nc1ccc(cc1[N+](=O)[O-])C(C)(C)C RF01602 c1cc(ccc1CNC(=O)N2CCOCC2)C#N HTS10945 CCOC(=O)C(c1ccccc1)NC(=O)C2CCC(CC2)c3ccc(cc3)Cl HTS10951 CCOC(=O)C(C)NC(=O)C1CCC(CC1)c2ccc(cc2)Cl HTS10953 CC(C(=O)O)N1C(=O)c2ccccc2C1=O HTS10163 Cc1ccc(cc1Cl)S(=O)(=O)Nc2ccc(nc2)OC HTS10810 COc1ccc(cc1OC)S(=O)(=O)Nc2ccc(nc2)OC HTS10811 Cc1ccc(cc1Cl)NCN2C(=O)CCC2=O CD04777 Cc1c(ncn1Cc2ccc(cc2)Cl)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F KM05035 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C\3/CCSC3 CD10441 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/Nc3c(cc(cc3Cl)Cl)Cl RF02022 c1cc(c(cc1OCC(F)(F)F)C(=O)N)OCC(F)(F)F RF04513 c1cc(ccc1S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)Cl HTS10850 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)SCC(=O)C GK00191 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3ccc(cc3)F HTS10072 c1cc(cnc1)NC(=O)Nc2ccc(cc2)F HTS10986 c1cc(c(cc1c2cc(on2)CO)Cl)Cl RF01801 CN(CCc1ccccn1)C(=O)c2c(nccn2)C(=O)O HTS09766 CC(C)(CC(=O)N1CCN(CC1)C2c3ccccc3-c4c2cccc4)CC(=O)O HTS09770 COc1ccc(cn1)NS(=O)(=O)c2ccc(cc2)F HTS10812 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CC(=O)N3CCOCC3 HTS10829 Cc1coc(=O)n1c2ccc(cc2Cl)Cl RF05403 Cc1ccc2cc(ccc2n1)NC(=O)C3CC(=O)N(C3)Cc4ccc(cc4)F HTS10904 Cc1c(c(c(n1C2CC2)C)C(=O)O)C(=O)C MO00624 c1cc(ccc1CCN2CC(CC2=O)C(=O)Nc3ccc(cc3)Cl)Cl HTS10905 Cc1ccc(cc1)N2C3(N(C(=O)/C(=C\c4ccccc4)/S3)c5ccccc5)SC(=N2)C(=O)Nc6ccccc6 HTS10481 c1cc(sc1/C=N/Nc2nc3c(s2)cc(cc3Cl)Cl)[N+](=O)[O-] RF02712 c1cc(ccc1CCN2CC(CC2=O)C(=O)O)Cl MO00129 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCC3CCCO3)Cc4cccc(c4)Br HTS11184 Cn1c2c(nc1NCCCCCO)n(c(=O)n(c2=O)Cc3ccc(cc3Cl)Cl)C HTS11186 CC1(Cc2c(c(sc2C(=O)Nc3ccc(cc3)Cl)SC)/C(=N/OC)/C1)C KM03602 c1ccc(cc1)C2C(=NOC23C(=O)c4ccccc4C3=O)C(=O)c5ccccc5 HTS10478 Cc1ccc(cc1)C2C(=NOC23C(=O)c4ccccc4C3=O)C(=O)c5ccccc5 HTS10479 CC(C)Sc1c(c(cc(n1)c2cccs2)C(F)(F)F)C#N RF01027 c1cnn(c1)c2ccc(cc2)CN CC18413 Cc1ccc(cc1)S(=O)(=O)N2CCN(CC2)CC(=O)N3CCOCC3 HTS10830 COC(=O)c1cc(ccc1OCS(=O)(=O)c2ccc(cc2)Cl)NC(=O)NC(=O)c3c(cccc3Cl)Cl RF03593 COC(=O)c1cn(cc(c1=O)F)Cc2ccncc2 HC00064 Cc1c(c(nc(=S)[nH]1)O)Oc2ccc(cc2)Cl SPB03974 CC(C)(C)c1c(cno1)C(=O)O SEW04589 COc1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)C(=O)Nc4ccccc4)c5ccccc5)c6ccccc6 HTS10483 COCCCn1c(cc(c1c2ccccc2)c3cccs3)c4ccc(cc4)Cl RG00098 CSc1nc(nc(n1)N2CCOCC2)NC(=O)NS(=O)(=O)c3ccccc3Cl RF02742 Cn1c2c(nc1NC3CCCC3)n(c(=O)n(c2=O)Cc4ccc(cc4)F)C HTS11188 CC1CCN(CC1)c2nc3c(n2C)c(=O)n(c(=O)n3C)Cc4cccc(c4)Br HTS11190 c1cc2c3c(c(ncn3)S)sc2nc1 MGH00222 CN(C)c1ccc(cc1)NC(=O)Nc2cccs2 HTS10999 CN(C)c1ccc(cc1)NC(=O)Nc2cc(ccc2OC)Cl HTS11000 COc1ccc(cc1OC)CCN2CC(CC2=O)C(=O)O MO00128 CSc1nc(nc(n1)NC(=O)NS(=O)(=O)c2ccccc2C(F)(F)F)c3ccccn3 RF02762 CNC(=S)NNC(=O)CN1c2cc(ccc2SCC1=O)C(F)(F)F KM08346 Cc1cc(nc2c1c3c(s2)c(ncn3)Sc4nnc(n4CC=C)c5ccc(cc5)Cl)C HTS11504 Cc1cc(cc(c1)NC(=O)NCc2ccc(cc2)C#N)C HTS10931 CC(C)(C)c1ccccc1NC(=O)NCc2ccc(cc2)C#N HTS10934 c1cc(ccc1CNC(=O)Nc2ccc(cc2)F)C#N HTS10935 CC(C)(C(=O)O)Oc1ccc(cc1)[N+](=O)[O-] CD04619 CCOC(=O)C1=NN(C2(S1)N(C(=O)/C(=C\c3ccccc3)/S2)c4ccccc4)c5ccc(cc5)C HTS10487 c1cc(ccc1C(=O)COC(=O)CC(C(=O)OCC(=O)c2ccc(cc2)C(F)(F)F)O)C(F)(F)F RF03435 c1cc(ccc1Cc2c(=O)nc3n(nc(n3n2)c4ccc(cc4Cl)Cl)c5ccc(cc5)[N+](=O)[O-])Cl HTS10489 Cc1cc(nc2c1c3c(s2)c(ncn3)Oc4ccc(cc4)Cl)C HTS11505 c1ccc(cc1)c2nnc3n2nc(cc3)Oc4ccc(cc4Cl)Cl RH00158 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCCc3ccccc3)Cc4ccccc4 HTS11183 COc1cc2cc(c(=O)oc2cc1OC)C(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 HTS10626 Cc1cc(nc2c1c3c(s2)c(ncn3)S)C HTS11503 c1cc(c(cc1F)F)NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F HTS10832 CC(C)C(=O)NNc1nc2c(n1Cc3ccc(cc3)Cl)c(=O)n(c(=O)n2C)C HTS11173 c1cc2c(cc1NC(=O)c3cc(cc4c3OCOC4)F)OCCO2 HTS10420 c1ccc(cc1)COC(=O)N2c3ccccc3CC2C(=O)Nc4ccc5c(c4)OCCO5 HTS10421 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS10423 c1ccc(cc1)c2c(cc(o2)c3ccc(cc3)Cl)c4cccs4 RG00090 c1ccn(c1)c2cccc(c2)C(=O)O CC21901 COc1cccc(c1)CC(=O)NNC(=O)c2ccc3c(c2)OCO3 HTS10673 Cc1c(snn1)C(=O)NNC(=O)Cc2cccc(c2)OC HTS10674 c1cc(=O)n(cc1[N+](=O)[O-])C2CCCCO2 BTB15252 Cc1cc(nn1C)c2nnc(n2c3cccc(c3)C(F)(F)F)SCc4ccc(cc4)Cl SPB00767 Cn1c(nnc1SCC#N)O SPB00782 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C/c3c(cccc3Cl)Cl)Cc4ccccc4 HTS11175 Cn1c2c(nc1N/N=C/c3ccc(cc3)Cl)n(c(=O)n(c2=O)Cc4ccc(cc4)Cl)C HTS11178 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C/c3ccccc3)Cc4ccccc4 HTS11181 COc1ccc(cn1)NS(=O)(=O)c2ccccc2 HTS10808 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)Nc3ccc(nc3)OC)C(F)(F)F HTS10815 COc1ccc(cn1)NC(=O)Nc2ccc(cc2)F HTS10817 CCOC(=O)N1CCC(CC1)NS(=O)(=O)c2cccs2 HTS10608 c1cc(ccc1F)S(=O)(=O)N2CCN(CC2)CC(=O)N3CCOCC3 HTS10828 Cc1c2cc(sc2n(n1)C)CO CC22909 COc1cccc(c1)CC(=O)NNC(=O)c2ccc3c(c2)nsn3 HTS10675 Cc1ccc(cc1)C2C3(C(=NN2c4ccc(cc4)[N+](=O)[O-])c5ccc(cc5Cl)Cl)C(=O)c6ccccc6C3=O HTS10488 COc1cccc(c1)Cc2nnc(o2)c3ccc(s3)c4cccs4 HTS11125 c1cnc(nc1)N2CCC(CC2)CO CC20709 CC1(CC(=O)CC(=O)S1)C KM04035 COc1cccc(c1NC(=O)N2CCOCC2)OC RF00510 c1cc(cc(c1)[N+](=O)[O-])NC(=N)NC(=N)N.Cl RJF01382 Cc1c(c(n[nH]1)C)Cc2csc3c2cc(cc3)Cl.Cl MWP00801 c1cc(ccc1C#N)Oc2c(cncc2Cl)Cl SPB07095 c1cc(ccc1S(=O)(=O)c2nc3cc(ccc3s2)Cl)Cl EN00209 Cn1c2c(nc1NCCc3ccc(cc3)O)n(c(=O)n(c2=O)C)C HTS11182 CCOC(=O)N1CCC(CC1)NC(=O)c2cc(cc(c2)C)C HTS10805 CCOC(=O)N1CCC(CC1)NC(=O)C2CCCCC2 HTS10616 CCOC(=O)N1CCC(CC1)NC(=O)c2cc(sc2Cl)Cl HTS10617 c1cc(sc1)NC(=O)N2CCN(CC2)C(=O)C3CCCO3 HTS10765 CN(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS11003 c1ccc2c(c1)cccc2NC(=O)NCc3ccc(cc3)C#N HTS10939 c1ccc(cc1)NC(=O)NCc2ccc(cc2)C#N HTS10940 c1ccc2cc(ccc2c1)c3csc(n3)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F.Br CD03069 Cc1cccc(c1C)n2c(nnn2)c3cnccc3C(F)(F)F RF04548 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=N/OC(=O)Nc3cccc(c3)Cl RF01891 C#CCOC(=O)Nc1cc(c(nc1)Sc2ccccc2)C(F)(F)F RF05315 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3cccc(c3)C(F)(F)F HTS10958 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccc(cc3)C(=O)OC HTS10965 CN(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)F HTS10992 Cc1c2c(cc(s2)c3ccc(cc3)F)sc1C(=O)OC GK01960 COc1ccc(cc1OC)C(=O)NCc2ccc(cc2)C#N HTS10943 Cc1ccc(cc1)N2C3(N(C(=O)/C(=C\c4ccccc4)/S3)c5ccccc5)SC(=N2)C(=O)c6ccccc6 HTS10485 Cc1cc(cc(c1CN(C)C(=O)c2cnc(cc2C(F)(F)F)Oc3ccc(cc3)Cl)Cl)Cl RF05044 COc1c(c(ccn1)C(F)(F)F)C(=O)NCc2c(cc(cc2Cl)Cl)Cl RF05060 c1ccc(c(c1)C(=O)Nc2cc(ccc2N3CCCC3)C(F)(F)F)C(=O)O HTS09435 CN(C)c1ccc(cc1)NC(=O)c2cccs2 HTS11004 c1cc(oc1)CN2CC(CC2=O)C(=O)Nc3ccc(cc3)F HTS11014 Cc1ccc2cc(ccc2n1)NC(=O)C3CC(=O)N(C3)Cc4ccco4 HTS11015 c1ccc(c(c1)C(F)(F)F)n2c(nnn2)c3cc(cc(c3)Cl)Cl RF04634 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3ccc(cc3)OC(F)F HTS10068 Cc1cccc(c1F)CSc2ccccc2C3=NCCCN3.Br CD05942 CC(C)(C)C1=C(C(C(=C(O1)NC(=O)NC(=O)c2c(cccc2F)F)C#N)c3cccs3)C#N CD06696 CC1(OC(=O)C(=Cc2ccc(c(c2)OC)OCc3ccccc3)C(=O)O1)C CD06764 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NCc3ccc(cc3)C#N HTS10949 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)NN KM08892 c1cc(ccc1CN2CC(CC2=O)C(=O)NCc3ccc4c(c3)OCO4)F HTS10902 CN(C)c1ccc(cc1)NC(=O)c2ccc(cc2)Cl HTS11255 c1cc(oc1)CNCCn2cnc3c2ncnc3N HTS11211 c1ccc(cc1)C2C(N(N=C2c3ccccc3)c4ccccc4)c5c(cn(n5)c6ccccc6)C#N HTS10482 CC(=O)Nc1ccc(cc1)S(=O)(=O)N2CCCc3c2cccc3 HTS10622 CCOC(=O)c1ccc(c(c1)N)NC MO00109 CCOC(=O)c1ccc2c(c1)nnn2C MO00117 CN(Cc1c(cccc1OC)OC)C(=O)c2cnccc2C(F)(F)F RF05437 CC(=O)c1ccccc1OC(=O)c2ccc(cc2)Cl RG00013 c1ccc(c(c1)C(=O)CC(=O)c2ccc(cc2)Cl)O RG00014 CCOC(=O)c1c(c(c([nH]1)C)CO)C CC23009 c1ccc(cc1)c2csc(n2)O RF03025 Cc1ccccc1Oc2nc3c(n2C)c(=O)n(c(=O)n3C)Cc4ccccc4Cl HTS11196 c1ccc(cc1)C2=NOC(C2)COC(=O)c3cccc(n3)C(=O)OCC4CC(=NO4)c5ccccc5 HTS11198 c1ccc(cc1)COc2ccc(cc2)NC(=O)Nc3ccc(nc3)Oc4c(cccc4Cl)Cl HTS09446 c1ccc2c(c1)c(c(s2)C(=O)N3CCN(CC3)C(=O)C4CCCO4)Cl HTS10891 CSc1nc(nc(n1)N2CCOCC2)NC(=O)NS(=O)(=O)Oc3ccc(cc3Cl)Cl RF02805 Cc1nc(nc(n1)N/N=C/c2c(cccc2Cl)F)N RF02943 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)c3ccc4c(c3)OCO4 HTS10022 c1cc(cc(c1)Cl)NC(=O)Nc2ccc3c(c2)snn3 RF03269 CSC1=N/C(=C\Nc2ccccc2)/C(=O)N1Cc3ccccc3Cl RF03507 CSC1=N/C(=C\Nc2ccc(cc2)Cl)/C(=O)N1Cc3ccco3 RF03552 c1c(cc(c(c1Br)NC(=N)NC(=N)N)Br)F.Cl RJF00741 c1cc(c(c(c1)Cl)C(CN2CCSCC2)O)F.Cl JM00165 c1ccc(cc1)C(=O)C(CC(=O)c2ccc(cc2)Cl)c3cccs3 RG00055 CN(CCc1ccccn1)S(=O)(=O)c2ccc3c(c2)CCO3.Cl HTS10667 c1cc(c(c(c1)F)C(=O)NC(=O)C(=O)Nc2ccc(cc2F)Br)F RF03984 Cc1cc(c(c(n1)O)C#N)C(=O)O RF00953 c1cc(ccc1[N+](=O)[O-])Oc2ccc(cn2)C(F)(F)F SPB03029 c1cc(ccc1SC(=O)c2ccc(o2)Oc3cc(cc(c3)Cl)Cl)Cl SPB03132 CC(c1cc(no1)c2ccc(cc2Cl)Cl)O SPB04879 c1ccc(c(c1)C(=O)O)N2CCOCC2 CC24301 c1cc2c(cc1CNCCn3cnc4c3ncnc4N)OCO2 HTS11197 COc1ccc(cc1)Cc2c(=O)nc3n(nc(n3n2)c4ccc(cc4Cl)Cl)c5ccc(cc5)[N+](=O)[O-] HTS10490 CC1SCC(=O)C(S1)C(=O)OC CD09909 CCOC(=O)c1cnn(c1NC(=O)Nc2ccccc2)c3ccccc3 HTS11498 CCOC(=O)C1=NN(C(=C2C(=O)c3ccccc3C2=O)S1)c4ccccc4 HTS10484 CC(C)(C)NC(=O)C(=O)NC(=O)c1c(cccc1Cl)F RF03987 CN(C)c1ccc(cc1C(=O)O)N CD06952 CC(=O)Nc1ccc(cc1Br)C(C)(C)C RF01504 c1ccc(cc1)CN2CCC3(CC2)Nc4ccccc4S3 HTS09421 c1cc(c(cc1C(F)(F)F)NC(=O)COCC(=O)O)N2CCCC2 HTS09433 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCc4c3cccc4 HTS10623 C/C(=N/Nc1nc2c(n1C/C=C\c3ccccc3)c(=O)n(c(=O)n2C)C)/c4ccc(cc4)Cl HTS11174 c1ccc(cc1)n2c(c(c(n2)c3ccc(cc3)Cl)N=O)N KM09661 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(\C#N)/c3ccccc3 RF00856 CCOC(=O)N1CCC(CC1)NC(=O)c2ccc(cc2)Cl HTS10613 COc1cccc(c1)Cc2nnc(o2)c3ccc4c(c3)nsn4 HTS11122 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(nc2)Oc3c(cccc3Cl)Cl HTS11138 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)Nc3ccc(nc3)Oc4c(cccc4Cl)Cl HTS11140 Cn1c2c(nc1N/N=C/c3ccc4ccccc4n3)n(c(=O)n(c2=O)Cc5ccccc5Cl)C HTS11176 Cc1cc(nn1C)c2nnc(n2c3ccc(cc3)Cl)SCc4ccc(cc4)Cl SPB00766 CCc1ccccc1n2c(nnn2)c3cnccc3C(F)(F)F RF04523 Cc1ccc(cc1)NC(=O)c2cnccc2C(F)(F)F RF04528 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3ccc(nc3)Oc4c(cccc4Cl)Cl HTS09450 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)Oc3c(cccc3Cl)Cl HTS11137 Cc1cc(c(c(c1)Cl)OC(=O)c2c(cccc2Cl)Cl)Cl CD07518 Cc1cc(sc1)C(=O)NN GK01990 c1ccc(c(c1)NC(=O)c2ccnc(c2)N3CCC(CC3)(c4ccc(cc4)Cl)O)N5CCOCC5 HTS10899 CN(C)c1ccc(cc1)NC(=O)c2c(c3ccccc3s2)Cl HTS11007 Cc1cc(cc(c1CN(C)C(=O)c2cnc(cc2C(F)(F)F)Oc3ccccc3)Cl)Cl RF05043 c1cc(ccc1CN2CC(CC2=O)C(=O)Nc3ccc(cc3)Cl)F HTS10900 Cc1ccc(cc1)NC(=O)C2CC(=O)N(C2)Cc3ccc(cc3)F HTS10903 Cc1c(snn1)C(=O)Nc2ccc(cc2)N(C)C HTS11006 CC(=O)c1c(cc(s1)c2ccc(cc2)F)Br GK01958 Cc1c(c(no1)c2ccc(cc2)OC)C(=O)O MO00392 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCCCOC)Cc3cccc4c3cccc4 HTS11187 CCOC(=O)c1cnn(c1NC(=O)CSc2nnc(o2)c3cccs3)c4ccccc4 HTS12388 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccc(cc3)OC HTS10957 Cc1cc(c(c2c1sc(c2C(=O)O)C(=O)OC)C)Cl.NN PD00001 CC(=O)Nc1ccc(cc1Cl)C(C)(C)C RF01505 COC(=O)c1ccc(s1)[N+](=O)[O-] RF01742 Cc1cc(nc2c1c(c(s2)c3nnc(n3CC=C)SCc4ccc(cc4)F)N)C HTS12408 Cc1cc(nc2c1c(c(s2)c3nnc(n3CC=C)SCC(=O)c4ccccc4)N)C HTS12409 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccccc3 HTS10961 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccc(cc3)NC(=O)C HTS10962 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccc(cc3)CC(=O)C HTS10963 CN(C)c1ccc(cc1)NC(=O)Nc2ccccc2 HTS10991 c1ccc2c(c1)C=C(CO2)C(=O)O CC24101 C=CCn1c2c(c(ncn2)Sc3nnc(o3)c4ccc(cc4)Cl)sc1=S HTS12634 C/C(=N\NC(=S)N)/c1cc(cc(c1O)Cl)Cl CD03802 c1c(cc(c(c1[N+](=O)[O-])NNC(=O)C2CC=CC2C(Cl)Cl)[N+](=O)[O-])C(F)(F)F CD03799 c1ccc2c(c1)N(C(=O)CS2)CC(=O)N/N=C/c3cccs3 HTS13164 c1ccc(cc1)Cn2c(n[nH]c2=S)CN3c4ccccc4SCC3=O HTS13166 CCOC(=O)C1=NN(C2C1C(=O)N(C2=O)c3ccccc3)c4cccc(c4)Cl HTS12230 c1cnccc1c2nnc3n2C(=O)CS3 HTS13242 Cc1ccc(cc1)NC(=O)C2CC(=O)N(C2)Cc3ccco3 HTS11013 c1ccc(cc1)Cn2c(cnc2S)CO MO00213 CCN(CC)CC(=O)Nc1c(cnn1c2ccccc2)C#N HTS12638 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccccc3)CCC2C(=O)OCC HTS12637 c1cc(sc1)c2cc(no2)CO CC23109 Cc1nc(cs1)c2cc(no2)CO CC14009 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2ccc(cc2)C#N HTS10936 CC(C)(C)c1ccc(cc1)NC(=O)NCc2ccc(cc2)C#N HTS10937 c1ccc(cc1)COc2ccc(cc2)NC(=O)NCc3ccc(cc3)C#N HTS10938 c1ccc(cc1)c2cc3c(s2)[nH]c(=O)n(c3=O)c4cccc(c4)Cl HTS13147 CC1CC(CC(C1)(C)C)NC(=O)C(=O)Nc2cccc(c2)C(F)(F)F JPV00093 CCCc1c(nc(nc1OC(=O)N(C)C)SCc2c(cccc2Cl)F)C RJF00100 Cn1c2c(nc1N3CCc4ccccc4C3)n(c(=O)n(c2=O)C)C HTS11189 CCCNc1nc2c(n1Cc3cccc4c3cccc4)c(=O)n(c(=O)n2C)C HTS11193 Cn1c2c(nc1Oc3cccc4c3nccc4)n(c(=O)n(c2=O)C)C HTS11194 CCOC(=O)c1cc(sc1NC(=O)Nc2ccc(cc2)C)c3ccccc3 HTS13153 CCOC(=O)c1cc(sc1NC(=O)Nc2ccc(c(c2)Cl)Cl)c3ccccc3 HTS13155 c1cc(ccc1SCc2nnc(o2)c3cc(cc(c3)Cl)Cl)Cl SPB01784 CC(=O)c1c(c2c(s1)nsc2SCCN3CCCC3)N HTS13178 c1ccc(cc1)c2cn(c(n2)SCC(=O)NC(=O)Nc3ccccc3)c4ccccc4 HTS13189 COc1cccc(c1)n2cc(nc2SCC(=O)c3cccs3)c4ccc(cc4)F HTS13191 c1cc(c(cc1NC(=S)Nc2ccc(c(c2)Cl)F)Cl)F RJF00159 CCOC(=O)c1cc(sc1NC(=O)Nc2ccccc2)c3ccccc3 HTS13151 CCOC(=O)c1c(cc(nc1O)C)O SEW00539 CSc1nc(nn1CCC#N)N CD10145 CC(C)c1ccc(cc1)NC(=N)NC(=N)N.Cl RJF00585 CN(C)NC(=O)c1ccc(o1)Oc2ccc(cc2Cl)Cl JM00117 c1ccc2c(c1)N(C(=O)CS2)CC(=O)N/N=C/c3ccc(cc3Cl)Cl HTS13159 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)c2cccnc2Oc3ccc(cc3)Cl HTS10672 COc1cccc(c1)CC(=O)NNC(=O)c2ccc3c(c2)nccn3 HTS10676 COc1cccc(c1)Cc2nnc(o2)c3ccc4c(c3)OCO4 HTS11120 c1cc(c(cc1OCC(F)(F)F)C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OCC(F)(F)F RF04507 c1cc(ccc1NC(=O)c2cnccc2C(F)(F)F)F RF04521 c1cc(sc1)c2cc([nH]c(=O)c2C#N)c3cccs3 HTS12392 c1cc(ccc1C#N)C2Nc3ccc(cc3C(=O)N2)[N+](=O)[O-] BTB05571 c1ccc(c(c1)CO)N2CCOCC2 CC24309 CC(C)(C)c1ccc(cc1)c2nnn(n2)CC(=O)NN SPB01128 c1ccc2c(c1)nc(s2)N/N=C/c3cccs3 HTS12643 CCOC(=O)C1(C(C(=NN1c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3Cl)Cl)c4ccccc4)C#N HTS10491 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N(C)Cc3ccccc3)Cc4ccccc4Cl HTS11167 C1CSCCN1C/C(=N/O)/N CD08263 CC(C)(C)c1ccc(cc1)C(=O)Oc2c(cncc2Cl)Cl RF01221 CC(C)(C)OC(=O)C(C)(C)ONC(=O)Nc1cc(cc(c1)Cl)Cl RF04667 c1cc(cc(c1)C(F)(F)F)c2nn(c(=O)o2)c3c(cccn3)C(F)(F)F RF04895 CC(=O)N1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)OC HTS12424 c1ccc2c(c1)CCC3C2=NN(C3c4cccs4)C(=O)Nc5ccc(cc5)Cl HTS12428 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccc(cc3)C HTS10959 Cc1ccc(cc1)S(=O)(=O)NC(=O)OCC2CN(CCO2)Cc3ccccc3 HTS11076 c1ccc(cc1)C2=N/C(=C/c3ccco3)/C(=O)N2 RG00111 CCOC(=O)c1ccc(c(c1)N)N.Cl.Cl RDP00141 c1ccc(c(c1)C(=O)O)SC(CC(=O)c2cccc(c2)F)c3ccc(cc3)F PD00282 Cc1cccc2c1N(CCC2)C(=O)Nc3cccs3 HTS09417 CC(C)S(=O)(=O)c1csc(c1N)C(=O)Nc2ccc(cc2)OC HTS10255 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C(=N/OC(=O)/C=C/C(=O)O)/N CD04514 Cc1nc(nc(n1)OC)NC(=O)NC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F RF04516 Cc1cc(nc2c1c(c(s2)c3nnc(n3Cc4ccccc4)SC)N)C HTS12412 CCOC(=O)CSc1nnc(n1C)c2c(c3c(cc(nc3s2)C)C)N HTS12413 c1ccc2c(c1)CCC3C2=NN(C3c4ccc(cc4)F)C(=O)CN5CCCCC5 HTS12430 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccc(cc3)C#N HTS10960 Cn1c2ccc(cc2nn1)CO CC23509 c1ccc(cc1)N2CCN(CC2)c3ncc(c(n3)N)C#N HTS12599 c1c(c(nc(n1)N2CCCCC2)N)C#N HTS12600 c1ccc2c(c1)CCN2C(=O)C(Cc3ccccc3Cl)C(=O)N4CCc5c4cccc5 HTS12603 Cc1c(cccc1Cl)NC(=S)NCCc2ccccn2 S04490 c1ccn(c1)c2cccc(c2)CO CC21909 Cc1cc(nc2c1c(c(s2)c3nnc(n3Cc4ccccc4)SCC(=O)C)N)C HTS12410 c1ccc2c(c1)CCN2C(=O)CN3CCOCC3 HTS12464 c1ccc(cc1)n2c(nnc2SCC(=O)N)Cn3c4ccccc4nn3 HTS12468 c1ccc(c(c1)CSc2nnc3n2CCCN3C(=O)c4cccs4)Cl HTS12640 CCN(CC)CC(=O)Nc1c(c2c(s1)CN(CC2)C(=O)OCC)C(=O)OCC HTS12642 c1ccc2c(c1)-n3c(nn(c3=O)CC(=O)c4cccs4)CS2 HTS13172 CC(C)(C)C(=O)Nc1cc(ccc1N2CCC(CC2)C(F)(F)F)C(F)(F)F SPB06390 Cc1c(c(on1)C)S(=O)(=O)N2CCN(CC2)C(=O)C3CCCO3 HTS10893 c1cc(cnc1)C(=O)C(CC(=O)c2ccc(cc2)Cl)c3cccs3 RG00073 c1ccc(cc1)c2cc3c(s2)[nH]c(=O)n(c3=O)c4ccccc4 HTS13150 COc1cccc(c1)C(=O)c2c(c3c(s2)nsc3SCc4ccc(cc4)F)N HTS13177 CC(=O)c1c(c2c(s1)nsc2SCCN3CCOCC3)N HTS13179 CCOC(=O)c1cc(sc1NC(=O)CSc2[nH]c3ccccc3n2)c4ccccc4 HTS13143 CCOC(=O)c1cc(sc1NC(=O)CN2CCN(CC2)C)c3ccccc3 HTS13145 CCOC(=O)c1cc(sc1NC(=O)Nc2ccc(cc2)Cl)c3ccccc3 HTS13152 c1cc(ccc1CN2CC(CC2=O)C(=O)O)F MO00127 Cc1cccc(c1)/C(=N/[N+](C)(C)C)/N=C(/Nc2ccc(c(c2)Cl)Cl)\[S-] MBE00065 c1ccc2c(c1)N(C(=O)CS2)CC(=O)N/N=C\c3ccc4c(c3)OCO4 HTS13157 COc1cccc(c1)NC(=O)Nc2ccc(nc2)Oc3c(cccc3Cl)Cl HTS09444 c1ccc(c(c1)C(=O)O/N=C(/c2ccc(cc2)[N+](=O)[O-])\N)Cl BTB04195 c1ccc(cc1)Cc2n[nH]c(=S)n2C3CCCCC3 HTS12440 c1cc(ccc1C(=O)c2c(c3c(s2)nsc3SCCN4CCOCC4)N)Cl HTS13182 c1ccc(cc1)n2c(ccn2)C(=O)O CC24501 c1ccc2c(c1)N(C(=O)CS2)CC(=O)N/N=C/c3ccco3 HTS13163 CCOC(=O)c1c2c(sc1NC(=O)CN3CCc4c3cccc4)CN(CC2)C(=O)OCC HTS12641 CCOc1c(c(c2c(n1)-c3ccccc3C2)c4cccs4)C#N HTS12444 c1ccc(cc1)C(=O)c2c(c3c(c4c(nc3o2)-c5ccccc5CC4)c6ccco6)N HTS12447 CCOC(=O)c1c2nc(c3ccccc3n2nn1)SCC(=O)N HTS12450 COc1ccc(cc1OC)CCNC(=S)Nc2cc(cc(c2)Cl)Cl RJF00147 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)N3CCN(CC3)C(=O)C4CCCO4 HTS10894 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CCN(CCO)Cc3ccccc3 HTS11168 COc1ccc(cc1)C2=NOC(C2)COc3ccc(cc3)[N+](=O)[O-] HTS11172 c1cc(sc1)CNC(=O)NCc2cccs2 HTS12605 CCOC(=O)c1cnn(c1NC(=O)CSc2nnc(n2c3ccccc3)c4cccs4)c5ccccc5 HTS12389 c1ccc2c(c1)CCN2C(=O)CN3CCCC3 HTS12461 c1ccc(cc1)N2CCN(CC2)CC(=O)N3CCc4c3cccc4 HTS12462 CN1CCN(CC1)CC(=O)N2CCc3c2cccc3 HTS12463 c1c(c(cc(c1Cl)Cl)Cl)NC(=N)NC(=N)N.Cl RJF00666 Cn1c2c(nc1N/N=C/c3ccc(cc3)Br)n(c(=O)n(c2=O)Cc4cccc(c4)F)C HTS11177 CN(Cc1ccc(cc1OC)OC)C(=O)c2cnc(cc2C(F)(F)F)OC RF04478 c1ccc(cc1)CN2CCOC(C2)COC(=O)Nc3ccc(cc3)OCc4ccccc4 HTS11075 CC(C)N(Cc1ccccc1)S(=O)(=O)c2cccs2 HTS07914 Cn1c2ccc(cc2nn1)C(=O)O CC23501 c1ccc(cc1)c2cc(cnc2)C(=O)O CC24201 C1C(=O)N=C(S1)CC(=O)N CD09799 CC(C)(C)S(=O)(=O)c1cn[nH]c1N KM08647 CSC(=C(C#N)C(=O)c1cccc(c1)[N+](=O)[O-])SC KM01802 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4cccs4)C HTS12394 Cc1cc(nc2c1c(c(s2)C(=O)c3ccc(cc3)Cl)NC(=O)C)C HTS12396 CN(C)c1ccc(c(c1)SCc2cccc(c2)C(F)(F)F)C3=NCCCN3.Cl CD03649 Cc1cccc(c1n2c(nnn2)c3cnccc3C(F)(F)F)C RF04549 CCOC(=O)c1cn[nH]c1NC(=S)NCc2ccccc2 HTS12500 CCOC(=O)c1cn[nH]c1NC(=S)Nc2ccc(cc2)Cl HTS12503 CCOC(=O)c1cn[nH]c1NC(=S)Nc2cccc(c2)C(F)(F)F HTS12504 c1ccc2c(c1)nnn2Cc3n[nH]c(=S)o3 HTS12508 c1ccc2c(c1)CCC3C2=NN(C3c4ccc(cc4)F)C(=O)c5ccc(cc5)F HTS12427 CC(=O)CSc1nc2ccccc2s1 RF00504 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2C(=O)Nc5ccc(c(c5)Cl)Cl HTS12429 c1ccc(cc1)Cc2n[nH]c(=S)n2Cc3ccccc3 HTS12437 c1ccc(cc1)Cn2c(=O)n-3c(n2)CSc4c3cccc4 HTS13171 COc1cccc(c1)C(=O)CSc2c(c(sn2)SCC(=O)c3cccc(c3)OC)C#N HTS13185 c1cc(ccc1C(=O)CSc2c(c(sn2)SCC(=O)c3ccc(cc3)Cl)C#N)Cl HTS13186 CCOC(=O)CSc1nc(cn1c2ccccc2)c3ccccc3 HTS13188 CCOc1cc(nc(n1)c2csc(n2)C)C SPB04581 CCn1c(nnc1SCC(=O)Nc2c(cnn2c3ccccc3)C(=O)OCC)c4cccs4 HTS12387 c1ccc2c(c1)CCN2C(=O)CSc3nnc(o3)c4ccncc4 HTS12496 c1ccc(cc1)c2c(nnc(n2)SCC(=O)N3CCc4c3cccc4)c5ccccc5 HTS12498 c1ccc(cc1)Cn2c(n[nH]c2=S)c3ccc(cc3)Cl HTS12533 C=CCC(C(=O)N1CCc2c1cccc2)C(=O)N3CCc4c3cccc4 HTS12537 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2C(=O)c5cccs5 HTS12425 c1ccc2c(c1)CCC3C2=NN(C3c4ccc(cc4)F)C(=O)c5ccco5 HTS12426 c1ccc(cc1)C2C3=C(c4ccccc4CC3)N=C5N2C(=O)CS5 HTS12433 c1ccn2cc(nc2c1)c3cccc(c3)N RDR01518 Cc1ccc(cc1)n2c(=O)c3cc(sc3[nH]c2=O)c4ccccc4 HTS13146 c1ccc(cc1)c2cc3c(s2)[nH]c(=O)n(c3=O)c4ccc(cc4)Cl HTS13149 c1ccc(cc1)Cc2n[nH]c(=S)n2c3cccc(c3)C(F)(F)F HTS12438 c1ccc(cc1)C2=NN(/C(=C\3/C(=O)N(C(=S)N3c4ccccc4)c5ccccc5)/S2)c6ccccc6 HTS12200 CCOC(=O)c1cc(sc1NC(=O)CN2CCOCC2)c3ccccc3 HTS13142 c1cc(ccc1c2n[nH]c(=S)o2)Cl HTS12509 c1cc(oc1)c2n[nH]c(=S)o2 HTS12510 CN1CCN(CC1)c2ncc(c(n2)N)C#N HTS12513 CCOC(=O)c1cc(sc1NC(=O)CN2CCCCC2)c3ccccc3 HTS13144 CCOC(=O)c1cc(sc1NC(=O)Nc2cccc(c2)Cl)c3ccccc3 HTS13154 CCn1c(n[nH]c1=S)Cc2ccccc2 HTS12436 c1ccc2c(c1)CCC3=C2N=C4N(C3c5cccs5)C(=O)CS4 HTS12434 c1ccc(c(c1)C(=O)NN)Br RDP00172 CCOc1c(c(=O)c1=O)Nc2ccccc2C(=O)O RDP00175 c1cc(c(c(c1)Cl)Cl)/N=C\2/N(C(=O)CS2)Cc3cccnc3 S04489 C=CCSc1nnc2n1CCCN2 HTS11916 Cc1c(n2ccsc2n1)C(=O)NN MO00121 c1ccc2c(c1)N(C(=O)CS2)CC(=O)N/N=C/c3ccc(cc3)F HTS13160 c1ccc2c(c1)N(C(=O)CS2)CC(=O)N/N=C/c3cccnc3 HTS13161 COc1cc(cc(c1OC)OC)/C=N/NC(=O)CN2c3ccccc3SCC2=O HTS13162 CC(=O)C1=NN(C2(S1)N(C(=O)CS2)c3ccccc3)c4ccc(cc4)Cl HTS12215 Cc1ccc(cc1)c2c(c-3n(c2C(=O)c4cccs4)CCc5c3cc(c(c5)OC)OC)C#N HTS12227 c1c(cc(cc1Cl)Cl)Nc2n[nH]c(=S)s2 S04532 Cn1c(nnc1Sc2c3c(c(c4n2c5ccccc5n4)C#N)CCC3)c6ccccc6 HTS11914 COc1cccc(c1)/C=N/NC(=O)CN2c3ccccc3SCC2=O HTS13156 Cc1ccc(o1)/C=N/NC(=O)CN2c3ccccc3SCC2=O HTS13158 CN(C)c1ccc(cc1)/C=C/2\C(=O)NC(=S)S2 RDP00176 CCOC(=O)c1c(cn(n1)c2ccc(cc2)C)C#N HTS12207 c1ccc(cc1)NC(=O)c2c(nn(c2N)c3ccc(cc3)[N+](=O)[O-])c4cccs4 HTS12212 Cc1ccc(cc1)N2C3(N(C(=O)CS3)c4ccccc4)SC(=N2)C(=O)c5ccccc5 HTS12214 c1ccc(c(c1)/C=N/c2ccc(cc2)N3CCOCC3)O S04547 c1ccc(cc1)c2n[nH]c(=S)n2/N=C/c3cccs3 HTS12519 CNC(=O)NC(=O)CSc1nnc(n1c2ccc(cc2)Cl)Cc3ccccc3 HTS12520 CCOc1ccc2c(c1)sc(n2)/N=C/c3ccccc3O S04540 c1ccc(c(c1)/C=N/c2ccc(cc2)S(=O)(=O)Nc3ncccn3)O S04544 Cc1nc2c(c(=O)n1/N=C/c3ccccc3)sc(=S)n2C HTS11915 Cc1nc(cs1)c2ccccc2.Br CD00563 CCOC(=O)CSc1nnc(n1c2ccccc2)c3ccncc3 HTS11938 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)C(c4c([nH]c(=S)[nH]c4=O)N)c5c([nH]c(=S)[nH]c5=O)N HTS11941 c1ccc(cc1)CN(Cc2ccccc2)c3ncc(c(n3)N)C#N HTS12514 Cc1cc(cc(c1F)C)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ccc(cc3F)F RJF00783 c1ccc2c(c1)CCN2c3ncc(c(n3)N)C#N HTS12515 CNC(=O)NC(=O)Cn1c(=O)n-2c(n1)CSc3c2cccc3 HTS13174 c1cc(sc1)c2n[nH]c(=S)n2C3CCCCC3 HTS12530 c1ccc(cc1)c2n[nH]c(=S)n2N HTS12534 CC1(CC2=C(C(C3=C(N2)CC(CC3=O)(C)C)c4ccc(c(c4)Cl)Cl)C(=O)C1)C S04453 c1ccc(c(c1)c2cc([nH]n2)c3cc(cc(c3O)Cl)Cl)Cl RG00070 c1cc(c(nc1)N2CCOCC2)N CC24614 Cc1ccccc1n2cc(nc2SCC(=O)N)c3ccc(cc3)Br HTS13192 CCn1c(nnc1SCC(=O)NC(=O)Nc2ccccc2)c3ccco3 HTS12523 CNC(=O)NC(=O)CSc1nnc(n1Cc2ccccc2)c3ccncc3 HTS12526 c1ccc(cc1)C(=O)c2c(c3c(s2)nsc3SCCN4CCOCC4)N HTS13183 c1ccc2c(c1)c(=O)n(c(n2)SCc3c(cccc3Cl)F)c4ccc(cc4F)F RJF00114 CCNC(=S)Nc1cc(cc(c1)Cl)Cl RJF00125 CC(=O)c1ccc(c(c1)CSc2nnc(n2Cc3ccco3)c4ccc(cc4)C(F)(F)F)OC HTS11112 c1ccc2c(c1)CCCN2C(=O)c3ccc(cc3)C(=O)N4CCCc5c4cccc5 HTS10621 CCOC(=O)c1c2nc(c3ccccc3n2nn1)Sc4nnc(n4C)c5ccncc5 HTS12552 c1ccc(cc1)c2cc3c(s2)ncnc3SCC(=O)c4cccs4 HTS13193 c1ccc(cc1)C(=O)Oc2cc(=O)oc3c2c(=O)n4c5c3cccc5CCC4 HTS12597 c1ccc(cc1)c2n[nH]c(=S)n2/N=C/c3ccc(cc3)Cl HTS12517 C=CCn1c(nnc1SCC(=O)NC(=O)Nc2ccccc2)c3ccc(cc3)Cl HTS12522 c1cc(cnc1)CNC(=S)Nc2ccc(cc2)Cl S04483 c1cc(cnc1)CN\2C(=O)CS/C2=N\c3ccc(cc3)Cl S04485 COc1ccc(cc1)/C=N/N2C(=N/C(=C\c3cccs3)/C2=O)c4ccccc4 HTS13203 c1ccc(cc1)c2c(nnc(n2)N3CCN(CC3)c4ccccc4)c5ccccc5 HTS12481 CC(=O)CN1C(=N/C(=C\c2cc(c(c(c2)OC)OC)OC)/C1=O)c3ccccc3 HTS13211 COc1cccc(c1)CC(=O)NNC(=O)c2ccc(s2)c3cccs3 HTS10669 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2cccc3c2nsn3 HTS10679 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)c4cccs4)N)c5ccco5 HTS12399 Cc1ccc2c(c1)c3c(c(n2)C)CCN3c4ccccc4 HTS12384 Cc1cc(n(n1)c2ccccc2)NC(=O)CN3CCCCC3 HTS12385 C=CCn1c(=O)n-2c(n1)CSc3c2cccc3 HTS13226 C=CCSc1c(c(sn1)SCC(=O)c2ccc(cc2)[N+](=O)[O-])C#N HTS13229 c1ccc(cc1)C2C3CCc4ccccc4C3=NN2c5ccccc5 HTS12419 CC(=O)N1C(C2CCc3ccccc3C2=N1)c4cccs4 HTS12421 CCOC(=O)Cn1nc(nn1)Cc2c(cccc2Cl)Cl RJF00343 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)Cl)/C(=O)N2Cc4ccc(cc4)Cl HTS13212 CCOC(=O)Cn1c(=O)n-2c(n1)CSc3c2cccc3 HTS13173 c1ccc(cc1)COc2ccc(cc2)/C=C/3\C(=O)N(C(=N3)c4ccccc4)CC(=O)c5cccs5 HTS13213 CCOC(=O)CSc1nc(c(nn1)c2ccccc2)c3ccccc3 HTS12487 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCC(=O)N HTS12488 Cn1c(=S)nc2c(n1)c3ccccc3n2CC(=O)c4ccc(cc4)Br HTS12604 C/C(=N\NC(=O)CN1c2ccccc2SCC1=O)/c3ccco3 HTS13223 CCn1c(n[nH]c1=S)CN2c3ccccc3SCC2=O HTS13224 Cc1cc(nc2c1c(c(s2)c3nnc(n3C)SCc4ccc(cc4)[N+](=O)[O-])N)C HTS12414 CC(=O)N1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)Cl HTS12423 Cc1cc(nc2c1c(c(s2)c3nnc(n3Cc4ccccc4)SCc5ccccc5)N)C HTS12411 c1ccc(cc1)N2CCN(CC2)CC(=O)N3C(C4CCc5ccccc5C4=N3)c6cccs6 HTS12431 COc1cc2c(cc1OC)C(=O)N(CC2)Cc3c(cccc3Cl)Cl GK02021 c1ccc(cc1)c2cn(c(n2)SCc3n[nH]c(=S)n3c4ccccc4)c5ccccc5 HTS13237 CCOC(=O)c1cnc(nc1N)N2CCOCC2 HTS13239 c1ccn2c(c1)nnc2S MO07000 c1cc(c(c(c1)Cl)Cc2nnn(n2)CC(=O)NN)Cl RJF00344 CCOC(=O)c1c2nc(c3ccccc3n2nn1)SCC(=O)C HTS12453 CCOC(=O)C1=NN(C2C1C(=O)N(C2=O)c3ccc(cc3)OC)c4ccc(cc4)Cl HTS12232 CCOC(=O)c1c2nc(c3ccccc3n2nn1)SCc4ccc(cc4)[N+](=O)[O-] HTS12456 CCOC(=O)c1c(c2c(=O)n(c(=S)n(c2s1)c3ccccc3)c4ccccc4)O HTS11918 COc1ccc(c(c1)OC)n2cc(nc2SCc3n[nH]c(=S)n3CC=C)c4ccccc4 HTS13233 c1ccc2c(c1)CCC3=C2N=C4N(C3c5ccccc5Cl)C(=O)CS4 HTS12435 COc1ccc(cc1)c2c3cc(ccc3no2)Br SCR00095 Cc1cccc(c1NC(=S)SCC(=O)N)C RF00463 c1cc2c(c(c1)C(F)(F)F)NC(=O)C2=O RF00952 c1ccc(cc1)C(Cc2cccnc2)(c3ccccc3)O.Cl RF00993 COc1ccc(cc1)/C=C/2\C(=O)N(NC(=N2)c3ccccc3)Cc4ccccc4 HTS13240 c1cc(cc(c1)C(=O)O)c2cccs2 MO07003 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4cccnc4)C HTS12395 Cc1cc(nc2c1c3c(s2)c(=O)n(nn3)/N=C/c4cccc(c4)OC)C HTS12397 CCOC(=O)c1c(c2c(cc(nc2s1)C)C)NC(=O)Nc3ccc(cc3)Cl HTS12398 CC1=C(C(NC(=S)N1)c2ccc(cc2)Cl)C(=O)OC HTS12458 Cc1ccc(cc1)n2c3nc(=O)c(nn3c(n2)C(=O)c4cccs4)Cc5ccc(cc5)OC HTS12266 c1ccc(cc1)Cc2c(=O)nc3n(nc(n3n2)C(=O)c4ccccc4)c5cccc(c5)Cl HTS12267 c1ccc(cc1)C(=O)c2nn(c3n2nc(c(=O)n3)Cc4ccc(cc4)Cl)c5ccccc5 HTS12268 CC1CCc2c(sc3c2c4nncn4cn3)C1 HTS11932 CCOC(=O)c1cnn(c1NC(=O)CSc2nc3ccccc3o2)c4ccccc4 HTS12390 CCOC(=O)c1cnn(c1NC(=O)CSc2nc3ccccc3s2)c4ccccc4 HTS12391 c1ccc(cc1)C(=O)COc2c(c(cc(n2)c3ccc(cc3)[N+](=O)[O-])c4cccs4)C#N HTS12393 c1cnc(nc1C(F)(F)F)N2CCC(CC2)C(=O)O AW01250 Cc1cc(nc2c1c(c(s2)c3nnc(n3CC=C)SCc4ccccc4Cl)N)C HTS12407 CCOc1ccc(cc1)NC(=O)C2CCN(CC2)C(=O)C SCR00123 c1cc(cnc1)/C=N/NC(=O)c2c(c3c(cc(nc3o2)c4ccco4)c5ccco5)N HTS12400 c1ccc(c(c1)Cn2c3c(c(ncn3)N/N=C/c4cccs4)nn2)Cl HTS12404 c1ccc(c(c1)/C=N/c2ccc(cc2)S(=O)(=O)Nc3nccs3)O S04541 Cc1cc(no1)C(=O)NN SPB01196 c1cc(cnc1)/C=N/n2c(n[nH]c2=S)c3ccc(cc3)Cl HTS12518 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])Oc2ccc(cc2)C3SCCS3 SPB01878 CC(=O)c1ccc(c(c1)/N=C/c2cc(ccc2O)Br)Cl CD03530 CC(=O)c1c(c2c(s1)nsc2SCCN3CCCCC3)N HTS13175 c1cc(sc1)C(=O)c2c(c3c(s2)nsc3SCCN4CCCCC4)N HTS13176 c1cc(oc1)C(=O)c2c(c3c(s2)nsc3SCCN4CCOCC4)N HTS13228 CCn1c(n[nH]c1=S)CSc2nc(cn2c3ccc(cc3)C)c4ccc(cc4)Cl HTS13234 CNC(=O)NC(=O)CSc1nnc(n1c2ccc(cc2)Cl)c3cccs3 HTS12527 c1ccc2c(c1)C(OC2=O)CC(=O)c3cc(ccc3Cl)Cl S04567 c1ccc2c(c1)[nH]c(n2)Sc3c4c5c(sc4ncn3)CCCC5 HTS11936 CC(=O)N1CCC(CC1)C(=O)Nc2nc3ccc(cc3s2)Cl SCR00104 c1ccc(c(c1)/N=C/2\NC(=O)C(S2)CC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl S04555 c1cc(oc1)c2n[nH]c(=S)n2c3ccc(cc3)F HTS12561 CCOC(=O)c1cc(sc1NC(=O)CN2CCCC2)c3ccccc3 HTS13222 CC(=O)Cn1c(=O)n-2c(n1)CSc3c2cccc3 HTS13227 c1cc(ccc1C2CCCCC2)OC(=O)c3ccc(cc3)Cl S06077 CNC(=O)NC(=O)CSc1nnc(n1CC=C)c2ccncc2 HTS12521 c1ccc(c(c1)/C=N/c2ccc(cc2)S(=O)(=O)/N=C/c3ccccc3O)O S04542 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)OC)Cl)[N+](=O)[O-] BTB07725 c1cc(ccc1CN2CCS(=O)(=O)CC2)N MO00124 CCOC(=O)CSc1nc(cn1c2ccc(cc2)C)c3cccs3 HTS13187 CCOC(=O)c1cnn2c1[nH]c3c(c2=O)CCCC3 HTS12473 CCOC(=O)c1cnn2c1[nH]c(cc2=O)C HTS12474 c1ccc(cc1)c2c(nnc(n2)N3CCCC3)c4ccccc4 HTS12479 COc1ccc(cc1Br)C(CC(=O)c2ccc(cc2)F)CC(=O)c3ccc(cc3)F S04423 COc1ccc(cc1)/C=C\2/C(=O)N(C(=N2)c3ccccc3)/N=C/c4ccc5c(c4)OCO5 HTS13201 c1ccc(cc1)n2c(nnc2SCC(=O)c3ccc(cc3)Cl)Cn4c5ccccc5nn4 HTS12469 CCOC(=O)CSc1nnc(n1c2ccc(cc2)F)Cn3c4ccccc4nn3 HTS12470 CCn1c(nnc1SCC(=O)c2ccc(cc2)Br)Cn3c4ccccc4nn3 HTS12472 c1cc(c(c(c1)Cl)C(=O)NC(=O)NCCc2ccc(cc2)Cl)Cl BTB04896 CCOc1c(c(c2c(n1)-c3ccccc3C2)c4ccc(cc4)F)C#N HTS12441 COc1c(c(c2c(n1)-c3ccccc3C2)c4ccccc4Cl)C#N HTS12442 CCOc1c(c(c2c(n1)-c3ccccc3C2)c4ccc(cc4)OC)C#N HTS12443 c1cc(c(nc1)N2CCOCC2)CO CC24609 c1cc(cnc1)CNC(=S)Nc2cc(cc(c2)Cl)Cl RJF00168 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3c(onc3c4ccccc4)C)C HTS11101 c1ccc(cc1)c2cc3c(=O)n(c(=O)n(c3s2)CC(=O)N)c4cccc(c4)Cl HTS13220 c1ccc(cc1)C2=N/C(=C\c3ccco3)/C(=O)N2/N=C/c4ccc(cc4)F HTS13200 c1ccc(cc1)c2cc3c(ncnc3s2)Nc4ccccc4 HTS13216 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)F)/C(=O)N2CC(=O)c4ccco4 HTS13214 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)Cc5cc(cc6c5OCOC6)Cl HTS10663 CCOC(=O)c1c2nc(c3ccccc3n2nn1)SC(C(=O)C)C(=O)OCC HTS12452 CCOC(=O)c1c2nc(c3ccccc3n2nn1)SCc4ccccc4Cl HTS12455 c1ccc2c(c1)CCN2CC(=O)N3CCc4c3cccc4 HTS12459 c1ccc2c(c1)CCC3C2=NN(C3c4ccccc4Cl)C(=O)c5cccs5 HTS12420 Cc1c2c(c3cc(ccc3n1)F)N(CC2)c4ccccc4 HTS12383 Cn1ccnc1SCC(=O)N2CCc3c2cccc3 HTS12492 c1ccc2c(c1)c3c([nH]2)nc(nn3)SCc4ccc(cc4)F HTS12490 CNC(=O)NC(=O)CSc1nc(cn1c2ccccc2)c3ccc(cc3)Cl HTS13230 c1ccc(cc1)c2cn(c(n2)SCC(=O)NN)c3ccccc3 HTS13231 C=CCn1c(n[nH]c1=S)c2cccs2 HTS12529 COc1ccc(cc1)n2c(nnc2SCC(=O)NC(=O)Nc3ccccc3)c4cccs4 HTS12528 COc1ccc(cc1)n2c(n[nH]c2=S)c3cccs3 HTS12531 c1ccc(cc1)Cc2n[nH]c(=S)n2c3ccc(cc3)Cl HTS12439 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=O)Cc3ccccc3 HTS12445 c1ccc(cc1)NC(=O)NC(=O)Cn2c(=O)n-3c(n2)CSc4c3cccc4 HTS13170 COc1ccc(cc1)/C=C(/C(=O)N/N=C/c2ccc3c(c2)OCO3)\NC(=O)c4ccccc4 HTS13206 CCOC(=O)COc1c2c(=O)n(c(=S)n(c2sc1C(=O)OCC)c3ccccc3)c4ccccc4 HTS11920 c1cc(sc1)c2n[nH]c(=S)n2c3ccc(cc3)Cl HTS12601 Cc1cc(n(n1)c2ccccc2)NC(=O)CN3CCOCC3 HTS12386 c1ccc2c(c1)-n3c(nn(c3=O)CC(=O)NN)CS2 HTS13225 Cn1c(nnc1SCC(=O)NC(=O)Nc2ccccc2)c3ccncc3 HTS12524 Cc1cc(nc2c1c(c(s2)c3nnc(n3C)SCc4ccc(cc4)Cl)N)C HTS12415 CC(=O)N1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)F HTS12422 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3cccc(c3)F HTS10956 Cc1ccc(cc1)n2cc(c(n2)C(=O)c3cccs3)C#N HTS12206 c1ccc(cc1)N2C(=O)CSC23N(N=C(S3)C(=O)c4cccs4)c5ccc(cc5)Cl HTS12213 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)[N+](=O)[O-])/C=N/n4c(n[nH]c4=S)c5ccncc5 HTS11973 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)/C=N/n4c(n[nH]c4=S)c5ccncc5 HTS11974 c1cc(sc1)c2nnc3n2N=C(CS3)c4ccc(cc4)Cl HTS11978 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3CC=C)c4ccc(cc4)Cl HTS12036 CCN(CC)C(=O)Sc1c(cc(cc1Br)Br)Br S06006 CCOC(=O)c1cn[nH]c1NC(=S)Nc2ccccc2 HTS12501 c1ccc2c(c1)CCN2C(=O)CSc3[nH]c4ccccc4n3 HTS12499 CCOC(=O)c1cn[nH]c1NC(=S)Nc2ccc(cc2)OC HTS12502 COc1cc2c(cc1OC)-c3c(c(c(n3CC2)C(=O)c4cccs4)c5ccc(cc5)Cl)C#N HTS12226 CC(=O)C1=NN(C2C1C(=O)N(C2=O)c3ccccc3)c4cccc(c4)Cl HTS12229 c1ccc(cc1)C2=Nn3c(nnc3SC2)c4cccs4 HTS11979 c1ccc(cc1)c2ccc(cc2)C3=Nn4c(nnc4SC3)c5cccs5 HTS11980 c1ccc(cc1)C(=O)c2c(c3c(s2)nsc3SCCN4CCCC4)N HTS13184 CC(=O)CSc1nc(cn1c2cccc(c2)OC)c3ccc(cc3)F HTS13190 c1ccc(cc1)c2cc3c(s2)[nH]c(=O)n(c3=O)c4ccc(c(c4)Cl)Cl HTS13148 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)[N+](=O)[O-])/C=N/n4c(n[nH]c4=S)c5cccs5 HTS11987 CC(=O)c1ccc(cc1)N2C(=O)CSC2=S S06019 c1ccc2c(c1)c(cs2)NC(=O)Nc3ccncc3 HTS12332 Cc1cc(no1)CNC(=O)Nc2csc3c2cccc3 HTS12348 CCOC(=O)c1c(cn(n1)c2cccc(c2)Cl)C#N HTS12360 CC(=O)N1C(OC(=N1)c2ccncc2)c3cn(nc3c4ccc(cc4)[N+](=O)[O-])c5ccccc5 HTS11989 c1ccc(cc1)n2cc(c(n2)c3cccs3)/C=N/NC(=O)c4ccncc4 HTS11991 Cc1c(n2ccccc2n1)C(=O)NNC(=S)Nc3ccccc3 HTS11912 Cc1c(cn(n1)c2ccccc2)/C=N/N=C/3\NC(=O)CS3 HTS11921 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/N=C/4\NC(=O)CS4 HTS11922 c1cc2c(cc1c3csc(n3)c4ccc5c(c4)OCCO5)OCCO2 SCR00135 c1ccc(cc1)Oc2ccc(cc2)NC(=O)/C=C/C(=O)O S01648 c1cc(oc1)CN2CN(C(=S)SC2)Cc3ccco3 S01962 CC(=O)Nc1cccc(c1)CCCC(=O)O TL00756 c1ccc2c(c1)C(N(C2=O)Cc3ccco3)C(=O)NC4CCCCC4 HTS11911 c1ccc(cc1)Cn2c(n[nH]c2=S)c3ccncc3 HTS11929 Cc1nnc2n1cnc3c2c4c(s3)CC(CC4)C HTS11933 CCNc1cc([n+](c2c1c(n[nH]2)N)CC)N.[Cl-] CD01550 Cc1c(c(no1)c2ccccc2Br)C(=O)NC(=S)Nc3ccc4ccccc4c3 S02185 CC1(CC2=C(C(c3c([nH]c(=S)[nH]c3=O)N2)c4ccc(cc4)OC)C(=O)C1)C HTS12057 Cc1ccc(c(c1)NC(=S)Nc2c(cccc2Cl)Cl)C S04600 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)[N+](=O)[O-])C(c4c([nH]c(=S)[nH]c4=O)N)c5c([nH]c(=S)[nH]c5=O)N HTS11942 Cc1cc(c(c(c1C)OC)C)C RF01253 c1cc2c(cc1c3csc(n3)c4ccc5c(c4)OCCO5)OCCCO2 SCR00142 CCCCCCC/N=C(\C)/c1ccccc1O S04747 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)N2CCN(CC2)C(=O)c3ccc(cc3)S(=O)(=O)N(CCC)CCC S06084 c1ccc(cc1)C(=O)CC(C(=O)N2CCc3c2cccc3)C(=O)N4CCc5c4cccc5 HTS12536 Cn1c(=S)nc2c(n1)c3ccccc3n2CC=C HTS12538 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc3c(c2)c4ccccc4o3 HTS00633 c1cc(cc(c1)F)NC(=S)NCCO S04560 CCCN(CCC)S(=O)(=O)c1ccc(cc1)c2nc3ccc(cc3c(=O)o2)C S06081 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)F S01413 Cc1c(c(n(n1)c2ccccc2)C)C(=O)O MO00744 CNC(=O)NC(=O)CSc1c2cc(sc2ncn1)c3ccccc3 HTS13194 c1ccc(cc1)c2cc3c(=S)[nH]cnc3s2 HTS13195 COc1ccc(cc1)/C=C\2/C(=O)N(C(=N2)c3ccccc3)/N=C/c4cccnc4 HTS13199 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=O)CSc3nnc(n3c4ccccc4)c5ccncc5 HTS11953 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nnc(n3Cc4ccccc4)c5ccncc5)C1 HTS11954 c1cc(cc(c1)F)N2C(=O)/C(=C\c3cccs3)/SC2=O S06116 CCOC(=O)C1=NN(C2C1C(=O)N(C2=O)c3ccc(cc3)Cl)c4ccc(cc4)C HTS12231 c1ccc(cc1)N2C(C3CCc4ccccc4C3=N2)c5ccccc5Cl HTS12416 c1ccc(cc1)C(=O)N/C(=C\c2cccs2)/C(=O)N/N=C/c3cccs3 HTS13208 c1ccc(cc1)/C=C(/C(=O)N/N=C/c2ccccc2)\NC(=O)c3ccccc3 HTS13209 Cn1c(=O)n-2c(n1)CSc3c2cccc3 HTS13169 COc1ccc(cc1)/C=C(/C(=O)N/N=C/c2cccnc2)\NC(=O)c3ccccc3 HTS13205 CC(=O)CSc1nc(c(nn1)c2ccccc2)c3ccccc3 HTS12485 c1ccc(cc1)c2c(nnc(n2)SCC(=O)N)c3ccccc3 HTS12486 Cc1ccc(cc1)Cc2c(=O)nc3n(nc(n3n2)C(=O)c4cccs4)c5ccc(cc5)Cl HTS12264 CCOC(=O)c1cnn(c1NC(=O)CN2CCN(CC2)c3ccccc3)c4ccccc4 HTS12022 c1ccc(cc1)Nc2c3cnn(c3[nH]c(=S)n2)c4ccccc4 HTS12024 CC(=O)CSc1nc2c(c3ccccc3[nH]2)nn1 HTS12491 c1cc(sc1)C(=O)c2c(cn(n2)c3ccc(cc3)Cl)C#N HTS12205 c1ccc(cc1)c2cc(n3c(n2)ncn3)Nc4cccc(c4)C(F)(F)F HTS11994 c1ccc(cc1)Cc2c(=O)nc3n(nc(n3n2)C(=O)c4cccs4)c5ccccc5 HTS12271 CC(=O)N1CCC(CC1)C(=O)Nc2ccc(cc2)c3cnco3 SCR00117 c1ccc(cc1)N2C(C3CCc4ccccc4C3=N2)c5ccc(cc5)F HTS12417 c1ccc(cc1)NC(=O)NC(=O)CSc2nnc(n2C3CCCCC3)c4cccs4 HTS12525 CCOC(=O)c1c(c2c(c3c(nc2o1)-c4ccccc4CC3)c5cccnc5)N HTS12446 Cc1ccc(cc1)Nc2cc(nc3n2ncn3)c4ccccc4 HTS11995 c1ccc(cc1)c2cc(n3c(n2)ncn3)Nc4ccc(cc4)Cl HTS11996 Cc1ccccc1N/C(=C/2\CCOC2=O)/C HTS11999 C/C(=C\1/CCOC1=O)/Nc2ccc(cc2)[N+](=O)[O-] HTS12001 CC(=O)CSc1nnc(n1Cc2ccccc2)Cn3c4ccccc4nn3 HTS12471 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CC4)OC(=O)c5ccco5 HTS12476 CCOC(=O)/C(=C/c1cn(nc1c2ccc(cc2)[N+](=O)[O-])c3ccccc3)/C#N HTS12002 c1ccc(cc1)n2c3c(cn2)c(=O)n(c(=O)[nH]3)c4ccccc4 HTS12009 c1ccc(cc1)n2c3c(cn2)c(=O)n(c(=O)[nH]3)c4ccc(cc4)Cl HTS12010 Cc1cc(cc(c1)NC(=O)C2CCN(CC2)C(=O)C)C SCR00121 CC(=O)N1CCC(CC1)C(=O)Nc2ccc(cc2)N3CCOCC3 SCR00101 CCOC(=O)c1c2nc(c3ccccc3n2nn1)S HTS12449 CCOC(=O)c1c2nc(c3ccccc3n2nn1)SCC=C HTS12451 c1ccc(cc1)n2c3nc(=O)c(nn3c(n2)C(=O)c4cccs4)Cc5ccc(cc5)Cl HTS12262 Cn1cnc2c(c1=O)cnn2c3ccccc3 HTS11923 CCN(CC)c1c2cnn(c2ncn1)c3ccccc3 HTS11925 c1ccc(cc1)n2c(n[nH]c2=S)c3ccncc3 HTS11930 CC1CCc2c(sc3c2c(ncn3)Oc4ccccc4)C1 HTS11931 c1ccc(cc1)n2c3c(cn2)c(=O)n(c(=O)[nH]3)c4ccc(c(c4)Cl)Cl HTS12011 CC(=O)CSc1nc(c2cnn(c2n1)c3ccccc3)Nc4ccccc4 HTS12012 Cc1c2c(c3cc(ccc3n1)F)N(CC2)c4ccc(cc4)Cl HTS12014 Cc1cccc2c1nc(c3c2N(CC3)c4ccccc4F)C HTS12016 Cc1ccc2c(c1)cc(s2)C(=O)O MO00911 c1cc(ccc1C(=O)CSc2nnc3n2CCCN3)[N+](=O)[O-] HTS11917 CSc1nc(c(nn1)c2ccccc2)c3ccccc3 HTS12483 Cc1ccc(c(c1)NC(=S)Nc2ccccc2Cl)C S04590 Cc1cccc2c1nc(c3c2N(CC3)c4ccc(cc4)Cl)C HTS12017 c1cc(cc(c1)Cl)n2c3nc(=O)c(nn3c(n2)C(=O)c4cccs4)Cc5ccc(cc5)Cl HTS12263 COc1ccc(cc1)Cc2c(=O)nc3n(nc(n3n2)C(=O)c4cccs4)c5ccccc5 HTS12265 CCOC(=O)CSc1nnc(n1C)c2ccncc2 HTS11937 c1ccc(cc1)c2c(cn(n2)c3ccccc3)C(c4c([nH]c(=S)[nH]c4=O)N)c5c([nH]c(=S)[nH]c5=O)N HTS11940 c1cc(c(c(c1C#N)OCC(F)(F)F)C#N)OCC(F)(F)F MWP01166 C=CCSc1c2c(c(c3n1c4ccccc4n3)C#N)CCC2 HTS11913 Cc1ccc(c(c1)NC(=S)Nc2ccccc2F)C S04589 CC12c3cc(c(cc3CCN1C(=NN2c4ccccc4)C(=O)c5cccs5)OC)OC HTS12368 CCOC(=O)C1=NN(C2(N1CCc3c2cc(c(c3)OC)OC)C)c4ccc(cc4)C HTS12369 c1cc(c(nc1)Cl)C(=O)Nc2cccnc2Cl TG00169 c1ccc2c(c1)nc(s2)CN.Cl CC06013 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)[N+](=O)[O-])/C=N/NC(=O)c4ccncc4 HTS11992 Cc1ccc2cc(ccc2n1)NC(=O)C3CCN(CC3)C(=O)C SCR00105 Cc1c(c(no1)c2ccccc2Cl)c3nnnn3c4cccc(c4)C(F)(F)F S03333 Cc1cc(ccc1NC(=O)c2c(onc2c3ccccc3Cl)C)F S03358 c1cc(ccc1c2csc(n2)c3ccc4c(c3)OCCO4)N5CCOCC5 SCR00144 c1cc(c(c(c1)Cl)N2C(=O)C=CC2=O)Cl S01327 CC(C)NC(=S)N1CCCN(CC1)c2c(cccn2)[N+](=O)[O-] SCR00153 CCOC(=O)/C(=N/Nc1cc(ccc1N2CCOCC2)C(F)(F)F)/C SP01160 CCc1ccc(cc1)NC(=S)NNC(C)(C)C S06243 COc1cc(cc(c1OC)OC)C(=O)Nc2c(cccc2F)F S06353 c1ccc2c(c1)C(=O)N(C2=O)CCSC(=N)N.Br S06360 Cc1cc(cc(n1)Cl)C(=O)NNc2ccc(cc2)Cl RF03771 c1ccc(cc1)n2c(n[nH]c2=S)c3ccc(cc3)Cl HTS11926 Cc1ccc(cc1)Sc2ccccc2NC(=O)c3c(cccc3F)F S06333 c1ccc(cc1)C(=O)NC(=S)Nc2ccccc2Cl S02076 CCOC(=O)c1cnc2c(cnn2c1N)C(=O)OCC HTS12465 C=CCSc1nnc(n1c2ccc(cc2)Cl)Cn3c4ccccc4nn3 HTS12466 CCN(CC)c1ccc(c(c1)C)NC(=S)N2CCN(CC2)C(=S)Nc3ccc(cc3C)N(CC)CC S06102 Cc1ccc(cc1)n2cc(nc2SCc3n[nH]c(=S)n3c4ccc(cc4)OC)c5cccs5 HTS13236 Cc1ccc(cc1)n2cc(nc2SCc3n[nH]c(=S)n3c4ccc(cc4)F)c5cccs5 HTS13238 c1cc(ccc1c2n[nH]c(=S)n2N)Cl HTS12535 c1cc(cc(c1)S(=O)(=O)N)C(F)(F)F CD03845 c1cc(cc(c1)N2C(=O)C=CC2=O)C(F)(F)F S02722 c1cc(c(c(c1)Cl)Cc2n[nH]nn2)Cl RJF00335 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N/N=C/c4ccncc4 HTS12542 Cc1ccc(cc1)/N=C\2/c3ccccc3N(C2=O)C HTS12043 Cc1c2c(n(n1)c3ccccc3)NC4=C(C2c5ccc(cc5Cl)Cl)C(=O)CC(C4)(C)C HTS12044 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N/N=C/c4ccc(cc4)Cl HTS12549 COCc1cc(nc(n1)SCc2ccc(c(c2)Cl)F)O RJF00523 Cc1ccc(cc1)N2C3C(C(=N2)C(=O)C)C(=O)N(C3=O)c4ccc(cc4)OC HTS12233 CCOC(=O)c1cnc(nc1NC(=O)Nc2ccc(cc2)Cl)N3CCOCC3 HTS13196 c1ccc(cc1)c2nc(c(=O)n(n2)CN3CCOCC3)C(CN4CCOCC4)c5ccccc5 HTS13197 c1c2c(ncnc2nc(n1)N3CCOCC3)N HTS13198 CSc1cccc(c1)N2C(=O)CSC2=O S06108 COc1ccc(cc1)/C=N/NC(=O)Cn2c(=O)nc(c(n2)c3ccccc3)c4ccccc4 HTS12556 c1ccc2c(c1)c3c([nH]2)nc(nn3)N/N=C/c4ccc5c(c4)OCO5 HTS12557 CCC1c2c(nn(c2NC3=C1C(=O)CC(C3)(C)C)c4ccccc4)C HTS12049 Cc1ccc(cc1)/C=C/2\C(=O)N(C(=O)S2)c3cccc(c3)SC S06109 c1ccc(cc1)C2=CS/C(=C\3/C(=NNC3=O)c4ccccc4)/O2 HTS12237 c1ccc(cc1)c2c3c4c(c(=O)n(cn4)/N=C/c5ccc6c(c5)OCO6)sc3nnc2c7ccccc7 HTS10013 c1ccc(cc1)C(=O)N/C(=C\c2ccccc2Cl)/C(=O)N/N=C/c3ccc(cc3)Cl HTS13210 c1ccc(cc1)/C=N/N2C(=N/C(=C\c3cccs3)/C2=O)c4ccccc4 HTS13204 COc1ccc(cc1)Cc2c(=O)nc3n(nc(n3n2)C(=O)c4ccccc4)c5ccc(cc5)Cl HTS12269 c1ccc(cc1)Cc2c(=O)nc3n(nc(n3n2)C(=O)c4cccs4)c5ccc(cc5)Cl HTS12270 Cn1c(=S)nc2c(n1)c3ccccc3n2Cc4ccc(cc4)F HTS12563 Cn1c(=S)nc2c(n1)c3ccccc3n2Cc4ccccc4 HTS12564 CN1CCN(CC1)c2c3cc(sc3ncn2)c4ccccc4 HTS13217 c1ccc2c(c1)-n3c(nn(c3=O)CC(=O)N/N=C/c4ccncc4)CS2 HTS13218 c1ccc(cc1)c2cc(n3c(n2)ncn3)SCc4ccc(cc4)[N+](=O)[O-] HTS11967 c1ccc(cc1)C(=O)CSc2nc3c(c4ccccc4[nH]3)nn2 HTS12489 CC(=O)c1c(cn(n1)c2ccccc2)C#N HTS12203 Cc1ccc(cc1)n2cc(c(n2)C(=O)C)C#N HTS12204 CCOC(=O)c1cnn(c1NC(=O)CSc2nnc(o2)c3ccncc3)c4ccccc4 HTS12027 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3c4ccccc4)c5ccc(cc5)Cl HTS12029 C=CCN1c2ccccc2/C(=N/c3ccc(cc3)Cl)/C1=O HTS12042 c1ccc(c(c1)Cn2c(=O)n-3c(n2)CSc4c3cccc4)Cl HTS13167 c1ccc2c(c1)-n3c(nn(c3=O)Cc4ccc(cc4)F)CS2 HTS13168 COc1cccc(c1)C(=O)c2c(c3c(s2)nsc3SCc4ccccc4)N HTS13180 c1cc(ccc1C(=O)c2c(c3c(s2)nsc3SCCN4CCCCC4)N)Cl HTS13181 Cn1c(nnc1SCc2ccc(cc2)F)c3c(c4c(cc(nc4o3)c5ccccc5)c6ccco6)N HTS12078 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3ccc(cc3)F)N)C HTS12091 CCO/C=C/1\C(=O)N(C(=S)S1)c2ccc(cc2C)C S03726 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3ccccc3Cl)N)C HTS12088 Cc1ccc(c(c1)NC2=NCCS2)C S04613 Cc1ccc(c(c1)NC(=S)NCCCN2CCOCC2)C S04614 CCOC(=O)C1(C(C(=NN1c2ccc(cc2)[N+](=O)[O-])c3cccs3)c4ccccc4)C#N HTS12362 CCOC(=O)CCC(=O)OC(c1ccccc1)C(=O)c2ccccc2 SS00043 Cc1cc2c(cc1C)nc([nH]2)c3cccc4c3cccc4 S03660 Cc1ccc2c(c1)nc([nH]2)c3cccc4c3cccc4 S03661 COc1ccc(cc1OC)/C=C/2\C(=O)N(C(=S)S2)c3ccc(c(c3)F)F S03845 c1ccc(c(c1)CNC(=O)c2cnc(cc2C(F)(F)F)Cl)Cl RF04325 c1cc(c2c(c1)OCCO2)CO CC01409 CSc1cccc(c1)N2C(=O)c3cccc4c3c(cc(c4)[N+](=O)[O-])C2=O S03300 c1ccc(cc1)NC(=S)N2c3ccccc3Sc4c2cccc4 HTS12545 Cc1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)C S04617 c1c(cc(nc1OCC(F)(F)F)Cl)C(=O)O RF04919 c1cc2c(cc1c3nc(cs3)c4ccc(c(c4)Cl)Cl)OCCO2 SCR00133 CCOC(=O)C(=CNNc1ccsc1C(=O)OC)C(=O)OCC GK01775 CC1(CC2=C(C(c3c([nH]c(=S)[nH]c3=O)N2)c4ccc(cc4)[N+](=O)[O-])C(=O)C1)C HTS12056 Cc1cc(nn1C(C)(C)C)C(=O)Nc2ccc3c(c2)OCCO3 HTS11317 c1cc(ccc1NNC(=O)c2cc(nc(c2)Cl)OCC(F)(F)F)F RF04963 CCO/C=C\1/C(=O)N(C(=S)S1)c2ccc(cc2)Cl S02878 Cc1c(c(no1)c2ccccc2Cl)c3nnnn3c4ccccc4 S03334 c1cc(ccc1C2(CCN(CC2)C(=O)c3cc(cc4c3OCOC4)F)O)Cl HTS11374 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2ccc(s2)c3cc(n(n3)C)C(F)(F)F HTS11118 CC1CN(CC(O1)C)c2ccc(cc2OC)NC(=O)c3cccs3 CD07157 Cc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3c(onc3c4c(cccc4Cl)Cl)C S06421 COc1cccc(c1O)/C=N\c2ccccc2N3C(=O)c4ccccc4C3=O S05529 c1cc(cc(c1)F)NCN2C(=O)c3ccc(cc3C2=O)[N+](=O)[O-] S05544 Cc1ccc(cc1)N2C(=O)CSC23c4ccccc4NC3=O HTS12063 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S06213 CSc1c2c(ncn1)n(nn2)Cc3ccccc3Cl HTS12149 Cc1ccc2c(c1)c(=O)oc(n2)C(c3ccccc3)(c4ccccc4)O S04768 c1ccc2c(c1)C=CC(N2C(=O)c3c(cccc3F)F)C#N S06271 CCNc1c2cnn(c2[nH]c(=S)n1)c3ccccc3 HTS12023 Cc1ccc(c(c1)NC(=S)Nc2c(cccc2C)C)C S04603 c1cc(ccc1NC(=S)NC2CCCCC2)Cl S04698 CCOC(=O)C1=NN(/C(=C/C2=NCCc3c2cc(c(c3)OC)OC)/S1)c4ccc(cc4)Cl HTS12380 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3Cc4ccccc4)c5ccncc5 HTS12028 CC(=O)CSc1nnc(n1c2ccccc2)c3ccco3 HTS11946 Cn1c(nnc1SCC(=O)N/N=C/c2cccnc2)c3ccncc3 HTS11949 Cc1cc(nc2c1c3c(s2)c(ncn3)N4CCOCC4)C HTS12121 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(o3)c4cccs4 HTS12032 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(o3)c4ccncc4 HTS12033 Cc1ccc(c(c1)/N=C/c2ccccc2O)C S04615 Cc1ccc(c(c1)/N=C/c2cc(ccc2O)Br)C S04616 c1ccc(cc1)n2c(n[nH]c2=S)c3cccs3 HTS11944 Cc1cccc(c1NC2=NCCS2)C S01189 c1ccc(cc1)n2c(nnc2SCC(=O)N/N=C/c3ccc(cc3)Cl)c4ccncc4 HTS11952 CC(C)c1ccc(cc1)/C=N/N=C\2/NC(=O)C(S2)CC(=O)O S04708 c1cc(oc1)/C=N/N=C\2/NC(=O)C(S2)CC(=O)O S04709 Cc1c(cn(n1)c2ccccc2)/C=N/n3c(n[nH]c3=S)c4ccncc4 HTS11976 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3c4ccccc4)c5ccncc5 HTS12030 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3cccnc3)N)C HTS12096 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nccn3C HTS12035 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3C)c4ccncc4 HTS12037 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N/N=C/c4ccc5c(c4)OCO5 HTS12550 CCOC(=O)c1c2nc(c3ccccc3n2nn1)Sc4nc5ccccc5o4 HTS12551 Cc1c2c(n(n1)c3ccccc3)NC4=C(C2c5ccccc5Cl)C(=O)CC(C4)(C)C HTS12046 Cc1ccc2c(c1)c3c(c(n2)C)CCN3c4ccc(cc4)F HTS12019 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S06183 CC1CCc2c(sc(c2C#N)NC(=O)CSc3[nH]cnn3)C1 HTS11964 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3c4ccccc4)c5ccco5 HTS12034 Cc1cc(nc2c1c3c(s2)c(ncn3)Sc4nnc(n4c5ccccc5)c6cccs6)C HTS12104 C=CCNC(=S)NNC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4ccco4)N HTS12110 Cc1ccc(c(c1)NC(=S)NC2CC(CC(C2)(C)C)C)C S04643 c1ccc(cc1)n2cc(c(n2)c3cccs3)/C=N/NC(=O)CSc4nnc(n4c5ccccc5)c6ccncc6 HTS11950 C/C(=N\OC(=O)NC)/C=C/c1ccccc1 EN00225 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nnc(n3c4ccccc4)c5cccs5)C1 HTS11958 c1cc(sc1)c2nnc3n2N=C(CS3)c4ccc(cc4)[N+](=O)[O-] HTS11977 Cc1c2c(c3cc(ccc3n1)F)SCC2 HTS12006 Cc1cccc2c1nc(c3c2COC3)C HTS12007 c1ccc(cc1)n2cc(c(n2)c3cccs3)/C=N/n4c(n[nH]c4=S)c5cccs5 HTS11984 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/n4c(n[nH]c4=S)c5cccs5 HTS11986 CN1c2ccccc2/C(=N/c3ccc(cc3)Cl)/C1=O HTS12041 c1ccc(cc1)CNC(=S)NNC(=O)c2c(c3c(cc(nc3o2)c4ccccc4)c5ccco5)N HTS12111 Cc1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)NNC(=S)Nc4ccccc4)N)c5ccco5 HTS12112 CCOC(=O)c1cnn(c1NC(=O)CN2CCOCC2)c3ccccc3 HTS12020 Cc1c2c(n(n1)c3ccccc3)NC4=C(C2c5ccc(c(c5)OC)O)C(=O)CC(C4)(C)C HTS12050 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3nnc(n3c4ccccc4)c5cccs5 HTS12031 c1ccc(cc1)c2cc3c(=O)n(c(=O)n(c3s2)Cc4ccccc4Cl)c5ccccc5 HTS13219 Cc1cc(nc2c1c3c(s2)c(ncn3)N(Cc4ccccc4)Cc5ccccc5)C HTS12116 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nnc(n3C)c4ccncc4)C1 HTS11959 c1ccc(cc1)c2ccc(cc2)C(=O)COc3c(c(cc(n3)c4cccs4)c5cccs5)C#N HTS12072 c1ccc(cc1)c2cc(c3c4c(c(=O)n(cn4)/N=C/c5ccc6c(c5)OCO6)oc3n2)c7ccco7 HTS12114 CCc1cccc(c1NC(=O)Nc2ccccc2)C(C)CC CD06443 Cc1ccc(cc1)NC(=O)CC2C(=O)N/C(=N/c3c(cccc3F)F)/S2 S05493 C=CCn1cnc2c(c1=O)cc(s2)c3ccccc3 HTS13221 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CC4)OC(=O)c5ccccc5 HTS12477 CN1CCN(CC1)c2nc(c(nn2)c3ccccc3)c4ccccc4 HTS12478 c1ccc(cc1)c2cc(n3c(n2)ncn3)SCC(=O)c4ccc(cc4)Br HTS11969 CC(=O)CSc1cc(nc2n1ncn2)c3ccccc3 HTS11971 Cc1cc(nc2c1c3c(s2)c(ncn3)N4CCCCC4)C HTS12117 c1cc(c(c(c1)F)/N=C\2/NC(=O)C(S2)CC(=O)Nc3ccc(cc3)Cl)F S05492 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)C3CC3 RJF01040 CC1(CC2=C(C(c3c(=O)[nH]c(nc3N2)SCc4ccc(cc4)Cl)c5ccc(cc5)OC)C(=O)C1)C HTS12052 c1ccc(cc1)c2cc(n3c(n2)ncn3)Sc4nnc(n4c5ccccc5)c6ccncc6 HTS11966 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4ccccc4)C HTS12080 CCOC(=S)SCc1cc(ccc1OC)C(=O)C CD06452 CCOC(=O)COc1c(sc2c1c(=O)n(c(=S)n2c3ccccc3)c4ccccc4)C#N HTS11919 Cc1ccc(c(c1)NC(=S)Nc2cccc(c2C)Cl)C S04602 c1ccc(cc1)c2c(nnc(n2)N3CCc4c3cccc4)c5ccccc5 HTS12480 Cc1ccc(c(c1)NC(=S)Nc2cccc(c2)C(F)(F)F)C S04597 Cc1ccc(c(c1)NC(=S)Nc2cccc(c2)SC)C S04598 Cc1c(nc(nc1C)S)C RF00381 CC1(CC2=C(C(c3c([nH]c(=S)[nH]c3=O)N2)c4cccs4)C(=O)C1)C HTS12061 Cc1cc(nc(c1C#N)N2CCN(CC2)c3ccccc3)C HTS12066 Cc1cccc(c1C)NC(=O)c2cnc(cc2C(F)(F)F)Cl RF04377 COc1ccc(c(c1)/C=C/2\C(=O)OC(=N2)c3ccccc3)OC S02897 c1cc(c(cc1NC(=O)CC2C(=O)NC(=N)S2)F)F S03905 CC(C)c1nn(c(=O)o1)c2c(cccn2)C(F)(F)F RF04906 COc1nn(c(=O)o1)c2c(cc(cn2)C(F)(F)F)Cl RF04957 c1cc(c(cc1NC(=O)/C=C/C(=O)O)C(=O)O)Cl S06239 c1cc(c(cc1N2C(=O)C=CC2=O)C(=O)O)Cl S06240 Cn1c(cnc1Sc2c(cccn2)[N+](=O)[O-])c3ccc(cc3)Cl TG00117 c1cc(c(c(c1)F)N2C(=O)C=CC2=O)F S05486 CSc1cccc(c1)NC(=O)CC2C(=O)N/C(=N\c3ccc(c(c3)F)F)/S2 S03907 Cc1cccc(c1NC(=O)c2cnc(cc2C(F)(F)F)Cl)C RF04378 c1cc(cc(c1)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)N)C(F)(F)F HTS08365 C/C(=N\O)/C(C)(C)Nc1cccc(c1)F HTS11324 c1cc(c2c(c1)OCCO2)C(=O)O CC01401 c1cc(c(c(c1)F)CSC(=N)N)F.Cl S05645 Cc1ccc(cc1)NC(=S)Nc2ccc(cc2)C(=O)C S00642 c1c(c(c(cc1Cl)Cl)O)/C=N/CC2CCC(CC2)C/N=C/c3c(c(cc(c3)Cl)Cl)O S00781 COc1ccc(cc1)c2csc(n2)c3ccc4c(c3)OCCO4 SCR00147 CCOc1ccc(cc1)NC(=S)NC2CCCCCCCCCCC2 S01397 COc1cc(cc(c1OC)OC)NC(=N)N[N+](=O)[O-] S03967 CC(C)c1ccc(cc1)/N=C\2/N(C(=O)CS2)CCc3ccc(c(c3)OC)OC S03640 Cc1ccc(cc1NCN2C(=O)c3ccccc3C2=O)I S01446 CCOC(=O)c1ccc(cc1Nc2ccc(cc2C(=O)OCC)[N+](=O)[O-])Cl S06225 c1cc2c(cc1c3csc(n3)c4ccc5c(c4)OCCO5)OCO2 SCR00136 CSc1cccc(c1)/N=c\2/c(c(ss2)SC)c3ccccc3 S03954 c1ccc(cc1)Oc2ccccc2C(=O)N/N=C/c3ccccc3O S04719 Cc1cc2c(cc1C)nc([nH]2)c3ccc(cc3)OC S03662 CCOC(=O)c1c(nc(s1)Br)C MO00750 CN(C)c1ccc(cc1)/C=N/N S04745 CC1(CC2=C(C(c3c([nH]c(=S)[nH]c3=O)N2)c4ccc(cc4)OCc5ccccc5)C(=O)C1)C HTS12058 CC(=O)c1ccccc1/N=C/c2cc(cc(c2O)Cl)Cl S04725 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccc(cc3)Cl)c4ccco4)N HTS12125 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccc(cc3)C)c4ccco4)N HTS12126 c1ccc(cc1)C(c2ccccc2)(c3nc4cc(ccc4c(=O)o3)[N+](=O)[O-])O S04767 CC1(CC2=C(C(c3c([nH]c(=S)[nH]c3=O)N2)c4cccc(c4)OC)C(=O)C1)C HTS12060 c1ccc(cc1)N2C(=O)CSC23c4ccccc4NC3=O HTS12062 CSc1c2c(ncn1)n(nn2)Cc3ccccc3 HTS12154 c1cc(cc(c1)F)NC(=S)NCc2ccc3c(c2)OCO3 S04647 C/C(=C\1/CCOC1=O)/Nc2ccccc2F HTS11998 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)N(C(=O)S2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F S06118 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4ccco4)N HTS12129 CC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4cccs4)N HTS12131 CCOC(=O)c1c2nc(c3ccccc3n2nn1)Nc4ccc(cc4)Cl HTS12541 Cc1c2c(n(n1)c3ccccc3)NC4=C(C2c5cccnc5)C(=O)CC(C4)(C)C HTS12047 Cc1c2c(n(n1)c3ccccc3)NC4=C(C2c5cccc(c5)OC)C(=O)CC(C4)(C)C HTS12048 CCn1c(n[nH]c1=S)c2cccs2 HTS11943 Cc1ccc(cc1)N/C(=C/2\CCOC2=O)/C HTS11997 Cc1cccc2c1nc(c3c2N(CC3)c4cccc(c4)C(F)(F)F)C HTS12018 Cc1cccc2c1nc(c3c2SCC3)C HTS12004 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4cccs4)N HTS12127 Cc1cc(nc2c1c(c(s2)c3n[nH]c(=S)n3CC=C)N)C HTS12145 c1ccc(c(c1)Cn2c3c(c(ncn3)Sc4nc5ccccc5s4)nn2)Cl HTS12146 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=O)c3c(c4c(cc(nc4o3)c5cccs5)c6ccco6)N HTS12139 Cc1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)N/N=C/c4ccccc4)N)c5ccco5 HTS12140 c1ccc(cc1)Cn2c3c(c(=S)[nH]cn3)nn2 HTS12157 c1ccc(c(c1)Cn2c3c(c(=S)[nH]cn3)nn2)Cl HTS12158 CN1CCN(CC1)c2c3c(ncn2)n(nn3)Cc4ccccc4Cl HTS12167 c1ccc(c(c1)CN\2C(=O)CS/C2=N\c3cc(c(cc3Cl)Cl)Cl)Cl S04654 c1ccc(c(c1)CN\2C(=O)CS/C2=N\c3cccc(c3)F)Cl S04657 CNC(=O)O/N=C/C(=O)c1ccc(cc1)Cl RF00950 CCOC(=O)c1cnn(c1NC(=O)CSc2nnc(n2c3ccccc3)c4ccc(cc4)Cl)c5ccccc5 HTS12026 CCn1c(n[nH]c1=S)c2c(c3c(cc(nc3o2)c4ccccc4)c5ccco5)N HTS12142 c1ccc2c(c1)c3c([nH]2)nc(nn3)N/N=C/c4cccs4 HTS12558 c1ccc2c(c1)c3c([nH]2)nc(nn3)N/N=C/c4ccc(cc4)F HTS12559 c1ccc(cc1)/C=N/Nc2nc3c(c4ccccc4[nH]3)nn2 HTS12560 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nc4ccccc4o3)C1 HTS11963 Cc1ccc2c(c1)c3c(c(n2)C)CCS3 HTS12005 CCOC(=O)NC(=S)N/N=C/c1ccccn1 S04735 C1CCCCCC(CCCCC1)NC(=O)/C=C/C(=O)O S01368 C1CCCCCC(CCCCC1)N2C(=O)C=CC2=O S01369 CCOc1ccc(cc1)/N=C/c2ccc(cc2)OC S04673 COc1cc2c(cc1OC)C3N(CC2)C(=NN3c4ccccc4)C(=O)c5cccs5 HTS12366 c1cc(cnc1)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)Cl HTS12069 CCOC(=O)COc1c(c(cc(n1)c2ccco2)c3ccco3)C#N HTS12070 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3cccs3)N)C HTS12095 COc1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)c4ccc(cc4)Cl)N)c5cccnc5 HTS12073 Cn1c(nnc1SCC(=O)N2CCc3c2cccc3)c4ccncc4 HTS12494 C=CCn1c(nnc1SCC(=O)N2CCc3c2cccc3)c4ccc(cc4)Cl HTS12495 c1ccc(cc1)SCC(=O)N2CCc3c2cccc3 HTS12497 c1ccc(cc1)c2cc(c(c(n2)OCC(=O)c3ccccc3)C#N)c4cccs4 HTS12071 Cc1cc(nc2c1c3c(s2)c(ncn3)Sc4nnc(n4Cc5ccccc5)c6ccncc6)C HTS12101 CCn1c(nnc1SCc2ccc(cc2)Cl)c3c(c4c(cc(nc4o3)c5ccccc5)c6ccco6)N HTS12077 c1ccc2c(c1)c3ccccc3n2CC(=O)O HTS11415 CCOc1ccc(cc1)NC(=S)Nc2cc(ccc2C)C S04642 CC(=O)C1=NN(C2(N1CCc3c2cc(c(c3)OC)OC)C)c4ccc(cc4)Cl HTS12367 Cc1ccc(cc1)S(=O)(=O)Nc2c(cccc2C(C)C)C CD06407 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3cn(nc3c4cccs4)c5ccccc5)N)C HTS12081 c1ccc2c(c1)C(=O)N(C2=O)c3ccccc3/N=C\c4cc(cc(c4O)Cl)Cl S05507 CCN(CC)c1ncc(c(n1)N)C#N HTS12511 c1ccc2c(c1)CCCN2C(=O)CN3CCc4c3cccc4 HTS12506 c1ccc(cc1)N2CCN(CC2)CC(=O)N3CCCc4c3cccc4 HTS12507 c1cc(ncc1C(=O)NN)N2CCOCC2 CC17527 Cc1c(nn(n1)c2ccccc2)C(=O)N3CCC(CC3)(c4ccc(cc4)Cl)O HTS11378 CC(=O)Nc1cc2cc(ccc2oc1=O)NC(=O)c3ccccc3C(F)(F)F SCR00155 CSc1cccc(c1)NC(=O)CC2C(=O)N/C(=N\c3cccc(c3)SC)/S2 S03904 c1ccc2c(c1)ccc(c2/C=N/Cc3cccnc3)O S04164 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)NNc3c(cccc3Cl)Cl)Cl HTS11405 c1c(cc(cc1Cl)Cl)CNC(=O)c2cnc(cc2C(F)(F)F)Cl RF04314 CCc1cccc(c1N(CC)C(=O)c2cnccc2C(F)(F)F)CC RF04407 CCN(CC)CCCNS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F CD05655 CN(CCN(C)S(=O)(=O)c1ccc(c(c1)Cl)N2C(=O)CC3(C2=O)CCCC3)S(=O)(=O)c4ccc(c(c4)Cl)N5C(=O)CC6(C5=O)CCCC6 SCR00154 c1ccc(cc1)Cn2c3c(c(ncn3)N4CCN(CC4)c5ccccc5)nn2 HTS12169 CN(C)C(=S)NCc1cccnc1 S04773 COc1cc2c(cc1OC)C3N(CC2)C(=NN3c4ccccc4)c5ccccc5 HTS12217 C[n+]1c(ccc2c1cccc2)/C=C/c3ccc(cc3)N(C)CCC#N.[I-] S04052 c1cncc(c1)/C=N/N=C/c2cnccc2 S04056 c1cc(c(c(c1)Cl)Cc2nc(cs2)C(=O)O/N=C/c3c(cccc3Cl)Cl)Cl HTS11406 CN(C)c1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccccc3 S06435 c1ccc(c(c1)C2=NCCCN2)SCc3cccc(c3)C(F)(F)F.Cl CD05714 c1ccc(cc1)N2CCN(CC2)C(=O)CSc3nnnn3c4ccc(cc4)O SCR00160 Cc1c(cnn1c2ccccc2)S(=O)(=O)N3CCCC3c4ccc(cc4)F SCR00186 Cc1ccc(cc1)C(=O)c2cc3c([nH]2)nsc3Nc4ccccc4OC SCR00158 Cc1c(c(on1)c2ccccc2)NC(=O)Nc3ccc(cc3)Cl SCR00346 c1cc(cc(c1)NC(=S)Nc2cccc(n2)NC(=S)Nc3cccc(c3)C(F)(F)F)C(F)(F)F S04082 Cc1cc(no1)/N=C/c2cc(ccc2O)Br S04779 COc1ccccc1C2C(CCC(=O)N2)[N+](=O)[O-] S06327 CCOC(=O)c1c(nc(s1)NC(=O)c2cccs2)C S06447 c1cc(c(cc1N2C(=O)CSC2=S)F)F S03822 c1cc(c(cc1/C=C/2\C(=O)N(C(=S)S2)c3ccc(c(c3)F)F)Cl)Cl S03842 CCOC(=O)c1c(c(sc1NC(=O)Nc2cccc(c2)Cl)C)c3ccccc3 SCR00215 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc(cc2)Oc3ccc(cc3)Cl S06238 CCOC(=O)c1c(n[nH]c1N/N=C/c2cccnc2)C S06450 c1cc(cc(c1)[N+](=O)[O-])/C=C/2\C(=O)N(C(=S)S2)c3ccc(c(c3)F)F S03844 Cc1ccc(cc1F)NC(=S)Nc2cccc(c2Cl)Cl S04128 c1cc2c(cc1CNC(=S)Nc3cc(c(cc3Cl)Cl)Cl)OCO2 S04646 c1ccc(cc1)C(c2ccccc2)NC(=S)Nc3cc(c(cc3Cl)Cl)Cl S04649 Cc1ccc(cc1)n2c(=O)c3c(c4c(cc(nc4s3)C)C)[nH]c2=O HTS12122 CSc1ccccc1NC(=S)Nc2ccc(cc2)Cl S04089 c1ccc(c(c1)CNC(=S)Nc2cc(c(cc2Cl)Cl)Cl)Cl S04648 c1ccc(cc1)C(c2ccccc2)NC(=S)Nc3cccc(c3)F S04650 c1cc(c(cc1NC(=S)NC2CCCC2)Cl)Cl S04692 Cc1cc(nc2c1c3c(s2)c(ncn3)N4CCN(CC4)c5ccccc5)C HTS12118 Cc1cc(nc2c1c3c(s2)c(ncn3)N4CCN(CC4)C)C HTS12119 CCN(CC)c1c2c(c3c(cc(nc3s2)C)C)ncn1 HTS12120 Cc1c(c(c(c(c1C)C)CSc2ccccc2NC(=O)/C=C/C(=O)O)C)C S03874 c1ccc(cc1)C/N=C/c2c3ccccc3ccc2O S04165 CSc1cccc(c1)NC(=S)NCCCO S04186 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4cn(nc4C)c5ccccc5)C HTS12084 c1cc(ccc1Cn2c(c(nn2)C(=O)N)N)Cl HTS12087 CNC(=S)N1C(C2CCc3ccccc3C2=N1)c4ccccc4Cl HTS12177 COc1ccc(cc1)NC(=S)N2C(C3CCc4ccccc4C3=N2)c5ccc(cc5)F HTS12178 Cc1cc(nc2c1c3c(s2)c(=O)n(c(=O)[nH]3)c4cccc(c4)Cl)C HTS12123 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccco3)c4ccco4)N HTS12124 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)c4ccc(cc4)Br)N)c5cccs5 HTS12133 CCOC(=O)CSc1nnc(n1c2ccccc2)c3ccco3 HTS11945 CC1CCc2c(sc(c2C#N)NC(=O)c3ccc(cc3)F)C1 HTS11947 CC1CCc2c(sc(c2C#N)N)C1 HTS11948 c1cc(c(c(c1)Cl)NC(=O)/C=C/C(=O)O)Cl S01326 c1ccc(cc1)c2cc(n3c(n2)ncn3)SCc4ccccc4Cl HTS11968 C/C(=C\1/CCOC1=O)/Nc2ccc(cc2)F HTS12000 CCOC(=O)/C(=C/c1cn(nc1c2ccc(cc2)C)c3ccccc3)/C#N HTS12003 CCOC(=O)c1c(c2c(cc(nc2o1)c3cccs3)c4ccco4)N HTS12128 c1cc(oc1)c2cc(c3c(c(oc3n2)C(=O)c4ccc(cc4)Cl)N)c5cccs5 HTS12130 c1cc(oc1)c2cc(nc3c2c(c(o3)C(=O)c4cccs4)N)c5cccs5 HTS12132 COc1cccc(c1)/C=N/NC(=O)c2c(c3c(cc(nc3o2)c4ccccc4)c5ccco5)N HTS12136 c1cc2c(c(sc2nc1)C(=O)O)N MO00759 CCNC(=S)N1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)F HTS12180 c1ccc(cc1)COC(=O)/C(=C/c2cccnc2)/C#N S05455 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)c4ccccc4)N)c5cccs5 HTS12134 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)N/N=C/c4cccnc4)N)c5ccco5 HTS12135 c1ccc2c(c1)C(=O)N(C2=O)Nc3ccc(cc3)N4CCOCC4 S04625 Cc1cc(nc2c1c(c(s2)C(=O)c3cccs3)N)C HTS12074 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=N/O RF01469 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nc4ccccc4s3)C1 HTS11955 CCn1c(nnc1SCC(=O)Nc2c(c3c(s2)CC(CC3)C)C#N)c4cccs4 HTS11957 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)/C=N/n4c(n[nH]c4=S)c5cccs5 HTS11983 c1ccc(cc1)Nc2c3cnn(c3nc(n2)SCc4ccc(cc4)Cl)c5ccccc5 HTS12013 Cn1c(n[nH]c1=S)c2c(c3c(cc(nc3o2)c4ccccc4)c5ccco5)N HTS12141 c1cc(ccc1Cn2c3c(c(ncn3)N4CCOCC4)nn2)F HTS12170 c1ccc2c(c1)CCC3C2=NN(C3c4ccc(cc4)F)C(=S)NC5CCCCC5 HTS12179 c1cc2c(c(c1)S(=O)(=O)N3CCCC3c4ccc(cc4)F)non2 SCR00182 CCOC(=O)c1c2n(c(=O)c3ccccc3n2nn1)C HTS12188 CCOC(=O)c1c2n(c(=O)c3ccccc3n2nn1)CC=C HTS12189 c1cc(sc1)c2n[nH]c(=S)o2 HTS11965 CC1CCc2c(sc(c2C#N)NC(=O)CSc3[nH]c4ccccc4n3)C1 HTS11961 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nnc(n3CC=C)c4ccccc4)C1 HTS11962 Cc1ccc(cc1Cl)c2nc(cc(n2)O)COC RJF01066 CC12c3cc(c(cc3CCN1C(=NN2c4ccc(cc4)Cl)NC(=O)c5ccccc5)OC)OC HTS12371 CCn1c(nnc1SCC(=O)c2ccccc2)c3c(c4c(cc(nc4o3)c5ccccc5)c6ccco6)N HTS12076 c1ccc2c(c1)CCC3C2=NN(C3c4ccc(cc4)F)C(=S)Nc5ccc(cc5)Cl HTS12181 C=CCNC(=S)N1C(C2CCc3ccccc3C2=N1)c4cccs4 HTS12182 COc1ccc(cc1)C2=CC=C(CS2)C(=O)OC SCR00162 c1ccc2c(c1)CCN2C(=O)CCC(=O)Nc3ccc(cc3)I SCR00161 c1ccc(cc1)Oc2ccc(cn2)S(=O)(=O)N3CCCC3c4ccc(cc4)F SCR00185 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=S)NC3CC(CC(C3)(C)C)C SCR00171 c1ccc2c(c1)C(=O)N(C2=O)c3ccccc3NC(=S)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F S05520 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3ccc(c(c3)OC)O)N)C HTS12089 c1ccc(cc1)Cn2c3c(c(ncn3)Nc4ccc(cc4)Cl)nn2 HTS12164 CN1CCOc2c1cc(cc2)S(=O)(=O)N3CCCC3c4ccc(cc4)F SCR00183 c1cc(ccc1c2cnco2)S(=O)(=O)N3CCCC3c4ccc(cc4)F SCR00184 c1cc(cc(c1)NC(=O)/C=C/C(=O)O)NC(=O)/C=C/C(=O)O S01819 c1ccc(c(c1)N2C(=O)C=CC2=O)[N+](=O)[O-] S02158 Cc1cccc(c1)/C=C\2/C(=O)N(C(=S)S2)/N=C/c3ccc(cc3Cl)Cl S04287 c1cc(c(cc1Br)Cl)Nc2n[nH]c(=S)s2 S04198 CCOC(=O)CSc1[nH]c(=O)c2c(n1)NC3=C(C2c4ccc(cc4)[N+](=O)[O-])C(=O)CC(C3)(C)C HTS12053 CC(=O)CSc1[nH]c(=O)c2c(n1)NC3=C(C2c4cccc(c4)OC)C(=O)CC(C3)(C)C HTS12054 c1ccc(cc1)COC(=O)N2CCCC(C2)C(=O)O CC24701 c1cc(c(cc1F)F)NC(=O)CC2(CCCCC2)CC(=O)O SCR00329 c1cc2c(cc1NC(=O)CC3(CCCCC3)CC(=O)O)OCCCO2 SCR00328 CCOC(=O)c1nn(c2n1c3ccccc3n2)c4ccc(cc4)C HTS12202 Cc1ccc(cc1C)n2c(nnn2)SCC(=O)c3ccc(cc3)c4ccccc4 S05734 CC\1=NN(C(=O)/C1=C/2\N(N=C(S2)C(=O)c3ccccc3)c4ccc(cc4)Cl)c5ccccc5 HTS12248 c1cc(sc1C(=O)O)[N+](=O)[O-] RF01631 Cn1cc(c(n1)C(F)(F)F)C(=O)O GK00761 c1c(cc(cc1C(F)(F)F)NC(=O)CC2(CCCCC2)CC(=O)O)C(F)(F)F SCR00332 Cc1c(snn1)C(=O)N2CCC(CC2)(c3ccc(cc3)Cl)O HTS11371 CC(C)N(Cc1ccccc1)C(=O)c2ccccc2C(=O)O HTS07901 CC(=O)Nc1ccc(cc1)C2=N/C(=C/c3ccc(cc3)N(C)C)/C(=O)O2 S06437 CC\1=NN(C(=O)/C1=C/2\N(N=C(S2)C(=O)c3cccs3)c4ccccc4)c5ccccc5 HTS12249 c1cc(c(cc1F)NC(=O)CC2(CCCCC2)CC(=O)O)Cl SCR00326 CCCCCC/N=C(\C)/c1ccccc1O S04748 CCN(CC)c1c2c(ncn1)n(nn2)Cc3ccccc3 HTS12168 Cc1cccc(c1NC(=S)NC2CCCC2)Cl S04693 Cc1cc(nc2c1c3c(s2)c(ncn3)SCC(=O)c4ccc(cc4)Br)C HTS12099 c1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)N3CCCCCC3 S05661 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(c(s3)C(=O)OCC)C HTS10581 CC1(CC2=C(C(C3=C(N2)CC(CC3=O)(C)C)c4cc(ccc4OC)OC)C(=O)C1)C S06315 c1ccc(c(c1)CNC(=S)Nc2cccc(c2)F)Cl S04651 c1cc2c(cc1CN\3C(=O)CS/C3=N\c4cc(c(cc4Cl)Cl)Cl)OCO2 S04652 CC\1=NN(C(=O)/C1=C/2\N(N=C(S2)C(=O)Nc3ccccc3)c4ccccc4)c5ccccc5 HTS12250 CCOC(=O)C1=NN(/C(=C\2/C(=NNC2=O)c3ccccc3)/S1)c4ccc(cc4)Cl HTS12251 c1cc(ccc1CNC(=N)N[N+](=O)[O-])C#N S03970 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N4CCN(CC4)c5ccccc5 HTS12194 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N4CCOCC4 HTS12196 Cc1cc(nc(c1C#N)Sc2c3c(c4c(cc(nc4s3)C)C)ncn2)C HTS12106 Cc1cc(nc2c1c3c(s2)c(ncn3)Sc4nccn4C)C HTS12107 c1ccc(cc1)Cn2c3c(c(ncn3)Sc4nnc(o4)c5ccncc5)nn2 HTS12150 Cc1cc(nc(c1C#N)Sc2c3c(ncn2)n(nn3)Cc4ccccc4)C HTS12152 c1ccc2c(c1)C3(C(=O)N2)N(C(=O)CS3)c4ccc(cc4)Cl HTS12064 CC(=O)Nc1ccc(cc1)C2=N/C(=C/c3ccccc3OC)/C(=O)O2 S06331 Cc1cc(nc2c1c3c(s2)c(ncn3)SCC=C)C HTS12098 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3ccc(cc3)Cl)N)C HTS12097 Cc1cc(nc2c1c3c(s2)c(ncn3)Sc4nnc(o4)c5ccncc5)C HTS12103 Cc1c(c(c(c(c1C)C)CSc2cccc(c2)NC(=O)/C=C/C(=O)O)C)C S03971 CCOC(=O)c1c(c(sc1NS(=O)(=O)c2ccc(cc2)C)C)c3ccccc3 SCR00221 CNC(=S)NNC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4ccco4)N HTS12108 c1cc(cnc1)C2CCCN2S(=O)(=O)c3ccc(cc3)Cl SCR00231 Cc1ccc(cc1)S(=O)(=O)N2CCCC2c3cccnc3 SCR00233 c1cc(cc(c1)NC(=O)n2c3ccncc3c(n2)C(F)(F)F)C(F)(F)F SCR00206 Cc1c(cnn1c2ccccc2)c3csc(n3)c4ccc5c(c4)OCCO5 SCR00143 CCNC(=S)Nc1c(c2c(s1)CC(CC2)C)C#N HTS12065 c1cc(ccc1Cn2c3c(c(=S)[nH]cn3)nn2)F HTS12159 Cc1ccc(cc1)Nc2c3c(ncn2)n(nn3)Cc4ccccc4 HTS12163 c1ccc(cc1)CNC(=O)CC2(CCCCC2)CC(=O)O SCR00228 CCn1c(nnc1Sc2c3c(c4c(cc(nc4s3)C)C)ncn2)c5cccs5 HTS12105 CCNC(=S)NNC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)c4ccco4)N HTS12109 Cc1c(c2c(s1)cc(s2)C(C)(C)C)C(=O)OC GK01845 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)Oc3cc(c(cc3Cl)Cl)Cl)Cc4ccccc4 HTS12287 CC(C)C[C@@H](C(=O)O)NC(=O)COc1ccc(cc1Cl)Cl HTS12320 CS(=O)(=O)c1ccc(cc1)c2csc(n2)c3ccc4c(c3)OCCO4 SCR00150 CCOC(=O)c1ccc(cc1)n2c3ccccc3[nH]c2=S SCR00164 CC(=O)Nc1ccc(cc1)C2=N/C(=C/c3ccc(o3)c4ccc(cc4)[N+](=O)[O-])/C(=O)O2 S05404 CC(=O)Nc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3ccccc3 S01294 CCOc1cc2c(cc1OCC)C3(N(CC2)C(=NN3c4ccccc4)C(=O)c5ccccc5)C HTS12372 c1ccc(cc1)c2cc(c3c4c(c(=O)n(cn4)/N=C/c5ccc(cc5)F)oc3n2)c6ccco6 HTS12113 CCOc1c2c(c3c(cc(nc3s2)C)C)ncn1 HTS12115 c1cc(ccc1S(=O)(=O)n2c3ccncc3c(n2)C(F)(F)F)Cl SCR00211 CCOC(=O)c1c(c(sc1NC(=O)Nc2c(c(c(s2)C)c3ccccc3)C(=O)OCC)C)c4ccccc4 SCR00222 Cc1ccc2c(c1)c(=O)n(c(n2)SCC#C)c3ccc(cc3Cl)Br S06530 c1cc(ccc1CNC(=O)CC2(CCCCC2)CC(=O)O)C(F)(F)F SCR00226 c1cc(ccc1NC(=S)N\2CCN/C2=N\c3ccc(cc3)Cl)Cl SCR00165 Cc1ccc(cc1)Sc2ccccc2NC(=O)c3ccccc3Cl S06334 c1cc(cc(c1)C(F)(F)F)CNC(=O)CC2(CCCCC2)CC(=O)O SCR00225 COc1ccc(cc1)C2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 S01353 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)C RJF01032 Cc1cc(nc2c1c(c(s2)c3n[nH]c(=S)n3C)N)C HTS12143 c1ccc(cc1)n2c(nnc2Sc3c4c(ncn3)n(nn4)Cc5ccccc5Cl)c6cccs6 HTS12147 CCOC(=O)N/N=C(\CN1C(=O)c2ccccc2C1=O)/c3ccc(cc3)OC HTS10912 c1cc(cc(c1)NC(=O)NNC(=O)c2ccc[nH]2)C(F)(F)F SCR00156 c1cnccc1CNC(=O)CC2(CCCCC2)CC(=O)O SCR00227 C(CCNC(=O)/C=C/C(=O)O)CCCNC(=O)/C=C/C(=O)O S02583 COc1cccc(c1)n2c(=S)[nH]nn2 S03209 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)Cc3ccc(cc3)C#N S03993 Cn1c(nnc1Sc2c3c(ncn2)n(nn3)Cc4ccccc4)c5ccccc5 HTS12151 CSc1c2c(ncn1)n(nn2)Cc3ccc(cc3)F HTS12156 c1cc(ccc1Cn2c3c(c(=S)[nH]cn3)nn2)Cl HTS12160 c1ccc(cc1)NC(=S)N2C(C3CCc4ccccc4C3=N2)c5ccc(cc5)Cl HTS12183 c1cc(ccc1CN2C(=O)CSC2=S)C#N S03749 COc1ccccc1Nc2n[nH]c(=S)s2 S03056 c1cc2c(cc1[N+](=O)[O-])cc(s2)C(=O)O MO00646 Cc1cccc(c1)NC2=NCCCS2 S03481 c1ccc2c(c1)CCC3=C2NC(=S)NC3c4ccc(cc4Cl)Cl HTS12668 CCc1ccc(cc1)/N=c\2/c(c(ss2)SC)c3ccccc3 S03960 c1ccc(cc1)C(=S)Nc2ccc3c(c2)OCO3 S06700 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/Cn2nc(nn2)N3CCOCC3)\c4ccc(cc4)Cl SCR00170 CC(=O)c1c(c(c-2n1CCc3c2cc(c(c3)OC)OC)C#N)c4ccc5c(c4)OCO5 HTS12220 Cc1ccc(cc1)/N=N/c2c(n3c(c2C#N)-c4cc(c(cc4CC3)OC)OC)C HTS12221 CCc1c(c([nH]c1C(=O)OCc2ccccc2)C)C SCR00163 c1ccc(cc1)C(=O)Cn2c(=O)c(=O)n3c4ccccc4sc3n2 HTS12853 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccccc3)CN(CC2)C(=O)OCC HTS12856 c1ccc(cc1)n2c(c(cn2)c3nnc(o3)SCc4ccc(cc4)Cl)N HTS12648 c1ccc(cc1)Cn2c(n[nH]c2=S)c3cnn(c3N)c4ccccc4 HTS12650 Cc1c2c(c3cc(cc(c3n1)OC)OC)SCC2 HTS12651 Cc1cc(c(cn1)C(=O)O)C(F)(F)F RF04298 c1ccc(c(c1)NC(=O)CC2(CCCCC2)CC(=O)O)n3cccn3 SCR00366 c1cc2c(ccs2)cc1NC(=O)CC3(CCCCC3)CC(=O)O SCR00355 COc1cc2c(cc1OC)-c3c(c(c(n3CC2)c4cccs4)/N=N/c5ccccc5)C#N HTS12222 Cc1c(c(on1)c2ccccc2)NC(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 SCR00336 CC(=O)C1=NN(C2C1c3cccc4c3c2ccc4)c5ccccc5 HTS12234 Cc1cc(cc(c1)NC(=S)N/N=C/c2cc(cc(c2O)Cl)Cl)C S04739 c1cc(ccc1c2cn3c(n2)SCC3)NC(=O)CC4(CCCCC4)CC(=O)O SCR00358 c1ccn(c1)c2nnc(s2)SCc3c(cccc3Cl)F CD05937 CCOC(=O)c1c(c2c(cc(nc2s1)C)C)NC(=O)Nc3cccc(c3)Cl HTS12660 c1cc(oc1)c2cc(nc3c2c(c(o3)C(=O)NN)N)c4ccco4 HTS12662 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)NN)N)c4ccco4 HTS12663 C[C@@H](C(=O)NCC(C)C)NC(=O)c1ccc(cc1Cl)Cl HTS12322 Cc1c(c(on1)c2ccccc2)NC(=O)Nc3ccc(cc3)OC SCR00334 CCOC(=O)C1=NN(C2C1c3cccc4c3c2ccc4)c5ccc(cc5)C HTS12236 c1cc(cc(c1)S(=O)(=O)N2CCCC2c3cccnc3)C(F)(F)F SCR00232 c1ccc(c(c1)NC(=O)N2CCCC2c3cccnc3)F SCR00234 c1cc(ccc1F)S(=O)(=O)n2c3ccncc3c(n2)C(F)(F)F SCR00212 c1cc(cc(c1)Cl)NC(=O)OC2CN3CCC2CC3 SCR00296 c1ccc2c(c1)C=CN(C2C#N)C(=O)c3c(cccc3F)F S06266 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3ccc(cc3)OCc4ccccc4)N)C HTS12093 C=CCSc1nnc(n1Cc2ccccc2)c3c(c4c(cc(nc4o3)c5ccccc5)c6ccco6)N HTS12079 Cc1cc(nc2c1c3c(s2)c(=O)n(nn3)/N=C/c4ccc(cc4Cl)Cl)C HTS12082 CC\1=NN(C(=O)/C1=C/2\N(N=C(S2)C(=O)C)c3ccccc3)c4ccccc4 HTS12246 CSc1cccc(c1)n2c(=O)c3ccccc3nc2SC S04393 CC1(Cc2cccc(c2O1)C(=O)O)C CC27201 CCO/C=C\1/C(=O)N(C(=S)S1)/N=C/c2cccc(c2)Cl S04280 C[n+]1c(ccc2c1cccc2)/C=C/c3ccc(cc3)Cl.[I-] S05922 C/C(=N\C(c1ccccc1)c2ccccc2)/c3ccccc3O S04658 c1ccc(c(c1)CNC(=S)Nc2ccc(cc2)Cl)Cl S04659 Cc1cc(nc2c1c3c(s2)c(=O)n(nn3)/N=C/c4ccccc4Cl)C HTS12083 c1ccc(c(c1)Cn2c3c(c(ncn3)N4CCCCC4)nn2)Cl HTS12171 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3ccc(cc3)OC)N)C HTS12090 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3cccc(c3)OC)N)C HTS12092 c1ccc(c(c1)NC(=O)OC2CN3CCC2CC3)Cl SCR00295 c1c(cc(c(c1/C=N/CCCC2C=NNC2=O)O)Cl)Cl CD02880 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)N(CC=C)CC=C CD05281 c1cc(ccc1c2c(snn2)N)C(F)(F)F MO00656 Cc1ccc2cc(ccc2n1)NC(=O)c3ccc(nc3C)C(F)(F)F HTS11350 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2C(=S)NCc5ccccc5 HTS12184 c1ccc2c(c1)CCC3C2=NN(C3c4cccs4)C(=S)NC5CCCCC5 HTS12185 CNC(=S)N1C(C2CCc3ccccc3C2=N1)c4ccc(cc4)OC HTS12186 c1cc(cc(c1)S(=O)(=O)n2c3ccncc3c(n2)C(F)(F)F)C(F)(F)F SCR00210 Cn1c(cc(n1)c2ccc(s2)CO)C(F)(F)F MO00643 COc1ccc(c(c1OC)C=C(C#N)C#N)[N+](=O)[O-] S04224 Cc1cc(c(c(c1)O)/C(=N/Cc2ccc(cc2)C#N)/C)C S04296 CC1(N=C(N=C(N1c2cccc(c2)C(F)(F)F)N)N)C.Cl S04343 COc1ccc(c(c1)Sc2ccc(cn2)[N+](=O)[O-])OC CD05135 Cc1c(cnn1c2ccc(cc2)F)CO MO00765 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N4CCCCC4 HTS12192 Cc1ccc2cc(ccc2n1)NC(=O)c3cccc(c3)F HTS11352 Cc1ccc2cc(ccc2n1)NC(=O)c3c(c4ccccc4s3)Cl HTS11351 CCOc1ccc(cc1)C(=O)CC2c3ccccc3C(=O)O2 S05770 c1ccc(c(c1)CN2CCCC2)c3nc(no3)c4ccc(cc4)Cl CD06164 C=CCNC(=S)N1C(C2CCc3ccccc3C2=N1)c4ccccc4Cl HTS12174 c1ccc(cc1)c2csc(n2)c3ccc4c(c3)OCCO4 SCR00151 Cc1ccc(cc1N2C(=O)C=CC2=O)[N+](=O)[O-] S01606 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1F)NC(=O)OCC BTB13196 c1ccc-2c(c1)Cc3c2ccc(c3)C(=O)Cc4ccc(cc4)Br BTB10536 Cc1c(c(c(c(c1C)C)CNC(C)(C)C#C)C)C CD00838 CCOC(=O)c1c(c(sc1NC(=O)Nc2ccc(cc2)Cl)C)c3ccccc3 SCR00216 c1ccc(cc1)c2c3c([nH]c(=O)c2C#N)-c4ccccc4CC3 HTS12688 c1ccc(cc1)/C=N/NC(=O)Cn2c3ccccc3nn2 HTS12689 c1ccc2c(c1)nnn2CC(=O)N/N=C/c3ccc(cc3)Cl HTS12690 c1cc(oc1)CNC(=O)CC2(CCCCC2)CC(=O)O SCR00316 CCN(CC)c1c2ccccc2n3c(n1)c(nn3)C(=O)OCC HTS12191 c1ccc2c(c1)C(=O)N(C2=O)c3c(nns3)c4ccc(cc4)Cl HTS10920 COc1ccc(cc1)c2c(snn2)N3C(=O)c4ccccc4C3=O HTS10913 COc1ccc(cc1)C(=O)CN2C(=O)c3ccccc3C2=O HTS10918 Cc1csc(c1C(=O)OC)NC(=O)CSCc2c(cccc2Cl)F SCR00159 CCOC(=O)/C(=C/1\N(C(=CS1)c2ccc(cc2)C)CC=C)/C#N SCR00157 Cc1c(c(c(c(c1C)C)CSc2nc3ccc(cc3s2)[N+](=O)[O-])C)C S04263 c1cc(nc(c1)NC(=S)Nc2ccc(cc2)F)NC(=S)Nc3ccc(cc3)F S04081 c1cc2c(ccnc2cc1Cl)SCC(=O)O KM10750 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)C4N(C(=O)CS4)Cc5ccco5 SCR00169 COc1ccc(cc1)CNC(=O)CC2(CCCCC2)CC(=O)O SCR00224 c1ccc2c(c1)OCC(O2)CNC(=O)CC3(CCCCC3)CC(=O)O SCR00314 c1ccc(cc1)C(=O)Oc2cc(=O)oc3c2c(=O)n4c5c3cccc5CC4 HTS12693 c1cc(ccc1n2ccnc2)O AC17979 COc1ccc(cc1)CSC(=N)Nc2ccccc2Cl.Cl S05993 c1ccc(cc1)S(=O)(=O)c2cscc2NC(=O)CC3(CCCCC3)CC(=O)O SCR00359 COc1ccc(cc1)n2c(=O)c3cn[nH]c3[nH]c2=S HTS12691 c1cc(ccc1n2c(=O)c3cn[nH]c3[nH]c2=S)Cl HTS12692 Cc1nc2c(cnn2c3ccccc3)c(=O)n1N HTS12936 c1ccc(cc1)C\2=NNC(=O)/C2=C/3\N(N=C(S3)C(=O)Nc4ccccc4)c5ccccc5 HTS12253 COc1ccc(cc1NC(=O)CC2(CCCCC2)CC(=O)O)C(F)(F)F SCR00325 Cc1ccc2cc(ccc2n1)NC(=O)c3cccnc3Sc4ccccc4 HTS11353 c1cc(ccc1C(=O)CSc2nnnn2c3cc(c(cc3Cl)Cl)Cl)Cl S05738 c1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)Sc3ccc(cc3)Cl S04685 c1ccc(cc1)Cn2c(n[nH]c2=S)c3cc(sc3N)c4ccccc4 HTS12890 CCOC(=O)/C(=C(\C)/NCc1ccco1)/C(=S)Nc2ccccc2 HTS12316 Cc1ccsc1c2ccc(cc2)CNC(=O)CC3(CCCCC3)CC(=O)O SCR00320 CCC(C)(C)NC(=S)Nc1ccc(cc1)OCC S05744 c1ccnc(c1)CNC(=O)CC2(CCCCC2)CC(=O)O SCR00318 c1cocc1CNC(=O)CC2(CCCCC2)CC(=O)O SCR00317 CCOC(=O)c1c(nc(s1)c2ccc(s2)c3ccno3)C HTS10580 COc1ccc(cc1OC)CC/N=C/c2cc(cc(c2O)Cl)Cl CD00891 CCCCC(C(=O)N/N=C/c1c(ccc(c1)Br)O)C(=O)N/N=C/c2c(ccc(c2)Br)O S04751 C1CCC(CC1)NC(=S)NC2CCCC2 S04695 c1ccc(c(c1)/C=N/N=C\2/NC(=O)C(S2)CC(=O)O)Cl S04711 CCOC(=O)C1=NN(/C(=C/C2=NCCc3c2cc(c(c3)OC)OC)/S1)c4ccc(cc4)C HTS12258 COc1cc2c(cc1OC)C(=NCC2)/C=C\3/N(N=C(S3)C(=O)c4ccccc4)c5ccc(cc5)Cl HTS12260 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)c3ccc(cc3)C(F)(F)F HTS11881 CCOC(=O)N/N=C(\CN1C(=O)c2ccccc2C1=O)/c3ccc(cc3)Cl HTS10919 Cc1cc(=O)oc2c1ccc(c2)NC(=O)c3ccccc3C(=O)O HTS07014 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)Nc3cccc(c3)S(=O)(=O)N)C HTS06640 c1ccc2c(c1)c(c(c(=O)[nH]2)C#N)O BTB12479 CCOc1ccc2c(c1)cc([nH]2)C(=O)OCC SP01227 Cc1ccc(cc1C)n2c(=S)[nH]nn2 S05727 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nnc(o3)NC(=O)C S04377 C#CCSc1nc2ccccc2c(=O)n1c3ccc(cc3)Cl S04389 c1cc(c(c(c1)Cl)CSc2nc3ccc(cc3s2)[N+](=O)[O-])Cl S04262 CCOC(=O)/C(=N/Nc1ccc(c(c1)C)C)/C SP01147 CCOC(=O)c1c(n[nH]c1N/N=C/c2cc(c(c(c2)OC)OC)OC)C S06465 c1cc(ccc1C#N)c2csc(n2)c3ccc4c(c3)OCCO4 SCR00149 c1ccc(cc1)c2cc(on2)c3csc(n3)c4ccc5c(c4)OCCO5 SCR00148 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccco2)C S06463 CCOC(=O)c1nn(c2n1c3ccccc3n2)c4ccc(cc4)Cl HTS12201 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3Br)Cl S06551 Cc1c(cnn1c2ccc(cc2)OC)NC(=O)N3CCOCC3 HTS12353 Cc1c(cnn1c2ccc(cc2)OC)NC(=O)NCc3cccs3 HTS12354 Cc1c(cnn1c2ccc(cc2)OC)NC(=O)N3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS12358 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccc(cc2)[N+](=O)[O-])C S06462 c1ccc(c(c1)CNC(=O)CC2(CCCCC2)CC(=O)O)F SCR00019 c1ccc(cc1)C(=O)Nc2cccnc2Cl TG00159 c1cc(ccc1NC(=S)N\2CCN/C2=N\c3ccc(cc3)F)F SCR00166 c1cc(ccc1CNC(=O)CC2(CCCCC2)CC(=O)O)F SCR00223 c1ccc2c(c1)c(cs2)NC(=O)NCc3cccs3 HTS12329 Cc1c(cnn1c2ccc(cc2)OC)NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS12352 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N4CCN(CC4)C HTS12193 CCOC(=O)c1c2nc(c3ccccc3n2nn1)Nc4cccc(c4)OC HTS12198 c1ccc(c(c1)NC(=O)c2ccc3c(c2)scn3)F SCR00004 c1cc(cc(c1)Cl)NC(=O)c2ccc3c(c2)scn3 SCR00002 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(c(c3)C)Br S06542 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3C)Br S06544 c1ccc(cc1)n2c(n[nH]c2=S)CN3c4ccccc4Sc5c3cccc5 HTS12653 COc1cc(cc(c1OC)OC)C(=O)NNC(=S)N S05628 c1cc(ccc1NC(=O)c2ccc3c(c2)scn3)Cl SCR00003 c1ccc(cc1)Nc2c3c4c(sc3[nH]c(=S)n2)CCCC4 HTS12645 Cc1ccc2c(c1)c(=O)n(c(n2)SC)c3ccc(cc3)Br S06526 Cc1cc(n(c(=O)c1C#N)/N=c\2/n(cc(s2)c3ccccc3)C4CCCCC4)C SCR00167 c1cc(c(c(c1)F)/N=C/c2ccc(s2)[N+](=O)[O-])F S06368 c1ccc(cc1)C(=O)NC(=S)Nc2c(cccc2F)F S05490 Cc1c(cnn1c2ccc(cc2)OC)NC(=O)NCc3ccccn3 HTS12359 CCOC(=O)c1c(nc(s1)NC(=O)C)C S06594 CCOC(=O)c1c(n[nH]c1N/N=C(\C)/c2ccc(cc2)Br)C S06599 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)N/N=C/c4ccco4 HTS12654 Cc1cc(n(n1)c2ccccc2)NC(=O)CSc3[nH]c4ccccc4n3 HTS12656 c1ccc(c(c1)NC(=O)/C=C/C(=O)O)Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F S03898 CC(=O)Nc1ccc(cc1)/C=C/c2ccc3ccccc3[n+]2C.[I-] S05918 COc1ccc(cc1)C2=Nn3c(=O)c4cc(sc4nc3SC2)c5ccccc5 HTS12841 COc1ccc(cc1)C2=Nn3c(=O)c4c5c(sc4nc3SC2)CCCC5 HTS12846 CCOC(=O)Cn1c(=O)c(=O)n2c3ccccc3sc2n1 HTS12851 CNc1c2c3c(sc2nc(n1)SCC(=O)c4ccccc4)CCCC3 HTS12647 COc1cc(c(cn1)C(=O)Nc2ccc(cc2)Cl)C(F)(F)F RF04301 Cc1c2c(c3cc(ccc3n1)Cl)SCC2 HTS12652 c1ccc2c(c1)nc(s2)c3csc(n3)c4ccc5c(c4)OCCO5 SCR00138 c1ccc2c(c1)c(co2)c3csc(n3)c4ccc5c(c4)OCCO5 SCR00146 c1cc2cccnc2c(c1)S(=O)(=O)N3CCCC3c4ccc(cc4)F SCR00181 CC(C)(C#C)NC(=N)N[N+](=O)[O-] S03966 COc1ccc(c(c1)OC)S(=O)(=O)N2CCC(=CC2)c3ccccc3 SCR00422 c1cc2c(cc1N)N3CCN=C3S2 AC12308 Cc1cc(nc2c1c3c(s2)C(=O)N(CC(=O)N3)c4cccc(c4)C(F)(F)F)C HTS12902 Cc1ccc(cc1)N2C3c4cc(c(cc4CCN3C(=N2)C(=O)C)OC)OC HTS12218 CCOc1cc2c(cc1OCC)C3N(CC2)C(=NN3c4ccc(cc4)Cl)C(=O)OCC HTS12219 c1ccc(c(c1)C(F)(F)F)NC(=O)N2CCCC2c3cccnc3 SCR00267 c1ccc2c(c1)-n3c(nnc3c4ccncc4)CS2 HTS12905 c1ccc2c(c1)-n3c(nnc3c4cccs4)CS2 HTS12906 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc(s3)c4ccno4 SCR00079 c1ccc(cc1)c2c(c(=O)nc3n2c(nn3c4ccccc4)c5ccccc5)C#N HTS12240 Cc1ccc(cc1)N2/C(=C\3/C(=NN(C3=O)c4ccccc4)c5ccccc5)/SC(=N2)C(=O)c6cccs6 HTS12245 CCOC(=O)c1c(c(sc1NS(=O)(=O)c2ccc(cc2)F)C)c3ccccc3 SCR00220 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CCN3CCOCC3 HTS12309 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4ccc(cc4)Cl)C1 HTS12862 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc4c(c3)OCCCO4 SCR00072 Cc1ccccc1NC(=O)c2ccc3c(c2)scn3 SCR00007 Cc1cc(cc(c1)NC(=O)NCc2c(onc2c3ccccc3)C)C SCR00090 Cc1ccc(cc1)N2/C(=C/C3=NCCc4c3cc(c(c4)OC)OC)/SC(=N2)C(=O)c5cccs5 HTS12259 CCOC(=O)c1nn(c2n1c(c(c(=O)n2)C#N)c3ccccc3)c4ccccc4 HTS12241 CCn1c(=O)c2c(c(sc2[nH]c1=S)C)C HTS12827 Cn1c2c(nc1Oc3ccc(cc3)F)n(c(=O)n(c2=O)Cc4ccccc4)C HTS12290 c1ccc2c(c1)ccc(n2)NC(=O)CC3(CCCCC3)CC(=O)O SCR00353 COc1ccc2c(n1)sc(n2)NC(=O)CC3(CCCCC3)CC(=O)O SCR00351 c1cc(ccc1C(=O)O/N=C/c2ccc(c(c2)Cl)F)C(F)(F)F SEW02046 Cc1c(sc(c1C#N)NC(=O)CN2CCOCC2)C HTS12833 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3cccc(c3)c4ccnc(n4)C SCR00078 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4ccc(cc4)C)C1 HTS12863 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4ccc(c(c4)Cl)Cl)C1 HTS12864 c1ccnc(c1)c2ccc(s2)S(=O)(=O)N3CCCC3c4ccc(cc4)F SCR00180 c1ccc(cc1)NNC(=S)N/N=C/c2ccc(s2)[N+](=O)[O-] S05863 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)CC(=O)N)C1 HTS12871 Cc1c(c(on1)c2ccccc2)NC(=O)Nc3ccc4c(c3)ccs4 SCR00343 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc(cc3F)F SCR00061 Cc1c(c(no1)c2ccccc2)CNC(=O)c3c(onc3c4ccc(cc4)F)C SCR00042 C=CCn1c(nnc1Sc2ncc(c(n2)N)C#N)c3cccs3 HTS12722 c1ccc(cc1)Cn2c(nnc2Sc3ncc(c(n3)N)C#N)c4ccc(cc4)Cl HTS12723 Cc1c(c(no1)c2ccccc2)CNC(=O)C3CCCCC3 SCR00021 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2C(=O)CSc5nnc(o5)c6ccncc6 HTS12673 Cc1c(sc(n1)C)S(=O)(=O)NCc2c(onc2c3ccccc3)C SCR00068 Cc1c(c(on1)C)S(=O)(=O)NCc2c(onc2c3ccccc3)C SCR00063 CCOC(=O)c1c2c(sc1NC(=S)N3CCOCC3)CN(CC2)C(=O)OCC HTS12876 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccccc3 SCR00058 COc1ccc(c(c1)OC)Nc2ncc(c(n2)N)C#N HTS12727 COc1cccc(c1)Nc2ncc(c(n2)N)C#N HTS12728 CCOC(=O)C1CCN(CC1)Cc2nc(no2)c3ccc(cc3)Cl CD02888 CC1=C(C(NC(=S)N1)c2ccc(cc2)F)C(=O)OC HTS12878 CC1=C(C(NC(=S)N1)c2ccc(cc2)OCc3ccccc3)C(=O)OC HTS12879 c1ccc2c(c1)nc(s2)Sc3ncc(c(n3)N)C#N HTS12725 COc1ccc(cc1)C2=Nn3c(nnc3SC2)c4ccccc4 HTS12734 CC1=Nn2c(nnc2SC1)c3ccc(cc3)Cl HTS12737 c1ccc2c(c1)CCC3=C2N=C4N(C3c5ccc(cc5)Cl)C(=O)CS4 HTS12674 COc1ccc(cc1)/C=C(\C#N)/C(=O)N HTS12676 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2ccc(c(c2)Cl)Cl S06727 c1cc(ccc1C(F)(F)F)NC(=O)c2ccc3c(c2)scn3 SCR00010 COc1ccc(cc1)NC(=O)c2ccc3c(c2)scn3 SCR00009 CC(=O)COc1c(c(c2c(n1)-c3ccccc3CC2)c4ccco4)C#N HTS12680 c1ccc(cc1)c2nnc3n2N=C(CS3)c4cccs4 HTS12739 COc1ccc(cc1)C2=Nn3c(nnc3SC2)c4ccc(cc4)Cl HTS12740 c1ccc-2c(c1)CCc3c2[nH]c(=O)c(c3c4ccc(cc4)Cl)C#N HTS12684 COc1cc(cc(c1OC)OC)CN2CCCN(C2c3ccc(c(c3)Cl)Cl)Cc4cc(c(c(c4)OC)OC)OC S04321 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)OC(=O)c5cccs5 HTS12707 c1cc(sc1)C2=Nn3c(nnc3SC2)c4ccc(cc4)Cl HTS12738 COc1ccc(cc1)c2c3c(nc(c2C#N)OC)-c4ccccc4CC3 HTS12678 c1ccc-2c(c1)CCc3c2[nH]c(=O)c(c3c4cccnc4)C#N HTS12686 COC(=O)c1cc2cc(ccc2s1)N MO00936 CC(C)(C)c1ccc(cc1)/N=C/c2ccc(c(c2)Cl)Cl S06755 CC(C(=O)Nc1ccc(cc1)C(C)(C)C)Oc2ccc(cc2Cl)Cl S06790 c1ccc2c(c1)nnn2Cc3nnc4n3N=C(CS4)c5ccc(cc5)Cl HTS12703 c1ccc(cc1)C2=Nn3c(nnc3SC2)Cn4c5ccccc5nn4 HTS12704 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)OC(=O)c5ccccc5 HTS12709 c1ccc2c(c1)C(OC2=O)CC(=O)c3cccc(c3)[N+](=O)[O-] S05975 c1ccc2cc(ccc2c1)C(=O)CSc3nnnn3c4cccc5c4cccc5 S05798 C/C(=N\N=C/1\NC(=O)C(S1)CC(=O)O)/c2ccc(cc2)F S04356 C/C(=N\N=C/1\NC(=O)C(S1)CC(=O)O)/c2ccccc2Cl S04363 COc1cccc(c1)N2CC(=O)N(CC2=O)N HTS12916 COc1cccc(c1)N2CC(=O)N(CC2=O)NC(=O)Nc3cccc(c3)Cl HTS12924 COc1cccc(c1)N2CC(=O)N(CC2=O)NC(=O)NC3CCCCC3 HTS12925 Cc1ccc(cc1)N2CC(=O)N(CC2=O)NC(=O)Nc3ccc(c(c3)Cl)Cl HTS12926 CC1(N=C(N=C(N1c2cc(c(cc2Cl)Cl)Cl)N)N)C.Cl S04349 Cc1ccc2c(c1)c(=O)n(c(n2)C(F)(F)F)c3ccc(cc3)Cl S04351 c1ccc-2c(c1)CCc3c2[nH]c(=O)c(c3c4cccs4)C#N HTS12683 c1ccc-2c(c1)CCc3c2[nH]c(=O)c(c3c4ccco4)C#N HTS12687 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3ccccc3 SCR00378 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)OC(=O)c5cccc(c5)[N+](=O)[O-] HTS12710 c1ccc(cc1)NC(=O)NC(=O)CSc2nnc(o2)c3ccncc3 HTS12714 CCOC(=O)c1c(c(sc1NS(=O)(=O)c2ccc(cc2)C(F)(F)F)C)c3ccccc3 SCR00218 c1cc(cc(c1)Cl)CNC(=O)CC2(CCCCC2)CC(=O)O SCR00017 c1ccc(cc1)C(c2ccccc2)N3CC(C3)C(=O)Nc4nc5ccc(cc5s4)Cl SCR00197 COC(=O)c1ccc(nc1)N2CCOCC2 CC17522 Cc1c(c(no1)c2ccccc2)CNC(=O)Nc3ccc(c(c3)OC4CCCC4)OC SCR00092 C/C(=N\N=C/1\NC(=O)C(S1)CC(=O)O)/c2ccc(cc2)Br S04364 c1cc(ccc1c2ccsc2)C(=O)O MO07004 c1cc(ccc1NC(=O)CC2(CCCCC2)CC(=O)O)N3CCCCC3 SCR00327 c1cc(c(cc1NC(=O)CC2(CCCCC2)CC(=O)O)Cl)N3CCOCC3 SCR00324 c1cc(sc1)c2ccc(cc2)CNC(=O)CC3(CCCCC3)CC(=O)O SCR00321 COc1ccc(cc1)n2c(n[nH]c2=S)c3cc(sc3N)c4ccccc4 HTS12888 Cc1ccc(cc1)N2CC(=O)N(CC2=O)NC(=O)CN3CCN(CC3)c4ccccc4 HTS12893 c1ccc2c(c1)CCN2CC(=O)NN3CC(=O)N(CC3=O)c4ccc(cc4)Cl HTS12894 Cc1cccc(c1)C(=O)Nc2nnc(s2)SCC#C S06831 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3cccc(c3)Br SCR00081 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3c(nc4n3ccs4)Cl SCR00080 Cc1c(c(no1)c2ccccc2)CNC(=O)Nc3ccc(cc3F)F SCR00089 Cc1c(c(no1)c2ccccc2)CNC(=O)Nc3cccc(c3)OC SCR00088 c1cc(cc(c1)N2CC(=O)N(CC2=O)NC(=O)Nc3ccc(cc3)Cl)C(F)(F)F HTS12930 c1ccc(cc1)n2c3c(cn2)c(ncn3)n4c(c(cn4)C#N)N HTS12933 c1cc(ccc1CNC(=O)CC2(CCCCC2)CC(=O)O)Cl SCR00018 C=CCn1c(n[nH]c1=S)c2cc(sc2N)c3ccccc3 HTS12889 Cc1c(c(no1)c2ccccc2)CNC(=O)Nc3ccc(cc3)C(F)(F)F SCR00091 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3ccccc3F SCR00421 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3cccs3 SCR00418 Cc1c(c(no1)c2ccccc2)CNC(=O)NC3CCN(CC3)C(=O)OCc4ccccc4 SCR00085 Cc1c(c(no1)c2ccccc2)CNC(=O)Nc3cccc(c3)Cl SCR00082 C[C@@H](C(=O)NCc1ccco1)NC(=O)c2ccc(cc2Cl)Cl HTS12326 Cc1ccc(cc1)Cn2c3c(nc2NCc4cccnc4)n(c(=O)n(c3=O)C)C HTS12274 CCN1CCN(CC1)c2nc3c(n2Cc4c(cccc4Cl)Cl)c(=O)n(c(=O)n3C)C HTS12275 Cc1c(c(on1)c2ccccc2)NC(=O)NCc3c(onc3c4ccccc4)C SCR00087 c1ccc(cc1)COc2ccc(cc2)/C=C/3\C(=O)OC(=N3)c4ccccc4 HTS13058 CCn1c(n[nH]c1=S)c2cc(sc2N)c3ccccc3 HTS12891 c1cc(ccc1n2cncn2)O AC18635 c1c(c(=O)[nH]c(=O)[nH]1)N2CCCCCC2 HTS12299 Cc1c(cnn1c2ccccc2)S(=O)(=O)NCc3c(onc3c4ccccc4)C SCR00075 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2cccc(c2)[N+](=O)[O-] S06853 Cc1ccc(o1)/C=N/NC(=O)c2cc(sc2N)c3ccccc3 HTS13008 c1ccc(cc1)C(=O)N/C(=C/c2ccccc2Cl)/C(=O)NN HTS13060 CN(C)c1ccc(cc1)c2ccncc2 HTS12311 Cc1cc(ccc1Cl)Oc2nc3c(n2C)c(=O)n(c(=O)n3C)Cc4ccccc4 HTS12281 Cc1cc(cc(c1Cl)C)Oc2nc3c(n2C)c(=O)n(c(=O)n3C)C HTS12282 c1ccc(c(c1)NC(=O)c2ccc3c(c2)scn3)Cl SCR00001 c1ccc(cc1)C\2=NOC(=O)/C2=C/3\N(N=C(S3)C(=O)c4cccs4)c5ccc(cc5)Cl HTS12254 Cn1c2c(nc1NCc3ccccn3)n(c(=O)n(c2=O)C)C HTS12276 Cc1c(c(no1)c2ccccc2Cl)c3nnc(o3)NC(=O)C S04380 c1ccc2c(c1)nc(s2)SCc3ccc(cc3)CSc4nc5ccccc5s4 HTS12302 c1cc(c(cc1Cl)Cl)COc2ccncc2 HTS12304 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc(cc3)n4cccn4 SCR00076 Cc1ccc(cc1)N2CC(=O)Nc3c4c(cc(nc4sc3C2=O)C)C HTS12903 Cc1cccc(c1)/N=C/c2ccc(s2)[N+](=O)[O-] S05792 Cc1c(c(nn1c2ccc(cc2)[N+](=O)[O-])c3cccs3)C(=O)C HTS12208 CCCCOc1ccc(cc1)Oc2nc3c(n2Cc4c(cccc4Cl)Cl)c(=O)n(c(=O)n3C)C HTS12284 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)Oc3ccc(cc3)OCc4ccccc4)Cc5c(cccc5Cl)F HTS12285 Cc1ccc(cc1)N2CC(=O)N(CC2=O)NC(=O)c3c(c4c(cc(nc4s3)C)C)N HTS12900 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3cc4ccccc4s3 SCR00070 c1ccc(cc1)c2nnc3n2-c4ccccc4SC3 HTS12907 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccc(c(c2)Cl)Cl HTS12910 c1cc(ccc1NC(=O)c2ccc3c(c2)scn3)F SCR00006 CCOC(=O)C1=NN(C2N1CCc3c2cc(c(c3)OC)OC)c4ccccc4 HTS12216 CCOC(=O)C1=NN(C2C1c3cccc4c3c2ccc4)c5cccc(c5)Cl HTS12235 c1cc(cnc1)c2nc(on2)CCCC(=O)O DP01249 c1ccc2c(c1)CCC3=C2NC(=S)NC3c4ccc(cc4)Cl HTS12669 c1ccc2c(c1)C(=O)N(C2=O)/N=C/c3ccco3 S05898 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc4c(c3)N(CCO4)C SCR00073 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc4c(c3)OCCO4 SCR00065 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3cccc(c3)Cl SCR00062 COc1cc(cc(c1OC)OC)C2OC(=O)c3ccccc3S2 S04250 COc1ccc(cc1Br)C2OC(=O)c3ccccc3S2 S04252 CCOC(=O)c1cc(sc1NC(=S)OCC)c2ccccc2 HTS12830 Cc1ccc(cc1)S(=O)(=O)NCc2c(onc2c3ccccc3)C SCR00060 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccccc3[N+](=O)[O-] SCR00059 c1ccc(cc1)c2cc(=O)nc3n2c(nn3c4ccccc4)C(=O)c5cccs5 HTS12239 Cc1c(c(no1)c2ccccc2)CNC(=O)C3CCN(CC3)c4nccc(n4)C(F)(F)F SCR00026 c1cc(sc1)c2nc(cs2)CNC(=O)CC3(CCCCC3)CC(=O)O SCR00313 Cc1c(c(on1)c2ccccc2)NC(=O)Nc3ccccc3 SCR00333 c1cc(cc(c1)C(F)(F)F)CN2CCOCC2.Cl CD03196 Cc1cc(ccc1NC(=S)NCCO)F S06000 c1cc(ccc1c2nc3c(c(n2)O)CS(=O)(=O)CC3)C(F)(F)F RF03922 Cc1nn(c(=O)o1)c2c(cc(cn2)C(F)(F)F)Cl RF04816 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(c(c3)Cl)Br S06547 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)CC(=O)c4ccc(cc4)Br)C1 HTS12866 c1ccc2c(c1)CCCN2C(=O)CSc3nc4ccccc4o3 HTS12700 c1ccc2c(c1)nnn2Cc3nnc4n3N=C(CS4)c5ccc(cc5)[N+](=O)[O-] HTS12702 CC(=O)COc1c(c(c2c(n1)-c3ccccc3CC2)c4ccc(cc4)Cl)C#N HTS12677 CCOC(=O)N1CCc2c(sc3c2c(=O)n4c(n3)SCC(=N4)c5ccc(cc5)OC)C1 HTS12872 c1ccc2c(c1)C(=O)N(C2=O)CNc3ccccc3Br S06765 CC1=C(C(N2C(=C(SC2=N1)C#N)N)c3ccc(cc3)F)C(=O)OC HTS12881 CCOC(=O)c1c(n[nH]c1N/N=C(\C)/c2ccccc2)C S06602 c1ccc(cc1)C(=O)NNC2=Nc3ccccc3SC2 HTS12885 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)OC(=O)c5ccc(cc5)Cl HTS12705 CC1CN(CC(O1)C)CCCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD06129 CC(C)(C)c1ccc(cc1)Nc2n[nH]c(=S)s2 S06750 CCOC(=O)c1c2c(sc1NC(=S)N3CCCc4c3cccc4)CN(CC2)C(=O)OCC HTS12877 c1cc(cc(c1)NC(=O)OC2CN3CCC2CC3)C(F)(F)F SCR00301 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)OC(=O)c5ccco5 HTS12708 c1ccc2c(c1)nc(s2)c3ccc(cc3)NC(=O)c4ccno4 SCR00396 CC(C)(C)c1ccc(cc1)NC(=O)C(C)(C)C S06749 C=CCn1c(n[nH]c1=S)c2cccc(c2)[N+](=O)[O-] HTS12912 c1ccc(cc1)n2c(n[nH]c2=S)c3cccc(c3)[N+](=O)[O-] HTS12913 Cc1nc2c(cc(s2)c3ccccc3)c(=O)o1 HTS12914 CNc1c2c3c(sc2[nH]c(=S)n1)CCCC3 HTS12644 CCOC(=O)CSc1nc(c2c3c(sc2n1)CCCC3)NC HTS12646 CSC1=C(C(=O)NC(S1)c2ccc(cc2)[N+](=O)[O-])C#N CD01346 CCOC(=O)c1c(n[nH]c1N/N=C/c2c(cccc2Cl)F)C S06601 c1cc2c(cc1Cl)c(c(nn2)C(=O)N)N HTS12655 c1ccc(cc1)C(=O)CSc2nnc(o2)c3cnn(c3N)c4ccccc4 HTS12649 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4ccc(cc4)F)C HTS12658 CSc1c(/c(=N/c2ccc(c(c2)F)F)/ss1)c3ccccc3 S03955 c1ccc(cc1)c2ccc(cc2)c3cc(c(c(=O)[nH]3)C#N)c4ccccc4 S06683 c1c(cnc2c1sc(c2N)C(=O)O)C(F)(F)F SEW04490 c1cc(ccc1CSc2ncc(c(n2)N)C#N)Cl HTS12716 c1cc(cc(c1)F)NC(=O)c2ccc3c(c2)scn3 SCR00005 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)F)/C(=O)N2 HTS13052 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4ccccc4)C1 HTS12996 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)C)C1 HTS12998 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)CC=C)C1 HTS12999 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)NC(=N2)c3ccccc3 HTS13048 c1ccc(cc1)/C=C(\C(=O)NN)/NC(=O)c2ccccc2 HTS13059 c1cc(oc1)c2cc(nc3c2c4c(o3)c(=O)[nH]cn4)c5ccc(cc5)Cl HTS12661 c1cc(oc1)c2cc(nc3c2c(c(o3)C(=O)NN)N)c4ccc(cc4)Cl HTS12665 CCOC(=O)c1c(cc([nH]1)C)C KM10848 c1ccc2c(c1)c(cs2)c3csc(n3)c4ccc5c(c4)OCCO5 SCR00140 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)c4ccc(cc4)Cl)C1 HTS13001 c1ccc(cc1)/C=C/2\C(=O)NC(=N2)c3ccccc3 HTS13055 COc1ccc(cc1)/C=C/2\C(=O)NC(=N2)c3ccccc3 HTS13056 c1cc(oc1)C2N(CCCN2Cc3ccc(cc3)F)Cc4ccc(cc4)F SCR00444 c1ccc2c(c1)nc(s2)c3ccc(cc3)NC(=O)Nc4ccc(cc4Cl)Cl SCR00397 c1cc2c(cc1F)c(c[nH]2)CC(C(=O)O)N AC11968 CCNc1cc(=N)n(c2c1c(n[nH]2)N)CC CD03750 CCOC(=O)c1c2c(sc1NC(=S)N3CCN(CC3)C)CN(CC2)C(=O)OCC HTS13003 c1ccc(cc1)c2cc(c(s2)N)C(=O)N/N=C/c3ccccc3Cl HTS13007 c1cc(ccc1N2CC(=O)N(CC2=O)NC(=O)CN3CCOCC3)Cl HTS12895 Cc1nc2c(cnn2c3ccccc3)c(=O)n1/N=C/c4cccs4 HTS12896 c1ccc2c(c1)CCC3=C2NC(=S)NC3c4cccnc4 HTS12666 COc1ccc(cc1)n2c(n[nH]c2=S)c3ccc(cc3)Cl HTS12898 CC(C)(C#C)NC(=O)Nc1cnccc1C(F)(F)F RF04022 c1ccc(cc1)c2cc(=O)nc3n2c(nn3c4ccc(cc4)[N+](=O)[O-])c5ccco5 HTS12238 CCc1ccnc(c1)NC(=O)CC2(CCCCC2)CC(=O)O SCR00352 c1cc(ccc1C(F)(F)F)NC(=O)OC2CN3CCC2CC3 SCR00302 Cc1cc(nn1C)C(=O)NCc2cc(cc3c2OCOC3)F SCR00648 Cc1cc(nn1C)C(=O)NCc2cc(oc2C(F)(F)F)C SCR00646 Cc1cc(nc2c1c3c(s2)c(=O)n(c(n3)C)/N=C/c4ccc(cc4)Cl)C HTS12915 C=CCn1c(nnc1SCC(=O)Nc2c(cnn2c3ccccc3)C#N)c4ccncc4 HTS12755 CNC(=O)Nc1cnccc1C(F)(F)F RF03993 c1ccc(cc1)C(=O)N/C(=C\c2cccs2)/C(=O)N/N=C/c3ccc(cc3Cl)Cl HTS13067 CN1C(=N/C(=C/c2cc(c(c(c2)OC)OC)OC)/C1=O)c3ccccc3 HTS13069 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)CC(=O)C)C1 HTS12869 Cc1c(c(on1)c2ccccc2)NC(=O)Nc3ccc(cc3)c4nc5ccccc5s4 SCR00399 c1ccc(cc1)n2c(c(cn2)C#N)NC(=O)CSc3nnc(o3)c4ccco4 HTS12746 c1ccc(cc1)n2c(c(cn2)C#N)NC(=O)CSc3nnc(o3)c4ccc(cc4)Cl HTS12747 CN(C)Cc1c[nH]c2c1cc(cc2)OC AC12586 c1ccc(cc1)n2c(c(cn2)C#N)NC(=O)CSc3nc4ccccc4s3 HTS12749 CCOc1cc2c(cc1OCC)-c3c(c(c(n3CC2)c4ccccc4)/N=N/c5ccccc5)C#N HTS12223 COc1cc2c(cc1OC)-c3c(c(c(n3CC2)C(=O)c4ccccc4)c5ccc6c(c5)OCO6)C#N HTS12224 Cc1c(sc2c1c(=O)n3c(n2)SCC(=N3)c4ccc(cc4)OC)C HTS12823 Cc1ccccc1n2c(=O)c3cc(sc3[nH]c2=S)c4ccccc4 HTS12829 c1ccc(c(c1)N2CC(=O)N(CC2=O)N)F HTS12917 c1cc(cc(c1)N2CC(=O)N(CC2=O)N)C(F)(F)F HTS12918 c1cc(ccc1N2CC(=O)N(CC2=O)N)Cl HTS12919 c1cc(sc1)c2nnc(n2c3ccc(cc3)Cl)Sc4ncc(c(n4)N)C#N HTS12721 c1cc(ccc1N2CC(=O)N(CC2=O)NC(=O)NC3CCCCC3)Cl HTS12923 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3Cl)Cl)/C(=O)N2 HTS13050 Cc1ccc(o1)/C=C/2\C(=O)NC(=N2)c3ccccc3 HTS13051 c1ccc(cc1)C(=O)CSc2nnc3n2CCCN3 HTS12769 CC(C)(C)c1ccc(cc1)/N=C/c2cc(ccc2O)Cl S06786 c1ccc(cc1)CN(Cc2ccccc2)c3c4cc(sc4ncn3)c5ccccc5 HTS13102 COc1ccc(cc1)/C=C/2\C(=O)N(C(=N2)c3ccccc3)Cc4ccc(cc4)F HTS13079 COc1ccc(c(c1)OC)n2cc([nH]c2=S)c3ccccc3 HTS13083 c1ccc(cc1)C2=N/C(=C/c3cccs3)/C(=O)N2Cc4ccc(cc4)Cl HTS13080 CCOC(=O)c1c2c(sc1NC(=S)N3CCc4c3cccc4)CN(CC2)C(=O)OCC HTS12874 CNc1nnc(s1)SCc2ccc(cc2)Cl S06812 c1cc2c3c(c1)c4c(c(cc(=O)o4)OC(=O)c5ccco5)c(=O)n3CC2 HTS12695 Cc1ccc(cc1)N2CC(=O)N(CC2=O)N HTS12920 Cc1ccc(cc1)NC(=O)NN2CC(=O)N(CC2=O)c3ccc(cc3)Cl HTS12921 c1ccc(cc1)NC(=O)NN2CC(=O)N(CC2=O)c3ccc(cc3)Cl HTS12922 c1cc(ccc1Nc2ncc(c(n2)N)C#N)F HTS12726 CN1CCN(CC1)CC(=O)Nc2c(cnn2c3ccccc3)C#N HTS12760 Cc1ccc(cc1)NC(=O)N2CCCn3c2nnc3SCC(=O)c4ccccc4 HTS12764 c1ccc(cc1)CN2CCCC(C2)O.Cl AC13425 c1ccc(cc1)C2=N/C(=C/c3ccccc3Cl)/C(=O)N2 HTS13054 c1c(c(cc2c1[nH]c(=S)[nH]2)Cl)C(F)(F)F S05816 c1ccc2c(c1)CCC3=C2NC(=S)NC3c4ccccc4Cl HTS12670 COc1ccc(cc1)C2C3CCc4ccccc4C3=NN2C(=O)CN5CCOCC5 HTS12672 Cc1ccc(c(c1)C)n2c(noc2=O)c3cnc(cc3C(F)(F)F)OC RF05245 Cc1ccc(cc1)N2CC(=O)N(CC2=O)NC(=O)Nc3cccc(c3)C(F)(F)F HTS12927 c1cc2c(cc1F)[nH]cc2CC(C(=O)O)N AC14674 c1c(cc(cc1Cl)Cl)NC(=O)CC2(CCCCC2)CC(=O)O SCR00330 c1cc2c(cc1/C=N/Nc3nc4c(ncnc4n3[C@@H]5[C@H]([C@H]([C@@H](O5)CO)O)O)N)OCO2 HTS12292 c1ccc(cc1)c2cc3c(ncnc3s2)N/N=C/c4ccncc4 HTS13112 CC(=NNc1nc2c(n1C)c(=O)n(c(=O)n2C)C)C HTS12295 C/C(=N\Nc1nc2c(n1C)c(=O)n(c(=O)n2C)C)/c3ccccc3 HTS12296 Cn1c2c(nc1NN=C3C(=O)NC(=O)NC3=O)n(c(=O)n(c2=O)C)C HTS12297 Cc1nc2c(cnn2c3ccccc3)c(=O)n1NC(=O)Nc4ccc(c(c4)Cl)Cl HTS12937 COc1cc(cc(c1OC)OC)/C=N/NC(=O)c2cc(sc2N)c3ccccc3 HTS12884 c1ccc2c(c1)N=C(CS2)NNC(=O)c3cccs3 HTS12886 CCOC(=O)c1c(c(sc1NC(=S)N2CCOCC2)C)C HTS12982 c1ccc(c(c1)N2CC(=O)N(CC2=O)NC(=O)Nc3ccc(cc3)Cl)F HTS12929 c1ccc(cc1)NC(=O)NN2CC(=O)N(CC2=O)c3cccc(c3)C(F)(F)F HTS12931 c1ccc2c(c1)-n3c(n[nH]c3=O)CS2 HTS12932 CC1=Nn2c(nnc2SC1)c3ccccc3 HTS12736 COc1cccc(c1CNC(=O)c2cnc(cc2C(F)(F)F)OC)OC RF04465 CCOC(=O)COc1c(c(c2c(n1)-c3ccccc3CC2)c4ccco4)C#N HTS12679 c1ccc-2c(c1)CCc3c2[nH]c(=O)c(c3c4ccc(cc4)F)C#N HTS12681 c1ccc2c(c1)c(cs2)NC(=O)Nc3ccc4c(c3)OCCCO4 HTS12333 c1ccc(cc1)c2cc(c(s2)N)c3n[nH]c(=S)n3c4ccc(cc4)F HTS13015 c1ccc(cc1)c2cc(c(s2)N)c3n[nH]c(=S)n3C4CCCCC4 HTS13016 CSc1c(c(nn1C(=O)C2CC2)N)c3ccccn3 SCR00489 c1ccc(c(c1)CSc2nnc3n2CCCN3)Cl HTS12770 c1cc(sc1)C(=O)CSc2nnc3n2CCCN3 HTS12771 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COC(=O)c3ccc(c(c3)OC)OC)OC(=O)c4ccc(c(c4)OC)OC HTS12308 c1ccc(c(c1)c2n[nH]c(=S)n2c3cccc(c3)C(F)(F)F)Cl HTS12942 CCn1c(n[nH]c1=S)c2ccccc2Cl HTS12943 Cc1ccc(cc1)N2CC(=O)N(CC2=O)/N=C/c3ccncc3 HTS12946 c1ccc2c(c1)N=C(CS2)NNC(=O)c3ccc(cc3)Cl HTS13013 c1ccc2c(c1)N=C(CS2)NNC(=O)c3ccc(cc3)F HTS13014 Cn1c(nnc1S)c2c(cc(cn2)C(F)(F)F)Cl SPB05806 c1cc(c(cc1Cl)Cl)/C=N/N2C(=O)/C(=C/c3c(c(c(c(c3F)F)F)F)F)/SC2=S S04288 CCOC(=O)c1c(n[nH]c1N/N=C(\C)/c2ccccc2Cl)C S06600 c1ccc(cc1)c2cc(c(s2)N)C(=O)NN HTS13018 CCC(C)[C@@H](C(=O)O)NC(=O)c1ccco1 HTS12321 CN1CCN(CC1)CC(=O)NN2CC(=O)N(CC2=O)c3ccc(cc3)Cl HTS13019 c1ccc2c(c1)-n3c(nnc3c4ccc(cc4)F)CS2 HTS13025 c1ccc2c(c1)-n3c(nnc3c4ccc(cc4)Cl)CS2 HTS13026 c1ccc2c(c1)C(=O)N(C2=O)c3c(nns3)c4ccc(cc4)C(F)(F)F HTS11883 C1COCCN1CCCNc2nc3c(=O)[nH]c(nc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS12310 CCOC(=O)c1c2c(sc1NC(=O)CN3CCCC3)CN(CC2)C(=O)OCC HTS12778 CCOC(=O)c1cc(sc1N)c2ccccc2 HTS12824 c1ccc(cc1)c2cc3c(s2)[nH]c(=S)n(c3=O)c4ccccc4 HTS12826 COc1ccc(c(c1)OC)n2c(=O)c3cc(sc3[nH]c2=S)c4ccccc4 HTS12828 c1cc(oc1)/C=N/N2CC(=O)N(CC2=O)c3ccc(cc3)Cl HTS12951 Cc1ccc(o1)/C=N/N2CC(=O)N(CC2=O)c3cccc(c3)OC HTS12953 c1cc(cnc1)/C=N/N2CC(=O)N(CC2=O)c3ccc(cc3)Cl HTS12954 Cc1cc(c(cc1Cl)C)SCc2nc(on2)c3c(noc3C)C SEW00844 COc1cccc(c1)N2CC(=O)N(CC2=O)NC(=O)CN3CCCC3 HTS13021 CCCN/C(=C(\C(=S)Nc1ccc(cc1)OCC)/C(=O)OCC)/C HTS12314 Cc1cc(nc2c1c(c(s2)C(=O)NN3CC(=O)N(CC3=O)c4cccc(c4)C(F)(F)F)N)C HTS13023 Cc1cccc(c1NC(=O)c2cnccc2C(F)(F)F)C RF04375 c1ccc(cc1)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)F S06672 c1cc(sc1)c2csc(n2)c3ccc4c(c3)OCCO4 SCR00141 c1ccc(cc1)c2cc3c(s2)nc4n(c3=O)N=C(CS4)c5cccs5 HTS12839 c1ccc2c(c1)-n3c(nnc3c4cccc(c4)[N+](=O)[O-])CS2 HTS13027 CCCN/C(=C/C(=S)Nc1cccc2c1cccc2)/c3ccc(cc3)OC HTS12315 CC(C)C[C@@H](C(=O)O)NC(=O)c1ccc(cc1Cl)Cl HTS12319 Cc1cc(nc2c1c3c(s2)c(=O)n(c(n3)C)NC(=O)Nc4ccccc4)C HTS13028 Cc1nc2c(c(=O)n1NC(=O)CN3CCN(CC3)C)ncn2c4ccccc4 HTS13033 CC(C)N(Cc1ccccc1)S(=O)(=O)c2ccc(s2)CNC(=O)c3ccc(cc3)Cl HTS07891 c1ccc(cc1)COc2ccc(cc2)/C=C/3\C(=O)N(C(=N3)c4ccccc4)CC(=O)N HTS13068 CCOC(=O)CN1C(=N/C(=C/c2ccc(o2)C)/C1=O)c3ccccc3 HTS13072 CCOC(=O)c1cc(sc1NC(=S)N2CCN(CC2)c3ccccc3)c4ccccc4 HTS12831 CN1CCc2c(sc3c2c(nc(n3)SCC(=O)c4ccccc4)SCC(=O)c5ccccc5)C1 HTS12791 Cc1cc(nc2n1nc(c2Cl)c3ccc(cc3)C(C)(C)C)C(F)(F)F KM02453 CC(=O)c1c(c(c(s1)SC)C#N)c2cccs2 KM05441 Cc1cc(nc2c1c3c(s2)c(=O)n(c(n3)C)/N=C/c4ccc5c(c4)OCO5)C HTS13029 C[C@@H](C(=O)NC1CCCCC1)NC(=O)c2ccc(cc2Cl)Cl HTS12323 C[C@@H](C(=O)NCCOC)NC(=O)c1ccc(cc1Cl)Cl HTS12324 Cc1c(sc2c1c(=O)n(c(n2)C)N)C HTS13032 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)F)/C(=O)N2Cc4ccc(cc4)F HTS13073 c1ccc(cc1)C2=N/C(=C\c3ccccc3Cl)/C(=O)N2CC(=O)c4ccccc4 HTS13075 CCOC(=O)CN1C(=N/C(=C/c2ccc(cc2)OC)/C1=O)c3ccccc3 HTS13078 Cc1ccc(cc1)n2c(=O)c3cc(sc3n(c2=O)CC=C)c4ccccc4 HTS13125 c1cc2c(cc1NC(=O)CC3(CCCCC3)CC(=O)O)C(=O)OC2 SCR00360 Cc1nc2c(c(=O)n1NC(=O)CN3CCCC3)ncn2c4ccccc4 HTS13034 Cc1nc2c(c(=O)n1NC(=O)CN3CCCCC3)ncn2c4ccccc4 HTS13035 c1ccc(cc1)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S05072 Cc1ccc(cc1)n2cc([nH]c2=S)c3cccs3 HTS13081 c1ccc2c(c1)-n3c(nn(c3=O)CC(=O)N/N=C/c4ccc(cc4)Cl)CS2 HTS13117 c1ccc(cc1)c2cc3c(=O)n(c(=O)n(c3s2)Cc4ccc(cc4)F)c5ccccc5 HTS13121 c1ccc(cc1)c2cc3c(=O)n(c(=O)n(c3s2)CC(=O)c4ccccc4)c5ccccc5 HTS13123 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)Cc4ccccc4Cl HTS13134 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)Cc4ccc(cc4)F HTS13127 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)CC(=O)c4cccs4 HTS13128 CC(C)(C)NC(=O)Nc1ccc(cc1)Cl S04975 c1ccc(cc1)c2nc(sn2)N3CCCN(CC3)CC(C(F)(F)F)O SCR00707 Cc1ccc(cc1C)NC(=O)c2cnc3ccccc3n2 SCR00737 CC(C)(C)c1ccc(cc1)NC(=O)c2cccs2 S06752 CC(C)(C)c1ccc(cc1)NC(=O)c2c(cccc2Cl)F S06753 COc1ccc2c(c1)sc(n2)/N=C/c3ccccc3O S04983 Cc1ccc(cc1Cl)NC(=S)N/N=C/c2cccnc2 S06893 c1ccc2c(c1)ccc3c2ccc4c3ccc(c4)/N=C/c5cc(ccc5O)Br S05061 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2ccc(cc2)C(F)(F)F S05041 c1cc(ccc1C(F)(F)F)NC(=O)/C=C/C(=O)O S05032 Cc1ccccc1n2cc([nH]c2=S)c3ccc(cc3)Br HTS13085 CCOC(=O)c1cc(sc1NC(=O)CSc2nccn2C)c3ccccc3 HTS13139 Cc1ccn2c(c1)nc(c2c3nnco3)C HTS12817 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)NN)N)c4cccs4 HTS12609 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)CC(=O)c4ccccc4 HTS13129 CC(=O)Cn1cnc2c(c1=O)cc(s2)c3ccccc3 HTS13130 CC(C)(C)c1ccc(cc1)/N=C/c2ccc(cc2)OC S06756 CC(C)c1ccc(cc1)NC(=S)N/N=C/c2cccnc2 S06890 c1cc(c(cc1C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl)Cl S05040 c1ccc(cc1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S05039 c1cc(ccc1C(F)(F)F)N2C(=O)C=CC2=O S05033 Cn1c2c(nc1Oc3ccccc3Br)n(c(=O)n(c2=O)Cc4ccccc4)C HTS12273 CCOC(=O)c1c(nn(c1c2ccccc2)c3ccc(cc3)[N+](=O)[O-])c4cccs4 HTS12209 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)Br MO00859 Cn1c2c(c(=O)n(c1=O)C)[nH]c(n2)NCc3ccccc3 HTS12280 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N3CCOCC3)C/C=C/c4ccccc4 HTS12279 c1ccc(cc1)C\2=NOC(=O)/C2=C/3\N(N=C(S3)C(=O)c4ccccc4)c5ccccc5 HTS12256 c1ccc(cc1)C\2=NOC(=O)/C2=C/3\N(N=C(S3)C(=O)c4ccccc4)c5ccc(cc5)Cl HTS12257 Cc1ccc(cc1)NC(=O)c2ccc3c(c2)scn3 SCR00008 c1ccc2c(c1)ncc(n2)C(=O)NCc3ccc(cc3)c4cccs4 SCR00729 Cc1c(cc(cc1Cl)F)S(=O)(=O)N2CCC(=CC2)c3ccccc3 SCR00413 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)Cl)/C(=O)N2 HTS13053 CCOC(=O)c1cc(sc1NC(=O)c2ccccc2)c3ccccc3 HTS13092 CCOC(=O)c1cc(sc1NC(=O)c2ccco2)c3ccccc3 HTS13093 CC(C)(C)c1ccc(cc1)NC(=O)c2ccc(cc2)Cl S06788 c1ccc(cc1)c2cc3c(ncnc3s2)N4CCc5c4cccc5 HTS13103 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc(cc3)c4cnco4 SCR00074 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc(s3)c4ccccn4 SCR00066 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2cccnc2 S06858 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3ccc4c(c3)OCCO4 SCR00417 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3ccc4c(c3)CCO4 SCR00415 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3cc(cc(c3)Cl)Cl SCR00414 Cc1c(c(no1)c2ccccc2)CNC(=O)C3CCN(CC3)C(=O)C SCR00093 Cc1c(c(no1)c2ccccc2)CNC(=O)CCC(=O)O SCR00056 Cc1c(c(no1)c2ccccc2)CNC(=O)c3ccccc3C(=O)O SCR00055 Cc1c(c(no1)c2ccccc2)CNC(=O)C3CCC3 SCR00043 Cc1c(c(no1)c2ccccc2)CNC(=O)c3cc4ccccc4o3 SCR00034 Cc1c(c(no1)c2ccccc2)CNC(=O)c3c(onc3c4ccccc4)C SCR00027 Cc1cc(nc2c1c(=O)n(s2)C(=O)C)C HTS12962 c1ccc(cc1)/C=N/n2cnc3c(c2=O)cc(s3)c4ccccc4 HTS12965 Cc1ccc(o1)/C=N/n2cnc3c(c2=O)cc(s3)c4ccccc4 HTS12966 CCn1c(nnc1SCC(=O)N2CCCc3c2cccc3)c4cccs4 HTS12699 Cn1c(nnc1Sc2ncc(c(n2)N)C#N)c3ccncc3 HTS12724 Cn1c(nnc1SCC(=O)Nc2c(cnn2c3ccccc3)C#N)c4ccncc4 HTS12754 c1cc(sc1)CNS(=O)(=O)Cc2ccc(cc2)Cl SCR00429 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)/N=C/c4ccc5c(c4)OCO5 HTS13041 c1ccc(cc1)/C=N/NC(=O)/C(=C/c2cccs2)/NC(=O)c3ccccc3 HTS13066 c1c(cc(c2c1COCO2)CNC(=O)CC3(CCCCC3)CC(=O)O)F SCR00315 c1ccc(cc1)c2cc3c(ncnc3s2)N4CCOCC4 HTS13106 CCOC(=O)c1cnn(c1N)c2c3c4c(sc3ncn2)CCCC4 HTS12842 c1ccc2c(c1)n3c(=O)c(=O)n(nc3s2)CN4CCCCC4 HTS12844 c1cc2c3c(c1)c4c(c(cc(=O)o4)OC(=O)c5ccc(cc5)F)c(=O)n3CC2 HTS12696 c1cc2c3c(c1)c4c(c(cc(=O)o4)OC(=O)c5ccc(cc5)Cl)c(=O)n3CC2 HTS12697 Cc1c(sc2c1c(=O)n(c(n2)C)/N=C/c3cccs3)C HTS12970 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)/N=C/c4cccs4 HTS12972 C=CCn1c2ccccc2c3c1nc4nncn4n3 HTS12729 c1ccc2c(c1)c3c(n2Cc4ccc(cc4)F)nc5nncn5n3 HTS12730 CCOC(=O)C1=NN(/C(=C\2/C(=NN(C2=O)c3ccccc3)c4ccccc4)/S1)c5ccccc5 HTS12243 CCOC(=O)C1=NN(/C(=C\2/C(=NN(C2=O)c3ccccc3)c4ccccc4)/S1)c5cccc(c5)Cl HTS12244 c1ccc2c(c1)CCC3=C2N=c4n(c(=O)/c(=C\c5cccnc5)/s4)C3c6ccccc6Cl HTS12675 Cc1ccc(cc1)c2c(nco2)C(=O)N SEW01998 c1ccc2cnc(cc2c1)NC(=O)CC3(CCCCC3)CC(=O)O SCR00350 c1ccc2c(c1)c(cs2)NC(=O)N3CCOCC3 HTS12328 c1ccc(cc1)Cn2c(nnc2SCC(=O)N3CCCc4c3cccc4)c5ccncc5 HTS12701 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)OC(=O)c5ccc(cc5)F HTS12706 CCOC(=O)c1cc(sc1NC(=S)Nc2ccc(cc2OC)OC)c3ccccc3 HTS12980 c1ccc(cc1)c2nnc3n2N=C(CS3)c4ccc(cc4)[N+](=O)[O-] HTS12733 c1ccc(cc1)C2=Nn3c(nnc3SC2)c4ccc(cc4)Cl HTS12735 c1ccc(cc1)C(=O)N/C(=C/c2cccs2)/C(=O)NN HTS13063 Cc1ccc(o1)/C=N/NC(=O)/C(=C/c2ccccc2Cl)/NC(=O)c3ccccc3 HTS13064 Cc1cc(n(n1)c2c3c(ncn2)n(nn3)Cc4ccccc4Cl)C HTS12745 Cn1c2c(nc1Oc3ccc(cc3)Br)n(c(=O)n(c2=O)Cc4ccc(cc4)Br)C HTS12288 Cc1ccc(o1)/C=N/NC(=O)Cn2c(=O)n-3c(n2)CSc4c3cccc4 HTS13115 c1ccc2c(c1)CCN2c3ncc4c(n3)[nH]c(=S)[nH]c4=S HTS12795 CCOC(=O)N1CCc2c(sc3c2c(=S)[nH]c(=S)[nH]3)C1 HTS12804 c1ccc2c(c1)n3c(=O)c(=O)n(nc3s2)Cc4ccc(cc4)F HTS12850 CCOC(=O)c1c(c(sc1NC(=S)N2CCN(CC2)C)C)C HTS12983 CNC(=O)NC(=O)CSc1nnc(o1)c2ccc(cc2)Cl HTS12711 CNC(=O)NC(=O)CSc1nnc(o1)c2ccco2 HTS12712 CNC(=O)NC(=O)CSc1nnc(o1)c2ccccc2 HTS12713 c1ccc(cc1)n2c(c(cn2)C#N)NC(=O)CN3CCCCC3 HTS12756 Cc1c(sc2c1c(=O)n(c(n2)C)/N=C/c3ccc(cc3)Cl)C HTS13043 COc1cccc(c1)/C=N/n2c(=O)c3cc(sc3nn2)c4ccccc4 HTS13044 Cn1c(nnc1Sc2c3c(ncn2)n(c(=S)s3)CC=C)c4ccncc4 HTS12742 COc1ccc(cc1)c2c3c([nH]c(=O)c2C#N)-c4ccccc4CC3 HTS12685 c1ccc2c(c1)c(cs2)NC(=O)Nc3ccc(cc3)OC(F)(F)F HTS12327 CCC(C)NC(=O)CSCCS(=O)(=O)c1ccccc1 KM01730 c1ccc(cc1)NC(=O)NC(=O)CSc2nnc(o2)c3cccs3 HTS12715 c1cnccc1c2nnc(o2)Sc3ncc(c(n3)N)C#N HTS12717 Cc1cc(nc2c1c(=O)n(s2)C(=O)c3cccs3)C HTS13039 c1ccc(cc1)n2c(c(cn2)C#N)NC(=O)CSc3nnc(n3c4ccc(cc4)F)c5ccco5 HTS12751 Cc1cc(nc(c1C#N)SCC(=O)Nc2c(cnn2c3ccccc3)C#N)C HTS12752 C=CCn1c(=O)c(=O)n2c3ccccc3sc2n1 HTS12852 c1ccc2c(c1)n3c(=O)c(=O)n(nc3s2)CC(=O)c4ccc(cc4)Cl HTS12854 c1ccc(c(c1)CSc2nnc3n2c4ccccc4s3)Cl HTS12809 CCOC(=O)CSc1nnc2n1c3ccccc3s2 HTS12810 c1ccc(cc1)c2nnc3n2N=C(CS3)c4ccccc4 HTS12741 COc1cc(c(cn1)C(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F RF04383 CCc1cccc(c1NC(=O)c2cnccc2C(F)(F)F)CC RF04401 c1cc2c(cc1Br)c(c[nH]2)CC(C(=O)O)N AC10751 CCOC(=O)c1c(n[nH]c1N/N=C/c2ccc(c(c2)Cl)Cl)C S06613 CC(C)(C)c1ccc(cc1)/N=C/c2ccccc2O S06737 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)CO MO00853 Cc1cc(nc2c1c(c(s2)C(=O)NN3CC(=O)N(CC3=O)c4cccc(c4)OC)N)C HTS12899 COc1ccc(cc1)C(=O)Nc2ccc(cc2)c3nc4ccccc4s3 SCR00393 c1ccc(cc1)n2c(c(cn2)C#N)NC(=O)CN3CCOCC3 HTS12761 CC(=O)CSc1c2cnc(nc2nc(n1)SCC(=O)C)N3CCCC3 HTS12762 CC(=O)CSc1nnc(o1)c2cnn(c2N)c3ccccc3 HTS12818 CCOC(=O)c1c2c(sc1NC(=O)Nc3cccc(c3)Cl)CN(CC2)C(=O)OCC HTS12859 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)C)CN(CC2)C(=O)OCC HTS12860 Cc1cc(ccc1Br)NC(=S)N/N=C/c2cccnc2 S06889 Cc1cc(nc2c1c3c(s2)C(=O)N(CC(=O)N3)c4cccc(c4)OC)C HTS12901 c1ccc(c(c1)c2nnc3n2-c4ccccc4SC3)Cl HTS12904 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccc(cc2)Cl HTS12908 CCOC(=O)Cc1csc(n1)NC(=O)Nc2ccc(cc2)C HTS12909 CCOC(=O)c1cccc(c1O)O MO00786 c1cc(ccc1c2cc(c(c(=O)[nH]2)C#N)c3ccc(c(c3)Cl)Cl)Cl S06649 c1ccc-2c(c1)CCc3c2[nH]c(=O)c(c3c4ccccc4Cl)C#N HTS12682 c1ccc2c(c1)nc(s2)c3ccc(cc3)NC(=O)c4cccc5c4OCCCO5 SCR00394 CCn1c(n[nH]c1=S)c2cccc(c2)[N+](=O)[O-] HTS12911 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4ccc(cc4)Cl)CS2 HTS12572 c1ccc2c(c1)CCN(C2)S(=O)(=O)Cc3ccc(cc3)Cl SCR00425 COc1cc(cc(c1OC)OC)/C=N/N2CC(=O)N(CC2=O)c3ccc(cc3)Cl HTS12955 COC(=O)c1cc2cc(ccc2s1)Br MO00965 Cc1cc(nc2c1c3c(s2)c(=O)n(c(n3)C)/N=C/c4ccccc4)C HTS13030 CC(=O)c1c(c2c(c3c(nc2o1)-c4ccccc4CC3)c5ccc(cc5)Cl)N HTS12568 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4cccnc4)CS2 HTS12569 c1cc(ccc1n2c(nnn2)c3cnccc3C(F)(F)F)F RF04525 c1ccc2c(c1)n3c(=O)c(=O)n(nc3s2)CC(=O)c4cccs4 HTS12990 CCOC(=O)c1c2c(sc1NC(=S)NCC=C)CN(CC2)C(=O)OCC HTS12994 CCOC(=O)c1c2c(sc1NC(=S)NCc3ccccc3)CN(CC2)C(=O)OCC HTS12995 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3ccc4ccccc4c3 SCR00379 CC1=Nn2c(nnc2SC1)Cn3c4ccccc4nn3 HTS12627 c1ccc(c(c1)NC(=O)c2cnccc2C(F)(F)F)Cl RF04518 CCOC(=O)c1cc(sc1NC(=O)c2cccs2)c3ccccc3 HTS13099 CCOC(=O)Cn1c(=O)c2c(cc(nc2s1)C)C HTS12959 Cc1cc(nc2c1c(=O)n(s2)C(=O)c3ccco3)C HTS12961 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3ccc(cc3)F SCR00381 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3cccc(c3)C(F)(F)F SCR00380 c1cn(cn1)CC\2CCCC/C2=N/O HTS11404 CCOC(=O)c1cn[nH]c1N/C=C(\C#N)/C(=O)OCC HTS12625 CC(C)(C)c1ccc(cc1)C(=O)Nc2ccc(cc2)C(C)(C)C S06739 CC(C)(C)c1ccc(cc1)C(=O)NCc2cccnc2 S06741 CC(C)(C)c1ccc(cc1)NC(=S)NCCO S06744 Cc1nc2c(cnn2c3ccccc3)c(=O)n1/N=C/c4ccc(cc4)Cl HTS12897 c1ccnc(c1)CN(Cc2ccccn2)C(=O)c3cccnc3Oc4ccc(cc4)Cl SCR00624 CN1CCN(CC1)c2ccc(cc2)CNC(=O)c3ccc4c(c3)OCCO4 SCR00791 Cc1c2cc(sc2n(n1)C)C(=O)NCc3ccc(cc3)N4CCN(CC4)C SCR00788 c1ccc(cc1)C2=CCN(CC2)C(=O)c3ccc4c(c3)cco4 SCR00408 CCN(CC)c1c2cc(sc2ncn1)c3ccccc3 HTS13100 c1ccc(cc1)c2nc(cs2)CNC(=O)c3cc(cc4c3OCOC4)F SCR00563 c1cc(sc1)c2nc(cs2)CNC(=O)c3cc(cc4c3OCOC4)F SCR00556 Cc1cc(no1)CNC(=O)c2cc(cc3c2OCOC3)F SCR00555 c1ccnc(c1)CN(Cc2ccccn2)C(=O)c3ccc4c(c3)nsn4 SCR00629 CS(=O)(=O)n1cc(c2c1cccc2)C(=O)C(F)F SCR00508 c1cc(ccc1CN2CCCN(C2c3ccc4c(c3)CCO4)Cc5ccc(cc5)F)F SCR00443 Cc1cc(nn1C)C(=O)NCc2ccc(cc2)N3CCOCC3 SCR00655 CN1CCN(CC1)c2ccc(cc2)CNC(=O)C3=Cc4ccccc4OC3 SCR00780 c1cc(sc1)c2c(c(n(n2)c3ccc(cc3)[N+](=O)[O-])N)C#N HTS12210 CCOC(=O)c1c(nn(c1N)c2ccc(cc2)[N+](=O)[O-])c3cccs3 HTS12211 c1ccc(cc1)C\2=NOC(=O)/C2=C/3\N(N=C(S3)C(=O)c4ccc5ccccc5c4)c6ccccc6 HTS12255 Cc1cc(no1)NS(=O)(=O)c2cccs2 JW00050 Cc1nc2c(c(=O)n1/N=C/c3cc(c(c(c3)OC)OC)OC)ncn2c4ccccc4 HTS13022 c1ccc(c(c1)c2nnc3n2-c4ccccc4SC3)F HTS13024 COc1ccc(cc1)/C=N/c2ccc(cc2)Cl S04897 c1ccc2c(c1)c(cs2)NC(=O)Nc3ccc(c(c3)Cl)F HTS12343 c1c(cnc(c1Cl)N2CCN(CC2)CC(C(F)(F)F)O)C(F)(F)F SCR00805 c1ccc2c(c1)n3c(s2)nnc3SCc4ccc(cc4)F HTS12808 c1ccc(cc1)NC(=O)NC(=O)CSc2nnc3n2c4ccccc4s3 HTS12812 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(cc3)Cl)C SCR00512 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(cc3)C(F)(F)F)C SCR00511 Cc1cc(nc2c1c(=O)[nH]s2)C HTS12963 COc1cccc(c1)/C=N/n2cnc3c(c2=O)cc(s3)c4ccccc4 HTS12964 COc1ccc(cc1)/N=C/c2ccc(c(c2)Cl)Cl S04896 c1ccc2c(c1)c(cs2)NC(=O)Nc3ccc(cc3F)F HTS12330 c1ccc2c(c1)c(cs2)NC(=O)NCC3COc4ccccc4O3 HTS12347 Cc1c(c(no1)c2ccccc2)CNC(=O)Nc3csc4c3cccc4 HTS12341 CC1CCN(CC1)C(=O)Nc2csc3c2cccc3 HTS12337 c1ccc(cc1)S(=O)(=O)N2CCc3c2ccc(c3)[N+](=O)[O-] HTS11325 CCc1ccc(cc1)Oc2nc3c(n2Cc4ccccc4Cl)c(=O)n(c(=O)n3C)C HTS12283 C=CCN1C(=N/C(=C/c2ccccc2Cl)/C1=O)c3ccccc3 HTS13074 c1ccc(cc1)C2=N/C(=C/c3ccco3)/C(=O)N2CC(=O)N HTS13077 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)CC(=O)c4ccccc4)C1 HTS12865 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)Cc4ccc(cc4)Cl)C1 HTS12867 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)Cc4ccc(cc4)F)C1 HTS12868 c1cc(ccc1CSc2nnc(s2)Nc3ccc(cc3)Cl)Cl S06814 Cc1cc(nn1C)C(=O)Nc2nc3ccc(cc3s2)Cl SCR00698 c1cc(ccc1C(=O)C2CCN(CC2)CC(C(F)(F)F)O)F SCR00803 c1ccc2c(c1)c(cs2)NC(=O)NCc3ccccn3 HTS12336 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3ccc(s3)c4ccno4 SCR00846 CCOC(=O)CSc1nnc(o1)c2cnn(c2N)c3ccccc3 HTS12819 CC(C)(C)c1ccc(cc1)c2nnc(s2)SCc3ccc(cc3)Cl S06913 COc1cc(cc(c1)/N=C/c2ccccc2O)C(F)(F)F S04927 CCOC(=O)c1cnn(c1N)c2c3c4c(sc3ncn2)CN(CC4)C(=O)OCC HTS12973 Cc1c(sc2c1c(=O)n3c(n2)SCC(=N3)c4cccs4)C HTS12974 Cc1cc(nn1C)C(=O)Nc2ccc(cc2)N3CCOCC3 SCR00696 COc1cccc(c1)C(=O)CN2C(=N/C(=C\c3ccco3)/C2=O)c4ccccc4 HTS13076 Cc1cc(n(n1)c2c3cc(sc3ncn2)c4ccccc4)C HTS13109 C/C(=N\Nc1nc2c(n1Cc3ccccc3)c(=O)n(c(=O)n2C)C)/c4ccncc4 HTS12293 C/C(=N\Nc1nc2c(n1Cc3ccccc3)c(=O)n(c(=O)n2C)C)/c4ccc(cc4)Cl HTS12294 Cc1ccc(cc1)n2cc([nH]c2=S)c3ccc(cc3)Cl HTS13084 CCOC(=O)c1c2c(sc1NC(=S)N3CCCCC3)CN(CC2)C(=O)OCC HTS12875 CC1=C(C(NC(=S)N1)c2cc(c(c(c2)OC)OC)OC)C(=O)OC HTS12880 c1ccc(cc1)/C=N/NC(=O)c2cc(sc2N)c3ccccc3 HTS12882 CCNC(=S)Nc1c(c(c(s1)C)C)C(=O)OCC HTS12979 Cc1cc(nc2c1c3c(s2)c(=O)oc(n3)C)C HTS12938 CC(=O)NCCc1c[nH]c2c1cc(cc2)O AC22693 Cc1c(sc2c1c(=O)n3c(n2)SCC(=N3)C)C HTS12975 Cc1cc(ccc1n2c(=O)c3ccccc3[nH]c2=S)F S04950 CCOC(=O)c1cc(sc1NC(=S)Nc2ccccc2)c3ccccc3 HTS12981 Cn1c(ccn1)NC(=O)CN(Cc2ccccc2)CC(=O)O SCR00483 CNNC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F S05088 CCOC(=O)c1c2c(sc1NC(=S)NC(=O)OCC)CCCC2 S05191 Cc1cc(nc2c1c(=O)[nH]cn2)C AC27191 Cc1ccccc1NC(=O)/C=C/C(=O)O S05218 CC(=O)c1ccc(c(c1)N2C(=O)C=CC2=O)Cl S05225 c1cc(ccc1c2cn(c(=S)[nH]2)c3ccc(cc3)F)[N+](=O)[O-] HTS13088 c1ccc2c(c1)N=C(CS2)NNC3=Nc4ccccc4SC3 HTS13089 C/C(=N\Nc1nc2c(n1C)c(=O)n(c(=O)n2C)C)/c3cccs3 HTS12298 c1c(c(=O)[nH]c(=O)[nH]1)N2CCOCC2 HTS12300 Cc1ccc(cc1)S(=O)(=O)N2CCCCC2c3cccnc3 HTS12303 Cc1c(n(c(=O)n(c1=O)Cc2ccc(cc2)Br)Cc3ccc(cc3)Br)C HTS12305 C=CCn1c(n[nH]c1=S)c2ccccc2Cl HTS12940 c1ccc(c(c1)c2n[nH]c(=S)n2C3CCCCC3)Cl HTS12941 c1cc(ccc1c2cc(=O)c3ccc(cc3o2)OCC(CS(=O)(=O)c4ccc(cc4)C(F)(F)F)O)Cl SEW02774 c1cc(cnc1)CNS(=O)(=O)Cc2ccc(cc2)Cl SCR00428 Cc1c(c(no1)c2ccccc2)CN3CCS(=O)(=O)CC3 SCR00597 CCN(CC)CC(=O)Nn1c(nc2c(c1=O)ncn2c3ccccc3)C HTS13037 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)/N=C/c4ccccc4Cl HTS13040 Cc1cc(nn1C)C(=O)Nc2ccc(cc2)c3cnco3 SCR00703 Cc1cc(nn1C)C(=O)N2CCN=C(C=C2)C(F)(F)F SCR00690 c1c(c2[nH]c3c(c(=O)n2n1)CCCC3)C#N HTS12586 c1c(c2[nH]c3c(c(=O)n2n1)CCC3)C#N HTS12587 c1ccc(cc1)C(=O)NC(=S)Nc2ccc3c(c2)OCCO3 S05246 c1ccc(cc1)CSc2nnc3n2CCCN3C(=O)c4ccco4 HTS12775 c1ccc(cc1)CSc2nnc3n2CCCN3C(=O)c4cccs4 HTS12776 Cc1c(sc2c1c(=O)n3c(n2)SCC(=N3)c4ccc(cc4)F)C HTS12822 Cc1ccnc(c1)n2c(=O)c3c(c(sc3[nH]c2=S)C)C HTS12825 CCOC(=O)c1c2c(sc1NC(=O)CN3CCOCC3)CN(CC2)C(=O)OCC HTS12780 c1ccc(c(c1)/C=N/N2CC(=O)N(CC2=O)c3ccccc3F)Cl HTS12947 c1ccc(c(c1)N2CC(=O)N(CC2=O)/N=C/c3cccs3)F HTS12948 COc1cccc(c1)N2CC(=O)N(CC2=O)/N=C/c3ccccn3 HTS12949 c1ccc(cc1)C2=N/C(=C/c3cccs3)/C(=O)N2 RG00110 c1ccc2c(c1)nnn2CC(=O)N/N=C/c3cccs3 HTS12623 c1ccc(cc1)c2c(nnc(n2)S)c3ccccc3 HTS12595 c1cc(c2c(c1)OCCCO2)C(=O)NCc3cccnc3 SCR00534 c1cc(cc(c1)N2CC(=O)N(CC2=O)/N=C/c3cccnc3)C(F)(F)F HTS12950 COc1cccc(c1)/C=N/N2CC(=O)N(CC2=O)c3ccccc3F HTS12952 COc1cccc(c1)N2CC(=O)N(CC2=O)/N=C/c3ccc(cc3)Cl HTS12956 Cc1c(c(n(n1)C(=O)c2cccc(c2)Cl)C)Br CD07247 CC(C)c1ccccc1NC(=O)/C=C/C(=O)O S05002 CC(=O)NCCc1c[nH]cn1 AC22864 CCOC(=O)N/N=C(/CN1C(=O)c2ccccc2C1=O)\c3ccc(cc3)C(F)(F)F HTS11882 c1cc(c(c(c1)Cl)Sc2[nH]c(nn2)N)[N+](=O)[O-] HTS11403 CCN(CC)CC(=O)Nc1c(c2c(s1)CN(CC2)C(=O)OCC)C#N HTS12785 CCOC(=O)c1c2c(sc1NC(=O)CSc3nnc(o3)c4ccccc4)CN(CC2)C(=O)OCC HTS12788 c1ccc(cc1)CN2CCc3c(sc4c3c(=S)[nH]c(=S)[nH]4)C2 HTS12793 Cc1c(sc(c1C#N)NC(=O)CN(Cc2ccccc2)Cc3ccccc3)C HTS12832 Cc1ccc(cc1)N2CC(=O)N(CC2=O)/N=C/c3ccc4c(c3)OCO4 HTS12957 Cc1cc(nc2c1c(=O)n(s2)C(=O)c3ccccc3)C HTS12960 Cc1c(sc(n1)C)S(=O)(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00841 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3ccc4c(c3)CCO4 SCR00839 COc1ccc(cc1)CN2CCCN(C2c3cccnc3)Cc4ccc(cc4)OC SCR00751 COc1ccc(cc1)CN2CCCN(C2c3ccsc3)Cc4ccc(cc4)OC SCR00750 COc1ccc(cc1)CN2CCCN(C2c3cccc(c3)Cl)Cc4ccc(cc4)OC SCR00749 COc1ccc(cc1)CN2CCCN(C2c3ccccc3)Cc4ccc(cc4)OC SCR00747 CCCCOc1ccc(cc1)N2C(=O)CSC2=S S04923 Cc1ccc(cc1C)C(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00800 c1ccc2c(c1)c(cs2)NC(=O)Nc3cccc(c3)n4cccc4 HTS12351 C=CCN1C(=N/C(=C/c2ccc(cc2)OCc3ccccc3)/C1=O)c4ccccc4 HTS13070 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)F)/C(=O)N2CC(=O)N HTS13071 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)Cc3cccc(c3)C(F)(F)F SCR00834 Cc1c(sc(c1C#N)NC(=O)CN2CCN(CC2)c3ccccc3)C HTS12834 Cc1c(sc(c1C#N)NC(=O)CN2CCc3c2cccc3)C HTS12835 c1ccc(cc1)c2cc3c(=O)n(c(=O)n(c3s2)CC(=O)c4cccs4)c5ccccc5 HTS13120 CC(=O)Cn1c2c(cc(s2)c3ccccc3)c(=O)n(c1=O)c4ccc(c(c4)Cl)Cl HTS13122 COc1cccc(c1O)/C=N/c2ccc(cc2)S(=O)(=O)NC(=N)/N=C/c3cccc(c3O)OC S04866 Cc1ccc(cc1F)S(=O)(=O)N2CCC(=CC2)c3ccccc3 SCR00382 Cc1cc(nn1C)C(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00657 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(C(F)(F)F)O SCR00712 COc1ccc(c(c1)C(=O)NCCc2ccc(c(c2)OC)OC)Br S07385 CCOC(=O)N1CCc2c(sc(c2C#N)NC(=O)CN3CCN(CC3)c4ccccc4)C1 HTS12781 CN1CCN(CC1)CC(=O)N2C(C3CCc4ccccc4C3=N2)c5ccc(cc5)OC HTS12617 c1ccc2c(c1)CCC3=C2N=c4n(c(=O)/c(=C\c5ccc(cc5)F)/s4)C3c6cccs6 HTS12619 CCOC(=O)N1CCc2c(sc(c2C#N)NC(=O)CN3CCc4c3cccc4)C1 HTS12782 CCOC(=O)Cn1cnc2c(c1=O)cc(s2)c3ccccc3 HTS13135 CCOC(=O)c1cc(sc1NC(=O)CSc2nc3ccccc3s2)c4ccccc4 HTS13136 CCOC(=O)c1cc(sc1NC(=O)CSc2nnc(o2)c3ccco3)c4ccccc4 HTS13137 COc1cccc2c1oc(c2)C(=O)O AC35494 Cc1cc2ccccc2c(c1C#N)/N=C/c3cc(cc(c3O)Cl)Cl S05157 Cc1c(c(no1)c2ccccc2)NC(=O)OCC#C S07272 c1ccc2c(c1)nc(s2)c3ccc(cc3)NC(=O)CSCC(=O)O SCR00400 c1cc(c2c(c1)OCCO2)C(=O)N MO00789 Cc1cc(nc2c1c3c(s2)c(=O)n(nn3)/N=C/c4ccc(cc4)OC)C HTS12565 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)Cc3ccc(cc3)Cl SCR00833 Cc1ccc(cc1S(=O)(=O)NCc2ccc(cc2)N3CCN(CC3)C)F SCR00829 c1ccc(c(c1)CSc2nc3c(c4ccccc4[nH]3)nn2)Cl HTS12596 c1ccc(cc1)n2cc([nH]c2=S)c3ccc(cc3)Cl HTS13086 c1ccc(cc1)c2cn(c(=S)[nH]2)c3ccccc3 HTS13087 c1ccc(cc1)Cn2c3c(cc(s3)c4ccccc4)c(=O)n(c2=O)c5ccccc5 HTS13124 CNC(=O)NC(=O)Cn1cnc2c(c1=O)cc(s2)c3ccccc3 HTS13131 c1cc2c(cc1CN3CCN(CC3)CC(C(F)(F)F)O)OCO2 SCR00821 c1cc(sc1)c2nc(cs2)CNCC(C(F)(F)F)O SCR00913 CCOC(=O)c1c2c(sc1NC(=O)CSc3nccn3C)CN(CC2)C(=O)OCC HTS12786 CCOC(=O)c1c2c(sc1NC(=O)CSc3nc4ccccc4o3)CN(CC2)C(=O)OCC HTS12787 c1ccc2c(c1)nnn2Cc3nnc4n3N=C(CS4)c5ccc(cc5)Br HTS12630 c1ccc2c(c1)C3(C(=O)N2)N(C(=O)CS3)c4cccc(c4)C(F)(F)F HTS12607 Cc1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)NN)N)c4ccco4 HTS12608 c1ccc(c(c1)Cn2c3c(c(ncn3)N/N=C/c4cccnc4)nn2)Cl HTS12610 Cc1ccc(cc1)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)S(=O)(=O)Nc4nccs4 S04815 Cc1nnc2n1c3ccccc3s2 HTS12987 CC1=NN(C(=O)C1)c2c3c4c(sc3ncn2)CCCC4 HTS12988 Cc1cc(nn1C)C(=O)NCC2COc3ccccc3O2 SCR00647 CCOC(=O)c1c(nc(s1)Nc2ccc(cc2)Cl)C S05023 c1cc(ccc1CS(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)Cl SCR00426 c1cc(ccc1c2n[nH]c(=S)o2)[N+](=O)[O-] HTS13090 C1CCc2c(c3c(nc(nc3s2)S)S)C1 HTS12777 c1ccc(cc1)/C=C\2/C(=O)N(C(=N2)c3ccccc3)/N=C/c4ccccc4 HTS13046 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)CC(=O)NC(=O)Nc4ccccc4 HTS13132 c1ccc(cc1)c2cc3c(=O)[nH]cnc3s2 HTS13133 c1cc2ccc(nc2c(c1)O)C(=O)O AC34762 CCOC(=O)c1cc(sc1NC(=O)c2ccc(cc2)Cl)c3ccccc3 HTS13094 c1ccc(c(c1)/C=N/c2c(c3c(s2)CCC3)C#N)O S05141 Cc1c(c(sc1c2ccccc2)/N=C/c3cc(cc(c3O)Cl)Cl)C#N S05137 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4ccc(cc4)F)CS2 HTS12570 C/C(=N\Cc1ccccc1)/c2ccc(cc2O)Cl S05015 Cc1nc(c(o1)C(F)(F)F)C(=O)NNc2ccc(cc2)F RF04648 c1ccnc(c1)CN(Cc2ccccn2)C(=O)c3cccc4c3OCCCO4 SCR00586 c1ccc2c(c1)CCC3=C2N=C4N(C3c5ccc(cc5)F)C(=O)CS4 HTS12618 CCOc1c(c(c2c(n1)-c3ccccc3C2)c4ccco4)C#N HTS12622 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)Cc4ccccc4)C1 HTS13000 c1ccc2c(c1)n3c(=O)c(nnc3s2)N4CCOCC4 HTS13004 CC(C)c1ccccc1NC(=S)NCCCN2CCOCC2 S05019 CCc1ccc(cc1)NC(=S)Nc2ccccc2C(C)C S05009 Cc1ccc(o1)/C=N/N2C(=N/C(=C\c3ccccc3Cl)/C2=O)c4ccccc4 HTS13047 c1ccc(cc1)COc2ccc(cc2)/C=C/3\C(=O)NC(=N3)c4ccccc4 HTS13049 Cc1ccc(cc1)/C=C/2\C(=O)NC(=N2)c3ccccc3 HTS13057 CCOC(=O)c1cc(sc1NC(=O)c2cccc(c2)[N+](=O)[O-])c3ccccc3 HTS13095 CCOC(=O)c1cc(sc1NC(=O)c2ccccc2Cl)c3ccccc3 HTS13096 CCOC(=O)c1c2c(sc1NC(=S)N3CCOCC3)CCCC2 HTS12837 c1ccc(cc1)n2c(ccn2)/N=C/c3cc(ccc3O)Br S04802 CC(C)c1ccccc1NC2=NCCS2 S05014 CC(C)c1ccccc1NC(=S)NCCO S05012 c1ccc2c(c1)c3ccncc3[nH]2 AC12926 c1ccc2c(c1)c(cs2)NC(=O)NC3CC3 HTS12344 CC1=C(C(N2C(=C(SC2=N1)C#N)N)c3cccs3)C(=O)OC HTS13005 c1ccc(cc1)c2cc(c(s2)N)C(=O)N/N=C/c3cccs3 HTS13006 COc1cccc(c1)/C=N/NC(=O)c2cc(sc2N)c3ccccc3 HTS13009 c1ccnc(c1)CN(Cc2ccccn2)S(=O)(=O)c3ccc(cc3)n4cccn4 SCR00617 c1ccc2c(c1)c(c3c(n2)CCCC3)N AC13350 c1ccc(cc1)C(=O)N/C(=C/c2ccco2)/C(=O)NN HTS13062 Cn1c(ccn1)NC(=O)CC2(CCCCC2)CC(=O)O SCR00356 c1cc(c(cc1NC(=O)CC2(CCCCC2)CC(=O)O)Cl)F SCR00331 c1cc(ccc1NC(=O)OC2CN3CCC2CC3)F SCR00294 c1cc2c(c(c1)NC(=O)CC3(CCCCC3)CC(=O)O)nsn2 SCR00361 CC1=Nn2c(=O)c3cc(sc3nc2SC1)c4ccccc4 HTS12838 c1ccc(cc1)c2cc3c(s2)nc4n(c3=O)N=C(CS4)c5ccccc5 HTS12840 c1ccc(cc1)c2cc3c(ncnc3s2)N/N=C/c4cccs4 HTS13110 c1ccc(cc1)n2c3c(cn2)c(=S)[nH]c(=S)[nH]3 HTS12800 c1ccc2c(c1)n3c(=O)c(=O)n(nc3s2)CN4CCOCC4 HTS12845 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccccc3)CN(CC2)C(=O)OCC HTS12992 c1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)SCCC#N S04838 Cc1c(cnn1c2ccccc2)S(=O)(=O)N(Cc3ccccn3)Cc4ccccn4 SCR00609 c1ccc2c(c1)c(cc(n2)O)O AC13220 Cc1cc(nn1C)C(=O)NCc2csc(n2)c3cccs3 SCR00651 Cn1c(cc(n1)C(F)(F)F)O AC29083 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4ccc(cc4)Cl)CO2 HTS12573 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=C(C#N)C#N)OC S04945 c1cc2c(cc1CN3CCS(=O)(=O)CC3)OCCCO2 SCR00606 CCOC(=O)c1c2c(sc1NC(=S)NC(=O)/C=C/c3ccccc3)CCCC2 S05189 CSc1c(c(nn1C(=O)c2cccs2)N)c3ccccn3 SCR00490 CCn1c(nnc1SCC(=O)Nc2c(cnn2c3ccccc3)C#N)c4cccs4 HTS12748 C=CCn1c(nnc1SCC(=O)Nc2c(cnn2c3ccccc3)C#N)c4ccco4 HTS12750 CCn1c(c(c(n1)C)[N+](=O)[O-])c2nnnn2c3ccc(cc3)Cl SPB02918 c1ccc2c(c1)n3c(=O)c(=O)n(nc3s2)CC(=O)N HTS12847 c1ccc(c(c1)Cn2c(=O)c(=O)n3c4ccccc4sc3n2)Cl HTS12848 Cn1c(=O)c(=O)n2c3ccccc3sc2n1 HTS12849 c1ccc2c(c1)n3c(s2)nnc3SCC(=O)c4ccc(cc4)Cl HTS12811 c1ccc2c(c1)nc(s2)N/N=C/c3cccnc3 HTS12815 c1ccnc(c1)CN(Cc2ccccn2)S(=O)(=O)c3ccc(cc3)c4cnco4 SCR00611 c1ccnc(c1)CN(Cc2ccccn2)S(=O)(=O)c3ccc(cc3)Cl SCR00613 c1ccnc(c1)CN(Cc2ccccn2)S(=O)(=O)c3ccc(s3)c4ccno4 SCR00616 c1ccc(c(c1)C(=O)NNC2=Nc3ccccc3SC2)F HTS13011 CN(C)c1c2c([nH]cn2)ncn1 AC22646 c1c(c(n2c(n1)c(cn2)C#N)N)C#N HTS12582 CCOC(=O)c1cnn2c1ncc(c2N)C#N HTS12583 CCOC(=O)c1cnn2c1[nH]c3c(c2=O)CCC3 HTS12585 CC(C)(C)C(=O)Nc1ccncc1 MO00094 c1ccc(cc1)/C=N\c2cccc3c2cccc3 AC33318 c1cc(ccc1CSc2nnc(s2)NC(=O)c3ccc(cc3)Cl)Cl S06825 CCN(CCC#N)C(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F JP00908 CCOc1ccc(cc1)NC(=O)c2cc(n(n2)C)C SCR00704 COC(=O)c1cc(ccc1N2CCOCC2)/N=C/c3ccccc3O S05214 C/C(=N\N=C(\c1c(cccc1)O)/C)/c2c(cccc2)O S05156 c1cc(sc1)C2N(CCCN2Cc3ccc(cc3)F)Cc4ccc(cc4)F SCR00446 c1ccc(cc1)CN(Cc2ccccc2)CC(=O)Nc3c(cnn3c4ccccc4)C#N HTS12757 c1ccc(cc1)n2c(c(cn2)C#N)NC(=O)CN3CCN(CC3)c4ccccc4 HTS12758 CCN(CC)c1ncc2c(n1)nc(nc2SCC(=O)N)SCC(=O)N HTS12763 CCOC(=O)c1cnn(c1N)c2c3cnn(c3ncn2)c4ccccc4 HTS12855 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)Cl)CN(CC2)C(=O)OCC HTS12857 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(c(c3)Cl)Cl)CN(CC2)C(=O)OCC HTS12858 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4cccc(c4)Cl)C1 HTS12861 c1ccc(cc1)C2=CCN(CC2)S(=O)(=O)c3ccc4c(c3)OCCCO4 SCR00420 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4ccncc4)CO2 HTS12574 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CC4)OC(=O)c5ccc(cc5)F HTS12590 CC(=O)Oc1c2cccc3c2n(c(=O)c1c4ccccc4)CC3 HTS12593 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3ccccc3 SCR00824 c1ccc2c(c1)-n3c(nn(c3=O)CC(=O)N/N=C/c4ccc5c(c4)OCO5)CS2 HTS13118 c1ccc2c(c1)-n3c(nn(c3=O)CC(=O)N/N=C/c4cccs4)CS2 HTS13119 Cc1ccc(cc1)N2CC(=O)N(CC2=O)/N=C/c3cn(nc3c4ccc(cc4)Cl)c5ccccc5 HTS12945 c1cnc(nc1)N2CCN(CC2)S(=O)(=O)Cc3ccc(cc3)Cl SCR00427 c1ccc(cc1)c2c(c[nH]n2)CN3CCC(CC3)C(=O)c4ccc(cc4)F HTS05682 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4ccccc4Cl)CO2 HTS12580 c1ccc2c(c1)cccc2Cc3nnc(n3c4ccc(cc4)Cl)S S07434 COc1ccc(cc1)C(=O)CSc2nnc3n2CCCN3C(=O)Nc4ccccc4 HTS12765 c1cc(ccc1S(=O)(=O)/C(=N/OS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N)Cl KM01356 Cc1ccc(n1CCN2CCN(CC2)S(=O)(=O)Cc3ccc(cc3)Cl)C SCR00431 c1cc(ccc1C2(CCN(CC2)CC(C(F)(F)F)O)O)Cl SCR00708 Cc1c(sc2c1c(=O)n(c(n2)C)/N=C/c3cccnc3)C HTS13042 CC(C)c1ccc(cc1)N2C(=O)/C(=C\c3ccc(o3)c4ccc(cc4)[N+](=O)[O-])/SC2=S S05381 c1ccc2c(c1)ncc(n2)C(=O)Nc3ccc(cc3Cl)F SCR00621 Cc1cc(nn1C)C(=O)NCc2cccn2C SCR00658 Cc1cc(nn1C)C(=O)NCc2ccc3c(c2)OCCCO3 SCR00654 Cc1cc(nn1C)C(=O)NCc2cc3ccccc3s2 SCR00652 CSc1nc2ccccc2c(=O)n1c3ccc4c(c3)OCCO4 S05361 c1cc(ccc1c2ccc(o2)/C=C(\C#N)/C(=O)N)[N+](=O)[O-] S05378 CCNC(=O)/C(=C/c1ccc(c(c1)Cl)Cl)/C#N S05387 c1ccc2c(c1)cccc2Cc3nnc(n3c4cc(cc(c4)C(F)(F)F)C(F)(F)F)S S07435 CCOC(=O)c1cc(sc1NC(=O)c2ccccc2F)c3ccccc3 HTS13091 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(c(c3)Cl)Cl)C SCR00507 c1ccc(cc1)C(=O)NC(=C(C#N)C#N)Nc2cccc(c2)Cl TL00105 CSc1c2c(nc[nH]2)nc(n1)N AC10402 c1c(cc(c(c1/C=N/c2c(c3c(s2)CCC3)C#N)O)Cl)Cl S05136 CCOc1ccc(cc1)NC(=S)NC(=O)COc2cc(c(cc2Cl)Cl)Cl S05322 CC(C)(C(=O)NC1CCCCNC1=O)Oc2ccc(cc2)Cl SCR00987 CCOC(=O)c1cnn(c1N)c2c3cc(sc3ncn2)c4ccccc4 HTS13107 c1ccc(cc1)c2cc3c(ncnc3s2)n4c(c(cn4)C#N)N HTS13108 Cc1ccc(o1)/C=N/Nc2c3cc(sc3ncn2)c4ccccc4 HTS13111 CCOC(=O)c1c2c(sc1N)CCCCC2 AC29286 Cc1[nH]c2ccc(cc2n1)C(=O)O AC29314 Cc1cccc(c1)C(=O)Nc2nnc(s2)SC S06829 c1cc(ccc1CSc2nnc(s2)c3ccncc3)Cl S07107 Cc1c2cc(sc2n(n1)C)C(=O)N(Cc3ccccn3)Cc4ccccn4 SCR00632 c1cc(c(cc1N2Cc3cc(c(cc3N=C2)Cl)Cl)Cl)Cl S04869 c1ccc2c(c1)N=C(CS2)NNC(=O)c3cccc(c3)[N+](=O)[O-] HTS13012 c1cc2c(cc1c3ccnc(n3)SCC(C(F)(F)F)O)OCCO2 SCR00931 c1ccc(cc1)n2cnnc2SCC(C(F)(F)F)O SCR00934 Cc1ccc(cc1)C(C[N+](=O)[O-])Sc2ccccc2N S05113 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(cc3F)F)C SCR00505 CCOC(=O)c1cc(sc1NC(=O)c2ccc(cc2)F)c3ccccc3 HTS13097 COc1ccc(c(c1)OC)Nc2c3cc(sc3ncn2)c4ccccc4 HTS13101 c1ccc(cc1)c2cc3c(ncnc3s2)N4CCN(CC4)c5ccccc5 HTS13104 c1ccc(cc1)c2cc3c(ncnc3s2)N4CCCC4 HTS13105 c1cc(cc(c1)Cl)NC(=O)c2cc(cc3c2OCOC3)F SCR00567 CCc1ccc(cc1)NC(=O)NC(C)(C)C S04977 c1ccc2c(c1)cccc2CC(=O)NC3CCCCNC3=O SCR00988 CC(C)(C)c1cc(n(n1)C)C(=O)NC2CCCCNC2=O SCR00990 c1ccc(cc1)N2CCN(CC2)c3ncc4c(n3)[nH]c(=S)[nH]c4=S HTS12798 CN1CCN(CC1)c2ncc3c(n2)[nH]c(=S)[nH]c3=S HTS12799 CCOC(=O)N1CCc2c(sc(c2C#N)N)C1 HTS12802 c1cc2c(cc1O)CC(NC2)C(=O)O AC30194 c1ccc2c(c1)c(c3ccccc3n2)C(=O)O AC40022 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2ccc3c(c2)OCO3 S06854 c1ccc(cc1)c2cc(c(s2)N)c3n[nH]c(=S)n3c4ccccc4 HTS13017 Cc1nc2c(c(=O)n1NC(=O)CN3CCOCC3)ncn2c4ccccc4 HTS13036 c1ccc2c(c1)cccc2C3CC(=Nc4ccccc4S3)c5ccc(cc5)F S05106 c1ccc2c(c1)cccc2C(CC(=O)c3ccc(cc3)F)Sc4ccccc4N S05104 c1ccc2c(c1)nc(s2)CNC(=O)c3cc(cc4c3OCOC4)F SCR00554 CCOC(=O)c1ccc(c(c1)NC(=S)N(C)C)Cl S05422 CCOC(=O)Cc1csc(n1)NC(=O)c2ccc(cc2)F HTS13541 c1ccc(cc1)S(=O)(=O)n2c3ccccc3cc2/C=C\4/c5ccccc5NC4=O SCR01013 c1ccc2c(c1)c(ccn2)/C=C\3/c4ccccc4NC3=O SCR01014 c1ccc2c(c1)c(cs2)/C=C\3/c4ccccc4NC3=O SCR01016 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)CCCN3CCOCC3 S07012 c1ccc(cc1)COC(=O)/C(=C/c2ccc(c(c2)Cl)Cl)/C#N S05454 Cc1ccc2cc(ccc2n1)NC(=O)c3cc(n(n3)C)C SCR00699 Cc1c(cc(o1)S(=O)(=O)NC2CCCCNC2=O)C(=O)OC SCR00888 Cc1c(cc(o1)S(=O)(=O)NCc2csc(n2)c3cccs3)C(=O)OC SCR00883 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)N3CCCCCC3 SCR00938 c1ccc2c(c1)cccc2S(=O)(=O)NC3CCCCNC3=O SCR00976 Cc1c2cc(sc2n(n1)C)C(=O)NC3CCCCNC3=O SCR00994 c1ccc2c(c1)nc(s2)N/N=C/c3ccco3 HTS12813 COc1cc(cc(c1OC)OC)/C=N/Nc2nc3ccccc3s2 HTS12814 Cc1c(cn(n1)c2ccccc2)/C=N/Nc3nc4ccccc4s3 HTS12816 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(cc3)S(=O)(=O)N)C SCR00510 c1ccc(cc1)SC(C(=O)c2cnc3n2cccc3)(F)F SCR00589 c1ccc(cc1)/C(=N\N=C\c2ccccn2)/C(=O)c3ccccc3 S04906 COc1cc(cc(c1)N2C(=O)CSC2=S)C(F)(F)F S04921 Cc1c(sc2c1c(=O)n(c(n2)C)/N=C/c3ccc4c(c3)OCO4)C HTS12969 c1ccc(cc1)c2cc3c(s2)ncn(c3=O)/N=C/c4ccco4 HTS12971 c1ccc(cc1)c2c(nco2)C(=O)N(Cc3ccccn3)Cc4ccccn4 SCR00630 Cc1c(cc(o1)S(=O)(=O)NCc2ccc(cc2)S(=O)(=O)N)C(=O)OC SCR00898 Cc1c(cc(o1)S(=O)(=O)N2CCSC2)C(=O)OC SCR00897 Cc1c(cc(o1)S(=O)(=O)N2CCC(CC2)C(=O)N)C(=O)OC SCR00894 Cc1c(cc(o1)S(=O)(=O)N2CCC(CC2)Cc3ccccc3)C(=O)OC SCR00891 c1cc(ccc1N2CCN(CC2)CC(C(F)(F)F)O)F SCR00918 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)Nc3cccc(c3)C(=O)O SCR00960 COc1cccc(c1)C(c2c([nH]c(=S)[nH]c2=O)N)c3c([nH]c(=S)[nH]c3=O)N HTS13261 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)c4ccc(cc4)Cl HTS13259 Cc1[nH]c(=O)c2c(n1)Oc3c4ccccc4oc(=O)c3C2c5cccs5 HTS13258 c1ccc(cc1)c2cc(=O)n3c(n2CC(=O)NN)ncn3 HTS13255 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccc(cc3)Cl)c4ccccc4)NC(=O)Nc5ccccc5 HTS13256 Cc1cc(nn1C)C(=O)NCc2c(onc2c3ccccc3)C SCR00645 c1ccnc(c1)CN(Cc2ccccn2)S(=O)(=O)c3ccc(s3)c4cc(on4)C(F)(F)F SCR00612 Cc1c(c(no1)c2ccccc2Cl)C(=C(C#N)C#N)OC S04940 Cc1cc(n(n1)c2ccccc2)n3c(=O)c4c(c(sc4[nH]c3=S)C)C HTS12976 CCOC(=O)c1c(c(sc1NC(=S)Nc2cc(nn2c3ccccc3)C)C)C HTS12978 Cc1c(cc(o1)S(=O)(=O)N2CCN(CC2)c3c(cncc3Cl)Cl)C(=O)OC SCR00890 Cc1c(cc(o1)S(=O)(=O)NCCc2c[nH]c3c2cccc3)C(=O)OC SCR00880 COc1ccc(cc1)C(c2c([nH]c(=S)[nH]c2=O)N)c3c([nH]c(=S)[nH]c3=O)N HTS13262 Cc1c(c(no1)c2ccccc2)/C=C\3/c4ccccc4NC3=O SCR01010 COc1ccc(cc1OC)CC(=O)NC2CC2 SCR00761 c1cc(sc1)CNC(=O)c2cc(cc3c2OCOC3)F SCR00559 CCN(CC)c1ccc(c(c1)C)NC(=S)NCCO S05035 c1ccc2c(c1)ncc(n2)C(=O)Nc3ccc(cc3)N4CCOCC4 SCR00735 CCOc1ccc(cc1)NC(=O)c2cnc3ccccc3n2 SCR00734 c1ccc(cc1)/C=C/2\C(=O)N(C3(S2)N(N=C(S3)C(=O)c4cccs4)c5ccc(cc5)Cl)c6ccccc6 HTS13243 CCc1ccccc1n2c(=O)c3ccccc3nc2SCC(C(F)(F)F)O SCR00923 Cc1c(cc(o1)S(=O)(=O)NCc2ccc(cc2Cl)Cl)C(=O)OC SCR00878 COc1ccc(c(c1)S(=O)(=O)NC2CCCCNC2=O)OC SCR00973 Cc1cc(c(o1)C(F)(F)F)S(=O)(=O)NC2CCCCNC2=O SCR01000 c1cc(ccc1S(=O)(=O)NC2CCCCNC2=O)Cl SCR00997 CC(C)(CO)NC(=O)c1c(cccc1Cl)F S07029 c1cc(c2c(c1)OCCCO2)C(=O)NCc3ccc4c(c3)OCO4 SCR00579 c1cc(cc(c1)S(=O)(=O)N)NC(=O)c2cccc3c2OCCCO3 SCR00584 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)N3CCOCC3 SCR00946 CC1CCc2c(sc(c2C#N)NC(=O)CN(Cc3ccccc3)Cc4ccccc4)C1 HTS13252 c1ccc2c(c1)CCC(=C2)N3CCN(CC3)c4ccc(cc4)F HTS13250 c1ccc(cc1)c2ccc-3c4ccccc4c(c3o2)C(=O)C(F)(F)F HTS13249 c1cc(c(c(c1)Cl)CN2CCN(CC2)CC(C(F)(F)F)O)F SCR00916 c1ccc(cc1)C2=CCN(CC2)C(=O)CN3C(=O)c4ccccc4C3=O SCR00940 Cc1c(c(on1)c2ccccc2)CNc3c4ccccc4nc(n3)c5ccccc5 SCR01033 Cc1cc(nn1C)C(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4 SCR00687 c1ccc(cc1)c2c(n[nH]c(=O)n2)c3ccccc3 HTS13520 COc1ccc(c(c1)C(=O)Nc2ncccn2)Br S07528 Cc1c(c(n(n1)C)C)CNC(=O)Nc2csc3c2cccc3 HTS12349 CN1CCC(CC1)CNC(=O)Nc2csc3c2cccc3 HTS12339 c1ccc2c(c1)-n3c(nn(c3=O)CC(=O)N/N=C/c4cccnc4)CS2 HTS13116 Cc1cc(nc2c1c3c(s2)c(=O)n(c(n3)C)N)C HTS12939 c1ccc(cc1)c2ccccc2NC(=S)NCCO S04956 c1ccc(cc1)/C(=C/C(=C(/C#N)\c2ccc(cc2)[N+](=O)[O-])/c3ccccc3)/CC(=O)c4ccccc4 HTS13248 c1ccc(cc1)C(=O)C/C(=C\C(=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])\c3ccccc3)/c4ccc(cc4)Cl HTS13246 CN1CCN(CC1)c2ccc(cc2)CNC(=O)c3ccc4c(c3)nsn4 SCR00785 c1cnc(nc1C(F)(F)F)N2CCCN(CC2)CC(C(F)(F)F)O SCR00818 Cc1cc(no1)CNC(=O)CN2C(=O)c3ccccc3C2=O SCR00954 COc1ccc(c(c1)C(=O)Nc2cc(cc(c2)Cl)Cl)Br S07536 c1cc2c(c(c1)N)C(=O)NC2=O AC40100 CCOC(=O)CN(c1ccc(cc1)F)C(=O)COc2c(c(cc(n2)C)C)C#N HTS13315 CCOC(=O)CN(c1ccccc1)C(=O)COc2c(c(cc(n2)C)C)C#N HTS13316 CCOC(=O)CN(c1ccc(cc1)Cl)C(=O)COc2c(c(cc(n2)C)C)C#N HTS13317 COc1cccc(c1)c2csc(n2)NNC(=O)c3ccncc3 HTS13318 CC(=O)CSc1c2c3c(sc2nc(n1)SCC(=O)C)CCC3 HTS13331 CCOC(=O)Cn1c(=O)nc(c(n1)c2ccccc2)c3ccccc3 HTS13521 CCNc1c2c3c(sc2nc(n1)SCC(=O)NC(=O)NC)CN(CC3)C HTS13524 CCNc1c2c3c(sc2nc(n1)SCC(=O)NC(=O)Nc4ccccc4)CN(CC3)C HTS13526 COc1cccc(c1)c2csc(n2)NNC(=O)c3ccc(cc3)Cl HTS13466 c1ccc(cc1)n\2c(cs/c2=N\Cc3cccnc3)c4ccc(cc4)[N+](=O)[O-] HTS13533 COc1ccc(cc1)CN2CCCN(C2c3ccc(cc3)F)Cc4ccc(cc4)OC SCR00745 CCOC(=O)c1c(nc(s1)Nc2cccc(c2)Cl)C S05021 C/C(=N\Cc1ccccc1Cl)/c2ccc(cc2O)Cl S05016 CC(C)c1ccccc1/N=C/c2cc(ccc2O)Br S05011 c1ccc2c(c1)cccc2CC(=O)Nc3cc(cc(c3)Cl)Cl S07542 C/C(=C\c1ccc(o1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/[N+](=O)[O-] S05358 CCOC(=O)CN(c1cccc(c1)C(F)(F)F)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13390 c1ccc2c(c1)CCCN2CC(=O)Nc3ccc(cc3)S(=O)(=O)N HTS13332 CN1CCN(CC1)CC(=O)Nc2ccc(cc2)S(=O)(=O)N HTS13333 c1ccc2c(c1)CCN2CC(=O)Nc3ccc(cc3)S(=O)(=O)N HTS13334 Cc1ccc(o1)/C=c\2/c(=O)n3c(s2)nc(=O)c(n3)C HTS13405 Cc1cccc(n1)/N=c\2/n(c(cs2)c3cccs3)Cc4ccccc4 HTS13537 CCn\1c(cs/c1=N\c2cc(ccn2)C)c3ccc(cc3)[N+](=O)[O-] HTS13538 CCOC(=O)Cc1csc(n1)NC(=O)c2cccc(c2)[N+](=O)[O-] HTS13540 Cc1c(c2ccccc2o1)CC(=O)NCC=C S07740 c1ccc(cc1)CN(CC(=O)Nc2ccc3c(c2)OCCCO3)CC(=O)O SCR00479 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(c(c3)Cl)F)C SCR00506 c1ccc(c(c1)/C=N/c2ccccc2C(F)(F)F)O S04930 CC(c1ccccc1)/N=C/c2ccccc2O S04931 Cc1c(c(no1)c2ccccc2)C(=C(C#N)C#N)OC S04934 Cc1cc(ccc1NC2=NCCS2)F S04936 Cc1cc(ccc1Nc2n[nH]c(=S)s2)F S04939 CCN(CC)CC(=O)Nc1c2c(cs1)c3ccccc3oc2=O HTS13324 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)c4cccc(c4)[N+](=O)[O-] HTS13326 COc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3cccs3 HTS13327 c1cc(sc1)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)F HTS13328 COc1cc(cc(c1OC)OC)c2nnc(n2CC=C)SCC(=O)NC(=O)Nc3ccccc3 HTS13397 CCNc1c2c3c(sc2nc(n1)SCC(=O)NC(=O)NCc4ccccc4)CN(CC3)C HTS13528 CCNc1c2c3c(sc2nc(n1)SCc4ccc(cc4)Cl)CN(CC3)C HTS13529 CN1C(=O)C(=Cc2cn(nc2c3ccc(cc3)OC)c4ccccc4)C(=O)N(C1=O)C HTS13530 CCNc1c2c3c(sc2nc(n1)SCc4ccc(cc4)F)CN(CC3)C HTS13523 c1ccc(c(c1)CNC(=O)C(C(C(=O)O)(F)F)(F)F)Cl SCR00278 CC1(Cc2cccc(c2O1)C(=O)Nc3ccncc3)C SCR00501 Cc1cc(c(s1)C)S(=O)(=O)Nc2ccc3c(c2)OCC4N3CCC4 SCR01120 c1ccn(c1)c2cccc(c2)NC(=O)c3cccc4c3OCCCO4 SCR00582 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3ccc(cc3Cl)Cl)/s2 HTS13406 CCOC(=O)c1c2c(sc1/N=C/c3cc(cc(c3O)Cl)Cl)CCC2 S05134 Cc1c(snn1)C(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00794 c1ccc(cc1)CN2CCC(CC2)NCC(C(F)(F)F)O SCR00907 CN1C(=O)C(=Cc2cn(nc2c3cccs3)c4ccccc4)C(=O)N(C1=O)C HTS13253 CCOC(=O)N1CCc2c(sc(c2C#N)NC(=O)CN(Cc3ccccc3)Cc4ccccc4)C1 HTS12783 COc1cccc(c1)c2c3c(nc(c2C#N)OC)-c4ccccc4C3 HTS12621 c1cc(cc(c1)n2c(=O)c3cn[nH]c3[nH]c2=S)C(F)(F)F HTS12626 CCOC(=O)c1cc(sc1NC(=O)CN2CCc3c2cccc3)c4ccccc4 HTS13138 CCOC(=O)c1cc(sc1NC(=O)CN2CCN(CC2)c3ccccc3)c4ccccc4 HTS13140 c1ccc(cc1)n2c(c(cn2)C(=O)N/N=C/c3cccnc3)N HTS12606 CCOc1nc(nc(n1)NC)N AC35726 COc1ccc(cc1)c2cc(c3c(ncnc3n2)N)c4ccccc4 HTS13340 Cn1c(nnc1SCC(=O)NN2CC(=O)N(CC2=O)c3cccc(c3)Cl)c4ccncc4 HTS13268 CCOC(=O)CN(c1ccccc1)C(=O)CSc2c(c(cc(n2)C)C)C#N HTS13274 COc1cc(cc(c1OC)OC)c2nn3cc(nc3s2)c4ccccc4 HTS13282 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3ccc(cc3)Cl)/s2 HTS13413 CCOC(=O)Cc1csc(n1)NC(=O)c2ccccc2F HTS13542 COc1ccc(cc1)c2cc(c(c(n2)N)C#N)c3ccccc3 HTS13543 c1cc(oc1)c2cc(nc(c2C#N)N)c3ccco3 HTS13545 CCOC(=O)CN(c1ccc(cc1)F)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13384 CCOC(=O)CN(c1ccccc1)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13388 c1cc(c2c(c1)OCCCO2)C(=O)Nc3ccc(cc3)C(=O)N SCR00580 CN1CCN(CC1)c2ccc(cc2)CN3CCS(=O)(=O)CC3 SCR00607 CN1CCN(CC1)c2ccc(cc2)CNC(=O)c3ccc(cc3)OC SCR00777 C/C(=N\Cc1ccccc1Cl)/c2cc(cc(c2O)Cl)Cl S05130 c1ccc2cc(ccc2c1)C(=O)CSc3nnnn3c4ccc(cc4)F S05122 COc1cc(ccc1O)C(c2c([nH]c(=S)[nH]c2=O)N)c3c([nH]c(=S)[nH]c3=O)N HTS13260 Cc1c(cc(o1)S(=O)(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4)C(=O)OC SCR00889 CCn1c(nnc1SCC(=O)Nc2c(c3c(s2)CN(CC3)C(=O)OCC)C#N)c4cccs4 HTS12789 c1c2c([nH]c(=S)[nH]c2=S)nc(n1)N3CCOCC3 HTS12794 c1ccc2c(c1)CCC3=C2NC(=S)NC3c4ccc(cc4)F HTS12616 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)NCc3ccc(cc3)N4CCN(CC4)C SCR00783 Cc1c2c([nH]n1)OC(=C(C23CCN(CC3)C)C#N)N HTS13257 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/NC(=O)c4c(nc5n4ccc(c5)C)C HTS13263 COC(=O)c1c[nH]c2c1cccc2 AC30928 c1c([nH]nc1C(F)(F)F)C(F)(F)F AC31181 c1cc(sc1)c2nc(cs2)CN3CCS(=O)(=O)CC3 SCR00604 CC(C)(C)NC(=O)NCCO S04973 CC(C)(C)NC(=O)N1CCOCC1 S04978 c1c(c(c(cn1)Cl)N2CCN(CC2)CC(C(F)(F)F)O)Cl SCR00806 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)N3CCN(CC3)Cc4ccc5c(c4)OCO5 SCR00941 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)N3CCN(CC3)c4ccc(cc4)F SCR00943 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)CN3C(=O)c4ccccc4C3=O SCR00944 COc1ccc(cc1)c2nnc(n2c3cccc(c3)OC)SCC(C(F)(F)F)O SCR00924 CCCc1c(c(on1)C)C(=O)O RG00002 c1ccc2c(c1)c(cs2)NC(=O)Nc3ccc(cc3)F HTS12345 CCOc1ccc(cc1)NC(=S)NC(c2ccccc2)c3ccccc3 S05116 C/C(=N\Cc1ccccc1)/c2cc(cc(c2O)Cl)Cl S05114 CN(C)c1ccc(cc1)C(CC(=O)c2ccc3ccccc3c2)Sc4ccccc4N S05105 c1cc(c(nc1)N2CCOCC2)Cl HTS11332 COc1ccc(cc1)C2=Nc3ccccc3SC(C2)c4cccc5c4cccc5 S05102 Cn1cccc1CNCC(C(F)(F)F)O SCR00911 Cc1cccc(n1)C2N(CCCN2Cc3ccc(cc3)OC)Cc4ccc(cc4)OC SCR00746 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3ccc(cc3)Cl SCR00827 CCOC(=O)C1CCN(CC1)C(=O)CN2C(=O)c3ccccc3C2=O SCR00947 COc1ccc(cc1OC)CC(=O)N2CCN(CC2)c3ncccn3 SCR00765 CC1(Cc2cccc(c2O1)C(=O)N3CCC(CC3)C(=O)c4ccc(cc4)Cl)C SCR00527 CC(C)(C)NC(=O)Nc1ccc2ccccc2c1 S04984 COc1ccc2c(c1)sc(n2)/N=C/c3cc(ccc3O)Br S04987 c1ccc(cc1)NNC(=S)N/N=C/c2cc(cc(c2O)Cl)Cl S04989 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3ccsc3 SCR00843 c1cc(ccc1CC#N)N2C(=O)C=CC2=O S05217 Cc1ccccc1N2C(=O)C=CC2=O S05219 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)NCc3ccsc3 SCR00957 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)NCc3ccc(cc3)N4CCOCC4 SCR00958 c1ccc(cc1)OCCNC(=O)CN2C(=O)c3ccccc3C2=O SCR00959 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)NC3CCCCC3 SCR00961 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)Nc3ccccc3N4CCOCC4 SCR00963 Cn1c2ccccc2nc1S(=O)(=O)O AC27651 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3ccc(o3)C(=O)OC SCR00847 Cc1cc(c(s1)C)S(=O)(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00845 Cc1c(c(no1)c2ccccc2)CNC(=O)CN3C(=O)c4ccccc4C3=O SCR00948 Cc1cc(c(o1)C(F)(F)F)CNC(=O)CN2C(=O)c3ccccc3C2=O SCR00949 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)NCC3COc4ccccc4O3 SCR00950 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)Nc3cccc(c3)n4cccc4 SCR00964 Cc1ccc2cc(ccc2n1)NC(=O)c3cccc4c3OC(C4)(C)C SCR00525 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(cc3)N4CCN(CC4)C)C SCR00523 COc1ccc(cc1OC)CC(=O)Nc2ccc(cc2)c3cnco3 SCR00759 CSc1cccc(c1)NC(=S)NNC(=S)NNc2ccccc2 S04990 c1ccc(cc1)n2c(ccn2)/N=C/c3cc(cc(c3O)Cl)Cl S04801 c1cc(ccc1N2C(=O)/C(=C\c3cc(ccc3Cl)Cl)/SC2=S)S(=O)(=O)Nc4nccs4 S04818 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3cccc(c3)F SCR00831 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3ccc(cc3Cl)F SCR00830 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3cc(ccc3OC)OC SCR00828 CCc1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00826 c1ccc(cc1)/C(=C/C(=C(/C#N)\c2ccc(cc2)[N+](=O)[O-])/c3ccc(cc3)Cl)/CC(=O)c4ccc(cc4)Cl HTS13247 c1ccc(cc1)C(c2ccccc2)(c3nnc(n3c4ccc(cc4)F)SCC(C(F)(F)F)O)O SCR00925 Cc1ccc(c(c1)Cl)NC(=O)CSCC(C(F)(F)F)O SCR00926 c1ccc(cc1)c2nc(nn2c3ccccc3)SCC(C(F)(F)F)O SCR00928 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)NCc3ccc4c(c3)OCO4 SCR00951 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4cccnc4)CO2 HTS12578 c1ccc2c(c1)-c3c(c(c(c(=O)[nH]3)C#N)c4ccccc4Cl)CS2 HTS12581 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC(C)(C)CO S07032 CSc1nnc(s1)NC(=O)c2c(cccc2Cl)Cl S06820 CCOC(=O)c1c2c(sc1NC(=S)N3CCN(CC3)c4ccccc4)CCCC2 HTS12986 c1ccc(cc1)CN(CC(=O)Nc2cccnc2)CC(=O)O SCR00482 CN1CCN(CC1)c2ccc(cc2)CNS(=O)(=O)c3cccc4c3non4 SCR00842 Cn1cc(nc1)S(=O)(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00840 Cc1csc(c1C(=O)N)NC(=O)CN2C(=O)c3ccccc3C2=O SCR00965 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)Nc3ccc(cc3)F SCR00969 c1cc(c(cc1S(=O)(=O)NC2CCCCNC2=O)F)F SCR00972 Cc1ccc(cc1S(=O)(=O)NC2CCCCNC2=O)F SCR00974 c1cc2c(cc1n3c(=O)c4cc(cc(c4[nH]c3=S)Br)Br)OCCO2 S05301 COC(=O)c1ccccc1NC(=S)Nc2ccc(cn2)Cl S04833 CC(C)c1cccc(c1NC(=O)c2ccccc2)C(C)C S05038 CCOc1ccc(cc1)n2c(=O)c3cc(cc(c3[nH]c2=S)Br)Br S05298 Cc1cc(c(s1)C)S(=O)(=O)NC2CCCCNC2=O SCR00981 Cc1c2cc(ccc2sc1S(=O)(=O)NC3CCCCNC3=O)Cl SCR00982 c1cc(cc(c1)S(=O)(=O)NC2CCCCNC2=O)C(F)(F)F SCR00983 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CC4)OC(=O)c5cccs5 HTS12589 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CC4)OC(=O)c5ccc(cc5)Cl HTS12592 Cc1cc(=O)n2c(n1CC(=O)NN)ncn2 HTS13254 COc1ccc(cc1)CN2CCCN(C2c3csc4c3cccc4)Cc5ccc(cc5)OC SCR00744 c1cc(ccc1OC(F)(F)F)S(=O)(=O)NC2CCCCNC2=O SCR00975 c1cc(c(c(c1)Cl)CSc2nnc(s2)c3ccncc3)F S07108 c1cc(c(c(c1)Cl)C(=O)N/N=C/c2cccnc2)Cl S06945 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4ccc(cc4)F)c5ccccc5 HTS13391 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4ccc(cc4)Cl)c5ccccc5 HTS13393 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4cccc(c4)Cl)c5ccccc5 HTS13394 Cn1c(nnc1SCC(=O)c2cccs2)c3cc(c(c(c3)OC)OC)OC HTS13396 c1cc(ccc1NC(=O)CN2CCCCC2)S(=O)(=O)N HTS13519 c1ccc2c(c1)CCN2CC(=O)Nc3c4c(cs3)c5ccccc5oc4=O HTS13475 COc1cccc(c1)C(=O)COc2c(c(cc(n2)c3cccs3)c4ccco4)C#N HTS13487 c1cc(oc1)c2cc(nc3c2c(c(o3)C(=O)c4ccc(cc4)F)N)c5cccs5 HTS13491 CC(=O)Nc1ccc(cc1)C2C(CCC(=O)N2)[N+](=O)[O-] S05374 Cc1c(c(no1)c2ccccc2)C(=O)N(Cc3ccccn3)Cc4ccccn4 SCR00627 c1ccc(cc1)c2nc(cs2)C(=O)N(Cc3ccccn3)Cc4ccccn4 SCR00631 COc1ccc(cc1OC)CC(=O)NCC2COc3ccccc3O2 SCR00770 Cc1cc(c(o1)C(F)(F)F)CNC(=O)Cc2ccc(c(c2)OC)OC SCR00769 COc1ccc(cc1OC)CC(=O)Nc2ccc(cc2)S(=O)(=O)N SCR00755 c1ccc2c(c1)cccc2CC(=O)NNC(=O)Nc3ccc(cc3)Cl S07422 COc1cccc(c1)c2cs/c(=N\Cc3cccnc3)/n2c4ccccc4 HTS13534 Cc1cccc(n1)/N=c\2/n(c(cs2)c3ccco3)c4ccccc4 HTS13539 COc1cc2c(cc1OC)CN(CC2)S(=O)(=O)c3ccc(c(c3)F)F SCR01113 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4ccccc4)C HTS13312 Cc1ccc(cc1)c2cc(c(c(=O)[nH]2)C#N)c3cccs3 HTS13329 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3ccc(cc3)OC)/s2 HTS13407 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3cccc(c3)OC)/s2 HTS13409 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3cc(c(c(c3)OC)OC)OC)/s2 HTS13412 COc1ccc(cc1)n\2c(cs/c2=N\Cc3cccnc3)c4cccc(c4)OC HTS13532 c1ccnc(c1)/N=c\2/n(c(cs2)c3cccs3)c4ccc(cc4)F HTS13536 Cc1c(cnn1c2ccc(cc2)OC)C(=O)Nc3ccc4c(c3)nccn4 SCR01279 c1cc(ccc1c2nnc3n2C(=O)CS3)Cl HTS13349 Cc1ccccc1N2CC(=O)Nc3c4c(cc(nc4sc3C2=O)C)C HTS13363 CCNc1c2cnc(nc2nc(n1)SCc3ccc(cc3)[N+](=O)[O-])N(CC)CC HTS13383 c1cc2c(cc1[N+](=O)[O-])c(ns2)N AC34541 COc1ccc(cc1OC)CC(=O)Nc2ccc(cc2)C(=O)O SCR00753 c1cc(cc(c1)F)NC(=S)Nc2ccc(cn2)Cl S04879 Cc1cc(ccc1n2c(=O)c3ccccc3[nH]c2=S)Br S04884 CNC(=O)NC(=O)CSc1nnc(n1CC=C)c2cc(c(c(c2)OC)OC)OC HTS13398 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2c3ccccc3 HTS13399 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2C3CCCCC3 HTS13403 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2Cc3ccccc3 HTS13404 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2c3ccc(cc3)Cl HTS13400 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3cccs3)/s2 HTS13408 Cc1ccc(cc1)/C=c\2/c(=O)n3c4ccccc4nc3s2 HTS13421 COc1cc2c(cc1OC)CN(CC2)S(=O)(=O)c3ccc(cc3)Cl SCR01112 CC1(CCc2cc(ccc2O1)S(=O)(=O)N3CCc4cc(c(cc4C3)OC)OC)C SCR01111 CCOC(=O)CSc1c2c3c(sc2nc(n1)SCC(=O)OCC)CCC3 HTS13330 Cc1cc(ccc1NC(=S)NCCCN2CCOCC2)Br S04891 Cc1cc(cc(c1)NC(=S)Nc2ccc(cc2C)Br)C S04892 c1ccc2cc(ccc2c1)NC(=S)Nc3cccc(c3)F S04894 c1ccc2cc(ccc2c1)NC(=S)Nc3cc(c(cc3Cl)Cl)Cl S04895 c1cc(c(c(c1)Cl)N2C(SCC2=O)c3cccnc3)F S07593 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)NC3CCCCNC3=O SCR00991 c1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)C(=O)NC4CCCCNC4=O SCR00992 Cc1ccc(cc1C)C(=O)NC2CCCCNC2=O SCR00995 C=CCSc1ncc2c(n1)[nH]c(=S)[nH]c2=S HTS12796 CCN(CC)c1ncc2c(n1)[nH]c(=S)[nH]c2=S HTS12797 Cn1c2ccccc2oc1=S AC29729 CSc1nc2ccccc2c(n1)N AC29790 C1CSCCC1(C(=O)O)N.Cl AC36050 Cc1ccc(cc1)CSc2nnc(s2)Nc3ccc(cc3)Cl S06844 CCNc1c2c3c(sc2nc(n1)SCC(=O)N)CN(CC3)C HTS13527 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3ccc(cc3)F)/s2 HTS13415 Cc1ccc(o1)/C=c\2/c(=O)n3c(c(nc3s2)c4ccccc4)c5ccccc5 HTS13416 c1ccc(cc1)c2c(n3c(=O)/c(=C/c4cccs4)/sc3n2)c5ccccc5 HTS13417 c1ccc2c(c1)nc3n2c(=O)/c(=C/c4ccc(cc4)F)/s3 HTS13419 c1ccc2c(c1)nc3n2c(=O)/c(=C/c4cccs4)/s3 HTS13420 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2Cl)Cl)C HTS13449 c1ccc(cc1)C2=N/C(=C\c3ccccc3Cl)/C(=O)NN2 HTS13458 c1ccc2c(c1)/C(=C/c3ccc4c(c3)nsn4)/C(=O)N2 SCR01015 c1ccc2c(c1)/C(=C/c3cc(cc4c3OCOC4)F)/C(=O)N2 SCR01008 CN1CCOc2c1ccc(c2)/C=C\3/c4ccccc4NC3=O SCR01009 c1ccc2c(c1)/C(=C/c3ccc4c(c3)OCCO4)/C(=O)N2 SCR01012 CCOC(=O)c1ccc(c(c1)NC(=S)NN)Cl S05418 COc1ccc(cc1)/N=C/c2c3ccccc3ccc2O S04899 Cc1cc(nn1C)C(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 SCR00686 Cc1cc(nn1C)C(=O)N2CCN(CC2)c3ncccn3 SCR00688 Cc1cc(nn1C)C(=O)Nc2ccccc2N3CCCCC3 SCR00697 Cc1c(cc(o1)S(=O)(=O)N2CCN(CC2)c3ccc(cc3)OC)C(=O)OC SCR00899 Cc1c(cc(o1)S(=O)(=O)N(C)Cc2ccccc2)C(=O)OC SCR00892 c1ccc2c(c1)/C(=C/c3ccc(nc3)N4CCOCC4)/C(=O)N2 SCR01017 c1ccc(cc1)Oc2ccsc2/C=C\3/c4ccccc4NC3=O SCR01018 CC(C)(C)C(=O)Nc1c(cccn1)/C=C\2/c3ccccc3NC2=O SCR01019 CCOC(=O)c1c2c(sc1N)CN(CC2)C(=O)OCC HTS12803 c1ccc2c(c1)n3c(nnc3s2)S HTS12805 CC1(Cc2cccc(c2O1)C(=O)Nc3ccc(cc3)c4csnn4)C SCR00522 CNC(=O)NC(=O)CSc1nnc2n1c3ccccc3s2 HTS12807 CC1(CC(=O)CC(N1)(C)C)C AC42061 CC(C)(C)c1ccc(cc1)NC(=S)Nc2nc[nH]n2 S06867 CC(C)(C)c1ccc(cc1)/N=C(/NCc2cccnc2)\SC S06868 c1ccc(cc1)c2csc(n2)NNC(=O)c3ccc(cc3)Cl HTS13465 COc1cccc(c1)c2csc(n2)NNC(=O)c3cccs3 HTS13467 c1nc2c3c4c(sc3ncn2n1)CCC4 HTS13468 Cc1ccc(cn1)C2N(C(=O)CS2)c3ccc(cc3)Br S07682 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)NCCc3ccccn3 SCR01252 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4cc(cc5c4OCOC5)F SCR00542 CCN(CC)CC(=O)NN1CC(=O)N(CC1=O)c2cccc(c2)Cl HTS13272 c1c2c(ncnc2nc(n1)N3CCCC3)N HTS13265 c1c2c(=O)[nH]cnc2nc(n1)N3CCOCC3 HTS13266 c1cc(ccc1N2CC(=O)N(CC2=O)NC(=O)CN3CCCCC3)F HTS13267 CN1CCN(CC1)CC(=O)NN2CC(=O)N(CC2=O)c3ccc(cc3)F HTS13270 c1ccc(cc1)C2=N/C(=C/c3cn(nc3c4cccs4)c5ccccc5)/C(=O)O2 HTS13470 c1ccc2c(c1)c3cc(c(c(c3c(=O)o2)N)C#N)c4cccs4 HTS13472 c1ccc2c(c1)c3cc(c(c(c3c(=O)o2)N)C#N)c4ccc(cc4)Cl HTS13473 c1cc(sc1)c2nc(cs2)CNC(=O)c3ccc4c(c3)nsn4 SCR01305 Cc1c(snn1)C(=O)NCc2csc(n2)c3cccs3 SCR01304 c1cc(oc1)C(=O)NCc2csc(n2)c3cccs3 SCR01303 c1cc(sc1)c2nc(cs2)CNC(=O)c3ccc4c(c3)CCO4 SCR01302 c1cc(cnc1)/C=N/NC(=O)c2ccncc2 S07083 c1ccc(cc1)Oc2ccc(cc2)/N=C/c3ccccc3O S05065 c1ccc(cc1)C(=O)Nc2c3c(cs2)c4ccccc4oc3=O HTS13481 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)c4ccc(cc4)F HTS13482 COc1cc(cc(c1OC)OC)C(=O)Nc2c3c(cs2)c4ccccc4oc3=O HTS13483 Cc1ccc(c(c1)Cl)N2C(SCC2=O)c3cccnc3 S07760 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)Nc4cccc(c4)Cl HTS13496 c1cc(sc1)c2nc(cs2)CNC(=O)C3CC3 SCR01296 c1cc(sc1)c2nc(cs2)CNC(=O)C3CCCCC3 SCR01295 c1cc(cc(c1)Cl)C(=O)NCc2csc(n2)c3cccs3 SCR01294 Cc1ccc(cc1C)C(=O)NCc2csc(n2)c3cccs3 SCR01316 COc1cc2c(cc1OC)CN(CC2)S(=O)(=O)c3cccs3 SCR01106 COc1ccc(c(c1)S(=O)(=O)N2CCc3cc(c(cc3C2)OC)OC)OC SCR01114 Cc1c(sc(n1)C)S(=O)(=O)NCc2csc(n2)c3cccs3 SCR01204 CCOC(=O)CN(c1ccc(cc1)Cl)C(=O)CSc2c(c(cc(n2)C)C)C#N HTS13275 c1cc(sc1)c2nnc3n2C(=O)CS3 HTS13348 Cc1cc(nc2c1c(c(s2)C(=O)Nc3nnc(s3)c4cccs4)N)C HTS13283 C=CCn1c(nnc1SCC(=O)Nc2nnc(s2)c3cccs3)c4ccco4 HTS13285 Cc1cc(nc(c1C#N)SCC(=O)Nc2nnc(s2)c3cccs3)C HTS13287 c1ccc2c(c1)c3cc(c(c(c3c(=O)o2)N)C#N)c4cccnc4 HTS13474 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3c4c(cs3)c5ccccc5oc4=O HTS13476 c1cc(oc1)c2cc(nc(c2C#N)OCc3ccc(cc3)F)c4cccs4 HTS13489 C=CCOc1c(c(cc(n1)c2cccs2)c3ccco3)C#N HTS13490 COc1cccc(c1)C(=O)c2c(c3c(cc(nc3o2)c4cccs4)c5ccco5)N HTS13492 c1cc(sc1)c2nc(cs2)CNC(=O)C3CCC3 SCR01313 c1ccc2c(c1)C=C(CO2)C(=O)NCc3csc(n3)c4cccs4 SCR01311 c1ccc(cc1)c2nc(cs2)C(=O)NCc3csc(n3)c4cccs4 SCR01310 c1cc(sc1)c2nc(cs2)CNC(=O)c3ccsc3 SCR01309 Cc1cc(no1)C(=O)NCc2csc(n2)c3cccs3 SCR01308 CC(C)c1ccc(cc1)NC(=O)c2cc(cc3c2OCOC3)F SCR00575 c1ccc(cc1)Oc2ccc(cc2)/N=C/c3cc(cc(c3O)Cl)Cl S05064 c1ccc2c(c1)ccc3c2ccc4c3ccc(c4)/N=C/c5ccccc5O S05060 c1ccc2c(c1)ccc3c2ccc4c3ccc(c4)/N=C/c5cc(cc(c5O)Cl)Cl S05059 c1c(cc(cc1C(F)(F)F)NC(=O)COc2cc(c(cc2Cl)Cl)Cl)C(F)(F)F S05058 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)Nc4ccc(c(c4)Cl)Cl HTS13498 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)Nc4ccc(cc4)Cl HTS13499 c1ccc(cc1)NC(=O)Nc2c3c(cs2)c4ccccc4oc3=O HTS13500 c1ccc-2c(c1)Cc3c2ccc(c3)Br BTB10462 CN1C2CCC1CC(C2)O BTBG00136 CNc1ccc(cc1)S(=O)(=O)O JFD03588 Cc1c(c2ccccc2o1)CNC(=O)Nc3ccc(cc3)Br S07649 Cc1c(c2ccccc2o1)CNC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F S07651 CN1C2/C(=C\c3ccc(cc3)F)/C(=O)/C(=C/c4ccc(cc4)F)/C1CC2 SCR01116 c1cc(oc1)c2nnc(s2)NC(=O)CSc3nnc(o3)c4ccc(cc4)Cl HTS13291 Cc1cc(nc2c1c(c(s2)C(=O)NN3CC(=O)N(CC3=O)c4ccccc4)N)C HTS13358 CCOC(=O)CN(c1ccccc1)C(=O)COc2c(c(cc(n2)c3cccs3)c4ccco4)C#N HTS13299 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4ccccc4)c5ccccc5 HTS13300 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4cccc(c4)OC)c5ccccc5 HTS13301 C1CCN(CC1)CC(=O)Nc2c(c3c(s2)CCC3)C#N HTS13493 c1ccc(cc1)Nn2cnc3c(c2=N)c4c(s3)CCC4 HTS13503 Cc1cc(nc2c1c(c(s2)C(=O)Nc3ccc(cc3)S(=O)(=O)N)N)C HTS13504 c1ccc(cc1)n2c(nnc2SCC(=O)Nc3ccc(cc3)S(=O)(=O)N)c4ccco4 HTS13505 c1ccc2c(c1)C=C(CO2)C(=O)Nc3ccc4c(c3)OCC5N4CCC5 SCR01117 COc1ccc(c(c1)C(=O)NCc2ccc(cc2)Cl)Br S07104 COc1ccc(c(c1)C(=O)NCc2ccc(cc2Cl)Cl)Br S07106 c1ccc2c(c1)c(c3c(n2)CCCC3)C(=O)O AC42043 c1cc(ccc1C(=O)NCc2ccc(s2)S(=O)(=O)NCCN3CCCC3)Cl SCR00664 Cc1ccccc1S(=O)(=O)NCc2ccc(cc2)N3CCN(CC3)C SCR00825 CCOC(=O)CN(c1ccc(cc1)Cl)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13386 c1ccc(cc1)c2c(n3c(=O)/c(=C/c4cccnc4)/sc3n2)c5ccccc5 HTS13418 c1ccc(cc1)COc2ccc(cc2)/C=C/3\C(=O)NNC(=N3)c4ccccc4 HTS13455 Cc1c(c2ccccc2o1)CNC(=O)N S07654 c1cc2c(c(c1)S(=O)(=O)NCc3csc(n3)c4cccs4)non2 SCR01205 c1ccc(cc1)Oc2ccc(cn2)S(=O)(=O)NCc3csc(n3)c4cccs4 SCR01211 CN(C)c1cccc2c1cccc2S(=O)(=O)NCc3ccc(cc3)S(=O)(=O)N SCR01146 Cn1c(nnc1SCC(=O)c2ccco2)c3cc(c(c(c3)OC)OC)OC HTS13302 c1ccc(cc1)c2cn3c(n2)sc(n3)c4cccs4 HTS13372 Cc1c(c(c2c(c1C)[nH]c(n2)c3ccc4c(c3)OCO4)C)C SCR01506 C=CCn1c(nnc1SCC(=O)Nc2ccc(cc2)S(=O)(=O)N)c3cccs3 HTS13508 COc1cc(cc(c1OC)OC)/C=c\2/c(=O)n3c(nnc3s2)c4cccs4 HTS13369 c1ccc(cc1)CS(=O)(=O)NCc2ccc(cc2)S(=O)(=O)N SCR01147 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2CC=C HTS13401 CCOC(=O)CN(c1cccc(c1)Cl)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13387 CCOC(=O)CN(c1cccc(c1)OC)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13389 c1ccc(cc1)c2nnc(o2)SCC(=O)Nc3ccc(cc3)S(=O)(=O)N HTS13511 c1cc(ccc1C(=S)N)Oc2ccc(cn2)C(F)(F)F SPB03013 c1cnc(nc1C(F)(F)F)NN HAN00391 Cc1cc(cc(c1)NC(=O)NCc2csc(n2)c3cccs3)C SCR01337 c1cc(sc1)c2nc(cs2)CNC(=O)Nc3ccc(cc3F)F SCR01336 COc1ccccc1CC(=O)NCc2ccc(cc2)c3cccs3 SCR01427 Cc1c(c(on1)C)NC(=O)Nc2cccc(c2)S(=O)(=O)N SCR01491 Cc1cc(c(o1)C(F)(F)F)CNC(=O)Nc2c(noc2C)C SCR01489 Cc1c(c(on1)C)NC(=O)NC(c2ccccc2)c3ccccc3 SCR01485 Cc1c(c(on1)C)NC(=O)NCCOc2ccccc2 SCR01484 Cc1c(nn(n1)c2ccccc2)CNC(=O)c3ccc4c(c3)nsn4 SCR01436 Cc1c(c2ccccc2o1)CC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F S07532 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NCc3ccc(cc3)S(=O)(=O)N SCR01149 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)Nc3cc(n[nH]3)c4ccc(cc4)Cl SCR01227 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccc3c(c2)OCCO3 SCR00634 Cc1c(c(on1)C)NC(=O)NC2CCCCNC2=O SCR01477 c1cc(cnc1)CN2CCN(CC2)C(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl SCR01068 COc1cc2c(cc1OC)CN(CC2)S(=O)(=O)c3ccccc3 SCR01103 Cn1c(cc(n1)c2ccc(s2)S(=O)(=O)NC3CCCCNC3=O)C(F)(F)F SCR00996 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)NC3CCCCNC3=O SCR00979 Cn1c(nnc1SCC(=O)NC(=O)NCc2ccccc2)c3cc(c(c(c3)OC)OC)OC HTS13303 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4ccc(cc4)Cl)C HTS13313 c1ccc(cc1)c2cs/c(=N\Cc3cccnc3)/n2c4ccccc4 HTS13535 c1cc(sc1)c2nc(cs2)CNS(=O)(=O)Cc3ccc(cc3)Cl SCR01214 Cn1cc(nc1)S(=O)(=O)NCc2csc(n2)c3cccs3 SCR01202 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)NCc3cc(cc4c3OCOC4)F SCR00952 Cn1c(cc(n1)C2CC2)NC(=O)CN3C(=O)c4ccccc4C3=O SCR00967 c1ccnc(c1)CCNS(=O)(=O)c2ccc(s2)c3ccccn3 SCR01248 c1ccc(cc1)n2c(c(cn2)C(=O)Nc3ccc4c(c3)nccn4)C(F)(F)F SCR01271 c1ccc2c(c1)cccc2CC(=O)Nc3ccc4c(c3)nccn4 SCR01273 c1cc(ncc1S(=O)(=O)N2CCSCC2)N3CCOCC3 SCR01191 c1cc(ncc1S(=O)(=O)N2CCC(CC2)C(=O)N)N3CCOCC3 SCR01190 c1cc2c(c(c1)S(=O)(=O)NCc3ccc(cc3)S(=O)(=O)N)non2 SCR01153 c1cc(sc1)c2csc(n2)NNC(=O)c3ccc(cc3)Cl HTS13319 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)c4cccs4 HTS13325 c1ccc(c(c1)/C=c\2/c(=O)n3c4ccccc4nc3s2)Cl HTS13422 c1ccc2c(c1)c3cc(c(c(c3c(=O)o2)N)C#N)c4ccc(cc4)F HTS13322 Cc1ccc(cc1)c2cc3c4ccccc4oc(=O)c3c(c2C#N)N HTS13323 c1cc(cc(c1)C(F)(F)F)CS(=O)(=O)NCc2csc(n2)c3cccs3 SCR01215 Cc1nc2c3c4c(sc3ncn2n1)CCC4 HTS13469 c1cc(c(nc1)Oc2ccc(cc2)Cl)C(=O)Nc3ccc4c(c3)nccn4 SCR01280 c1cc(cnc1)C2CCCCN2S(=O)(=O)c3ccc4c(c3)nsn4 SCR00454 Cc1cc(cc(c1)NC(=S)NCCc2ccc(c(c2)OC)OC)C S05281 CC1(Cc2cccc(c2O1)C(=O)Nc3cccc4c3CCCC4)C SCR00521 c1ccc2c(c1)CCN2CC(=O)Nc3nnc(s3)c4cccs4 HTS13432 c1ccc(cc1)CN(Cc2ccccc2)CC(=O)Nc3nnc(s3)c4cccs4 HTS13433 c1ccnc(c1)CCNC(=O)c2csc(n2)Cc3c(cccc3Cl)Cl SCR01265 CC(C)(C)c1cc(n(n1)C)C(=O)Nc2ccc3c(c2)nccn3 SCR01272 c1cc(c(cc1Cl)Cl)CNS(=O)(=O)c2ccc(nc2)N3CCOCC3 SCR01174 Cc1c(cnn1c2ccc(cc2)OC)C(=O)NCCc3ccccn3 SCR01262 c1ccnc(c1)CCNC(=O)c2cccnc2Oc3ccc(cc3)Cl SCR01260 c1ccnc(c1)CCNS(=O)(=O)c2ccc(cc2)OC(F)(F)F SCR01258 COc1ccc(c(c1)S(=O)(=O)NCCc2ccccn2)OC SCR01257 c1ccnc(c1)CCNS(=O)(=O)c2ccc(s2)c3ccno3 SCR01256 CCOC(=O)Cn1c(c(nc1c2cccnc2)c3ccccc3)c4ccccc4 HTS13437 CCOC(=O)CN(c1cccc(c1)Cl)C(=O)COc2c(c(cc(n2)C)C)C#N HTS13453 CC(C)(C)c1ccc(cc1)C(=O)NCCc2ccc(c(c2)OC)OC S07384 c1cc2c(cc1Cl)oc(n2)O AC29726 c1c(nc2c(nc(nc2n1)N)N)CO.Cl AC29806 c1c(cc(c(c1/C=N/CCO)O)Cl)Cl S04960 CCOc1ccc(cc1)NC(=O)NC(C)(C)C S04972 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)/N=C/c4c5ccccc5ccc4O S04967 CCOC(=O)C1=C(NC(=O)NC1c2ccc(o2)C)C HTS13445 CCOC(=O)C1=C(NC(=O)NC1c2ccccn2)C HTS13446 CCOC(=O)C1=C(NC(=O)NC1c2cccnc2)C HTS13447 c1cc(cc(c1)Cl)CNC(=O)C(C(C(=O)O)(F)F)(F)F SCR00279 c1cc(sc1)c2ccc(cc2)CNC(=O)c3cc(cc4c3OCOC4)F SCR00557 c1ccc(cc1)S(=O)(=O)NCc2csc(n2)c3cccs3 SCR01195 Cc1ccc(cc1)/C=C/2\C(=O)NNC(=N2)c3ccccc3 HTS13454 COc1cc(cc(c1OC)OC)/C=C\2/C(=O)NNC(=N2)c3ccccc3 HTS13456 c1ccc(cc1)C2=N/C(=C\c3ccc(cc3)Cl)/C(=O)NN2 HTS13457 c1ccc(cc1)c2nc(c(=O)n(n2)CN3CCOCC3)C(CN4CCOCC4)c5ccc(cc5)Cl HTS13343 Cc1ccc(cc1)C(CN2CCOCC2)c3c(=O)n(nc(n3)c4ccccc4)CN5CCOCC5 HTS13346 c1ccc2c(c1)ncc(n2)C(=O)NCc3cccnc3 SCR00533 CC1(Cc2cccc(c2O1)C(=O)NC3CCN(CC3)Cc4ccccc4)C SCR00503 COc1ccc(cc1OC)CC(=O)NCc2cc3ccccc3s2 SCR00774 COc1ccc(cc1OC)CC(=O)NCc2csc(n2)c3cccs3 SCR00773 c1ccc2c(c1)cc(s2)CNCC(C(F)(F)F)O SCR00713 c1ccc(cc1)n2c(ccn2)/N=C/c3ccccc3O S04803 c1ccnc(c1)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)S(=O)(=O)Nc4nccs4 S04811 COc1cc(cc(c1OC)OC)C(CN2CCCCC2)c3c(=O)n(nc(n3)c4ccccc4)CN5CCCCC5 HTS13342 c1ccc(cc1)C2=N/C(=C\c3ccco3)/C(=O)NN2 HTS13461 c1cc(ccc1n2c(=N)c3cnc(nc3[nH]c2=O)N4CCCC4)Cl HTS13462 c1ccc(cc1)N2CC(=O)N(CC2=O)NC(=O)CN3CCc4c3cccc4 HTS13354 COc1ccc(cc1)c2cc(c3ccccc3n2)C(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F S07778 COc1ccc(cc1)c2cc(c3ccccc3n2)C(=O)Nc4cc(cc(c4)Cl)Cl S07781 COc1ccccc1CC(=O)NCc2csc(n2)c3cccs3 SCR01299 c1ccc(cc1)c2nc(c(=O)n(n2)CN3CCCCC3)C(CN4CCCCC4)c5ccccc5Cl HTS13344 Cc1nccc(n1)c2cccc(c2)NC(=O)c3nc4ccccc4s3 SCR01081 c1ccc2c(c1)cc(s2)S(=O)(=O)NCc3csc(n3)c4cccs4 SCR01206 c1cc(sc1)c2nc(cs2)CNS(=O)(=O)c3cccs3 SCR01207 c1cc(sc1)c2nc(cs2)CNS(=O)(=O)c3ccc4c(c3)OCCCO4 SCR01208 CN1CCOc2c1cc(cc2)S(=O)(=O)NCc3csc(n3)c4cccs4 SCR01209 Cc1c(cn(n1)c2ccccc2)/C=c\3/c(=O)n4c5ccccc5nc4s3 HTS13281 c1ccc(cc1)c2nnc3n2C(=O)CS3 HTS13350 c1cnccc1c2[nH]c(nn2)SCC(=O)O HTS13378 c1ccc(cc1)c2cc3c4ccccc4oc(=O)c3c(c2C#N)N HTS13471 Cc1cc(nc2c1c(c(s2)C(=O)NN3CC(=O)N(CC3=O)c4cccc(c4)Cl)N)C HTS13359 c1ccc(cc1)n2c3c(cn2)c(ncn3)N4CCc5c4cccc5 HTS13361 Cc1cc(nc2c1c3c(s2)C(=O)N(CC(=O)N3)c4cccc(c4)Cl)C HTS13362 COc1ccc(cc1OC)CC(=O)Nc2ccccc2N3CCCCC3 SCR00758 COc1ccc(cc1OC)CC(=O)Nc2ccc(cc2)N3CCOCC3 SCR00757 COc1ccc(cc1OC)CC(=O)Nc2cccc(c2)Cl SCR00754 COc1ccc(cc1)/C=C/2\C(=O)N(C(=S)S2)c3ccc(cc3)S(=O)(=O)Nc4nccs4 S04817 c1ccc(cc1)S(=O)(=O)N(Cc2ccccn2)Cc3ccccn3 SCR00610 CC1(CCc2cc(ccc2O1)S(=O)(=O)N(Cc3ccccn3)Cc4ccccn4)C SCR00614 c1ccc(cc1)N2CCN(CC2)CC(=O)NN3CC(=O)N(CC3=O)c4cccc(c4)Cl HTS13353 CCOC(=O)CN(c1ccc(cc1)F)C(=O)CSc2c(c(cc(n2)C)C)C#N HTS13355 CCOC(=O)CN(c1cccc(c1)Cl)C(=O)CSc2c(c(cc(n2)C)C)C#N HTS13356 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)CN4CCCCC4 HTS13478 Cc1ccc(cc1)/C=c\2/c(=O)n3c(nnc3s2)c4ccco4 HTS13367 CCOC(=O)CN(c1ccccc1C)C(=O)CSc2c(c(cc(n2)C)C)C#N HTS13357 Cc1cc(nc2c1c(c(s2)C(=O)NN3CC(=O)N(CC3=O)c4ccc(cc4)F)N)C HTS13360 CC(C)(C)OC(=O)NCC1CCN(CC1)Cc2ccccc2 MO00974 CC(C)(C)c1ccc(cc1)C(=O)NCc2cccs2 S07671 Cc1c2cc(ccc2sc1S(=O)(=O)NCc3ccc(cc3)S(=O)(=O)N)Cl SCR01164 CCOC(=O)CN(c1ccc(cc1)C)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13298 CC(=O)Nc1c2c(cs1)c3ccccc3oc2=O HTS13485 COc1cccc(c1)c2cc(c(c(=O)[nH]2)C#N)c3cccs3 HTS13486 c1cc(sc1)c2nn3cc(nc3s2)c4ccc(cc4)F HTS13374 c1ccc(cc1)NC(=O)NC(=O)CSc2[nH]c(nn2)c3ccncc3 HTS13376 CCOC(=O)CSc1[nH]c(nn1)c2ccncc2 HTS13377 c1ccc(cc1)C(=O)NCc2csc(n2)c3cccs3 SCR01314 C=CCSc1nc2c(cnc(n2)N3CCOCC3)c(n1)Nc4ccc(cc4)Cl HTS13379 Cc1ccc(cc1)N2CC(=O)Nc3c4c(cc(nc4oc3C2=O)c5ccccc5)C HTS13395 Cn1c(n[nH]c1=S)c2cc(c(c(c2)OC)OC)OC HTS13402 CCOC(=O)Cc1ccc(cc1)[N+](=O)[O-] RH01326 c1cc(cc(c1)NNC(=S)Nc2ccc3c(c2)OCCO3)C(F)(F)F S05311 c1cc(ccc1N2CCN(CC2)C(=O)c3cc(cc4c3OCOC4)F)F SCR00544 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)N(Cc3ccccn3)Cc4ccccn4 SCR00615 Cc1c(c(on1)C)S(=O)(=O)N(Cc2ccccn2)Cc3ccccn3 SCR00618 c1ccc2c(c1)nc(s2)SCCO S04857 Cc1ccc(o1)/C=c\2/c(=O)n3c(nnc3s2)c4ccco4 HTS13368 c1ccc(cc1)/C=c\2/c(=O)n3c(nnc3s2)c4cccs4 HTS13370 c1cc(sc1)c2nnc3n2c(=O)/c(=C/c4ccc(cc4)Cl)/s3 HTS13371 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3c(c4c(s3)CCC4)C#N HTS13495 CCn1c(nnc1SCC(=O)Nc2ccc(cc2)S(=O)(=O)N)c3cccc(c3)[N+](=O)[O-] HTS13509 CN1CCOc2c1cc(cc2)S(=O)(=O)NCc3ccc(cc3)S(=O)(=O)N SCR01155 c1cc(oc1)c2nnc(o2)SCC(=O)Nc3nnc(s3)c4cccs4 HTS13284 Cn1c(nnc1SCC(=O)Nc2nnc(s2)c3cccs3)c4ccncc4 HTS13286 c1ccc(cc1)Cn2c(nnc2SCC(=O)Nc3nnc(s3)c4ccco4)c5ccncc5 HTS13290 CCOC(=O)CN(c1ccccc1)C(=O)CSc2[nH]c(nn2)c3ccncc3 HTS13292 c1ccc(cc1)CSc2nc3c(cnc(n3)N4CCOCC4)c(n2)Nc5ccc(cc5)Cl HTS13380 c1cc(ccc1Oc2ccc(cc2[N+](=O)[O-])C(=O)O)Cl SPB01167 CCCOc1c(cc(cc1Cl)C(=O)O)Cl SPB00180 c1cc(ccc1C(C(CO)NC(=O)C(Cl)Cl)O)[N+](=O)[O-] JFD01781 CSc1ccc(cc1)OCc2ccc(cc2)C(=O)O S08036 CN/N=C/c1cc(cc(c1O)Cl)Cl S05344 CN/N=C/c1ccc(s1)[N+](=O)[O-] S05345 c1cc(cnc1)C2C(CCC(=O)N2)[N+](=O)[O-] S05369 c1ccc(cc1)c2cc(cc(=O)[nH]2)c3ccc(cc3)Cl SCR01082 c1ccc(c(c1)/C=N/c2ccc(cc2)S(=O)(=O)NC(=N)/N=C/c3ccccc3O)O S04863 CC(C)c1ccccc1NC(=S)N(C)C S05027 c1cc(ccc1c2cc([nH]n2)NC(=O)c3ccc4c(c3)nsn4)Cl SCR01228 c1ccc(cc1)n2c(nnc2SCC(=O)Nc3ccc(cc3)S(=O)(=O)N)c4ccncc4 HTS13513 c1cc(ccc1c2nnc(o2)SCC(=O)Nc3ccc(cc3)S(=O)(=O)N)Cl HTS13515 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3ccc(cc3)S(=O)(=O)N HTS13518 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3ccccc3Cl)/s2 HTS13410 Cc1c(cnn1c2ccc(cc2)OC)C(=O)NCc3ccc(cc3)c4cccs4 SCR01425 c1ccc(cc1)c2c(nco2)C(=O)NCc3ccc(cc3)c4cccs4 SCR01424 c1ccc2c(c1)C=C(CO2)C(=O)NCc3ccc(cc3)c4cccs4 SCR01421 Cc1c(c(on1)C)NC(=O)Nc2ccccc2N3CCOCC3 SCR01493 Cc1c(c(on1)C)NC(=O)Nc2ccc(cc2)N(C)C SCR01492 c1cc(c(cc1NC(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F)C(=O)O)N4CCOCC4 HTS11145 c1cc2c(c(c1)S(=O)(=O)NCc3ccc(cc3)S(=O)(=O)N)nsn2 SCR01152 Cc1c(sc(n1)c2cnccn2)C(=O)Nc3cc(n[nH]3)c4ccc(cc4)Cl SCR01230 COc1cccc(c1)c2cc3c4ccccc4oc(=O)c3c(c2C#N)N HTS13320 c1cc(ccc1CNC(=O)c2cc(cc3c2OCOC3)F)N4CCOCC4 SCR01510 c1c(cc(cc1Cl)Cl)S(=O)(=O)N BTB05603 CC(=O)c1ccn(c1)S(=O)(=O)c2ccccc2 BTB07103 c1ccc2c(c1)/C(=C/c3ccc4c(c3)CCO4)/C(=O)N2 SCR01011 c1ccc2c(c1)nc3n2c(=O)/c(=C/c4cccnc4)/s3 HTS13423 Cc1ccc(o1)/C=c\2/c(=O)n3c4ccccc4nc3s2 HTS13424 c1cc(sc1)c2nc(cs2)CNC(=O)Nc3cc(cc4c3OCOC4)F SCR01332 Cc1cc(nc(c1C#N)SCC(=O)Nc2ccc(cc2)S(=O)(=O)N)C HTS13514 Cc1ccc(cc1)c2cc(c(c(n2)N)C#N)c3ccccc3 HTS13544 Cc1ccc(cc1S(=O)(=O)Nc2ccc3c(c2)OCC4N3CCC4)F SCR01119 c1ccc(cc1)OCC(=O)Nc2ccc3c(c2)OCC4N3CCC4 SCR01118 CC(C)(C)c1ccc(cc1)C(=O)N2CCCCCC2 S06993 c1cc(ccc1C2CC23C(=O)C4CCN3CC4)C(F)(F)F SCR01246 c1cc(oc1)c2cc(nc(c2C#N)N)c3cccs3 HTS13338 c1cc(sc1)c2nnc(s2)NC(=O)CN3CCOCC3 HTS13434 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4ccc(cc4)F)C HTS13310 CCOC(=O)Cc1csc(n1)NC(=O)c2cccs2 HTS13337 Cc1ccccc1N2CC(=O)Nc3c4c(cc(nc4oc3C2=O)c5ccccc5)C HTS13392 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3ccccc3)/s2 HTS13414 CCN(CC)c1ncc2c(n1)nc(nc2Nc3ccc(cc3)OC)SCC(=O)OCC HTS13297 COC(=O)c1c(ccs1)S(=O)(=O)NCc2ccc(cc2)S(=O)(=O)N SCR01160 Cc1c(c(n(n1)C)C)CNS(=O)(=O)c2ccc(nc2)N3CCOCC3 SCR01177 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc(nc3)N4CCOCC4 SCR01179 COc1cccc(c1)/C=c\2/c(=O)n3c4ccccc4nc3s2 HTS13426 c1cc(oc1)c2nnc(s2)N HTS13431 c1ccc2c(c1)c3csc(c3c(=O)o2)NC(=O)CN4CCOCC4 HTS13479 c1ccc(cc1)c2c(nc([nH]2)c3cccs3)c4ccccc4 HTS13439 COc1cc(ccc1O)c2[nH]c(c(n2)c3ccccc3)c4ccccc4 HTS13440 CN1CCN(CC1)CC(=O)Nc2c3c(cs2)c4ccccc4oc3=O HTS13477 c1cc(oc1)c2cc(nc(c2C#N)OCC(=O)c3ccc(cc3)F)c4cccs4 HTS13488 Cc1ccc(cc1)NC(=O)Nc2c3c(cs2)c4ccccc4oc3=O HTS13497 Cc1c(c2ccccc2o1)CNC(=O)Nc3ccc(cc3)Oc4ccc(cc4)Cl S07650 c1ccc(c(c1)c2[nH]c3ccccc3n2)/N=C\c4cc(cc(c4O)Cl)Cl S05441 c1ccc(cc1)N2CCN(CC2)CC(=O)Nc3nnc(s3)c4ccco4 HTS13435 CCOC(=O)Cn1c(c(nc1c2cccs2)c3ccccc3)c4ccccc4 HTS13436 C=CCn1c(c(nc1c2cccs2)c3ccccc3)c4ccccc4 HTS13438 CCOC(=O)C1=C(NC(=O)NC1c2ccco2)C HTS13450 Cc1cc(c(o1)C(F)(F)F)CNS(=O)(=O)c2ccc(nc2)N3CCOCC3 SCR01180 c1cc(ncc1S(=O)(=O)NCC2CCCO2)N3CCOCC3 SCR01178 c1cc(sc1)c2nc(cs2)CNS(=O)(=O)c3ccc(nc3)N4CCOCC4 SCR01176 c1cc(ncc1S(=O)(=O)NCc2cc(cc3c2OCOC3)F)N4CCOCC4 SCR01175 c1ccc(cc1)S(=O)(=O)n2cc(c3c2cccc3)C(=O)NCCc4ccccn4 SCR01261 Cc1c2cc(ccc2sc1S(=O)(=O)NCCc3ccccn3)Cl SCR01255 c1ccc(cc1)c2c(nc([nH]2)c3cccnc3)c4ccccc4 HTS13442 c1ccc(cc1)c2c(nc([nH]2)c3ccco3)c4ccccc4 HTS13444 c1ccc(cc1)/C=C\2/C(=O)NNC(=N2)c3ccccc3 HTS13459 COc1ccc(cc1)/C=C\2/C(=O)NNC(=N2)c3ccccc3 HTS13460 CN1CCOc2c1cc(cc2)S(=O)(=O)NC3CCCCNC3=O SCR01006 CCOC(=O)c1c(c(c([nH]1)C)S(=O)(=O)NC2CCCCNC2=O)C SCR01004 c1cc2c(cc1S(=O)(=O)NC3CCCCNC3=O)OCCCO2 SCR01002 c1ccc2c(c1)c(c[nH]2)C3CCN(CC3)CC(C(F)(F)F)O SCR00709 CCOC(=O)CN(c1ccccc1C)C(=O)COc2c(c(cc(n2)C)C)C#N HTS13451 CCOC(=O)CN(c1cccc(c1)C(F)(F)F)C(=O)COc2c(c(cc(n2)C)C)C#N HTS13452 c1ccc(cc1)c2nc(cs2)C(=O)Nc3ccc4c(c3)nccn4 SCR01276 c1ccc(cc1)c2csc(n2)NNC(=O)c3cccs3 HTS13464 c1cc2c(nc1)sc(n2)S RH00329 Cc1c(nn(n1)c2ccccc2)CNC(=O)COC SCR01445 Cc1c(nn(n1)c2ccccc2)CNC(=O)Cc3ccc(c(c3)OC)OC SCR01444 Cc1c(nn(n1)c2ccccc2)CNC(=O)CC(C)(C)C SCR01443 c1ccc2c(c1)c(cs2)C(=O)NCc3ccc4c(c3)CCO4 SCR01385 CCc1ccc(cc1)S(=O)(=O)NC2CCCCNC2=O SCR00998 c1ccc(cc1)CS(=O)(=O)NCc2csc(n2)c3cccs3 SCR01197 c1ccc(cc1)n2c3c(cn2)c(ncn3)N4CCCC4 HTS13277 c1ccc(cc1)/C=c\2/c(=O)n3c(nnc3s2)c4ccc(cc4)Cl HTS13278 c1cc(oc1)c2nnc3n2c(=O)/c(=C/c4ccc(cc4)F)/s3 HTS13279 c1ccc(cc1)c2nnc(o2)SCC(=O)NN3CC(=O)N(CC3=O)c4cccc(c4)Cl HTS13352 c1cc(ccc1c2[nH]c(nn2)SCC(=O)O)Cl HTS13294 CNC(=O)NC(=O)CSc1[nH]c(nn1)c2ccncc2 HTS13293 c1cc(sc1)c2ccc(s2)CNC(=O)c3ccc(nc3)N4CCOCC4 SCR01376 c1cc(ncc1C(=O)NCc2cc(cc3c2OCOC3)F)N4CCOCC4 SCR01373 c1ccc(c(c1)CSC(=N)N)Cl.Cl S01437 c1cnc(c(n1)C(=O)NN)N HAN00435 CC(C(=O)O)SCc1ccccc1 BTBG00017 Cc1c(nn(n1)c2ccccc2)CNC(=O)c3ccc(cc3)N(C)C SCR01439 CCOC(=O)c1c(c(c([nH]1)C)S(=O)(=O)NCc2c(nn(n2)c3ccccc3)C)C SCR01461 CC(=O)N[C@@H]1[C@H]([C@@H]([C@H](O[C@@H]1O)CO)O)O SB01966 CC(C)(C)OC(=O)N1CSC[C@H]1C(=O)O SB02065 CCOC(=O)c1c(c2c(cc(nc2s1)C)C)N RF00051 c1ccnc(c1)SC/C(=N/O)/N CD09642 c1ccc2c(c1)cc(c(n2)N)C#N SEW05329 c1ccc(cc1)COc2cccnc2N BTB08555 Cc1c(c2ccccc2o1)CNC(=O)Nc3ccc(cc3)C(C)(C)C S07653 Cc1c(cnn1c2ccccc2)S(=O)(=O)NCc3csc(n3)c4cccs4 SCR01210 c1ccc(cc1)c2[nH]c(nn2)SCC(=O)O HTS13295 c1cc(ccc1c2nnc(s2)N)Cl HTS13308 Cc1cc(nc2c1c3c(s2)C(=O)N(CC(=O)N3)c4ccc(cc4)F)C HTS13365 Cc1cc(nc2c1c3c(s2)C(=O)N(CC(=O)N3)c4ccccc4)C HTS13366 c1ccc2c(c1)N(c3ccccc3S2)Cc4nc([nH]n4)SCC(=O)N HTS13305 CC(=O)CSc1[nH]nc(n1)CN2c3ccccc3Sc4c2cccc4 HTS13306 COc1ccc(cc1)NC(=O)c2ccc(nc2)N3CCOCC3 SCR01360 c1cc(ccc1NC(=O)c2ccc(nc2)N3CCOCC3)n4cncn4 SCR01358 Cc1c(c(on1)C)NC(=O)N2CCN(CC2)c3ncccn3 SCR01470 Cn1c(nnc1S)c2ccncc2 ML00396 c1cc(ccc1Sc2ccc(cc2[N+](=O)[O-])C(=O)O)Cl BTB06747 c1ccc2c(c1)cc(s2)CNC(=O)c3ccc(nc3)N4CCOCC4 SCR01368 c1ccc(cc1)OCC(CN2CCNCC2)O BTB12336 CS(=O)(=O)c1ccc2c(c1)sc(n2)N XBX00319 c1cc(ccc1CNS(=O)(=O)c2ccc(c(c2)F)F)S(=O)(=O)N SCR01167 Cn1c(ccc1S(=O)(=O)NCc2ccc(cc2)S(=O)(=O)N)C(=O)OC SCR01166 c1ccc(cc1)S(=O)(=O)NCc2ccc(cc2)S(=O)(=O)N SCR01145 CCOC(=O)Cn1c(c(nc1c2ccco2)c3ccccc3)c4ccccc4 HTS13309 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4cccc(c4)C(F)(F)F)C HTS13311 CCOC(=O)CSc1nc2c(cnc(n2)N3CCOCC3)c(n1)Nc4ccccc4 HTS13381 CCOC(=O)c1ccccc1Nc2ccc(cc2C(=O)OCC)[N+](=O)[O-] S06221 Cc1cc(c(s1)C)S(=O)(=O)NCc2ccc(cc2)c3cccs3 SCR01419 c1cc(c(c(c1)Cl)C(=O)NC(=O)N2CCSCC2)Cl BTB04460 CC(=O)C1=CN=C(SC1)c2ccc(cc2)Cl BTB05406 COc1ccc(c(c1)CCC(=O)O)OC BTB02098 CCC(C)Sc1nnc(s1)S JFD03143 COC(=O)c1c(c(c(s1)SC)S(=O)(=O)c2ccc(cc2)Cl)N KM01163 c1cc(ncc1C(=O)N2CCN(CC2)c3c(cncc3Cl)Cl)N4CCOCC4 SCR01351 CCCCCCC#Cc1cc(cnc1)C(=O)O KM09448 c1cc(ccc1C#N)OCc2ccc3c(c2)non3 KM07235 c1ccc2c(c1)[nH]c(n2)SCC(=O)O DP01042 c1cc(ccc1COc2ccc(c(c2)Cl)Cl)C(=O)O S08027 c1cc2c(cc1CNS(=O)(=O)c3ccc(c(c3)F)F)CCO2 SCR01407 CN(C)c1ccc(cc1)C(=O)NCc2ccc3c(c2)CCO3 SCR01392 CC(C)C[C@@H](C(=O)OCc1ccc(cc1)CC(=O)O)NC(=O)OC(C)(C)C JFD01596 C/C(=N\OCc1ccc(cc1)Br)/c2ccc(c(c2)[N+](=O)[O-])Sc3ccccn3 JP00690 c1cc(cc(c1)Cl)NC(=O)NCc2csc(n2)c3cccs3 SCR01330 COc1ccc(cc1OC2CCCC2)NC(=O)NCc3csc(n3)c4cccs4 SCR01335 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)c2ccno2 SCR01320 c1cc(sc1)c2ccc(cc2)CNC(=O)C3CCC3 SCR01420 Cc1c(c(on1)C)NC(=O)NCc2csc(n2)c3cccs3 SCR01481 Cc1c(c(on1)C)NC(=O)NCc2cc(cc3c2OCOC3)F SCR01480 Cc1c(c(on1)C)NC(=O)NCc2ccc(cc2Cl)Cl SCR01479 Cc1c(c(on1)C)NC(=O)NCc2ccc3c(c2)OCO3 SCR01476 COc1ccccc1CC(=O)NCc2ccc3c(c2)CCO3 SCR01391 Cc1ccc(cc1C)C(=O)NCc2ccc3c(c2)CCO3 SCR01388 c1cc2c(cc1CNC(=O)C3CCC3)CCO2 SCR01387 CC(C)(C)c1cc(n(n1)C)C(=O)NCc2ccc3c(c2)CCO3 SCR01386 Cc1c(cnn1c2ccc(cc2)OC)NC(=O)Nc3ccc4c(c3)OCCCO4 HTS12356 CCOC(=O)c1c(c(sc1NC(=S)Nc2cc(ccn2)C)C)C HTS12977 CC(C)(C)OC(=O)N1CCN(CC1)c2ccc(cn2)NC(=O)c3ccc(cc3)OC HTS07825 c1cc2c(cc1C(=O)OCc3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)CCO2 HTS03027 c1ccc(cc1)n2c(c(cn2)C(=O)N/N=C/c3ccc(cc3)[N+](=O)[O-])N HTS07447 COc1cc2c(cc1OC)CN(CC2)C(=O)c3cccs3 SCR01096 c1ccc(cc1)n2c(c(cn2)C(=O)NC3CCCCNC3=O)C(F)(F)F SCR00986 c1ccc2c(c1)c3c([nH]2)C(NCC3)c4ccc(cc4)F.Cl SCR01193 CC1(C2CCC(C2)(C1N)C)C.Cl RH01534 c1ccc2c(c1)c(cs2)C(=N)N.Cl CC12331 c1ccc(c(c1)/C=N/CCCNC(=O)c2c(cccc2F)F)O CD03936 C=CCn1c(nnc1SCC(=O)Nc2ccc(cc2)S(=O)(=O)N)c3ccc(cc3)Cl HTS13506 CC1CCCN(C1)S(=O)(=O)c2ccc(nc2)N3CCOCC3 SCR01185 CN(Cc1ccccc1)S(=O)(=O)c2ccc(nc2)N3CCOCC3 SCR01184 c1cc(sc1)c2ccc(s2)CNS(=O)(=O)c3ccc(nc3)N4CCOCC4 SCR01183 c1cc2c(cc1CNS(=O)(=O)c3ccc(nc3)N4CCOCC4)OCO2 SCR01181 c1cc(oc1)CNC(=O)c2cc(cc3c2OCOC3)F SCR01509 c1ccc-2c(c1)Cc3c2ccc(c3)c4csc(n4)N JFD03223 Cc1c(c(n(n1)C)C)S(=O)(=O)NCc2ccc(cc2)c3cccs3 SCR01412 Cc1c(sc(n1)C)S(=O)(=O)NCc2ccc(cc2)c3cccs3 SCR01410 c1ccc(cc1)c2c(oc(n2)S)c3ccccc3 SB01351 c1cc(c2c(c1)OCCCO2)C(=O)NCc3csc(n3)c4cccs4 SCR01301 Cc1c(cc(o1)C(C)(C)C)C(=O)NCc2csc(n2)c3cccs3 SCR01315 c1cc(sc1)c2nc(cs2)CNC(=O)c3ccc(cc3Cl)F SCR01317 CCN(CC)CC(=O)Nc1ccc(cc1)S(=O)(=O)N HTS13516 c1cc(c(c(c1)Cl)C2=N/C(=C/c3ccc4c(c3)OCO4)/C(=O)O2)F S06427 COc1cccc(c1OC)c2cc(nc(c2C#N)O)c3ccc(cc3)F S06553 c1ccc2c(c1)nc(s2)C(=O)Nc3ccccc3N4CCOCC4 SCR01080 c1ccnc(c1)CCNS(=O)(=O)c2ccc(cc2)S(=O)(=O)N3CCCC3 SCR01254 c1ccnc(c1)CCNS(=O)(=O)c2ccc(cc2)S(=O)(=O)N3CCOCC3 SCR01253 c1ccnc(c1)CCNS(=O)(=O)c2ccc3c(c2)OCCCO3 SCR01250 c1ccnc(c1)CCNS(=O)(=O)c2cccc3c2nsn3 SCR01249 CC(CCC(=O)OC)[C@H]1CCC2[C@@]1([C@H](CC3C2[C@@H](CC4[C@@]3(CC[C@H](C4)O)C)O)O)C SB01788 Cc1c(c(n(n1)C)C)CNC(=O)c2ccc(nc2)N3CCOCC3 SCR01372 c1cc2c(cc1CNC(=O)c3ccc(nc3)N4CCOCC4)OCO2 SCR01371 Cc1cc(c(s1)C)S(=O)(=O)NCc2ccc3c(c2)CCO3 SCR01403 Cc1c(c(n(n1)C)C)S(=O)(=O)NCc2ccc3c(c2)CCO3 SCR01405 CN1CCOc2c1cc(cc2)S(=O)(=O)NCc3ccc(cc3)c4cccs4 SCR01411 c1cc(cc(c1)S(=O)(=O)NCc2csc(n2)c3cccs3)C(F)(F)F SCR01198 c1cc(sc1)c2nc(cs2)CNS(=O)(=O)c3ccc4c(c3)CCO4 SCR01200 c1ccnc(c1)c2ccc(s2)S(=O)(=O)NCc3csc(n3)c4cccs4 SCR01201 c1cc2cccnc2c(c1)S(=O)(=O)NCc3csc(n3)c4cccs4 SCR01203 CCn1c(nnc1SCC(=O)NN2CC(=O)N(CC2=O)c3ccc(cc3)F)c4cccs4 HTS13271 Cc1c(nn(n1)c2ccccc2)CNC(=O)COc3ccccc3 SCR01449 Cc1c(nn(n1)c2ccccc2)CNC(=O)c3c(ocn3)c4ccc(cc4)OC SCR01447 c1ccc(cc1)NC(=O)c2ccc(nc2)N3CCOCC3 SCR01356 CN(C)c1ccc(cc1)NC(=O)c2ccc(nc2)N3CCOCC3 SCR01355 Cc1c(c(on1)C)NC(=O)NC2Cc3ccccc3C2 SCR01487 c1ccc(cc1)Oc2ccc(cc2)N3C(SCC3=O)c4cccnc4 S07619 Cc1cc(c(s1)C)S(=O)(=O)NCc2csc(n2)c3cccs3 SCR01212 CC1(CCc2cc(ccc2O1)S(=O)(=O)NCc3csc(n3)c4cccs4)C SCR01213 c1cc(sc1)c2nc(cs2)CNS(=O)(=O)c3ccc(cc3)Cl SCR01216 c1cc(sc1)c2nc(cs2)CNS(=O)(=O)c3ccc(s3)c4ccno4 SCR01217 c1ccc(cc1)n2c(nnc2SCC(=O)Nc3nnc(s3)c4cccs4)c5ccco5 HTS13288 c1cc(c(cc1C(=O)O)[N+](=O)[O-])S(=O)(=O)c2cc(ccc2Cl)Cl BTB06762 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)N AW00805 Cc1c(cccc1Cl)SCC(=O)O BTB08831 c1ccc(cc1)OCc2ccc(cc2)C(=O)O CC63701 CS(=O)(=O)c1c(c(cs1)c2ccccc2)C#N KM02063 Cc1c(nn(n1)c2ccccc2)CNC(=O)c3c(ocn3)c4ccccc4 SCR01435 CC(C)(C(=O)N1CCC2(CC1)NC(=O)c3ccccc3O2)Oc4ccc(cc4)Cl SCR01382 CC(C)(C)c1ccc(cc1)c2nnnn2c3cc(ccc3Cl)Cl S07842 Cc1c(c(on1)C)NC(=O)Nc2cccc(c2)n3cccc3 SCR01490 Cc1c(sc(n1)c2cccs2)C(=O)C SPB02598 Cc1c(c2ccccc2o1)CNC(=O)Nc3ccc(cc3Cl)Cl S07666 COc1ccccc1NC(=O)c2cc3cc(ccc3cc2OC)Br S07696 COc1ccc(cc1)N2CCN(CC2)S(=O)(=O)c3ccc(nc3)N4CCOCC4 SCR01189 c1cc(ncc1S(=O)(=O)NCc2ccsc2)N3CCOCC3 SCR01182 CCOC(=O)CSc1[nH]nc(n1)CN2c3ccccc3Sc4c2cccc4 HTS13304 CSc1ccc(cc1c2cc[nH]n2)[N+](=O)[O-] KM03224 c1cc(sc1)C2N(C(=O)CS2)c3ccc(cc3F)F S07843 COc1ccc(c(c1)S(=O)(=O)NCc2ccc3c(c2)CCO3)OC SCR01404 c1cc(cnc1)c2c(c[nH]c(=O)n2)C(=O)O MO00826 Cc1ccc(n1c2c(ccs2)C(=O)NN)C GK02967 c1cc(ncc1C(F)(F)F)OCC#N HAN00271 c1ccc2c(c1)C=C(CO2)C(=O)NCc3ccc4c(c3)CCO4 SCR01384 c1ccc(cc1)n2c(c(cn2)C(=O)NCc3ccc(cc3)c4cccs4)C(F)(F)F SCR01431 CC(C)(C)c1cc(n(n1)C)C(=O)NCc2ccc(cc2)c3cccs3 SCR01429 c1cc(ccc1NC(=O)CN2CCOCC2)S(=O)(=O)N HTS13335 CN1CCc2c(sc3c2c(nc(n3)SCc4ccc(cc4)Cl)NCC=C)C1 HTS13336 c1ccc(cc1)N2CC(=O)N(CC2=O)NC(=O)CSc3nnc(o3)c4ccc(cc4)Cl HTS13351 CCN(CC)c1ncc2c(n1)nc(nc2NCc3ccccc3)SCc4ccccc4 HTS13382 c1cc(sc1)c2nnc(s2)N HTS13430 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3ccc(nc3)N4CCOCC4 SCR01455 c1csc2c1sc(c2)C(=O)O SEW01931 c1cc(sc1)c2ccc(cc2)CNS(=O)(=O)c3cccs3 SCR01415 Cc1nc(cn1C)S(=O)(=O)NCc2ccc(cc2)c3cccs3 SCR01414 c1cc(sc1)c2ccc(cc2)CNS(=O)(=O)c3ccc(nc3)N4CCOCC4 SCR01413 c1ccn(c1)c2ccc(cc2)F CD02331 CNc1ccc(cc1C(=O)NN)Cl DP01825 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN CD01867 Cc1c(sc(n1)c2cnccn2)C(=O)N3CCc4cc(c(cc4C3)OC)OC SCR01098 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)Nc3ccc(cc3)C(=O)N SCR00962 COc1cc2c(cc1OC)CN(CC2)C(=O)COc3ccccc3 SCR01092 c1ccc2c(c1)cccc2CC(=O)NCc3csc(n3)c4cccs4 SCR01312 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)S(=O)(=O)c4ccc(nc4)N5CCOCC5 SCR01186 Cc1c2cc(sc2n(n1)C)C(=O)NCCc3ccccn3 SCR01264 Cc1c(sc(n1)c2cnccn2)C(=O)NCCc3ccccn3 SCR01263 CN(C)c1cccc2c1cccc2S(=O)(=O)NCCc3ccccn3 SCR01247 Cc1c(c(on1)C)NC(=O)NCCN2CCOCC2 SCR01475 Cc1c(c(on1)C)NC(=O)N2CCN(CC2)c3ccc(cc3)OC SCR01472 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3cc(ccc3OC)OC SCR01465 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3cccc4c3cccc4 SCR01464 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3c(c(cs3)C(=O)OC)OC SCR01463 C1Cc2c(sc3c2c(nc(n3)SCC(=O)N)SCC(=O)N)C1 HTS13501 Cc1cccc(c1)NC(=O)/C=C/C(=O)O S07160 c1cc(cnc1)C2N(C(=O)CS2)c3ccc(cc3F)I S07756 c1cc(ncc1S(=O)(=O)NC2CCCCC2)N3CCOCC3 SCR01171 c1ccc(cc1)n2c3c(cn2)c(ncn3)N4CCCCC4 HTS13276 COc1ccc(cc1)COc2ccc(cc2)CC#N BTB07334 CSc1nc2ncc(c(n2n1)N)C(=O)O BTB08394 c1cc(ccc1n2c(c(cn2)C#N)N)Cl BTB07485 c1ccc2c(c1)c(c(s2)Cl)CC(=O)O MWP00105 c1cnc(nc1C(F)(F)F)N2CCCNCC2 AW00488 c1cc(ccc1c2csc(n2)CC#N)F CD02890 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3c(nn(c3C)C)C SCR01454 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3c(nc(s3)C)C SCR01452 c1ccc(c(c1)NC(=O)c2ccc(nc2)N3CCOCC3)N4CCOCC4 SCR01357 COC(=O)c1c(c(cs1)C#N)N KM00977 CC(C)(C)S(=O)(=O)CC#N KM01834 CC(C)(C)S(=O)(=O)c1cnc(nc1N)N KM02686 CC(C)n1cc(c(=O)n(c1=O)Cc2ccccc2)C#N KM07738 COc1cccc(c1C#N)OCc2ccccc2Cl MWP00988 c1ccc(cc1)c2nc(sn2)N3CCNCC3 HAN00371 c1c(c(nc(n1)N2CCOCC2)N)C#N HTS12516 c1c(cncc1Br)C(=O)NN RDP00027 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4ccc(nc4)N5CCOCC5 SCR01348 Cc1c(nn(n1)c2ccccc2)CNC(=O)C3CCC3 SCR01432 Cc1c2cc(sc2n(n1)C)C(=O)NCc3c(nn(n3)c4ccccc4)C SCR01434 c1cc(sc1)c2ccc(cc2)CNS(=O)(=O)c3ccc4c(c3)OCCCO4 SCR01416 Cc1ccc(cc1NC(=O)c2c(onc2c3ccccc3Cl)C)NC(=O)C BTB01571 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)c4ccccc4 SPB05191 COc1ccc2c(c1)c(ccn2)[C@H]([C@@H]3C[C@@H]4CCN3C[C@@H]4C=C)O.Cl SB01805 c1cc(c(cc1Cl)Cl)OCC#N SPB00370 COc1ccc(cc1C#N)C(=O)OC TL00306 c1cc(ccc1C2SCCS2)C(=S)N RF02581 c1cncc(c1C(F)(F)F)N RF03857 C1CCC(CC1)c2c(c(=O)[nH]c(=S)[nH]2)C#N RH00269 Cc1cc(c2ccccc2n1)N3CCNCC3 RH02136 CCOC(=O)/C(=C/Nc1ccccc1Cl)/C#N RH02178 CCc1cccc(c1N2C(=O)C=CC2=O)CC S02113 c1ccc(cc1)c2nc(cs2)CC(=O)O RH01225 CC1=CCC(C(C1)C(=O)Nc2cc(cc(c2)Cl)Cl)C(=O)O S07818 CC(C)(C)c1ccc(cc1)c2nnnn2c3ccc(cc3Cl)Cl S07839 c1cc(ccc1CC(=O)O)F RH01845 Cc1c(c(on1)C)NC(=O)NCc2cc3ccccc3s2 SCR01482 Cc1c(c(on1)C)NC(=O)NC2CCCc3c2cccc3 SCR01486 CC(=O)N[C@@H]1[C@H]([C@H]2[C@@H](COC(O2)c3ccccc3)O[C@@H]1OCc4ccccc4)O RH01184 c1ccc2c(c1)c(=O)c(cs2)Cc3ccc(c(c3)Cl)Cl BTB14855 COc1ccc(cc1)c2cc[nH]n2 SEW03385 COC(=O)C/C(=N\NC(=O)CCc1nc(no1)c2ccc(cc2)Cl)/C(=O)OC BTB03642 Cn1c(nnc1SCC(=O)Nc2cccc(c2)C(F)(F)F)SCC(=O)Nc3cccc(c3)C(F)(F)F BTB08558 Cc1ccc(cc1)C(=O)OCCN2C(=O)c3cccc4c3c(ccc4)C2=O BTB14689 Cc1c(c(on1)C)S(=O)(=O)NCc2ccc3c(c2)CCO3 SCR01401 CCc1ccc(cc1)S(=O)(=O)NCc2ccc3c(c2)CCO3 SCR01400 CC1(C2CCC1(c3c2c(nc(n3)N)C(F)(F)F)C)C BTB14926 CC(=O)OCc1ccccc1Sc2ccccc2C(=O)Nc3ccc(cc3)OC BTB14928 c1cc2cccc(c2c(c1)I)I BTB14941 c1ccc(cc1)C(=O)C(NC(=O)c2ccccc2)n3cnccc3=O BTB14948 c1cc(ccc1CC(N2CCN(CC2)c3nc4ccc(cc4s3)Cl)O)[N+](=O)[O-] AW00626 c1cc(ccc1OCC(CN2CCN(CC2)c3nc4ccc(cc4s3)Cl)O)OC(F)(F)F AW00627 c1ccc(cc1)C(CN2CCN(CC2)c3nc4ccc(cc4s3)Cl)O AW00646 c1cc(c(c(c1)Cl)Cl)NC(=O)N2CCCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F AW00663 Cc1ccc(cc1NS(=O)(=O)c2ccc3c(c2)c(=O)sn3C)C(=O)OC BTB03648 c1ccc(cc1)C(=O)CSCC(=O)c2ccccc2 BTB03675 Cc1ccc(cc1)C(=O)CSCC(=O)c2ccc(cc2)C BTB03681 c1c2c(cc(c1Cl)F)nc[nH]2 BTB03697 CNC(=S)N(C)/N=C/c1cc(cc(c1O)Cl)Cl BTB03833 CC(C)(C)SC(=S)SCC(=O)c1ccc(cc1)[N+](=O)[O-] BTB03855 c1cc(ccc1NC(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl BTB08628 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NS(=O)(=O)c3ccc(cc3)C)C BTB08641 COc1ccc(c(c1)CNC(=O)Cc2cccs2)OC BTB08690 Cc1ccc(cc1)Sc2c(cccn2)C3=N/C(=C\c4ccc(cc4)C(F)(F)F)/C(=O)O3 BTB08788 c1ccc2c(c1)C(=O)N(C2=O)CCC(=O)Nc3ccccc3C(F)(F)F BTB14781 CN1C2C[C@@H](CC1CC2)NC(=O)CSc3ccccc3 BTB14824 CN1C2C[C@@H](CC1CC2)NC(=O)CSCc3ccc(cc3)OC BTB14830 c1ccc(cc1)c2c(c(=O)c3ccccc3o2)OS(=O)(=O)c4ccc(cc4)Br BTB14844 CC12CC3CC(C1)(CC(C3)(C2)C(=O)NN)C BTB14963 Cc1c(cn(n1)c2ccccc2)/C=N/n3c(nnc3SCC(=O)c4ccccc4)c5ccncc5 HTS11982 c1ccc(c(c1)NC(=O)Nc2ccccc2F)N3CCCCC3 HTS08439 Cc1nc2c(cnn2c3ccccc3)c(=O)n1/N=C/c4ccc5c(c4)OCO5 HTS07452 c1cc(sc1)CC(=O)NCc2ccc(o2)c3ccc(cc3F)F BTB08691 CCOC(=O)C(=CNc1cc(no1)C)C(=O)OCC BTB08700 COc1ccc(c(c1)Sc2c(cccn2)C(=O)NCC(=O)OC)OC BTB08749 Cc1cc(n2cnnc2n1)O BTB08753 CC(C)(C)OC(=O)NC(Cc1c[nH]c2c1cccc2)C(=O)OC BTB15190 Cc1ccc(c2c1C(=O)c3ccccc3C2=O)C BTB15203 CCCOc1cccc(c1)C2CCCCN(C2=O)C BTB15234 C1CCC(C(C1)C(=O)N)C(=O)O BTBG00083 C1C2CC3(CC1CC(C2)(C3)Br)Br BTBG00087 CC(C)(CC(=O)O)C(CCC(=O)O)C(=O)O BTBG00152 c1cc(c(cc1OCC(CN2CCC(CC2)O)O)Cl)Cl AW00664 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccc(nc3)Oc4ccc(cc4)Cl BTB03883 c1cc(c(c(c1)Cl)Oc2ccc(cc2)[N+](=O)[O-])Cl BTB03902 CN\1C(=O)CS/C1=N/N=C/c2cn(nc2c3ccccc3)c4ccccc4 HTS09979 Cc1ccc(cc1)S(=O)(=O)N(CC=C)c2ccccc2C3=N/C(=C\c4cccc(c4)C)/C(=O)O3 BTB08802 CN(c1cnn(c(=O)c1Cl)c2ccc(c(c2)Cl)F)NC(=O)c3ccc(cc3)Cl BTB08819 Cc1cc(n2c(n1)nc(n2)S(=O)(=O)C)OC BTB08884 CC(C)(C)OC(=O)C(C)(C)Sc1ccc(cn1)C(F)(F)F BTB08902 C=CCNC(=O)NC(=O)C12CC3CC(C1)CC(C3)C2 BTB15003 C1CC2CCCC(C1)(C2)C(=O)N BTB15008 C/C(=N\O)/CC12CC3CC(C1)CC(C3)C2 BTB15013 CC12CC3(CC(C1)(CC(C2)(C3)CO)C)C BTB15026 c1cc(c(c2c1[nH]cc2O[C@H]3[C@@H]([C@H]([C@H]([C@H](O3)CO)O)O)O)Cl)Br BTB15126 CN(CCC#N)c1ccc(cc1)/C=N/NC(=O)C2CCN(CC2)C(=S)NC3CC4CC3C=C4 CD02150 CCOC(=O)c1cc(on1)c2csc(n2)N/N=C/c3c(cccc3Cl)Cl SPB04524 Cc1nc(c(o1)C(F)(F)F)C(=O)NNC(=O)c2ccc(cc2)Cl RF04208 Cc1ccc(cc1)S(=O)(=O)N(CC=C)c2ccccc2C(=O)NCC(=O)O BTB08766 Cc1ccc(cc1)Oc2c(cccn2)C3=N/C(=C\c4ccc(cc4)C(F)(F)F)/C(=O)O3 BTB08782 CC(C)(C)OC(=O)C(C)(C)S(=O)(=O)c1ccccn1 BTB08908 CSc1c(c(nc(n1)c2ccccc2)Sc3cccc(c3)C(F)(F)F)C#N BTB08926 CSc1c(c(nc(n1)c2ccccc2)Sc3ccc(cc3Cl)Cl)C#N BTB08927 CSc1ncc(c(n1)C(=O)O)Br RH00785 COC(=O)/C=C/1\C(=O)NCC(CN1)O PD00242 COC(=O)c1cccc(c1)NC(=S)NC(=O)c2cc(sc2Cl)Cl DFP00290 c1ccc(cc1)n2cc(c(n2)c3cccs3)/C=N/n4c(n[nH]c4=S)c5ccncc5 HTS11975 c1cc2cccc(c2c(c1)CO)I NRB00699 CSc1c(c(c(s1)C(=O)O)c2cccc(c2)Cl)C#N KM02576 CC(C)(C)S(=O)(=O)c1cnc(nc1N)N2CCCCC2 KM02675 CC1(C=Cc2cc(ccc2O1)C#N)C KM06599 CN1CC2C(N(N=C2/C(=C/c3ccccc3Cl)/C1)C)c4ccccc4Cl.Cl.Cl S07782 Cc1ccc(cc1)S(=O)(=O)N2CCCCCC2 BTB08940 c1cc(cc(c1)Cl)C(=O)OCCS(=O)(=O)c2ccc(cn2)Cl BTB08983 Cc1c2c(onc2c(=O)[nH]n1)/C=C/c3ccsc3 BTB08998 c1ccc(cc1)c2cc(c(o2)N)C#N AW01254 c1c2cc(c(=O)oc2c(cc1Cl)Cl)C(=O)O BTB01254 c1cc2c(cc1C(F)(F)F)nc([nH]2)CCCO BTB05684 Cc1c(cc(cc1Cl)[N+](=O)[O-])Cl KM08058 c1cc2c(cc1C(F)(F)F)c(cc(n2)C(F)(F)F)O KM09514 c1cc(sc1)S(=O)(=O)CC(=S)N KM03009 CSC(=C(C#N)C#N)SC CD00793 c1ccc(cc1)c2ccccc2NC(=O)NCc3csc(n3)c4cccs4 SCR01331 c1c(cnc(c1[N+](=O)[O-])O)Br SPB06123 c1cc(cc(c1)C(F)(F)F)CSc2nnc(s2)S TL00206 CCOC(=O)c1c(n(c(c1CNC(=O)c2ccc(nc2)N3CCOCC3)C)C4CC4)C SCR01377 Cc1ccccc1n2c(c(cn2)C(=O)O)C MO00434 c1ccc2c(c1)c(c[nH]2)OS(=O)(=O)[O-].[K+] AC33706 Cc1c(cc(c(n1)O)C#N)C(=O)C BTB09128 C1CCN2CCC[C@H]([C@H]2C1)CO BTB15228 c1cc(ccc1c2csc(n2)CC#N)Cl CD02848 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3ccc(s3)c4ccno4 SCR01457 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3cn(c(n3)C)C SCR01456 c1cc(ncc1C(=O)NCc2ccsc2)N3CCOCC3 SCR01367 COc1ccc(cc1)C(=O)NCc2ccc(cc2)c3cccs3 SCR01426 Cc1c(nn(n1)c2ccccc2)CNC(=O)C3=Cc4ccccc4OC3 SCR01433 Cc1c(nn(n1)c2ccccc2)CNC(=O)c3cccs3 SCR01440 COc1ccc(cc1)C(=O)NCc2csc(n2)c3cccs3 SCR01297 c1cc(ccc1NC(=O)c2ccc(nc2)N3CCOCC3)F SCR01361 c1cc(sc1)c2nc(cs2)CNC(=O)Nc3ccc4c(c3)OCCCO4 SCR01333 c1cc(ncc1C(=O)N2CCCC2)N3CCOCC3 SCR01346 CC(C)[C@@H](C(=O)O)NC(=O)OCc1ccccc1 SB02029 COc1ccccc1N2CCN(CC2)C(=O)c3ccc(cc3)N RH01624 CC(=O)c1csc(n1)CS(=O)(=O)c2ccccn2 SPB03551 Cc1c(c(no1)c2ccccc2)c3ccn[nH]3 SPB04970 Cc1nc(cs1)c2nc(cs2)C(=O)C SPB03623 Cn1c2ccc(cc2[nH]c1=S)C(F)(F)F TG00013 Cc1c(nn(n1)c2ccccc2)CNC(=O)c3c(nc(s3)c4ccc(cc4)C(F)(F)F)C SCR01442 Cc1cc(c(s1)C)S(=O)(=O)NCc2c(nn(n2)c3ccccc3)C SCR01466 Cn1c(cnc1S)c2ccc(cc2)Cl TG00105 c1ccc(cc1)C(C#N)N2CCOCC2 XBX00113 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)n2cccc2 BTB05942 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)NN BTB05972 c1cc(ccc1/C=C(\C#N)/C(=S)N)O CD02967 c1cc(cnc1)C2N(C(=O)CS2)c3c(cc(cc3F)F)F S07871 COc1ccc(cc1)C(=O)NCc2ccc3c(c2)CCO3 SCR01390 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)CS(=O)(=O)C SCR01462 c1ccc(cc1)N2CC(=O)N(CC2=O)NC(=O)CN3CCOCC3 HTS13273 COc1ccc(cc1)C(CN2CCOCC2)c3c(=O)n(nc(n3)c4ccccc4)CN5CCOCC5 HTS13347 CS(=NC(=S)NC(=O)Oc1ccccc1)(=O)c2ccc(cc2)Cl KM04270 Cc1cc(c(cc1C)/N=C\2/NC(C(=C)S2)(C)C)C BTB01404 Cc1cc2c(cc1C)CSC(SC2)(C)c3ccccc3 BTB01438 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2NS(=O)(=O)c3cccc(c3)C(F)(F)F)C BTB01468 c1ccc(cc1)N(Cc2c(cccc2Cl)F)NC(=O)NC(=O)c3ccccc3F BTB06013 Cc1cc(c2cc(ccc2n1)F)Oc3nc4c(s3)cc(cc4Cl)Cl BTB06089 Cc1nc(nc(n1)OC)N/C=N/O BTB06125 c1cc2c(cc1Cl)nc3n(c2=O)c4cc(ccc4s3)Cl BTB06127 Cc1cc(c(cc1Cl)Cl)Sc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] BTB06237 c1ccc(cc1)c2c(c(c(n(c2=O)c3ccccc3)c4ccccc4)Br)O BTB11806 c1ccc(cc1)c2c(c3ccc(cc3[nH]c2=O)F)O BTB11816 CCn1c2ccc(cc2c3c1ccc(c3)Cl)Cl BTB11851 CC(C)CCn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br BTB11856 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])C(=O)N BTB11884 CCCN(CCC)CC(Cn1c2ccc(cc2c3c1c(cc(c3)Br)Br)Br)O BTB12234 COc1ccc(cc1)C(CC(=O)N)CC(=O)O CD02971 CS/C(=N\S(=O)(=O)c1ccccc1)/N2CCCC2 CD03052 c1cc(cnc1)/C=N/NC(=S)NC2CC3CC2C=C3 CD03332 CC1(O[C@@H]2[C@H]([C@H](O[C@@H]2O1)C(CO)O)O)C BTB11978 Cc1ccc(cc1)NC(=O)CCC(=O)O BTB12145 Cc1ccc(cc1)NC(=O)CCC(=O)OC BTB12146 Cc1c(c(=O)n(n1C)c2ccccc2)NS(=O)(=O)c3ccc(cc3)NC(=O)C BTB12150 CCCCN(CCCC)CC(Cn1c2ccc(cc2c3c1ccc(c3)Br)Br)O BTB12227 c1ccc2c(c1)cc(c(=O)o2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB01485 c1ccc(c(c1)/C=C\2/C(=O)NC(=S)S2)Cl BTB01515 Cc1ccc(c(c1)C(=O)N/N=C/c2cc(c(c(c2)OC)OC)OC)[N+](=O)[O-] BTB01689 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)c2ccc(cn2)[N+](=O)[O-] BTB06254 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)c2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB06263 Cc1ccc(c(c1)C(C)Sc2c(cccn2)C(=O)O)C BTB06325 CCSc1c(cccn1)C(=O)N BTB06390 c1cc2c(cc1Cl)c3cc(ccc3n2CC(CN4CCCCC4)O)Cl BTB12253 COc1ccc(cc1OC)c2c3ccc(cc3c(=O)n(c2N)Cc4ccccc4)[N+](=O)[O-] BTB12298 CC(C)(C)c1ccc(=O)[nH]n1 BTB12376 c1ccc(cc1)C(CO)(CO)[N+](=O)[O-] BTB12380 CCCCN(CCCC)CC(Cn1c2ccccc2c3c1cccc3)O BTB12243 COC(=O)C1(C2C3C4CC5C3C1C6C5C4C62)C(=O)OC BTB12410 CCCCOC(=O)c1cccc2c1-c3ccccc3C2=O BTB12458 CCOC(=O)CCCSc1nnc(s1)S BTB12607 Cc1c(c(no1)c2ccccc2)NC(=O)N(CCC#N)Cc3cccs3 HTS06092 c1cc2c(cc1F)cc([nH]2)C(=O)O RH01182 CSc1nc(nc(n1)N2CCCC2)N RF02733 Cc1c(c2c(cc1Br)nsn2)C RDP00093 COC(=O)c1ccc(o1)CSc2ccc(cn2)C(F)(F)F KM06162 c1ccc(cc1)c2nc(sn2)N3CCCNCC3 AW00426 Cc1c(c(on1)C)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F SEW05939 c1cc(ccc1CO)OCCCCC(=O)O MO01083 Cc1cc(=O)n2ccccc2n1 BTB12654 c1cc2c(cc1S(=O)(=O)N3CCCN(CC3)c4c(cncc4Cl)Cl)CCO2 HTS04999 c1ccc(cc1)NC(=O)Nc2ccc(cc2)C#N HTS05107 c1cc(ccc1C#N)NC(=O)CCCC(=O)O HTS05120 Cn1c2c(c3c(cc4ccccc4n3)c(=O)n2c5ccccc5)c(=O)n(c1=O)C BTB13070 c1cc-2c(cc1[N+](=O)[O-])C(=C(C#N)C#N)c3c2c(cc(c3)[N+](=O)[O-])C(=O)N4CCCCC4 BTB13127 c1ccc2c(c1)-c3ccccc3C2=NO BTB13141 c1cc(c(c(c1)Cl)C(C#N)N2CCSCC2)Cl CD08301 C(C#N)Sc1nc(sn1)SCC#N CD08311 c1cc(c(c(c1)F)C#N)NCCc2ccc(cc2)Cl CD08314 CCOC(=O)c1c(c(sc1N2C(=O)CCC2=O)C)c3ccccc3 AW01012 COc1ccc(cc1)C(=O)CC2(c3cc(ccc3N(C2=O)CN4CCCCC4)Br)O BTB02036 Cc1ccc(c(c1)C(=O)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)[N+](=O)[O-] BTB02224 c1ccc2c(c1)C(=O)NC(N2)C3CCC=CC3 BTB02264 c1ccc(cc1)n2c(c3c(n2)cc(nc3O)O)N BTB02276 C#Cc1cccc(c1)NC(=O)NC(=O)c2ccccc2Cl BTB04456 c1ccc(cc1)S(=O)(=O)c2ccc(c(c2)OS(=O)(=O)c3cc(cc(c3)Cl)Cl)[N+](=O)[O-] BTB06577 CC(C)NC(=O)/C(=C/N(C)C)/C#N BTB06620 Cc1ccc(cc1)CNC(=O)c2cccnc2Sc3cccc(c3)Cl BTB06631 COc1cccc(c1)c2nnc(o2)c3ccccc3NC(=O)c4ccc(cc4)C(F)(F)F BTB06979 CCC(=NOc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])CC BTB12759 CC1(CC(c2cccc3c2c1ccc3)(C)c4cccc5c4cccc5)C BTB12803 c1cc(c(cc1N)S(=O)(=O)O)/C=C/c2ccc(cc2S(=O)(=O)O)N BTB12832 C(C(C(F)(F)F)C(F)(F)F)(C(=O)O)N BTB12858 C/C(=C/C(=O)O)/C=C/c1cccnc1.Cl BTB12916 CCOC(=O)c1cnc(nc1c2ccccc2)c3ccc(cc3)Cl CD08047 c1ccc(c(c1)C(=O)Nc2ccc(c(c2Cl)Cl)Cl)F CD08067 Cc1c(c(c(c(c1C)C)S(=O)(=O)Oc2cc(cc(c2)Cl)Cl)C)C CD08082 c1cc(oc1)c2cc(c(c(n2)O)C#N)c3cccs3 HTS10305 CCNC(=N)SCc1c(c(c(c(c1C)C)C)C)C.Cl CD00213 c1cc(cc(c1)NC(=O)CC#N)C(F)(F)F CD00242 c1cc(cc(c1)O)C=C2C(=O)NC(=O)NC2=O CD00397 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C(F)(F)F)NC(=O)c2cccc(c2)Cl BTB13214 c1ccc(cc1)C(=O)CC2(c3ccccc3NC2=O)O BTB13298 c1ccc(cc1)CNS(=O)(=O)c2ccc-3c(c2)C(=O)c4c3ccc(c4)S(=O)(=O)NCc5ccccc5 BTB13354 c1cc(ccc1C#N)S(=O)(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00993 COc1ccccc1NC(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F AW01017 c1ccc2c(c1)c(=O)oc(n2)c3cccs3 BTB02495 c1ccc(c(c1)C(=O)Nc2ccc(cc2)F)NC(=O)c3ccco3 BTB02496 COc1ccccc1NC(=O)CS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02516 C/C(=N\NC1=NCCCN1)/c2ccc(cc2)Cl BTB02527 COc1cccc(c1)c2nnc(o2)c3ccccc3NS(=O)(=O)c4cc(cc(c4)Cl)Cl BTB06982 Cc1ccc(=O)n(n1)Cc2ccc(cc2)Cl BTB06985 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CSc4ccc(cn4)C(F)(F)F BTB09507 c1cc(c(cc1COc2ccc(cc2[N+](=O)[O-])C3SCCS3)Cl)Cl BTB09610 c1cc(cnc1)Oc2ccc(cn2)NC=C(C#N)C#N BTB07238 COc1cc(ccc1O)/C=C\2/C(=O)NC(=O)N2 BTBS00035 c1ccc(cc1)NC(=O)c2cccc-3c2C(=O)c4c3cccc4 BTB13175 c1ccc(cc1)OS(=O)(=O)c2cc3c(c(c2)[N+](=O)[O-])-c4c(cc(cc4[N+](=O)[O-])S(=O)(=O)Oc5ccccc5)C3=NO BTB13184 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C(F)(F)F)NC(=O)OCC BTB13205 C#CC1(CCCCC1)NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 CD00598 COc1ccc(cc1/C=C/2\c3ccccc3NC2=O)Br CD00744 COc1ccc(cc1OC)/C=C/2\c3ccccc3NC2=O CD00745 COc1ccc(cc1Br)/C=C/2\c3ccccc3NC2=O CD00753 Cc1ccc(cc1)NS(=O)(=O)c2ccc-3c(c2)Cc4c3ccc(c4)S(=O)(=O)Nc5ccc(cc5)C BTB13629 c1ccc(cc1)N2C(CC(=N2)c3ccc4ccccc4c3)c5ccc6c(c5)OCO6 BTB13683 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01155 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCN(CC4)c5nccc(n5)C(F)(F)F AW01161 Cc1ccc(c(c1)C)NC(=S)/N=C/N(C)C BTB04780 CCOC(=O)/C(=C/Nc1nc2ccc(cc2s1)F)/C#N BTB04813 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02670 c1ccc2c(c1)c(c(s2)C(=O)Nc3cccc(c3)C#N)Cl BTB02755 c1ccc(c(c1)C(=O)c2ccc(c(c2)[N+](=O)[O-])N)C(=O)O BTB02773 Cc1cccc(c1NC(=O)CSC(C)C(=O)OC)C BTB02790 C/C(=N\OC(=O)c1ccc(cc1)C(F)(F)F)/c2ccc[nH]2 BTB07256 Cc1ccc(nn1)n2c(cc(n2)C)C BTB07293 CCOC(=O)c1cc(=O)c2c(ccc(c2o1)C(C)(C)C)OCc3ccccc3 BTB10111 CCCc1c(ccc2c1OC(CC2=O)(C)CCC(=O)OC)O BTB10119 Cc1cccc(c1C(=O)NC(=O)Nc2c(cc(cc2F)F)F)C BTB07480 CC(C)(C)c1ccc(c(c1)Cl)Oc2ccc(cn2)[N+](=O)[O-] BTB07489 c1cc(c(c(c1)Cl)C=C2C(=O)NC(=S)NC2=O)Cl CD00610 c1cc(c(cc1[N+](=O)[O-])S(=O)(=O)[O-])/C=C/c2ccc(cc2S(=O)(=O)[O-])[N+](=O)[O-].[Na+].[Na+] BTB13476 CN1c2ccccc2C(=O)C(C1=O)(Cl)Cl BTB13502 CC(=O)NC(CC(=O)N)C(=O)O BTB13545 CCC(C)[C@@H](C(=O)O)NC(=O)C BTB13548 CC(C)CC(C(=O)O)NC(=O)C(C)N BTB13577 COc1ccc(cc1OC)CC/N=C/c2ccccn2 CD00925 CC(C)(C)NS(=O)(=O)c1ccc(c(c1)Cl)N2C(=O)CC3(C2=O)CCCC3 AW01062 c1cc(c(cc1S(=O)(=O)NCC2CC2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01063 c1cc(cc(c1)C(F)(F)F)C(=O)ON=C2CCC3(CC2)OCCO3 BTB13759 CCOc1ccc2c(c1)nc([nH]2)SCc3c(c(c(c(c3F)F)F)F)F BTB13802 COc1cc(cc(c1OC)OC)C2Nc3ccccc3S2 CD01595 c1cc(c(cc1/C=N/N=C(N)N)Cl)O BTB13987 CCN1C(=O)/C(=C\c2ccc(c(c2)Cl)OCc3ccc(cc3)F)/SC1=S BTB14000 COc1ccc2c(c1)cc([nH]2)C(=O)O BTB14051 CCCCCc1ccc(cc1)C(=O)NCc2cccs2 BR00008 Cc1cc(cc(c1Cl)C)Oc2ccc(cc2NC(=O)C(Cl)(Cl)Cl)C(F)(F)F BTB02831 c1cc(cc(c1)NC(=O)c2ccncc2)C#N BTB02864 c1cc(sc1)c2nnc(n2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Sc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB03041 c1ccc(cc1)Oc2c(cccn2)C(=O)NNC(=S)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F BTB03068 COC(=O)/C=C(/C(=O)OC)\O/N=C(/c1ccc(cc1)Cl)\N BTB05315 CC(C)(C)c1ccc(c(c1)Cl)Oc2c(cccn2)[N+](=O)[O-] BTB07491 CCCn1c(nnc1SC)SC.I BTB07525 Cc1c(c(no1)c2ccccc2Cl)C(=O)NN BTB07542 CSc1nnc(n1CCNC(=O)c2c(cccc2Cl)Cl)SC BTB07548 c1ccc2c(c1)-c3ccc(cc3C2=O)Br BTB10475 Cc1ccc(cc1)C(=O)OCCS(=O)(=O)c2ccc(cn2)C(F)(F)F BTB07936 CCOc1ccc(cc1)/C=C/2\c3ccccc3NC2=O CD01001 CC(CCC(=O)OC1CC2CC=CC1C2)C3CCC4C3(CCC5C4CC=C6C5(CCC(C6)O)C)C BTB13785 c1cc(ccc1CO)C(=O)O BTB13819 Cc1ccc(cc1)NC(CC(=O)C2CC2)c3ccccc3 BTB13847 c1ccc(cc1)n2cc(cn2)C(=O)c3ccccc3O BTB13941 COc1cccc(c1)CC(=O)NC2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW01184 CC1(OC(C(O1)C(c2ccccc2)(c3ccccc3)O)C(c4ccccc4)(c5ccccc5)O)C BTB14055 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=O)c2c(c3ccccc3s2)Cl CD01984 c1cc(cc(c1)Cl)C(C(=O)O)O BTB14381 c1ccc2c(c1)c3ccc4c(c3[nH]2)non4 BTB14394 c1ccc(cc1)C(=O)c2ccc3ccccc3n2 BTB14404 CCNC(=Nc1ccc(cc1)Cl)NCC BTB14420 CN(C)c1ccc(c(c1)Cl)/C=N/NC(=O)c2ccncc2 BTB00392 Cc1cc2c(cc1C)CSC(SC2)c3ccccc3 BTB00415 Cc1cc2c(cc1C)CSC(SC2)c3ccc(cc3Cl)N(C)C BTB00422 c1c(cc(cc1C(F)(F)F)NC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F AW00197 c1ccc(cc1)c2csc3c2c(ncn3)Sc4ccccc4N AW00217 c1ccc2c(c1)-c3c(nc4ccc(cc4n3)Cl)C2=O BTB05337 c1cc(c(c(c1)F)C(=O)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F)F BTB05356 Cc1c(nn(n1)c2ccccc2)C(=O)ONC(=O)Cc3ccccc3 BTB03355 CN(C)c1ccc(cc1)CC(C#N)C#N BTB03400 c1cc(c(c(c1)F)C(=O)Nc2cc3cc(ccc3oc2=O)[N+](=O)[O-])F BTB03415 CCOC(=O)/C(=C/NCCc1ccncc1)/C#N BTB03431 Cc1ccc(cc1)NC(=O)c2cnccc2C(=O)OC BTB07961 CC(C)NC(=O)c1cccc2c1-c3ccccc3C2=O BTB10976 Cc1nc2ccccc2c(=O)n1c3ccccc3 BTB10993 Cc1ccc(cc1)c2[nH]c3ccccc3n2 BTB10994 Cc1ccc(cc1)C(=O)N2C(=O)C(CN(C2=S)c3ccccc3OC)(C)C BTB08258 c1cc(c(cc1F)F)Oc2cc3c(cc2[N+](=O)[O-])C(=O)NC3=O BTB08299 COc1ccc(cc1)OCCC(=O)NNC(=S)Nc2cc(ccc2Cl)Cl CD01776 COc1ccc(cc1)OCC(=O)Nc2ccc(cc2)C(=O)O BTB14128 Cc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cc(on2)C BTB14273 Cc1cc(ccc1Cl)OCc2c(c(c(c(c2C)C)C)C)C CD02212 c1cc(ccc1C(C2CC2)O)Br XBX00143 CCCCc1ccc(c(c1)C)NC(=O)N2CCCN(CC2)c3nc(ns3)c4ccccc4 AW00481 c1cc(ccc1C(=O)COC(=O)c2ccc(c(c2)Cl)F)Cl BTB03724 c1ccc(cc1)OCC(=O)Nc2cccc(c2C(=O)O)F BTB03730 Cc1ccc(cc1)N/C=C(\C#N)/c2[nH]c3ccccc3n2 BTB08365 C1CCN(C1)C(=O)C(C(C(=O)N2CCCC2)O)O BTB14422 CC(=O)c1ccc(c(c1)CSc2ccc(cc2)Cl)OC CD02434 CC(=O)c1ccc(c(c1)CSC#N)OC CD02443 COc1ccccc1C2CCN(CC2)Cc3cccc(c3)[N+](=O)[O-] BTB14603 c1ccc(cc1)Oc2ccc(cc2)OC(=O)c3ccc(cc3)[N+](=O)[O-] BTB14629 c1ccc(cc1)c2csc3c2c(ncn3)Sc4ccc(cc4)F AW00219 CC(=O)Nc1ccc(cc1C#N)[N+](=O)[O-] BTB00737 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCCCC3 AW00419 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCCN(CC3)c4nc(ns4)c5ccccc5 AW00445 CC(=O)C(C)(C)OC(=O)NCc1cccs1 BTB05610 CC(=O)C(C)(C)OC(=O)NCc1ccccn1 BTB05612 c1ccc2c(c1)c(=O)nc([nH]2)c3ccc(cc3)C#N BTB05668 Cc1cccc(c1NC(=S)N2CCOCC2)C DSHS01233 CC1CN(CC(O1)C)C(=S)Nc2ccccc2OC DSHS01250 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccc4c(c3)OCO4 DSHS01254 Cc1cccc(c1)NC(=S)N(CCC#N)C2CCCCC2 DSHS01268 CC1(CN(C(=S)N(C1=O)C(=O)c2c(cccc2Cl)F)c3ccccc3OC)C BTB08260 Cc1cc(nc(n1)S/C=C/C(=O)c2ccccc2F)C BTB11389 CCc1ccc(cc1)C(=O)/C=C/Nc2cccc(c2)Cl BTB11394 CC(=O)OCc1cccc2c1c(ccc2)Sc3ccccc3C(=O)NC BTB11479 c1cc(ccc1NC(=O)c2ccc(o2)S(=O)(=O)N3CCOCC3)S(=O)(=O)N HTS00422 c1cc(c(c(c1)F)C(=O)O)NC(=O)CCCC(=O)O HTS00457 Cc1c(c(c(c(c1C)C)CSC(=Nc2cccc(c2)OC)N(CCC#N)CCC#N)C)C CD02225 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)S(=O)(=O)c4ccc(cc4)C#N BTB14546 CC1(C2CCC(C2)(C1NC(=O)c3ccc(cc3)Cl)C)C BTB14560 CN1C2CCC1CC(C2)NS(=O)(=O)c3ccc(cc3)Cl BTB14569 Cc1c(ccc(n1)C(F)(F)F)c2nnc(o2)SCc3ccc(cc3)OC(F)(F)F AW00493 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)c4nc(ns4)c5ccccc5 AW00558 c1cc(ncc1[N+](=O)[O-])N2CCCN(CC2)C(=O)C3CCC3 AW00596 c1ccc(cc1)NC(=S)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl AW00667 CC(C)(C)NC(=S)N/N=C/c1cccc(c1O)OC BTB03761 c1cc(c(cc1C(=O)Nc2c(cc(cc2Br)F)F)Cl)Cl BTB03962 c1ccc(c(c1)C(=O)NC(=O)Nc2ccc(cc2)Br)N3CCCCC3 BTB03991 Cc1ccn2c(c1)ncc(c2=O)C(=O)O BTB08395 Cn1ccnc1SCC(=O)c2cccc(c2)[N+](=O)[O-] BTB08488 Cc1nc(c(=O)[nH]n1)Cc2ccc(cc2)OC BTB11725 c1cc2cccnc2c(c1)S(=O)(=O)N3CCCN(CC3)Cc4c(cccc4Cl)F HTS00681 c1cc2c(c(c1)S(=O)(=O)N3CCCN(CC3)Cc4c(cccc4Cl)F)non2 HTS00682 C/C(=N\OC(=O)c1ccc(cc1)[N+](=O)[O-])/c2ccc(c(c2)CN3CCCC3)OC CD02705 COC(=O)c1c(ccs1)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS04892 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])NC(=O)c3cc(on3)C HTS04901 c1c(cc(c(c1[N+](=O)[O-])NNC(=O)CC#N)[N+](=O)[O-])C(F)(F)F CD03571 Cc1c(cccc1Cl)NC(=O)N2CCCN(CC2)c3c(cccn3)[N+](=O)[O-] AW00452 Cc1cccc(c1NC(=S)N2CCc3ccccc3C2)C BTB01013 Cc1ccccc1NC(=S)NNC(=O)CCc2ccc(cc2)O BTB01052 CNc1nnc(s1)Sc2c(cccn2)[N+](=O)[O-] CD07979 Cc1cc(=O)oc2c1ccc(c2)OCc3c(cccc3Cl)F CD08040 c1c(cc(cc1C(F)(F)F)NC(=O)NC(=O)c2cc(sc2)[N+](=O)[O-])C(F)(F)F DFP00079 Cc1cc(sc1)C(=O)NNC(=O)c2ccc(cc2)C(C)(C)C GK02264 Cc1cc(sc1)C(=O)O/N=C(/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)\N GK02270 CC(C)(C)c1cc(cc(n1)c2ccc(cc2)Cl)SC EN00243 c1cc(c(c(c1)Cl)CS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl EN00245 Cc1csc2c1ncnc2N3CCN(CC3)C(=O)c4ccc(cc4)C(C)(C)C GK02677 CCOC(=O)C(=CN(C)c1ccccc1)C(=O)OCC GK02808 c1cc(ccc1C(=O)NNS(=O)(=O)c2ccc(cc2)Cl)[N+](=O)[O-] HTS00485 c1cc(ccc1C(=O)NNS(=O)(=O)c2ccc(cc2)F)[N+](=O)[O-] HTS00486 COCc1cc(nc(n1)SCCS(=O)(=O)c2ccc(cc2Cl)Cl)O HTS02277 Cc1nc(cn1C)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS02338 CN(C)c1ccc(cc1)n2c(nnn2)SC(c3ccccc3)c4ccccc4 HTS00792 c1cc(ccc1CC#N)NC(=O)CCCC(=O)O HTS04727 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3ccc(cc3)OC HTS04747 CCc1ccccc1NNC(=O)CCc2ccccc2 HTS04753 CCCc1ccc(cc1)C(=O)NNc2ccc(cc2)F HTS04770 c1ccc2c(c1)CC(=C2)N3CCN(CC3)c4ccc(c(c4)Cl)Cl HTS06841 Cc1c(ccc(n1)C(F)(F)F)C#N AW00676 c1ccc(cc1)NC(=O)N2CCCN(CC2)c3ccc(cn3)[N+](=O)[O-] AW00803 CC(C)(C)c1ccc(cc1)C(=O)NCCNc2nccc(n2)C(F)(F)F AW00815 c1cc(cc(c1)C(F)(F)F)C(=O)NCCNc2nccc(n2)C(F)(F)F AW00818 Cc1ccc(cc1C)OCC(CNCc2ccco2)O AW00832 CC(=O)Nc1c(cccc1Cl)F BTB04051 CC(=O)CSCC(=O)Nc1ccc(cc1F)F BTB04074 CC1CCN(CC1)S(=O)(=O)c2cc(c(c(c2)Cl)Oc3ccc(cc3Cl)[N+](=O)[O-])Cl BTB04103 c1cc(sc1)C(=O)Oc2ccc(cc2)F BTB04115 Cc1c(c(nc(n1)c2ccccc2)SCc3ccccc3[N+](=O)[O-])C#N HTS02504 c1cc(ccc1NC(=O)Nc2nc(cs2)c3ccc(c(c3)F)F)OC(F)(F)F HTS02514 Cc1cn(c2c1cccc2)CCC(=O)Nc3ccc(cc3)F HTS01096 c1cc(ccc1C2(CCN(CC2)C(=O)CC34CC5CC(C3)CC(C5)C4)O)Cl HTS01104 c1cc(cc(c1)Cl)C(=O)O/N=C(/c2c(cccc2Cl)Cl)\N CD03679 CCCCNC(=S)Nc1ccc(cc1)F CD03731 c1ccc(c(c1)C(=O)O)SCc2cccc(c2)C(F)(F)F CD03738 c1ccc(c(c1)C(=O)NCC2CC2)NS(=O)(=O)c3cccc(c3)C(F)(F)F HTS05145 COc1cc(ccc1CN2CCC(CC2)C(=O)c3ccc(cc3)F)OCc4ccccc4 HTS05159 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)N2CCN(CC2)CCN3CCOCC3 HTS05173 CCCCNC(=O)O/N=C/c1cc(sc1)[N+](=O)[O-] DFP00100 c1cc(ccc1c2cnco2)[N+](=O)[O-] DFP00101 Cc1ccc(cc1Cl)NC(=S)Nc2ccc(cc2[N+](=O)[O-])Cl DFP00139 c1ccc(cc1)c2nc(sn2)n3ccc(n3)c4cccs4 AW00838 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])n2ccc(n2)C(F)(F)F AW00851 COC(=O)c1c(ccs1)Oc2nccc(n2)C(F)(F)F AW00863 CC(C)(C)NC(=S)N/N=C/c1cc(cc(c1O)I)I BTB04126 c1cc(c(c(c1)Cl)CSCC(=O)Nc2ccc(c(c2)Cl)F)Cl BTB04179 c1cc(ccc1[N+](=O)[O-])OCC(CNCc2ccc3c(c2)OCO3)O HTS00972 Cn1c2cccc(c2c(n1)NC(=O)C3CCN(CC3)C(=O)OCc4ccccc4)OC HTS02638 Cn1cc(c(n1)c2cccc(c2)NC(=O)CCC(=O)O)Br HTS02656 CCOC(=O)C1=C(Oc2ccc(cc2C1C(C#N)C(=O)OCC)Cl)N HTS02701 COc1ccc(cc1N/C=C/c2nnnn2c3ccc(cc3)Br)C(F)(F)F HTS06848 c1cc(sc1)c2ccnc(n2)SCCS(=O)(=O)c3ccc(cc3)F HTS04959 c1cc(c(nc1)N2CCN(CC2)C(=O)Nc3ccc(cc3)OC(F)(F)F)C#N HTS04987 CC(C)(C)OC(=O)N[C@@H](CCC(=O)OCc1ccccc1)C(=O)N SB01934 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)CSCC(=O)O HTS01146 c1cc(sc1)S(=O)(=O)NCCN2CCNC2=O HTS02795 COc1ccccc1NC(=O)NCCN2CCNC2=O HTS02808 CC(=O)CNC(=O)Cc1ccccc1 BTB09315 Cc1ccc(c2c1CCC2)Oc3c(cccn3)[N+](=O)[O-] BTB09388 c1cc(c(c(c1)Cl)CO/N=C/c2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl CD04192 c1cc(c(c(c1)F)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F CD04254 C#CCSc1c(c(sn1)SCC#C)C#N CD00503 c1cc(ccc1C=C2C(=O)NC(=O)NC2=O)Cl CD00546 c1cnc(nc1C(F)(F)F)NCCN2C(=O)CC3(C2=O)CCCC3 AW00891 c1cc(oc1)C(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F AW01023 CC(C)(C)OC(=O)NC1CCN(CC1)S(=O)(=O)c2ccc(c(c2)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01047 COc1ccccc1Oc2ccccc2[N+](=O)[O-] BTB04185 c1cc(ccc1/C(=N/O)/N)[N+](=O)[O-] BTB04188 c1cc(sc1)c2nc(no2)c3ccc(cc3)[N+](=O)[O-] BTB04197 Cc1ccc(c2c1nc(cc2Oc3c(cc(cc3[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-])C)Cl BTB04487 CN(c1cccc(c1C#N)F)NC=C(C#N)C#N BTB04500 CCc1cccc(c1/N=C\2/NC(C(=C)S2)(C)C)CC BTB04521 Cc1c2c(c(=O)n(nc2c3ccccc3)c4ccccc4)no1 BTB09043 CC(C(=O)OC)Sc1nc(c2n1cccc2)C(=O)C(F)(F)F BTB09068 CN(C)CCCNC(=O)c1c(cccc1F)NC(=O)c2cccc(c2)C(F)(F)F BTB09176 Cc1c(cc2c(c1[N+](=O)[O-])C(CC2(C)C)(C)C)NN=C3C(=O)CC(CC3=O)(C)C CD03984 COC(=S)Nc1cccc(c1)C(F)(F)F CD03989 c1cc(cc(c1)[N+](=O)[O-])C(=O)/C=C/2\c3cc(ccc3NC2=O)Br BTBT00048 COc1ccc(cc1OC)CC2c3cc(c(cc3CCN2/N=N/c4cccc(c4)Cl)OC)OC BW00087 COc1ccc(cc1)/C=N/NC(=O)c2cccnc2 BW00105 c1cc(cnc1)c2cc(c3cc(ccc3n2)Br)C(=O)O BW00138 Cc1ccc(c2c1CCC2)OCC(=O)O RH01724 CN(CCO)c1cc(nc2c1cccc2)C(F)(F)F KM08215 CC(C)Cc1ccc(cc1)C(C)C(=O)NN SEW06461 c1ccc2c(c1)nc(c(n2)c3ccco3)c4ccco4 BTB09595 c1ccc(cc1)C(=O)C2=C(c3cccc4c3c(ccc4)C2=O)Cl BTB12966 Cc1cccc(c1)NC2=NCC(S2)(C)C BTB13021 c1ccc2c(c1)[nH]c(=O)c(n2)C(F)(F)F BTB13028 COc1ccc(c(c1OC)Cl)/C=C/2\C(=O)NC(=S)S2 BTB09822 C1CCCCC(C(=O)C(CCCC1)CCC(=O)O)CCC(=O)O BTB09925 Cc1cc(=O)oc2c1ccc(c2CC=C)O BTB09991 c1ccc2c(c1)cccc2/C=C/3\c4ccccc4NC3=O CD00758 Cc1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N/N=C/c2ccco2 CD00811 c1cc([nH]c1)C=C2C(=O)NC(=S)NC2=O CD00862 CC(C)(C)NC(=O)NCCc1ccccc1 CD00898 c1cc2c(cc1[N+](=O)[O-])NC(N2)c3ccc(s3)[N+](=O)[O-] BTB02216 c1cc(oc1)C(=O)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02222 Cc1c(c(nc(n1)c2ccccn2)NC3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)Cl AW01165 COc1cccc(c1)CC(=O)NC2CCN(CC2)c3nccc(n3)C(F)(F)F AW01178 c1ccc2cc(ccc2c1)c3csc4c3c(ncn4)O AW01192 CCCCCC(=O)Nc1ccccc1c2nnc(o2)c3ccc(cc3)Cl BTB06925 CS/C(=N\S(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)/N4CCCC4 BTB06972 CC(=O)Nc1cc2cc(ccc2oc1=O)n3cccc3 BTB04915 c1ccn(c1)c2cc3cc(ccc3oc2=O)[N+](=O)[O-] BTB04926 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccc(cc3C(=O)C)F BTB04937 C=CCSc1nnnn1c2ccc(cc2)O BTB09652 c1c(cncc1C(=O)O)C(=O)O BTB09654 CCCCCCCCCCCOC(=O)c1cc(cc\2c1-c3ccc(cc3/C2=N\O)[N+](=O)[O-])[N+](=O)[O-] BTB13159 CC(C)OC(=O)c1cccc-2c1C(=O)c3c2cccc3 BTB13172 CCCc1c(ccc2c1sc(cc2=O)C(=O)OC)O BTB10135 Cc1c(c(c(c(c1C)C)CN2CCCCC2)C)C CD00077 COc1cccc(c1OC)/C=C/2\c3ccccc3NC2=O CD00662 COc1cccc(c1)NC(=S)NNc2ccc(cc2)[N+](=O)[O-] CD00714 CC(C)(C)NC(=O)NCCCN1CCOCC1 CD00719 CN(C)c1ccc(cc1)/C=C/2\c3ccccc3NC2=O CD00741 CCCc1cc(=O)c2c(o1)cccc2OCC#C BTB10076 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1Cl)NC(=O)c2cccc(c2)Cl BTB13211 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1F)NC(=O)c2cccc(c2)Cl BTB13212 c1ccc2c(c1)C(c3ccccc3O2)C(=O)O/N=C/c4ccc5c(c4)OCO5 BTB10312 c1ccc(cc1)c2c(oc(n2)c3ccccc3)c4ccccc4 BTB10410 c1ccc(cc1)CC2=NN=C(NN2)Cc3ccccc3 BTB10416 CCNc1cc([n+](c2c1c(n[nH]2)/N=C/c3cc(cc(c3O)Cl)Cl)CC)N.[Cl-] CD01551 CCC(c1ccccc1)(c2ccccc2N)O CD01753 Cc1c(c(c(c(c1C)C)C(=O)c2ccc(cc2)[N+](=O)[O-])C)C CD01754 COc1cc(cc(c1OC)OC)/C=N/NC(=S)NC2CC3CC2C=C3 CD01773 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3cccs3)/C#N)C#N)n4cccc4 BTB02401 CCOC(=O)C1CCN(CC1)c2ccc(cc2NC(=S)Nc3cc(ccc3Cl)Cl)C(=O)C BTB02473 CCCCCCCc1ccc(cc1)C(=O)Nc2ccc(c(c2)Cl)F BR00011 CCCCCCCc1ccc(cc1)NC(=O)Nc2ccc(cc2)F BR00017 c1cc(sc1)C(=O)NC2=NCCS2 BR00046 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/c2cc(ccc2OC(=O)c3ccccc3F)F BTB04938 c1cc(cc(c1)Cl)Oc2ccc(cn2)[N+](=O)[O-] BTB07176 c1cc(cnc1)Oc2ccc(cn2)N BTB07204 c1c(cc(cc1Cl)Cl)NC(=O)CC#N BTB05105 Cc1cc(c(c(c1)C)NC(=S)NN=C2CCCCCC2)C BTB05126 c1cc(c(cc1NC(=O)C/C(=N/O)/N)Cl)F BTB05153 Cc1ccc2c(c1)C(=O)C(CO2)C(=O)C BTB10145 c1cc(ccc1C(=S)N2CCOCC2)Cl BTB10172 COC(=O)c1ccc(cc1)C(=O)NN BTB10177 CCCc1ccc(cc1O)SC(=O)N(C)C BTB10197 COc1ccccc1C2CCN(CC2)C(=O)C3CCCCC3 BTB13389 Cc1c(c2ccccc2[nH]1)CC#N BTB13427 CCCCCCC(=O)c1ccc-2c(c1)Cc3c2cccc3 BTB10534 CC(=O)/C(=N\O)/c1ccccc1 CD01161 c1ccc(cc1)c2csc(n2)N3CCOCC3.Br CD01172 COc1cc(cc(c1OC)OC)C(=O)NNC(=N)c2ccccn2 CD01223 CN(C)c1ccc(cc1)/C=N/c2ccccc2C(=O)NCCc3ccc(c(c3)OC)OC CD01376 CC(C)(C)c1ccc(cc1)OC(C)(C)C(=O)O JM00278 Cc1c(cnc(n1)c2ccccc2)CO CC20209 CN(C)CC1CCCCC1=O.Cl BTB10417 c1ccc(cc1)S(=O)(=O)Cc2ccsc2[N+](=O)[O-] BTB10426 CCCCCCc1ccc-2c(c1)Cc3c2ccc(c3)C#N BTB10461 c1cc(sc1)C(=NOC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3cccs3 BTB10715 Cc1c(c(sc1Br)Br)c2ccccc2 BTB10741 CCOC(=O)c1cnc(nc1O)S BTB10802 Cc1ccc-2c(c1)NNc3n2cnn3 BTB10874 COc1cccc(c1OC)/C=N/NC(=S)NC2CC3CCC2C3 CD02063 c1ccc(cc1)CC(=NO)Cc2ccccc2 CD02115 c1ccc(cc1)CC(=NOC(=O)c2ccc(c(c2)Cl)Cl)Cc3ccccc3 CD02176 c1cc(c(c(c1)Cl)CSC(=O)c2ccc(o2)[N+](=O)[O-])Cl BR00082 CCCCCCCc1ccc(cc1)C(=O)NC(=S)Nc2cc(on2)C BR00116 Cc1cc2c(cc1C)CSC(SC2)c3ccc(cc3)N(C)CCC#N BTB00423 Cc1cc2c(cc1C)CSC(SC2)(C)c3ccc(cc3)OC BTB00432 c1ccc(cc1)CNC(=S)NNC(=O)C2CCCNC2=O BTB00468 CC(C)(C)NC(=S)Nc1cccc(c1)SC BTB02982 Cc1cc(cc(c1Cl)C)OCOc2cc(c(c(c2)C)Cl)C BTB05156 c1cc(ccc1/C=N/Nc2ccc(cn2)[N+](=O)[O-])Cl BTB05157 CC(C)(C)c1csc(n1)N/N=C/c2ccc3c(c2)OCO3.Br BTB05188 c1cc(ccc1CC#N)OCc2cc(cc(c2)Cl)Cl BTB07443 c1cc(ccc1C#N)C2Nc3cc(ccc3O2)Cl BTB05377 COC(=O)c1cccc(c1c2c(cccc2[N+](=O)[O-])C(=O)OC)[N+](=O)[O-] BTB10591 Cc1cc(n[nH]c1=O)c2ccsc2 BTB10623 Cc1cccc(c1c2c(cccc2[N+](=O)[O-])C)[N+](=O)[O-] BTB10650 CCCCCCCCCCCCN1c2ccccc2C(C1=O)(c3ccc(c(c3)C)O)c4ccc(c(c4)C)O BTB13812 Cc1c(snn1)C(=O)ON=C2CCCCCCCCCCC2 BTB11033 CN(C)c1ccc(cc1)C(=O)NNC(=S)Nc2cccc(c2)OC CD01826 C1CC(OC1)CN(CCC#N)C(=S)NC2CC3CC2C=C3 CD01840 c1cc(c(c(c1)Cl)CSC(=C(C#N)C#N)SCc2c(cccc2Cl)Cl)Cl CD01912 c1ccc(cc1)CC(c2ccccc2)(c3ccccc3NC(=S)NC4CC5CC4C=C5)O CD01958 CC(=O)Nc1ccc(cc1)c2cc(c3ccccc3n2)C(=O)O RH00767 Cc1c(nc(o1)C(=O)NN)c2ccccc2 SEW01708 c1ccc(cc1)c2c3c(c(=O)c(c[nH]3)C(=O)O)sc2C(F)(F)F SEW03172 COc1ccc2cc(ccc2c1)c3ccn[nH]3 SEW04502 c1cc(ncc1C(F)(F)F)S(=O)(=O)CC#N KM04876 Cc1ccc2c(c1)nnc3n2c(=S)[nH]n3 BTB10876 c1ccc2c(c1)c(=O)n3c(n2)OCC3 BTB13943 CCOC(=O)CCn1cnc2c1c(=O)n(c(=O)n2C)C BTB13946 c1ccc(cc1)C(C=C2c3ccccc3-c4c2cccc4)C=C5c6ccccc6-c7c5cccc7 BTB11132 c1ccc(cc1)c2cc(c3c(c2C(=O)c4ccc(cc4)Cl)C(=O)CCCC3)c5ccc(cc5)Cl BTB11355 C/C(=N\O)/c1ccc(c(c1)CN2CCOCC2)OC CD02464 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)ONC(=O)c3ccccc3 CD02492 Cc1c(c(c(c(c1C)C)CO/N=C/c2cccs2)C)C CD02526 c1ccc(c(c1)C(=O)NNC(=S)Nc2cccc(c2)Cl)n3cccc3 CD02594 Cc1cc(ccc1Cl)C(=O)CSC#N BTB03006 c1cc(ccc1/C(=N/O)/N)Oc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB03015 COC(=O)c1cccc(c1C(=O)OC)[N+](=O)[O-] BTB00762 c1ccc2c(c1)CCCN2C(=O)c3c(c4ccccc4s3)Cl BTB00790 c1cc(c(cc1c2cnc3cc(ccc3n2)Cl)Cl)Cl BTB05385 CCc1cccc(c1NC(=O)NC(=O)c2c(c(cc(c2OC)Br)Cl)OC)CC BTB07740 CN(C)/C=N/c1nnc(s1)SCC#N BTB07772 c1cc(cc(c1)Cl)S(=O)(=O)N(c2ccc(nc2)Oc3cc(cnc3)Cl)S(=O)(=O)c4cccc(c4)Cl BTB07790 CCOC(=O)/C(=C/Nc1cc(c(c(c1)Cl)OS(=O)(=O)c2cc(cc(c2)Cl)Cl)C)/C#N BTB05662 c1ccc2c(c1)c(c(s2)C(=O)ON=C3CCCCCCCCCCC3)Cl BTB11034 c1cc(cnc1)C(=O)NNC(=S)NC23CC4CC(C2)CC(C4)C3 BTB11154 CN1CCN(CC1)c2cc(nc3c2cccc3)c4ccccc4 BTB14088 c1ccc(c(c1)C(=O)Nc2nc(cs2)CC(=O)O)Cl BTB14097 C[C@@H]1[C@H]([C@H]([C@@H](O1)n2cnc3c2ncnc3N)O)O BTB14111 CNC(=O)c1cccc2c1c(ccc2)Sc3ccccc3 BTB11487 c1ccc(c(c1)c2ccccc2C(=O)O)C(=O)Nc3ccc(cc3)F CD02261 COc1cc(c(cc1N2C(=O)C=CC2=O)Cl)OC CD02264 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3cccc(c3)C(F)(F)F CD02310 Cc1c(c(c(c(c1C)C)C(=O)/C(=N/N)/c2ccccc2)C)C CD02397 Cc1ccc(cc1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3)SC KM10242 c1ccc2c(c1)CCCN2c3nc(nc(n3)N4CCOCC4)N5CCOCC5 BTB01165 c1ccn(c1)c2ccc(cc2)CN CC25513 Cc1c(c(n(n1)C)O)/C=C/2\C(=NN(C2=O)C)C BTB06164 CC\1=NN(C(=O)/C1=C/c2ccc(cc2Cl)Cl)c3ccccc3 BTB06176 CC1(CC2=C(CC3=C(O2)CC(CC3=O)(C)C)C(=O)C1)C BTB14351 CNc1c(n(c(=O)[nH]c1=O)Cc2ccccc2)N BTB11737 CCN(CC)C(=O)Nc1ccc(cc1)OC BTB11746 CCc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2Cl)Cl BTB11787 COc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2Cl)Cl BTB11788 CC(=O)Nc1nc(cs1)c2cccs2 AW00005 CCOc1ccc(cc1)/C=N/NC(=S)NCCCOC CD02749 COc1ccccc1NC(=S)NNC(=O)CC#N CD02843 c1cc(sc1)/C=C(\C#N)/c2nc(cs2)c3ccc(cc3)Cl CD02864 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)Nc3ccc(c(c3C#N)Cl)N(C)C BTB03300 c1ccc2c(c1)NC=C(C(=N2)N)C#N.Cl BTB03346 c1cc(ccc1CCC(=O)NNC(=S)Nc2ccc(c(c2)Cl)Cl)O BTB01054 CS(=O)(=O)N1CCc2ccccc2C1 BTB01056 c1ccc(cc1)C(=O)NCc2ccc(cc2)Cl BTB01080 Cc1ccc(cc1N(S(=O)(=O)C)S(=O)(=O)C)[N+](=O)[O-] BTB01160 c1cc(cc(c1)S(=O)(=O)N(CCC#N)Cc2ccco2)C(F)(F)F BTB08202 Cc1ccc(cc1)n2c3c(cccn3)c(=O)nc2SCC#C BTB08211 c1ccc(cc1)c2c(=S)ssc2Sc3c(cccn3)[N+](=O)[O-] BTB08240 Cc1cc(sc1)C(=O)O/N=C/c2ccc(cc2)C#N GK02271 COC(=O)c1cc(c(cc1Br)C(=O)OC)Br BTB11563 c1ccc(cc1)C2OC[C@@H]3[C@@H](O2)[C@@H](C=CO3)O BTB11577 c1ccc2c(c1)c3ccccc3c4c2nc5nnnn5n4 BTB11718 c1ccc(cc1)C2(CCC3C2CCC3(c4ccccc4)O)O BTB14457 c1(c(c(c(c(c1F)F)F)F)C(=O)O)C(=O)O BTB14467 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)c4c(cccc4Cl)Cl BTB14538 c1ccc(cc1)NC(=S)NNC(=O)CC#N CD02667 Cc1c(c(c(c(c1C)C)CSc2nnc(n2c3ccccc3)/C(=C/c4ccc(cc4Cl)Cl)/C#N)C)C CD02679 Cc1cc(ccc1Cl)OCc2cc(ccc2OC)C(=O)C CD02687 Cc1ccc(cc1/N=C/c2ccc(cc2)OC)NS(=O)(=O)C BTB01176 Cc1ccccc1NC(=S)NNC(=O)c2ccccc2Cl BTB01234 COc1ccccc1NC(=S)NNC(=O)c2ccccc2Cl BTB01238 CCOC(=O)CCc1cc(c(c(c1)/N=C/c2c(c(cc(c2)Cl)Cl)O)O)/N=C/c3c(c(cc(c3)Cl)Cl)O BTB01260 c1ccnc(c1)/C=C/2\C(=O)NC(=S)S2 BTB01743 c1c(cc(c(c1/C=C\2/C(=O)NC(=S)S2)O)Cl)Cl BTB01744 c1ccc(c(c1)C(=O)Nc2cccc(c2)F)Cl BTB06193 c1cc(c(cc1c2nnnn2c3ccc(c(c3)Cl)Cl)Cl)Cl BTB06216 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2ccc(cc2)Cl BTB06223 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2cc(c(cc2Cl)Cl)C BTB06226 Cc1cc(c(cc1Cl)C)SCc2c3c(cc(=O)oc3[nH]n2)C BTB06377 CC\1=NN(C(=O)/C1=C/c2ccc(cc2Cl)Cl)c3cccc(c3)Cl BTB06417 c1ccc(cc1)Oc2c[nH]nc2c3ccc(cc3O)O BTB11794 Cc1ccc(c(c1)Br)OC(=O)c2cccs2 BTB14578 CN1C2C[C@@H](CC1CC2)NC(=O)Nc3ccc(cc3)Br.Cl BTB14595 Cc1c(cnn1c2ccc(cc2)F)C(=O)Nc3c4c(cccc4OC)n(n3)C HTS02615 Cc1c(cnn1c2ccc(cc2)F)C(=O)NCCSCc3cccc(c3)C(F)(F)F HTS02630 CCc1ccnc(c1)NC(=O)Nc2ccccc2C(C)(C)C HTS04809 Cc1c(cccc1Cl)NC(=S)NNC(=S)NCCCOC CD02872 CC(C)(C)OC(=O)NCCNC(=O)Nc1ccc(cc1)C(F)(F)F AW00390 CC(C)c1ccc(cc1)NC(=S)NC(=N)N CD03798 Cc1c(c(no1)c2ccccc2Cl)NC(=O)Nc3cc(cc(c3)OC)C(F)(F)F CD03854 c1cc(c(cc1S(=O)(=O)N2CCSCC2)Cl)Cl CD07832 Cc1c(c(c(c(c1C)C)S(=O)(=O)N2CCSCC2)C)C CD07854 Cc1ccc(cc1NC(=S)Nc2ccc(cc2)OC)NS(=O)(=O)C BTB01174 c1cc(cc(c1)NC(=S)N2CCOCC2)C(F)(F)F DSHS01229 c1cc(cc(c1)Cl)NC(=O)Nc2cc(sc2)[N+](=O)[O-] DFP00171 c1cc(ccc1c2cnco2)NC(=O)Nc3ccc(c(c3Cl)Cl)Cl DFP00216 c1cc(sc1)C(=O)C=C2SCCS2 EN00170 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)NC(=O)C(F)(F)F GK02429 c1cc(ccc1NC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)[N+](=O)[O-])F GK02433 CCCCNC(=O)c1cc(oc1C)S(=O)(=O)N2CCCCC2 HTS00393 COC(=O)c1ccsc1N2C(=O)c3ccccc3C2=O GK02874 CC(C)Nc1c2ccsc2ncn1 GK02878 Cc1cc(on1)NC(=O)C(=O)c2ccc(o2)CN3C(=O)c4ccccc4C3=O HTS02358 Cc1ccc(cc1)S(=O)(=O)CCN2CCN(CC2)c3ccccn3 HTS02439 CCc1ccccc1CSc2nnc(n2c3ccccc3C(F)(F)F)O HTS02457 Cn1cc(nc1)S(=O)(=O)NCc2c(cccc2Cl)Oc3ccccc3 HTS04650 c1cc(ccc1CC#N)NC(=O)c2c(nccn2)C(=O)O HTS04721 Cc1cc(cc(c1)NC(=S)Nc2ccc(cc2)Oc3ccc(cc3)OC(F)(F)F)C AW00237 c1cc(ccc1NS(=O)(=O)c2cc(c(cc2Cl)Cl)Cl)Oc3ccc(cc3)OC(F)(F)F AW00253 c1cc(cc(c1)Cl)N2CCN(CC2)c3nc(cs3)c4ccc(cc4)Cl HTS06850 Cc1cc2nccc(n2n1)c3ccco3 HTS06869 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3c(onc3c4ccccc4)C)C HTS06878 C/C=C(\C)/C(=O)NC(=S)NNC(=O)c1cccnc1 BTB01781 C/C=C(\C)/C(=O)NC(=S)NNC(=O)c1cc(c(c(c1)OC)OC)OC BTB01784 COc1cc(cc(c1OC)OC)C2Nc3ccc(cc3C(=O)N2)[N+](=O)[O-] BTB01827 c1cc2c(nnc(n2c1)C(F)(F)F)O RF03111 CC\1=NN(C(=O)/C1=C/c2ccc(cc2)Br)c3cccc(c3)Cl BTB06419 CCc1nn2cc(nc2s1)C(C)(C)C BTB06486 c1ccc(cc1)Sc2ccc(c(c2)OCC#N)[N+](=O)[O-] BTB06533 CCOC(=O)c1cnn(c1N)C EN00291 COC(=O)c1c(c(cs1)Br)O GK01940 c1cc(sc1)S(=O)(=O)CC#N KM01280 CC1c2cc(c(cc2CCN1C(=O)c3c(c4ccccc4s3)Cl)OC)OC HTS04857 Cc1c(cc(o1)C(C)(C)C)C(=O)N2CCN(CC2)c3ccccc3OC HTS04878 c1cc(ccc1F)S(=O)(=O)NC2CCS(=O)(=O)C2 HTS02839 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)C(=O)NCc3ccc4c(c3)OCO4 HTS02885 c1cc2c(cc1COCc3ccc4c(c3)CCO4)CCO2 HTS02910 C#Cc1cccc(c1)NC(=O)C(Cl)(Cl)Cl CD07867 Cc1cc(c(c(c1)Br)NC(=O)C(Cl)Cl)Br CD07893 Cc1cc(c(c(c1)Br)NC(=O)c2cccs2)Br CD07898 c1c(cc(cc1C(F)(F)F)S(=O)(=O)NCCCNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F CD04333 Cc1c(c(c(c(c1C)C)CN2CCCCCC2)C)C CD04377 c1c(cc(cc1C(F)(F)F)NCN2C(=O)CCC2=O)C(F)(F)F CD04438 c1cc(ccc1CSc2nc3cc(ccc3s2)Cl)Cl EN00193 c1ccc2c(c1)c(c(s2)C(=O)Nc3cc(ccc3N4CCCCC4)C(F)(F)F)Cl BTB01901 c1ccc(cc1)CNc2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB01954 CCOC(=O)C(=CNc1cc(ccc1NCc2ccccc2)C(F)(F)F)C(=O)OCC BTB01956 c1ccc2c(c1)C(=O)N(C2=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS00734 Cn1cccc1CN(Cc2ccc(cc2)OC)S(=O)(=O)c3cccc(c3)C(F)(F)F HTS00762 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)C3CCC3C(=O)O HTS00767 Cc1c(nn(n1)c2ccccc2)c3nnc(o3)c4ccc(cc4)Cl BTB06547 CCOC(=O)C1=C(Oc2c(cc(cc2OC)Br)C1C(C#N)C(=O)OCC)N HTS02703 Cc1ccc(n1c2cc(ccc2N3CCN(CC3)C(=O)c4ccc(cc4)F)[N+](=O)[O-])C HTS04914 CC(C)(C)c1ccc(cc1)C2=NC(=O)C(S2)CC(=O)O HTS04921 c1cc(c(nc1)NNC(=O)CSCC(=O)O)C#N HTS04936 c1cc(sc1)C(=O)/C=C/2\NC(=O)CS2 CD07664 Cc1ccc(c(c1)OC(=O)/C=C/C(=O)Oc2cc(ccc2C)C)C CD07707 c1ccc(c(c1)NC(=O)C(Cl)(Cl)Cl)Sc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] CD04032 c1cc(oc1/C=N/NC(=O)CC#N)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04152 c1cc(cnc1)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD04190 Cc1c(noc1NC(=O)NC(=O)c2cc(c(c(c2)F)N(C)C)F)C SEW01753 C1CN(C(=O)N1)CCNC(=O)CCC(=O)O HTS02473 c1csc(c1Br)C(=S)N SEW03535 CCOC(=O)C1=C(OC(=C(C1c2ccc3c(c2)CCO3)C#N)N)C MO00266 c1ccc(cc1)C2CCC(=O)/C(=C\Nc3cccc(c3)C(F)(F)F)/C2=O KM05261 CSc1c-2c(c(s1)C(=O)N)CCc3c2onc3 KM05283 c1cc2c(cc1S(=O)(=O)N3CCN(CC3)c4nc5cc(ccc5s4)Cl)CCO2 HTS03275 c1ccc(c(c1)NC(=O)CN2CCN(CC2)c3nc4cc(ccc4s3)Cl)Oc5ccc(cc5Cl)Cl HTS03280 CC(C)(C)c1csc(n1)c2ccc(s2)c3ccccn3 HTS03331 C=CCn1c2c(c(=O)[nH]cn2)sc1=S HTS09062 c1cc(ccc1Cn2c3c(c(=O)[nH]cn3)nn2)F HTS09091 c1cc[n+](cc1)CC(=O)c2c(cccc2F)F.[I-] CD04770 Cc1ccc(n1c2ccsc2COC(=O)c3c(onc3c4c(cccc4Cl)F)C)C CD08865 COc1ccc(cc1)/C=C(\C#N)/C(=O)N2CCOCC2 DP00493 CCO/C=N\C1=C(C(c2ccc3ccccc3c2O1)c4ccc(cc4)Cl)C#N FM00130 CCOC(=O)Cc1cnc(s1)NN=C2C3CC4CC(C3)CC2C4 FM00166 c1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccccc3)/CC2 DP00959 c1c(ccc(c1)Cl)/C=C\2/C(=O)/C(=C/c3ccc(cc3)Cl)/CC2 DP00964 CCOC(=O)CSc1[nH]c2ccccc2n1.Cl DP00997 COc1cc(c(s1)C(=O)OC)OC(=O)c2cccs2 GK03021 COC(=O)c1c(ccs1)NCc2ccccc2 GK03119 Cn1c(ccn1)NC(=O)/C=C/C(=O)O GK03197 c1cc(c(cc1Cl)NC(=O)N/C=C/c2ccsc2)F GK03206 CCOC(=O)c1ccc(cc1)NC(=S)N GK03261 c1cc(c(cc1F)NC(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl)F HTS01151 CCOC(=O)c1c2c(sc1NC(=O)NC(C)(C)C)CN(CC2)C HTS02982 c1cc(ccc1NC(=O)NCc2ccc3c(c2)OCO3)OC(F)(F)F HTS03100 CC(C)c1cc(c(c(c1)Br)NC(=O)NCc2ccc3c(c2)OCO3)Br HTS03101 c1ccc2c(c1)CC(C2)NC(=O)CCCO HTS03104 c1cc(oc1)C(=O)N2CCN(CC2)CCN3CCOCC3 HTS05175 c1ccc2c(c1)c(c(s2)C(=O)Nc3nnc(s3)C4CC4)Cl HTS03422 c1ccc(cc1)c2c(nnn2c3ccc(cc3)[N+](=O)[O-])C(=O)O CD04612 c1c(cc(cc1Br)Br)CN2CCOCC2 CD08468 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])SC2=NCCS2 CD08585 c1cc(ccc1SCCSc2ccc(cc2)Cl)Cl CD05014 COc1ccc(cc1OC)S(=O)(=O)Oc2ccc(cc2)C#N CD05035 Cc1c(c(n(n1)C)NNC(=O)c2c(cccc2Cl)Cl)[N+](=O)[O-] EN00276 Cc1c(c(n(n1)C)n2c(c(cn2)C#N)N)[N+](=O)[O-] EN00284 COC(=O)c1ccccc1NC(=O)COc2ccc(cc2Cl)Cl EN00299 c1cc2c(cc1[N+](=O)[O-])NC(O2)c3ccc(s3)[N+](=O)[O-] BTB02164 Cc1ccc(c(c1)N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB02189 CCOC(=O)C(=CNNc1ccccc1)C(=O)OCC BTB02201 c1cc(ccc1OCC(CNCc2ccc3c(c2)OCO3)O)SC(F)(F)F HTS00987 COC(=O)c1c(ccs1)S(=O)(=O)Nc2cc(sc2C(=O)OC)c3cccs3 HTS01043 CN(C)/C=N/c1nnc(s1)SCC(=O)Nc2cc(cc(c2)Cl)Cl BTB06772 C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/c2ccc(c(c2)F)F BTB06877 CS/C(=N/S(=O)(=O)c1ccc(cc1)n2c(cc(n2)C(F)(F)F)c3cccs3)/N/N=C/c4ccccc4 BTB06881 c1cc(c(c(c1)Cl)CNS(=O)(=O)c2ccc(s2)c3ccno3)Sc4ccc(cc4)Cl HTS05265 c1cc(c(c(c1)Cl)CNC(=O)c2ccc3c(c2)CCO3)Sc4ccc(cc4)Cl HTS05266 c1cc2c(c(c1)S(=O)(=O)NN3CCOCC3)non2 HTS03661 Cc1ccc(cc1S(=O)(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)[N+](=O)[O-] HTS03692 Cc1ccc(cc1NS(=O)(=O)c2ccc(c(c2)Cl)NC(=O)C)S(=O)(=O)N(C)C HTS05509 c1ccc(c(c1)C(=O)NC(=O)SCc2c(cccc2Cl)F)Oc3ccc(cc3Cl)Cl CD08929 CN(C)c1ccc(cc1)/C=C(\C#N)/C(=O)c2cccs2 CD05224 c1cc(oc1)C(=O)/C(=N/O)/C#N CD05265 Cc1cccn(c1=O)Cc2c(cccc2Cl)Cl CD09416 C1COCCN1S(=O)(=O)c2c(c(sc2Cl)Cl)Br CD09581 c1cc(cc(c1)OC(=O)Nc2ccc(cc2)Cl)N3CCOCC3 CD09596 CNc1ccc(cc1C(=O)NC2CCCCC2)Cl DP01006 c1csc(c1NC(=O)C(Cl)Cl)C(=O)O GK00011 CCOC(=O)C(=CNc1ccsc1)C(=O)OCC GK00016 c1cc(ccc1c2nc(on2)CCC(=O)O)Cl DP01167 CCc1nc(no1)c2ccc(cc2)Cl DP01237 COC(=O)c1c(ccs1)NC(=O)NC(=O)c2c(cccc2Cl)Cl GK00380 Cc1ccccc1C(=O)Nc2ccc(cc2)S(=O)(=O)Nc3cc(on3)C GK03436 CC(C)Nc1c2cnn(c2ncn1)C GK03457 COc1cccc(c1)Nc2c3cc(c(cc3ncn2)OC)OC GK03503 Cn1c2c(cn1)c(ncn2)NNS(=O)(=O)c3ccc(cc3)Cl GK03543 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Nc3ccc4c(c3)OCO4 HTS01365 c1cc(oc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS01399 CCOC(=O)C1CCN(CC1)c2ccccc2CN3CCCc4c3ccc(c4)C HTS03469 CCCc1c(cnn1c2ccccc2)C(=O)NC3CCN(CC3)Cc4ccccc4 HTS03517 c1cc(ccc1c2c(c[nH]n2)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)F HTS05419 c1cc(ccc1c2c(c[nH]n2)CN3CCC(CC3)(c4ccc(cc4)Cl)O)F HTS05426 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)CC(COc4ccc(cc4)c5csnn5)O HTS03849 CC1=C(C(=O)OC1c2c(cccc2Cl)Cl)O CD09144 Cc1cc(ccc1Cl)OS(=O)(=O)CS(=O)(=O)Oc2ccc(c(c2)C)Cl CD09829 CNC(=O)N1CCCC(C1)Cn2cccc2 CD09942 c1ccc(c(c1)n2ccnc2S)Cl CD09952 c1cc(c(cc1S(=O)(=O)NC2CC2)Cl)Cl BTB04269 CCOC(=O)c1cnc(nc1N)SCC(=O)c2ccc(c(c2)C)Cl BTB04329 c1ccc2c(c1)c(nc(n2)O)O BTB02356 c1ccc(cc1)CCNC(=S)NNC(=O)CCc2ccc(cc2)O BTB02367 CC(=O)C(=CNc1ccc(cc1)F)C(=O)C BTB02370 Cn1c(nnc1S)c2ccco2 BTB02377 c1ccc(c(c1)C(=O)c2cc(ccc2NC(=O)c3cccc(c3)F)Cl)Cl BTB09237 c1cc2c(cc1Br)[nH]c(=O)s2 BTB09256 CC1(c2cc(ccc2OC1N3CCOCC3)O)C BTB09297 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(C)c3c4c(nn3C)CCCC4 BTB07101 c1cc(c(cc1Cl)Sc2ccc(cn2)[N+](=O)[O-])Cl BTB07160 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNc3ccccc3OC HTS05544 Cc1cccc(c1C(=O)O)NC(=O)c2cc3ccccc3s2 HTS05567 COc1ccc(cc1)SCCC(=O)NNS(=O)(=O)c2ccc(s2)CNC(=O)c3ccccc3 HTS05875 Cc1cc(cc(c1)NC(=O)Nc2ccc3ccccc3n2)C HTS05969 c1cc(c(cc1OS(=O)(=O)c2c(c(sc2Cl)Cl)Br)Cl)Cl CD09629 Cc1c(c(n(n1)C)C)NC(=O)c2ccccc2NC(=O)Nc3ccc(cc3)Cl CD10051 CCOC(=O)c1cnn(c1C)c2c(cc(cc2Cl)Cl)Cl CD10067 CC1SCC(=NOCc2c(cccc2Cl)F)CS1 CD10161 Cn1ccc(n1)NC(=O)NC(=O)c2c(cccc2F)F GK00384 c1c(c([nH]n1)NC(=O)C(Cl)Cl)Br GK00505 c1csc(c1N)C(=O)NN GK00508 Cc1csc(c1C(=O)NC)NC(=O)C(F)(F)F GK00521 COC(=O)c1c(ccs1)S(=O)(=O)Nc2ccc(cc2)F GK00888 Cc1ccsc1/C=C/C(=O)O/N=C/c2c(cccc2Cl)Cl GK00984 CC(C)(C)c1cc(c(s1)C(=O)N)NC(=O)/C(=C/c2ccc(cc2)Cl)/C#N GK01079 c1cc(oc1)CNc2nccc(n2)C(F)(F)F HAN00244 Cn1c(ccc1S(=O)(=O)N2CCN(CC2)c3ccc(cn3)C(F)(F)F)C(=O)O HTS01557 c1ccc2c(c1)cc(o2)c3csc(n3)NNC(=O)c4ccc(cc4)Cl HTS01567 c1ccc(cc1)c2csc(n2)c3cccs3 HTS01588 COc1cc2c(cc1OC)nc(sc2=O)NC(=O)c3ccc(cc3)OC(F)(F)F HTS01598 CC(C)(C)c1ccc(cc1)NC(=O)COc2c3ccc(cc3ncn2)Cl HTS06416 CC(C)(C)c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cc3)F HTS05804 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2c(n(n(c2=O)c3ccccc3)C)C HTS05807 CCOC(=O)c1c(c2cc(ccc2n1C)[N+](=O)[O-])NC(=O)Nc3ccc(cc3)C(C)(C)C HTS06011 Cc1ccc(nc1)NC(=O)CC(CC(=O)O)c2ccccc2 HTS06031 Cc1c(c(n(n1)C)C)N/C(=N/C#N)/SC CD09979 COC(CNc1cccc(c1C#N)F)OC CD09994 Cc1c(c(n(n1)C)C)NC(=O)CC#N CD10002 CC1SCC(=NOCc2c(cccc2Cl)Cl)CS1 CD10044 Cc1cc(no1)NC(=O)C(=O)N CD10336 Cc1c(cnn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NC CD10345 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3cccc(c3)[N+](=O)[O-])/C#N)C#N)n4cccc4 BTB02392 c1ccc(c(c1)C#N)n2c(c(cn2)C#N)N BTB04531 COc1cc(cc(c1OC)OC)C(=O)c2ccccc2C#N BTB04552 c1ccc(cc1)c2nc3c(cc(cc3Br)Br)c(=O)o2 BTB02538 C/C(=N\NC1=NCCN1Cc2ccccc2)/c3ccc(cc3)Br BTB02546 C/C(=N\NC1=NCCN1Cc2ccccc2)/c3ccc(cc3)Cl BTB02547 c1cc(cc(c1)Oc2ccc(cn2)[N+](=O)[O-])C(F)(F)F BTB07166 Cc1ccc(c2c1CCC2)OC(C)(C)C(=O)Nc3ccc(nc3)Oc4ccc(cc4F)F BTB09673 Cc1ccc(nn1)N(C)NC(=O)NC(=O)c2c(cccc2Cl)F BTB07306 Cn1c(=O)c(c(cn1)SCc2ccccc2)Cl BTB07372 c1cc(c(cc1C(F)(F)F)[N+](=O)[O-])Oc2cc(cnc2)Cl BTB07420 c1cc2c(c(c1)S(=O)(=O)Nc3ccc4c(c3)OCCO4)non2 HTS06021 CCCc1c(cnn1c2ccccc2)C(=O)Nc3cc(ccc3C)S(=O)(=O)N(C)C HTS06221 Cc1ccc(cc1NC(=O)CCc2ccccc2)S(=O)(=O)N(C)C HTS06231 c1cc(c(c(c1)F)C#N)N2CCC(CC2)C(=O)N CD10249 Cc1c(nnn1c2ccc(c(c2)Cl)Cl)C(=O)C CD10511 Cc1c(nnn1c2cc(ccc2Cl)Cl)C(=O)/C=C/N(C)C CD10581 CS/C(=N\S(=O)(=O)/C=C/c1ccccc1)/NN CD10589 Cc1c(cnn1c2ccc(c(c2)Cl)Cl)C(=O)C CD10634 CC(C)(C)c1cc(c(s1)C(=O)N)NC(=O)/C(=C/c2ccc(cc2)C#N)/C#N GK01081 c1cc(ccc1/C(=N/OC(=O)/C=C/c2cc(sc2)[N+](=O)[O-])/N)Cl GK01196 CCCc1c(cnn1c2ccccc2)c3nc(no3)c4ccc(cc4)C(C)(C)C GK01543 c1cc(ccc1n2c(c(cn2)NC(=O)Nc3ccc(cc3Cl)Cl)C(F)(F)F)Cl GK01560 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)CCC(=O)O HTS01717 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc4c(c3)OCO4)C HTS01777 Cc1ccc(cc1)S(=O)(=O)Nc2ccc(nc2)Oc3ccc(cc3C4CCCCC4)Cl HTS01793 c1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)Nc3cccnc3 HTS01795 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=O)CC(CC(=O)O)c3ccccc3 HTS06056 Cc1cc(no1)C(=O)NNc2c(cccc2Cl)Cl HTS06169 c1ccc(c(c1)NC(=O)C2=CCCCC2C(=O)O)N3CCCCC3 HTS06209 c1ccc(cc1)N(C2CCCCC2)C(=O)CN3CCN(CC3)C(=O)C4COc5ccccc5O4 HTS06263 c1ccc2c(c1)OCC(O2)C(=O)N3CCN(CC3)CC(=O)Nc4cccc(c4)C#N HTS06266 Cc1cnnn1c2c(nn(c2C)C)C CD10365 c1cc(cc(c1)Cl)CNC(=O)C(=O)NC2CCCCNC2=O CD10480 Cc1c(c(sc1C#N)C(=O)NC(=O)OCC#Cc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C CD10493 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)C#N CD10698 Cc1cc(cc(n1)NN/C(=N\S(=O)(=O)c2ccccc2)/SC)C(F)(F)F CD10707 c1ccc(c(c1)C(=O)NCC(=O)NNC=C(C#N)C#N)[N+](=O)[O-] BTB02612 CC(C)(C)c1cs/c(=N\c2ccc(cc2)Cl)/n1c3ccc(cc3)Cl BTB04960 Cc1cc(cc(c1Cl)C)OCc2nc(no2)c3cccc(c3)[N+](=O)[O-] BTB02943 Cc1cc(ccc1Cl)C(=O)c2cc3ccccc3o2 BTB02951 Cc1cc(ccc1Br)NC(=S)NC(C)(C)C BTB02974 c1cc(ccc1C(F)(F)F)S(=O)(=O)Nc2ccc(nc2)Oc3ccc(cc3Cl)Cl BTB07429 CCSc1c(cccn1)C(=O)Oc2cc(nn2c3ccccc3)C BTB07658 COc1c(cc(c(c1C(=O)NC(=O)Nc2cc(cc(c2)Cl)Cl)OC)Br)[N+](=O)[O-] BTB07712 COc1ccc(c(c1C(=O)OC)OC)n2cccc2 BTB07737 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)F HTS06245 c1ccc(c(c1)C(=O)NCCCN2CCOCC2)NC(=O)c3cc(cc(c3)Cl)Cl HTS06334 c1cc(c(nc1)Oc2c3ccc(cc3ncn2)Cl)[N+](=O)[O-] HTS06408 c1ccc(cc1)C(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl HTS06418 Cc1c(c(on1)C)S(=O)(=O)/N=C(\NCC#C)/SC CD10649 Cc1c(c(on1)C)S(=O)(=O)/N=C(\NNC(=O)Nc2ccc(cc2)Cl)/SC CD10652 c1cc(c(cc1C(=O)NCc2cc(cc(c2)Cl)Cl)Cl)Cl CD10794 CS/C(=N\C#N)/NCc1c(cccc1F)N CD10870 COc1ccc(cc1)n2c(=O)c3ccccc3c(n2)C(=O)Oc4ccc(cc4)[N+](=O)[O-] CD11093 c1cc(ccc1NC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl)OC(F)(F)F GK01567 c1cc(ccc1n2c(c(cn2)C(=O)Sc3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(F)(F)F)Cl GK01592 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)OC)NC(=O)c3ccccc3 HTS01891 c1cc(c(cc1NC(=O)CSCC(=O)O)C(F)(F)F)Br HTS01931 Cc1cc(n(n1)C)C(=O)NC2(C(=O)c3ccccc3C2=O)O HTS01976 c1ccc2c(c1)C(=O)C(C2=O)(NC(=O)c3c(cccc3Cl)Cl)O HTS01978 CC(C)(C)OC(=O)N1CCC(CC1)CNS(=O)(=O)c2cccs2 HTS02033 Cc1c(snn1)C(=O)Nc2ccc3ccccc3n2 HTS06275 c1ccc(cc1)C(CC(=O)Nc2ccc(cc2)C#N)CC(=O)O HTS06302 Cn1c(ccn1)NC(=O)CC(CC(=O)O)c2ccccc2 HTS06319 CC(C)(C)c1ccc(cc1)NNC(=O)c2ccno2 HTS06472 Cc1ccc2nc(cn2c1)c3ccc(cc3)F HTS06528 Cc1ccc(cc1)c2cn3cc(ccc3n2)C HTS06531 CC(C)(C)C(=N)NC(=O)c1ccc(o1)[N+](=O)[O-] BR00126 CCc1cc2c(cc1C(=O)CC3(c4cc(ccc4NC3=O)Br)O)C(CCC2(C)C)(C)C BTB00084 CC(C)(C)NC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F BTB02978 c1cc(sc1)C(=O)Oc2ccc(cc2)c3ccc(cc3)OC(=O)c4cccs4 BTB05202 C/C(=N\N=C(/N=C/N(C)C)\SC)/c1ccc(cc1)F BTB05221 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Oc2c(cccc2OC)C BTB03157 COc1ccc(c(c1C(=O)OC)OC)[N+](=O)[O-] BTB03225 c1cc(sc1)C(=NOC(=O)c2cccs2)c3cccs3 BTB10696 CC(=O)Nc1ccc-2c(c1)CCc3c2cccc3 BTB10710 c1ccc(cc1)/C=C/C(=O)Nc2cccnc2Oc3ccc(cc3)F BTB08113 c1ccc(cc1)C(c2ccccc2)C3CCN(CC3)C(=O)C(Cl)(Cl)Cl BTB08145 CSc1c(c([s+]s1)SC)c2ccccc2.[I-] BTB08163 CSc1c(/c(=N/c2cccc(c2)C(F)(F)F)/ss1)c3ccccc3 BTB08195 c1ccc(cc1)C(=O)NNc2cc(cc(c2)Cl)Cl HTS06461 CCc1ccc(cc1)C(=O)NNc2ccc(cc2)C(C)(C)C HTS06467 CC1(OC(=O)C(=Cc2ccc(cc2)Br)C(=O)O1)C CD06805 c1cc(cnc1)Oc2ccc(c(c2C#N)Oc3cccnc3)[N+](=O)[O-] CD07413 c1cn(cn1)CCCNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD07434 c1c(cc(cc1Cl)Cl)C(=O)c2cc(cc(c2)Cl)Cl CD07463 CN(C)/C=C/C(=O)c1ccc(cc1)Br CD11131 CN(C)c1cc(oc(=O)c1Cl)c2ccc(cc2Cl)Cl CD11157 CC(=O)c1c(c2ccccc2nc1O)O CD11244 CC(C)(C)Sc1ccc(cc1[N+](=O)[O-])C(=O)N(Cc2ccc3c(c2)OCO3)c4ccc(cc4)F DSHS00953 CC(C)Sc1ccc(cc1C(=O)Nc2ccncc2)[N+](=O)[O-] DSHS01005 Cc1c(c(c(c(c1C)C)CSCc2n[nH]c(=S)n2c3cccc(c3)C(F)(F)F)C)C DSHS01021 Cc1c2c(cc(s2)C(C)(C)C)sc1C(=O)Nc3ccc(cc3)F GK01849 COC(=O)c1c(ccs1)OS(=O)(=O)c2ccc(cc2)C(F)(F)F GK01932 c1c(c(nc(n1)N2CCSCC2)C(F)(F)F)C(=O)OCC3CC3 GK02056 c1ccc(cc1)n2c(c(cn2)C(=O)NNC(=O)c3cc(cc(c3)Cl)Cl)C(F)(F)F GK02069 c1csc(c1Cl)C(=O)NN2CC(=O)N(CC2=O)c3cc(cc(c3)Cl)Cl HTS02092 Cc1ccc2c(c1)CCCN2CC(=O)Nc3ccc(cc3C(=O)NCc4cccs4)Cl HTS02131 COc1ccc(cc1OC)CCNC(=O)c2cc3ccccc3s2 HTS02161 c1ccc2c(c1)cc(s2)C(=O)N(Cc3ccccn3)Cc4ccccn4 HTS02162 c1cc(sc1)C(=O)c2[nH]ccn2 HTS02197 Cc1c(cc(o1)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N)C(=O)OC HTS06652 CCOC(=O)C1CCN(CC1)C(=O)c2c(nc(s2)c3ccccc3)C HTS06677 Cc1ccc(cc1C)C(=O)N2CCNC(=O)C2CC(=O)Nc3ccc(cc3)OC HTS06724 Cc1c(c2ccccc2[nH]1)SCC(=O)NNC(=O)c3cccs3 KM07815 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCCn3cc(c(=O)[nH]c3=O)C#N KM07836 Cc1ccc(cc1)CSc2nc3c(c4cc(ccc4[nH]3)Br)nn2 BTB00501 CC(=O)Nc1ccc(cc1NC(=S)Nc2ccccc2Cl)OC BTB00546 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F AW00318 Cc1cccc(c1NC(=O)N2CCCN(CC2)c3c(cccn3)C(F)(F)F)Cl AW00335 COc1cc(c(cc1Cl)OC)/N=C\c2ccc3c(c2)OCO3 BTB00826 Cc1ccc(cc1)C(=O)CCN2CCOCC2 BTB03284 c1cc(c(cc1c2cnc3cc(ccc3n2)F)Cl)Cl BTB05386 c1cc(c(cc1c2cnc3cc(ccc3n2)C(F)(F)F)Cl)Cl BTB05388 CC(=O)OCc1csc(n1)c2ccc(cc2)Cl BTB05432 Cc1c(nn(n1)c2ccccc2)C(=O)Sc3ccccn3 BTB03581 c1ccc2c(c1)nc(s2)c3ccc(cc3)CSc4ccccn4 BTB03599 c1cc2c(c-3c(cc2)/C(=C/C(/C=C\4/c5c(c6c(cc5)cccc6)-c7c4cccc7)/C=C\8/c9c(c2c(cc9)cccc2)-c2c8cccc2)/c2c3cccc2)cc1 BTB11078 Cc1ccc(cc1)c2cc(c(=O)[nH]n2)Cc3cccn3c4ccc(cc4)Cl HTS04529 CC(C)(C)c1ccc(cc1)NC(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl HTS04543 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4cccnc4Sc5ccc(cc5)Cl HTS04583 CSC1=C(C(=O)NC(S1)c2c(cccc2Cl)Cl)C#N CD07552 Cc1ccc(cc1)S(=O)(=O)NC(=O)Nc2nc(c(s2)C)c3ccc(c(c3)Cl)C HTS06900 c1cc(sc1)C(=O)Nc2nc(cs2)c3ccc(c(c3)F)F HTS06922 C1COCCN1C(=O)C(Cl)(Cl)Cl DSHS01059 c1ccc(cc1)C23c4ccccc4C(=O)N2CCN3C(=S)Nc5cccc(c5)Cl DSHS01080 Cc1c(c(no1)c2ccccc2)C(=O)NCC3COc4ccccc4O3 HTS10755 CC(C)(C)c1ccc(cc1)NC(=O)Nc2c(ccs2)c3nc4ccccc4s3 HTS10884 c1ccc2c(c1)nc(s2)c3ccsc3NC(=O)Nc4cccc(c4)Cl HTS10887 CC(=O)NC12CC3CC(C1)CC(C3)(C2)NC(=O)C JFD02057 c1ccc(cc1)CNC(=O)CNC(=O)COc2ccccc2 JFD02071 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NC(=S)N/N=C\2/c3cc(ccc3NC2=O)Br)OC(=O)C)OC(=O)C)OC(=O)C JFD02097 COC(=O)C(c1ccc(cc1)NC(=O)Nc2cccc(c2)Cl)(C(F)(F)F)O JFD02173 c1ccc(cc1)NC(=O)CSCCS(=O)(=O)c2ccc(cc2)Cl KM01723 c1ccc(cc1)S(=O)(=O)CCSCC(=O)Nc2ccc(cc2)Cl KM01725 c1cc(cc(c1)Cl)S(=O)(=O)CC#N KM01728 COC(=O)c1c(c(c(s1)SC)C#N)c2ccc(s2)Br KM01764 CS/C(=C(/C#N)\C(=O)c1ccc(cc1)Cl)/NCC2CC2 KM01814 Cc1cccc(c1)c2c(c([nH]n2)S(=O)(=O)C)C#N KM01865 c1ccc(cc1)C(=O)OCC#Cc2ccc(s2)c3ccccn3 KM07840 c1cc(cc(c1)Oc2c(nccn2)/C(=N/OC(=O)Nc3ccc(cc3)Cl)/N)C(F)(F)F KM07856 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)SCc3ccccc3 KM07901 Cc1c2ccccc2sc1CN3CCC(CC3)C(=O)c4ccc(cc4)F HTS06970 CCCCc1ccc(cc1)NC(=O)Nc2ccc(cc2)N3CCCCC3 HTS06978 COc1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)S BTB00882 c1ccc(c(c1)N)SC(CC(=O)c2cccs2)c3cccs3 CD07715 c1c(cc(c(c1[N+](=O)[O-])Sc2nnc(s2)N)[N+](=O)[O-])C(F)(F)F CD07813 CC1CN(CC(O1)C)C(=N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD07818 CCOC(=O)c1cc2cc(ccc2o1)Cl BTB05722 c1cc(ncc1[N+](=O)[O-])NCCCCCO BTB05733 c1ccn(c1)c2ncc(s2)[N+](=O)[O-] BTB05772 Cc1nnc(s1)N/C=N/O BTB05816 CSC(=C(C#N)c1ccccc1)SC EN00061 c1ccc(cc1)C2(c3ccccc3C(=O)O2)c4ccccc4 EN00129 CCOc1ccsc1C(=O)NN GK02493 Cc1ccc(cc1NS(=O)(=O)C)NC(=O)Nc2ccc(cc2)C(F)(F)F HTS04606 CCOC(=O)c1cc(ccc1N2CCCCC2)NS(=O)(=O)c3ccc4c(c3)CCO4 HTS04640 CS(=O)(=O)/C(=C/Nc1cccnc1)/C#N KM01935 CCOC(=O)Cn1c(=O)c2ccsc2c3c1sc(c3C#N)SC KM01996 c1ccc(c(c1)NS(=O)(=O)c2ccc(cc2F)F)SCCS(=O)(=O)c3ccc(cc3)Cl KM02009 CCOC(=O)C1CCCN(C1)S(=O)(=O)c2cc(cs2)S(=O)(=O)c3ccccc3 HTS06914 Cc1c(nn(n1)c2ccccc2)C(=O)Nc3nc(cs3)c4ccc(c(c4)F)F HTS06926 Cc1c(nn(n1)c2ccccc2)C(=O)NNC(=O)c3cccc4c3cccc4 HTS07094 CCOC(=O)C1CCN(CC1)S(=O)(=O)c2ccc3ccccc3c2 HTS07102 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)NCc3ccc4c(c3)OCO4 HTS07184 COc1ccc(cc1)c2c(snn2)NC(=O)c3ccccc3CO HTS10917 CCOC(=O)c1cn2c(n1)ccc(n2)Oc3ccc(cc3)N4CCN(CC4)C(=O)C HTS10964 CC(=O)CSc1nc(sn1)SCC(=O)C CD08325 c1cc(c(c(c1)Cl)C#N)NCCc2ccc(cc2)Cl CD08344 c1cc(c(c(c1)Cl)CO/N=C(/CN2CCSCC2)\N)F CD08401 Cn1c(nnc1SCc2cc(cc3c2OCOC3)F)C(F)(F)F CD08467 Cc1cc(ccc1NC(=O)Nc2cccc(c2)Cl)C(C(=O)OC)(C(F)(F)F)O JFD02174 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2OC)C(C(=O)OCC)(C(F)(F)F)O JFD02188 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccccc1C)O JFD02268 COC(=O)C1=C(Oc2c(cc(cc2Br)Br)C1C(C#N)C(=O)OC)N FM00186 Cc1cc2nc(c(c(n2n1)N)C#N)SC KM02086 CS(=O)(=O)c1csc(c1Cl)C(=O)NCc2cccnc2 KM02102 Cc1c(c(sc1C(=O)OC)SC)c2ccn(n2)C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F KM02103 CC(=NOC(=O)c1c(c(cs1)S(=O)(=O)C)Cl)C KM02148 Cc1nccc(n1)c2cccc(c2)NC(=O)c3ccc(cc3)Cl KM02171 c1ccc(cc1)N/N=C(\C#N)/C(=O)C2CC2 KM02184 c1cc(cc(c1)S(=O)(=O)Nc2ccc(cc2)N3CCCCC3)C(F)(F)F HTS06985 c1cc(ccc1NS(=O)(=O)c2ccc(cc2F)F)N3CCCCC3 HTS06989 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)N3CCN(CC3)CCN4CCOCC4 HTS05174 CCOC(=O)N1CCC(CC1)NC(=O)Nc2cc(ccc2OC)Cl HTS05186 CC(C)(C)C(=O)NCc1c(cccc1Cl)Sc2ccc(cc2)Cl CD11895 CN(C)/C=C/C(=O)c1cccc(c1F)Cl CD11925 c1cc(c(cc1Cl)Cl)n2c(c(cn2)c3n[nH]nn3)N CD11935 c1cc(c(cc1OS(=O)(=O)c2ccc(c(c2)Cl)Cl)Cl)Cl CD08085 CC(C)(C)N(C(=O)C(Cl)(Cl)Cl)OC(=O)c1ccccc1 CD08165 c1ccc2c(c1)C/C(=C\c3ccc[nH]3)/C2=O FM00012 COc1c(c(c2c(n1)-c3ccccc3C2=O)c4cccs4)C#N FM00028 c1ccc\2c(c1)CC/C2=N\OS(=O)(=O)c3ccc(cc3)Cl FM00066 c1ccc(c(c1)NC(=O)c2cccs2)SCCS(=O)(=O)c3ccc(cc3)Cl KM02019 c1ccc(cc1)NC(=O)Nc2ccccc2SCCS(=O)(=O)c3ccc(cc3)Cl KM02023 COc1ccc(cc1)c2c(c(nc(n2)N)SC)C#N KM02060 c1ccnc(c1)S(=O)(=O)/C(=C/Nc2ccc(cn2)Cl)/C#N KM02207 Cc1nccc(n1)c2cccc(c2)NC(=O)Nc3ccccc3 KM02243 CCCS(=O)(=O)c1csc(c1Cl)C(=O)OC KM02318 CC(C)N(Cc1ccccc1)C(=O)c2ccc3c(c2)OCO3 HTS07189 COc1ccc(cc1OC)CCNC(=O)Nc2csc3c2cccc3 HTS07204 c1ccc(cc1)c2ccc(cc2)NCC(=O)Nc3ccc(cc3C(=O)c4ccccc4Cl)Cl HTS05298 Cc1ccc(cc1Cl)NC(=O)N2CCCN(CC2)c3c(cccn3)C#N HTS05329 c1ccc2c(c1)C(=O)N(C2=O)c3c(cccn3)OCc4ccc(c(c4)Cl)Cl HTS05377 CC1c2ccsc2CCN1S(=O)(=O)c3ccc(s3)Cl DFP00367 COc1cc(cc(c1OC)OC)/C=N/NC(=O)CC#N DP00076 COc1ccc(cc1)/C=N/NC(=O)CC#N DP00077 Cc1ccc(n1c2ccsc2COC(=O)Nc3c(onc3c4c(cccc4Cl)Cl)C)C CD08956 c1cc(cc(c1)Cl)NC(=O)C23CC4CC(C2)CC(C4)C3 CD09045 Cc1cc(cc2c1C(=O)/C(=C\c3cccnc3)/S2)Cl CD09065 CC\1=C2CCCC2CC/C1=N\NC(=O)N FM00216 CC\1=C2CCCC2CC/C1=N\Nc3nc(cs3)c4ccccc4 FM00223 C1C2CC3CC1CC(C2)C3=NNC(=S)N FM00224 c1cc(c(cc1c2n[nH]nn2)Cl)Cl GK02984 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2cc(c(cc2C)Cl)C GK03004 COC(=O)c1c(ccs1)NC(=O)CC(=O)Nc2ccsc2C(=O)OC GK00081 c1ccc(cc1)CN2CCN(CC2)c3ccc(cc3)NC(=O)Nc4ccc(cc4)C(F)(F)F HTS01158 CN1CCN(CC1)c2ccc(cc2)NC(=O)Nc3ccc(cc3)C(F)(F)F HTS01159 Cc1c(c(c(o1)C)S(=O)(=O)NCc2ccc(cc2)OC)C(=O)OC HTS01162 c1ccc2c(c1)cc(o2)C(=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS01199 CSc1c(cccn1)C(=O)NNc2cc(ccc2Cl)Cl HTS02916 Cn1cc(nc1)S(=O)(=O)NCc2c(cccc2Cl)Sc3ccc(cc3)Cl HTS05264 c1ccc(cc1)c2cnnn2c3cc(cc(c3)C(F)(F)F)C(F)(F)F CD04519 c1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4ccc(cc4)F HTS05430 c1ccc2c(c1)ccc(n2)NC(=O)c3ccco3 HTS05481 CCc1ccc(cc1)S(=O)(=O)Nc2cccc(c2)S(=O)(=O)N HTS05507 COC(=O)c1cccc(c1)NC(=S)NC(=O)c2ccccc2Cl DFP00278 COc1ccc(cc1)OCC(CNC2CCN(CC2)c3c4c(csc4ncn3)c5ccccc5)O AW00945 c1ccc(cc1)c2csc3c2c(ncn3)N4CCN(CC4)c5nccc(n5)C(F)(F)F AW00961 CC1CN(CC(O1)C)C(=O)c2cc3ccccc3oc2=O BTB04383 Cc1c(c(no1)c2ccccc2)C(=O)Nc3cc(ccc3Oc4ccccc4OC)C(F)(F)F BTB04415 Cc1cc(cc(c1Sc2ncc3n2cccc3)[N+](=O)[O-])[N+](=O)[O-] BTB04426 CC(C)S(=O)(=O)c1csc(c1Cl)C(=O)NN KM02381 CCOC(=O)c1cnc2c(c1NCc3ccco3)c(nn2C)C KM02387 c1ccc(cc1)c2csc(n2)NC(=O)c3cc(oc3C(F)(F)F)c4ccc(cc4)Cl HTS01314 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3ccncc3 HTS01317 c1ccc(cc1)CN2CCN(CC2)CCNC(=O)Nc3ccc(cc3F)F HTS03186 c1c(cc(cc1C(F)(F)F)N2C3(C4CC(C3N=N2)C5C4CCC5)N6CCOCC6)C(F)(F)F CD04653 c1ccc(cc1)c2c(nnn2c3ccc(cc3)[N+](=O)[O-])C(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F CD04666 c1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4cc(ccn4)C(F)(F)F HTS05678 CN1CCN(CC1)Cc2c[nH]nc2c3ccc(cc3)OC HTS05688 c1cc(ccc1S(=O)(=O)c2ccc(cc2[N+](=O)[O-])Cl)Cl CD05116 CCC(CC)(C#C)NC(=O)Nc1ccccc1 DP00746 c1ccc(cc1)/C/2=N/CCOC(=O)c3c2cccc3 DP00774 c1ccc(cc1)C(=O)NC(=S)Nc2nncs2 DP00858 CN(C)c1cccc(c1CN/C(=N\S(=O)(=O)c2ccccc2)/SC)N(C)C CD09806 c1cc(ccc1c2csc(=N)n2c3ccc(cc3Cl)Cl)Cl.Cl DP01088 Cc1ccc(cc1)/C(=N/NC(=S)NC)/C DP01127 CC1CCCN(C1)c2ccc3nncn3n2 GK00203 Cc1csc(c1C(=O)N)NC(=O)CSCC(=O)OC GK00214 CCOC(=O)c1c(csc1NC(=O)c2ccccc2Cl)C GK00235 Cn1c(ccn1)NS(=O)(=O)c2ccc(cc2Cl)F GK03381 CCC(C)Nc1c2c3c(sc2ncn1)CCCC3 GK03386 c1ccc2c(c1)nc(s2)/C(=C/c3ccc(cc3)Cl)/C#N GK00532 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)c3c(nccn3)C(=O)O HTS01413 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)F)NC(=O)Nc3ccc(cc3F)F HTS01418 Cn1c(c(c(n1)C(F)(F)F)c2cccc(c2)C(F)(F)F)NC(=O)Nc3cccc(c3)OC HTS01425 Cc1c(snn1)C(=O)NNc2ccccc2C(F)(F)F HTS03406 c1ccc(c(c1)C(F)(F)F)NNC(=O)c2cccs2 HTS03407 COCCCNC1=NC(=O)C(S1)CC(=O)Nc2cc(ccc2Cl)Cl CD04884 c1ccc(cc1)OCC(=O)Nc2c(cc(cc2F)Br)F CD04972 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OCC#C CD05290 c1cc(c(c(c1)Cl)CS(=O)(=O)c2ccc(cc2)Cl)F CD05336 CCOC(=O)c1c(c(sc1NC(=O)/C=C/C(=O)O)C)c2ccccc2 AW00967 c1cc(c(c(c1)Cl)/C=C\2/C(=O)NC(=S)S2)F BTB02087 c1ccc(cc1)c2csc3c2c(ncn3)N4CCCC4 AW01079 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCCN2CCN(CC2)Cc3c(cccc3Cl)F AW01120 CCOC(=O)C(=CNc1ccc(cc1)S(=O)(=O)c2ccc(cc2)NC=C(C(=O)OCC)C(=O)OCC)C(=O)OCC BTB06665 Cc1cc(ccc1N)/N=N/c2cccc(c2)C(F)(F)F BTB06669 CC(=O)N1CCN(CC1)c2ccc(cc2[N+](=O)[O-])C(F)(F)F BTB04710 COC(=O)/C=c\1/c(=O)n2c3ccccc3nc2s1 BTB04712 C/C(=N\Nc1c(cc(cc1Cl)Cl)Cl)/C=N/OC(=O)c2cc3ccccc3s2 BTB04742 Cc1c(c(no1)c2ccccc2)C(=O)Nc3ccc(c(c3)C(=O)OC)N4CCOCC4 HTS01358 COc1ccccc1NC(=O)NCCN2CCN(CC2)Cc3ccccc3 HTS03188 Cc1cc(=O)c2cc(ccc2s1)Cl HTS01507 CC1(c2ccccc2N3C1=CC4(C(c5ccccc5N4CC3=O)(C)C)C)C HTS01524 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc(cc3)C(=O)O)C(=O)OC HTS03553 COc1ccc(cc1)C(=O)/C=C(/c2ccccc2)\C(=O)c3ccccc3 CD05154 Cc1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C(=N/O)/C CD05200 Cc1c(snn1)C(=O)Nc2cccnc2 CD05417 Cc1c(snn1)C(=O)Nc2cccc(c2)Cl CD05493 Cc1c(c(on1)C)NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F CD05524 c1ccc2c(c1)cccc2/C=N/NC(=O)c3ccccc3N DP01139 c1ccc(c(c1)C(=O)N/N=C/c2cccc(c2)[N+](=O)[O-])N DP01146 c1ccc(c(c1)C(=O)NNC(=O)c2ccccc2N)N DP01161 COc1ccc(cc1OC)CCNC(=O)c2[nH]c(=O)c3ccccc3n2 DP01484 CC(=C(C#N)C#N)c1ccc(cc1)NC(=O)C DP01501 c1ccc(cc1)CNC(=N)c2ccc(cc2)Cl.I DP01658 Cn1ccc(n1)NC(=O)Nc2ccc(cc2)Cl GK00535 c1ccc(cc1)c2cc(c(s2)C(=O)N)NC(=O)c3ccco3 GK03728 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)C(=O)Nc4cc(cc(c4)Cl)Cl GK03762 c1csc(c1C#N)NC(=O)/C=C/C(=O)O GK03786 c1cc(ccc1Sc2c3c(ccs3)ncn2)Cl GK03790 c1cc(sc1)c2csc3c2c(=O)[nH]cn3 HAN00487 Cc1c(ccc(n1)C(F)(F)F)C(=O)Nc2nc3ccccc3c(=O)s2 HTS01620 c1cc2c(cc1CN3CCN(CC3)S(=O)(=O)c4cc(sc4Cl)Cl)OCO2 HTS03693 c1ccc2c(c1)cc(s2)NC(=O)NC3Cc4ccccc4C3 HTS03759 CC1=C(C(C2=C(N1)CCCC2=O)c3ccc4c(c3)OCO4)C(=O)OC HTS03817 c1ccc(cc1)NC(=O)N2CCN(CC2)c3ccc(cc3)F HTS05803 Cc1c(snn1)C(=O)NNC(=O)c2cccs2 CD05345 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)ONC(=O)c3ccc(cc3)F CD05372 c1cc(c(c(c1)Cl)C#N)NCc2ccc(cc2)Cl CD05691 c1cc(n(c1)c2ccc(cc2)Cl)/C=C(\C#N)/C(=O)O CD05694 c1ccc(c(c1)C2=NCCCN2)SCc3c(cccc3Cl)F.Br CD05711 c1ccc(cc1)C(c2ccccc2)(C(=O)NNC(=S)Nc3ccc(cc3)F)O BTB02300 CC(=O)c1c(c2cc(ccc2nc1O)Cl)c3ccccc3 BTB02345 c1cc(cc(c1)C(F)(F)F)C(=O)NCCCN2CCN(CC2)Cc3c(cccc3Cl)F AW01205 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)C2CCN(CC2)c3nccc(n3)C(F)(F)F AW01259 Cc1ccc(cc1)/C(=N\Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-])/CCC(=O)OC BLT00007 c1cc(c(cc1C2=CSC3=NCCN23)F)F.Br BTB07004 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Nc3cccc(c3)Cl BTB07052 Cc1cc(cc(c1Cl)C)Oc2cc(nc3c2cccc3)C BTB04992 c1ccc2c(c1)cc(s2)C(=O)Oc3ccccc3Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F BTB05050 c1ccc2c(c1)CCN2C(=O)NC(=O)c3c(cccc3Cl)Cl BTB05079 c1cc(cc(c1)NC(=S)NN)C(F)(F)F BTB05094 CC(C)(C)c1cc(n(n1)C)C(=O)NCc2ccc3c(c2)OCO3 HTS03590 Cc1ccc(cc1Cl)NNC(=O)c2c(noc2C)C HTS03640 Cc1cc(ccc1NNC(=O)c2ccc(cc2F)F)Cl HTS03648 c1cc(ccc1c2csnn2)OCC(CNCc3ccc4c(c3)OCO4)O HTS03850 Cn1cnc(c1Sc2ccc(cc2)F)[N+](=O)[O-] HTS03862 Cc1cc(ccc1NNC(=O)c2c(ccs2)Br)Cl HTS03872 Cc1cccc(c1F)CS(=O)(=O)c2ccc(cc2)Cl CD05592 Cc1c(snn1)c2nc(cs2)c3ccc(cc3)F.Br CD05595 Cc1cc(n(n1)c2cccc(c2C#N)Cl)C CD05681 c1ccc(cc1)c2c(nnn2c3ccc(cc3)[N+](=O)[O-])NC(=O)Nc4c(n(nn4)c5ccc(cc5)[N+](=O)[O-])c6ccccc6 CD05960 CC(C)NC(=O)NCc1c(cccc1Cl)F CD06056 c1cc(c(cc1Cl)Cl)/C=N/OCC(=O)NNC(=S)Nc2cc(ccc2Cl)Cl CD06082 c1cc(ccc1c2cn3c(n2)sc(n3)C(F)(F)F)Cl DP01671 c1ccc(cc1)CN2CCNC(C2=O)CC(=O)Nc3ccc(cc3)Cl DP01686 c1ccc(cc1)S(=O)(=O)c2ccc(cc2Cl)N DP01992 c1ccc(c(c1)/C=N/c2ccc(cc2Br)F)O DP02018 CCOC(=O)c1c(c2cc(ccc2s1)NC(=O)C)C DP02038 CCCN(CCC)C(=S)NC(=O)c1cccc(c1)[N+](=O)[O-] HR00030 COc1ccc(cc1OC)CCNC(=S)NC2CC3CCC2C3 HR00060 CCCN(CCC)C(=S)NC1CC2CC1C=C2 HR00086 c1cc(c(cc1/C=N/N=C/2\c3cc(ccc3NC2=O)Br)Cl)Cl HR00125 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCc3nc(no3)c4ccc(cc4)C(F)(F)F HTS00081 c1cc2c(cc1CNS(=O)(=O)c3ccc4c(c3)OCC4)OCO2 HTS03974 c1cc(cc(c1)NC(=O)Nc2cccc(c2)Cl)C(=O)O HTS03990 CC(C)(CC(=O)N1CCCN(CC1)c2nccc(n2)C(F)(F)F)CC(=O)O HTS03991 c1cc2c(cc1S(=O)(=O)N3CCCN(CC3)c4nccc(n4)C(F)(F)F)CCO2 HTS03998 Cc1cc(c(nc1)NC(=O)c2ccccc2)Br HTS04001 CCOC(=O)/C(=N/OC(=O)c1c(onc1c2c(cccc2Cl)Cl)C)/C#N CD05950 c1cc(sc1)CNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD05987 CS/C(=N\c1ccccc1F)/Nc2ccccc2F.I CD06207 c1cc(cc(c1)Cl)C(=O)NNC(=O)CO/N=C/c2ccc(cc2Cl)Cl CD06211 CCc1cccc(c1NS(=O)(=O)c2ccc(cc2)C)C(C)C CD06411 CCOC(=S)SCc1ccccc1C(=O)Oc2c(cccc2Cl)Cl CD06438 CC(=O)c1cc(cc(c1OC(=O)c2cccc(c2)C(F)(F)F)Cl)Cl BLT00267 Cc1nc2c(cc(cc2Br)Br)c(=O)n1c3ccc(cc3)F BTB02535 C/C(=N\N=C(\c1cc2c(cc1)cccc2)/C)/c3cc4c(cc3)cccc4 BTB00227 COc1cc(ccc1OC(=O)c2ccccc2)/C=N/Nc3ccccc3 BTB00287 COc1cc(cc(c1OC)OC)/C=N/NC(=O)c2cccnc2 BTB00360 c1cc(cnc1)C(=O)N/N=C/c2ccco2 BTB00364 c1ccn2c(c1)c(nc2SCc3ccc(cc3)Cl)C(=O)C(F)(F)F BTB05099 Cc1cccc(n1)NC(=O)c2ccc(cc2[N+](=O)[O-])Cl BTB07298 c1cc(ccc1c2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-])Oc4ccc(cn4)[N+](=O)[O-] BTB05223 CCc1c(nc2cc(c(cc2n1)C)C)CC BTB05241 c1cc(c(cc1NC(=O)Cc2ncon2)Cl)F BTB05259 COC(=O)c1c(c2ccccc2s1)OC(=O)c3cccs3 BTB05277 CCc1ccc(cc1)C(=O)NNc2ccc(cc2)C(C)C HTS03879 CC(C)(CC(=O)NCc1csc2c1cc(cc2)Cl)CC(=O)O HTS03890 COc1ccc(cc1)Cc2cc(n[nH]c2=O)c3ccc(cc3)F HTS03960 Cc1ccsc1CNS(=O)(=O)c2ccc3c(c2)CCO3 HTS04017 Cc1nc(cn1C)S(=O)(=O)Nc2ccc(cc2)n3c(cc(n3)C(F)(F)F)c4cccs4 HTS04039 COc1ccc(cc1)C(=O)Nc2ccc(cc2)CN3CCS(=O)(=O)CC3 HTS04106 Cc1c(c(c(c(c1C)C)/C=C/2\c3ccccc3NC2=O)C)C CD06091 Cc1c(c(c(c(c1C)C)S(=O)(=O)NCCCN2CCOCC2)C)C CD06139 c1cc(sc1)C(=O)C2CCCCC2 CD06156 c1ccc(c(c1)C(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)F CD06864 c1cc(c(cc1Br)C(=O)NCCc2ccncc2)O CD06865 c1ccn(c1)c2cccc(c2C#N)Cl CD06868 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3ccccc3C(=O)C CD06876 Cc1c(c(c(c(c1NC(=O)c2c(onc2c3ccccc3Cl)C)C)C)NC(=O)c4c(onc4c5ccccc5Cl)C)C DSHS00154 Cc1c(c(sc1c2ccc(c(c2)OC)OC)/N=C/c3cc(cc(c3O)Br)Br)C#N DSHS00322 c1ccc(cc1)CNC(C#N)c2ccc(c(c2)Cl)Cl DSHS00561 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3ccc(cc3)[N+](=O)[O-])Cl DSHS00643 c1ccc(cc1)C(=O)c2cc(ccc2NC(=O)c3ccco3)Cl DSHS00648 c1c(cc(cc1Cl)Cl)NC(=O)CC(=O)Nc2cc(cc(c2)Cl)Cl HTS00098 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)c4cc(cc(c4)Cl)Cl HTS00110 CCc1ccc(cc1)S(=O)(=O)Nc2cc(c(cc2OCC)N3CCOCC3)OCC HTS00112 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)C4CCC4 HTS00116 c1cc(ccc1c2nc(on2)CSc3nncn3c4ccc(cc4)C(F)(F)F)C5SCCS5 HTS00214 c1cc(ccc1C(=O)NCc2ccc(s2)S(=O)(=O)NCc3cc(cc4c3OCOC4)F)Cl HTS04162 c1cc(ccc1S(=O)(=O)NCc2csc3c2cc(cc3)Cl)Cl HTS04203 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)NCc3csc4c3cc(cc4)Cl HTS04204 c1cc(ccc1N2C(=O)CCC2=O)S(=O)(=O)Nc3ccc4c(c3)C(=O)OC4 HTS04219 COc1ccc(cc1OC)C(=O)NCc2csc3c2cc(cc3)Cl HTS04228 CCOC(=O)CSC(=O)NC(=O)c1c(nns1)C CD06715 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(C)(C)C CD06797 c1ccc(cc1)c2cc(n(n2)CCC#N)NS(=O)(=O)c3ccc(c(c3)Cl)Cl CD06933 c1cc(c(cc1/N=C\2/NC(CS2)(CO)CO)Cl)F CD07012 CCOC(=O)NCc1c(cccc1Cl)Cl CD07039 c1ccc(c(c1)C(=O)NCc2c(cccc2Cl)Cl)N CD07143 c1ccc(cc1)C(C(=O)c2ccc(cc2)Cl)Sc3ccc(cc3)Cl BTB02889 c1ccn(c1)c2cccc(c2)c3nc(on3)c4cccs4 BTB02910 Cc1ccc(c(c1)[N+](=O)[O-])NC(=O)C BTB00582 COc1nc(nc(n1)OC)Nc2cccc(c2)C(F)(F)F BTB00587 COc1ccc(cc1)NC(=O)/C=N/O BTB00634 c1cc(sc1)C(SCC(=O)O)SCC(=O)O BTB00636 Cc1nc2cc(ccc2c(=O)n1c3ccc(cc3)F)Cl BTB00700 CN(C)/C=N/c1cc(c(cc1Oc2ccc(cc2)Cl)n3cccc3)Cl BTB07557 COc1ccc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC)[N+](=O)[O-] BTB07575 CC(=O)C(=CNc1c(cc(c(c1OC)OC)OC)C(=O)OC)C(=O)C BTB05447 c1ccc2c(c1)c(=O)oc(n2)c3ccc(o3)[N+](=O)[O-] BTB05483 c1ccc(cc1)Oc2c(cccn2)C(=O)O/N=C(/c3ccc(cc3)Oc4ccc(cc4[N+](=O)[O-])C(F)(F)F)\N BTB05537 c1cc2c(cc1CN3CCN(CC3)C(=O)CSCC(=O)O)OCO2 HTS04128 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS04165 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)COCC(=O)O HTS04273 Cc1c(cnn1c2ccc(cc2)OC)C(=O)NCc3c(cccc3Cl)Oc4ccccc4 HTS04307 c1ccc(cc1)NC(=O)NCc2c(cccc2Cl)Oc3ccccc3 HTS04315 CSc1cccc(c1)NC(=O)c2ccccc2F CD06912 CCN1CCCC1CNC(=O)c2c(onc2c3c(cccc3Cl)Cl)C CD06940 COc1ccc(cc1)Oc2cccc(c2C#N)Cl CD11650 Cc1cc(cc(n1)n2c(c(cn2)/C(=N/OC(=O)c3ccc(cc3)Cl)/C)C)C(F)(F)F CD11715 Cc1c(sc(n1)c2ccc(cc2F)F)C(=O)C CD11788 c1c(c(cc(c1Cl)Cl)Cl)S(=O)(=O)N2CCCCC2 DSHS00683 COc1cc(c(cc1Cl)OC)NC(=O)/C=C/c2ccccc2Cl DSHS00700 COc1ccc(cc1)C(=O)CSc2nnc3n2CCCN3C(=O)c4cccc(c4)[N+](=O)[O-] HTS12774 CC(=O)CSc1nnc2n1c3ccccc3s2 HTS12806 c1c(cnc(c1C(F)(F)F)N)C(F)(F)F HTS12821 Cc1nc(cs1)c2nnc(n2C)SCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS00220 c1ccc(cc1)C(=O)NCc2ccc(s2)S(=O)(=O)N3CCN=C(C=C3)C(F)(F)F HTS00234 CN(c1nc(cs1)c2ccc(s2)Cl)C(=O)C3CCC3C(=O)O HTS00260 CCCCCCCCOc1ccc(cc1)C(=O)O JFD03911 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(cc3OC)OCc4ccccc4)C(=O)OC HTS04348 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc4c(c3)CCC(O4)(C)C)C(=O)OC HTS04350 c1ccc2c(c1)CC(C2)NCC(=O)Nc3ccc(cc3C(=O)c4ccccc4Cl)Cl HTS04394 Cc1cc(n(n1)C)NC(=O)CCCC(=O)O HTS04438 CC(C)Cc1ccc(cc1)C(=O)C(C)Sc2nnc(n2C)c3ccc4ccccc4c3 HTS04518 Cn1c(ccn1)c2cc(cc(c2O)Cl)Cl CD07342 COCCCNc1ccc(c(c1C#N)NCCCOC)[N+](=O)[O-] CD07396 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3ccccc3 HTS08499 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3ccccc3C(=O)O HTS08512 c1ccc(cc1)Oc2c(cccn2)c3nnc(s3)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F BTB03137 Cc1ccc(cc1)S(=O)(=O)CC(=O)C BTB00889 c1cc(sc1)C(=O)NCCc2ccncc2 BTB03434 Cc1ccc(cc1)SCC(=O)NCc2cccs2 BTB03459 c1cc(c(cc1[N+](=O)[O-])c2nnc(o2)c3ccc(cc3Cl)Cl)Oc4cc(cnc4)Cl BTB08057 c1cc(ccc1/C=C\2/C(=O)NC(=O)N2)OC(=O)c3ccc(cc3)Cl BTB08072 c1c(cc(cc1Cl)Cl)NC(=O)Cc2n[nH]nn2 BTB05820 c1ccc2c(c1)cc(c(=O)o2)C(=O)NCC3CC3 BTB05873 c1cc(c(cc1F)F)S(=O)(=O)NCC2CC2 BTB05880 c1ccc(c(c1)NC(=O)NCC2CC2)F BTB05893 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccc(o3)CN4C(=O)c5ccccc5C4=O)C(=O)OC HTS04321 c1ccc(c(c1)C(=O)NCCCN2CCOCC2)NC(=O)c3ccc(cc3)F HTS06333 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccc(cc3)c4cn5c(n4)SCC5 HTS06795 Cc1nc(cn1C)S(=O)(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS06798 CCOc1ccccc1N2CCN(CC2)C(=O)c3cc4c(cc(cc4[nH]3)C)C HTS06810 c1cc(c(c(c1)F)C#N)N2CCC(CC2)C#N CD11791 c1ccc(cc1)NC(=O)NCc2c(cccc2Sc3ccc(cc3)Cl)F CD11846 CC(c1ccccc1)n2c(nnc2SCC(=O)c3ccc4c(c3)OCCO4)OC(=O)N(C)C HTS08654 Cc1c(snn1)c2nnc(n2C3CC3)SCC(=O)c4ccc(cc4)F HTS08684 CC(=O)N1CCN(CC1)c2ccc(cc2)OC(=O)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl HTS08755 CCOC(=O)N1CCc2c(sc3c2c(=O)[nH]cn3)C1 HTS12870 Cc1nc2c(cnn2c3ccccc3)c(=O)o1 HTS12935 c1ccc(cc1)NC(=O)NC(=O)Cn2c(=O)c(=O)n3c4ccccc4sc3n2 HTS12989 CCOC(=O)/C(=C/c1ccc2c(c1)OCO2)/C#N JA00060 CCOC(=O)/C(=C/c1ccc(c(c1)OC)OCc2ccccc2)/C#N JA00075 Cc1ccc2c(cc(nc2c1)c3cccc(c3)[N+](=O)[O-])C(=O)O JA00103 Cc1ccncc1S(=O)(=O)O JFD03918 CC[n+]1c(ccc2c1cccc2)C.[I-] JFD03940 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2ccc(c3)[N+](=O)[O-] JFD03948 c1cc(cc(c1)[N+](=O)[O-])NC(=O)C(C(=O)Nc2cccc(c2)[N+](=O)[O-])C34CC5CC(C3)CC(C5)C4 JFD03971 c1cc(oc1C(=O)Oc2c(cc(cc2Br)C#N)Br)Br JFD03977 Cn1c(nnc1SC)c2cccs2 KM04555 Cn1c(nnc1SC)c2cc(sc2)S(=O)(=O)Nc3cccc(c3)C(F)(F)F KM04606 CN(C)n1cccc1/C=C(\C#N)/S(=O)(=O)C KM04609 CO/N=C/1\CCCc2c1c(sc2C(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F)SC KM04632 Cc1c(sc2c1C(=C(S(=O)(=O)N2C)C(=O)Nc3ccccc3)O)C KM04707 CS(=O)(=O)c1cc2ccccc2oc1=O KM04867 c1cc2c(cc1C(=O)CSc3nnc(n3C4CC4)O)OCCO2 HTS08641 CC(c1ccccc1)n2c(nnc2SCC(=O)c3cc(no3)c4ccccc4)O HTS08648 c1ccc2c(c1)cccc2C(=O)NNC(=O)c3ccc4c(c3)OCO4 HTS08786 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3cc(nn3Cc4ccccc4)C(C)(C)C)C HTS08818 CC(=O)Nc1ccc(cc1)NS(=O)(=O)c2cn(cn2)C HTS08942 CN1C(c2cc(ccc2OC1=O)Cl)O BTB03510 CCOC(=O)c1cc(c(c(c1)Cl)NC(=O)c2ccc(cc2)[N+](=O)[O-])Cl BTB03530 CSc1cc(nn1C(=O)c2ccccc2)c3ccc(cc3)Oc4ccccc4 CD11991 c1ccnc(c1)N/N=C/c2cc(sc2)[N+](=O)[O-] DFP00004 c1cc(cc(c1)Cl)NC(=O)c2cc(sc2)[N+](=O)[O-] DFP00057 Cc1ccc(c(c1)C)NC(=S)NCc2cccnc2 DSHS01293 Cc1cc(cc(c1OCC(=O)NNC(=O)c2cccc(c2)C(F)(F)F)C)c3c4ccccc4c(=O)n(n3)C BTB08309 COC(=O)COc1ccc(cc1)SC(F)(F)F BTB08346 COc1c(csc1C(=O)NNC(=O)c2cccc(c2)[N+](=O)[O-])Br GK02585 c1ccc(cc1)C(c2ccccc2)N3CCN(CC3)C(=O)c4cccs4 HTS00647 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)OCC)C1=O HTS06835 Cc1cc2ncc(c(n2n1)C)c3ccnc(n3)SCCS(=O)(=O)c4ccccc4 KM04765 c1ccc(cc1)N/N=C(\C#N)/C(=O)c2ccccc2OC(F)(F)F KM04879 COC(=O)c1c(c2cccnc2s1)N KM05066 c1ccc(cc1)Oc2ccc(cc2)NC(=O)Nc3cccs3 HTS08760 CN(CCc1ccccn1)C(=O)Nc2cc(cc(c2)Cl)Cl HTS08776 Cn1c(nnc1SCC(=O)NNC(=O)Nc2ccccc2)c3ccccc3 HTS09019 Cc1cc(=O)n2c(n1CC(=O)N/N=C/c3ccc(cc3)Cl)ncn2 HTS09030 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccc(cc3)Cl)c4ccccc4)NC(=O)Nc5ccc(c(c5)Cl)Cl HTS09041 c1ccc(c(c1)/C=N/N=C/2\c3ccccc3NC2=O)Cl JA00122 CCOc1ccc(cc1)NC(=O)/C=N/O JA00162 CCOC(=O)/C(=C(/NCC=C)\SCC(=O)c1ccccc1)/C#N DP00143 Cc1cccc(c1NC(=O)CC#N)Cl DP00171 CC1CCCN(C1)S(=O)(=O)c2cc(ccc2Cl)Cl DP00322 COC(=O)c1ccc(o1)Oc2ccc(c(c2)Cl)Cl JM00077 CNC(=O)NNC(=O)c1ccccc1 JM00238 CC1(N=C(N=C(N1c2ccc(cc2)Cl)N)N)C.Cl JM00274 Cc1c2cccc(c2nc(c1Cl)O)Cl JM00482 c1ccc(c(c1)NC(=O)c2ccc(cc2Cl)Cl)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F JP00468 Cc1ccc(cc1)S(=N/C=C/2\C(=O)c3c(ccs3)N(S2(=O)=O)C)(=O)C KM05133 COc1ccc(cc1)NC=C2C(=O)CC(CC2=O)c3cccs3 KM05152 c1cc(cnc1)c2ncc(c(n2)N)S(=O)(=O)c3ccc(cn3)C(F)(F)F KM05158 CC1(CCc2cc(ccc2O1)/C=N/OC(=O)c3ccc(cc3)Cl)C KM05219 c1ccc(cc1)Oc2cccc(c2)c3[nH]c4ccccc4c(=O)n3 HTS02969 c1ccc(cc1)n2c3c(cn2)c(=O)n(nn3)/N=C/c4ccc(cc4)[N+](=O)[O-] HTS08983 c1ccc(cc1)c2c3c(c(sc3nnc2c4ccccc4)C(=O)N/N=C/c5ccc(cc5)[N+](=O)[O-])N HTS08990 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)Nc2cccnc2)C CD04575 Cc1cc(ccc1NCN2C(=O)CCC2=O)Cl CD04594 c1ccc(cc1)c2c(nnn2c3cc(cc(c3)C(F)(F)F)C(F)(F)F)C(=O)Nc4ccccc4 CD04597 Cc1c(c(n(n1)C)NCc2cccs2)[N+](=O)[O-] EN00018 CS/C(=N/C(=O)c1c(cccc1Cl)Cl)/NCCSCc2c(cccc2Cl)Cl EN00056 CC(C)(C)c1ccc(cc1)C(=O)NC(=S)Nc2cccc(c2)C(=O)OC DFP00280 COC(=O)c1cccc(c1)NC(=S)Nc2ccccc2C(F)(F)F DFP00320 CC1c2ccsc2CCN1S(=O)(=O)c3ccccc3 DFP00360 Cc1nc(cs1)c2ccc(s2)S(=O)(=O)N3CCN(CC3)C(c4ccccc4)c5ccccc5 HTS00661 COc1ccccc1NC(=O)N2CCN(CC2)C(c3ccccc3)c4ccccc4 HTS00666 CCOC(=O)c1cnc(nc1C(F)(F)F)Nc2ccc(cc2)F GK02949 CCOC(=O)c1cnc(nc1C(F)(F)F)NNS(=O)(=O)c2ccc(cc2)OC GK02971 CSc1c2c(c(s1)C(=O)/C(=N/Nc3cccc(c3)C(F)(F)F)/C#N)CCC=C2 KM05067 CSc1c2c(c(s1)C(=O)/C(=C/c3ccc(cc3)Cl)/C#N)CCC=C2 KM05231 CC1(Cc2c(c(sc2C(=O)OC)SCCOC(=O)c3cccc(c3)C(F)(F)F)C(=O)C1)C KM05238 CC1(Cc2c(c(sc2C(=O)OC)SCCOC(=O)Nc3ccc(cc3)OC(F)(F)F)C(=O)C1)C KM05244 CS(=NC(=O)NC(=O)c1ccc(cc1)Cl)(=O)c2ccc(cn2)C(F)(F)F KM05572 COc1ccc(cc1)NS(=O)(=O)c2ccc(s2)S(=O)(=O)c3c(cc(cn3)C(F)(F)F)Cl KM05576 Cc1cc(no1)NS(=O)(=O)c2ccc(s2)S(=O)(=O)c3c(cc(cn3)C(F)(F)F)Cl KM05703 CSc1c(c(c(s1)c2ccnc(n2)SCCS(=O)(=O)C)c3ccccc3)C#N KM05762 c1cc2c(cc1c3cc(n4c(n3)cc(n4)C5CC5)C(F)(F)F)CCC2 KM10522 COC(=O)c1ccc2c(c1)nnn2C3CCN(CC3)Cc4ccccc4 KM10572 CC(C)(C)OC(=O)NCc1nnc(n1C)SCC(=O)N2CCOCC2 KM10618 Cc1ccc(cc1NC(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5)F HTS09207 CCCc1cnc(nc1)N2CCN(CC2)C(=O)Nc3ccc(cc3)F HTS09256 c1ccc(cc1)c2cn3ccccc3n2 JFD00397 Cc1c(ncnc1OC)OC JFD02419 c1ccc(cc1)N2C3=C(CCCC3)CCC2=O JFD00499 C1CCc2c(c(c(s2)N)C#N)C1 JFD00504 c1cc(cnc1)C(=O)NCn2cncn2 JFD00507 c1cc(ccc1C(=O)c2ccc3c(c2)CCC3)/N=C/c4cc(cc(c4O)Cl)Cl JPV00032 Cc1cc(nc2n1nc(c2)c3ccc(cc3)Cl)C(F)(F)F KM02445 c1ccc(cc1)SCCS(=O)(=O)c2ccc(cc2)Cl KM00071 Cc1ccc(cc1)S(=O)(=O)CCS(=O)(=O)c2ccc(cc2)Cl KM00079 Cc1cc(n(n1)C(C)(C)C)NC(=O)c2ccccc2 KM00089 c1ccc(cc1)C(=O)/C(=C/N2CCc3c2cccc3)/C#N KM05386 c1ccc(cc1)S(=O)(=O)C(=C2SCCCCS2)C#N KM05411 COc1ccc(cc1)Oc2c(ccs2)[N+](=O)[O-] KM05487 CC(=O)Nc1ccc(cc1)Br KM05555 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccsc3)C HTS07241 CC1(CCc2cc(ccc2O1)c3ccnc(n3)SCc4ccc(cc4)Cl)C KM05849 Cc1c2cc(ccc2sc1C(=O)CSc3nnc(n3C4CC4)O)Cl HTS09143 CC(C)(C)c1ccc(cc1)c2nc(on2)CSc3nnc(n3C4CC4)O HTS09144 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)Nc5cccc(c5)C(F)(F)F HTS09198 Cc1ccc(cc1)Cn2c3c(nc2Oc4ccc(cc4Cl)Cl)n(c(=O)n(c3=O)C)C HTS11219 Cc1ccc(cc1)n2c(nnn2)c3cn[nH]c3c4ccc(cc4)C(F)(F)F HTS09298 Cc1c(sc(n1)N/N=C/2\CCCc3c2cccc3)C FM00245 c1ccc(c(c1)CSc2[nH]c3ccccc3n2)Cl.Cl DP01070 c1cc(ccc1c2csc(=N)n2c3ccc(c(c3)Cl)Cl)Cl.Cl DP01085 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2nnc(o2)N3CCCC3 GK00256 Cc1c(c(n(n1)CC/C(=N/OC(=O)c2cc(cc(c2)Cl)Cl)/N)C)Oc3ccc(cc3)Cl HTS01502 Cn1c2ccccc2c(n1)NC(=O)CC34CC5CC(C3)CC(C5)C4 HTS01641 Cc1cc(nc2c1c3c(s2)c(=O)sc(n3)NC(=O)c4ccc(nc4C)C(F)(F)F)C HTS01654 Cc1c(snn1)C(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl HTS01671 COc1ccc(cc1)C(=O)/C(=C/N=S(=O)(C)c2ccc(cn2)C(F)(F)F)/C#N KM05816 CC(C)CSc1nnc(n1C)CSCc2nc(cs2)c3ccc(cc3)Cl KM05978 COc1ccccc1C(=O)N=S2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl KM06038 COc1ccccc1C(=O)N=S2CCN(CC2)S(=O)(=O)c3ccc(cc3)Cl KM06055 Cc1cnn2c1ncc3c2-c4ccccc4C3=O HTS09273 c1ccc(cc1)C(=O)c2cc(ccc2N/C=C/c3nnnn3c4ccc(cc4)F)Cl HTS09289 c1cc(ccc1c2c(cn[nH]2)c3nnnn3c4ccc(cc4)Cl)F HTS09295 Cc1ccc(c2c1CCC2)Oc3c(cccn3)NC(=O)CC(CC(=O)O)c4ccccc4 HTS09497 c1cc(sc1)CNC(=O)c2ccc3c(c2)nccn3 HTS09581 CC(=O)OC[C@@H]([C@H]([C@H]([C@@H](c1[nH]nnn1)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00520 Cc1c2ccccc2ncc1c3nnnn3c4ccc(cc4)I JFD00600 CCOC(=O)C(c1c2ccccc2n(c(=O)c1[N+](=O)[O-])c3ccccc3)C(=O)C JFD00853 Cc1cc(n(n1)c2ccccc2)NC(=O)c3cc(cc(c3)Cl)Cl KM00188 c1ccc(cc1)C(CS(=O)(=O)c2ccc(cc2)Cl)N3CCCCC3 KM00198 Cc1ccc(cc1)/C=C(\C#N)/C(=O)C2CC2 KM00333 c1cc(cc(c1)Cl)/C=C(\C#N)/C(=O)C2CC2 KM00334 CN(C)c1ccc(cc1)/C=C(\C#N)/C(=O)C2CC2 KM00335 c1ccc(cc1)c2csc(n2)CSCC(=O)NN KM05922 c1cc(ccc1/C=C(\C#N)/C(=O)C2CC2)O KM05952 C/C(=N\OCC(=O)Nc1ccc(cc1)OC(F)(F)F)/c2ccc(cc2)Cl KM05958 c1ccc(c(c1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)OCc3c(cccc3Cl)Cl KM05968 CS(=O)(=O)/C(=C/c1ccccc1OCc2c(cccc2Cl)Cl)/C#N KM05969 c1ccnc(c1)CNC(=O)c2cccnc2SCCS(=O)(=O)c3ccc(cn3)C(F)(F)F KM06188 c1cc(oc1)Cn2c(nnc2SCC(=O)c3ccc(cc3)C#N)O HTS09454 c1cc(oc1)Cn2c(nnc2SCC(=O)c3ccc4c(c3)OCCCO4)O HTS09460 Cc1c(sc(n1)Nc2ccccc2)C(=O)c3cc4ccccc4s3 HTS09478 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3)C#N HTS09695 CCOC(=O)c1c(csc1NC(=O)CC#N)C GK00564 CSc1cc(nc(c1)c2cccs2)c3ccc(cc3)Cl GK00591 CC(=O)c1c(cc(s1)c2ccc(cc2)Cl)NC(=O)C(Cl)(Cl)Cl GK00644 Cn1cc(c(n1)C(F)(F)F)C(=O)O/N=C/c2c(cccc2Cl)F GK00820 c1cc(ccc1n2c(nnn2)SCC(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)O HTS01669 Cc1c(c(c(o1)C)S(=O)(=O)NCc2ccc(cc2)Cl)C(=O)OC HTS01714 c1ccc(cc1)c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc4c(c3)OCO4 HTS01798 c1ccc(cc1)CCN2CCCN(CC2)S(=O)(=O)c3cccs3 HTS01802 Cc1nc(cn1C(C)C(=O)c2ccc(cc2)c3ccccc3F)[N+](=O)[O-] HTS01861 CCOC(=O)c1c2c(c(s1)/S(=N/C(=O)Nc3ccccc3Cl)/C)C=CCC2 KM06073 CSc1ccc(cc1)OC(=O)Nc2ccccc2 KM06347 c1c2c(cc(c1Cl)Cl)nsn2 KM06366 c1cc(ccc1Sc2c(nccn2)/C(=N\O)/N)Cl KM06392 CC(=O)Nc1ccc(cc1[N+](=O)[O-])Br KM06404 Cc1c(c(n(n1)Cc2cccc(c2)C(=O)O/N=C(/c3ccc(cc3)Cl)\N)C)Br KM06408 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3cccc(c3)C(F)(F)F HTS09631 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)Nc3cccc(c3Cl)Cl HTS09635 c1ccc(cc1)n2c(nnc2SCC(=O)NN)c3ccncc3 HTS09851 CC1CCc2c(sc3c2c(ncn3)SCC(=O)N/N=C/c4ccc(cc4)OCc5ccccc5)C1 HTS09854 c1ccc2c(c1)NC(S2)[C@@H]([C@H]([C@H](CO)O)O)O JFD00891 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC([C@H](COC(=O)C)OC(=O)C)[C@H]([C@@H](C#N)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00925 Cc1cccc(c1)C(=O)C2=NNCC2c3ccc(cc3)Cl JFD01090 CC(/C=C/c1cccc[n+]1C)O.[I-] JFD01143 c1cc(c(cc1c2ccc(c(c2)[N+](=O)[O-])N)[N+](=O)[O-])N JFD01175 Cc1cc(n2c(n1)cc(n2)c3ccc(cc3)C(C)(C)C)C KM00338 CC(C)(C)c1ccc(cc1)c2cc3[nH]c(cc(=O)n3n2)c4ccccc4 KM00348 c1ccc(cc1)c2cc([nH]n2)NC(=O)c3ccccc3 KM00359 c1cc(ccc1N/N=C(\C#N)/C(=O)C2CC2)Br KM00382 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2ccc(cc2)Cl KM00549 c1ccc(cc1)OC(=O)c2ccc(o2)CSc3ccc(cn3)C(F)(F)F KM06313 CC(=O)N1CSCC1C(=O)NNS(=O)(=O)c2cccc(c2)C(F)(F)F KM06316 Cc1cc(c(c(c1)C)S(=O)(=O)O)C.CS(=N)(=O)c1ccc(cc1)OC(=O)c2ccc(cc2)Cl KM06334 CS(=NS(=O)(=O)c1cccs1)(=O)c2ccc(cc2)OC(=O)c3ccc(cc3)Cl KM06561 Cc1c(c(no1)c2c(cccc2Cl)F)c3nnc(o3)c4cccc5c4cccc5 HTS09761 Cn1c2c(nc1N/N=C/c3cccs3)n(c(=O)n(c2=O)Cc4ccccc4)C HTS09821 CN1CCN(CC1)c2nc3c(=O)[nH]c(nc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09823 CCNc1c2c3c(sc2nc(n1)SCc4ccc(cc4)[N+](=O)[O-])CC(CC3)C HTS09841 Cc1nc2c(c(n1)N3CCN(CC3)C)sc(=S)n2c4ccccc4 HTS09903 Cc1csc(c1NC(=O)CN2CCCCC2)C(=O)OC GK01335 C1CCc2c(c(c(s2)N3C(=O)CCC3=O)C#N)C1 GK01346 Cc1csc(c1Cl)NC(=O)Nc2ccc(cc2)C(F)(F)F GK01359 COc1ccc(cc1)C(=O)Nc2ccc3c(c2)OCCO3 HTS01866 c1cc(cnc1)CNC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl HTS01875 Cc1ccsc1CNC(=O)Nc2ccccc2 HTS04012 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)Nc2cc(ccc2OC)Cl HTS02040 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCC(=O)c5ccc(cc5)c6ccccc6 HTS02046 Cn1c(nnc1SCc2ccc(cc2Cl)Cl)CSCCOc3ccccc3 KM06508 c1cc(c(c2c1nsn2)[N+](=O)[O-])N3CCOCC3 KM06731 CS(=N/C=C(\C#N)/C(=O)c1ccco1)(=O)c2ccc(cc2)Oc3ccc(cn3)[N+](=O)[O-] KM06756 c1ccc2c(c1)OCC(O2)c3nc(cs3)c4ccc(cc4)Cl KM06769 CSc1nc2ccccc2s1 KM06784 c1cc(c(c2c1nsn2)[N+](=O)[O-])SCCO KM06791 Cc1[nH]c(=O)c2c(n1)Oc3c4ccccc4oc(=O)c3C2c5ccccc5Cl HTS09878 CCOC(=O)c1c(=O)n(c(=S)n(c1S)c2ccccc2)c3ccccc3 HTS09888 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)/C=N/NC(=S)N HTS09898 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)NNC(=O)Nc4ccc(cc4)Cl)C#N HTS09973 c1ccc(cc1)NC(=O)N2CCCn3c2nnc3SCC(=O)c4ccc(cc4)[N+](=O)[O-] HTS09977 c1ccc(cc1)C(C#CC(c2ccccc2)(c3ccccc3)O)(c4ccccc4)O JFD01265 c1ccc(cc1)c2c(c(sc2c3ccccc3)c4ccccc4)c5ccccc5 JFD01272 CN(C)c1ccc(cc1)C(=S)c2ccc(cc2)N(C)C JFD01489 c1ccc(cc1)/C(=N\O)/c2ccccn2 JFD01559 Cn1c2ccccc2c\3c1CCC/C3=N\OC(=O)c4cccc(c4)C(F)(F)F JFD01618 c1cc(ccc1F)S(=O)(=O)CCS(=O)(=O)c2ccc(cc2)Cl KM00574 COc1c(csc1Cl)C(=O)O/N=C(/c2cccs2)\N KM00614 c1ccc(c(c1)c2nc(no2)c3cccc(c3)CS(=O)(=O)c4ccc(cc4)Cl)Cl KM00643 c1cc(oc1)C(=O)C(=C2SCCCS2)C#N KM00824 Cc1cc2nc(nc(n2n1)N)SC KM00833 c1cc2c(c(c1)S(=O)(=O)Nc3ccc(cc3)OC(F)(F)F)non2 KM06573 C/C(=N/OC(=O)c1ccccc1)/c2ccc3c(c2)CCO3 KM06619 Cc1ccccc1NC(=O)O/N=C(/C)\c2ccc3c(c2)CCO3 KM06633 c1ccc(cc1)OCCSCC(=O)NCc2cccs2 KM06690 Cc1ccc(cc1)Sc2ccc(c3c2non3)[N+](=O)[O-] KM06815 CSc1c2c(c(c3n1c4ccccc4n3)C#N)CCCC2 HTS09912 Cc1cc(n2c3ccccc3nc2c1C#N)N(C(=O)C)C(=O)C HTS09914 Cn1c(nnc1SCC(=O)N/N=C/c2cn(nc2c3ccc(cc3)[N+](=O)[O-])c4ccccc4)c5ccncc5 HTS09929 Cc1c(n2ccccc2n1)C(=O)N/N=C/c3cn(nc3c4cccs4)c5ccccc5 HTS09936 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC(=O)c3ccc4c(c3)OCCCO4 HTS10030 Cc1csc2c1ncnc2NC(C)C GK01644 Cc1csc2c1ncnc2Sc3ccccc3NC(=O)c4cc(cc(c4)C(F)(F)F)C(F)(F)F GK01694 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCc5ccc(cc5)F HTS02050 Cc1c(c(nc(n1)c2ccccn2)SCC(=O)c3ccc(cc3)OC)Cl HTS02086 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)Nc3ccc(cc3F)F)F HTS02213 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)Nc3ccc(cc3)F)F HTS02216 CCOC(=O)CC1C(=Nc2ccccc2S1)SCCS(=O)(=O)c3ccc(cc3)Cl KM06814 COC(=O)c1ccc2c(c1)CCO2 KM07044 Cc1ccc(cc1)OC(=O)c2cc(cc3c2OCC3)Br KM07174 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)O KM07304 c1ccc(cc1)c2c(c(=O)n(nc2c3ccccc3)CC(=O)N/N=C/c4cn(nc4c5ccccc5)c6ccccc6)C#N HTS09983 c1ccc2c(c1)C(=O)N(S2(=O)=O)CC3CC(=NO3)c4ccccc4Cl HTS12291 Cn1c(cc(n1)c2ccccc2)NC(=O)Nc3ccc(cc3)F HTS10227 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)CC(=O)C)C HTS10294 Cc1cc(nc(c1C#N)SCc2ccccc2)C HTS10314 COc1ccccc1N2CCN(CC2)C(=O)Nc3ccc(cc3)Br JFD01740 CCO/C=C\1/c2ccc(cc2C(=O)N(C1=O)c3ccccc3)OC JFD01788 COc1ccc(cc1OC)c2c3ccc(cc3c(=O)n(c2N)c4ccccc4)[N+](=O)[O-] JFD01853 CSc1nnc(n1c2ccccc2)Nc3ccccc3 JFD01896 c1ccnc(c1)N/C=C(\C#N)/C(=O)C2CC2 KM00844 CC(C)(C)C(=O)C(=C1SCCS1)C#N KM00867 c1cc(oc1)C(=O)C(=C2SCCS2)C#N KM00870 Cc1cc2nc(c(c(n2n1)c3ccccc3Cl)C#N)SC KM00873 Cn1c(c(c(n1)c2ccco2)C#N)SC KM00886 c1ccnc(c1)S(=O)(=O)/C(=C/Nc2cc(cc(c2)Cl)Cl)/C#N KM01167 CC(C)(C)C(=O)n1c(c(c(n1)c2cccs2)C#N)SC KM01194 COc1ccccc1Nc2ccc(c3c2non3)[N+](=O)[O-] KM06819 c1cc(cc(c1)F)Nc2ccc(c3c2non3)[N+](=O)[O-] KM06822 c1cc(sc1C2=NN(CC2)CCC(=O)c3ccc(s3)Cl)Cl KM06916 CC1(C=Cc2cc(ccc2O1)/C(=N/O)/N)C KM06957 CC(C)(C)c1cc2nc(cc(n2n1)OC)C(F)(F)F KM07417 c1cc(c(cc1F)F)CNC(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD10769 c1cc(c(cc1F)F)S(=O)(=O)NCc2cc(cc(c2)Cl)Cl CD10787 c1ccc(c(c1)C(=O)NC(=O)NNc2cc(ccc2Cl)C(F)(F)F)Cl CD11292 COCC(=O)C(/C=N/c1ccc(cc1Cl)Cl)C(=O)OC CD11313 Cc1csc(c1N/N=C/c2ccc(cc2)C#N)C(=O)OC GK01799 c1cc(oc1)COC(=O)c2cnc(nc2C(F)(F)F)N3CCOCC3 GK02076 c1ccc(cc1)n2c(c(cn2)C(=O)NNS(=O)(=O)c3ccc(cc3)F)C(F)(F)F GK02081 c1cc(ccc1COC(=O)c2cnc(nc2C(F)(F)F)NNC(=O)C(F)(F)F)Cl GK02111 CC(C)C(C#N)c1ccc(c(c1)OC)OC GK02118 Cc1csc2c1c(ncn2)N3CCCCC3 GK02163 Cc1c(cc(o1)S(=O)(=O)N2CCCC2)c3nc(no3)c4ccc(cc4)F HTS02238 c1cc(ccc1F)S(=O)(=O)CCN2CCN=C(C=C2)C(F)(F)F HTS02264 c1ccnc(c1)N2CCN(CC2)CCS(=O)(=O)c3ccc(cc3)F HTS02269 CC1(CC(=O)C(=CNc2ccccc2Cl)C(=O)C1)C KM01521 CCCS(=O)(=O)/C(=C\OCC)/C#N KM01615 c1ccc2c(c1)c(cc(n2)C(F)(F)F)SCC(=O)O KM07648 CCOC(=O)NC(=O)/C(=C/Nc1ccc(cc1)OC)/C#N KM07698 Cn1cc(c(=O)[nH]c1=O)C#N KM07702 Cn1c(nnc1S)CSc2cc(nc3c2cccc3)C(F)(F)F KM07717 CN1C(=O)C(=Cc2cn(nc2c3ccc(cc3)Cl)c4ccccc4)C(=O)N(C1=O)C HTS10326 C=CCSc1[nH]c(=O)c(c(n1)N)C(c2ccc(cc2Cl)Cl)c3c(nc([nH]c3=O)SCC=C)N HTS10329 c1ccc(cc1)C(=O)CC(c2ccc(cc2)Cl)Sc3ccc(cc3Cl)Cl HTS10474 c1ccc(cc1)COC(=O)N[C@H]2C[C@@H]2NC(=O)OCc3ccccc3 HTS10492 Cc1ccc(cc1)c2nc(=O)c3ccccc3o2 HTS10506 CC(C)(C)c1cc2c(c(c1)Cc3cc(cc(c3OC)Cc4cc(cc(c4O)Cc5cc(cc(c5OC)C2)C(C)(C)C)C(C)(C)C)C(C)(C)C)O JFD01915 c1ccc(c(c1)C2=N/C(=C/c3ccc(c(c3)Cl)Cl)/C(=O)O2)I PD00471 CCOC(=O)C1C(C(C(NC1(C(F)(F)F)O)(C(F)(F)F)O)C(=O)OCC)c2cc(c(c(c2)I)O)OC PD00521 CSc1cccc(c1)N2C(=O)CC(CC2=O)c3ccc(cc3)C(F)(F)F PD00535 CC(=NOc1ccccc1[N+](=O)[O-])C KM01261 c1ccc(c(c1)C(=O)O/N=C(/CS(=O)(=O)c2ccccn2)\N)Cl KM01281 CN1c2ccccc2C(=O)/C(=C\Nc3cccnc3)/S1(=O)=O KM01349 c1cc(sc1)c2nnc(o2)S KM01386 CS(=O)(=O)c1c(c(n[nH]1)c2cccc(c2)Cl)C#N KM01433 COc1ccc(cc1)NC(=S)NC(=O)c2ccccc2Cl RF01992 c1ccc(c(c1)C(=O)NC(=S)Nc2cccc(c2)C(F)(F)F)Cl RF01993 c1cc(c(cc1F)Cl)Oc2cc(nc3c2c(cc(c3)Cl)Cl)C(F)(F)F KM07479 CC(C)Oc1cc(nc2c1cc(cc2)CSc3[nH]c4ccccc4n3)C(F)(F)F KM07488 c1cc(ccc1Oc2cc(nc3c2cc(cc3)Br)C(F)(F)F)F KM07541 c1c(cnc(c1Cl)C(=O)O)C(F)(F)F KM07561 CS(=O)(=O)C/C(=N/OC(=O)c1c(cc(cn1)C(F)(F)F)Cl)/N KM07592 CCOC(=O)/C(=C/N(C)/N=C/c1ccccc1)/C#N RJC00562 c1cc(ccc1CCN2CC(CN(C2)CCc3ccc(cc3)Cl)(C#N)C(=O)O)Cl CD11501 CS(=O)(=O)n1c(ccn1)c2ccc(cc2)Oc3cccc(c3C#N)Cl CD11533 Cc1c(c(n(n1)C)Sc2ccccn2)[N+](=O)[O-] CD11597 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)S(=O)(=O)c5ccc(cc5)n6cccn6 HTS10653 Cc1c(c(no1)c2ccccc2)C(=O)NNC(=O)Cc3cccc(c3)OC HTS10670 CC(=O)c1c(cc(s1)C(C)(C)C)NC(=O)/C=C\C(=O)O GK02213 COC(=O)C(c1ccc(cc1)N2C(=O)c3ccccc3C2=O)(C(F)(F)F)O JFD02149 CCOC(=O)C(c1ccc(c(c1)C)NC(=O)Nc2ccc3ccccc3c2)(C(F)(F)F)O JFD02158 CCOC(=O)C(c1ccc(c(c1)C)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2ccc(cc2)C)(C(F)(F)F)O JFD02167 CC(C)NC(=O)c1c(c(c(s1)SC)C#N)c2cccs2 KM01700 c1cc(ccc1SCC(=O)Nc2cscc2S(=O)(=O)c3ccc(cc3)Cl)Cl KM01720 c1cc(ccc1O)Oc2c(cncc2Cl)Cl RF02613 c1cc(c(c(c1)Cl)C(=O)CS(=O)(=O)c2ccc(cc2)Cl)F RF02869 CC(C)NC(=O)CSc1nnc(n1C)CSc2cc(nc3c2cccc3)C(F)(F)F KM07749 COC(=O)c1c2c(cs1)c(cc(n2)C(F)(F)F)N3CCCCC3 KM07903 CNc1c(c(ncn1)Oc2ccc(cc2)OC)[N+](=O)[O-] KM07928 CCOC(=O)Cn1c(=O)c(cn(c1=O)C(C)C)c2nc(cs2)c3ccccc3 KM07932 COc1cc(nc2c1cc(cc2)C#CCO)C(F)(F)F KM07945 COc1ccccc1NC(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS10536 Cc1ccccc1NC(=O)Nc2cc(nn2C)c3ccccc3 HTS10592 CC(C)CNC(=S)NC(C)(C)C NH00217 CC(C)CNC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F NH00218 COc1ccc(cc1OC)S(=O)(=O)Nc2ccccc2C#N NH00243 c1cc(c(cc1S(=O)(=O)N2CCOCC2)Cl)Cl NH00310 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)CNc4ccc(c(c4)C)Br PD00566 COc1ccc(cc1OCc2ccccc2)/C=C/3\CCc4ccccc4C3=O PD00583 c1ccc-2c(c1)CCc3c2sc(c3)C(=O)NNC(=O)c4ccccc4[N+](=O)[O-] PD00659 c1ccc2c(c1)C(C(N(C2=O)Cc3ccc4c(c3)OCO4)c5cccnc5)C(=O)O PD00718 c1cnccc1CNC(=O)/C=C/C(=O)O PD00762 COC(=O)c1c(noc1C(=O)OC)c2c(cccc2Cl)Cl RF02041 COC(=O)c1c(noc1NC(=O)NCc2ccccc2)c3c(cccc3Cl)Cl RF02257 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N RF02364 CC(C)(C)C(=O)OC/C(=N/OC(=O)c1ccc(c(c1)Cl)Cl)/N RF03003 c1cc(ccc1c2[nH]c3ccc(cc3n2)c4ccc5c(c4)[nH]c(n5)c6ccc(cc6)C(=O)O)C(=O)O RJC00553 c1cc(ccc1n2c(cc(=O)[nH]c2=O)N)Cl RJC00572 Cc1c(cc(s1)c2ccccc2)C(=O)C RJC00609 CC(C)(C)C(=O)/C=C/1\C(=O)Nc2ccccc2N1 RJC00761 c1cc(ccc1Cn2ccnc2COC(=O)Nc3ccc(cc3)Cl)Cl KM08020 c1cc(oc1)CNC(=O)c2ccsc2 HTS10698 c1cc2c(c(c1)S(=O)(=O)Nc3nc([nH]n3)SCc4ccc(cc4)Cl)non2 HTS10721 c1ccc2c(c1)OCC(O2)CNC(=O)c3cc(sc3Cl)Cl HTS10752 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc(cc2)N(C)C HTS10994 CN(C)c1ccc(cc1)NC(=O)c2ccccc2 HTS11005 c1cc2c(cc1S(=O)(=O)N3CCCN(CC3)c4ccc(cn4)C(F)(F)F)CCO2 HTS11046 Cc1c(nc(=O)[nH]n1)SC JFD02305 COc1ccc2c(cc(=O)oc2c1)c3ccccc3 JFD02373 CCOc1ccc2c(cc(=O)oc2c1)c3ccccc3 JFD02374 c1cc(ccc1c2ccc(o2)C=C3C(=O)NC(=O)NC3=O)[N+](=O)[O-] JFD02395 c1cc(ccc1C(=O)N2CCSC2COc3ccc(cc3)[N+](=O)[O-])C(F)(F)F FM00262 COc1c(cc(c(c1C(=O)O/N=C(/c2ccc(o2)[N+](=O)[O-])\N)OC)Cl)Cl RF02893 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N RF02895 Cc1cc(no1)N(Cc2cccc(c2Cl)Cl)C(=O)c3ccccc3 RF03216 c1cc(sc1)CN(Cc2ccc(cc2)Cl)C(=O)c3ccc(cc3)Cl RF03302 CSC1=N/C(=C\c2cccc(c2)Cl)/C(=O)N1Cc3ccc(cc3)Cl RF03332 COC(=O)c1c(ccs1)n2cc(c(=O)[nH]c2=O)C#N KM07976 c1ccc(cc1)SC2CS(=O)(=O)c3c2cccc3 KM08137 c1ccc(cc1)S(=O)(=O)C2CS(=O)(=O)c3c2cccc3 KM08140 CC(C)(C)c1cc2nc(cc(n2n1)SCCOC(=O)Nc3ccccc3)C(F)(F)F KM08148 COc1ccc(cc1)C(=O)CSC2=NCCc3c2cccc3.Br KM08240 c1cc(c(c(c1)Cl)Cl)NS(=O)(=O)c2ccc(c(c2)Cl)Cl NH00313 c1cc(ccc1c2csc(n2)NC(=O)c3ccc(cc3)Cl)Br NH00361 CNC(=S)N(C)NC(=S)NCc1cccs1 NH00448 Cn1c2c(nc1NCc3ccccc3)n(c(=O)n(c2=O)Cc4ccccc4Cl)C HTS11185 Cn1c2c(nc1Oc3ccccc3OC)n(c(=O)n(c2=O)Cc4ccc(c(c4)Cl)Cl)C HTS11195 Cn1c2c(c(=O)n(c1=O)C)CN(CN2)CCOc3ccc(cc3)OC PD00838 c1cc(oc1)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00019 Cn1c2c(c(=O)n(c1=O)C)C(=O)/C(=C/Nc3ccc(cc3)Cl)/C(=O)N2c4ccccc4 JFD02466 COc1ccccc1CC(=O)N2CCN(CC2)c3cccc4c3cc[nH]4 JFD02500 c1ccnc(c1)CCN2C(=O)CNC2=S RF03154 c1cc(ccc1CN2C(=O)CNC2=S)Cl RF03172 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)c3ccc(cc3)Cl KM02458 CCSc1c(c(c(s1)C(=O)O)c2ccc(cc2)Cl)C#N KM02480 c1ccc2c(c1)c(cc(n2)C(F)(F)F)NNC(=O)Nc3ccc(cc3)OC(F)(F)F KM08035 c1ccc(cc1)COC(=O)N2CCN(C(=O)C2)Cc3c(cccc3Cl)Cl KM08051 c1ccc(cc1)C#Cc2ccc(s2)c3ccn(n3)S(=O)(=O)c4ccc(cc4)Cl KM08072 c1ccc(cc1)n2c(nnn2)SCC(=O)NCCSCc3ccco3 KM10422 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccccc3C(C)(C)C)C HTS07244 Cc1ccc(n1c2ccc(cc2)C(=O)NNC(=O)c3ccc4c(c3)OCO4)C HTS11102 CCCSc1c(cccn1)C(=O)Nc2c(onc2c3ccccc3)C HTS11158 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(c3ccccc3)O CD08685 Cc1c(c(n(n1)C)O)C(=O)c2c(onc2c3ccccc3Cl)C CD08715 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(c3ccc(cc3)F)O CD08728 c1ccc(cc1)C(=O)c2ccc(c(c2)[N+](=O)[O-])n3cccc3 CD08766 c1ccc(c(c1)C(=O)O)SCC(=O)c2ccc(cc2)[N+](=O)[O-] FM00286 COc1c(c(c(c(n1)N)C#N)c2cccc(c2)C(F)(F)F)C#N FM00320 c1ccc2c(c1)-c3c(cc(nn3)c4ccc(cc4Cl)Cl)C2=O FM00339 COc1cc2c(cc1OC)ncnc2NCCCN3CCOCC3 GK03296 CCOC(=O)c1c2c(sc1N3C(=O)C=CC3=O)CCCC2 GK03299 CNC(=S)N(Cc1cccnc1)Cc2cccs2 RF03356 CC(C)S(=O)(=O)c1cnc(nc1N)N2CCCC2 KM02592 c1cc(sc1)SCC(=O)Nc2ccc(cc2F)F KM02689 CSCCC(C(=O)NNC(=O)c1ccccc1Cl)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02754 c1ccc2c(c1)CC(C2)NC(=O)C3CC3 KM10498 COc1ccc(cc1)c2cn3cccc(c3n2)OCc4ccc(c(c4)Cl)Cl HTS07274 CC(C)(C)c1cn2cccc(c2n1)OCc3ccc(c(c3)Cl)Cl HTS07275 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCNC(=O)C2CC(=O)Nc3ccsc3C(=O)OC HTS07293 Cn1c2c(nc1Oc3cccc(c3)Cl)n(c(=O)n(c2=O)Cc4ccc(cc4Cl)Cl)C HTS11218 c1ccc(cc1)C(=O)C2(C3C2CCCC3)C(=O)c4ccccc4 JFD00204 Cn1c(n[nH]c1=S)c2ccc(cc2)Cl HTS11927 c1cc(sc1)/C=N/NC(=O)CSc2c3c4c(sc3ncn2)CCCC4 HTS11934 CCC(c1c([nH]c(=S)[nH]c1=O)N)c2c([nH]c(=S)[nH]c2=O)N HTS11939 c1cc(ccc1C(=O)N2CCC(CC2)NC(=O)C3CCCCC3)Cl JFD02504 c1c(cc(cc1C(F)(F)F)N/N=N/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F JP00904 c1ccc2c(c1)CC3C2=Nc4ccccc4SC3c5cccc(c5)Cl JFD02640 Cc1cccc(c1)C(=O)Nc2ccccn2 JFD02664 c1ccc(c(c1)C(=O)Nc2cccc(c2)C(F)(F)F)I JFD02672 COc1cc(cc(c1OC)OC)C(=O)NC2CCCCC2 JFD02690 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)Nc3ccc(cc3)Cl KM02487 Cc1nccc(n1)c2cccc(c2)N/N=C(\C#N)/C(=O)c3ccc(cc3)Cl KM02502 CC1(OC(=O)C(=CNc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)O1)C KM02529 c1cc(ccc1c2csc(c2C#N)S(=O)C3CCCCC3)Cl KM02782 Cn1c(cc(n1)c2ccc(s2)C(=O)Nc3ccc(cc3)Cl)C(F)(F)F KM02904 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccsc3)C HTS07247 c1ccc(cc1)NC(=O)NCC(COc2ccc(cc2)[N+](=O)[O-])O HTS07263 CCOC(=O)C1=NN(C2(C1c3ccc(cc3)C)C(=O)c4ccccc4C2=O)c5ccccc5 HTS09117 CCOC(=O)c1c(nc2n1ccc(c2)C)C HTS07415 CCOC(=O)/C(=C/1\c2cc(ccc2NC1=O)Br)/C#N DP00507 c1ccc2c(c1)c(nnc2O)c3ccc(cc3)Cl DP00603 c1ccn(c1)c2c(c(c(o2)c3cccs3)C#N)c4ccc(cc4)C#N CD09256 c1ccn(c1)c2c(c(c(o2)c3cccs3)C#N)c4cccs4 CD09257 c1ccc(cc1)c2c(c[nH]n2)c3nc(no3)c4ccc(cc4)Cl CD09386 CNc1ccccc1C(=O)NCc2ccco2 DP01030 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3nnc(o3)c4ccc(cc4)Cl GK00263 CC(C)(C)c1ccc(cc1)c2cc(c(s2)C(=O)N)NS(=O)(=O)c3ccccc3 GK03562 CC(C)(C)c1cc2c(s1)c(ncn2)N3CCOCC3 GK03578 c1cc(ccc1CNCC(Cn2ccc(n2)C(F)(F)F)O)C(F)(F)F HAN00285 CSCCC(C(=O)NNS(=O)(=O)c1ccccc1Cl)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02774 CSc1c(cccn1)C(=O)N=S(=O)(C)c2ccc(cc2)Cl KM02930 Cn1c(cc(n1)c2ccc(s2)C(=O)N)C(F)(F)F KM03001 CC(C)S(=O)(=O)c1c([nH]nc1SC)N KM03016 c1cc(c(c(c1)Cl)/C=C(\C#N)/S(=O)(=O)Cc2ccco2)F KM03085 c1ccnc(c1)N/C=C(\C#N)/S(=O)(=O)Cc2ccco2 KM03111 c1ccc2c(c1)cccc2C(=O)NNC(=O)COc3c4ccc(cc4ncn3)Cl HTS07341 c1ccc2c(c1)cccc2C(=O)NNC(=O)c3cc(cnc3)c4cccs4 HTS07377 Cc1c2c([nH]n1)OC(=C(C2c3cccc(c3)OC)C#N)N HTS07490 Cc1c2c([nH]n1)OC(=C(C2c3ccc4c(c3)OCO4)C#N)N HTS07491 CNC(=S)NNC(=O)CN1c2ccccc2Sc3c1cccc3 HTS07501 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nnc(n3c4ccccc4)c5ccco5)C1 HTS11956 CC1CCc2c(sc(c2C#N)NC(=O)CSc3nccn3C)C1 HTS11960 c1ccc(cc1)/N=C\2/c3ccccc3NC2=O HTS12039 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)CC=C)C HTS12075 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4cn(nc4c5cccs5)c6ccccc6)C HTS12085 COc1cc(cc(c1OC)OC)C(=O)Nc2cccc3c2cccc3 JFD02700 c1ccc(cc1)C(=O)O/N=C/c2ccc3c(c2)OCO3 JFD02711 CCS(=O)(=O)CS(=O)(=O)CC JFD02735 c1ccc\2c(c1)CCC/C2=N\c3ccccc3C(F)(F)F JFD02864 c1cc(c(cc1Cl)[N+](=O)[O-])c2ccc(o2)C(=O)O JFD02879 COc1cc(cc(c1OC)Br)C(=O)O JFD02899 c1ccc2c(c1)nc(s2)c3cccc(c3)Cl JFD02908 CSCCC(C(=O)NNC(=O)Nc1ccccc1)NC(=O)c2ccc(cc2)C(F)(F)F KM02877 CC(C)(CCNC(=O)Cc1ccsc1)C(=O)N/N=C/c2ccccc2 KM02909 COC(=O)c1c(c(c(s1)N2CCOCC2)C#N)N KM02915 c1cc(oc1)CS(=O)(=O)Cc2nc(cs2)c3ccc(cc3)Cl KM03218 CC(C)S(=O)(=O)c1csc(c1Cl)NC(=O)N=S(=O)(C)c2ccc(cc2)Cl KM03259 CCOC(=O)CSc1nnc(n1c2ccccc2)c3ccccc3 HTS07433 Cc1nc2c(cnn2c3ccccc3)c(=O)n1/N=C/c4ccccc4 HTS07449 Cn1c(nnc1SCc2n[nH]c(=S)n2Cc3ccccc3)c4ccccc4 HTS07460 c1ccc(cc1)CNC(=S)NNC(=O)c2c(c3c(cc(nc3o2)c4ccc(cc4)Cl)c5ccccc5)N HTS07550 c1ccc(c(c1)C(=O)N/N=C/c2ccc3c(c2)OCO3)N DP01043 Cc1ccc(cc1C)CSC2NCC(N2)C.Cl DP01062 c1ccc(cc1)N2C(=O)CC(C2=O)n3cnc4c3cccc4 DP01241 CN(C)c1ccc(c(c1)Cl)C2Nc3cc(ccc3O2)Cl DP01271 COc1cc(cc(c1OC)OC)C2Nc3ccccc3O2 DP01283 COCCCN1CNC(=S)NC1 DP01314 c1cc(c(c(c1)Cl)Cl)S(=O)(=O)Nc2ccc(cc2)n3ccc(n3)C(F)(F)F HAN00365 COC(=O)c1ccccc1CSc2nccc(n2)C(F)(F)F HAN00418 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2c(nccn2)N HAN00438 C1Cc2c(sc(c2C(=O)N)N)C1 HR00227 CNc1nc(cs1)c2ccc(s2)Cl HTS00001 Cn1c(c(c(n1)C(F)(F)F)c2ccc(cc2)Br)NC(=O)Cc3ccccc3F HTS00010 COC(=O)c1cscc1OS(=O)(=O)c2ccc(cc2)Cl KM03207 CSc1c2c(c(s1)C(=O)NN)CCCC2O KM03384 CSc1c(cc(s1)C(=O)NN)C#N KM03408 Cc1cc2nnc(c(n2n1)C)C(=O)/C=C/N(C)C KM03432 CC(C)S(=O)(=O)/C(=N/Nc1c(csc1C(=O)OC)S(=O)(=O)Cc2ccco2)/C#N KM03452 c1ccc2c(c1)N(c3ccccc3S2)CC(=O)N/N=C/c4ccc(cc4)[N+](=O)[O-] HTS07510 c1ccc2c(c1)[nH]c3n2c(=O)c4c(c3C#N)CCC4 HTS07553 C=CCn1c(nnc1Sc2c3c(nc4n2ncn4)CCC3)c5ccccc5 HTS07593 c1ccc(cc1)Cn2c3c(c(=O)n(cn3)Cc4ccc(cc4)F)nn2 HTS07635 CC1CCc2c(sc3c2c(=O)n(c(=O)[nH]3)c4ccc(cc4)Cl)C1 HTS07652 c1cc(ccc1Cn2c(c(nn2)C(=O)N)N)F HTS12086 Cc1cc(nc2c1c(c(s2)C(=O)N/N=C/c3ccccc3)N)C HTS12094 COc1cccc(c1)Nc2c3c(ncn2)n(nn3)Cc4ccc(cc4)Cl HTS12172 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=C/4\CCc5ccccc5C4=O HTS12173 CCOC(=O)c1c2nc(c3ccccc3n2nn1)N(Cc4ccccc4)Cc5ccccc5 HTS12195 c1cc(ccc1F)S(=O)(=O)/C(=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C#N KM01394 CCOC(=O)C(C(CC(=O)C1CC1)c2ccccc2)C(=O)OCC JFD03008 c1cc(cc(c1)[N+](=O)[O-])c2ccc(o2)C=C3C(=O)NC(=O)NC3=O JFD03080 c1ccc(cc1)C(=O)NC(=S)NC23CC4CC(C2)CC(C4)C3 JFD03120 CCCCc1c(nc2ccccn2c1=O)O JFD03137 Cc1c(nc2ccccn2c1=O)O JFD03144 CC(C)Sc1c2c(c(s1)C#N)CC(CC2=O)(C)C KM03312 CCOC(=O)c1c2c(c(s1)SCc3ccc(cc3)Cl)C(=O)CCC2 KM03346 CN(C)/C=C/1\CCc2c(sc(c2C1=O)SC)C#N KM03376 CCOC(=O)CSc1c2c(c(s1)C(=O)OCC)CCCC2O KM03377 CSc1c\2c(c(s1)C#N)CCC/C2=N/O KM03507 Cc1csc2c1c(c(s2)C=C(C#N)C#N)C KM03526 Cc1cc(nc2c1c(c(o2)c3nnc(n3C)SCc4ccc(cc4)Cl)N)c5ccccc5 HTS07551 Cn1c(nnc1SCC=C)c2c(c3c(cc(nc3o2)c4ccccc4)c5ccccc5)N HTS07552 c1ccc2c(c1)nc3n2c(c4c(c3C#N)CCCC4)N5CCOCC5 HTS07561 Cc1ccc2nc(cn2c1)c3cc(no3)c4ccccc4 HTS07690 c1ccc(c(c1)c2csc(n2)c3ccc(cc3)Cl)Cl DP01413 Cc1ccc(cc1)CSC2=NCCCN2C3CCCCC3.Cl DP01438 c1ccc(cc1)CN2CCNC(C2=O)CC(=O)NN DP01702 c1ccc2c(c1)ccc(c2/N=N/c3c(c(cc(c3Cl)Cl)Cl)Cl)O DP01713 c1ccc2c(c1)C(=O)NNC(=S)N2 DP01824 c1ccc(c(c1)C(=O)NNc2ccccc2Cl)N DP01883 c1cc(c(cc1C(F)(F)F)C(=O)O)Cl DP01924 c1ccc(cc1)N(C2CCCCC2)C(=O)CN3CCN(CC3)c4ccc(cn4)[N+](=O)[O-] HTS00019 c1cc(sc1)C(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS00079 Cn1c(nnc1SCC(=O)N2CCOCC2)CSc3ccnc4c3ccc(c4)Cl HTS00158 COC(=O)c1c(ccs1)NC(=O)CSc2ccccn2 HTS00161 CCCCCc1ccc(cc1)S(=O)(=O)NCc2nc(no2)c3ccc(cc3)C(F)(F)F HTS00177 Cc1csc2c1c(c(s2)COC(=O)c3ccccc3Cl)C KM03503 c1ccc(cc1)/C=N/C(=C(/C#N)\NCc2ccccc2Sc3ccc(cc3)Cl)/C#N KM03648 COC(=O)c1c(ccs1)N/C=C(\C#N)/C(=O)C2CC2 KM03696 Cc1c2c(c(sc2sc1C(=O)C)[N+](=O)[O-])C KM03799 CS(=O)(=O)c1c2c(c(s1)Br)CCCC2=O KM03820 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(cc3)C)CC(CC2)C HTS07656 c1ccc(cc1)/C=N/NC(=O)Cn2cnc3c(c2=O)c4c(s3)CCCC4 HTS07670 c1ccc(cc1)C(=O)Nc2nnc(s2)C3CC3 HTS07889 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)c5cccnc5Oc6ccc(cc6)Cl HTS07938 CN(CCc1ccccn1)C(=O)c2c(c3ccccc3s2)Cl HTS07945 CCOC(=O)c1c2nc(c3ccccc3n2nn1)Nc4cccc(c4)C(F)(F)F HTS12197 CCOC(=O)c1c(n(nc1/C=C/c2ccccc2)c3ccccc3)C HTS12228 c1ccc2c(c1)nc(n2Cc3ccc(cc3Cl)Cl)SCc4ccc(cc4Cl)Cl HTS12301 c1ccc2c(c1)c(cs2)NC(=O)N3CCSCC3 HTS12346 CCOC(=O)C1(C(C(=NN1c2ccc(cc2)[N+](=O)[O-])c3cccs3)c4ccc(cc4)OC)C#N HTS12363 c1ccc(cc1)C(c2ccc3ccccc3c2)O JFD03195 CC(C(=O)NNC(=S)Nc1ccccc1)Oc2ccc(cc2Cl)Cl JFD03196 CC(C(=O)NNC(=S)NC)Oc1ccc(cc1)Cl JFD03200 CC1=C(C(C2=C(N1)CC(CC2=O)(C)C)c3ccccc3Cl)C#N JFD03300 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/O JFD03327 c1cc(ccc1N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl)OC(F)(F)F KM03576 CC1(Cc2c(c(sc2C(=O)O)SC)/C(=N\OC)/C1)C KM03586 COC(=O)c1cc(c(s1)SC)c2nc(cs2)c3ccc(cc3Cl)Cl KM03603 c1cc2c(cc1c3csc(n3)N)OCCO2 HTS07721 CCCCN1Cc2c(n(c3cc(nn3c2=O)c4ccccc4)CC(=O)c5ccc(cc5)OC(F)(F)F)C1=O HTS07741 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)C3CCCCC3)C HTS07782 c1ccc(cc1)CN2CCc3c(ccs3)C2c4ccc(cc4)OC(F)(F)F HTS07828 c1ccc(cc1)n2c(nnc2SCCS(=O)(=O)c3ccc(cc3)F)O HTS07990 CC(C)(C)NC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl DP01979 COc1cc(cc(c1OC)OC)C(=O)N2CCCN3C2c4ccccc4C3=O DSHS00344 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)C3CCN2CC3 DSHS00355 c1ccc(c(c1)/C=C\2/C(=O)C3CCN2CC3)Cl DSHS00407 CC1(C(=C)S/C(=N\c2ccccc2Cl)/N1C(=O)c3ccc(cc3)[N+](=O)[O-])C DSHS00458 C#CC1(CCCCC1)NS(=O)(=O)c2cc(ccc2Cl)Cl DSHS00531 CC(C)(CC(=O)Nc1ccsc1C(=O)OC)CC(=O)O HTS00186 c1cc(ccc1C2(CCN(CC2)C(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)O)Cl HTS00202 Cc1ccc(n1c2cc(ccc2n3ccnc3)[N+](=O)[O-])C HTS00294 Cc1c(c(nc(n1)c2ccccc2)SCCCOc3ccc(cc3)Cl)C#N HTS00304 c1cc(ccc1n2c(c(cn2)C#N)NC(=O)C3CCCCC3)F HTS00328 CC1(CC(=O)C=C(S1)SCC(=O)Nc2ccccc2Cl)C KM03964 CC1(Cc2c(c(sc2c3ccn(n3)C(=O)Nc4ccc(cc4)Cl)SC)/C(=N/OC)/C1)C KM04068 Cc1cc(nc2c1c(nn2C)C)N/N=C/c3ccccc3Cl KM04107 CN1c2ccccc2-c3c(c(sc3C(=O)N4CCOCC4)SC)S1(=O)=O KM04136 c1cc(c(cc1F)F)NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS07956 c1cc(ccc1NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl)F HTS07958 CN1CCc2c(sc(c2C(=O)c3ccc(cc3)OC)N)C1 HTS08117 c1ccc(c(c1)C#N)NS(=O)(=O)c2ccc(cc2)F HTS08145 CC12c3cc(c(cc3CCN1C(=NN2c4ccccc4)C(=O)c5ccccc5)OC)OC HTS12370 CCn1c(n[nH]c1=S)c2ccco2 HTS12532 CCOC(=O)c1c2nc(c3ccccc3n2nn1)Sc4[nH]c5ccccc5n4 HTS12553 CCOC(=O)c1c(c2c(cc(nc2s1)C)C)NC(=O)Nc3ccccc3 HTS12567 Cc1ccc(o1)C(CC=C)NCc2ccccc2 JFD03357 CC1=C(C(C(=C(N1)C)C#N)c2cc(ccc2O)Br)C#N JFD03362 COC(=O)CCN1CCCc2c1ccc(c2)/N=N/c3ccc(cc3)C#N JFD03384 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(COc3ccccc3C(=O)N)O JFD03569 c1ccc(cc1)CN(c2cccc3c2cccc3)C(=S)Nc4ccccc4 JFD03582 CC(=O)c1ccc2ccc3ccccc3c2c1 JFD03589 CC1(CC(=O)C=C(S1)SCC(=O)c2ccc(cc2)Cl)C KM04009 CN1c2ccccc2-c3c(c(sc3C(=O)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F)SC)S1(=O)=O KM04014 CC(C)S(=O)(=O)c1cc(sc1SC)C(=O)Nc2cccc(c2)C(F)(F)F KM04016 CSc1c(c(on1)c2ccc(s2)S(=O)(=O)NCc3ccccc3)C#N KM04023 Cc1c(c(n(n1)Cc2nnc(n2C)SCC(=O)c3ccc(cc3)Cl)C)[N+](=O)[O-] KM04212 CC(C)c1ccc(cc1)NC(=O)CSc2nnc(n2c3ccccc3)O HTS07994 Cn1c(cc(n1)c2ccc(cc2)Cl)NC(=O)CCCC(=O)O HTS08052 CCOC(=O)Cc1csc(n1)NC(=O)CC(C)(C)CC(=O)O HTS08089 CCOC(=O)Cc1csc(n1)NS(=O)(=O)c2cn(cn2)C HTS08093 Cn1cc(nc1)S(=O)(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08274 COc1ccc(cc1OC)CCNC(C#N)c2ccco2 DSHS00559 c1ccc(c(c1)NC(=O)COc2cc(c(cc2Cl)Cl)Cl)Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00744 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3ccccc3Sc4ccc(cc4[N+](=O)[O-])Cl DSHS00749 c1ccc(c(c1)NC(=O)c2ccco2)Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00751 COc1cc(cc(c1OC)OC)C(=O)N(CCC#N)C2CCCCC2 DSHS00778 CC(=O)Nc1c(c(nn1C)C(F)(F)F)c2ccc(cc2)OC HTS00341 c1cc(c(cc1Cl)NC(=O)CC2C(=O)NCCN2)Cl HTS00380 CC1(CC(=C(C(=O)N1)C#N)c2ccccc2)c3ccccc3 JFD03987 CC(C)(C)c1ccc(cc1)C(=O)NC2CCNCC2 JFD04004 CSc1cccc(c1)N/C(=N/C#N)/SC JFD04018 Cc1cc(nc(n1)N/C=C/2\C(=O)c3c(ccs3)N(S2(=O)=O)C)C KM04190 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/OC(=O)Nc3ccc(cc3)Cl KM04381 CSc1c-2c(c(s1)C(=O)Nc3ccc(cc3)Cl)CCc4c2nc(nc4)SC KM04397 COC(=O)c1cc(=O)nc2n1ccs2 KM04412 CNC(=S)NNC(=O)CSc1ccccc1 KM04425 COc1cscc1C(=O)NNC(=O)c2ccc(cc2)Cl KM04434 CCCCc1ccc(c(c1)C)NC(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl HTS08222 Cc1cc(no1)C(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08254 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)c3ccco3)C(F)(F)F HTS08396 c1ccc(c(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F)N3CCCCC3 HTS08436 c1ccc(c(c1)NC(=O)Nc2cccs2)N3CCCCC3 HTS08447 C/C(=N\Nc1nc(c(nn1)c2ccccc2)c3ccccc3)/c4ccco4 HTS12594 COc1ccc(cc1)C2C3=C(c4ccccc4CC3)NC(=S)N2 HTS12667 c1ccc2c(c1)CCC3=C2NC(=S)NC3c4cccs4 HTS12671 COc1ccc(cc1)c2cc(cc(n2)c3ccccc3)c4ccccc4 NRB03343 c1ccc(cc1)C(=O)C/C(=C\C(=O)c2ccccc2)/c3ccc(cc3)Cl NRB03363 Cc1ccc(cc1)Sc2cc(c(cc2[N+](=O)[O-])C)N3CCOCC3 NRB03393 [C@@H]1([C@@H]([C@H](OC([C@@H]1O)O)C(=O)O)O)O JFD03599 c1ccc2c(c1)c(cc(n2)c3cc(ccc3Cl)Cl)C(=O)O JFD03602 CCOC(=O)CNC(=O)c1cc2cc(ccc2o1)Br JFD03614 c1ccc(cc1)c2c(nc(nc2O)S)N RDR01717 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N/c3ccc(cc3Cl)Cl RDR01748 Cc1cc(ccc1Br)NC(=S)NCCc2ccc(c(c2)OC)OC RDR01768 Cc1c(c(n(n1)Cc2nnc(n2C)SCC(=O)Nc3ccccc3Cl)C)[N+](=O)[O-] KM04222 Cc1c(c(n(n1)Cc2nnc(n2C)SCc3c(cccc3Cl)Cl)C)[N+](=O)[O-] KM04225 CS(=NC(=S)NC(=O)Oc1ccccc1)(=O)c2ccccc2 KM04269 Cc1c(sc2c1C(=O)/C(=C\Nc3ccc(cc3)Cl)/S(=O)(=O)N2C)C KM04331 c1c(c(cc2c1OCO2)[N+](=O)[O-])/C=C/[N+](=O)[O-] RH00774 CC(c1ccccc1)n2c(nnc2SCC(=O)c3ccc4c(c3)OCCO4)O HTS08336 Cc1cc(c(c(c1)C)n2c(nnc2SCC(=O)c3ccc4c(c3)OCCO4)O)C HTS08337 Cc1cccc(c1C)C(=O)Nc2ccc(cc2)S(=O)(=O)N HTS08350 CC(=O)Nc1ccc(cc1)S(=O)(=O)N(C)C2CCCCC2 HTS08352 c1ccc(cc1)C#Cc2cc(cnc2)C(=O)NC(=S)Nc3cccc(c3)C(F)(F)F KM09955 Cc1c(c(c(c(c1C)C)CSCC(=O)NN)C)C DSHS00856 CCOC(=O)N1CCc2c(sc3c2c(=O)n(c(=S)[nH]3)c4ccccc4)C1 HTS13002 Cc1nc2c(c(=O)n1NC(=O)CN(Cc3ccccc3)Cc4ccccc4)ncn2c5ccccc5 HTS13038 C=CCn1c(nnc1SCC(=O)NN2CC(=O)N(CC2=O)c3ccccc3)c4cccs4 HTS13269 COc1ccc(cc1OC)/C=N/N2C(=O)c3ccccc3C2=O JA00043 CCCC(C(=O)O)NC(=O)C(C)N JFD04033 CCOC(=O)c1ccc(c(c1)[N+](=O)[O-])SCC(=O)Nc2ccc(c(c2)Cl)C JP00549 COc1cc(c(cc1Cl)OC)NC(=S)N2CCOCC2 JP00555 CC(=O)c1ccc(c(c1)[N+](=O)[O-])N2CCc3ccccc3C2 JP00677 CC(C)Sc1ccc(cc1[N+](=O)[O-])C(=O)C JP00698 Cc1cc(nc(n1)C)N/C=C/2\C(=O)c3c(c(sc3N(S2(=O)=O)C)C)C KM04449 Cc1c2ccccc2oc1C(=O)O/N=C(/c3ccc(cc3)OC(F)(F)F)\N RH00884 c1cc2c(cc[nH]2)cc1NC(=S)NCC3CC3 RH00904 c1cc2c(cc[nH]2)cc1NC(=S)Nc3ccc4c(c3)OCCO4 RH00907 CC(=O)OC(c1ccccc1)C(=O)O RH00919 COc1cccc(c1)NC(=O)Nc2ccc(nc2)Oc3cccc(c3)C(F)(F)F HTS08493 CC(C)(C)c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3ccc(cc3)C(F)(F)F HTS08498 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)Cl KM10269 COc1cccc(c1)NC(=O)NCCSCc2ccco2 KM10275 c1cc2c(cc1c3cc(nc(n3)N)C(F)(F)F)CCC2 KM10321 CN(c1ccc(cc1Cl)[N+](=O)[O-])C2CCCCC2 NRB03412 CC(=O)/C(=C\N(C)C)/c1nnnn1c2ccc(cc2)Cl NRB03495 CN(C)/C=C(/c1nnnn1c2ccc(cc2)F)\C(=O)c3ccccc3 NRB03502 CC(=O)OC1CCC2(C3CCC4(C(C3CC=C2C1)CCC4OC(=O)c5ccccc5)C)C NRB03675 CCC(=O)O[C@@H]1CC2(C(C[C@H]([C@@]2(C(=O)C)O)C)C3C1C4(CCC(C[C@@H]4CC3)OC(=O)CC)C)C NRB03726 CN(C)C(=O)Oc1ccc2c(cc(=O)oc2c1)c3ccccc3 RDR01779 COc1cccc(c1C(=O)Nc2ccccc2F)OC RDR01952 COc1c(cc(cc1Cl)Cl)c2cn3ccccc3n2 RDR02046 c1ccc(cc1)N2C(CC(=N2)c3ccc(cc3)Cl)c4ccc(c(c4)Cl)Cl RDR02306 Cc1ccc(cc1)C2CC(=NN2c3ccccc3)c4ccccc4Cl RDR02309 Cc1cc(nc(n1)N2CCCC2)O RDR02326 Cc1cc(ccc1[N+](=O)[O-])c2nnc(o2)CSc3nnc(s3)NC(=O)c4ccc(s4)Cl RH00788 Cc1ccc2c(c1)c3c([nH]2)CCCCC3 RH00820 Cc1cc(n(n1)c2ccccc2)Nc3ccccc3C(=O)O RH00834 Cc1cc(n(n1)c2ccc(cc2)OC)Nc3ccccc3C(=O)O RH00838 Cc1ccc(cc1n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3)C(=O)OC KM09994 COc1c(cc(c2c1nccc2)Cl)I KM10003 COc1ccc(cc1)CNC(=O)Nc2cccc(c2)SC KM10206 CNC(=S)NNC(=O)c1ccc2c(c1)cccn2 KM10266 CCCCc1ccc(cc1)NC(=O)NC2Cc3ccccc3C2 KM10453 CCOc1ccccc1/C=N/N2C(=O)c3ccccc3C2=O JA00047 CN(/C=C/C=C(C#N)C#N)c1ccccc1 JFD00036 CCOC(=O)C1=C(NC(=O)C1)C JFD00048 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)O JFD00160 c1ccc(cc1)[C@H]2[C@@H](C(=O)c3ccccc3O2)O JFD00176 CCOC(=O)C(=C1CCCC1)C#N JP00765 Cc1cccnc1NC2c3ccccc3C(=O)O2 JP00795 c1ccc(cc1)CN2CCC(CC2)Nc3c4c5c(sc4ncn3)CCCC5 GK03330 CC(C)Nc1c2c(ccs2)ncn1 GK03338 Cn1c(ccn1)NC(=O)CCc2ccccc2 GK03350 COc1cc2c(cc1OC)ncnc2NCCO GK03358 CC1=C(C(CC(=O)N1)c2ccc(cc2)C(C)C)C(=O)OC RH00949 CCCCCCCCCC(=O)Nc1nc-2c(s1)CCc3c2ccc(c3)OC RH01163 CCOC(=O)c1c[nH]c2ccccc2c1=O RH01193 Cc1cc(no1)C(=O)Nc2nc-3c(s2)CCc4c3cccc4 RH01200 CC(C)/C=C/C1=CC2=C(C1)Cc3c2cccc3 RH01201 Cc1c(nc(s1)c2ccccc2)CC(=O)NNC(=O)Nc3ccc(cc3)OC(F)(F)F RH01255 COc1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4S(=O)C KM10373 c1csc(n1)c2cc(nc(n2)N)C(F)(F)F KM10391 COc1ccc(cc1)c2cc(n3c(n2)cc(n3)c4ccco4)C(F)(F)F KM10414 COc1ccc(cc1)CNC(=O)Nc2ccccc2C(F)(F)F KM10509 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc4c(c3)CCC4 KM10521 CC(=O)OC1CCC2(C3C(CC[C@]2(C1)C)C4CCC(=O)C4(CC3=O)C)C NRB03739 CC(C1CCC2C1(CCC3C2CC[C@@H]4C3(CCC(=O)C4)C)C)OC(=O)C NRB03875 C[C@@]1(CCC2C1(CCC3C2CCC4C3(C/C(=C\c5ccccc5)/C(C4)O)C)C)O NRB03879 CC1=C(C(=O)OC1(C)COC)C(=O)OC JFD00220 COc1ccc(cc1)OC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02329 c1cc(ccc1Nc2nnc(s2)C(F)(F)F)Cl RDR02364 CC(C)(C)C(=O)OCc1nc(on1)c2ccccc2 RF02992 COc1cc2c(c(c1OC)OC)C(=O)CC2 JP00916 COc1cc(cc(c1OC)OC)/C=N/NC(=O)C(=O)Nc2ccc(c(c2)Cl)Cl JPV00018 c1cc(ccc1C(=O)c2ccc3c(c2)CCC3)[N+](=O)[O-] JPV00026 c1cc(sc1)c2nnc3n2N=C(CS3)CC(=O)NN RH01068 c1ccc(cc1)c2csc(n2)c3cccnc3.Br RH01083 c1ccc(cc1)CCNC(=O)c2ccco2 RH01094 COc1ccc-2c(c1)CCc3c2nc(s3)NC(=O)c4ccco4 RH01143 Cc1c(c2ccccc2[nH]1)SCc3nnc(n3C)SCC(=O)Nc4cccc(c4)C(F)(F)F KM07997 Cn1c(cc(n1)C(F)(F)F)c2ccc(s2)/C=C(\C#N)/S(=O)(=O)c3ccc(cn3)C(F)(F)F KM05352 COc1ccc(cc1NC(=O)Nc2ccccc2)Cl KM10454 c1ccc(cc1)C(=O)NC2Cc3ccccc3C2 KM10474 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC3Cc4ccccc4C3 KM10487 CCOc1ccccc1NC(=O)NC2Cc3ccccc3C2 KM10496 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(c(c3)Cl)F NH00503 CC(C)(C)c1ccc(cc1)NC(=O)CSc2nnc(n2c3cccnc3)O HTS09137 c1ccc2c(c1)C(=O)/C(=C\c3ccc(cc3)Cl)/S2 JFD00189 Cc1ccc(cc1)c2c(nc3cc(c(cc3n2)C)C)c4ccc(cc4)Cl DP00619 CN(c1ccc(cc1)/C=N/NC(=O)N/N=C/c2ccc(cc2)N(CCC#N)C)CCC#N DP00689 c1ccc(cc1)C(=O)Nc2ccccc2C(=O)Nc3ccncc3 DP00699 Cc1csc(n1)N/N=C/2\CCCc3c2ccc(c3)OC FM00227 COc1cccc(c1)SCC(=O)N2CCN(CC2)c3ccccc3 HTS01203 c1ccc(cc1)C2=NN=C(C=C(C2)c3ccc(cc3)F)c4ccccc4 HTS01277 c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4ccc(cc4)OC(F)(F)F GK03601 Cc1ccc(cc1)C(=O)NNc2c3c(cc(s3)C(C)(C)C)ncn2 GK03634 CC(C)(C)c1cc(=O)n2c([nH]1)c(c(n2)C(F)(F)F)c3ccc(cc3)OC HTS01429 CCCCCCNC(=O)NCCCCCC RH01432 COc1ccc(cc1OC)CCNC(=O)C2CCCO2 RH01459 COc1ccccc1C2CCN(CC2)c3cc(ccc3[N+](=O)[O-])O RH01481 COc1ccccc1C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C4OCCO4 RH01483 C=CCCOc1ccccc1C(=O)N RH01489 CCCCOc1ccc(cc1)S(=O)(=O)NC(Cc2c[nH]c3c2cccc3)C(=O)OC RH01617 c1cc(cnc1)c2nc(cs2)c3ccc(cc3)Br.Br ML00079 c1cc(cnc1)c2nc(cs2)c3ccc(cc3)[N+](=O)[O-].Br ML00081 c1ccc(c(c1)Nc2nc(cs2)c3ccc(cc3)F)Cl.Br ML00086 c1ccc(cc1)/C=N/NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 ML00096 CC(c1ccccc1)NC(=O)/C=C/C(=O)O NRB00620 CC1([C@@H](NC(S1)c2ccc(cc2)OC)C(=O)O)C NRB04487 CC1([C@@H](NC(S1)c2ccc(cc2)[N+](=O)[O-])C(=O)O)C NRB04493 CC(C)(C)c1ccc(cc1)C(=O)CC(C(=O)O)Sc2ccc(cn2)C(F)(F)F NRB04690 CN1C(=O)C(OC1=O)c2ccccc2 NRB04783 c1ccc(cc1)/C=C/2\C(=O)N3CCCCSC3=N2 NRB04871 CC(C)c1ccc(cc1)NCC(CSc2ccccc2)O RDR03295 c1cc(cnc1)n2ccnc2SCc3ccc(cc3)Br RDR03307 Cc1c(c(no1)c2c(cccc2Cl)Cl)C3=NCCO3 RDR03685 Cc1cc(nc(n1)c2ccccn2)Oc3cc(cc(c3)Cl)Cl RDR03747 c1cc(c(cc1Cl)Cl)CS(=O)(=O)C2CCCCC2O RDR03789 c1cc(c(cc1F)F)Cc2nc(on2)N RDR03833 Cc1ccccc1NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)c4ccccc4OC RH01574 Cc1ccc(cc1)S(=O)(=O)NC(Cc2c[nH]c3c2cccc3)C(=O)OC RH01575 c1cc(c(cc1[N+](=O)[O-])CC(CO)C#N)N2CCOCC2 RH01587 c1cc(ccc1F)S(=O)(=O)CCN2CCOCC2 KM08563 COC(=O)C(Cc1c[nH]c2c1cccc2)NC(=O)CN3CCCCC3 RH01692 c1ccc2c(c1)nc(c(n2)O)O MGH00027 CNc1c2ccccc2oc(=O)c1[N+](=O)[O-] MGH00119 c1cc(c(cc1F)F)C(=O)NC(=O)N2CCCCC2 MGH00237 c1cc(ccc1c2csc(n2)c3ccncc3)Br.Br ML00034 c1cc(oc1)C(=C(C#N)C#N)C#N NRB00510 CCOc1ccccc1/C=N/NC(=S)N ML00166 COC(=O)[C@@H](Cc1ccccc1)NC(=O)c2cccc3c2cccc3 JFD00457 c1ccc(cc1)CC(=O)NC2CCN(CC2)S(=O)(=O)c3cc(c(cc3Cl)Cl)Cl JFD02531 CC(C)(C)c1cc2c(c(c1)Cc3cc(cc(c3O)Cc4cc(cc(c4O)Cc5cc(cc(c5O)C2)C(C)(C)C)C(C)(C)C)C(C)(C)C)O JFD00633 c1ccc(cc1)c2ccnc3c2ccc4c3nccc4c5ccccc5 JFD00692 c1ccc(cc1)S(=O)(=O)CCN2CCOCC2 KM00012 C1CCC2(CC1)C3CCCCC3=NC(=C(N2)C#N)C#N KM00026 Cc1c(c(n(n1)C)NC(=O)c2ccc(cc2Cl)Cl)Cl KM00038 CS(=O)(=O)c1c(c(cs1)c2ccccc2Cl)C#N KM02577 COc1cccc(c1)c2c(nnc3n2nc(c3)c4ccccc4)C(=O)N KM00225 c1ccc(cc1)c2cc([nH]n2)NN=C(C#N)C#N KM00228 c1ccc2c(c1)cccc2CSCC(=O)NNC(=O)C(F)(F)F RH01661 CCOC(=O)C(=C(Nc1ccc(cc1)Cl)SC)C(=O)OCC KM08718 CCOC(=O)C1=C(OCC1=O)Nc2ccc(cc2)Cl KM08750 Cc1ccc(c2c1c(ccn2)O)C RH01798 c1ccc2c(c1)C(=O)N(C2=O)CCCO RH01831 CCCn1cnc2c1cccc2.Br NRB00676 CNC(=O)c1cccc2c1c(ccc2)I NRB00696 C/C(=N\NC(=O)N/N=C(/c1ccc(cc1)[N+](=O)[O-])\C)/c2ccc(cc2)[N+](=O)[O-] ML00294 CNC(=S)N/N=C/c1ccc(c(c1)Cl)Cl ML00309 CNC(=S)N/N=C/c1cc(cc(c1O)Cl)Cl ML00320 CNC(=S)N/N=C/c1ccccc1Cl ML00324 CC(=O)c1cc(c2c(c1)OCCO2)NC(=O)C NRB00895 Cc1cc2c(cc1C)Nc3c(c(=O)c3=O)N2 RDP00177 C1CCN(CC1)c2c(c(=O)c2=O)N3CCCCC3 RDP00193 CC1CCc2c(c3ccccc3[nH]2)C1 NRB05266 CCOC(=O)/C(=C/c1ccc(cc1)SC)/C#N P00095 c1cc(ccc1/C=N/NC(=S)Nc2cc(ccc2Cl)Cl)Cl RDR00385 c1cc(cnc1)C(=O)Oc2ccc(cc2)CC#N RF04720 COC(=O)c1cnc(cc1C(F)(F)F)Oc2ccc(cc2)N RF04728 Cc1cc(c2c(c1)occ(c2=O)C3C4=C(CC(CC4=O)(C)C)OC5=C3C(=O)CC(C5)(C)C)C RF00078 Cc1cc(c2c(c1)occ(c2=O)c3cc(c4cc5ccccc5cc4n3)C(=O)O)C RF00088 COc1ccccc1C2CCN(CC2)c3ccc(cc3)/C=C/C(=O)Nc4ccc(cc4Br)F RH01731 CCOC(=O)CCSc1cc(c(cc1[N+](=O)[O-])Cl)n2cccc2 RH01733 CC(=O)Nc1cc(n[nH]1)c2ccc(cc2)[N+](=O)[O-] KM08843 CSc1c(cn(n1)c2ccccc2)C(=O)Sc3ccc(cc3)Cl KM08845 Cc1c(c(no1)c2ccccc2Cl)C(=O)NCCNc3ccc(cc3[N+](=O)[O-])C(F)(F)F RH01918 CCOc1ccccc1/C=N/Nc2nc(cs2)c3ccccc3.Cl ML00167 c1cc(cc(c1)n2c(=O)[nH][nH]c2=S)C(F)(F)F ML00213 Cc1cccc(c1)n2c(=O)[nH][nH]c2=S ML00219 CCOC(=O)N/N=C/c1ccc(cc1)F ML00224 c1ccc2c(c1)cccc2NC(=O)NCCC(=O)O NRB00825 c1ccc2c(c1)NC(=O)CCN2C(=O)c3ccc(cc3Cl)Cl NRB00834 CNC(=S)NNC(=O)c1ccncc1 ML00391 c1cc2c(cc1CC(=O)O)OCO2 JFD00708 COc1cc(cc(c1OC)OC)/C=N/N=C(N)N.Cl JFD00737 c1cc(sc1)/C=N/N=C(N)N JFD00741 C/C(=N\N=C(N)N)/c1ccc(cc1)Br JFD00742 c1cc2c(nc1)Nc3c(c(nc(n3)N)O)S2 JFD00941 Cc1ccc2c(c1)cc3c(n2)c4c(n(c3=O)C)n(c(=O)n(c4=O)c5ccccc5)c6ccccc6 JFD00968 CC(C)(C)CN/C(=C(/C#N)\N=C\c1c(cccc1Cl)Cl)/C#N KM00233 c1ccc(cc1)n2c(c(c(n2)C3CC3)Br)NC(=O)C(Cl)(Cl)Cl KM00261 CC(C)(C)n1c(cc(n1)C2CC2)NC(=O)Nc3ccccc3 KM00290 CC(C)(C)C(=O)/C=C/1\NC(=O)CS1 KM00385 CC(C)(C)c1ccc(cc1)C(=O)/C(=C/c2ccccc2)/C#N KM00393 CN1C=NC(c2c1ccc(c2)Cl)(c3ccccc3)O RH01841 COc1ccc2c(c1)c(ccn2)[C@@H]([C@H]3C[C@@H]4CCN3C[C@@H]4C=C)O RH01857 CC(=O)c1ccc(s1)C#CCOC(=O)c2ccccc2 KM09009 Cc1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)CCS(=O)(=O)c4ccccc4 KM09042 c1ccc2c(c1)nc3c4cc(ccc4n(c3n2)C(=O)c5c(cccc5Cl)F)F RH01988 CCC(=O)Nc1cc(cc(c1)OC)OC RH02001 C=CCNC(=S)NNC(=O)c1ccc(cc1)O NRB00962 Cn1c(n[nH]c1=S)c2ccc(cc2)O NRB00970 c1cc(sc1)C2N(CCO2)C(=O)Nc3ccc(cc3)Cl MWP00264 CS(=O)(=O)NNC(=O)c1csc(n1)Cc2c3cc(ccc3sc2Cl)Cl MWP00311 Cc1c2cc(ccc2sc1CC(=O)NNC(=O)Nc3ccc(cc3)Cl)Cl MWP00371 CC(C(c1ccccc1)NC(=O)c2ccccc2)O NRB01480 CSC(=N)Nc1c(cccc1Cl)Cl.I RDR00490 c1ccc(cc1)/N=c/2\[nH]c(=O)c3ccccc3o2 PD00138 COc1ccc(cc1)N/N=C(\C#N)/c2ccccn2 PD00170 c1ccnc(c1)/C(=N/Nc2ccc(cc2)F)/C#N PD00171 CSC(=C(C#N)c1ccccn1)SC PD00174 c1cc(ccc1c2csc(n2)NCC3CCCO3)F RDR00932 CC(C)Oc1cc(c(cn1)C(=O)N(C)Cc2c(cccc2OC)OC)C(F)(F)F RF05409 CN(Cc1c(cccc1OC)OC)C(=O)c2cnc(cc2C(F)(F)F)OCC(F)(F)F RF05412 Cc1cc(c2c(c1)occ(c2=O)/C=C/3\C(=O)N(C(=S)S3)c4ccc(cc4)F)C RF00684 c1cc(sc1/C=N/NC(=S)N)[N+](=O)[O-] RF00709 Cc1ccc(cc1)S(=O)(=O)NNC(=O)c2ccc(cc2)n3c(ccc3C)C RH01948 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc3ccccc3c2O RH01954 COc1ccc(cc1)NC(=O)NCc2ccccc2 KM09304 COc1ccc(cc1OC)S(=O)(=O)N(CCC#N)CC2CCCO2 KM09305 COCCNc1cc(nc2c1cccc2)c3ccccc3 RH02078 CCCn1c(n[nH]c1=S)c2ccncc2 ML00400 Cc1ccccc1C(=O)Nc2ccc3c(c2)oc(n3)C MWP00029 CN(C)c1ccc(cc1C(F)(F)F)[N+](=O)[O-] NRB01082 CC(=O)N1CCN(CC1)c2ccccc2 NRB01139 c1ccc(cc1)C(=O)SC2=NCCc3c2cccc3 MWP00478 Cn1ccnc1S/C(=C/C=C(C#N)C#N)/c2ccc(cc2)Cl JFD00979 c1cc(oc1)C(=O)NNC(=S)Nc2c(cc(cc2Cl)Cl)Cl JFD00989 c1ccc(cc1)C2CNN=C2C(=O)c3ccccc3 JFD01087 c1ccc2c(c1)ccc(n2)N/N=C/c3ccccn3 JFD01295 COc1ccc(cc1)C2CS(=O)(=O)CS(=O)(=O)C2 JFD01342 Cc1cc(n2c(n1)c(c(n2)c3ccccc3)Br)C KM00429 CCOC(=O)c1c(n2c(cc(n2)C)nn1)C KM00447 CCOC(=O)c1cnc2c(c1N3CCCCC3)c(nn2C)C4CC4 KM00474 CN1c2ccccc2C(=O)/C(=N\Nc3ccccc3Cl)/S1(=O)=O KM00518 CC1CN(CC(O1)C)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Br KM00674 CCOC(=O)c1c(nc(c(c1O)[N+](=O)[O-])O)C KM00684 CCCc1ccc(cc1)S(=O)(=O)Nc2c(cccn2)OCc3ccc(c(c3)Cl)Cl RH02033 c1cc2c(c(c1)S(=O)(=O)N(CC/C(=N/OC(=O)Nc3ccc(cc3)OC(F)(F)F)/N)Cc4ccco4)nsn2 KM09370 CCOC(=O)c1csc(n1)n2cccc2 RH02260 c1ccn(c1)c2cc(ccc2n3ccnc3)[N+](=O)[O-] RH02263 COc1ccc2c(c1)sc(n2)/N=C/c3ccccc3[N+](=O)[O-] NRB01496 c1ccc(cc1)CC2(c3ccccc3N(C2=O)Cc4ccccc4)c5ccccc5 NRB01548 Cc1c2cc(ccc2sc1/C=N/Nc3c(cc(cc3Cl)Cl)Cl)Cl MWP00671 Cc1c2ccccc2sc1C(=S)Nc3ccccc3Cl MWP00775 c1cc(ccc1NC2=NNC(=O)C2)F MWP00813 c1ccc(cc1)NCCC(=O)c2ccc(s2)Cl MWP00900 COc1cc(cc(c1OC)OC)/C=N/NC(=S)NCC2CCCO2 RDR00937 c1ccc(c(c1)NC(=O)CCC(=O)O)F RDR01042 Cc1cccc(c1)NC(=S)N/N=C/c2ccc(cc2)F PD00357 CN(C)C(=S)Nc1cc(cc(c1)OC)OC PD00367 COc1ccc(c(c1)OC)/C=C/2\C(=O)N(C(=S)S2)CCc3ccc(cc3)Cl PD00394 c1ccnc(c1)/C=C/2\C(=O)N(C(=S)S2)CCc3ccc(cc3)Cl PD00395 COc1ccc(c(c1)Sc2ccc3nnc(n3n2)c4ccccc4)OC RH00147 CCCCCCCc1c(c2cccc3c2n(c1=O)CCC3)O RH00167 CCOC(CNc1ccc2nnc(n2n1)c3ccccc3)OCC RH00171 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3c(cccc3Cl)F RF01315 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C(\C)/c3ccco3 RF01348 Cc1ccc(cc1)Sc2c(cccn2)NS(=O)(=O)c3cc(ccc3OC)OC RH02107 C1CC(OC1)CNC(=S)NNC(=O)CC#N RH02156 c1ccc(cc1)NC(=O)NNC(=O)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09415 c1cc(oc1)CN(CCC(=O)NNS(=O)(=O)c2cccs2)S(=O)(=O)c3ccc(cc3)Cl KM09421 c1cc(ccc1C(=O)COC(=O)c2cc(c(cc2Br)C(=O)OCC(=O)c3ccc(cc3)Br)Br)Br RJC00089 CC(C)NC(=O)n1c(ccn1)c2ccc(cc2Cl)[N+](=O)[O-] MWP00484 Cc1c2cc(ccc2sc1C(=O)/C(=C\c3ccc(cc3)[N+](=O)[O-])/C#N)Cl MWP00554 C1C2CC3(CC1CC(C2)(C3)Br)C(=O)N NRB01923 Cc1ccc(cc1)S(=O)(=O)OC2CC3CC2C(C3)[N+](=O)[O-] NRB02174 Cc1ccc(cc1)S(=O)(=O)NC(C)(C)C NRB02436 c1ccc(cc1)Sc2c(=O)c(=O)c2Sc3ccccc3 MWP00916 COc1cc(ccc1O)C2C(S(=O)(=O)CS(=O)(=O)C2C(=O)OC)C(=O)OC JFD01349 c1ccc(cc1)C(c2ccccc2)N3CC(C3)Oc4ccccc4 JFD01367 CC1CCC(C(C1)NC(=O)c2ccco2)C(C)C JFD01384 c1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(cc2)C(F)(F)F JFD01391 c1cc(ccc1C2SCCS2)NC(=O)CSc3ccc(cc3)Cl KM00711 Cc1cc(n2c(n1)c(cn2)/C(=N/OC(=O)NC(C)C)/N)C KM00765 CCCCNC(=O)Nc1ccc(cc1)C2SCCS2 KM00783 Cn1c(c(c(n1)c2ccccc2)C#N)SC KM00808 Cc1c(c(n(n1)CC(=O)NN)C)Br KM01023 Cc1cc(cc(c1)N/C=C(\C#N)/S(=O)(=O)Cc2ccc(cc2)Cl)C KM01036 CCOC(=O)COc1ccc(cc1C(=O)OC)Cl RH02265 CCCCC#Cc1ccc(o1)C(=O)N/N=C/c2cccc(c2)OC KM09524 c1ccc(cc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccccn4 KM09542 c1ccc(cc1)CN2CCN(CC2)CCS(=O)(=O)c3ccc(cc3)Cl KM09885 CN1CCC(=NOC(=O)Nc2ccccc2)CC1 KM09921 c1ccc(cc1)c2cc(=S)c3ccccc3o2 NRB02689 c1ccc2c(c1)c3c([nH]2)CCCCC3 NRB02757 Cc1ccccc1N/C=C\c2nnnn2c3ccc(cc3)F NRB03305 c1cc(ccc1N/C=C\c2nnnn2c3ccc(cc3)Cl)Cl NRB03326 Cc1cccc(c1n2c(=O)c3ccccc3nc2SC)C RDR01344 c1ccc(c(c1)CSc2nccn2c3cccc(c3Cl)Cl)Cl RDR01359 c1ccc2c(c1)C(=O)C(=Cc3ccncc3)C2=O S12977 c1ccc(cc1)N2C(=O)CC(C2=O)SCC(=O)O S12991 c1ccc2c(c1)c(cs2)CN3C(=O)c4ccccc4C3=O S13297 c1cc(sc1)CNC(=S)NNc2c(cncc2Cl)Cl RF01350 c1ccnc(c1)/C=N/Nc2c(cncc2Cl)Cl RF01356 Cc1cc(c2c(c1)occ(c2=O)C#N)C RF01381 c1cc(sc1)C(=O)Nc2nnc(s2)Sc3ccnc4c3ccc(c4)Cl RH00426 c1cc(ccc1N)n2c(cc(n2)C(F)(F)F)C(F)(F)F SEW04192 c1ccc2c(c1)NC(=O)CC(S2)c3ccsc3 SEW04201 c1cc(c(cc1C#N)[N+](=O)[O-])SCCO SEW04232 c1cc(ccc1C(=O)COC(=O)c2cc(ccc2I)Cl)Br RJC00107 Cc1c(c(=O)c2c(cc(cc2o1)O)O)c3ccccc3 RJC00209 CC(=O)c1ccccc1OC(=O)c2ccccc2 RJC00235 CC1(C2CCC1C(C2O)O)C RJC00236 Cc1ccccc1NC(=O)NCc2ccccc2 KM09674 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)c(c[nH]3)Cl SP01353 Cc1ccc(cc1)Oc2c(cccn2)C(=O)NC(=O)c3ccccc3O HTS10048 Cc1ccc(cc1)S(=O)(=O)Nc2cccc3c2cc(nn3)C HTS10060 c1ccc2c(c1)C(C(=O)N2)Cc3ccccn3 HTS10082 c1ccc(cc1)NC(=O)N2CCCc3c2cccc3 HTS10195 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4cn(nc4c5ccc(cc5)[N+](=O)[O-])c6ccccc6)C HTS10371 CCOC(=O)/C(=N/Nc1ccc(cc1)Br)/C(=O)C JFD01761 CCOC(=O)/C(=N/Nc1ccc(cc1)F)/C(=O)C JFD01763 c1ccc(cc1)/C=C/C=N/c2ccccc2 JFD01779 CCO/C=C\1/c2ccc(cc2C(=O)N(C1=O)c3ccc(cc3)C)OC JFD01786 CCCCCCCCC(=O)CCCCCCCCC(=O)OC JFD01973 c1cc(sc1S(=O)(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl KM01046 CSc1c(c(nc(n1)SC)c2cccs2)C#N KM01065 CC(C)Oc1cccc(c1)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM01127 Cn1c2c(c(cc(n2)O)COC)c(n1)c3ccccc3 KM01148 CSc1c(c(nc2c1c(c(s2)C(=O)c3ccccc3)N)N)C#N RH00564 CCOC(=O)COc1ccc(c2c1CCC2)C RH00583 c1ccc2c(c1)c(c[nH]2)CCNS(=O)(=O)c3cccc4c3nsn4 KM09925 CN1C(=O)/C(=N/Nc2ccc(cc2)C(F)(F)F)/C(=N1)Nc3ccccc3Cl MWP01012 CN(C)c1cc(c2ccccc2n1)NC(=O)Nc3ccccc3 MWP01055 CC(=O)OC[C@H]([C@H]([C@@H]([C@H](C(=O)N1CCOCC1)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C RJC00837 COc1ccc(cc1)NC(=S)NC2CCCCC2 S04694 C1CCN(C1)c2nnn(n2)CC(=O)O RJF01912 CC(C)(C)C(=O)COC(=O)Cn1nc(nn1)N2CCCC2 RJF01929 CCCc1cc(=O)oc2c1ccc(c2)OCC(=O)NNC(=O)NC(C)C RJF01994 c1cc(cc(c1)S(=O)(=O)NNC(=O)Cn2nc(nn2)c3cc(cc(c3)Cl)Cl)C(F)(F)F RJF02012 c1cc(ccc1C2c3ccsc3CCN2C(=O)c4ccc(cc4)C(F)(F)F)C(F)(F)F SEW01205 c1ccc2c(c1)c(nc(=O)o2)Nc3ccc(cc3)OC(F)(F)F S14029 CCOC(=O)C(C)c1ccc2cc(ccc2c1)OC S14045 c1ccc2c(c1)CCCC23CC(=O)N(C3=O)CN4CCOCC4 S14061 c1ccc2c(c1)CCC2(CC#N)C#N S14065 Cc1cc(no1)NC(=O)CCOc2ccc(cc2)F SEW01429 c1ccn(c1)c2cccnc2NNS(=O)(=O)c3ccc(c(c3)Cl)Cl SEW04305 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=O)COCC(=O)O)C(F)(F)F SEW06185 c1ccc2c(c1)nc(s2)SCC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl SEW06195 COCCCNC(=S)N/N=C/c1ccc(s1)c2ccc(cc2)OC SEW04651 Cc1c(c(no1)c2c(cccc2Cl)Cl)/C=C/3\c4ccccc4NC3=O SEW04685 Cc1c(cc(o1)S(=O)(=O)NCc2cccs2)C(=O)OC SP01429 c1ccc(cc1)n2c(nnn2)/C=C/Nc3ccccc3C#N RJC03189 CC1(O[C@@H]2[C@H](O[C@H](C2O1)n3cnc4c3ncnc4N)CO)C RJC03233 c1cc(ccc1C23CC4CC(C2)CC(C4)C3)[N+](=O)[O-] RJC00945 c1ccc(c(c1)n2c(c(cn2)c3nnnn3c4ccc(cc4)F)C(F)(F)F)Cl HTS10382 c1cc(cc(c1)Cl)N2CCN(CC2)/C=C/c3nnnn3c4ccc(cc4)F HTS10409 C/C(=N\O)/C(C)(C)Nc1ccc(cc1)Br HTS10429 c1cc(ccc1NC(=O)NCC2CC2)Cl HTS10467 Cc1ccc(cc1)Sc2cccc3c2c(nc(n3)N)N MWP01127 CCc1ccc(cc1)NS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F MWP01136 c1ccc(c(c1)CSc2nc3ccccc3s2)[N+](=O)[O-] JFD01988 CCOC(=O)CNC(=O)c1cc(c(c(c1)OC)OC)OC JFD02035 COc1ccc(cc1OCc2ccccc2)C3C4CCc5ccccc5C4=Nc6ccccc6S3 PD00591 CC(C)CC(C(=O)O)NCc1ccccc1O RH00617 Cc1cc2c3c(c1)c(c(c(=O)n3CCC2)c4ccccc4)OC(=O)c5c(cccc5Cl)F RH00703 COC(=O)c1cc(c(s1)Br)Br RH00748 CC1(CC(=O)Nc2ccccc2S1)C RJC00304 CCS(=O)(=O)c1ccc(cn1)C#N SEW04447 Cc1c(c(c(c(c1C)NC(=O)C)NC(=O)C)C)C SEW04472 c1ccc2c(c1)C(=O)C3(C2=O)N4[C@H](CS3)C(=O)N5[C@@H](C4=O)CSC56C(=O)c7ccccc7C6=O RJC00877 CNc1[nH]c2c(n1)n(c(=O)n(c2=O)C)C RJC03298 C(C(=O)O)N(CC(=O)O)[N+](=O)[O-] RJC00998 CCc1ccc2c(c1)c(=O)c3cc(c(nc3o2)N)C#N RJC01066 c1cnc(nc1)c2ncccn2 RJC01086 c1cc2c(cc1Cl)CCC2=O RJC01116 c1cc2c(cc1NC(=S)NCCO)OCCO2 S05269 c1ccc(cc1)CNC(=S)C(=O)Nc2ccccc2C#N NRB00073 Cc1ccc(cc1)SCC(=O)Nc2cc(cc(c2)Cl)Cl NRB00076 CSc1cccc(c1)NC(=O)C(=S)NC2CCCCC2 NRB00087 c1cc(ccc1SC(CC(=O)O)C(=O)O)Cl SEW01463 CCOc1ccccc1/C=C/2\C(=O)OC(=N2)c3ccc(cc3)Cl PHG00631 c1cc(cc(c1)[N+](=O)[O-])C(=O)NCC(=O)O PHG00644 c1ccc(c(c1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)[N+](=O)[O-])Cl PHG00687 COc1cc(cc(c1OC)OC)C(=O)NCC(=O)O PHG00717 c1ccc2c(c1)[nH]c(n2)/C(=C/c3cccc(c3)[N+](=O)[O-])/C#N PHG00722 CSc1c(c(sn1)SC)C(=O)NCCSCc2ccc(cc2)Cl SEW06367 c1cc(c(nc1)N2CCN(CC2)c3ccc(cn3)NC(=O)Nc4ccc(cc4)C(F)(F)F)C(F)(F)F SEW06382 Cc1ccc(cc1)C(=O)N2CCC(CC2)C(=O)c3c(cc(cc3C)C)C SEW06387 CC(=CC(=O)OCC(=O)c1ccc(cc1)C(F)(F)F)C RF03431 c1cc(ccc1C(=O)COC(=O)COCC(=O)OCC(=O)c2ccc(cc2)C(F)(F)F)C(F)(F)F RF03434 Cc1c(nc(s1)C)C23CC4CC(C2)CC(C4)C3.Cl RJC00962 C1CC2CC3CC1CC(C2)(C3)C(=O)N RJC00968 CCc1c(c(c(=O)n(c1c2ccccc2)c3ccccc3)C(=O)C)O RJC03392 c1cc2c3c(c1)C(=O)C(C(=O)N3CCC2)(Cl)Cl RJC03400 CCOC(=O)C1=C(NC(=C(C1c2ccc(c(c2)OC)OC)C(=O)OCC)C)C RJC03407 CCOC(=O)c1cc(cnc1)C#CC(C)(C)O KM08284 CNC(=S)N1CCOC1c2ccc(s2)[N+](=O)[O-] MWP01163 c1ccc(cc1)S(=O)(=O)NC(=S)Nc2ccc(c(c2)Cl)Cl NH00081 c1ccc(c(c1)C(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)NCc3ccccn3 NH00137 c1ccc2c(c1)C(=O)N3C2(NCC3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F NH00156 Cc1cc(c(c(c1)Br)NC(=S)NC(=O)C(C)(C)C)Br NH00563 Cc1ccc(cc1)N2C(CC(=N2)c3ccccc3)c4ccc5c(c4)OCO5 PD00625 c1ccc(c(c1)CSc2ccc(cn2)C(F)(F)F)C(=O)O PD00635 C=CCOc1ccc(cc1)C=C2C(=O)c3ccccc3C2=O PD00643 COc1ccc(c(c1OC)Cl)/C=C/2\CCc3ccccc3C2=O PD00645 CC(=O)Nc1ccc(cc1)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] PHG00074 c1cc(ccc1c2cc3cc(cc(c3oc2=O)Br)Br)[N+](=O)[O-] PHG00101 C/C(=N\OC(=O)Nc1ccccc1)/c2ccc3cc(ccc3c2)OC SEW04533 Cc1cc(c(o1)C)C(=O)Nc2ccc(cc2)OC(F)(F)F SEW04544 c1cc2c(cc1OCC(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl)OCO2 SEW06222 COc1cccc(c1OC)/C=N/Nc2c(cccn2)[N+](=O)[O-] SEW04733 c1cc(sc1)c2nc(on2)Cc3cc(cc(c3)F)F SEW04740 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NCc3ccccc3)CC(CN4CCN(CC4)Cc5ccccc5)O RJC03465 CCC(CNCCO)Nc1nc2c(n1Cc3ccccc3)c(=O)n(c(=O)n2C)C RJC03502 c1ccc(c(c1)C(=O)Nc2ccc3c(c2)C(=O)OC3)Cl KM08471 Cn1c(nnc1SCC(=O)Nc2cccc(c2)C(F)(F)F)c3cc(cnc3)C#Cc4ccccc4 KM08503 c1cc(ccc1NC(=O)OCCSCc2ccc3c(c2)ccc(n3)C(F)(F)F)Cl KM08528 CC(C)(C)c1ccc(cc1)NC(=O)C(=S)NCc2ccco2 NRB00158 Cc1cc(oc1C)/C=C\2/C(=O)NC(=S)S2 NRB00393 COc1ccc(cc1OC)/C=C(\C#N)/c2[nH]c3ccccc3n2 PHG00727 CN(C)N1C(=O)c2cccc3c2c(cc(c3)[N+](=O)[O-])C1=O PHG01005 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)CCCN4CCN(CC4)CCCN5C(=O)c6cccc7c6c(cc(c7)[N+](=O)[O-])C5=O)[N+](=O)[O-] PHG01009 c1cc2cc(cc3c2c(c1)C(=O)N(C3=O)CC(=O)O)[N+](=O)[O-] PHG01014 Cc1ccc(cc1C)NC(=S)Nc2ccc(c(c2)Cl)Cl RB00012 CSC1=N/C(=C\Nc2cccc(c2)Cl)/C(=O)N1Cc3ccccc3Cl RF03509 c1ccnc(c1)c2nc3c(c(n2)O)CSCC3 RF03877 COc1cc(c(cn1)C(=O)NCc2c(cccc2Cl)Cl)C(F)(F)F RF04360 c1cc2c(cc1C(F)(F)F)N(C(=O)CS2)CC(=O)NN KM08301 Cc1cc(no1)C(=O)N=S(=O)(C)c2cccs2 KM08349 COc1c(csc1S(=O)(=O)N=S(=O)(C)c2cccs2)C(=O)OC KM08429 CN(CCOC(=O)Nc1ccc(cc1)OC(F)(F)F)c2cc(nc3c2cccc3)C(F)(F)F KM08434 CCCNC(=S)NCCO NH00750 Cc1ccc(cc1)SCC(=O)Nc2ccc(cc2)I NRB00030 c1cc(c(cc1F)F)NC(=O)C(=S)N2CCOCC2 NRB00047 Cc1ccc(cc1)C(=O)/C=C/Sc2ccc(cc2)C NRB03902 CC(C)(C)OC(=O)N1CCCN(CC1)C(=O)Nc2cc(cc(c2)Cl)Cl HTS11281 Cc1[nH]nc(n1)c2cccc(c2)Cl HTS11299 CCCCN1C(=O)c2cccc3c2c(cc(c3)[N+](=O)[O-])C1=O PHG00252 c1cc(cc(c1)Cl)C(=O)NCC(=O)O PHG00472 COc1ccc(cc1)/C=C/2\C(=O)OC(=N2)c3cccc(c3)Cl PHG00497 C#CCSc1nc2ccccc2c(=O)n1c3ccc(cc3)F RDR02381 Cc1ccc(cc1)C(=O)NC(C)CCc2ccc(c(c2)OC)OC(=O)c3ccc(cc3)C JFD02574 CC(CCc1ccc(c(c1)OC)OC(=O)c2ccc(cc2)Cl)NC(=O)c3ccc(cc3)Cl JFD02577 c1cc(ccc1S(=O)(=O)CCC(=O)O)Cl SEW04754 CCOC(=O)c1c(nn(c1C)c2c(cccn2)NC(=O)Nc3cccc4c3cccc4)C SEW04761 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCCSCc2c(cc(cc2C)C)C SEW06445 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2cccc3c2cccc3)C SEW06451 CNC(=O)O/N=C/c1c(c[nH]n1)Br RF03961 c1ccc(c(c1)C(=O)NC(=O)C(=O)Nc2ccc(cc2F)Br)Cl RF03991 COc1ccc(cc1)C(=O)/C(=C/NC2CCN(CC2)Cc3ccccc3)/C#N KM08560 CCOC(=O)NC(=O)c1cn(c(=O)[nH]c1=O)Nc2ccc(cc2F)F KM08772 CCOC(=O)c1c(c2cc(ccc2nc1SC)Cl)Oc3ccccc3 KM08804 c1ccc(c(c1)NC(=O)CSc2c(c(cc(c2Cl)Cl)Cl)Cl)Cl KM08815 c1ccc2c(c1)c(cc(n2)C(F)(F)F)N3CCN(CC3)C(=O)Nc4cc(cc(c4)Cl)Cl KM08841 Cc1cc(oc1C)C=C2C(=O)OC(OC2=O)(C)C NRB00479 c1cc(oc1CS(=O)(=O)C(Cl)(Cl)Cl)[N+](=O)[O-] NRB00496 CNC(=O)c1ccccc1I NRB00705 COc1ccc(c(c1)C(=O)O)Sc2ccccc2C(=O)O NRB00728 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3ccc4c(c3)OCO4 RB00023 CC1=Nc2cc(c(cc2NC(C1)(C)C)Cl)Cl RDP00237 c1cc2c(cc1C(F)(F)F)nccn2 RDP00242 C1CCN(C1)c2c(c(=O)c2=O)N3CCCC3 RDP00244 c1ccc(cc1)CCN\2C(=O)CS/C2=N\c3cc(c(cc3Cl)Cl)Cl RDR00098 c1ccc(cc1)c2csc(n2)Nc3cccnc3 RDR03651 Cc1cccc(c1C)NC(=O)c2cnc(cc2C(F)(F)F)OC RF04388 c1ccc(cc1)NC(=O)NC(=O)c2cnccc2C(F)(F)F RF04461 COc1cc(cc(c1)OC)CNC(=O)c2cnc(cc2C(F)(F)F)OC RF04469 CC(=O)NNc1c(cc(cn1)C(F)(F)F)Cl RF04804 CCOC(=O)NNc1c(cccn1)C(F)(F)F RF04965 c1ccn(c1)C2CCN(CC2)C(=O)c3ccc(cc3)Cl KM08579 CC(C)(C)OC(=O)c1cccc(c1)NC(=O)Nc2ccc(cc2)OC(F)(F)F KM08589 c1ccc(cc1)C#Cc2cc(cnc2)NC(=O)Nc3cccc(c3)C(F)(F)F KM08617 c1ccc(cc1)C#Cc2ccc(o2)C(=O)Nc3ccc(cc3)Cl KM08631 Cc1c(c(c([nH]1)C)C(=O)OC)/C=C(\C#N)/C(=O)c2cccs2 KM08854 C/C(=N\O)/C(C)(C)Nc1ccccc1F HTS11323 Cc1cc(n(n1)c2nc3c(n2Cc4ccc(cc4Cl)Cl)c(=O)n(c(=O)n3C)C)C HTS11453 c1ccc(cc1)Cn2c3ccccc3[nH]c2=O HTS11479 c1ccc(cc1)c2c(c3nnnn3nc2c4ccccc4)c5nnc(o5)S JFD00400 CSc1nnc(n1/N=C/c2cn(nc2c3ccc(cc3)Cl)c4ccccc4)c5ccncc5 HTS11981 COc1ccc2c(c1)c(=O)cco2 JFD02610 Cc1c(c(c(c(c1C)C)C(=O)/C(=C/c2ccccn2)/C)C)C JPV00044 COc1cc(c(cc1OC)Br)OC JFD02748 Cc1c(c(=O)n(n1C)c2ccccc2)/N=C/c3ccc(o3)c4ccccc4[N+](=O)[O-] JFD02779 CC(C(C(=O)OC)NC(=O)OCc1ccccc1)O JFD02830 CN(C)C(=O)Nc1cnccc1C(F)(F)F RF03994 CCC(CC)(C#C)NC(=O)Nc1cnccc1C(F)(F)F RF04023 Cc1ccc(cc1)c2nnnn2c3ccccc3C(F)(F)F RF04542 Cc1ccc(c(c1)C)c2csc(n2)c3ccncc3.Br ML00036 COc1ccc(cc1)Nc2nnns2 ML00063 Cn1c(nnc1SCc2ccc(cc2)OC(F)(F)F)CSCC(=O)Nc3ccccc3 KM09093 c1cc(ccc1NC(=O)CSCC(=O)NNC(=O)Nc2cc(cc(c2)Cl)Cl)OC(F)(F)F KM09104 CC(=O)NC(=O)/C(=C/N1CCN(CC1)c2ccccc2)/C#N KM09188 c1csc(n1)/N=C/c2cc(cc(c2O)Cl)Cl ML00233 c1ccc2c(c1)nc3n2C(=O)CS3 NRB04602 Cc1ccc(cc1C#N)NC(=O)CSc2nnnn2c3ccccc3 NRB04686 C=CCn1c(n[nH]c1=S)COc2ccccc2 NRB00976 c1cnc(nc1)S(=O)(=O)[O-].[Na+] NRB01033 C[C@@H](C(=O)O)NC(=O)OC(C)(C)C NRB05199 c1ccc(cc1)/C(=C/C(=C/N2CCOCC2)/c3ccccc3)/C#N NRB05228 c1cc(ccc1C2=NCCO2)C(F)(F)F RDR03677 CC(C)CCCC(C)C1CCC2C1(CCC3C2CCC4=C/C(=N/NC(=S)Nc5ccc(cc5)F)/CCC34C)C RDR00517 CC(=O)CCCNc1nc(cs1)c2ccc(cc2)Cl.Br RDR00830 Cc1cc(nc(c1C#N)OC(=O)c2c(cccc2F)F)C RF00030 Cc1cc(nc(c1C#N)N2CCOCC2)C RF00043 c1c(c(n[nH]1)/C=N/O)[N+](=O)[O-] RF05017 COc1ccccc1N/C(=N\O)/c2ccccc2Cl RF05149 CCOC(=O)/C(=N/Nc1ccc(cc1)C)/C RH01686 c1ccn(c1)c2cc(c(cc2Cl)[N+](=O)[O-])Sc3[nH]c(nn3)N RH01687 CC(=O)c1ccccc1OC(=O)c2cccs2 RG00010 c1ccc(c(c1)c2cc(n[nH]2)c3ccc(cc3)Cl)O RG00016 c1c(c(sc1S(=O)(=O)N)N2CCCCC2)[N+](=O)[O-] KM08940 Cn1c2c3cccc(c3nc(c2c(=O)n1Cc4ccc(cc4)Cl)SC)Cl KM08964 CC(C)(C)c1cc2nc(cc(n2n1)N3CCNCC3)C(F)(F)F KM08987 COc1ccc(cc1)/C=N/NC(=S)NCCc2ccccc2 ML00122 c1c(cc(c(c1)Cl)Cl)/C=N/NC(=O)N/N=C/c2cc(c(cc2)Cl)Cl ML00133 c1cc(ccc1/C=N/NC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F)C(F)(F)F KM09321 c1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/n4c(n[nH]c4=S)c5cccs5 HTS11985 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/NC(=O)c4ccncc4 HTS11990 CCn1c(nnc1SCC(=O)Nc2cc(nn2c3ccccc3)C)c4cccs4 HTS12038 CCOC(=O)C(C(=O)C)Sc1c2c(c3c(cc(nc3s2)C)C)ncn1 HTS12100 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)N/N=C/c4ccccc4Cl)N)c5ccco5 HTS12137 c1ccc2c(c1)c(=O)c3ccc(cc3o2)O JFD02834 c1ccc(cc1)C(c2ccccc2)(c3ccccc3)N4C(=O)C(SC4=O)Cc5ccc(cc5)O JFD02849 Cc1cc(c(c(c1S(=O)(=O)NC(=N)NCCCC(C(=O)NC(CC(=O)OC(C)(C)C)C(=O)NC(CC(C)C)C(=O)NC(CCCCNC(=O)OC(C)(C)C)C(=O)NCC(=O)O)NC(=O)OCC2c3ccccc3-c4c2cccc4)C)C)OC JFD02948 CCN(c1c(cccc1C)C)C(=O)c2c(ccnc2OCC)C(F)(F)F RF04613 CCN(c1c(cccc1C)C)C(=O)c2c(ccnc2NC)C(F)(F)F RF04614 CC1CCC(C(C1)NCc2ccccc2)C(C)C.Cl RH01600 COc1ccccc1C2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RH01607 Cc1cccc(c1)C(=O)Nc2nccs2 ML00256 COc1ccc(cc1)c2nc(cs2)c3ccc(cc3)Br.Br ML00287 c1cc(cc(c1)C(F)(F)F)C(=O)NNC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F KM09384 c1cc(oc1)c2cc3nc(cc(n3n2)C(F)(F)F)c4ccncc4 KM09393 Cc1nc2ccc(cc2o1)NS(=O)(=O)c3ccccc3C(F)(F)F MWP00041 Cn1c2ccccc2c(c(c1=O)Cc3ccccc3)OS(=O)(=O)c4ccccc4 NRB05244 Cc1nc(c(o1)c2ccc(cc2)[N+](=O)[O-])c3ccc(cc3)S(=O)(=O)N/N=C\c4ccc(c(c4)OC)OC NRB01527 CCCCc1c(c2ccccc2n(c1=O)CCCC)O NRB01602 CCCCC1(C(=O)N(N(C1=O)c2ccccc2)c3ccccc3)COC(=O)c4ccc(cc4Cl)Cl PD00126 Cc1cc(nc(c1C#N)Sc2ccc(cc2)Cl)C RF00044 Cc1ccc(cc1C)/N=C/c2ccc(cc2)Cl RDR01060 Cc1ccc(cc1C)/N=C/c2ccc(cc2)OC RDR01061 Cc1ccc(cc1)S(=O)(=O)NNC(=S)NCCc2ccccc2 RDR01071 c1ccc(cc1)c2[nH]c(nn2)SCC(=O)c3ccc(cc3)Cl RF00495 CCCCCCCCCCCCSC(=S)Nc1ccc(cc1)OC RF00590 CC(C)(C(=O)Nc1ccccc1)Oc2ccc(cc2)C#N RH00012 CC1CCC(=C(C)C)/C(=N/O)/C1 RH01861 c1ccc(cc1)N/N=C/C(=N/Nc2ccccc2)/[C@H]([C@@H](CO)O)O RH01878 CSc1[nH]c2cc(c(cc2n1)Cl)Cl RH00196 c1cc2c(c(c1)S(=O)(=O)N(CCC#N)Cc3ccco3)nsn2 KM09330 CS(=O)c1ccc(cc1)n2c3c(c(=O)n(c2=O)Cc4ccccc4)[nH]cn3 KM09352 c1ccc(c(c1)n2c(n[nH]c2=S)c3ccco3)Cl ML00338 Cc1ccc(c(c1)C)C(=O)CSc2nnc(n2c3ccc(cc3)OC)c4ccncc4.Br ML00377 c1cc(sc1)C2=NOC(C2)(C(F)(F)F)O KM09440 c1cc2c(cc1Cl)c(cc(n2)C(F)(F)F)O KM09476 c1ccc(cc1)c2nnc(n2c3ccccc3)Sc4c5c(ncn4)n(nn5)Cc6ccccc6Cl HTS12148 c1ccc(cc1)Cn2c3c(c(ncn3)Nc4cccc(c4)C(F)(F)F)nn2 HTS12166 COc1ccc(cc1)C2C(=C3c4cc(c(cc4CCN3C(=C2C#N)N)OC)OC)C#N HTS12242 CC\1=NN(C(=O)/C1=C/2\N(N=C(S2)C(=O)c3ccccc3)c4ccccc4)c5ccccc5 HTS12247 c1ccc2c(c1)nc(s2)S/C(=C/C=C(C#N)C#N)/c3ccc(cc3)Br JFD03033 Cc1ccc(cc1)/C=N\Nc2c(nc3ccccc3n2)/C=C/c4cccs4 JFD03051 C(CSc1c(sc(=S)s1)SCCC#N)C#N JFD03079 c1cc(ccc1Nc2ccc(cc2)F)[N+](=O)[O-] JFD03234 c1ccc(cc1)COc2ccc(cc2)/C=C(\C#N)/C(=O)O JFD03249 COc1cc(c(cc1/C=C(\C#N)/C(=O)O)C(=O)OC)OC JFD03257 C#CCOC(=O)Nc1ccc(nc1)Sc2ccccc2 RF05314 c1cc(ccc1c2csc(n2)N/N=C\c3cc[nH]n3)Cl RF05375 c1cc(c(c(c1)Cl)c2nc(on2)c3ccno3)Cl RF05388 Cc1ccc(c2c1CCC2)OCc3nnc(n3c4ccccc4)SCC(=O)c5cccc(c5)Cl RH01734 c1cc(cc(c1)Cl)C(=O)c2cc3cc(ccc3o2)[N+](=O)[O-] RH01745 Cc1c2ccccc2sc1CC(=O)N(C)C MWP00132 c1ccc2c(c1)c(cs2)C/C(=N/O)/N MWP00245 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccccn3 KM09551 CC(=O)c1cc2c3ccccc3ccc2c4c1cccc4 KM09650 COc1ccc(cc1)/C=N/NC(=O)c2ccc3c(c2)non3 KM09653 CNC(=S)NNC(=O)c1ccc2c(c1)non2 KM09668 Cc1c2ccccc2sc1/C=N/Nc3ccccn3 MWP00622 c1ccc(cc1)C2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl PD00134 c1ccc(cc1)NC(=O)C2=Cc3ccccc3/C(=N/Nc4ccc(cc4)C#N)/C2=O NRB02905 COc1cccc(c1)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-] NRB02942 c1ccc(c(c1)C(=O)Nc2ccc(cc2)Br)[N+](=O)[O-] PD00340 COCCCNC(=S)Sc1ccc(cc1)Cl RF00612 c1ccc(c(c1)C(=O)Nc2cccc(c2)[N+](=O)[O-])O RDR01399 c1ccc(c(c1)C(=O)Nc2ccc(cc2)/N=C/c3ccc(cc3)Cl)O RDR01415 c1ccc(c(c1)C(=O)O)NC(=O)c2ccc(cc2)Cl RDR01446 Cc1cc(=O)oc2c1ccc(c2C)O RDR01466 Cc1cc(=O)oc2c1cc(c(c2)OC(=O)c3ccc(cc3)[N+](=O)[O-])Cl RDR01498 CC(C)(C)c1ccc(cc1)Oc2c(cccn2)NC(=O)c3ccccc3 RH02071 c1ccc(c(c1)C(F)(F)F)S(=O)(=O)Nc2c(cccn2)OCc3cc(cc(c3)F)F RH02077 c1ccc(c(c1)NC(=S)N2CCc3c2ccc(c3)[N+](=O)[O-])Cl RH00440 c1ccc(cc1)/C=C\2/C(=O)/C(=C/c3ccccc3)/CCC2 RH00503 CCOC(=O)c1cnc2c(c1N3CCC(CC3)n4cccc4)c(nn2C)C KM09482 Cc1c2ccccc2sc1c3ccn[nH]3 MWP00406 Cc1c2cc(ccc2sc1c3ccnc(n3)SCc4ccccc4)Cl MWP00472 CCOC(=O)c1c(c(c(=O)oc1C)Br)C KM09732 c1ccc(c(c1)Cn2c(=O)cc(n(c2=O)c3ccccc3C(F)(F)F)N)F KM09735 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)NC3CCCC3)Cc4cccc(c4)Br HTS12277 Cn1c2c(nc1Oc3ccccc3Cl)n(c(=O)n(c2=O)C)C HTS12286 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)Oc3ccc(cc3Br)Br)Cc4ccccc4 HTS12289 CC(=O)C1=NN(/C(=C\2/C(=NN(C2=O)c3ccccc3)c4ccccc4)/S1)c5ccc(cc5)Cl HTS12379 CCOC(=O)c1c2nc(c3ccccc3n2nn1)SCc4ccc(cc4)F HTS12454 CC1=C(C(C(=C(N1)C)C(=O)OC)c2ccc(cc2)OCc3ccccc3)C(=O)OC JFD03270 CCOC(=O)COc1ccc(cc1)C2C(=C(NC(=C2C#N)C)C)C#N JFD03275 Cc1ccc(cc1)C2C(=C(NC(=C2C#N)C)C)C#N JFD03277 CC(=O)c1ccc(cc1)/N=N/c2ccc3c(c2)CCCN3CCC#N JFD03408 c1ccc(cc1)/C=C/c2c[nH]c3c2cccc3 JFD03411 CCOC(=O)Cc1nnc(o1)c2ccc(cc2)Cl RH00091 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)c5c4CCCC5)OC(=O)c6ccc(cc6)[N+](=O)[O-] RH00121 Cc1ccc(n1c2ccc(cc2)C(=O)NNS(=O)(=O)c3ccccc3)C RH01962 c1ccc2c(c1)c3ccccc3n2CC(=O)NN RH01973 CC(=O)n1c2ccc(cc2c3c1nc4ccccc4n3)F RH01975 CC1NCCN(C1)Cc2ccccc2.C(=C/C(=O)O)\C(=O)O.C(=C/C(=O)O)\C(=O)O RH00316 Cc1c2cc(ccc2sc1C(=O)/C(=N/Nc3ccc(cc3)C(C)C)/C#N)Cl MWP00655 c1cc(c(nc1)Sc2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F)C(F)(F)F MWP01066 c1ccc(cc1)CNC(=O)N/N=C/c2cccs2 MWP01091 c1ccc(cc1)N/C=C\c2nnnn2c3ccccc3 NRB03222 CC(=O)SC1CC(=O)N(C1=O)c2ccc(cc2)Cl PD00352 COc1ccc(cc1)CNC(=S)NCCCO PD00356 Cc1cc(nc(c1)NC(=S)Nc2cccc(c2)F)C S04876 CC(C)(C)NC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F S04979 c1ccc(cc1)/N=N/c2nnc(s2)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F S04996 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccccc3C(C)C S05018 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3c(cncc3Cl)Cl RF01234 c1cc(cc(c1)NC(=O)c2cccs2)c3nnco3 SEW01223 c1cc(cc(c1)NC(=O)c2ccc(o2)[N+](=O)[O-])c3nnco3 SEW01224 CC(C)(C)C(=O)Nc1cccc(c1)c2nnco2 SEW01228 c1ccc(cc1)/C=C/2\Cc3ccccc3C2=O RH00518 CCCCc1ccc(c(c1)C)NC(=O)CSc2nc(c(o2)c3ccccc3)c4ccccc4 RH00533 c1ccc(cc1)c2c(nnc(n2)N3CCOCC3)c4ccccc4 RJC00063 CCCCCC(=O)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06205 C=CCNC(=S)Nc1ccc(nc1)N2CCN(CC2)c3ccc(cn3)C(F)(F)F SEW06209 CSc1nc(nc(n1)N)C2COc3ccccc3O2 KM09753 c1ccc(cc1)OS(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F KM09807 CN(C)S(=O)(=O)c1ccc(s1)c2cc(on2)C(F)(F)F KM09820 c1ccc(cc1)C(=O)N/N=C/C(=O)O RJC03266 CCOC(=O)c1c2nc(c3ccccc3n2nn1)Sc4nnc(o4)c5ccncc5 HTS12457 c1ccc2c(c1)CCCN2CC(=O)N3CCc4c3cccc4 HTS12460 c1ccc2c(c1)CCCN2CC(=O)N3CCCc4c3cccc4 HTS12505 c1cc2c3c(c1)c4c(c(cc(=O)o4)OC(=O)c5cccs5)c(=O)n3CC2 HTS12694 c1ccc(cc1)NC(=O)NC(=O)CSc2ncc(c(n2)N)C#N HTS12719 CC(c1ccccc1)NC(=O)c2ccccc2 JFD03426 c1ccc(cc1)CC(=O)Nc2ccc3ccccc3c2 JFD03487 Cn1c2c(c(=O)n(c1=O)C)n(cn2)CC(CN3CCCC3)O JFD03562 c1ccc2c(c1)CC(=C2)N3CCN(CC3)c4cccc(c4)Cl JFD03621 Cc1ccc(cc1)NC(=O)c2ccccc2 JFD03709 c1ccc(c(c1)C(=O)NNC(=O)CC#N)Cl RH00327 CCOC(=O)CSc1nc2cccnc2s1 RH00352 c1cc2c(ccnc2cc1Cl)N3CCCCC3 RH00412 Cc1c2c3ccccc3ccc2oc1C(=O)c4ccccc4 RH02204 CCc1ccc(cc1)C(=O)Nc2ccc3c(c2)ccc(n3)C RH02218 COc1cccc(c1C2=Nc3ccccc3SC(C2)c4ccccc4)O RJC00351 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N)CCCC(=O)O RJC03315 c1ccc(cc1)Cc2c(nc(sc2=O)c3ccccc3)O RJC03347 c1ccc(cc1)CNc2ccc(nn2)c3ccccc3 RJC03365 C/C(=N\c1ccccc1)/c2cccs2 RJC03366 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)F)C2=O S12973 c1ccc2c(c1)C(=O)C(=Cc3c(cccc3Cl)F)C2=O S12976 CCNC(=O)/C(=C/c1cccc(c1OC)OC)/C#N S05388 Cc1ccc(cc1)C2N(C(CS2)C(=O)O)C(=O)C S05423 c1cc(ccc1NCN2C(=O)c3ccc(cc3C2=O)[N+](=O)[O-])F S05534 c1ccc2c(c1)C3(C(=O)N2)OCCCO3 S13980 CN(C)/C=C/C(=O)c1ccccn1 SEW04035 c1ccc2c(c1)NC(=O)CC(S2)c3ccco3 SEW04041 Cc1c(oc(n1)C)c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl SEW01591 c1cc(c(cc1C(F)(F)F)Cl)/C=N/N2CCOCC2 SEW01609 c1cc(ccc1CC#N)c2nnco2 SEW01635 COCCCNC(=S)N/N=C/c1ccc[nH]1 SEW04552 c1ccc2c(c1)c3c([nH]2)C(N(CC3)C(=S)Nc4ccccc4OC(F)(F)F)C(F)(F)F SEW06217 Cc1cn(nc1c2cccs2)C(=O)c3c(nns3)C SP01256 c1ccnc(c1)SCc2nc(on2)COc3ccc(cc3Cl)Cl SP01265 c1cc(ncc1[N+](=O)[O-])Oc2cc(cc(c2)C(F)(F)F)C(F)(F)F SEW06415 CC(C)Cc1ccc(cc1)C(C)C(=O)NC(=O)Nc2ccc(cc2)OC SEW06427 CC[n+]1c(sc2c1cccc2)C.[I-] RJC03274 CC1=C(C(=O)C(=C(C1=O)C)C)C RJC03282 Cc1cccc(c1NC(=S)N2CCCC2=O)C RJF01800 c1ccc(c(c1)c2nnn(n2)CC(=O)NNC(=O)C3CC3)C(F)(F)F RJF01860 CCOC(=O)C1=C(NC(=C(C1c2ccc3c(c2)OCO3)C(=O)OCC)C)C RJC03409 Cc1cc(nc(c1C#N)Sc2ncc(c(n2)N)C#N)C HTS12720 c1ccc(cc1)n2c(=O)c3c4c(sc3[nH]c2=S)CCC4C(=O)O HTS12743 c1ccc(c(c1)CSc2nnc3n2CCCN3C(=O)c4ccc(cc4)F)Cl HTS12773 C/C(=N\Cc1ccc(cc1)OC)/C2CCOC2=O NRB03566 c1cc(sc1)c2cc(c(c(c2C#N)N)C#N)c3cccs3 JFD03794 Cc1ccc(cc1C)NC(=S)NCc2ccccn2 JFD03872 COc1cc(cc(c1OC)OC)C(=O)Oc2c(cc(cc2Cl)Cl)/C=N/c3cccc(c3)C(F)(F)F JFD03887 c1cc(oc1)CNc2ccc(cc2C(=O)O)[N+](=O)[O-] RDR02080 Cc1cc(ccc1NC(=O)c2ccc(cc2[N+](=O)[O-])Cl)Cl RDR02193 Cc1ccc(c(c1)OC(C)CC(=O)O)[N+](=O)[O-] RJC00386 CCCCCCCOc1ccc(nn1)S RJC00502 c1ccc(c(c1)NC(=S)Nc2cc(n[nH]2)c3cccs3)Cl KM09853 c1cc2c(cc(nc2c(c1)Cl)C(F)(F)F)N3CCCC3 KM09870 c1cc2c(ccc(c2nc1)NCCCO)[N+](=O)[O-] RJC03509 CC(CNc1ccc(c2c1nccc2)[N+](=O)[O-])O RJC03510 CC(C12CC3CC(C1)CC(C3)C2)Nc4ccc(c5c4nccc5)[N+](=O)[O-] RJC03518 c1cc(c(c(c1)C(F)(F)F)C(=O)N)C(F)(F)F RJC03569 c1cc(ccc1C(F)(F)F)NC(=S)Nc2ccc(cc2)S(=O)(=O)Nc3cc(ccc3F)F RJF02106 CCOC(=O)C(CSC1CC(=O)N(C1=O)c2ccc(cc2)OC(F)(F)F)N.Cl S13991 c1ccc(cc1)c2c(nn3c(n2)nnc3S)c4ccccc4 NRB04127 COc1ccc(cc1)Cc2c(=O)nc([nH]n2)SC NRB04131 c1ccc(cc1)C(=O)/C=C/Sc2ccccn2 NRB04153 c1ccc(cc1)C(=O)Nc2ccc3c(c2)C(=O)c4ccccc4C3=O NRB04166 c1c(ccc(c1)F)/C=C\2/C(=O)/C(=C/c3ccc(cc3)F)/COC2 SEW04554 c1cc(n(c1)S(=O)(=O)c2ccc(cc2F)F)C=C(C#N)C#N SEW04565 Cc1cccc(c1NC(=O)CCN2CCCCC2)C RDR02556 CN(C)CC(=O)Nc1nc(cs1)c2ccc(cc2)Cl RDR02625 c1c(cc(cc1C(F)(F)F)NC(=S)SCCSC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F RDR02630 c1c(cc(cc1C(F)(F)F)NC(=O)CN2CCCCC2)C(F)(F)F RDR02660 CC(=O)OC[C@@H]1[C@]2(CO[C@H]([C@@H]([C@H]2OC(=O)C)OC(=O)C)OC3[C@@H](CO1)O[C@H]([C@@H]([C@H]3OC(=O)C)OC(=O)C)OC)OC(=O)C RJC00890 COC(=O)Nc1[nH]c2ccc(cc2n1)c3c4ccccc4c(=O)[nH]n3 RJC00902 c1ccc(cc1)CCN2C(=O)CN(CC2=O)C(=O)C3CCCCC3 RJC00904 COc1ccccc1C2CCN(CC2)C(=O)CSc3nnc(s3)N RH01265 c1cc(cc(c1)N2CCCC2=O)C(F)(F)F RH01282 CC1=C(C(C(=C(N1)C)C#N)c2ccc(cc2Cl)O)C#N RJC03424 Cc1cccc(n1)C2C(=C(NC(=C2C(=O)OC)C)C)C(=O)OC RJC03437 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CC(=O)NNC(=S)Nc3ccc(c(c3)Cl)Cl RJF02020 Cn1c(nnc1SCC(=O)c2ccc(cc2)Cl)c3ccc4c(c3)cccn4 KM10640 CCCC(=O)c1ccc(c(c1)OC)OC NRB03602 CC(=O)OC1CCC2(C3C(CC[C@]2(C1)C)C4CC=C(C4(CC3OC(=O)C)C)OC(=O)C)C NRB03671 c1cc(c(c(c1)Cl)S/C=C/C(=O)c2ccc(cc2)I)Cl NRB03910 c1ccc2c(c1)[nH]c(n2)NCCO NRB03945 c1ccc(cc1)CCNC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02199 Cc1ccc(c(c1)C)NC(=O)C(C)Oc2ccc(cc2Cl)Cl RDR02206 C=CCOc1ccc(cc1Br)C(=O)OCC(=O)c2ccccc2 RDR02261 Cc1ccc(cc1)Cc2c(nc(nc2O)N3CCCC3)C RDR02417 c1ccc(cc1)S(=O)(=O)/C(=C/c2cccn2c3ccc(cc3)OC(F)(F)F)/C#N SEW06338 c1cc(c(c(c1)F)C(=O)NCCSCc2ccc(cc2)Cl)F SEW06360 c1ccc(cc1)C(=O)/C=C(\O)/C(=C/C(=O)c2ccccc2)/O RJC00790 C1C2C3C4C1C5C2C(=O)C3C4C5(F)F RJC00821 Cc1ccc(cc1)S(=O)(=O)CC(=O)c2ccccc2 RJC00863 c1cc(cc(c1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F)COc4ccc(cc4)Cl SEW06482 CCOC(=O)Cn1nc(nn1)c2cccc(c2)C(F)(F)F RJF02109 CC1(OC2[C@H](O[C@H](C2O1)n3cnc4c3ncnc4N)CO)C KM10862 CCCCNC(=O)c1cc2cc(ccc2[nH]1)CC KM11007 c1ccc(cc1)Nc2ccnc3c2ccc(c3)Cl KM11055 Cc1ccc(cc1Cl)c2ccc(c(c2)Cl)C MB00043 COc1cc2c(c(c1OC)OC)Cc3cc(c(c(c3C2)OC)OC)OC MB00114 CCc1c(c([nH]c1C(=O)OCC)C)C(=O)OCC NRB04228 CC(=O)O[C@H]1[C@H]2[C@@H](CO[C@H](O2)c3ccccc3)O[C@H]([C@@H]1OC(=O)C)OC(=O)C NRB04421 c1ccc(c(c1)C2N[C@@H](CS2)C(=O)O)C(=O)O NRB04468 COc1cc(cc(c1OC)OC)/C=N/N=C(N)N NRB04485 Cc1ccc(cc1)S(=O)(=O)Nc2c(cc(cc2C)I)C RDR02687 COc1cc(cc(c1OC)OC)/C=N/OC(=O)c2ccc(c(c2)Cl)Cl RDR02690 CC1CN(CC(O1)C)C(=O)COc2ccccc2OC(=O)N(C)C RDR03038 c1cc(cc(c1)[N+](=O)[O-])C(C(Cl)(Cl)Cl)O RDR03158 c1cc(c(cc1[N+](=O)[O-])CO)N2CCCCC2 RH01305 COC(=O)/C(=C/c1ccc(c(c1)[N+](=O)[O-])N2CCCCC2)/C#N RH01316 Cc1ccc(cc1)c2nnn(n2)CC(=O)O RH01367 c1cc(sc1c2cnc3c(n2)cc(cc3Cl)C(F)(F)F)Br RH01383 CC(CN1c2ccccc2Sc3c1cccc3)NC RH01503 Cc1ccc(cc1)C(=O)NNC(=O)CSCc2cccc3c2cccc3 RH01531 C=CCn1c(nnc1SCC(=O)c2ccc(cc2)Cl)c3ccc4c(c3)cccn4 KM10641 C=CCn1c(nnc1SCc2ccc(cc2)OC(F)(F)F)c3ccc4c(c3)cccn4 KM10673 Cn1c(nnc1SCc2ccccc2)CNC(=O)c3ccc(cc3)OC(F)(F)F KM10709 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3ccc(cc3)OC KM10762 CC(C)(C)c1ccc(s1)C(=O)NC(=O)Nc2ccccc2 MBE00188 c1ccc2c(c1)ccnc2C(=O)c3cccc(c3)C(F)(F)F NRB04079 CCOC(=O)NN(/C(=C\C=C\N1CCCC1)/c2nnn(n2)c3ccc(cc3)Cl)C(=O)OCC NRB04098 Cc1ccc(cc1)/C(=C/c2ccc(cc2)N(C)C)/C#N PHG00056 c1ccc(cc1)NC(=S)Nc2cccc(c2)C(F)(F)F JFD00422 c1ccc2c(c1)C3=C(C2=O)C(NC(=S)N3)c4ccc(cc4)[N+](=O)[O-] JFD00449 c1ccc2c(c1)c(c([nH]2)c3ccc(cc3)Cl)/C=N/NC(=S)Nc4cc(cc(c4)C(F)(F)F)C(F)(F)F RDR02525 c1ccc(cc1)CNC(=O)C(=O)Nc2cccc(c2)C(F)(F)F JPV00092 Cc1cccc(c1C)/N=C/c2cc(ccc2O)Br K00010 C/C(=C\c1ccc(c(c1)OC)OC)/[N+](=O)[O-] K00031 c1cc(cc(c1)[N+](=O)[O-])c2nnc(o2)/C=C/c3ccc(cc3)OC(F)(F)F SEW06491 CC(C)Cc1ccc(cc1)C(C)c2nc(no2)c3cccs3 SEW06492 CC(=NNc1ccc(cc1[N+](=O)[O-])[N+](=O)[O-])C RJC00976 c1ccc(cc1)/C=N/Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] RJC00977 c1ccc2c(c1)N/C(=C/C(=O)c3ccc(cc3)[N+](=O)[O-])/C(=O)O2 RJC00979 CC(C)(C)c1ccc(cc1)NC(=O)CSc2[nH]c(=O)c(c(n2)C3CCCCC3)C#N RH01392 c1ccc(cc1)NC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl SPB02952 Cc1c(sc(n1)C)C(=O)NNC(=O)c2ccc(cc2)Cl SPB02977 c1cc(ccc1c2nc(cs2)c3ccc(cc3)Cl)Oc4ccc(cn4)C(F)(F)F SPB03016 CCn1c(cc(n1)C)C(=O)Sc2cccc(c2)Br SPB03081 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)NNC(=O)Nc3ccccc3 SPB03118 CC1CN(CC(O1)C)c2ccccc2[N+](=O)[O-] S06454 c1ccc(cc1)N2C(SCC2=O)c3cccnc3 S06688 CC1(COC(=N1)c2ccc(cc2)C(C)(C)C)C.Cl S06921 c1cc(ccc1C(C[N+](=O)[O-])Sc2ccc(cc2)N)Cl S14251 CC1(OC(=O)C(=Cc2cc(ccc2OC)OC)C(=O)O1)C S14256 c1cc(ncc1C(F)(F)F)SCCS(=O)(=O)CCSc2ccc(cn2)C(F)(F)F SEW01881 c1ccc(cc1)c2csc(n2)c3ccc(cc3Cl)C(F)(F)F SEW01919 c1cc(c(cc1C(F)(F)F)Cl)c2nc(cs2)C(=O)O SEW01963 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=O)c2cccn2c3ccc(cc3)F SEW04777 c1cc(cc(c1)NC(=S)NNC(=O)c2cccn2c3ccc(cc3)F)C(F)(F)F SEW04784 c1ccc(cc1)CN2CCN(CC2)c3ccccc3/C=C(/C#N)\S(=O)(=O)c4ccccc4 SEW06545 CC(C)(C)c1cc(n(n1)C)C(C)(C)C SEW06558 c1cc(cc(c1)C(F)(F)F)CSCCNC(=O)c2ccc(c(c2)Cl)Cl SEW06564 COc1cccc(c1OC)/C=N/C2CCN(CC2)Cc3ccccc3 SEW06622 C1COCCN1/C(=N\O)/c2c(non2)N RJC01129 c1ccc2c(c1)-c3ccccc3NC(=O)N2 RJC01303 Cc1c2c(nc(nc2sc1C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F)c4ccccc4OC)C SPB05512 Cn1c2c(cc3ccc(cc3n2)C#C)c(=O)n(c1=O)C RJC03665 CN1c2ccccc2C(=O)/C(=C/Nc3ccccc3)/C1=O RJC03675 c1ccc(c(c1)C(F)(F)F)NS(=O)(=O)c2ccc(cc2)NC(=S)NC(=O)/C=C/c3cccs3 RJF02183 c1ccc\2c(c1)CC/C2=N\N=C(N)N NRB04548 COc1ccc(cc1OCc2ccccc2)CO NRB04550 CSC(=N)Nc1ccc(cc1)Cl.I NRB04583 c1ccc(cc1)N=c2[nH]c(nc(=O)n2c3ccccc3)N NRB04590 c1ccc2c(c1)C(=O)N(C2=O)CNc3cccc(c3)Cl RB00029 c1cc2c(cc1C(=O)CCN3CCCCC3)OCCCO2.Cl NRB05081 c1cc(ccc1NC(=O)COc2ccc(cc2)OC(F)(F)F)OC(F)(F)F RDR03487 c1cc(ccc1C(=C2SCCS2)C#N)Cl RDR03511 c1c(cc(cc1Cl)Cl)N2C(=O)CC3(C2=O)CCCC3 RDR03516 c1ccc(cc1)c2nc(sn2)Sc3ccc(cc3)Cl RDR03895 CS(=O)(=O)Cc1nnc(o1)c2cccc(c2)[N+](=O)[O-] SEW06660 Cc1cc([nH]c1c2cc[nH]n2)C SEW06694 Cc1ccc(cc1)S(=O)(=O)Oc2c(cc(cc2Cl)Cl)/C=N\c3cccc(c3)C(F)(F)F SJC00183 COc1cc(cc(c1OC)OC)C(=O)Oc2c(cc(cc2Cl)Cl)/C=N\c3ccc(cc3C#N)[N+](=O)[O-] SJC00213 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CCC4)O RJC01488 Cc1ccc(cc1)S(=O)(=O)NC(C)c2ccccc2 RJC03740 C1CCc2c(c3c(c4c2CCCC4)CCCC3)C1 RJC03788 CC(C)(C)c1ccc(cc1)C(=O)/C=C/C(=O)O RJC03868 CCCCN(CCCC)CCCn1cnc2c(c1=O)cccn2 RJC03954 Cc1c2c(c3ccccc3n(c2=O)C)n(n1)c4ccccc4 RJC03984 CCN(CC)c1ccc(cc1)/C=N/C(c2ccccc2)c3ccccc3 S00628 c1cc(cnc1)C2N(C(=O)CS2)Cc3cccs3 S07622 c1cc(sc1)CNC(=O)/C=C\C(=O)O S07623 c1cc(sc1)CN2C(=O)C=CC2=O S07624 CC(C)(C)c1ccc(cc1)NC(=S)Nc2ccc(cc2)S(=O)(=O)N3CCCCC3 S07956 c1ccc2c(c1)CCC/C(=C\c3ccc(cc3)Br)/C2=O S14665 c1cc2c(cc1Cl)C(=C(CS2)CN3CCCCC3)Cl SEW02217 c1cc(sc1)c2ccc(s2)c3ccn[nH]3 SEW02222 c1ccc(c(c1)CN/C=N/O)OC(F)(F)F SEW02237 c1cc(cc(c1)NC(=O)CS(=O)(=O)Nc2cccc(c2)C(F)(F)F)C(F)(F)F SEW02240 c1cc(ccc1C(F)(F)F)NC(=O)CC23CC4CC(C2)CC(C4)C3 SEW05134 c1cc(oc1)CNC(=S)N/N=C/c2cc(cc(c2O)Cl)Cl SJC00364 CC(C)(C)NC(=S)N/N=C/c1ccccc1O SJC00393 CCOC(=O)c1cc([nH]c1C)C SP00003 Cc1c(cc(o1)c2ccc(cc2)Cl)c3cc[nH]n3 SP00114 Cc1c2cnn(c(=O)c2c([nH]1)C)Cc3ccccc3Cl SP00126 c1cc(sc1)/C=C/C(=O)NC(=S)Nc2nc(cs2)c3ccc(cc3)Cl RJF02215 CC12CCCCC13NC(=O)CN3c4c2cccc4 RJC04045 COc1cccc(c1[N+](=O)[O-])/C=C/N2CCCC2 RJC04052 c1cc(c(cc1F)F)NC(=S)NN RJF00037 c1cc(c(cc1F)F)NC(=N)NC(=N)N.Cl RJF00041 Cc1cc(nc(n1)NC(=N)Nc2ccc(cc2F)F)O RJF00043 CC(=O)c1c(c2cccc3c2n(c1=O)c4c3cccc4)O NRB05103 Cc1ccc(cc1)C(=O)/C=C\Nc2ccc(cc2)OC(F)(F)F NRB05120 CCOc1ccc(cc1)C2N[C@@H](CS2)C(=O)O NRB05178 Cc1cc(c(cc1C)N/C(=N/CCCOC)/SC)C RDR00211 c1ccnc(c1)N2C(=O)CSCC2=O PD00053 c1cc(cnc1)NC(=O)CSCC(=O)O PD00054 Cc1cc(cc(c1N2C(=O)CC(C2=O)Sc3ccc(cc3)Cl)C)C(C)(C)C RDR03913 c1ccc(cc1)c2cc(n[nH]c2=O)c3ccc(cc3)F RDR04000 c1cc(nc(c1)n2c(=O)oc(n2)c3ccc(c(c3)Cl)Cl)C(F)(F)F RF05185 COc1ccc(c(c1)C(=O)Nc2cccc(c2Cl)Cl)Br RF00411 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)N)c3ccccc3 SP00373 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)NCCCN4CCOCC4 SP00380 CC(C)(C)c1ccc(cc1)c2nc(cs2)c3ccc(cc3)OC(F)F SP00388 CCC1C2=C(CCCC2=O)NC3=C1C(=O)CCC3 RJC01796 CC(=O)OCc1ccccc1Sc2ccc(cc2C(=O)O)[N+](=O)[O-] RJC01857 Cc1c(c(nc(n1)N2CCOCC2)O)Cc3c(cccc3Cl)F RJF00110 CNC(=S)Nc1ccc(cc1F)F RJF00130 c1cc(c(cc1NC(=S)NCCCN2CCOCC2)Cl)F RJF00176 COc1ccc(cc1OC)CCN2CN(C(=S)SC2)CCc3ccc(c(c3)OC)OC S01961 Cc1ccc(cc1N2C(=O)CC(C2=O)Sc3ccccc3N)Cl S02034 c1cc(cc(c1)NC(=O)/C=C/C(=O)O)C#N S09410 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3cccc(c3)C#N S09412 c1ccc(c(c1)NC(=O)CCC(=O)O)Oc2ccc(cc2Cl)Cl S09530 CC(C)(C)c1ccc(cc1)/C=C/2\CCc3cc(ccc3C2=O)OC S15135 COc1ccc2c(c1)CC/C(=C\c3cccc(c3)Br)/C2=O S15330 Cc1c(c(n(n1)C)O)/N=N/c2ccccc2OC(F)(F)F SEW02654 CC(=O)c1ccc(cc1OC(=O)c2ccc(cc2)Cl)OC(=O)c3ccc(cc3)Cl SEW02724 c1cc(c(cc1F)F)OCCC(=O)O SEW05376 Cc1ccc(cc1)c2csc(n2)c3ccc(cc3)Cl SEW05396 CCOC(=O)C(=CNc1ccc(cc1Cl)C(F)(F)F)C(=O)OCC SEW05405 c1cc(ccc1c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F)[N+](=O)[O-] SP00430 c1cc(ccc1c2csc(n2)c3ccc(cc3)Oc4ccc(cn4)C(F)(F)F)C(F)(F)F SP00446 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)c3ccc(cc3)C(F)(F)F SP00498 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1)C)NC(=O)Nc2ccccc2 RJC01997 CC1CN=C(S1)Nc2ccccc2F RJC02012 Cc1cc(c(cc1C)CSC(=N)N)CSC(=N)N S01533 c1cc(ccc1c2csc(n2)NC(=O)CN3CCSCC3)Cl RJF00197 c1cc(ccc1C(=O)Cn2nc(nn2)N3CCOCC3)Cl RJF00230 Cc1c(nc(nc1O)SCc2c(cccc2Cl)F)C RJF00269 CC(=O)Nc1nc(nc(n1)N2CCCCC2)NC(=O)C RJF00293 COC(=O)/C=C\1/C(=O)N=C(S1)c2ccccc2 PD00086 c1cc(ccc1NC(=O)c2cc(ccc2O)Br)F RDR00835 CC(C)NC(=S)N/N=C/c1cccnc1 RDR00899 CC(C)NC(=S)N/N=C/c1ccco1 RDR00908 c1ccnc(c1)/C(=C/c2cccnc2)/C#N PD00233 c1ccnc(c1)/C(=C/c2ccncc2)/C#N PD00234 Cc1cc(nc(c1C#N)Sc2c(c(c(c(n2)C)[N+](=O)[O-])C)C#N)C RF00430 Cc1cccc(c1NC(=O)Cc2ccc(cc2)[N+](=O)[O-])C RF00485 c1ccc2c(c1)c(=O)[nH]c3n2ncc3C#N RH00043 c1(c([nH]c(=O)[nH]c1=O)C(=O)O)[N+](=O)[O-] RH00056 c1ccc2c(c1)C(c3ccccc3O2)c4nnc(o4)S RH00058 c1cc(ccc1c2csnn2)c3nc(cs3)c4ccc(cc4)C(F)(F)F SP00520 c1cc(ccc1c2nc(cs2)c3ccc(cc3)C(F)(F)F)C4SCCS4 SP00534 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)C(C)(C)C)C(=O)O SP00572 c1ccc(c(c1)OCc2nc(cs2)c3ccc(c(c3)F)F)Cl SP00582 c1ccc2c(c1)cccc2C#CC(=O)O RJC02245 COc1ccc(cc1OC)CCNC(=S)NC2CC2 RJF00367 c1cc(sc1)CNC(=S)NC2CC2 RJF00369 Cc1c(c(nc(n1)c2ccc(c(c2)Cl)F)O)CC=C RJF00472 c1cc(cc(c1)Cl)NC(=S)Nc2cccc(c2)Cl S03280 COc1cc(cc(c1OC)OC)NC(=O)/C=C/C(=O)O S03340 c1c(cc(cc1C(F)(F)F)NC(=O)COCC(=O)O)C(F)(F)F S10461 c1cc(c(cc1C(F)(F)F)NC(=O)CSCC(=O)O)Cl S10511 c1cc(ccc1N2C(=O)CSCC2=O)Br S10516 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3cccs3 SCR01459 CC/C(=N\NC(=O)OCC)/c1ccccc1 SEW03357 CCOC(=O)c1c(nc(s1)c2cnccn2)C SEW03455 COc1ccc(cc1)/C=N/NC(=O)c2ccc[nH]2 SEW05631 c1cc([nH]c1)C(=O)NNC(=S)Nc2ccc(cc2)F SEW05633 CC(=O)C(=CNCC(=O)OC)C(=O)C SEW05636 c1cc(ccc1c2csc(n2)c3c(cc(cc3Cl)C(F)(F)F)Cl)OC(F)F SP00708 Cc1c(c(on1)C)c2nc(no2)c3ccccn3 SP00714 CC(C)(C)c1cc(n(n1)Cc2ccccc2)c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F SP00747 COc1ccc(cc1OC)/C=C/c2nc3ccccc3s2 RJC02415 CCOC(=O)CNC(=O)CSc1nnc(s1)C RJC02433 c1c(cc(c(c1Cl)NC(=S)N)Cl)Cl S02726 COc1cc(cc(c1OC)OC)c2c(c(nc(c2C#N)OC)N)C#N S02760 c1cc(ccc1NC(=S)NNC(=O)C2CC2)Cl RJF00606 Cc1cc(nc(n1)c2ccccc2)O RJF00618 c1cc(ccc1Nc2ncnc(n2)N)I RJF00659 Cc1cc(ccc1/N=C\2/N(C(=O)CS2)CCc3ccc(c(c3)OC)OC)Cl S03639 c1cc(ccc1CNC(=S)Nc2ccc(c(c2)Cl)Cl)C#N S03792 Cc1ccc(cc1)N2C(=O)C=C(C2=O)Sc3ccc(cc3)C(C)(C)C PD00238 c1ccc(cc1)COc2cccc(c2)/C=C(\C#N)/c3ccccn3 PD00305 Cc1ccc(cc1C)NC(=O)CCC(=O)O RDR01078 c1cc(ccc1c2csc(n2)N)[N+](=O)[O-] RDR01084 c1c(cc(c(c1Br)O)Br)/C=N/NC(=S)NCC2CCCO2 RDR01120 c1cc(c(cc1F)Br)NC(=S)NCCCCCCO PD00432 Cc1cc(nc(n1)c2cccnc2)O RF01002 c1cc(sc1)c2cc(c(c(n2)N3CCCCC3)C#N)C(F)(F)F RF01024 CCOC(=O)C(=CNc1ccc(c(c1)C#N)F)C(=O)OCC RH00251 CCOC(=O)c1cnn(c1n2cccc2)c3ccc(cc3)[N+](=O)[O-] RH00290 c1cc(sc1)CNC(=S)NNC(=O)CC#N RH00311 Cc1c(cc(n1CCCN2CCOCC2)c3ccccc3)C(=O)NCc4ccco4 SP00774 COc1ccc(c(c1)c2nc(no2)c3ccc(cc3)OC(F)(F)F)Br SP00821 CC(=O)c1ccc(cc1)NC(=O)CSc2ccc(cc2)Cl RJC02511 CCOC(=O)Cc1csc(n1)NC(=O)CSc2[nH]c(=O)c3ccccc3n2 RJC02517 CCCc1cc(nc(n1)SCC(=O)Nc2ccc(cc2)C(=O)OCC)O RJC02528 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(cc(c2)Cl)Cl RJF00745 CC(C)(C)c1ccc(cc1)NC(=S)NCCC(=O)O RJF00756 c1cc(c(cc1F)F)N2C(=O)C=CC2=O S03891 CSc1cccc(c1)N2C(=O)C3CC=CCC3C2=O S03928 c1ccc2cc(ccc2c1)C3=Nc4ccccc4SC(C3)c5ccsc5 S11130 c1cc(ccc1/C=C/[N+](=O)[O-])F S11468 CCOC(=O)/C(=C/c1ccc(cc1)F)/C#N S11470 c1ccc(cc1)NC(=O)NNC(=N)c2ccccn2 SEW00368 CCOC(=O)CSCc1nc(on1)COc2ccc(cc2Cl)Cl SEW00396 Cc1cc(c(n1c2ccc(cc2)C(F)(F)F)C)C=C(C#N)C#N SEW03582 c1c(csc1[N+](=O)[O-])C(=S)N SEW03585 CSc1ccc(s1)CNC(=O)c2ccc(cc2)Cl SEW03647 c1ccc(cc1)CC(C(F)(F)F)OC(=O)c2ccc(cc2Cl)Cl SEW03679 CC(C)(C)c1ccc(s1)C(=O)Nc2ccc(cc2)OC SEW05830 Cc1c(c(on1)C)S(=O)(=O)N2CCCCC2 SEW05837 Cc1c(c(on1)C)C(=O)Oc2ccccc2 SEW05848 Cc1ccc(cc1)NC(=O)c2cc(n(c2C)CCSC)c3ccccc3 SP00909 Cc1c(cc(n1CCSCc2c(cccc2Cl)F)c3ccccc3)C(=O)N4CCCC4 SP00932 Cc1ccccc1NC(=O)c2cc(n(c2C)CCSCc3c(cccc3Cl)F)c4ccccc4 SP00938 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)OCc2ccc(cc2)OC RJC02640 Cc1ccccc1N(C2=NCC(S2)C)C(=O)Nc3cccc(c3)Cl RJC02642 Cc1ccc(cc1)Sc2c(=O)c(=O)c2Sc3ccc(cc3)C MWP00918 c1cc(ccc1NS(=O)(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F)[N+](=O)[O-] MWP00978 CCCS(=O)(=O)c1ccc(cc1)NC(=O)Nc2ccc(cc2Cl)Cl MWP01002 CC(C(=O)NNC(=O)C(C)(C)C)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01867 c1ccc2c(c1)c(cs2)CNC(=O)Nc3ccc(c(c3)Cl)Cl PD00439 CN(C)NC(=S)NCc1ccc(cc1)F PD00442 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2csc3c2cccc3 PD00446 c1ccc(cc1)C(=O)COC(=O)c2ccccc2C(=O)c3ccccc3 RDR01502 c1ccc(cc1)c2c(=O)oc(nn2)c3ccc(cc3)Cl S13858 CC(=N/N=C\1/N=C(CS1)c2ccc(cc2)Cl)C RF01459 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2c(cccc2Cl)F RF01595 CC(=O)Nc1ccc(cc1NC(=O)C(Cl)(Cl)Cl)C(C)(C)C RF01651 c1c(c(=O)c(cn1CC(=O)NN)Cl)Cl RF01797 CC(=O)Nc1cccc(c1)C#C RF01853 Cc1c(cc(o1)C(C)(C)C)c2cc(n(n2)c3ccc(cc3)I)N SP00994 c1cc(ccc1c2cc(n(n2)c3ccc(cc3)I)NC(=O)C4CCC4)Cl SP01009 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)N3CCC(CC3)(c4ccc(cc4)Cl)O SP01050 CN(C)/C=N/n1cnc2c(c1=O)c3c(s2)CCCC3 RJC02769 Cc1ccc(cc1Cl)c2nc(cc(n2)OC(=O)N(C)C)COC RJF01078 c1ccc(c(c1)c2nnn(n2)CC(=O)NN)C(F)(F)F RJF01084 Cc1ccc(cc1Cl)c2n[nH]nn2 RJF01102 c1cc(cnc1)/C=N/N2C(=O)CSC2=S S04279 CCOc1ccc(cc1OC)/C=C(\C)/[N+](=O)[O-] S04283 Cn1c(c(c(=O)n(c1=O)C)C(C[N+](=O)[O-])c2ccc(cc2)OC)N S12158 c1ccc(cc1)CN2C(=O)CC(=O)NC2=O S12193 COc1ccc(cc1C2Nc3ccccc3C(=O)N2)Br S12246 CC(=O)C1CNc2ccc(cc2C1(c3ccccc3)O)Cl S12252 Cc1cccc(c1N2C(=O)CC(C2=O)N3CCSCC3)C S12381 c1ccc\2c(c1)CCC/C2=N/Nc3c(cc(cc3Cl)C(F)(F)F)Cl SEW03808 COc1ccc(cc1/C=N/Nc2c(cc(cc2Cl)C(F)(F)F)Cl)Br SEW03809 c1cc(sc1)/C=N/Nc2c(cc(cc2Cl)C(F)(F)F)Cl SEW03810 c1cc(sc1)CC2=NC(=O)CS2 SEW03845 COC(=O)c1c(ccs1)c2ccc(o2)/C=C/[N+](=O)[O-] SEW03887 c1cc(ccc1SCc2csc(n2)N3CCOCC3)Cl SEW03894 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)Nc3ccc(cc3)[N+](=O)[O-] SP01061 CCOC(=O)c1c(n(c(c1S(=O)(=O)NCc2ccccc2)c3ccccc3)c4ccccc4)C SP01127 CCOC(=O)c1c(oc(c1S(=O)(=O)N)C)C SP01166 Cc1c(cc(o1)c2ccccc2)C(=O)N3CCN(CC3)c4c(cccn4)C(F)(F)F SP01178 CC(C(=O)NNS(=O)(=O)C)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01873 CN(C)c1ccc(cc1)n2c(nnn2)S S05029 c1cc(cc(c1)[N+](=O)[O-])C(=O)Nc2cccc(c2)F S05044 c1ccc(cc1)C(=O)NC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F S05112 c1cc(ccc1n2c(=S)[nH]nn2)F S05119 c1ccc(cc1)/C=C/C(=O)NC(=S)NNC(=O)Cn2nc(nn2)N3CCOCC3 RJF02076 CCOC(=O)N1c2ccc(cc2C=CC1C#N)C(C)C S13862 c1ccc(cc1)C#CC(=O)Nc2ccc(cc2)OC(F)(F)F S13953 COC(=O)CSc1nc2ccc(cc2s1)Cl SEW01270 Cc1csc(n1)Cc2ccc(cc2)c3csnn3 SEW01318 c1cc(cc(c1)/N=C/c2ccc(cc2)[N+](=O)[O-])c3nnco3 SEW01362 CN1C(CC(=N1)c2ccc3ccccc3c2)c4ccc(cc4)C(F)(F)F S14219 CN(C)c1cc(cnc1C#N)C(F)(F)F SEW03922 CN(C)c1cc(cnc1C(=S)N)C(F)(F)F SEW03924 c1c(cc(cc1Cl)Cl)C(=O)OCCSCc2cc(cc3c2OCOC3)[N+](=O)[O-] SEW03966 c1cc(ccc1NC(=O)N2CCN(CC2)c3cc(ccn3)C(F)(F)F)Cl SEW03971 CN(c1cc(ccn1)C(F)(F)F)NC(=O)/C=C/C(=O)O SEW03974 c1cc(cc(c1)F)C2NC(CS2)C(=O)O RJC02834 Cc1c(cc(o1)c2ccccc2)C(=O)Nc3ccccc3 SP01181 Cc1c(cc(o1)c2ccccc2)C(=O)Nc3cccc(c3)[N+](=O)[O-] SP01183 Cc1c(cc(o1)c2ccccc2)C(=O)Nc3ccc(cc3)OC(F)(F)F SP01187 COc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccc(cc3Br)F SP01202 CCC(C)c1ccccc1NC(=O)c2cc3cc(ccc3[nH]2)OC SP01228 CCCc1c(c(nc(n1)S)O)CC=C RJF01574 CCCc1c2ccc(cc2oc(=O)c1Cc3c(cccc3Cl)F)OC(=O)N(C)C RJF01600 c1ccc(c(c1)c2nc(nc(n2)N)N)Cl RJF01628 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2ccccc2Oc3ccc(cc3Cl)Cl RJF01707 c1cc(oc1)C(=O)N(c2ccc(cc2F)F)C3=NCCCC(=O)S3 RJF01775 c1cc(c(cc1NC2=NCCC(=O)S2)Cl)F RJF01785 c1cc(c(cc1Cc2c(nc(nc2O)S)C(F)(F)F)Cl)Cl RJF02078 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2cc(ccc2F)F RJF02099 c1ccc(cc1)NN2C(=O)c3ccccc3C2=O S05558 Cn1c(=O)c2ccccc2c(n1)O S05568 CC(C)(C)NC(=S)NC1CCCCC1 S05699 CSc1cccc(c1)NC(=O)CSc2ccc(cn2)C(F)(F)F NRB00163 CN1C(CC(=N1)c2ccc3ccccc3c2)c4ccc(cc4)OC S14224 Cc1ccc(cc1)n2c(=O)c3cc(ccc3nc2SCC(=O)C(C)(C)C)C S14244 c1cc2c(cc1Cl)C(=C(CS2)C#N)Cl SEW01700 Cc1c(nc(o1)C(=O)NNC(=O)C)c2ccccc2 SEW01719 c1cc(sc1)SCCC(=O)Nc2ccc(cc2)Cl SEW01770 c1ccc2c(c1)[nH]c(n2)/C(=C/c3ccc(c(c3)Cl)Cl)/C#N PHG00735 c1ccc(cc1)C2=N/C(=C/c3ccc(s3)c4cccs4)/C(=O)O2 SP01247 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N/N=C/c3cccc(c3)[N+](=O)[O-] SPB00152 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3c(cccc3Cl)Cl SPB00190 COc1c(cc(cc1Br)c2nc(on2)CSC)Br SPB00232 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)N SPB00316 CCn1c2cc(c(cc2nc1SCC(=O)O)Cl)Cl SPB02604 COC(=O)c1cnn(c1/C=N/OC(=O)Nc2ccc(cc2)Cl)c3ccc(cc3F)F SPB05321 Cc1c(c(nc(n1)c2ccccc2OC)S)C(=O)C SPB05339 Cc1c(c(nc(n1)c2ccccc2OC)SCC#C)C(=O)C SPB05357 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)O SPB05427 CC1=C(C(N=C(N1)C(F)(F)F)(C)O)Oc2ccc(cc2)Cl SPB05458 C=CCSc1n[nH]c(=O)n1c2ccc3c(c2)OCCO3 SPB07902 c1c(cc(cc1C(F)(F)F)C(F)(F)F)c2[nH]nc(n2)S SPB00415 CC(C)(C)c1ccc(cc1)c2nc(on2)C(=O)NN SPB00452 c1cc(c(cc1Cl)Cl)OCCOC(=O)c2cc(cc(c2)Cl)Cl SPB00472 c1cc(c(c(c1)Cl)COc2c(cc(cc2Br)C#N)Br)F SPB00476 c1cc(c(c(c1)Cl)NNC(=O)c2ccc(o2)[N+](=O)[O-])Cl SPB00525 c1cc(c(cc1F)F)c2nc(cs2)CC(=O)O SPB02727 Cc1ccc(cc1NC(=O)CSc2nnc(s2)SCC(=O)Nc3cc(ccc3C)F)F NRB00189 CCC(C#N)(c1ccccc1)c2ccc(cc2)/N=C/c3cc(cc(c3O)Cl)Cl NRB00243 COc1ccc(cc1)c2c(c(=O)c3ccc(cc3o2)OC)O NRB00325 COC(=O)/C(=C(\C#N)/c1ccc(o1)Br)/C#N NRB00511 COc1ccc(cc1OC)/C=C/2\C(=O)OC(=N2)/C=C/c3ccccc3 PHG00753 Cc1cc2c(cc1C)nc([nH]2)c3cc4cc(cc(c4oc3=O)Cl)Cl PHG00765 c1ccc2c(c1)[nH]c(n2)c3cc4cc(ccc4oc3=O)Br PHG00766 CC(=O)N(c1ccc2c3c1cccc3CC2)C(=O)C PHG00865 CC(CN1C(=O)c2cccc3c2c(cc(c3)[N+](=O)[O-])C1=O)O PHG00997 c1cc(sc1)/C=N/c2ccc3c(c2)OCO3 RB00126 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)N/N=C/c3c(cccc3Cl)Cl SPB00329 c1cc(c(c(c1)Cl)NNS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Cl SPB00537 Cc1c(c(c(c(c1C)C)S(=O)(=O)NNc2c(cccc2Cl)Cl)C)C SPB00538 CCOC(=O)c1nc(no1)c2cccs2 SPB00567 CC(C)(C)c1ccc(cc1)c2nnc(n2CCCOC)SCC(=O)NNC(=O)C(Cl)Cl SPB00590 c1cc(cc(c1)C(F)(F)F)c2nnn(n2)Cc3ccc(c(c3)Cl)Cl RJF02130 CC(C)(C)C(=O)Cn1nc(nn1)c2cccc(c2)C(F)(F)F RJF02133 c1cc(ccc1c2nnc(o2)N3CCOCC3)Cl RJF02161 c1ccc(cc1)C2=N/C(=C\c3c(cccc3Cl)F)/C(=O)O2 S06348 CC1=N/C(=C\c2ccc3c(c2)OCO3)/C(=O)O1 S06429 c1ccc(cc1)NC2CC(=O)N(C2=O)c3ccccc3 S14265 c1ccc(cc1)S(=O)(=O)C2CC(=O)N(C2=O)c3cc(cc(c3)Cl)Cl S14294 CC1=C(C2(c3ccccc3NC2=O)C(=C(O1)N)C#N)C(=O)OCCOC S14431 CN(c1c(cc(cn1)C(F)(F)F)Cl)NC2c3ccccc3C(=O)O2 SEW01848 Cc1c(c(on1)C)C(=O)NC(=N)C23CC4CC(C2)CC(C4)C3 SEW01857 Cn1c(c(c(n1)C(F)(F)F)c2ccccc2)/N=C/c3cccc(c3)C(F)(F)F SEW04792 CC(C)(C)c1csc(n1)c2ccc(s2)c3cccs3 SEW04838 COC(=O)c1cc(ccc1N2CCOCC2)[N+](=O)[O-] SEW04885 c1cc(oc1)c2nnc(o2)c3cc(oc3C(F)(F)F)c4ccc(cc4)Cl SEW04925 CCc1cc2c(cc1c3csc(n3)c4cnccn4)C(CCC2(C)C)(C)C SEW06509 c1ccc(c(c1)CSCCNC(=O)c2ccc(c(c2)Cl)Cl)Cl SEW06544 c1cc(c(cc1Cl)Cl)C(Cn2cncn2)O RJC01325 CCOc1ccc(cc1)C2C(=C(NC(=O)N2)C)C(=O)OC RJC01425 CN(C)c1c(nc2ccccc2n1)N(C)C RJC01468 CCC1C(NC(CC1(c2ccc(cc2)F)O)c3ccccc3)c4ccccc4.Cl RJC03625 CCOC(=O)C(C(F)(F)F)(NC(=O)Nc1ccc(c(c1)Cl)Cl)OCC(F)(F)F RJC03642 Cn1c(ccc1S(=O)(=O)C)C=C(C#N)C#N NRB00519 c1cc(cc(c1)Sc2cccc(c2)C(=O)O)C(=O)O NRB00550 c1c(cc(c(c1C(=O)O)Sc2c(cc(cc2Cl)Cl)C(=O)O)Cl)Cl NRB00565 CS(=O)c1nc2ccccc2s1 NRB00584 c1ccc(cc1)Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] NRB00608 CC(=O)N1[C@@H](SC([C@@H]1C(=O)O)(C)C)c2ccccc2 NRB04499 c1cc(ccc1N2C(=O)C=CC2=O)Oc3ccc(cc3)Cl RB00150 CCc1cccc(c1N2C(=O)C(=C(C2=O)C)C)CC RB00296 CCOC(=O)c1ccc(cc1)NC(=O)/C(=C/C(=O)O)/C RDP00040 Cc1ccc(c(c1)C)/N=C/2\N(CCS2)C.I RDR00235 Cc1cc([nH]c1C=C(C#N)C#N)C SEW04972 Cc1cc(ccc1OC)CNCc2ccc(c(c2)OC)OC SEW04974 Cc1cc([nH]c1/C=N/Nc2ccc(cc2[N+](=O)[O-])C(F)(F)F)C SEW04991 Cc1cc([nH]c1/C=N/Nc2ccc(cc2)[N+](=O)[O-])C SEW05120 c1cc(ccc1CS(=O)(=O)CCNC(=O)c2ccc(cc2)Cl)F SEW06623 CC(C)(C)c1cc(n(n1)c2ccc(cc2)Br)C(C)(C)C SEW06656 CC(C)(C)C(=O)/C=C\1/c2cc(ccc2NC1=O)Br SPB00625 CCOC(=O)NNC(=S)Nc1ccccc1 SPB00710 COc1ccc(cc1)c2c(c(=O)c3ccccc3o2)Cl RJC01629 COc1cccc2c1C(=O)CC(O2)c3ccccc3 RJC01638 c1ccc2cc(ccc2c1)C(=O)C3=NNCC3c4ccc5c(c4)OCO5 RJC01643 COc1ccc(cc1OC)CCNC(=O)/C=C/C(=O)O S01354 c1ccc(cc1)CN2C(=O)C=CC2=O S01402 Cc1ccc(cc1)/C=C\2/C(=O)OC(=N2)c3ccccc3 S01412 Cc1ccc(cc1F)/N=C\2/NCCS2 S01470 c1ccc(cc1)C2=N/C(=C\c3ccco3)/C(=O)O2 S01515 Cc1cc(c(c(c1)C)n2c(nnn2)SCC#C)C S07173 CC(C)(C)NNC(=S)Nc1ccc(c(c1)Cl)Cl S07298 CCOC(=O)C(CSC1CC(=O)N(C1=O)c2ccccc2)N.Cl S14687 COc1ccc(cc1)/C=C/2\CCCc3ccccc3C2=O S14712 c1ccc(cc1)NNC(=O)N S14722 C=CCOc1ccc(cc1)C=C(C#N)C#N S14814 c1cc(sc1)CCNC(=O)c2ccc(cc2)OC(F)(F)F SEW02188 CC(C)c1nnc(o1)c2cc3c(s2)ccs3 SEW02203 COC(=O)c1ccccc1n2cccc2C(=O)OC SEW05135 COC(=O)CCCCCCCC(=O)Nc1nnc(s1)C(F)(F)F SEW05139 COc1ccc(cc1)CN(Cc2cc(c(c(c2)OC)OC)OC)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05140 c1cc2c(cc1F)c(c3c(n2)CCCC3)C(=O)O SEW05227 c1cc(c(c(c1)F)OCc2ccc(cc2)Cl)OCc3ccc(cc3)Cl SEW05242 Cc1ccc2c(c1)sc(n2)c3ccc(cc3)NC(=O)c4ccccc4O SJC00292 C=CCNC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC01713 c1ccc2c(c1)c3ccccc3n2CC(CN4CCNCC4)O.Cl.Cl RJC01739 c1ccc2c(c1)c3cc(ccc3n2CN4CCCCC4)Br RJC01748 c1ccc2c(c1)C(=C(C2=O)c3ccc(cc3)I)O RJC01752 C=CCC1(CCCCC1)Nc2ccc3ccccc3c2 RJC03990 CCOCCNS(=O)(=O)c1cccc2c1cccc2N NRB00859 COc1ccc(c2c1OCCO2)Br NRB00874 CC(=O)Nc1cc2c(cc1[N+](=O)[O-])OCCO2 NRB00894 CC(=O)/C(=C\N1CCCCC1)/c2nnnn2c3ccc(cc3)Cl NRB05010 c1cc(ccc1C(=O)O)N/C=C/C(=O)c2ccc(cc2)Cl NRB05050 c1cc(cc(c1)Cl)Nc2ccc(cc2)N=Nc3ccc(cc3)[N+](=O)[O-] NRB01168 Cc1cc(ccc1NC(=S)NCCCOC)Cl RDR00360 c1cc(cnc1)/N=C/c2cc(cc(c2O)Cl)Cl RDR00364 c1ccc(cc1)c2nc(sn2)N3CCCC3 RDR03890 COCCCNC(=S)Nc1ccc(cc1)Oc2ccc(cc2)Cl RDR00914 Cc1c(nc(s1)Nc2ccccc2)CC(=O)OC SEW05313 c1cc(ccc1c2cc(c(o2)C(F)(F)F)C(=O)Nc3ccc(cc3)Oc4ccc(cc4)Cl)Cl SEW05360 c1ccc(cc1)NC(=O)c2cc(oc2C(F)(F)F)c3ccc(cc3)Cl SEW05361 Cc1c(c(on1)C)C(=O)O/N=C/2\CCSc3c2cc(cc3)F SEW05369 Cc1c(cc(o1)c2ccc(cc2)Cl)C(=O)/C(=C/Nc3ccccc3)/C#N SP00157 c1cc2c(cc1Cl)c3c([nH]2)CCCC3 RJC03691 c1ccc(cc1)CC(C#N)c2ccccc2 RJC03710 Cc1cc2c(nc1)CCC(C2)Cc3ccc(cc3)OC RJC01931 CCOC(=O)C(C(F)(F)F)(Nc1nc2ccccc2s1)NC(=O)C RJC01979 CCOC(=O)C(C(F)(F)F)(Nc1cccc(n1)C)NC(=O)C RJC01994 Cc1cc(nc(n1)SCc2c(cccc2Cl)F)O RJF00079 c1ccc(cc1)C(=S)NCCO S02163 COc1ccc(cc1OC)CC/N=C\2/NCCS2 S02179 c1cc(cc(c1)F)c2nc3ccc(cc3c(=O)o2)[N+](=O)[O-] S02434 Cc1ccccc1c2nc3cc(ccc3c(=O)o2)Cl S02596 COc1ccc(cc1)C2C(=Cc3ccccc3O2)[N+](=O)[O-] S09107 c1cc(ccc1C2CCCCC2)N3C(=O)C=CC3=O S09389 COc1ccc2c(c1)CCC3=C2NC(=S)NC3c4cccc(c4)Br S15334 c1ccc2c(c1)C=C(C(O2)c3ccc(cc3)C4C(=Cc5ccccc5O4)[N+](=O)[O-])[N+](=O)[O-] S15345 CC(=O)N1CCc2c3ccccc3[nH]c2C1C(F)(F)F SEW02505 c1cc(sc1)Cc2cccs2 SEW02590 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)F SEW02648 CN(Cc1ccccc1)S(=O)(=O)c2c(cc(cc2Cl)C(F)(F)F)Cl SEW05432 Cc1c(c(on1)C)C(=O)Nc2ccc(c(c2)C(=O)OC)N3CCOCC3 SEW05451 c1cc(ccc1NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F SEW05464 CC(C)(C)c1cc(cc(c1O)C(C)(C)C)c2csc(n2)c3ccc(cc3)Cl SP00404 c1cc(ccc1c2nc(cs2)c3ccc4c(c3)OCCCO4)Oc5ccc(cn5)C(F)(F)F SP00426 CC1CN=C(S1)N(Cc2ccccc2)C(=O)Nc3ccccc3 RJC02026 c1ccc(cc1)C2=NN(C(C2)c3ccc(cc3)[N+](=O)[O-])c4ccccc4 RJC02118 C[C@H](C(=O)O)NC(=O)OC(C)(C)c1cc(cc(c1)OC)OC.C1CCC(CC1)N RJC02201 c1cc(cnc1)CN\2C(=O)CS/C2=N\c3cc(cc(c3)Cl)Cl RJF00177 c1cc(c(cc1NC(=S)N)Cl)F RJF00180 c1ccc(cc1)CC(Cc2ccccc2)(C#N)C#N NRB01312 Cn1c2ccccc2sc1=S NRB01427 CCOC(=O)Nc1ccccc1C(=O)OC P00099 c1ccc2c(c1)ccc3c2sc(c3)C(=O)NNS(=O)(=O)c4ccc(cc4)F PD00024 CN(C)CC1(CCCCC1)CC(c2ccccc2)OC(=O)c3ccc(cc3)[N+](=O)[O-].Cl NRB02288 c1cc(oc1)/C=C(\C#N)/c2ccc(cc2)Cl RDR00922 c1ccc(cc1)/C(=C/c2ccc(cc2)Cl)/C#N RDR00924 c1ccc(c(c1)c2csc(n2)NCC3CCCO3)Cl RDR00931 c1cc(ccc1C(=O)NCCOC(=O)c2ccc(cc2)[N+](=O)[O-])[N+](=O)[O-] RF00118 CCc1cccc(c1NC(=O)C(Cl)Cl)CC RF00335 Cc1cc(nc(c1C#N)SCC(=O)C)C RF00395 c1ccc(c(c1)/C=N/NC(=S)Nc2cccc(c2Cl)Cl)Cl RDR01131 CCOC(=O)N/N=C(/C(=N/NC(=O)OCC)/C)\C SEW05546 c1cc(ccc1Sc2ccc(c(n2)Sc3ccc(cc3)Cl)[N+](=O)[O-])Cl SEW05568 c1cc(nc(c1[N+](=O)[O-])N2CCN(CC2)CCO)N3CCN(CC3)CCO SEW05574 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2ccc(cc2)OC SEW05603 c1cc2c(cc1Cl)sc(n2)N3CCCCC3 SEW05613 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)c4ccc5c(c4)OCCCO5 SP00490 c1ccc(c(c1)/C=N/O)[N+](=O)[O-] RJC02279 CC(=O)[C@]1(CC[C@@H]2C1(CC[C@H]3[C@H]2CC[C@@H]4C3(CCC(=O)C4)C)C)O RJC02364 COC(=O)Cn1c(nnn1)c2ccc(cc2)Cl RJC02395 CCCCCCCCC(=O)NCc1ccco1 RJC02396 c1ccc(c(c1)/C=N/NC(=O)Cn2nc(nn2)N3CCCCC3)Cl RJF00312 c1ccnc(c1)SC2CC(=O)N(C2=O)c3ccc(cc3)[N+](=O)[O-] S03506 c1cc(cc(c1)[N+](=O)[O-])/C=N/c2ccc(cc2C#N)Cl S03546 COc1cc(cc(c1)OC)/C(=N/O)/N S03549 Cc1ccc(cc1)S(=O)(=O)NC(C(C)C)C(=O)O S03579 CCOC(=O)/C(=C/c1cccc(c1)Br)/C#N S10272 c1cc(cc(c1)Br)c2cc(c3c(cc(cc3n2)C(F)(F)F)C(F)(F)F)C(=O)O S10281 COc1ccccc1N/C(=N\C#N)/SC SEW00079 CCOC(=O)c1c(nc(n1c2ccccc2OC)SC)NC(=O)C(Cl)(Cl)Cl SEW00087 COc1ccccc1c2csc(n2)Nc3cccnc3 SEW03094 c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)NC(=O)Nc3cccc(c3)C(F)(F)F SEW03117 c1ccc(cc1)c2c(csc2C(F)(F)F)NC(=S)N SEW03168 CC(C)NC(=O)NNC(=O)c1ccc[nH]1 SEW05663 CN(C)c1ccc(c(c1)Cl)/C=C(\C#N)/S(=O)(=O)C SEW05682 c1cc([nH]c1)C(=O)NNC(=O)c2cc(cc(c2)Cl)Cl SEW05697 Cc1c(c(on1)C)NC(=O)N SEW05714 Cc1ccc(cc1)c2csc(n2)c3ccno3 SP00624 c1cc(cc(c1)F)c2csc(n2)c3ccno3 SP00633 c1cc(cc(c1)OC(F)F)c2csc(n2)c3ccc(cc3)C(F)(F)F SP00659 c1ccc(cc1)Oc2cc(c(cc2Oc3ccccc3)C#N)C#N RJC02436 c1cc(ccc1C(=O)NCC(=O)N)Cl RJC02448 Cc1nnc(s1)SCc2ccc(cc2)[N+](=O)[O-] RJC02492 CC(=O)c1ccc(cc1)NC(=O)CSc2nc3ccccc3o2 RJC02508 Cc1c(c(nc(n1)c2ccccn2)O)CC3CC3 RJF00482 COCc1cc(nc(n1)NC(=N)Nc2cc(ccc2Cl)C(F)(F)F)O RJF00548 c1ccc(cc1)/C(=N\O)/CN2CCOCC2 NRB02471 c1ccc(cc1)COc2ccccc2C(=O)[C@@H]3[C@@H](N3C4CCCCC4)c5ccc(cc5)[N+](=O)[O-] NRB02657 c1ccc(cc1)C\2=NOC(=O)/C2=C\c3ccc4c(c3)OCO4 PD00179 CC(=O)c1ccc(cc1)NC(=O)c2ccccc2C(=O)O PD00208 c1ccc2c(c1)c(=O)n3c(n2)SCCC3 PD00217 COc1ccc(cc1OCc2ccccc2)/C=C/[N+](=O)[O-] NRB03047 Cc1ccc(cc1)S(=O)(=O)Oc2ccccc2/C=N\NC(=S)Nc3cc(ccc3Cl)Cl RDR01248 c1ccc(cc1)C(=O)CSc2nc3ccccc3c(=O)n2Cc4ccco4 RDR01280 c1ccc(cc1)C\2=NOC(=O)/C2=C\c3c(cccc3Cl)Cl RF00973 CCCc1c(nc(nc1O)S)C RDR01510 c1ccc(c(c1)c2c(c[nH]n2)/C=C\3/c4ccccc4NC3=O)[N+](=O)[O-] SEW05803 COc1cccc(c1/C=N/Nc2ccc(cn2)[N+](=O)[O-])OC SEW05812 CC(C)(C)c1ccc(s1)C(=O)Nc2ccc(cc2)Cl SEW05829 CC1(CCC(c2c1ccc(c2)c3csc(n3)CS(=O)(=O)C(C)(C)C)(C)C)C SP00755 CC1(CCC(c2c1ccc(c2)c3csc(n3)c4ccc(cc4)Cl)(C)C)C SP00758 CCCc1ccc(cc1)c2nc(no2)c3ccc(cc3)C SP00766 c1cc(ccc1NC(=S)NNC(=O)Cn2nc(nn2)N3CCCC3)Cl RJF00336 CCCCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)OC RJC02611 CCOc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(n2)C RJC02635 c1csc(n1)NC(=N)NC(=N)N.Cl RJF00663 COc1cc(cc(c1)OC)NC(=N)NC(=N)N.Cl RJF00670 Cc1cccc(c1)c2nc(cc(n2)OC(=O)N(C)C)COC RJF00712 C/C(=C/c1cccc2c1cccc2)/[N+](=O)[O-] S03997 Cc1c(c(c(c(c1C)C)C/N=C(\C)/c2ccccc2O)C)C S04017 c1cc(ccc1NC(=O)N)Cl S04036 CC1CCC2C(C1)C(=O)N(C2=O)c3ccc(cc3)Cl S10865 CC(C)(C)OC(=O)/C(=C/c1cccs1)/C#N S10890 C/C(=N\N=C/1\NC(=O)C(S1)CC(=O)O)/c2ccccn2 S11076 CC(CC(=O)O)S(=O)(=O)c1ccc(cc1)Cl SEW00548 CCOC(=O)C1CSC(=C(N1)C)C(=O)OCC SEW00603 c1cc2c(cc1Cl)-c3c(snn3)CS2(=O)=O SEW00605 CC1(OC(=O)C(=Cc2ccc(s2)SC)C(=O)O1)C SEW03576 Cc1c(c(on1)C)C(=O)N2CCOCC2 SEW05862 CC(C)(C)c1ccc(cc1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05911 c1cc(ccc1c2nc(on2)c3ccc(o3)Oc4cc(cc(c4)Cl)Cl)OC(F)(F)F SP00826 CC(C)(C)c1cc(n(n1)Cc2ccccc2)c3nc(no3)c4ccc(cc4)C(F)(F)F SP00846 Cc1cc(ccc1Nc2ncnc(n2)N)Br RJF00566 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)Cl)F RJC02643 Cc1ccccc1C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2cccc(n2)C RJC02645 CCOC(=O)C(C(F)(F)F)(NC(=O)c1ccco1)O RJC02677 Cc1c(c(nc(n1)N)O)Cc2c(cccc2Cl)F RJF00816 c1ccn(c1)c2ncnc(n2)Nc3cc(cc(c3)Cl)Cl RJF00856 CN(/C=C/c1nnnn1c2ccc(cc2)OC)c3ccccc3 NRB03125 Cc1ccc(cc1)n2c(nnn2)/C=C/N3CCCCCC3 NRB03128 c1ccc(cc1)c2cc(c(c3c2CCCC3=O)C(=O)c4ccccc4)c5ccccc5 NRB03166 c1cc(ccc1n2c(nnn2)/C=C/N3CCCC3)Br NRB03212 CC(=O)Nc1ccc(cc1)S(=O)(=O)NCc2csc3c2cccc3 PD00430 c1cc(oc1)CNC(=S)N/N=C/c2ccncc2 RDR01605 Cc1cc(c(c(c1)C)NC(=S)NCCCN2CCOCC2)C RDR01622 c1ccc(c(c1)NC(=N)NC(=N)NN)F.Cl RDR01642 c1ccc(cc1)c2cc(=O)n3c(csc3n2)c4ccc(cc4)Cl RDR01714 Cc1c(c(c(cn1)Br)O)OCC(=O)O RF01402 c1cc(ccc1NC(=S)NNC(=O)c2cnc3n(c2=O)CCS3)F SEW01398 c1cc(c(nc1)N2CCN(CC2)C(=O)CSc3ccc(cc3)Cl)C(F)(F)F SEW05968 c1cc(ccc1C(=O)Nc2ccc(nc2)N3CCN(CC3)c4ccc(cn4)C(F)(F)F)Cl SEW05983 c1cc(c(nc1)N2CCN(CC2)C(=O)NC3CCCCC3)C(F)(F)F SEW06005 c1ccc(c(c1)c2cc(c(o2)C(F)(F)F)c3nc(no3)c4ccc(cc4)OC(F)(F)F)Cl SP00948 c1cc(oc1)c2cc(n(n2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)N SP00976 Cc1ccccc1OC(=O)Nc2ccc(cc2)Cc3ccc(cc3)NC(=O)Oc4ccccc4C RJC02870 CC1=C(C(NC(=O)N1C)c2ccccc2)C(=O)OCc3ccccc3 RJC02897 c1ccc(c(c1)NC(=N)NC(=N)N)F RJF01026 c1cc(c(cc1NC(=N)NC(=N)N)Cl)Cl RJF01034 Cc1cccc(c1)NC(=S)Nc2c(cccc2C(C)C)C(C)C S04432 Cc1c(cccc1Cl)NC(=S)NN(C)C S04444 c1c(cc(cc1Cl)Cl)NC2=NCCS2 S04530 CN(C)C(=S)Nc1cc(cc(c1)Cl)Cl S04545 C1CSCCN1C(=N)N[N+](=O)[O-] S12066 c1cc(ccc1N2C(=O)CSC2=O)Cl S12084 c1ccc(c(c1)C(=O)NCc2ccc(cc2)c3csnn3)C(F)(F)F SEW00849 CNC(=S)NCc1ccc(cc1)c2csnn2 SEW00859 CC(CC(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)C(Cl)(Cl)Cl SEW00885 c1c(cc(c(c1Br)N)Br)c2csnn2 SEW00894 CC1=NN(C(=O)C1)c2ccc(cc2)c3csnn3 SEW00895 Cc1cc(c(n1c2ccc(cc2)Cl)C)C(=O)C(F)(F)F SEW00986 c1cc(ccc1NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl)F SEW06006 Cc1ccc(n1c2ccc(cc2)n3c(cc(n3)C(C)(C)C)C(C)(C)C)C SEW06008 COc1ccccc1N2CCN(CC2)C(=O)c3c(cccc3Cl)F SEW06022 Cc1c(c(on1)C)c2nnc(o2)c3cccc(c3)C(F)(F)F SEW06034 CN(C)c1ccc(cc1)NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06039 c1cc2c(cc1C(=O)O)C(=O)N(C2=O)CC(=O)O RJC02908 CN(C)c1ccc(cc1)C2C3C(C(=O)N(C3=O)c4ccccc4Cl)ON2c5ccccc5 RJC02922 c1cc2c(cc1NC(=O)/C=C\C(=O)O)OCCO2 S05228 Cc1ccc(cc1)C(=O)CC(c2cccs2)C(=O)c3ccc(cc3)C(F)(F)F S13496 c1cc(ccc1NC(=O)Nc2ccc(cc2)SC(F)(F)F)SC(F)(F)F S13692 CSc1ccc(cc1)/C=C(\C#N)/C(=O)N S13822 c1cc(c(cc1N2CCCC2=O)Cl)Cl S13835 CC1CC(CC(C1)(C)C)/N=C/c2ccc(s2)[N+](=O)[O-] S05769 c1cc(ccc1SC(=O)c2cnc3n(c2=O)CCS3)Cl SEW01401 c1cc(ccc1c2c(nco2)C(=O)NN)Cl SEW01414 CC1=C(C(C(=C(N1)C)C(=O)OC)c2cccs2)C(=O)OC SEW04366 Cc1c(c(c(c(n1)C)C(=O)O)c2cccs2)C(=O)O SEW04369 COC(=O)c1cc2c(s1)-c3cc(ccc3S(=O)(=O)C2)Cl SEW01807 c1cc(cc(c1)Br)NC(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW06075 c1cc(sc1/C=N/O)Cl SEW06085 COc1ccccc1N2CCN(CC2)C(=O)C3CCCCC3 SEW06097 CC(C)c1ccccc1NC(=S)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06103 Cc1ccc(cc1)SCC(=O)N2CCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl SEW06126 c1ccc2c(c1)/C(=C/c3cccn3c4ccc(cc4)C(F)(F)F)/C(=O)N2 SEW06160 COCc1cc(nc(n1)c2ccc(cc2)Cl)O RJF01064 COc1ccccc1CC(=O)NC2CCN(CC2)Cc3ccccc3 RJC03042 COc1ccc(cc1OC)CCNS(=O)(=O)c2cccc(c2)C(F)(F)F RJC03063 CC1(c2ccccc2N3C1=CC(=O)C(C3=O)(c4ccccc4)O)C RJC03125 Cc1cc(c(c(c1)C)S(=O)(=O)Oc2ccc(cc2)C3SCCS3)C RJC03141 CCC(C)Cn1c(nnc1Sc2ncc(s2)[N+](=O)[O-])O SPB07592 CCOC(=O)NNC(=S)NC1CC2CC1C=C2 SPB07666 CC(C)(C)c1cc(n(n1)C)C(=O)Oc2ccc(cc2)Cl SPB07695 CC(C)(C)c1ccc(cc1)NC(=O)c2cc(nn2C)C(C)(C)C SPB07696 CC(C)(C)c1cc(n(n1)C)C(=O)O/N=C(/c2ccc(cc2)Cl)\N SPB07697 CC(C)(C)c1cc(n(n1)C)C(=O)Sc2ccccc2 SPB07706 c1ccc(cc1)C(=O)NC2CCN(CC2)Cc3ccc(c(c3)Cl)Cl RJC03004 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NNC(=O)c3csc(n3)C SPB02497 CCn1c(cc(n1)C)C(=O)NNC(=S)Nc2ccccc2 SPB02498 CCn1c(cc(n1)C)c2nnc(n2c3ccc(cc3)Cl)SCc4ccccc4 SPB02507 CCn1c(cc(n1)C)c2nnc(n2c3cccc(c3)C(F)(F)F)SCC(=O)c4ccccc4 SPB02539 CNNC(=S)NC1CC2CC1C3C2CC=C3 S06024 CC(c1ccccc1O)NCc2ccccc2 S06259 CC(=O)NC1=CC(=O)CC(C1)(C)C S06317 COc1ccc(cc1)C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-] S14109 Cc1ccccc1C(=O)N2C(SC(=N2)Nc3ccccc3)(C)C S14135 CCOc1nc2ccc(cc2c(=O)o1)C S14206 c1ccc(cc1)C(=O)/C=C/Sc2nc3ccccc3s2 NRB04232 CN(C)c1ccc(c(c1C#N)F)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl SEW01812 CN(C)/C=C/1\CSc2ccc(cc2C1=O)Cl SEW01818 COc1ccc(cc1)C(=O)n2cc3c(n2)-c4cc(ccc4SC3)Cl SEW01832 c1cc(c(c(c1)F)C(=O)OCc2cc(cc(c2)F)F)F SEW04693 c1ccc(cc1)C2=NC(OC2=O)C(F)(F)F SEW04708 c1ccc(cc1)/C=C/C(=O)O/N=C/c2ccc(cc2)Cl RJC03157 Cc1c(sc(n1)c2cccs2)c3ccnn3C(=O)NC(C)C SPB02625 c1cc(ccc1c2cnc(o2)SCC(=O)Nc3cc(cc(c3)Cl)Cl)Cl SPB02671 Cc1nc(cs1)c2nc(on2)c3ccc(cc3)C(F)(F)F SPB02688 Cc1ccc(cc1)C(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl SPB07914 CC(C)(C)c1ccc(cc1)c2nnc(n2CCCOC)SCC(=O)NNC(=S)NC SPB07954 Cc1cc(nn1C(C)(C)C)C(=O)O SPB07977 Cc1c2ccccc2sc1/C=C(/C(=O)O)\NC(=O)C SPB08007 CC(=O)Nc1cc2cc(cc(c2oc1=O)Br)Cl SPB08013 c1c(cc(cc1C(F)(F)F)C(F)(F)F)C(=O)NNC(=S)N SPB00409 CCn1c2cc(c(cc2nc1SCC(=O)OCC)Cl)Cl SPB02603 CC(C)n1c2ccc(cc2nc1SCC(=O)C(C)(C)C)C(F)(F)F SPB02750 CCn1c(c(c(n1)C)Br)C(=O)Sc2ccccc2Cl SPB02769 c1cc(ccc1CSc2ccc(cn2)C(F)(F)F)[N+](=O)[O-] SPB02841 c1cc(c(c(c1)Cl)CSc2ccc(cn2)C(F)(F)F)Cl SPB02843 c1cc(ccc1C(F)(F)F)NC(=O)c2ccno2 SPB02916 Cc1ccc(cc1)C(=O)/C=C/Nc2ccc(cc2Cl)Cl NRB04236 c1ccc2cc(ccc2c1)N/C=N/c3ccc4ccccc4c3 NRB04277 Cc1ccc(cc1)C(=O)/C=C/Sc2ccc(cn2)C(F)(F)F NRB04303 CCOC(=O)c1c(n(c(n1)S)CC(C)C)C(=O)OCC NRB04341 c1cc(c(c(c1)Cl)/C=N/NC(=N)Nc2[nH]cnn2)Cl NRB04441 COc1cccc(c1c2nc(nc(n2)N)N)Cl RDR02712 c1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)c3cc4cc(ccc4o3)Cl RDR02746 c1cc(ccc1c2cc3cc(ccc3o2)Cl)NS(=O)(=O)c4ccc(c(c4)Cl)Cl RDR02747 CC(C)(C)c1ccc(cc1)c2nc(nc(n2)N)N RDR02761 Cc1ccc(cc1)c2nc(cc(n2)OS(=O)(=O)c3ccc(cc3)C)C RDR02782 Cc1c(c(no1)c2c(cccc2Cl)Cl)CO/N=C(\C#N)/c3c(cccc3Cl)Cl SPB00917 Cc1c(c([nH]n1)c2cccs2)C(=O)NN SPB00947 Cc1cc(no1)c2c(c(no2)C)C(=O)N SPB03602 CCOC(CC(=O)NNC(=O)c1c(onc1c2c(cccc2Cl)F)C)OCC SPB06161 Cc1c(c(on1)COc2ccccc2)C(=O)Sc3ccc(cc3F)F SPB06259 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)N3CCCCC3 SPB08245 c1ccc(cc1)CC(=O)Nc2ccc(cc2)Cl SPB08371 c1ccc(cc1)C(=O)Nc2cccc(c2)[N+](=O)[O-] SPB08380 COc1ccc(cc1Cl)NC(=O)c2ccccc2 SPB08382 CC(C)c1ccc(cc1)n2c(nnc2SCc3ccc(cc3)[N+](=O)[O-])c4ccc(cc4)C(C)(C)C SPB01084 Cc1c(c(on1)c2c(nns2)C)C(=O)OC SPB03348 C/C(=N\NC(=S)N)/c1csc(n1)c2ccccc2 SPB03738 C/C(=N/Nc1nc(cs1)c2ccc(cc2)Cl)/c3csc(n3)c4ccccc4.Br SPB03739 CC(=O)Nc1ccc(cc1)S(=O)(=O)C[N+](=O)[O-] SPB03745 c1cc(cnc1)C2N(C(=O)CS2)Cc3ccc(cc3Cl)Cl S07097 c1cc(cnc1)C2N(C(=O)CS2)Cc3ccc(cc3)Cl S07098 CC(=O)c1ccccc1NC(=O)c2cc(ccc2Br)OC S07114 COc1ccc(c(c1)NC(=S)NC(=O)c2ccccc2)Br S07116 COC(=O)/C(=C/1\c2ccccc2NC1=O)/C#N S14435 CC1(CC2=C(CC1=O)C3(c4ccccc4NC3=O)C(=C(O2)N)C(=O)OC)C S14438 c1ccc(c(c1)c2c(nco2)C(=O)N)Cl SEW02025 c1cc(sc1)Sc2ccc(cc2C(=O)O)[N+](=O)[O-] SEW02074 c1ccc(c(c1)/C=N/c2ccc(cc2)Cl)OC(F)(F)F SEW02151 c1cc(ccc1/C=N/NC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(F)(F)F SEW04943 c1c(c(sc1S(=O)(=O)N2CCCCC2)Cl)Br SEW04947 Cc1cc(n2c(n1)nc(n2)SC/C(=N/O)/N)C SPB00995 c1c(c(cnc1O)C(=O)O)C(F)(F)F RF04283 Cc1cc(c(cc1Cl)Cl)SCc2cc(on2)C SPB01285 CN(CCOC(=O)c1ccc(cc1)Cl)c2c(cc(cn2)C(F)(F)F)Cl SPB06286 COC(=O)c1c(ccs1)NC(=O)C2CCCS2 SPB03842 CCOC(=O)C(=O)/C(=C/N(C)C)/Sc1ccc(cc1)Cl SPB03844 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(n3C)SCC(=O)c4ccccc4 SPB03945 CCc1ccc(cc1)S(=O)(=O)Nc2ccc(cc2)N3CCN(CC3)C SS00028 Cc1cccc(c1NC(=S)N(CCC#N)Cc2ccccc2)C SW00044 Cc1cccc(c1NC(=S)NC2CC(CC(C2)(C)C)C)C SW00048 Cc1ccc(cc1C)NC(=S)N2CCC(CC2)C SW00074 CCN(CC)c1ccc(c(c1)C)NCN2C(=O)c3ccccc3C2=O SW00100 CSc1cc([nH]c(=O)c1C#N)c2cccs2 SPB01100 Cc1coc(=O)n1c2ccc(c(c2)Cl)Cl RF05402 CCCCCCCCCCCc1nnc(n1c2ccccc2C(F)(F)F)SCc3ccc(cc3)C SPB01554 Cc1cc(nc(n1)O)C(=O)OC SPB06320 CCCNC(=O)Nc1ccc(nc1)N2CCC(CC2)C(F)(F)F SPB06333 CCOC(=O)c1c(=O)c(cn(n1)c2ccc(cc2)C(F)(F)F)Sc3nnc(n3C)C(F)(F)F SPB04012 Cc1cc(n(c(=O)c1C#N)Cc2ccccc2F)C SPB06580 c1cc(cc(c1)Cl)NC(=O)Cn2c3c(cccn3)oc2=O SPB06593 c1cc2c(nc1)n(c(=O)o2)CC(=O)Nc3ccc(cc3)C(F)(F)F SPB06613 CCCCCCCCCCCCSc1nnc(s1)N S08084 Cc1ccc(c(c1)C(=O)Nc2ccc(cc2)Cl)N S08551 c1cc(c(cc1NC(=O)CC(CC(=O)O)c2ccc(cc2Cl)Cl)Cl)F S08560 CN(C)/C=C\1/C(=O)N(C(=S)S1)c2ccc(cc2)Br S08742 C=CCOc1ccc(cc1)/C=C/[N+](=O)[O-] S14817 c1cc2c(c(c1)[N+](=O)[O-])C(=O)N(C2=O)c3ccc(cc3)OC(F)(F)F S14930 Cc1c(c2c(o1)c(c(c(c2F)F)F)F)C(=O)Oc3cccc(c3)C(F)(F)F SEW02397 Cc1ccccc1C(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F SEW02447 Cc1c(c(n(n1)C)O)/N=N/c2ccc(cc2)S(=O)(=O)C SEW02450 c1cc(sc1)c2ccc(s2)CNc3ccc(cn3)[N+](=O)[O-] SEW02492 CCc1c(nc(s1)c2ccc(cc2)Cl)C(=O)OC SEW05293 COc1ccc(cc1)/C=C/2\CSc3ccc(cc3C2=O)F SEW05298 c1c(cc(cc1Cl)Cl)OC/C(=N/O)/N SPB01312 c1c(sc(n1)Sc2nnc(n2C3CCCCC3)O)[N+](=O)[O-] SPB01625 CC(C)(C)C(=O)O/N=C(/CS(=O)(=O)c1ccc(cc1)Cl)\N SPB01704 CSc1c(c(nc(n1)CSc2ccc(cc2)Cl)C3CC3)C#N SPB06403 Cc1c(c[nH]n1)Sc2ccc(cc2)Cl SPB04120 C=CCSc1nnc(n1Cc2ccco2)c3cc(nc(c3)OCC(F)(F)F)OCC(F)(F)F SPB06676 CS(=O)(=O)Nc1ccc(cc1)C#N SPB06755 Cc1cc(c(nc1)N/C=N/O)Br XAX00109 CCOC(=O)C1=C(OC2=C(C1c3ccc(cc3Cl)Cl)C(=O)CC(C2)(C)C)N XAX00144 c1ccnc(c1)SCc2ccc(cc2)C(F)(F)F SPB01827 c1cc(ccc1COc2ccc(cc2)C#N)C(F)(F)F SPB01837 c1cc(ccc1CSc2nnc(o2)c3ccc(nc3)OCC(F)(F)F)Cl SPB06668 COC(c1ccc(c(n1)SC)C#N)OC SPB04329 Cc1ccc(cc1)C(=O)n2c(c(c(n2)C)Sc3ncccn3)C SPB04366 c1ccc(cc1)C(=O)CSc2nnc(o2)c3ccc(cn3)C(F)(F)F SPB06832 c1cc(ccc1C(=O)N2CCN(CC2)c3c(cncc3Cl)Cl)Cl SPB06844 c1ccc2c(c1)cc3ccccc3c2C=C(C#N)C#N S09746 COc1ccc(cc1)C(C[N+](=O)[O-])Sc2ccccc2N S09923 COc1ccc(cc1OC)CC(=O)NNC(=S)Nc2ccc(cc2)Cl S09964 CCOc1ccc(cc1)NC23c4ccccc4CCC2C(=O)CS3 S15364 C1C2CC3CC1CC(C2)C34NC(=O)CS4 S15377 c1ccnc(c1)c2nc(on2)c3cc(sc3)[N+](=O)[O-] SEW02749 c1ccc(cc1)c2c(c(ns2)N3CCCC3)C#N SEW02751 c1ccc(cc1)c2cn(nc2C(F)(F)F)C(=O)c3ccc(cc3)Cl SEW02810 c1ccc(cc1)c2c(nc(s2)NC(=O)c3cccs3)C(F)(F)F SEW02839 Cc1c(c(nc(n1)c2ccccn2)N3CCCC3)Cl SEW02969 c1ccc(cc1)Oc2ccc(cn2)C=C(C#N)C#N SEW05536 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)C(F)(F)F)Cc3cccnc3)C SPB01936 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)Nc3ccccc3)C#N SPB06801 c1cc(cc(c1)C(F)(F)F)/C=N/NC(=S)N SPB04514 Cc1ccccc1CSc2cnc(nc2C)C SPB04582 COC(=N)NC(=S)Nc1cccc(c1)C(F)(F)F SPB06995 COC(=N)NC(=S)Nc1ccc(cc1F)F SPB06997 Cn1c(nnc1SCc2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl)C(F)(F)F SPB01849 c1ccc(c(c1)NC(=O)Nc2cccc(c2)C(F)(F)F)Sc3c(cncc3Cl)Cl SPB06904 CCOC(=O)c1c(noc1c2csc(n2)c3cccc(c3)C(F)(F)F)C SPB04713 CCOC(=O)c1cnc(nc1Nc2ccccc2Cl)C(F)(F)F SPB04764 CCOC(=O)c1cnc(nc1N/N=C\c2c(cccc2Cl)Cl)C(F)(F)F SPB04767 c1ccc2c(c1)C(=O)N3C2(OC(=O)c4c3cccc4)O S10559 Cc1cc(no1)NC(=O)CCCC(=O)O S10663 CS(=O)(=O)c1c(c(sn1)S(=O)(=O)C)C#N SEW00144 CSc1c(c(sn1)SC)C(=O)O SEW00190 CSc1c(c(sn1)SC)C(=O)Nc2ccc(cc2)Cl SEW00240 CC(C)(C)C(=O)NNC(=O)CSc1nc2cc(ccc2s1)Cl SEW00272 c1cc(ccc1C(=O)Oc2ccc3c(c2)c(co3)[N+](=O)[O-])C(F)(F)F SEW03541 c1cc(ccc1S(=O)(=O)C2CS(=O)(=O)CC2O)Cl SEW03548 Cc1c(snn1)c2nc(cs2)C(=O)O SEW03560 CN(C)c1cnn(c(=O)c1Cl)c2cnc3ccccc3n2 SEW05735 CCOC(=O)c1cnn(c1C)c2ccc(cc2)[N+](=O)[O-] SEW05785 CCOC(=O)c1cc2c(ccc(c2OC)OC)c(c1)OC(=O)C SEW05798 c1cc(ccc1c2csc(n2)COc3ccc(cc3)C4SCCS4)Cl SPB01942 c1ccc(cc1)c2[nH]c(nn2)Sc3nc(ns3)c4cccs4 SPB07012 C/C(=N\NS(=O)(=O)c1ccc(cc1)Cl)/c2cc(no2)c3ccccc3 SPB04825 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)c4ccc(cc4)[N+](=O)[O-] SPB04837 Cc1c(n2ccccc2n1)c3ccnc(n3)SCC(=O)Nc4ccccc4 SPB04844 c1cc(c(c(c1)Cl)CSc2nnc(s2)SCC(=O)N3CCC(CC3)C(F)(F)F)Cl SPB07228 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NNS(=O)(=O)c3ccc(c(c3)Cl)F SPB02129 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)O/N=C(/c3ccc(cc3)Cl)\N SPB02369 c1ccc(c(c1)/C=N/NC(=S)Nc2cc(ccc2Cl)C(F)(F)F)O RJF00949 Cc1ccc(cc1)Cn2nc(nn2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJF00977 CCSc1nc(cc(n1)O)N RJF01002 CCOC(=O)c1ccc(cc1)NC(=S)Nc2cccc(n2)N S04083 c1cc(c(c(c1)Cl)Cl)NC(=S)NN S04124 COc1ccc(cc1)N2C(=O)CSC23c4ccccc4NC3=O S11707 C/C(=C\c1ccc(cc1Cl)Cl)/[N+](=O)[O-] S11816 c1ccc(c(c1)N)SC2CC(=O)N(C2=O)c3cccc(c3)C(=O)O S11820 CCc1cccc(c1NC(=O)CC(C)(C)CC(=O)O)C S12037 CCCS(=O)(=O)/C(=C/c1cc(cc(c1)C(F)(F)F)C(F)(F)F)/C#N SEW00697 c1cc(ccc1COc2ccc(cc2)Cl)c3csnn3 SEW00714 c1ccc(cc1)CC(C(F)(F)F)OC(=O)Nc2ccccc2 SEW03724 c1cc(sc1)c2nc(no2)c3cc(c(c(c3)Cl)N)Cl SEW03756 Cc1ccsc1C=C2C(=O)OC(OC2=O)(C)C SEW03785 Cc1c(c(on1)C)C(=O)NNC(=O)c2cccc(c2)C(F)(F)F SEW05948 Cc1c(c(on1)C)S(=O)(=O)Nc2ccccc2OC(F)(F)F SEW05951 Cc1c(sc(n1)c2cccs2)C(=O)NN SPB02247 Cc1c(sc(n1)c2cccnc2)C(=O)N/N=C/c3c(cccc3Cl)F SPB02284 CC(C)c1ccc(cc1)NC(=O)CSc2nccn2C SPB02458 Cc1c(n(c(c1S(=O)(=O)Cc2ccc(cc2)F)N)Cc3ccccc3Cl)C SPB02477 Cc1c(c(n(n1)C)C(=O)Sc2cccc(c2)C(F)(F)F)[N+](=O)[O-] SPB02488 Cc1c(c(n(n1)C)C(=O)Sc2ccc(cc2)OC)[N+](=O)[O-] SPB02489 CCOC(=O)c1c(c(nc(n1)C)Sc2[nH]c(nn2)c3ccc(cc3)C(C)(C)C)C SPB07261 C/C(=N\Nc1ccccc1)/c2csc(n2)c3ccc(nc3)OCC(F)(F)F SPB07488 Cc1ccc(cc1)/C(=N/OC(=O)c2cc(n(n2)C(C)(C)C)C)/N SPB07518 CCOC(=O)c1cc(cc(n1)C(=O)OCC)Sc2ccccc2 SPB07538 Cn1c(cc(n1)c2ccc(s2)C(=O)O)C(F)(F)F MO07338 Cc1c(c(on1)c2ccc(cc2)Cl)C(=O)Sc3cccc(c3Cl)Cl SPB02372 CNC(=S)NNC(=O)c1csc(n1)c2cccs2 SPB02377 Cc1c(c(no1)c2ccccc2)c3nc4cc(ccc4c(=O)o3)Cl S04147 Cc1cccc(c1)c2nc(cc(n2)OCCOC)COC RJF01203 CCCCc1c(nc(nc1O)c2ccc(cc2)Cl)COC RJF01210 C1CC1CNC(=S)NCC2CC2 RJF01267 CC1=CC(NC(=S)N1c2ccc(cc2)Cl)(C)C RJF01337 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N\c3ccc(cc3)F S12458 COc1cc(cc(c1)OC)N2C(=O)CC(C2=O)Sc3ccccc3N S12655 C/C(=N\N=C\1/NC(=O)CS1)/c2ccc(s2)Cl S12745 c1cc(ccc1C(=O)CC(C#N)C#N)Cl S12809 Cc1ccc(cc1N2C(=O)CSCC2=O)F S12871 COC(c1c(cc(c(n1)SCc2ccccc2)C#N)C(=O)OC)OC SPB05117 COC(c1c(cc2c(c(sc2n1)C(=O)OC)N)C(=O)OC)OC SPB05168 c1cc(ccc1/C(=N/O)/N)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05169 Cc1c(c(no1)c2ccc(cc2)Cl)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(C)C SPB05190 CN(C)/C=C/C(=O)c1cc(no1)c2cccc(c2)C(F)(F)F SPB05244 CSc1c(c(=O)[nH]c(=O)[nH]1)C#N SPB05754 c1cc(ccc1C(=O)O/N=C(/c2ccc(nc2)Oc3ccc(cc3)Cl)\N)Cl SPB05795 c1cc(ccc1c2csc(n2)c3ccc(cn3)C(F)(F)F)Cl SPB05831 Cc1c(c(n(n1)C(=O)C)C)Sc2nnnn2c3ccccc3 SPB05878 c1ccc2c(c1)cccc2C/C(=N/O)/N SPB00822 c1ccc(cc1)c2nc(on2)CSc3[nH]c(nn3)N SPB00853 COC(c1c(cnn1c2c(cccc2Cl)Cl)C(=O)OC)OC SPB05264 Cc1c(sc2n1nc(n2)C(F)(F)F)C(=O)O/N=C/c3ccccc3 SPB05558 c1ccc(cc1)/C=c/2\c(=O)n3c(s2)nc(n3)c4ccccc4 SPB05598 COC(c1cc(nc(n1)SCc2c(cccc2Cl)Cl)O)OC SPB05721 c1cc(ccc1OCC(=O)N)Cl SPB05735 c1cc(ccc1c2nnc(o2)c3ccc(cn3)C(F)(F)F)Cl SPB05740 CC(C)(C)c1ccc(cc1)c2nnc(n2c3cccc(c3)C(F)(F)F)SCc4ccc(cc4)[N+](=O)[O-] SPB00955 c1ccc2c(c1)ccc(c2C3SCCS3)OC(=O)COc4ccc(cc4Cl)Cl SPB01019 Cc1ccc(cc1)NC(=O)c2c(noc2c3c(nns3)C)C SPB03368 c1cc(cnc1)c2nnc(o2)c3ccc(cc3)OC(F)(F)F SPB03502 c1cc(ccc1NC(=O)N2CCC(CC2)C(F)(F)F)Cl SPB05933 CCOC(=O)C(C(=O)OCC)Nc1ccccc1 SPB06295 CCOC(=O)c1cc(nc(n1)Sc2ccc(cc2)NC(=O)C)C SPB06309 c1cc(ccc1c2nc(cs2)C34CC5CC(C3)CC(C5)C4)Oc6ccc(cn6)C(F)(F)F SPB08342 Cc1ccc(cc1)NC(=O)c2c(c(sn2)Cl)Cl SPB08361 COc1ccccc1NC(=O)c2ccccc2Cl SPB08368 c1cc(ccc1C2SCCS2)OC(=O)Nc3ccc(cc3)Cl SPB00875 CC(C)(C)c1cc(n(n1)C)C(=O)Sc2cccc(c2)Br SPB03152 CCOC(=O)c1cc(nn1C(=O)c2ccc(cc2)C)C SPB01245 Cc1cc(no1)CSCc2ccc(cc2)Cl SPB01283 CC(C)Oc1ccc(cc1)/C=C(/C(=O)O)\NC(=O)C SPB08026 COc1ccc(cc1)NC(=S)Nc2ccc(cc2)OC S00062 COc1ccccc1NC(=S)NC2CCCCCCCCCCC2 S00111 Cc1ccc(c(c1)C)NC(=S)Nc2cccc(c2)C(F)(F)F S00154 COc1ccc(cc1)n2c(=O)c3ccccc3[nH]c2=S S00447 CC(C)(C#C)NC(=O)/C=C\C(=O)O S06952 CC(C)(C)c1ccc(cc1)C(=O)NCC(=O)O S06998 CC1=CC(=O)N(C1=O)c2ccccc2C(C)(C)C S14485 c1cc(cnc1)C2N(C(=O)CS2)Cc3ccc(cc3)F S14507 c1cc(ccc1Cn2c(=S)[nH]nn2)F S14525 c1cc(c(cc1Cl)Cl)/C=N/N=C\2/NC(=O)CCS2 S14541 c1ccnc(c1)NC(=O)CCC(=O)O S14590 Cc1cccc(c1NC(=O)NC(=O)c2csc(n2)c3ccc(cc3Cl)C(F)(F)F)C SEW01980 CCOC(=O)c1c(ocn1)c2ccc(cc2)OC SEW01989 Cc1cc(c(c(c1)C)Nc2nc(cs2)C(=O)C)C SPB03563 Cc1cc(no1)c2c(c(no2)C)C(=O)NN SPB03592 COCCCn1c(nnc1SC)c2ccc(cc2)C(F)(F)F SPB01437 c1cc(ccc1Cn2ccnc2c3ccc(cc3)C(F)(F)F)F SPB01486 COc1ccc(cc1)NC(=O)Cc2ccccc2 SPB08370 CCOC(=O)c1cc(c(nc1C(F)(F)F)Sc2ccccc2)C#N SPB06426 Cc1c(nc(nc1Sc2[nH]c(nn2)c3cc(cc(c3)Cl)Cl)C(F)(F)F)C SPB06502 Cc1nc(cs1)C(=N)NC(=O)c2ccc(cc2)Cl SPB06505 c1cc(cc(c1)C(F)(F)F)/C(=N/OC(=O)c2cccc(n2)C(F)(F)F)/N SPB06514 Cc1nc(cs1)c2nc(nc(n2)OC)N SPB03617 Cc1c(c(no1)C(=O)NNC(=O)Nc2ccccc2)c3csc(n3)c4csc(n4)C SPB03716 Cc1c(sc(n1)C)C(=O)NNC(=O)c2ccc(cc2)C(C)(C)C SPB01610 Cc1c([nH]cn1)C(=O)N/N=C/c2c(cccc2Cl)Cl SPB01617 c1cc(sc1)c2[nH]c(nn2)Sc3ncc(s3)[N+](=O)[O-] SPB01622 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)c3nnc(n3C)SCC(=O)c4ccc(cc4)Cl SPB03946 c1cc(cnc1)C2N(C(=O)CS2)c3ccc(c(c3)Cl)Cl S07066 c1ccc2c(c1)C(=O)N(C2=O)CNc3ccc(cc3F)I S01584 Cc1ccc(cc1)CNc2cccnc2 S01604 CCOc1ccc(cc1)NC(=S)Nc2ccccn2 S01715 Cc1ccc(cc1C)N2C(=O)C=CC2=O S01742 COc1ccc(cc1)CNc2ccc(cc2)C(=O)O S01757 CN(C)/C=C/C(=O)c1ccc(cc1)F S14944 c1ccc(cc1)c2c3ccccc3c(=O)[nH]n2 S15065 c1ccc2c(c1)c(n[nH]c2=O)c3ccc(cc3)Cl S15079 CC(C)(C)c1ccc(cc1)/C=C\2/C(=O)C3CCN2CC3 S15122 Cc1c2ccccc2n3c1/C(=N\OC(=O)Nc4ccc(cc4Cl)Cl)/CC3 SEW02359 c1cc(cc(c1)Cl)c2nc(on2)c3ccsc3 SEW02376 Cc1cc(n(n1)C(C)(C)C)C(=O)/C(=N/Nc2cccc(c2)Cl)/C#N SPB03810 c1ccc(c(c1)C(F)(F)F)NC(=S)NNC(=O)Cn2nc(nn2)CSc3ccc(cc3)Cl SPB01807 CN1CCN(CC1)c2ccc(cc2)NC(=O)c3cccs3 SS00026 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)Nc3cccc(c3)C(F)(F)F)C#N SPB06803 CC(C)C(=O)NNC(=O)c1c(ccs1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB06818 c1cc(sc1c2cnc(s2)N/C=N/O)Br XAX00054 CC(C)(C)c1ccc(cc1)NC(=O)CN2CCCCC2 XAX00063 CC(C)(C)c1[nH]c(=O)cc(n1)CSc2nnc(n2C)C(F)(F)F SPB03964 Cc1c(c(nc(n1)NC(=O)C)O)Oc2ccc(cc2)Cl SPB04001 CC(C)(C)c1ccc(cc1)C(=O)OCc2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3Cl)Cl SPB01896 c1cc(ccc1C2SCCS2)OC/C(=N\OC(=O)Nc3ccc(cc3)Cl)/N SPB01906 Cn1ccnc1Sc2cnc(nc2c3ccccc3)S SPB04176 CCOC(=O)c1cc(on1)c2cccs2 SPB04177 C/C(=N\CCc1c[nH]c2c1cccc2)/c3ccccc3O S07987 CC(C)c1ccc(cc1)NC(=S)NCCO S02898 CSc1cccc(c1)N2C(=O)CC(C2=O)Sc3ccccc3N S03017 c1cc(cc(c1)Br)NC(=O)/C=C/C(=O)O S03225 Cc1ccc(cc1C)N2C(=O)CSC23CCCCC3 S15388 c1cc2c(c(nn(c2=O)CCO)O)nc1 S15408 CCCSC(=S)c1c(nn(c1O)c2ccccc2)C S15549 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3cccs3 SCR00071 c1cc(ccc1c2csc(n2)c3ccc4c(c3)OCCO4)F SCR00134 COc1cc(cc(c1OC)OC)N/C=C(\C#N)/C(=O)c2ccsc2 SEW02731 Cc1c(c(nc(n1)c2ccc(cc2)C(F)(F)F)O)Oc3cccc(c3)C(F)(F)F SPB04095 CC(=O)/C(=C\N(C)C)/Sc1ccc(cc1)Cl SPB04117 COC(=O)c1ccc(c(c1)Oc2ccc(cc2Cl)Cl)[N+](=O)[O-] SPB01989 CCOC(=O)Cc1csc(n1)COc2ccc(cc2)C3SCCS3 SPB02084 Cc1c(c(n(n1)C)C(=O)/C(=C(\C)/NC)/C(=O)OC)[N+](=O)[O-] SPB02127 CCn1c(cc(n1)C)C(=O)n2c(c(c(n2)C)Sc3ncccn3)C SPB04374 Cc1ccc(cc1)CSc2nnc(s2)N/C=N/O XAX00076 CC(C)C(=N)NC(=S)Nc1ccccc1 SPB07020 c1cc(cnc1)/C=C(\C#N)/C(=S)N SPB07051 CCc1cccc(c1NC(=O)c2c(c3c(c4c(nc3s2)CCCC4)c5cccs5)N)CC SPB07082 CCCCCCCCCCCC1=NCCN1CCO XBX00281 c1cc(c(cc1Cl)[N+](=O)[O-])/N=N\c2cc(cc(c2O)F)F XBX00329 Cn1ccnc1Sc2cnc(nc2c3ccc(cc3)Cl)SCc4ccc(cc4)Cl SPB04200 CCOC(=O)c1cc(c(nc1C)SC)C#N SPB04233 Cc1cc(nn1c2c(cc(cc2Cl)Cl)Cl)C(=O)NNS(=O)(=O)c3ccc(cc3)Cl SPB02130 CCOC(=O)c1cc(on1)CSc2nnc(n2c3ccccc3)O SPB02143 c1cc(c(c(c1)Cl)Cl)c2nc(cs2)C(=O)Nc3ccc(cc3)F SPB02188 c1ccnc(c1)S(=O)(=O)Cc2nc(cs2)c3ccc(cc3)[N+](=O)[O-] SPB02233 CCOC(=O)/C(=C/c1c(ccs1)C)/C#N S09710 COc1cc(cc(c1OC)OC)/C=C/2\C(=O)N(C(=S)S2)c3ccc(c(c3)F)F S03843 CSc1ccc(cc1)N2C(=O)C=CC2=O S03870 c1cc(c(cc1CN2C(=O)C=CC2=O)Cl)Cl S03873 CC(CC(=O)Nc1ccc(cc1)Br)CC(=O)O S10547 COC(=O)c1c(n(nn1)c2cccc(c2)Cl)C(=O)OC SEW00279 CC(C)(C)C(=O)Cn1nc(nn1)c2ccc(cc2)C(F)(F)F SEW00316 Cc1cc(c(n1c2ccc(cc2)C(F)(F)F)C)/C=C(\C#N)/S(=O)(=O)C SEW03476 c1ccc(cc1)c2c(csc2C(F)(F)F)S(=O)(=O)Oc3ccc(cc3)Cl SEW03511 c1cc2c(cc1OCc3c(snn3)Cl)OCO2 SEW03529 Cc1cccc(c1)N/N=C(/C(=O)c2cccs2)\C(=O)C(F)(F)F SPB04439 Cc1c(c(nc(n1)N)O)Oc2ccccc2 SPB04460 Cc1nc(cs1)C(=O)NN SPB02297 Cc1nc(cs1)C(=O)NNC(=O)c2ccc(cc2)C(C)(C)C SPB02304 Cc1nc(cs1)c2nnc(n2C)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F SPB02320 Cc1ccc(cc1)CSc2nnc(n2C)Cc3ccsc3 SPB02366 CC(C)(C)c1csc(n1)c2ccc(nc2)n3cncn3 SPB07280 c1cc(cc(c1)NC(=O)N2CCN(CC2)Cc3ccc4c(c3)OCO4)C(F)(F)F SPB07291 CC(C)(C)C(=O)CSc1nnc(s1)c2cnccn2 SPB07303 CCOC(=O)c1c(noc1c2csc(n2)Nc3ccc(cc3)Cl)C SPB04697 Cn1c(nnc1S)c2csc(n2)c3cccs3 SPB02378 Cn1c(nnc1SCC(=O)NN)Cc2ccsc2 SPB02383 Cc1nc(cs1)c2nnc(o2)SCc3ccc(cc3)Cl SPB02386 c1ccc(cc1)c2cc(on2)c3csc(n3)N/N=C/c4ccccc4Cl SPB04913 Cc1cc(ccc1NC(=O)CC(C)CC(=O)O)Cl S10552 c1cc(cc(c1)S(=O)(=O)N2CN3CN(C2)CN(C3)S(=O)(=O)c4cccc(c4)C(F)(F)F)C(F)(F)F S04172 c1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3Cl)Cl S04202 CCOC(=O)/C(=C/c1ccccc1OC)/C#N S04229 CC(C)(CC(=O)Nc1cc(ccc1Cl)Cl)CC(=O)O S11487 c1cc(ccc1C(=O)NCC(=O)O)Cl S11521 c1cc(ccc1c2csnn2)NC(=O)C3CC3 SEW00785 CCn1cc(c(=O)c2c1ccc(c2)C(F)(F)F)C(=O)N/N=C/c3ccc(cc3)Cl SEW00811 c1cc(ccc1CS(=O)(=O)Cc2nc(no2)c3ccsc3)Cl SEW03702 c1cc(sc1)C(=O)/C(=C/c2ccc(cc2)OCc3nc(no3)c4ccsc4)/C#N SEW03719 c1cc(ccc1/C=N/c2ccc(cc2)c3csnn3)Cl SEW00995 CCOC(=O)c1cnc(nc1N/N=C/c2ccc(cc2)Cl)C(F)(F)F SPB04768 Cc1c(nc(nc1Sc2ccc(cc2)Cl)C(F)(F)F)C SPB04775 COC(=O)c1cnn(c1/C=N/NC(=S)Nc2ccccc2)c3ccc(cc3F)F SPB05143 COC(c1c(cc2c(c(sc2n1)C#N)N)C(=O)OC)OC SPB05167 c1ccc(cc1)c2[nH]c(nn2)Sc3c(cc(cn3)Br)[N+](=O)[O-] SPB07416 c1cc(cc(c1)C(F)(F)F)CN(Cc2cccc(c2)C(F)(F)F)OC(=O)NC3CCC3 CD05730 Cc1cc(c(c(c1)C)Nc2nc(cs2)c3c(onc3c4ccccc4)C)C SPB05023 c1cc(ccc1C#N)C(N2CCSCC2)N3CCSCC3 S11562 c1cc2c(cc1)C(=O)OC2C/C(=N/N=C(\c3ccc(cc3)[N+](=O)[O-])/CC4OC(=O)c5c4cccc5)/c6ccc(cc6)[N+](=O)[O-] S04571 CN(C)C(=S)Nc1ccccc1F S04578 Cc1cccc(c1/C=N/NC(=S)NC)Cl SEW01048 COc1ccc(cc1)c2nc(no2)c3ccc(cc3)c4csnn4 SEW01078 CC(C)(C)c1csc(n1)c2ccc(cc2)c3csnn3 SEW01083 CCOC(=O)c1csc(n1)c2ccc(cc2)c3csnn3 SEW01096 c1ccnc(c1)CNC(=O)NC(=O)c2ccc(cc2)c3csnn3 SEW01151 Cc1nc(cs1)c2nnc(n2CCCOC)SCC(=O)Nc3ccc(cc3)Cl SPB02445 COC(=O)c1cc(c(nc1)Sc2ccccc2NC(=O)Nc3cc(cc(c3)Cl)Cl)[N+](=O)[O-] SPB07480 Cc1ccc(c(c1)Nc2n[nH]c(=S)s2)C S04611 Cc1c2ccccc2nc(c1C#N)Sc3nnc(n3c4cccc(c4)C(F)(F)F)c5ccc(cc5)C(C)(C)C SPB07736 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCC(=O)Nc4ccc(cc4)Cl SPB07875 c1ccc(cc1)COc2ccc(cc2)n3c(=O)[nH]nc3SCc4ccccc4 SPB07876 c1cc(c(c(c1)Cl)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4)Cl SPB07888 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCCOc3ccc(cc3)OC SPB08189 c1cc(ccc1c2nnc(o2)Sc3ncc(s3)[N+](=O)[O-])Cl SPB08198 c1ccnc(c1)S(=O)(=O)Cc2nc(cs2)c3ccc4c(c3)OCCO4 SPB08218 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccccc3Cl SPB08236 CC(C)(C)c1cc(n(n1)C)C(=O)NNC(=O)c2ccc(cc2)C(F)(F)F SPB03168 Cc1cc(no1)NC(=O)c2ccno2 SPB03184 c1cc(ccc1c2nc(on2)C(=O)NN)OC(F)(F)F SPB03238 c1cnoc1NC(=O)N2CCOCC2 SPB03340 CSc1n[nH]c(=O)n1c2ccc3c(c2)OCCO3 SPB07900 c1c(cc(cc1F)F)CC(C(=O)O)N SPB08033 Cc1c2ccccc2sc1C[C@@H](C(=O)O)N SPB08034 Cc1ccc(cc1C)/C=C/2\C(=O)OC(=N2)C SPB08053 COc1ccc(c(c1OC)OC)CN[C@@H](CO)c2ccccc2 SPB08159 Cc1ccc(cc1)S(=O)(=O)NC(=O)NNC(=O)c2cc(nn2Cc3ccc(cc3)F)C(C)(C)C SPB08179 c1cc(ccc1Nc2c3ccc(cc3ncn2)Cl)S(=O)(=O)O RH01822 Cc1cc(no1)C(=O)NCC(=O)OC SPB08427 c1cc(sc1)C(=O)NNC(=O)c2cc(ccc2OCC(F)(F)F)OCC(F)(F)F SPB08434 CC(C)(C)OC(=O)N1Cc2ccccc2C[C@H]1C(=O)NCCN3CCOCC3 SPB08450 CN1CCN(CC1)c2ccc(cc2)NC(=O)Cc3ccccc3 SS00019 Cc1ccc(cc1Cl)C(=O)C(C)Sc2ccc(cc2)Cl XAX00015 CCOc1ccc(cc1)C(=O)/C=C/C(=O)O XAX00029 CCC(=O)Oc1c(cc(c2c1cccc2)O)C XBX00249 C/C(=N\Nc1cc(ccn1)C(F)(F)F)/c2ccc(cc2)Oc3c(cncc3Cl)Cl SPB07114 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)c4ccc(cc4)C(F)(F)F SPB05033 C(=O)(C(F)(F)F)NNC(=O)C(F)(F)F SPB07304 Cc1nc(c(s1)C(=O)O/N=C(/c2cccc(c2)C(F)(F)F)\N)C(F)(F)F SPB07321 Cc1cccc(c1NC(=O)Nc2ccccc2)C(C)C CD06434 c1ccc2c(c1)CCC(O2)NC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F GK01989 CCOC(=O)c1cnn(c1C(F)(F)F)c2nc(cs2)c3ccccc3 SPB07364 CCCc1c(c(nc(n1)SCC(=O)c2ccc(cc2)Cl)OC(=O)N(C)C)C RJF01921 c1cc(c(cc1Br)Cl)NC2=NCCS2 S04199 c1ccc2c(c1)C(=O)OC(S2)c3ccc(cc3)Cl S04248 COc1ccc(cc1)/N=C(/Nc2ccccc2F)\SC.I CD06234 Cc1ccc(cc1)c2nc3c(o2)c4c(n(c3=O)C)n(c(=O)n(c4=O)C)C RJC03112 c1ccc2c(c1)cc(o2)c3csc(n3)c4ccc5c(c4)OCCO5 SCR00139 c1cc2c(c(c1)NC(=O)CC3(CCCCC3)CC(=O)O)non2 SCR00349 c1ccc(c(c1)C(=O)NNC(=O)c2csc(n2)c3c(cc(cn3)C(F)(F)F)Cl)C(F)(F)F SPB05961 Cc1ccc(cc1)c2nc(no2)c3ccc(nc3)OCC(F)(F)F SPB05969 CNC(=S)Nc1ccc(cc1)OCc2c(cc(cn2)C(F)(F)F)Cl SPB05993 CSC(=C(C#N)C#N)/N=C(\C(F)(F)F)/N SPB06022 Cc1c(c(nc(c1C#N)S)C)Cc2c(cccc2Cl)F CD09496 COc1ccc(cc1)C(=O)CCC(=O)c2ccccc2 JFD00235 Cc1c(oc(n1)c2ccccc2)C(=O)O CC18101 CNC(=S)NNC(=O)c1ccc(cc1Cl)Cl SPB06034 c1cc2c(cc1C(=O)CSc3ccc(c(c3)Cl)F)OCCO2 SPB08273 c1cc(c(cc1C(F)(F)F)N)N2CCC(CC2)C(F)(F)F SPB06376 Cc1cc(nc(n1)Sc2ccccc2NC(=O)Nc3cccc(c3)Cl)C(=O)OC SPB06398 c1cc(c(c(c1)CO)F)CO CD10664 Cc1cc(no1)C(=O)NCCN2CCCCC2 SPB08415 CCOC(=O)C1CCN(CC1)Cc2cccc(c2)[N+](=O)[O-] SPB08420 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(=N)c3ccc(cc3)Cl SPB06672 CC(C)N(CCC#N)C(=S)Nc1ccc(cc1)Cl SW00108 c1cc(c(c(c1)Cl)CN2CCC(CC2)NC(=O)c3cccs3)F TB00018 CC(=O)Nc1cccc(c1)C(=O)CCC(=O)O TL00749 Cc1ccc(c(c1)C)C(=O)c2cc(cc(c2)Cl)Cl TL00906 c1ccc(cc1)C(=O)NC(=S)NNc2c(cc(cn2)C(F)(F)F)Cl SPB06943 c1ccnc(c1)C2NN=C(S2)SCC(=O)Nc3cccc(c3)Cl SPB06990 CC1=C(S(=O)(=O)CCO1)C(=O)Nc2ccccc2 XBX00007 Cc1c(nc2ccccc2n1)C XBX00028 c1ccc(cc1)C(=O)CCCCC(=O)O XBX00050 c1c(c[nH]c(=O)c1Cl)Cl XBX00052 c1cc(c(c(c1)Cl)/C(=N/O)/Nc2ccc(cc2)OC(F)(F)F)Cl SPB07163 c1cc(ccc1C(=N)NC(=O)c2cnccc2C(F)(F)F)Cl SPB07188 c1cc(cc(c1)C(F)(F)F)/C(=N/OC(=O)N2CCOCC2)/N SPB07193 Cc1cccc(c1N/N=C(\C)/c2ccc(cc2)Oc3ncc(s3)[N+](=O)[O-])Cl SPB07218 c1cc(ccc1/C=N/Nc2ncc(s2)c3ccc4c(c3)OCCCO4)Cl SPB07376 c1ccnc(c1)SCc2cc(=O)oc3c2ccc(c3)O SPB07385 Cc1ccc(cc1)CN2C(=O)CNC2=S SPB07390 COc1cccc(c1C(=O)Nc2c(cccc2OC)OC)OC CD04270 CCNc1ccc2c3c1cccc3C(=O)N(C2=O)c4ccccc4 BTB11674 C/C(=N\NC(=S)Nc1ccccc1)/c2ccco2 S11089 CC1(CC(=CC(=O)C1)Nc2ccccc2SC)C SPB00811 c1cc(c(nc1)SCC(=O)Nc2ccc(cc2)C(F)(F)F)C(F)(F)F SPB03891 CNc1nnc(s1)Sc2nnc(s2)NC S06805 COc1ccccc1OCc2nc(cs2)c3ccc(cc3)Cl SPB08290 c1cc(ccc1c2c(c[nH]n2)Sc3ccc(cc3)Cl)OC(F)F SPB08303 c1cc(c(cc1F)Cl)SCC(=O)C23CC4CC(C2)CC(C4)C3 SPB08311 Cc1cc(c(c(c1)C)Cn2c(cc(n2)C(C)(C)C)C(=O)Oc3ccc(c(c3)C)Cl)C SPB08331 CS/C(=N\S(=O)(=O)c1ccccc1)/N/N=C/c2ccccn2 CD03030 Cc1nc(c(s1)C(=O)Sc2ccc(cc2)Cl)C(F)(F)F SPB07341 Cn1cccc1CNC(=O)CN2C(=O)c3ccccc3C2=O SCR00953 Cc1nc(cs1)c2nc(cs2)c3ccnc(n3)SCc4ccccc4Cl SPB03668 c1cc(cc(c1)Cl)S(=O)(=O)C[N+](=O)[O-] SPB03576 c1ccc(cc1)c2cc(c(s2)N)C(=O)N/N=C/c3ccncc3 HTS12883 CCOC(=O)c1cc(sc1NC(=O)c2ccc(cc2)[N+](=O)[O-])c3ccccc3 HTS13098 c1ccc2c(c1)c(c(s2)C(=O)Nc3c(cccn3)OCc4ccc(c(c4)Cl)Cl)Cl HTS04547 c1ccc(cc1)C(C2CCC2)(C(=O)O)N JFD00688 COc1cccc(c1O)C(C[N+](=O)[O-])Sc2ccccc2N S13944 c1cc(c(c(c1)Cl)Cl)NC(=N)NC(=N)N RJF01370 CNNC(=O)Cc1ccc(c(c1)OC)OC GK01229 CC1=CC(N=C(N1c2cccc(c2)Cl)SCC(=O)C(C)(C)C)(C)C RJF01410 COc1ccc(c(c1)[N+](=O)[O-])N2C(=O)C=CC2=O S08739 c1cc(ccc1c2cc(on2)c3ccnc(n3)SCC(=O)Nc4cc(cc(c4)Cl)Cl)Cl SPB05083 CSc1nnc(s1)SCC(=O)N2CCC(CC2)C(F)(F)F SPB07224 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2cc(ccc2Cl)C(F)(F)F S06185 c1cc2c(cc1F)/C(=N/N3CCOCC3)/C(=O)N2 SEW05215 c1cc(ccc1OC/C(=N/O)/N)Cl SEW05385 C=CCSc1[nH]c(nn1)c2ccc(cc2)[N+](=O)[O-] SPB00260 COc1c(cc(cc1Br)/C(=N/OC(=O)c2cccnc2SC)/N)Br SPB01649 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3Cl)Br S06528 c1ccc2c(c1)C(=O)N(C2=O)CC(=O)NCc3csc(n3)c4cccs4 SCR00955 CC1(CCc2cc(ccc2O1)S(=O)(=O)NCc3ccc(cc3)S(=O)(=O)N)C SCR01162 COC(=S)Nc1cccc(c1)Cl RH01095 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1F)F)NC(=O)c2cccc(c2)Cl BTB13583 c1ccc(cc1)C(c2ccccc2)N3CCC3 BTB15232 Cc1c(c(c(c(c1C)C)C(=O)c2c(c(c(c(c2Cl)Cl)Cl)Cl)C(=O)NCc3ccco3)C)C CD02144 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)N(C)/N=C/c3c(cccc3Cl)Cl CD06978 c1cc(sc1)c2cc3n(n2)C4=NCCN4C(N3)c5cc(cc(c5O)Cl)Cl CD07326 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NC(=N)N3CCOCC3 CD07769 c1ccc2c(c1)c(c(s2)C(=O)N3CCC(CC3)C(=O)O)Cl HTS08275 c1cc(ccc1CNS(=O)(=O)c2ccc(cc2)C(F)(F)F)N3CCOCC3 HTS09731 CCn1c(nnc1SCC(=O)N)c2c(c3c(cc(nc3o2)c4ccccc4)c5ccco5)N HTS11500 c1ccc(cc1)C(C(=O)O)O JFD03933 CCOC(=O)c1ccc(c(c1)NC(=O)c2cc(c(c(c2)OC)OC)OC)N3CCOCC3 JP00602 Cc1ccc(cc1)c2cncnc2N JM00018 CSc1cccc(c1)NC(=O)C(=O)NCc2ccncc2 JPV00074 c1cc(cc(c1)[N+](=O)[O-])c2c(c(c(c(n2)O)C#N)C(F)(F)F)[N+](=O)[O-] RF00866 CC1(C(=O)N(C(=O)NO1)c2ccccc2)C RF04662 Cc1ccc(cc1C)NC(=S)C2CC(OC(C2)C)C SW00002 c1ccc(c(c1)C(=O)Nc2ccc(cc2)NC(=O)/C=C/C(=O)O)O RDR01423 Cc1ccc(cc1)N/N=C(/C#N)\C(=O)C2CC2 KM02185 CC(C)(C)/N=C(/NCC1CC1)\SC.I RJF01251 Cc1ccc(cc1)S(=O)(=O)Oc2cc(=O)n(c3c2c(=O)n(c(=O)n3C)C)c4ccccc4 RJC01845 Cc1c(c(nc(n1)c2ccccn2)S)Cl RDR03820 c1ccc2c(c1)nc(s2)S/C=C/C(=O)c3ccc(cc3)F NRB04233 Cc1ccc(c(c1)C(=O)C)OC(=O)c2ccc(cc2)Cl NRB02831 CC(=O)N1CCN(CC1)c2cc(nc3c2cccc3)C(F)(F)F KM08929 CCOC(=O)c1cn(nc1N)C NRB02380 Cc1c([nH]c(c1C(=O)C)C)CC(C)C NRB02787 CCN(Cc1ccc(cc1)OC)C(=O)c2cnc(cc2C(F)(F)F)OC RF04338 c1cc(cc(c1)C(F)(F)F)C(=O)NC(=N)c2cccs2 SPB07000 Cc1c(sc(n1)Br)C(=O)O MO00751 c1ccc2c(c1)C(=O)N(C2=O)c3ccccc3N4C(=O)C=CC4=O S05510 c1cc2cn[nH]c2c(c1)[N+](=O)[O-] AC32877 c1ccc2c(c1)nc(s2)c3ccc(cc3)NC(=O)Nc4ccc(cc4)C(F)(F)F SCR00389 Cc1cc(c2ccccc2n1)N3CCN(CC3)CC(C(F)(F)F)O SCR00710 c1cc(c(nc1)N2CCC(CC2)/C(=N/O)/N)[N+](=O)[O-] CD11945 c1cc(cc(c1)OC/C(=N/O)/N)C(F)(F)F SPB02645 CCN(CC)CCNS(=O)(=O)c1c(c(c(c(c1C)C)C)C)C CD06141 CCO.c1ccc(cc1)NC(=O)Nc2cccnc2N3CCC(CC3)C(F)(F)F SPB06552 C1CCCC(CCC1)NC(=O)N XBX00189 Cn1c(cnc1SCC#C)c2ccc(cc2)Cl TG00110 c1cc(sc1)S(=O)(=O)c2cc(ccn2)C(F)(F)F KM05471 c1cc2c(cc1Cl)sc(n2)NS(=O)(=O)CS(=O)(=O)Nc3nc4ccc(cc4s3)Cl BTB06061 c1ccc2c(c1)CCN(C2)C(=O)c3c(c4ccccc4s3)Cl BTB00511 C/C(=N\NC(=O)c1cccc(c1)OC)/c2ccccc2O BTB08530 CC1(Cc2c(c(sc2Br)S(=O)C)C(=O)C1)C KM03781 Cc1c(c(n(n1)Cc2nnc(o2)c3ccccc3Cl)C)Br KM03797 CCOC(=O)c1c(csc1N)c2ccc(cc2)c3ccccc3 AW01211 Cc1ccc(cc1)Sc2c(cccn2)C(=O)N BTB08809 c1ccn2c(c1)c(nc2SCc3c(cccc3Cl)Cl)C(=O)C(F)(F)F BTB05055 c1ccc(cc1)S(=O)(=O)N=C(NNC(=O)c2ccc(cc2)F)NNC(=O)c3ccc(cc3)F CD03208 CC(=NNC(=N)NC(=S)Nc1ccccc1)C RJC00513 CCOC(=O)c1c(noc1C(=O)C)c2ccccc2 SPB06810 CCOC(=O)c1ccc2c(c1)sc(n2)NC=C(C#N)C#N RH00130 CC(C)(CN(Cc1ccccc1)Cc2ccccc2)C(C)(C)O BTBG00228 C/C(=N\O)/c1c(cc(n(c1=O)c2ccccc2)c3ccccc3)O RJC00801 Cc1cc([nH]n1)C(=O)NNC(=S)SC SPB01228 Cc1c(c(n(n1)C)C(=O)O/N=C/c2c(cccc2Cl)F)[N+](=O)[O-] SPB01657 COc1ccc(cc1)c2ccc(s2)C=C(C#N)C#N SEW04649 c1ccc(cc1)N2C(=O)CC(C2=O)Sc3ccc4ccccc4c3 S11231 CCOc1ccc(cc1/C=C\2/C(=O)N(C(=S)S2)CCc3ccc(c(c3)OC)OC)Br S02319 CCCCCc1c(nc(nc1O)c2ccccn2)C RJF01649 Cc1cccc(c1NC(=O)NNC(=O)Cc2csc(n2)c3csc(n3)C)C SPB03508 c1cc(cc(c1)NC(=O)/C(=C\c2cccs2)/c3ccsc3)C(F)(F)F SEW02111 c1ccc(cc1)CN2CCC(CC2)NC(=O)Nc3cc4ccccc4s3 HTS02960 Cc1c(c(no1)c2ccccc2)C(=O)NNc3ccc(cc3)F HTS05016 c1c(cc(c(c1/C=N/NC(=S)NC2CC2)O)Br)Cl BTB04029 c1ccc(cc1)C(=O)CSc2ncccn2 SPB04141 c1ccc(cc1)CCC(=O)NNc2ccc(cc2)Cl HTS05651 Cc1cc(c2cc([nH]c2c1)C(=O)Nc3ccccc3)C HTS06800 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccccc3)C HTS07250 CCOC(=O)c1csc(n1)c2ccc(cc2)Cl BTB06026 c1cc(cc(c1)C(F)(F)F)CSC2=NCCCN2.Cl CD03108 CSc1cccc(c1)NC(=S)Nc2ccccc2SCc3nc(no3)c4ccc(cc4)Cl CD03171 CSc1c2cccn2c3ccccc3n1 CD03386 CC(=O)C(=NNc1ccccc1SCCC#N)C(=O)C CD03684 Cc1c(c(c(c(n1)C)C(=O)OC)c2cc(sc2)S(=O)(=O)NN3CCOCC3)C(=O)OC SEW02160 Cc1ccc(cc1)c2nnc(o2)c3cc(on3)C SPB02792 c1c(csc1[N+](=O)[O-])C(=O)NC(=S)NN2CCCCC2 DFP00154 CNC(=S)NNC(=O)c1ccco1 BTB02369 c1cc(c(c(c1)Cl)C(=O)NC(=O)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-])F BTB05946 c1cc2c(cc1Br)c3cc(cc(c3n2CC(CO)O)Br)Br BTB11866 CC(C)(C)OC(=O)N1CCC(CC1)CNC(=O)c2ccccc2 HTS02025 Cc1cc(nc2c1c3c(o2)C(=O)N(CC(=O)N3)c4cccc(c4)Cl)C HTS13314 c1cc(oc1)c2nnc(o2)SCC(=O)Nc3ccc(cc3)S(=O)(=O)N HTS13510 CCNc1cc(ccc1C)NC(=O)C BTB13391 CN(C)c1ccc(cc1)C2Nc3ccccc3C(=O)N2CCc4ccc(c(c4)OC)OC CD01380 c1cc(oc1)C(=O)NNC(=S)NC2CC3CC2C=C3 CD01406 Cn1cc(nc1)S(=O)(=O)N=S(=O)(C)c2ccc(cc2)Cl KM06789 CSc1c(c(n[nH]1)N)c2ccccn2 PD00175 C[C@@H]1CC2C3CCC4=CC(=O)C=CC4(C3=CCC2([C@]1(C(=O)CO)O)C)C NRB03732 CCN(CC)CCNC1=C(C(=O)c2ccccc2C1=O)Cl BTB13991 COc1ccc(cc1OC)CCNC(=S)Nc2ccc(cc2F)F RJF00148 Cc1c(nc(nc1OC(=S)N(C)C)SCc2c(cccc2Cl)Cl)C RJF00268 Cc1ccc(cc1Cl)C(=N)N.Cl RJF01058 Cc1ccc(cc1C)c2ccc(c(c2)C)C JFD01276 Cc1cc(c(c(c1)C)NC(=O)N)C PHG00001 c1cc(sc1)/C=N/c2ccc(cc2)C(=O)O DSHS00501 c1ccc(c(c1)C(=O)/C(=N/Nc2ccc(c(c2)Cl)Cl)/C#N)OC(F)(F)F KM04873 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2csc3c2cccc3 PD00149 CC(=O)N1CCCC1C(=O)O HTS01510 COc1ccc2c(c1)CCC3C2=NN(C3)Cc4ccccc4 KM07040 Cc1ccc(cc1)c2csc(n2)N SEW05364 Cc1ccc(cc1)Oc2c(cccn2)C(=O)NCC(=O)O BTB08773 CC(=O)N[C@@H](Cc1ccccc1)C(=O)O BTB13559 Cc1c(c(on1)C)c2c(c(no2)C)C(=O)NNC(=O)c3c(cccc3Cl)F SPB02419 c1ccc2c(c1)cccc2c3nnc(o3)c4ccc5c(c4)nsn5 HTS09759 COC(=O)C(Cc1ccc(cc1)O)N BTB06642 c1ccc(cc1)COc2cc(ccc2N)[N+](=O)[O-] BTB13404 c1ccc(cc1)CSc2ccccc2C(=O)N JFD03097 c1cc2c(cc1[N+](=O)[O-])CCN2C(=S)NC3CC4CC3C5C4CC=C5 RH00442 Cc1c(csc1C(=O)NCc2csc3c2cc(cc3)Cl)S(=O)(=O)c4ccc(cc4)Cl HTS04227 COc1ccc(cc1OC)CCNC(=O)c2ccc(c(c2)Cl)Cl MB00250 c1ccc(cc1)C/N=C/c2cccc(c2)Br BTB00694 CC\1=NN(C(=O)/C1=C\c2ccc(cc2)C#N)c3cccc(c3)Cl BTB06323 CCCc1cc(nc(n1)SCC(=O)Nc2ccc(cc2)Br)O BTB06515 CCOC(=O)C(=CNC1CCCCNC1=O)C(=O)OCC BTB06521 COc1ccc(cc1)N2C(=O)C(=O)/C(=C(\N3CCN(CC3)/C(=C\4/C(=O)N(C(=O)C4=O)c5ccc(cc5)OC)/c6ccccc6)/c7ccccc7)/C2=O JFD02993 c1cc(c(cc1S(=O)(=O)NCCCNc2c(cc(cn2)C(F)(F)F)Cl)Cl)N3C(=O)CC4(C3=O)CCCC4 AW01089 Cc1ccccc1c2nc(c(c(n2)SCc3ccccc3)C(=O)C)C SPB05841 Cn1c(nnc1SCC(=O)NNC(=O)Nc2ccc(cc2)Cl)c3ccccc3 HTS07522 Cc1c(ccc(n1)C(F)(F)F)C(=O)OCc2ccc(o2)c3cc(cc(c3)C(F)(F)F)C(F)(F)F HTS03344 Cc1ccc2c(c1)[nH]c(=O)c(c2O)c3ccccc3 NRB01604 Cc1ccc(cc1)S(=O)(=O)Nc2ccccc2c3nc(no3)c4ccc(cc4)Cl BTB03476 CN(C)/C=C/C(=O)c1ccc(s1)Br KM02860 Cc1ccc(cc1Cl)NC(=O)Nc2ccc(cc2)C#N HTS05114 CC(C)(C)c1cc2[nH]c3c(c(=O)n2n1)CN(C3=O)Cc4ccccc4 HTS06825 CN(C)C(=O)NNC(=O)c1c(c(no1)c2c(cccc2Cl)Cl)C(=O)OC RF02177 c1ccc(c(c1)C(=O)Cn2ccccc2=O)Cl RDR01338 CC(=O)Nc1cc2cc(ccc2oc1=O)Cl SPB08012 c1ccc2cc(ccc2c1)c3cc(n4c(n3)cc(n4)c5cccs5)C(F)(F)F KM10593 Cc1ccc(cc1)S(=O)(=O)OCC(CNC2Cc3ccccc3C2)O HTS02900 CC(=O)O[C@@H]1[C@@H]2[C@H](O[C@@H]1C(C#N)OC(=O)C)OC(O2)(C)C NRB04849 CC(C)(C)c1csc(n1)c2ccc(cc2)/C=N/OC(=O)c3cccc(c3)C(F)(F)F KM04383 CCOC(=O)c1cnc2c(cnn2c1N)C#N HTS12584 c1ccc(c(c1)N2C(=O)C=CC2=O)Cl S01401 COc1cc(cc(c1)OC)C2NC(CS2)C(=O)O S12699 CC(C)NC(=O)NNC(=O)C(C)n1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01878 CCOC(=O)Cn1nc(nn1)c2cc(cc(c2)Cl)Cl RJF02003 c1ccc2c(c1)N(C(=O)CS2)CC(=O)N/N=C/c3ccc(cc3)Cl HTS13165 c1ccc(cc1)c2c(c3cccc4c3n(c2=O)CC4)OC(=O)c5cccc(c5)[N+](=O)[O-] HTS12591 CCc1ccc(cc1)n2c(=S)[nH]nn2 S07168 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)c3ccccc3)C HTS07037 c1ccc(cc1)COc2ccc(cc2)/C=N/NC(=O)c3cnn(c3N)c4ccccc4 HTS07444 CCOC(=O)c1cc(c(nc1C(F)(F)F)N2CCN(CC2)C(=O)c3cccc(c3)C(F)(F)F)C#N SPB06800 COC(=O)c1c(nccn1)N SEW03162 CC(C)(C)OC(=O)N1CCN(CC1)C(=O)Nc2ccc(cc2)C(F)(F)F AW01052 c1cc(c(cc1Cl)Cl)Oc2ccc(cn2)N BTB03827 CCCCCCCC(=O)Nc1nnc(s1)Sc2ccnc3c2ccc(c3)Cl RH00421 CC1(Cc2csc(c2C(=O)C1)S(=O)(=O)C)C KM03760 c1cc(ccc1c2[nH]c(nn2)S)C(F)(F)F SPB01423 Cc1c(c(no1)c2ccc(cc2Cl)Cl)C(=O)/C=C/N(C)C SPB05183 c1cc2c(cc[nH]2)cc1NC(=S)NC3CCCC3 RH00911 c1cc(ccc1C(=O)NC(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)c3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl CD05953 C1CC2CCC1C(C2C(=O)O)C(=O)O BTBG00143 Cc1c(c(on1)C)C(=O)Nc2cccc(c2SC)C(F)(F)F SEW03611 c1cc(ccc1c2nc(on2)CNC(=O)Nc3cc(cc(c3)Cl)Cl)C(F)(F)F HTS01223 CCOC(=O)C1CCN(CC1)c2cc(nc3c2cccc3F)C(F)(F)F KM10671 c1ccc(cc1)NC(=O)CSc2nnc(n2c3ccccc3)O HTS07995 c1ccc(c(c1)c2[nH]c3ccccc3n2)Cl BTB06799 c1c(cc(c2c1C(C(=C(O2)N)C#N)C(C#N)C#N)Br)Br FM00108 Cc1cc(c(c(c1)C)N2C(=O)C=CC2=O)C S02803 Cc1ccc(cc1)C(=O)c2c(c3c(s2)nsc3Nc4ccccc4OC)N DP00400 c1cc2c(c(c1)S(=O)(=O)NCc3ccc4c(c3)OCO4)non2 HTS03967 c1cc(ccc1C(=O)NNC(=O)c2csc(n2)c3cnccc3C(F)(F)F)C(F)(F)F SPB05782 c1cc2c(cc1F)c3c([nH]2)CCN(C3)S(=O)(=O)c4cc(c(cc4Cl)Cl)Cl RJC01949 CC(=O)NS(=O)(=O)c1ccccc1 CD09031 CCCCCCSc1ccc2c(c1[N+](=O)[O-])nsn2 KM06787 CC(=O)c1c(c2c(c3c(nc2o1)-c4ccccc4CC3)c5ccco5)N HTS12448 Cc1ccc(cc1)S(=O)(=O)Oc2ccc(cc2Br)C RH01474 c1cc(cnc1)CN2CNC(=NC2)SCc3ccc(cc3)Br.Br ML00417 c1cnccc1c2c(cnc(n2)O)C(=O)O MO00827 Cc1cc(c(cc1Cl)C)S(=O)(=O)Nc2cc(sc2C(=O)C)c3ccccc3 GK03717 Cc1cc(c(c(c1)C)CSCCNC(=O)Nc2ccc(cc2)C(F)(F)F)C SEW06453 Cc1c2ccccc2nc(c1C#N)Sc3ccccc3NS(=O)(=O)c4ccc(cc4)Cl SPB07792 Cc1ccc(c(c1)C)C2=NN(C(C2)c3ccc(cc3)OC)C(=O)C RJC04107 COc1ccc(cc1)n2cnc3c2c(=O)[nH]cn3 SEW01264 c1cc(ccc1NC(=O)c2ccc(c(c2)[N+](=O)[O-])Oc3ccc(cc3)Cl)Cl SPB02953 CN(C)/C=C/C(=O)c1cccs1 S14948 CCOC(=O)c1cc(c(nc1N2CCC(CC2)NC3CCCCC3O)C)C(=O)OC AW00880 COc1ccc(cc1)C(=O)Nc2cccnc2Sc3ccc(cc3)Cl RH02126 COC(=O)Cc1cc(=O)n2c([nH]1)nc(n2)SC HTS00828 CC(C)(C)c1ccc(cc1)c2nc(on2)c3ccc4c(c3)CCO4 HTS02101 c1ccc2c(c1)CC(C2)NC(=O)Nc3c(ccs3)n4cccc4 HTS04255 CCS(=O)(=O)c1ccc(c(c1)NC(=O)c2c(nccn2)C(=O)O)O HTS04065 COc1ccc(cc1OC)CCNC(=O)c2ccc3c(c2)nccn3 HTS09574 CC(C)(C)C(=O)N1CCN(CC1)C(c2ccccc2)c3ccccc3 HTS00651 COc1cccc(c1)C2(CCSc3c2cccc3)O HTS01427 Cc1cc(cc(n1)NN2C(=O)C(=C(C2=O)C)C)C(F)(F)F SCR01519 Cc1c(sc(n1)COc2cccc(c2)Cl)C(=O)/C=C/N(C)C SPB02569 CC(=O)Nc1ccccc1OCC(CN2CCC(CC2)C(=O)N)O HTS03305 Cn1c(nnc1SC)c2ccc(s2)S(=O)(=O)O KM09395 c1ccc(c(c1)OC(F)(F)F)S(=O)(=O)N2CCN(CC2)c3ccnc4c3ccc(c4)Cl KM11092 CCCCCc1ccc(cc1)C(=O)CSc2nccc(n2)c3cccs3 HTS04410 Cc1ccc2nc(cn2c1)c3ccc(c(c3)C)Cl HTS07133 c1ccc(c(c1)N2CCOCC2)N3C(=O)CCC3=O HTS06772 COc1ccc(cc1)NC(=O)N NRB04513 CNC(=S)Sc1ccc(cc1F)F RF03749 COc1ccc(cc1)n2c(nnn2)C/C=N/Nc3ccc(cc3[N+](=O)[O-])[N+](=O)[O-] NRB03180 CCOC(=O)c1ccc(cc1)OC(=O)c2ccc(cc2[N+](=O)[O-])Cl RDR02232 CC(C)(C)OC(=O)C(C)(C)Sc1nc(c(o1)c2ccccc2)c3ccccc3 RH02098 c1cc(ccc1C(F)(F)F)S(=O)(=O)NCc2ccc3c(c2)OCO3 HTS03976 c1cc(cnc1)n2c(noc2=O)c3ccc(cc3Cl)Cl RF05141 c1cc(cnc1)C(=O)C(CC(=O)c2ccc(cc2)Cl)c3ccc4c(c3)OCO4 RG00076 COC(=O)c1ccccc1Sc2nc3ccc(cc3s2)Cl SEW01269 COC(=O)c1c(cc(s1)c2cccs2)NC(=O)CCC(=O)O HTS01038 COc1ccc(cc1)C(=O)CSc2nccc(n2)c3cccs3 HTS04562 Cc1cccc(n1)NC(=O)Nc2cc(cc(c2)C)C HTS07029 CCS(=O)(=O)c1ccc2c(c1)[nH]c(=O)o2 HTS04185 c1cc(ccc1c2cn3c(n2)SCC3)N HTS06799 c1cc(cc(c1)C(F)(F)F)c2nnc(o2)c3ccc(cc3)Cl RJF02156 CS(=O)(=O)NNC(=O)Cn1nc(nn1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F RJF01024 Cc1c(n2ccccc2n1)C(=O)NNS(=O)(=O)c3ccc(s3)CNC(=O)c4ccccc4 HTS05868 c1ccc(c(c1)C#N)S(=O)(=O)Nc2ccc3c(c2)C(=O)OC3 HTS04223 CCOc1ccc(cc1)/C=C(\C#N)/c2cccc(c2)Cl PHG00582 CC(C)(C)c1ccc(cc1)OC(=O)c2ccc(cc2)Cl RDR01854 CCOC(=O)c1ccc(cc1)NC(=S)Nc2c(cccn2)C RB00092 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)C(F)(F)F SEW04324 c1ccc(c(c1)C(=O)N/N=C(/c2cnccn2)\N)Cl SPB07145 Cc1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(c(c3)OC)OC HTS13684 c1ccc(cc1)C(c2ccccc2)NS(=O)(=O)c3cccc4c3nccc4 HTS13685 c1ccc(cc1)S(=O)(=O)/N=C(\N/N=C/c2ccccc2O)/N3CCCC3 CD03651 Cc1c(c(n(n1)c2ccccc2)NC(=O)C(Cl)Cl)Br KM00151 c1ccc2c(c1)c(cn2Cc3cc(cc(c3)F)F)/C=C/C(=O)O RH02013 CC(=O)N1CCc2c1ccc(c2)S(=O)(=O)Nc3ccc(cc3)Cl KM05518 Cc1ccc(cc1)C(=O)Nc2cccc(c2)c3[nH]c4ccccc4n3 HTS00911 Cc1c(c(on1)C)C(=O)N2CCc3c(ccs3)C2c4ccc(cc4)C(F)(F)F SEW01207 Cc1c2ccccc2n3c1/C(=N\OC(=O)c4ccc(cc4Cl)Cl)/CC3 SEW02358 CSc1nnc(s1)/N=C/c2c3ccccc3ccc2O S15035 c1cc(cc(c1)NS(=O)(=O)c2ccc(cc2)N)C(F)(F)F RJF00766 c1cc(ccc1COc2ccc(cc2)c3nnco3)F SEW04807 CC(=O)Oc1ccc(cc1)NNc2ccccc2 XBX00146 c1c(cnc(c1Cl)S)C(F)(F)F SPB03806 Cc1cc(no1)C(=O)O/N=C(/c2c(onc2c3c(cccc3Cl)Cl)C)\N SPB06685 c1cc(c(c(c1)Cl)/C=N/NC(=O)c2cccn2c3ccc(cc3)F)F SEW04778 Cc1cc(n(n1)C)c2nc(no2)c3ccc(cc3)C(F)(F)F SPB01995 c1ccc2c(c1)c(nc3n2nnc3C(=O)NCc4ccncc4)N CD05126 CCOC(=O)C1CC(=O)C(CC1=O)C(=O)OCC BTB12681 c1cc(cc(c1)[N+](=O)[O-])C(=O)CSc2c(c(sn2)SCC(=O)c3cccc(c3)[N+](=O)[O-])C#N CD00482 COc1cccc(c1)c2nc(c(o2)N)C#N SEW05774 CCOC(=O)c1cc(=O)oc2c1ccc(c2)O BTB14939 C1C2CC3(CC1(CC(C2)(C3)Br)CC(=O)O)Br BTB14994 CCO/C=C\1/C(=O)N(C(=S)S1)CCc2ccccc2 S03087 Cc1cc(cc2c1nc[nH]2)Br MO07408 Cc1nc(cs1)c2nc(on2)C(=O)NNC(=O)Nc3cccc(c3)C(F)(F)F SPB02737 CC(=O)c1cc(no1)c2ccc(cc2)Cl SPB05654 Cc1c(c(nn1C)C(=O)Sc2ccc(cc2F)F)[N+](=O)[O-] SPB03816 c1ccc(c(c1)CN/C(=C(/C#N)\NCc2c(cccc2Cl)F)/C#N)Cl KM00430 Cc1c(cn(n1)c2ccccc2)/C=N/NC(=O)Cn3c(=O)n-4c(n3)CSc5c4cccc5 HTS13113 c1ccc(cc1)C(=O)n2ccc3c2cccc3 RJC03790 Cc1c(c(c(c(c1C)C)CSC(=N)N)C)C.Cl JFD04020 Cc1c(n(c(c1C#N)NC(=O)c2ccc(cc2)C(F)(F)F)CC3CC3)C SPB01910 Cc1c(c(no1)c2ccccc2)CNC(=O)c3ccccc3 SCR00044 CCOC(=O)C1=C(NC(=C(C1c2ccccc2)C(=O)OCC)C)C BTB14326 c1c(cncc1Br)CC(=O)O BTB14052 c1cc2c(cc[nH]2)c(c1)N3CCN(CC3)C(=O)c4ccc(cc4)[N+](=O)[O-] BTB14537 CCSc1c(cccn1)C(=O)N[C@@H](CCSC)C(=O)OC KM01823 Cc1ccc(cc1)S/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM00537 c1cc(ccc1C(=O)/C(=C/Nc2ccc(c(c2)Cl)Cl)/C#N)OC(F)(F)F KM04870 CSc1c2c(c(s1)c3ccnc(n3)SCc4c(cccc4Cl)Cl)CCCC2=O KM03937 COC(=O)c1c(ccs1)N/C=C(\C#N)/C(=O)c2cccc(c2)CSc3ccc(cc3)Cl KM05727 c1ccc(c(c1)C(=O)N2CCC(CC2)n3cccc3)Cl KM08580 c1cc(c(cc1S(=O)(=O)c2ccc(c(c2)Cl)Cl)Cl)Cl TL00145 CSc1c(c(c2c(n1)CCCC2)c3cccs3)C#N SPB07039 CCOC(=O)c1cc(c(nc1C(F)(F)F)Oc2cc(cc(c2)Cl)Cl)C#N SPB06476 Cc1csc2c1ncnc2S GK02666 Cn1cc(c(=O)n(c1=O)Cc2ccccc2)/C(=N/OC(=O)c3ccc(cc3)Cl)/N KM07753 COc1ccc(cc1OC)CC2c3cc(c(cc3CCN2C(=S)Nc4cccc(c4)C(F)(F)F)OC)OC BTB00971 Cc1c(c(no1)c2ccccc2Cl)C(=O)N=S(=O)(C)c3ccc(cc3)Cl KM02810 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)NCCc1ccc(cc1)OC BTB14243 CCCCCCC#Cc1cc(cnc1)c2nnc(n2C)SCc3ccccc3 KM09567 c1ccc2c(c1)OCC(O2)c3nc(cs3)C(=O)SCc4cccs4 KM06806 c1ccc(cc1)C(c2ccccc2)N3CC(C3)SCC(=O)NNC(=O)c4ccccc4 KM09095 c1cc(ccc1C2=NCCS2)OC/C(=N/O)/N SPB02435 COc1ccc(cc1OC2CCCC2)c3nc(on3)c4cccc(c4)C(F)(F)F KM09632 CCn1c(nnc1SCC(=O)Nc2nnc(s2)c3cccs3)c4cccs4 HTS13289 CCOc1ccc(c(c1)SCC(=O)O)C(=O)N XBX00168 CCOC(=O)c1cc(cnc1)C(=O)OCC JFD03996 c1cc2c(c(c1)S(=O)(=O)N3CCN(CC3)c4ccc(cc4)C#N)non2 HTS01295 CC(C)(C)c1cc(n(n1)Cc2ccc(cc2)F)C(=O)Nc3ccc(cc3)F HTS00913 Cc1cc(no1)n2cnc(n2)CC(=O)C CD09221 Cc1ccc(c(c1)[N+](=O)[O-])OCC2N(CCS2)C(=O)c3ccc(cc3)F FM00278 Cc1cc(n(n1)c2ccccc2)NC(=O)C(Cl)Cl KM00148 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3cccc4c3non4 SCR00069 COc1ccc(cc1)S(=O)(=O)N=S(=O)(C)c2ccc(cn2)C(F)(F)F KM05609 CSc1nc2ccc(cc2s1)[N+](=O)[O-] KM06788 CCOC(=O)Cc1cc(=O)n2c([nH]1)cc(n2)c3cccs3 KM09495 CC1CN(CC(O1)C)c2ccc(cc2C(=O)O)NS(=O)(=O)c3ccccc3 CD06976 Cn1cc(nc1)S(=O)(=O)N TL01003 CC(C)(C)OC(=O)N1CCC(=O)CC1 JFD01627 Cc1ccc(cc1)Sc2ccc(cn2)N BTB07163 COc1cccc(c1)c2cn3c(n2)sc(n3)c4cccs4 HTS13373 CC(C)(C)c1cc2nc(cc(n2n1)C(F)(F)F)c3ccc(cc3)Cl KM10404 c1cc(cc(c1)Cl)N2C(=O)CSC2=S S02963 CC1C(C1(Cl)Cl)(c2ccccc2)c3ccccc3 RJC03718 Cc1cccc(c1C)NC(=O)c2c(cccc2OC)OC RDR02727 CCOC(=O)Cc1csc(n1)NC(=O)CSc2ccc(cc2)Cl RJC02513 c1ccc(c(c1)CNC(=O)COc2ccccc2OC(=O)c3ccc(cc3)Cl)Cl RDR03035 COc1ccc(cc1OC)CCNS(=O)(=O)c2ccc(cc2)C#N RJC03060 CCC1(CC(=O)N(C(=O)C1)c2ccc(cc2)Cl)C S10925 CC(C)(C)c1ccc(cc1)c2nnc(s2)NC(=O)C(Cl)Cl SPB00177 c1ccc(cc1)NC(=O)N/N=C(/c2cnccn2)\N SPB07264 c1ccc(cc1)n2c(nnc2SCc3c(cc(cn3)C(F)(F)F)Cl)O SPB06210 CC(C)c1ccc(cc1)NNS(=O)(=O)c2ccc(c(c2)Cl)Cl SPB00464 c1cc(ccc1C(=O)/C=C/Sc2ccc(cc2)Cl)F BTB11773 c1cc(c(c(c1)F)C#N)NCCCn2ccnc2 CD07436 c1ccc2c(c1)C(CS2(=O)=O)N3CCCC3 KM08196 c1cc(ccc1N/C=C(\C#N)/C(=O)C2CC2)OC(F)(F)F KM03618 CCCCc1c(c2ccccc2oc1=O)O NRB02296 C/C(=N\NC(=O)c1cccnc1)/c2cccnc2 BW00100 Cc1c(cc(n1c2ccccc2)c3ccccc3)C(=O)Nc4cccc(c4)OC SP00342 CCOC(=O)Cc1c(cnc(n1)N)C(=O)OCC CD11442 CN(C)c1ccc(cc1)n2c(nnn2)SCC(=O)c3cc4ccccc4o3 HTS00789 c1ccc(cc1)OCC(CN2CCN(CC2)c3ccc(cn3)C(F)(F)F)O HTS00939 Cc1cc(c(cc1Cl)C)SCc2ccc(cc2Cl)[N+](=O)[O-] SPB01543 CC(C)(C)c1ccc(cc1)NC(=O)Nc2cccc(c2)S(=O)(=O)N HTS05225 Cc1ccc2nc(cn2c1)c3ccc(cc3)C(F)(F)F HTS07693 c1cc(cc(c1)[N+](=O)[O-])c2nnn(n2)Cc3ccc(cc3)Cl RJF01437 Cc1ccc2c(c1)c(=O)n(c(=S)[nH]2)c3ccc(cc3)S(=O)(=O)N4CCCCC4 S07903 CCOC(=O)C/C(=N/Nc1ccc(cc1)[N+](=O)[O-])/C(F)(F)F S15542 c1ccc(cc1)C(=O)Nc2ccn(c(=O)n2)[C@H]3CC[C@H](O3)CO BTB14104 c1cc2c(nc1)n3ccsc3nc2=S BTB08465 c1cc(ccc1C2CCCCC2)C3CCCCC3 BTB11188 CCCOc1ccc(cc1)C(=O)CCC(=O)O BTB10246 Cn1c(cnc1S(=O)CC#N)C(=O)OC KM06248 CC(=O)Nc1ccccc1OCCN(Cc2ccccc2)C(=S)NCCC3=CCCCC3 S14201 CC1=C(C(C(=C(N1)C)C(=O)OC)c2cc(ccc2OC)OC)C(=O)OC JFD03299 c1c(csc1[N+](=O)[O-])C(=O)NC(=O)NN2CCCCCC2 DFP00188 c1cc(ccc1C(=O)c2cc3cc(cc(c3o2)Cl)Cl)Br RH01782 COC(=O)c1cc(ccc1N2CCOCC2)NC(=O)c3cc(oc3C(F)(F)F)c4ccc(cc4)Cl HTS01355 CNC(=S)N(Cc1cccc(c1Cl)Cl)Cc2cccs2 RF03353 c1ccc(cc1)CN2CCN(CC2)CCCNS(=O)(=O)c3ccc(cc3)N4C(=O)CCC4=O AW01220 c1cc(c(c(c1)Cl)CN2CCN(CC2)CCCNC(=O)c3cn4cc(cc(c4n3)Cl)C(F)(F)F)F AW01206 c1ccc(cc1)C(CC(=O)NCC(c2ccccc2)O)CC(=O)O HTS05975 COC(=O)[C@H](Cc1ccc(cc1)O)NC(=O)c2ccc(cc2)Cl RJC02520 c1ccc(cc1)c2ccc(cc2)/C=C\3/C(=O)OC(=N3)c4ccccc4 S01295 CN(c1ccc(cn1)[N+](=O)[O-])NC(=O)c2ccccc2F CD07305 COc1cccc(c1CO)OC CD04716 Cc1c(nnn1c2cc(ccc2Cl)Cl)C(=O)C CD10569 COC(=O)c1c(c(c(s1)SC)C#N)c2cccc(c2)Cl KM02571 Cc1ccc(cc1)c2c(cno2)c3nnnn3c4ccccc4 JFD03659 CCOC(=O)c1ccc(c(c1)/N=C/c2cc(cc(c2O)Cl)Cl)NC3CCCCC3 SJC00249 COc1ccc(cc1)Cn2c(=O)c3c(nc[nH]3)n(c2=O)c4ccccc4C(F)(F)F KM10602 COC(=O)/C(=C/c1ccc(c(c1)Cl)Cl)/C#N S07697 c1cc(ccc1NC(=S)N(CCO)N)OC(F)(F)F S15294 c1ccc(cc1)c2nccc(n2)c3c(=O)ccn(n3)c4ccc(cc4)Cl SPB04433 c1ccc(cc1)C#Cc2cc(sc2)/C=N/Nc3ccccc3 KM08131 c1ccc2c(c1)c(c(s2)C(=O)NNC(=O)CSc3ccccc3[N+](=O)[O-])Cl DSHS00866 CC(C)(C)c1ccc(cc1)C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-] S14128 COc1cc(ccc1O)C(=O)c2cc(ccc2N)Cl RH01504 CS/C(=N\S(=O)(=O)c1ccccc1)/N2CCCCC2 CD03051 Cc1ccc(cc1)NC(=O)c2cc(n(c2C)CCCN3CCOCC3)c4ccccc4 SP00485 c1cc(c(cc1F)F)c2ccc(o2)/C=C/C(=O)O CD06617 c1cc(ccc1CC(=S)N)[N+](=O)[O-] DP01591 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F RDR00558 c1ccc(cc1)CN(Cc2ccccc2)C(=O)c3ccc(o3)Br JFD03981 Cn1c2c(cn1)c(ncn2)NNC(=S)Nc3ccc(cc3F)F GK03514 Cc1c(cc(o1)c2ccccc2)C(=O)NC3CCN(CC3)Cc4ccccc4 SP01189 CCCCCCCN/C(=C/1\C(=O)C(=O)N(C1=O)c2ccccc2)/c3ccccc3 RJC02213 Cc1nc(cs1)CSc2[nH]c(nn2)C(F)(F)F SPB02175 Cc1c(sc(n1)c2ccc3c(c2)CCO3)C(=O)Nc4cccc(c4)[N+](=O)[O-] SP00246 c1ccc(cc1)/C(=N/OC(=O)c2cccc(c2)Cn3cc(ccc3=O)C(F)(F)F)/N SPB06703 c1ccc(cc1)c2c[nH]cn2 SEW05612 c1ccnc(c1)CCNc2ccc(cn2)[N+](=O)[O-] CD06607 c1cc(ccc1C(=O)/C(=N/Nc2ccc(c(c2)Cl)Cl)/C#N)OC(F)(F)F KM04937 c1cc(ccc1NC(=O)CC#N)Br DP00459 CC(c1n[nH]c(=S)n1c2ccccc2)Oc3ccc(cc3Cl)Cl JFD03197 COC(=O)c1csc2c1nc(cc2C(F)(F)F)N3CCN(CC3)C(=O)c4ccco4 GK03759 c1ccc(cc1)N2CCN(CC2)C(=O)CSc3ccc(cc3)F HTS01204 Cc1ccc(cc1)NC(=O)c2cc(nn2Cc3ccc(cc3Cl)Cl)C(C)(C)C SPB08248 c1cc(c(cc1Br)/C=N/Cc2ccncc2)O S04181 c1cc(c(cc1F)NC(=O)/C=C/C(=O)O)F S03892 CC(C)(C)c1ccc(cc1)N2C(=O)CC(C2=O)CC=C S15212 CCOC(=O)c1cnc(nc1Sc2ccc(cc2)Cl)c3cccs3 SPB05903 Cc1c2c(c(sc2nc(c1/N=N/c3cc(cc(c3)Cl)Cl)C)C(=O)c4ccccc4)N SPB06749 Cn1ccnc1SCC(=O)c2ccc(c(c2)F)F BTB08487 Cc1ccc(cc1)c2nc(no2)c3cc(on3)C SPB04225 c1cc(ccc1/C(=C/c2ccncc2)/C#N)NC(=S)NC3CC4CC3C=C4 CD01848 c1ccc(cc1)c2cc(=O)c3cc(ccc3s2)Cl KM02030 c1cc2c(c(c1)S(=O)(=O)NCC(=O)N/N=C/c3ccc(cc3)Cl)nsn2 KM06431 c1ccc(cc1)NC(=O)CSCC(=O)NNC(=O)Nc2ccc(cc2)Cl KM08990 c1cc(c(cc1F)F)N2C(=O)CS(=O)(=O)CC2=O S10822 CN(C)c1c(cc(cn1)NC(=O)OCC#C)C(F)(F)F RF05256 c1cc(oc1)CNC(=O)CC(CC(=O)O)c2ccc(cc2)C(F)(F)F PD00529 c1cc(sc1)c2cc(nn2c3ccc(cc3)NS(=O)(=O)c4ccc(cc4)Cl)C(F)(F)F HTS04038 Cc1ccc(cc1)OC(=O)c2cc(nn2C(C)(C)C)C SPB03142 c1cc(cc(c1)NC(=S)NNC(=O)c2ccc(cc2)OC(F)(F)F)C(F)(F)F SPB03813 Cc1ccc(cc1)Cn2c(cc(c(c2=O)C#N)C)C SPB06577 COc1ccc(cc1)Oc2ccc(cn2)NC(=O)Nc3ccc(cc3)SC(F)(F)F BTB08362 c1cc(ncc1N)N2CCOCC2 CD04400 c1cc(ccc1C(=S)N2CCCCC2)Cl BTB10176 Cc1cc(cc(c1OCC(=O)NN)C)c2c3ccccc3c(=O)n(n2)C BTB08293 Cc1c(c(on1)C)C(=O)Nc2ccc(cc2)OC SEW05826 c1ccc(c(c1)CCOC(=O)c2ccc(cc2)F)/C=C\[N+](=O)[O-] RH01881 c1cc(ccc1C(F)(F)F)S(=O)(=O)CC(=S)N SPB02572 Cc1c(c(no1)c2c(cccc2Cl)Cl)c3csc(n3)c4ccccc4Cl SPB08287 Cc1cc(c(cc1Cl)C)S(=O)(=O)Cc2nc(on2)c3c(noc3C)C SEW00848 c1ccc2c(c1)C(OC2=O)CC(=O)c3ccc(cc3)Cl S04715 CS(=O)(=O)/C(=C/c1ccc(s1)c2cccs2)/C#N SEW02157 CC(C)(C)c1ccc(cc1)C(=O)O/N=C(/Cn2nc(nn2)N3CCCCC3)\c4ccc(cc4)Cl RJF00382 CC(C)(C)c1nccc(n1)c2c(=O)ccn(n2)c3ccc(cc3)F SPB04026 CC(C)(C)COS(=O)(=O)c1ccc(cc1)Br BTB12751 CCOC(=O)C(CCC(=O)O)(CCC(=O)O)C(=O)OCC BTBG00018 Cc1ccc(cc1)S(=O)(=O)N(C)CCCC#N BTBG00169 COc1ccc(cc1)CCC(=O)CCc2ccc(cc2)OC BTB09976 C1CCC2CC[C@H](C[C@@H]2C1)O BTBG00239 C1CC1C(=O)C(=C2SCCS2)C#N KM00866 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccccc3C(=O)NNc4ccc(c(c4)Cl)Cl BTB04940 c1cc(c(cc1)O)/C=N/CC/N=C/c2c(cccc2)O JFD03654 COc1ccc(cc1)Oc2cccc(c2CNC(=O)c3ccccc3)Cl CD11662 c1cc(c(cc1Cl)NC(=O)CC2C(=O)NCCCN2)Cl HTS00381 c1ccc(cc1)C(=O)NC(=S)NCC2CC2 GK03536 c1cc(ccc1CO)N2CCOCC2 CC17409 COc1ccc(cc1)OCCC#N SEW04595 CCOC(=O)c1c(sc(n1)c2ccccc2)c3ccnn3C(=O)NC(C)C SPB04634 c1ccc(cc1)CNS(=O)(=O)c2cc(c(s2)Br)Br SEW03594 c1ccc(cc1)C(=O)C2CCNCC2.Cl SEW04290 COC(Cn1c(nnc1SCC=C)c2ccc(cc2)Cl)OC SPB04891 c1ccc(cc1)CSc2n[nH]c(=O)n2C3CC4CC3C=C4 SPB07725 Cc1c(c(c(c(c1C)C)CSCC(=O)NNC(=S)NC2CC3CC2C=C3)C)C CD01700 CS(=O)(=O)c1c2c(c(s1)NC(=O)Nc3ccc(cc3)Cl)CCC=C2 KM04641 Cc1c(c(sc1C(=O)OC)SC)c2ccn(n2)S(=O)(=O)c3ccc(cc3)Cl KM02105 Cc1c(c(no1)c2ccccc2)C(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl SEW05978 CC(C)(C)c1ccc(cc1)C(=O)Nc2nc3ccsc3c(=O)s2 HTS01339 COc1ccc(cc1)C2c3ccsc3CCN2C(=O)c4ccc(cc4F)F SEW06421 c1ccc(cc1)CNC(=S)NNC(=O)c2cnn(c2N)c3ccccc3 HTS07438 CCOC(=O)CNc1ccc(cc1)OC(F)(F)F S14310 CCCc1c(c(nc(n1)SCc2ccc(cc2)F)OC(=O)N(C)C)CC=C RJF01612 Cc1ccc(n1c2ccc(cc2)C(F)(F)F)C SEW00970 c1ccc(cc1)NC(=O)O/N=C/c2ccc(c(c2)Cl)F SEW00878 Cn1c(nnc1Sc2ncc(s2)[N+](=O)[O-])O SPB01624 c1ccc(cc1)Cn2c(nnc2SCc3csc(n3)c4cccs4)O SPB02579 c1cc(ccc1C(=O)Nc2ccc(cc2)Oc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl SEW05457 c1ccc2c(c1)n(c(=O)o2)CCC(=O)Sc3ccc(cc3Cl)Cl SPB02720 Cc1c(cc(c(n1)SCCNC(=O)c2ccc(cc2)F)C#N)c3csc(n3)C BTB09489 c1cc(c(cc1F)C(F)(F)F)NN=C(C#N)C#N SEW06224 CC(C)(C)C(C)(C#N)Nc1ccc(cc1)Cl RJC03586 COc1c(cc(c(c1C(=O)NC(=O)Nc2c(cc(cc2Cl)[N+](=O)[O-])Cl)OC)Br)Cl BTB07755 COC(=O)CSc1c2c3c(sc2ncn1)CCCC3 GK03212 c1cc(ccc1C#N)NC(=O)COCC(=O)O HTS05121 CC(C)(C)c1ccc(cc1)c2nnc(o2)c3ccccc3NC(=O)/C=C\C(=O)O BTB06967 c1cc(sc1)CNC(=O)/C=C/C(=O)NCc2cccs2 CD07696 CCOC(=O)c1cc(on1)c2csc(n2)c3ccc(cc3)C(C)(C)C SPB04497 CCOC(=O)/C(=C\c1ccc(s1)Cl)/C#N SEW03828 CCOC(=O)c1c(nc(s1)COc2cccc(c2)Cl)C SPB01812 CC(C)NC(=O)n1c(c(cn1)S(=O)(=O)c2ccc(cc2)Cl)c3ccc(cc3)Cl SPB05385 Cc1c(c(no1)c2ccccc2Cl)C(=O)Nc3cccc(c3)C(F)(F)F DSHS01252 c1ccc(cc1)NC(=O)O/N=C/2\CCSC2 CD10147 CC(=O)N[C@@H](Cc1ccc(cc1)OC(F)(F)F)C(=O)O SPB08025 Cc1c(c(no1)c2ccccc2)c3ccnc(n3)N(C(=O)C)C(=O)C SPB05239 c1ccc(cc1)C(=O)NC(=O)N2CCc3c4ccccc4[nH]c3C2C(F)(F)F SEW06186 CCOC(=O)c1cc(n(c1C)c2ccc(cc2)c3csnn3)C SP01244 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NCc3ccc4c(c3)CCO4 SP01304 Cc1cscc1NC(=O)/C=C(\C)/C(=O)O GK02477 c1ccc(c(c1)NC(=O)/C=C\C(=O)O)Sc2nccc(n2)C(F)(F)F HAN00312 Cc1ccc(cc1)CSc2nnc(s2)N XAX00074 CSc1c(c(c(s1)c2ccno2)c3ccco3)C#N KM05475 c1cc(oc1)CN(CCC(=O)Oc2ccc(cc2)Cl)S(=O)(=O)c3ccc(cc3)Cl KM09550 COc1ccc(cc1)CSc2n[nH]c(=O)n2c3ccc4c(c3)OCCO4 SPB07889 Cc1ccc(cc1)S(=O)(=O)NNC(=O)Cn2cccc(c2=O)OC KM07199 CC(C)NC(=O)N1CCCN(CC1)c2nc3ccc(cc3s2)Cl SPB07929 CNC(=S)N(Cc1cccnc1)Cc2ccc(cc2Cl)Cl RF03483 c1cc(sc1)c2cc(n[nH]2)C(F)(F)F CD04898 CN(c1ccccc1Cl)C(=O)c2cc3cc(ccc3[nH]2)OC SP01200 CCCCc1[nH]cc(n1)CO SB02033 c1cc(oc1)CNC(=O)c2ccc3c(c2)nns3 KM10662 COC(=O)c1cc(c(s1)C(F)(F)F)c2ccc(cc2)S(=O)(=O)N3CCCCC3 HTS03242 Cc1cc(no1)C(=O)N2CCC3(CC2)OCCO3 HTS06997 COc1ccc(c(c1OC)OC)/C=C/2\Cc3cc(c(c(c3C2=O)OC)OC)OC SEW04092 CC(=O)O/N=C(/COc1ccc(cc1)c2nnco2)\N SEW04639 CC(C)(C)c1ccc(cc1)c2nnc(n2CCCOC)SCc3c(cccc3Cl)F SPB00457 c1cc(ccc1C#N)OS(=O)(=O)c2ccc(cc2)C#N CD10703 Cc1c(nnn1c2cccc(c2Cl)Cl)C(=O)/C=C/N(C)C CD09925 c1ccc(c(c1)c2nc(no2)c3ccc4c(c3)non4)Cl KM06764 c1cc(oc1)CN(CCC#N)S(=O)(=O)c2ccc(cc2)Cl KM09444 c1ccc(cc1)Cn2c(nnn2)c3ccc(cc3)[N+](=O)[O-] GK02980 CC(C)Cc1ccc(cc1)C(C)c2nc(no2)c3ccc(cc3)OC(F)(F)F SEW06260 CCCOc1ccccc1/C=N/NC(=S)Nc2ccc(cc2C)Br RDR01210 COc1ccc(cc1)S(=O)(=O)NNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl HTS00411 CCN1CN(C(=S)SC1)CC S01972 CC1(CCCCCCCCCCC1)O RJC03263 CC(=O)c1ccccc1NC(=O)/C=C\C(=O)O S04240 COc1cccc(c1)C2C(=Cc3cc(ccc3O2)Cl)[N+](=O)[O-] S14115 c1cc(c(nc1)Sc2ccc(cc2)Cl)C(=O)O BTB08734 CCOC(=O)c1c(c(c(=N)n(n1)c2ccccc2)C#N)C BTB09057 COC(=O)c1c(ccs1)NC(=O)C(F)(F)F CD08692 Cc1cccc(c1)NC(=S)NCc2ccncc2 DSHS01215 c1ccc(cc1)c2ccc(cc2)c3csc(n3)CS(=O)(=O)Cc4ccco4 KM03222 CCOC(=O)C1CCN(CC1)C(=S)Nc2ccc(cc2C)Br RH01382 c1ccc(cc1)C(=O)N2CCOCC2 SEW04620 CC(C)(C)c1ccc(cc1)c2cc3c(s2)c(ncn3)Nc4cccc(c4)Cl GK03741 CCOC(=O)c1cc(on1)C(=O)/C=C/N(C)C SPB04620 COCCCn1c(=O)c2ccc(cc2nc1S)Cl RDR01291 CC(C)(C)OC(=O)NCc1nnc(n1Cc2ccccc2)S KM10517 Cc1cc(=O)oc2c1ccc(c2)NS(=O)(=O)c3ccc4c(c3)CCO4 HTS06547 CC(C)(CC(=O)Nc1ccc(cc1)CC#N)CC(=O)O HTS04726 c1ccc(cc1)C(=O)C2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F SEW04342 c1ccc(cc1)C(=O)NC(=S)Nc2ccccc2Oc3ccc(cc3Cl)Cl S09526 c1cc(cc(c1)NC(=O)NC(=O)c2ccc(nc2)Oc3ccc(cc3)Cl)C(F)(F)F SPB06255 c1cc(c(nc1)Sc2[nH]c(nn2)c3ccc(cc3)Cl)[N+](=O)[O-] SPB00511 CCOC(=O)c1cc(ccc1Oc2cc(cnc2)Cl)NC(=O)Nc3cccc(c3)Cl BTB07890 c1ccc(c(c1)C(=O)NCC2CC2)NC(=O)NC(=O)c3c(cccc3Cl)Cl BTB05907 c1ccc(cc1)c2coc3cc(ccc3c2=O)OS(=O)(=O)c4ccc(cc4)Br JFD02648 CCOC(=O)c1c(n(c(c1S(=O)(=O)Nc2ccccc2)c3ccccc3)c4ccccc4)C SP01124 CC(=O)Nc1ccc(cc1N)C(F)(F)F BTB00739 CC(C)(C)OC(=O)/C(=C/c1ccc(cc1Cl)Cl)/C#N S10886 Cc1ccc(cc1)S(=O)(=O)NNC(=S)Nc2ccc(cc2)F RDR00474 c1cc(ccc1C(F)(F)F)/N=N/c2ccc3c(c2)CCCN3CCC#N JFD03372 Cn1c2ccccc2c(n1)NC(=O)COCC(=O)O HTS00768 c1cc(c(nc1)S)C(=O)O SB00659 CC(C)(C)c1ccc(cc1)NC(=O)CC(CC(=O)O)c2ccc(cc2Cl)Cl S08563 Cc1ccc(cc1)NC(=O)CC(CC(=O)O)c2cc(c(c(c2)OC)OC)OC S08598 CN(C)/C=C(\C#N)/C(=O)Nc1ccc(c(c1)Cl)F CD08646 c1ccc(cc1)C(C(=O)c2ccccc2)OC(=O)CCC(=O)O MO07610 CCOc1ccc(cc1/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])Br PHG00095 Cc1ccc(n1CCSCc2c(cc(cc2C)C)C)C SEW06535 c1ccc(c(c1)C(=O)N(Cc2ccccn2)Cc3ccccn3)C(=O)O HTS00606 c1ccc(cc1)/C(=N\O)/c2ccc(cc2)Cl CD02102 CCOC(=O)c1c(c2c(cc(nc2o1)c3ccccc3)C)NC(=O)Nc4ccc(cc4)Cl HTS07544 Cc1c(c(no1)c2ccccc2)CNS(=O)(=O)c3ccc(cc3OC)OC SCR00077 c1ccc(cc1)CN2CCN(CC2)Cc3ccc4c(c3)cco4 HTS13962 CC[C@@]12CCCN3[C@@H]1c4c(c5ccccc5n4C(=O)C2)CC3 HTS13967 Cc1c(c(c(c(c1C)C)CS/C(=C(/C#N)\C(=O)Nc2cccc(c2)C(F)(F)F)/Nc3ccccc3Cl)C)C CD01673 CC(C)(C)c1cc(c(s1)C(=O)OC)N GK00671 CC(C)(C)c1ccc(cc1)/C(=N/OC(=O)c2c(ccs2)Cl)/N GK01357 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)Nc3ccc(cc3)F HTS01375 Cc1c(sc(n1)c2ccc3c(c2)OCC3)C(=O)Nc4ccc5c(c4)OCCO5 HTS03215 Cc1ccc(cc1)S(=O)(=O)n2c(c(c(n2)C)/N=N/c3ccc(cc3)Cl)C BTB00946 c1cc(c(c(c1)Cl)CSC2=NCN(CN2)Cc3c(cccc3Cl)Cl)F.Br BTB03986 COc1ccc(c2c1c(=O)cc(o2)C(=O)O)OC BTB10024 Cc1cccc(c1NC(=O)CN2CCOCC2)C BTB13831 Cc1c(c(c(o1)C)S(=O)(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5)C(=O)OC HTS08764 c1ccc(cc1)C#Cc2ccc(o2)C(=O)N3CCCCC3 KM08686 CCN(CC)c1ccc(cc1)C=C2C(=O)c3ccccc3C2=O NRB01428 COC(CNC(=S)Nc1cc(ccc1Cl)Cl)OC RDR00369 COc1ccccc1N\2C(=O)CS/C2=N\N=C\c3ccccc3OC(=O)c4ccc(cc4)Cl RJF01000 c1cc(ccc1N2C(=O)CSC2=S)Cl S01224 COc1ccccc1C2CC(=Nc3ccccc3S2)c4ccccc4 S02348 CCOC(=O)c1c2c(sc1NC(=O)CN3CCN(CC3)C)CN(CC2)C(=O)OCC HTS12779 CCOC(=O)N1CCc2c(sc3c2c(=O)n(cn3)Cc4ccccc4Cl)C1 HTS12997 COc1ccc(cc1)/C=N/NC(=O)/C(=C/c2cccs2)/NC(=O)c3ccccc3 HTS13065 COc1ccc(cc1OC)CCN\2C(=O)CS/C2=N\c3ccc(cc3Cl)Cl S05287 COCc1c(c(nc(n1)c2ccccn2)O)CC3CC3 RJF01816 Cc1cc(no1)c2nnc(n2C)SCC(=O)c3ccccc3 SPB06299 CC1(CC2=C(C(C3=C(N2)CC(CC3=O)(C)C)c4ccc(s4)[N+](=O)[O-])C(=O)C1)C S06318 Cc1ccc(cc1)/C=C/c2ccc3ccccc3[n+]2C.[I-] S08179 CC(C)(C)c1ccc(cc1)c2nnc(n2Cc3ccco3)SCC=C SPB00784 c1cc(sc1)C(=O)Oc2ccc(cc2)C3SCCS3 SPB00849 c1cc(ccc1N2C(=O)C=CC2=O)Br S03021 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)/N=C\c3ccc(cc3)OC)C SEW04183 c1cc(c(cc1Cl)Cl)S(=O)(=O)NNC(=O)c2cc3c(s2)cc(cn3)C(F)(F)F SPB04798 c1cnc(nc1)N2CCN(CC2)S(=O)(=O)c3ccc(nc3)N4CCOCC4 HTS13694 c1ccc(cc1)OCC(=N)N.Cl MO07572 c1cc(ccc1CNC(=O)c2ccc(c(c2)Cl)Cl)C(F)(F)F CD10750 CC1=CC(=O)N(C1=O)c2ccnn2C(=O)C GK02803 Cc1ccc(cc1)/N=N/c2c(nn(c2O)C)C CD11020 CCOC(=O)c1cnc(nc1C(F)(F)F)NNC(=O)c2ccc(cc2)C(C)(C)C GK03032 c1cc(ccc1Nc2ccc3c(c2[N+](=O)[O-])nsn3)Cl KM06751 c1cc(ccc1CSc2[nH]nc(n2)NS(=O)(=O)c3ccc4c(c3)CCO4)Cl HTS10720 CC1CN(CC(O1)C)CN2C(=O)c3ccccc3C2=O NS00009 c1ccc(cc1)CN2CCN(CC2)Cc3cccnc3 HTS13961 Cc1ccc(n1c2c(c3c(s2)CCCC3)C(=O)NNC(=O)C)C GK03269 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)c3ccccc3)C HTS00994 CCOC(=O)c1csc(n1)Nc2ccncc2 SEW06613 CN(C)/C=N/NC(=O)c1cc(on1)COc2cc(cc(c2)Cl)Cl SPB01300 CCOC(=O)Cn1cnc2c3c(cc(nc3sc2c1=O)C)C HTS10293 Cn1c2c(cc(s2)C(=O)Nc3ccc(c(c3)Cl)F)c(n1)C(F)(F)F GK02687 Cc1c2c(cc(s2)C(C)(C)C)sc1C(=O)Nc3ccccc3 GK01908 CC(C)N(Cc1ccccc1)C(=O)c2ccc(cc2)OC(F)(F)F HTS07893 c1cc(ccc1n2ccc(=O)c(n2)C(=O)NN)F SPB04005 Cc1nc(cs1)c2ccc(cc2)C#N SP00460 c1ccc(cc1)N2C(C3CCc4ccccc4C3=N2)c5cccs5 HTS12418 c1ccc2c(c1)CCC3C2=NN(C3c4ccc(cc4)Cl)C(=O)CN5CCOCC5 HTS12432 CNC(=O)c1ccc(cc1)Cl HTS13706 c1ccc(cc1)NC(=S)C(C#N)C(=O)N RF02344 CN(C)Cc1c[nH]c2c1cc(cc2)OCc3ccccc3 AC10608 Cc1cc(nc(c1)NC(=S)Nc2cccc(c2)OC)C S04878 CC(C)c1ccccc1/N=C/c2cc(cc(c2O)Cl)Cl S05008 COc1cc(c(cc1Cl)OC)NC(=S)N/N=C/c2ccc(cc2O)O CD03234 Cc1nc2cc(ccc2c(=O)n1CC3CCCO3)Cl BTB01331 c1cc(ccc1N)S(=O)(=O)N2CCCCC2 TL00817 c1cc2c(c(c1)S(=O)(=O)NC3CCS(=O)(=O)C3)non2 HTS02825 CC(=O)c1c(cc(s1)c2ccc(cc2)C(C)(C)C)NS(=O)(=O)c3ccccc3 GK03549 c1ccc(c(c1)NC(=S)Nc2ccc(cc2)Cl)Sc3nccc(n3)C(F)(F)F HAN00308 CN(c1ccc(cc1)C(C(=O)OC)(C(F)(F)F)O)C(=O)Nc2ccc3ccccc3c2 JFD02157 c1cc(sc1)CC(=O)NCc2cc(cc(c2)Cl)Cl BTB08688 Cc1ccc(cc1)n2c(nnn2)/C=C\Nc3ccc(cc3)O NRB03424 c1cc(cc(c1)NC(=S)Nc2ccc(cc2)[N+](=O)[O-])C(F)(F)F RDR00047 CN(C)CCCN1c2ccccc2CCc3c1cc(cc3)Cl.Cl RJC01223 CCCCc1c(nc(nc1O)SC)C RDR02439 CN(C)/C=C(/c1nnnn1c2ccccc2)\C(=O)c3cc(cc(c3)F)F JFD00606 Cc1ccc(cc1)C(=O)Nc2ccccc2N3CCCCC3 HTS08456 CCN(CC)c1ccc(cc1)NC(=O)Nc2ccc(cc2)OCc3ccccc3 HTS03917 CC(=O)c1c(c(c(s1)SC)C#N)N KM03413 Cc1ccc(cc1)C2CC(=O)CC(=O)C2 CD11331 c1ccc2c(c1)ccnc2C#N BTB09817 Cc1ccccc1C(=O)Nc2cccc(c2)F RDR01806 CC(C(=O)Nc1ccc(cc1)Br)Oc2ccc(cc2)I RDR02316 CC(C)CC(C(=O)N)NC(=O)OC(C)(C)C JFD02955 c1cc(ccc1Nc2c3c(nc4n2ncn4)CCC3)Cl HTS07590 CC(C)(C)c1ccc(cc1)C(=O)NNC(=O)Cn2nc(nn2)c3cccc(c3Cl)Cl RJF02067 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNc3c(cncc3Cl)Cl HTS03086 Cc1ccc(n1C)CNC(=O)Nc2ccc(cc2)OC(F)(F)F HTS10879 c1c(cc(cc1C(F)(F)F)C(F)(F)F)/C=C/c2nc(on2)CN3CCCCCC3 CD04868 Cc1c(nnn1c2cccc(c2Cl)Cl)/C(=N/OCc3c(cccc3Cl)Cl)/C CD05156 c1cc(cc(c1)S(=O)(=O)NCc2ccc3c(c2)OCO3)Oc4cccc(c4C#N)Cl HTS03962 c1cc(ccc1C(=O)CN2CCN(CC2)c3nc4cc(ccc4s3)Cl)F HTS03290 c1cc(ccc1c2nc(on2)CCC(=O)O)C(F)(F)F SEW04217 c1ccc(cc1)c2c(c(=O)[nH]nc2c3ccccc3)C#N HTS09886 c1cc(c(cc1Cl)Cl)CNC(=O)c2cc3cc(ccc3[nH]2)Cl HTS09323 Cn1c2c(c(=O)n(c1=O)C)n(c(n2)N/N=C\3/c4ccccc4NC3=O)Cc5ccc(c(c5)Cl)Cl HTS11201 c1cc2cccc(c2c(c1)c3cccc4c3c(ccc4)C(=O)O)C(=O)O BTB10712 CCOC(=O)c1c2c(sc1NC(=O)Nc3ccc(c(c3)Cl)Cl)CC(CC2)C HTS10020 Cc1ccc2c(c1)c(c[nH]2)c3nnnn3c4ccc(cc4)Br HTS10405 c1ccc2c(c1)CCN2CC(=O)Nc3c(c4c(s3)CCC4)C#N HTS13494 CCOC(=O)C(c1cc(cc(c1)C(F)(F)F)C(F)(F)F)(c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O CD05395 c1ccc(cc1)C(=O)Nc2ccc(c(c2)C(=O)O)N3CCOCC3 HTS11146 c1ccc(cc1)c2c(nnc(n2)N/N=C/3\c4ccccc4NC3=O)c5ccccc5 HTS12554 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)Nc2ccc(cc2F)F S06194 c1ccc(cc1)S(=O)(=O)N2CCCC2c3cccnc3 SCR00229 CC1(Cc2cccc(c2O1)C(=O)N3CCC(CC3)(c4ccc(cc4)Cl)O)C SCR00532 COc1ccc(c(c1)c2cc(c3cc4ccccc4cc3n2)C(=O)O)OC S05343 c1c(c2csc(c2nc1C(F)(F)F)C(=O)O)O KM07538 CCOC(=O)N1CCc2c(sc(c2C#N)NC(=O)CSc3nnc(o3)c4ccco4)C1 HTS12790 CCOC(=O)N1CCC(CC1)NC(=O)Nc2ccc(cc2)F HTS05182 c1ccc(cc1)C\2=NOC(=O)/C2=N/Nc3c(cccc3Cl)F RF00976 Cc1nnc(s1)SCc2cccc(n2)CSc3nnc(s3)C RJC02450 c1ccc2c(c1)c(=O)c(co2)Br RF01262 c1ccc(cc1)c2cc(c(s2)N)C(=O)N/N=C/c3ccc(cc3)Cl HTS13010 COc1cc(nc(n1)NCC(C(=O)N)NC(=O)c2ccccc2)OC BTB09737 COc1ccc(cc1)/C=N/NC(=O)c2c(n(c(=S)s2)c3ccccc3)N HTS07571 CN(C1CCCCC1)C(=O)c2ccc3c(c2)OCO3 HTS07919 c1ccc(cc1)CN2CCC(=O)N(C2=O)c3ccccc3 HTS05900 CC(C)(C)N1CNC(=NC1)SC.Br DP01601 c1cc(ncc1C(F)(F)F)OCC(CSc2ccc(cn2)C(F)(F)F)O HAN00260 COc1ccc(c(c1)Nc2ncnc(n2)N)OC RJF00654 COc1ccc(cc1)CN2CCCN(C2c3cccc4c3OCO4)Cc5ccc(cc5)OC SCR00743 COc1cccc(c1)NC(=O)CN2C(=O)c3ccccc3C2=O SCR00970 COc1c(csc1S(=O)(=O)NC2CCCCNC2=O)C(=O)OC SCR00980 c1ccc(cc1)S(=O)(=O)NNC(=O)c2cnn(c2C(F)(F)F)c3ccc(cc3)Cl HTS00412 c1cc(cc(c1)Cl)NCC(=O)c2ccc(cc2)Cl BTB03148 CC(C)(C)C(=O)NNc1c2ccsc2ncn1 GK02927 Cc1cccc(c1NC(=O)NNC(=O)c2cc(n(n2)C(C)(C)C)C)Cl HTS00057 c1ccc2c(c1)nc3n2c(c(s3)C#N)/N=C/N4CCOCC4 HTS07536 CC(C(=O)Oc1ccc2ccccc2c1I)Oc3ccc(cc3Cl)Cl RDR02573 CS(=O)(=O)OCC(COS(=O)(=O)C)(C1CCCCC1)[N+](=O)[O-] RJC01323 Cc1c2cc3c(cc2ncc1c4nnnn4c5ccc(cc5)F)OCO3 HTS05459 COc1ccc(c(c1)C=C2C(=O)NC(=O)NC2=O)OC CD00548 c1cc(c(cc1N2C(=O)C3C4CC(C3C2=O)C=C4)F)F DSHS01086 c1cc(ccc1NS(=O)(=O)c2ccsc2C(=O)O)S(=O)(=O)N HTS00374 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)O/N=C(/c3ccc(o3)[N+](=O)[O-])\N RF02857 CCOC(=O)c1cc(nc(c1C#N)S)C RF00734 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)NNc3ccccn3 RF00929 CC\1=NNC(=O)/C1=N\Nc2ccc(cc2)F RJC02938 Cc1cn(c(=O)[nH]c1=O)Cc2ccccc2Cn3cc(c(=O)[nH]c3=O)C HTS09831 CSc1c(c(c(s1)c2ccnc(n2)S)c3ccccc3)C#N KM05733 CCOC(=O)N1CCN(CC1)CC(Cn2cnc3c2c(=O)n(c(=O)n3C)C)O NRB03540 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2cc(nn2CCC#N)c3ccccc3)C)C CD06946 Cc1cccc(c1NC(=O)c2cnc(cc2C(F)(F)F)OC)C RF04382 Cc1cc(nn1c2ccc(cc2)[N+](=O)[O-])CO JM00395 CC(C)(C)c1ccc(cc1)NC(=O)N2CCCc3c2cccc3 HTS10191 c1ccc(cc1)/C(=C/2\CCc3ccccc3C2=O)/CC(=O)c4ccccc4 NRB03368 Cc1c(sc(n1)c2ccccc2)C(=O)Nc3ccc4c(c3)OCCO4 HTS10413 c1cc(ccc1c2csc(n2)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)[N+](=O)[O-].Br CD03043 c1cc(sc1)SCC(=O)Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F KM02698 c1ccc(c(c1)C(=O)NC(=O)c2c(cccc2Cl)F)O HTS10463 CN(C1CCCCC1)C(=O)c2ccc3c(c2)nccn3 HTS08834 Cc1c(c(no1)c2c(cccc2Cl)F)C(=O)NNC(=O)c3ccc(cc3)C(F)(F)F HTS09187 c1cc(c(nc1)NCCNC(=O)CSCC(=O)O)C(F)(F)F HTS03482 c1cc(ccc1C(=O)N2CCNC(=O)C2CC(=O)Nc3cc(ccc3Cl)Cl)F HTS07975 CC1CCc2c(sc(c2C#N)NC(=O)CN3CCN(CC3)c4ccccc4)C1 HTS10332 CCc1cccc(c1NC(=O)c2cccs2)C(C)C CD06431 c1cc(ccc1NC(=S)NCCO)N2CCOCC2 S04604 c1ccc(cc1)c2cc(c3c(c(oc3n2)C(=O)N/N=C/c4ccc(cc4)F)N)c5ccco5 HTS12138 c1ccc(cc1)c2cc([nH]c(=O)c2C#N)c3ccc(cc3)Br S06666 c1ccc2c(c1)-c3ccccc3C2N4CCN(CC4)C(=O)Nc5ccc(cc5)OC(F)(F)F HTS09201 Cn1c2c(nc1NCc3ccccn3)n(c(=O)n(c2=O)Cc4cccc(c4)Br)C HTS12278 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2ccc(cc2)n3cccn3 HTS10680 Cc1c(c(nc(c1[N+](=O)[O-])C)O)C(=O)N RF00069 COc1cc(cc(c1)OC)C(=O)CC2c3ccccc3C(=O)O2 S05973 CC/C(=N\Cc1ccc(cc1)C#N)/c2ccccc2O S04267 c1c(c(n(n1)c2c3c4c(sc3ncn2)CCCC4)N)C#N HTS12934 c1cc-2c(cc1S(=O)(=O)N3CCCCCC3)C(=O)c4c2ccc(c4)S(=O)(=O)N5CCCCCC5 HTS13702 CC(=O)Nc1ccc(cc1)Oc2cc(c(cc2Cl)C#N)C#N HTS13705 Cc1ccc(cc1)NC(=O)NN2CC(=O)N(CC2=O)c3ccccc3F HTS12928 CCOC(=O)CN(c1ccccc1C)C(=O)COc2c(c(cc(n2)c3ccccc3)C)C#N HTS13385 c1cc(sc1)/C=c\2/c(=O)n3c(nnc3s2)c4ccc(cc4)Cl HTS13280 c1ccc(cc1)n2c(nnc2Sc3ncc(c(n3)N)C#N)c4ccco4 HTS12718 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccc(cc3)Cl)CN(CC2)C(=O)OCC HTS12993 Cc1c2cc(sc2n(n1)C)C(=O)NCc3ccc(cc3)c4cccs4 SCR01423 c1cc(ccc1C23CC4CC(C2)CC(C4)(C3)C(=O)O)[N+](=O)[O-] RJC00957 CCCc1c(cnn1c2ccc(cc2)Cl)C(=O)NCCc3ccccn3 GK01745 C[C@@H](C(=O)NCc1cccnc1)NC(=O)c2ccc(cc2Cl)Cl HTS12325 CCNC(=O)O/N=C(\C)/c1cnn(c1C)c2cc(cc(n2)C)C(F)(F)F CD11712 c1cc(c(c(c1)Cl)F)N/C=C(\C#N)/S(=O)(=O)c2ccc(cc2)Cl KM01235 Cn1c(cc(n1)c2ccccc2)NS(=O)(=O)c3ccc(cc3)C#N HTS10214 c1cc(sc1)CN2C3CCCC2CC(=NO)C3 KM08822 c1cc(ccc1C#N)c2c(c(n(c(=O)c2C#N)N)N)C#N P00086 CCCOc1cccc(c1)/C=N/Nc2nc3c(ncnc3n2[C@@H]4[C@H]([C@H]([C@@H](O4)CO)O)O)N HTS09791 CCC(=O)Nc1ccc(cc1C)c2nnc(o2)C(F)(F)F RH00950 CC(C)Oc1ccc(cc1)C[C@H](C(=O)O)NC(=O)C SPB08037 c1cc(c(cc1Cl)Cl)C(=O)NCCCl RDR03675 c1ccc(c(c1)NC(=O)Nc2ccc(s2)c3ccccn3)Cl KM02624 Cc1c(nn(n1)c2ccccc2)CNS(=O)(=O)c3ccc4c(c3)N(CCO4)C SCR01453 COc1cccc(c1C(=O)NNC(=O)c2cnc(s2)c3cccnc3)OC MWP01175 c1c(c(c(cn1)Cl)N2CCNCC2)Cl SPB06834 CCO/C=C/1\C(=NN(C1=O)c2cccc(c2)Cl)C BTB06421 c1cc(cc(c1)NN2C(=O)c3c(c(c(c(c3Cl)Cl)Cl)Cl)C2=O)C(F)(F)F S05560 Cc1c(cc(n1CCCN2CCOCC2)c3ccccc3)C(=O)O SP00344 c1cc(ccc1/C(=N/O)/N)Cl SPB06960 CC1(Cc2c(cnc(n2)SCC(=O)NCC=C)C(=O)C1)C KM04733 CC1(C=Cc2cc(ccc2O1)c3nc(on3)c4cccs4)C KM06996 CCOC(=O)c1cnn(c1C(F)(F)F)c2ccc(cc2)Cl GK01546 CCO/C=C(\C#N)/S(=O)(=O)c1ccccc1 KM00478 c1cc(ccc1Sc2ccc(s2)S(=O)(=O)N)Cl KM03958 CC(C)(C)c1c(cno1)C(=O)OC SEW04583 c1ccc2c(c1)C(=C(C2=O)c3ccc(cc3)Br)O RJC01751 c1cc(c(cc1C(F)(F)F)N)N BTB07340 COc1ccc(c(c1)C(=O)c2c3nc(c4c(n3nn2)cccc4Cl)N)Br CD07379 c1ccc(cc1)SCC(=O)N2c3ccccc3Sc4c2cccc4 HTS10265 c1cc2c(cc1C(=O)Nc3cc(ccc3N4CCCC4)C(F)(F)F)CCO2 HTS13704 c1ccc(c(c1)c2nnnn2c3ccc(cc3Cl)Cl)C(F)(F)F RF04531 Cn1c(n[nH]c1=S)CSc2nnc(n2CC=C)c3ccccc3 HTS07459 c1ccc(cc1)n2c3c(c(=O)[nH]cn3)sc2=S HTS07575 c1c(c(n[nH]1)C#N)Br RF05036 COc1ccc(cc1OC)/C=N/NC(=O)CSC2CN(C2)C(c3ccccc3)c4ccccc4 KM09566 C/C(=C(/C#N)\C(=O)N)/c1ccccc1 NRB04281 c1cc2cccc3c2c(c1)CC3O RDP00045 CC(C)(C)c1cc(n(n1)Cc2ccccc2)C(=O)Nc3ccccc3Cl SPB03054 Cc1c(c(no1)C(=O)NNC(=O)Nc2ccccc2)c3csc(n3)C SPB03394 c1ccc(cc1)COc2ccccc2C(=O)/C(=C/c3ccccc3)/[N+](=O)[O-] NRB04941 c1cc(ccc1C2c3ccsc3CCN2)C(F)(F)F SEW01183 CCOC(=O)CSC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F RDR02166 CCOC(=O)c1cc(on1)CSc2nnc(s2)SC SPB02627 CCOC(=O)c1c2c(sc1NC(=S)Nc3ccccc3)CN(CC2)C HTS11935 CC(C)(C)NC(=S)N1CCN(CC1)C(=S)NC(C)(C)C S06100 c1cc(c(c(c1)Cl)CN2C(SCC2=O)c3cccnc3)F S07597 c1ccc(cc1)NC(=O)O/N=C(/c2ccc(cc2)OCc3c(cc(cn3)C(F)(F)F)Cl)\N SPB05170 CC(C)(C)c1ccc(cc1)c2nc(on2)CCOc3ccc(cc3)F SEW01470 COc1ccccc1C2CCN(CC2)C(=O)c3ccccc3Cl RH01501 CCOC(=O)CC(=NNc1ccccc1[N+](=O)[O-])N NRB01448 c1cc(c(cc1C(F)(F)F)Cl)Oc2ccc(c(c2)F)N.Cl MO08102 c1ccc(cc1)C(=O)NNC(=S)Nc2ccccc2 HTS07429 c1ccc(cc1)c2c(sc(n2)Nc3ccc4c(c3)OCCO4)C(=O)c5ccc(cc5)F HTS10133 c1cc(c(cc1NCC(=O)NN)Cl)Cl NRB00020 COc1ccc(cc1)n2c(nnc2SCC(=O)c3ccc(cc3)c4ccccc4)c5ccncc5.Br ML00379 c1ccc2c(c1)CC(O2)C(=O)O CC23901 CCOC(=O)[C@H](C(C)C)NS(=O)(=O)c1cc(c(s1)Cl)Br HTS13696 CCOC(=O)[C@H](C(C)C)NS(=O)(=O)c1ccc(cc1)OC(F)(F)F HTS13695 CC1CCC(C(C1)N(Cc2ccccc2)C(=O)c3cccs3)C(C)C JFD02578 COc1ccc(c(c1)C(=O)Nc2ccc(cc2F)F)Br S07814 c1ccc(c(c1)COC(=O)NCCCC[C@@H](C(=O)O)N)Cl RJC01689 C[C@@H](c1ccccc1)Nc2c3c4c(sc3ncn2)CCCC4 GK03380 CC(C)c1ccc(cc1)NC(=S)NC(C)(C)CO RDR01688 Cc1nc(cs1)CC(=O)O CD12020 Cc1ccccc1NC2CC(NC(C2)(C)C)(C)C NRB00486 c1ccc2c(c1)-c3cccc(c3C2=O)C(=O)N4CCOCC4 HTS10473 c1ccc2c(c1)OCC(O2)C(=O)O CC01501 c1cc(ccc1C(=O)O)N2CCOCC2 CC17401 c1cc(c(nc1)N2CCOCC2)C(=O)O CC24601 CCc1ccccc1NC(=S)N HTS13955 CC(C)(C)c1nc(nc(n1)SC)N RF02694 C[C@H](CCCC(C)C)[C@H]1CC[C@@H]2[C@@]1(CC[C@H]3[C@H]2CCC4=CC(=O)CC[C@]34C)C SB01791 COC(=O)c1cc(n(n1)c2cc(cc(c2)C(F)(F)F)C(F)(F)F)O SEW00037 CN(C)CC#Cc1ccc(cc1)/C=N/O MO08250 CC1(C=CN(C(=S)N1)c2cccc(c2)OC)C SEW05412 Cc1c2c(onc2c(=O)n(n1)c3ccccc3)C SPB03609 CC(C)Sc1nnc(n1c2cccc(c2)C(F)(F)F)OC(=O)N(C)C SPB00871 Cc1c(c(no1)C(=O)OC)C(=O)/C=C/N2CCCCC2 SPB04601 Cc1cc(ccc1Br)NC(=N)NC(=N)N.Cl RJF00660 Cn1c(cc(n1)c2ccccc2)NC(=O)c3c(nccn3)C(=O)O HTS10209 c1ccc(cc1)c2c(c3nnnn3nc2c4ccccc4)C(=O)NN JFD00399 c1cc(ccc1C(=O)CCCN2CCC(CC2)(c3ccc(cc3)Cl)O)F BTBS00008 c1ccc(cc1)c2nc(c(=O)n(n2)CN3CCOCC3)C(CN4CCOCC4)c5ccccc5Cl HTS13345 CCOC(=O)C12CCC(CC1)(CC2)OS(=O)(=O)c3ccc(cc3)[N+](=O)[O-] NRB01949 Cc1ccc(cc1NS(=O)(=O)C)N BTB01378 c1cc(sc1)C(=O)Nc2ccc3c(c2)nsn3 HTS13734 c1ccc2c(c1)CC(O2)C(=O)Nc3ccc4c(c3)nsn4 HTS13735 c1ccc2c(c1)CC(CO2)C(=O)Nc3ccc4c(c3)nsn4 HTS13736 COC(=O)c1ccc(o1)COCOCc2ccc(o2)C(=O)OC NH00370 Cn1c(c(cn1)Br)c2cccc(c2)N MO08354 Cc1c(sc(n1)c2cc(nc(c2)Cl)Oc3ccc(cc3)Cl)/C(=N/Nc4ccccc4)/C SPB06736 c1ccc2c(c1)c(cs2)S(=O)(=O)Nc3ccc4c(c3)nsn4 HTS13790 c1ccc(cc1)NC(=O)c2cccc3c2nsn3 HTS13808 COc1ccc(cc1)NC(=O)c2cccc3c2nsn3 HTS13810 c1ccc2c(c1)CCCC2NC(=O)c3cccc4c3nsn4 HTS13811 c1cc2c(c(c1)NC(=O)c3cccc4c3nsn4)CCCC2 HTS13812 CC(C)(C)c1ccc(cc1)NC(=O)Nc2ccc3c(c2)nsn3 HTS13777 c1cc(c2c(c1)nsn2)C(=O)Nc3ccc4c(c3)CCC4 HTS13813 c1cc(c2c(c1)nsn2)C(=O)Nc3ccc(cc3)Cc4ccncc4 HTS13817 c1ccc(c(c1)NC(=O)c2cccc3c2nsn3)N4CCOCC4 HTS13818 c1ccc(c(c1)NC(=O)Nc2ccc3c(c2)nsn3)N4CCCCC4 HTS13765 c1ccc(c(c1)NC(=O)Nc2ccc3c(c2)nsn3)Cl HTS13778 c1ccc(c(c1)NC(=O)Nc2ccc3c(c2)nsn3)OC(F)(F)F HTS13779 c1ccc(c(c1)NC(=O)Nc2ccc3c(c2)nsn3)F HTS13780 CSc1cccc(c1)NC(=O)Nc2ccc3c(c2)nsn3 HTS13782 c1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)nsn3 HTS13783 Cc1ccc2cc(ccc2n1)NC(=O)c3cccc4c3nsn4 HTS13819 c1c(cncc1Br)C(=O)O SB01732 COc1ccc(cc1)OCCNC(=O)c2cccc3c2nsn3 HTS13820 CC(C12CC3CC(C1)CC(C3)C2)NC(=O)c4cccc5c4nsn5 HTS13821 c1cc(cc(c1)NC(=O)Nc2ccc3c(c2)nsn3)C(F)(F)F HTS13753 c1cc2c(cc1NC(=O)Nc3ccc4c(c3)ccs4)nsn2 HTS13766 Cc1nc(no1)c2cccc(c2)NC(=O)Nc3ccc4c(c3)nsn4 HTS13768 c1cc(cc(c1)NC(=O)Nc2ccc3c(c2)nsn3)CN4CCOCC4 HTS13769 Cc1nc(cs1)c2ccc(cc2)NC(=O)Nc3ccc4c(c3)nsn4 HTS13770 c1cc(cc(c1)Cl)C(=O)Nc2ccc3c(c2)nsn3 HTS13716 Cc1cccc(c1)C(=O)Nc2ccc3c(c2)nsn3 HTS13718 Cc1ccc(cc1)C(=O)Nc2ccc3c(c2)nsn3 HTS13719 COc1cccc(c1)C(=O)Nc2ccc3c(c2)nsn3 HTS13720 c1ccc(cc1)Oc2c(cccn2)C(=O)Nc3ccc4c(c3)nsn4 HTS13721 c1cc2c(cc1NC(=O)C3CCOCC3)nsn2 HTS13739 Cc1cc(sc1)C(=O)Nc2ccc3c(c2)nsn3 HTS13740 c1ccc(c(c1)c2cccs2)C(=O)Nc3ccc4c(c3)nsn4 HTS13741 Cn1c(c2ccccc2n1)C(=O)Nc3ccc4c(c3)nsn4 HTS13742 CC(C)c1ccc(cc1)NC(=O)Nc2ccc3c(c2)nsn3 HTS13755 CSc1ccc(cc1)NC(=O)Nc2ccc3c(c2)nsn3 HTS13756 c1ccc(c(c1)C#N)NC(=O)Nc2ccc3c(c2)nsn3 HTS13757 c1ccc(cc1)Oc2ccccc2C(=O)Nc3ccc4c(c3)nsn4 HTS13743 Cn1c(c(cn1)C(=O)Nc2ccc3c(c2)nsn3)Cl HTS13745 CCCc1ccc(cc1)C(=O)Nc2ccc3c(c2)nsn3 HTS13722 c1cc(sc1)c2nc(cs2)C(=O)Nc3ccc4c(c3)nsn4 HTS13731 c1ccc(cc1)c2c(nco2)C(=O)Nc3ccc4c(c3)nsn4 HTS13730 c1ccc(c(c1)C(C(=O)O)O)Cl RDR03335 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)nsn3 HTS13784 c1ccc2cc(ccc2c1)S(=O)(=O)Nc3ccc4c(c3)nsn4 HTS13786 Cc1c(oc(n1)c2ccc(cc2)c3nc(c(o3)c4ccccc4)C)c5ccccc5 SB01211 CC1([C@@H](N2[C@H](S1)[C@@H](C2=O)N)C(=O)O)C SB01619 CSc1ccccc1NC(=O)Nc2ccc3c(c2)nsn3 HTS13771 COc1ccc(cc1)NC(=O)Nc2ccc3c(c2)nsn3 HTS13773 c1ccc(cc1)Oc2ccc(cc2)NC(=O)Nc3ccc4c(c3)nsn4 HTS13774 c1cc(ccc1NC(=O)Nc2ccc3c(c2)nsn3)OC(F)(F)F HTS13775 CCCc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)nsn3 HTS13788 Cc1c(c(on1)C)NC(=O)Nc2ccc3c(c2)nsn3 HTS13759 c1cc(sc1)c2ccc(cc2)NC(=O)Nc3ccc4c(c3)nsn4 HTS13761 c1cc(sc1)NC(=O)Nc2ccc3c(c2)nsn3 HTS13762 c1cc2c(cc1NC(=O)Nc3ccsc3)nsn2 HTS13763 c1ccc(c(c1)C(F)(F)F)NC(=O)Nc2ccc3c(c2)nsn3 HTS13776 c1cc2c(cc1C(=O)Nc3ccc4c(c3)nsn4)nccn2 HTS13732 CC(C)(C(=O)Nc1ccc2c(c1)nsn2)Oc3ccc(cc3)Cl HTS13746 c1ccc(cc1)CCC(=O)Nc2ccc3c(c2)nsn3 HTS13747 c1cc(c(c(c1)Cl)C(=O)Nc2ccc3c(c2)nsn3)F HTS13749 c1cc(ccc1NC(=O)Nc2ccc3c(c2)nsn3)Cl HTS13750 c1ccc(cc1)NC(=O)Nc2ccc3c(c2)nsn3 HTS13751 Cc1c(cnn1c2ccccc2)NC(=O)Nc3ccc4c(c3)nsn4 HTS13764 c1cc(n(c1)c2ccc(cc2)OC(F)(F)F)/C=N/Nc3c(cc(cn3)C(F)(F)F)Cl SEW06337 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)NCc3cc(cc4c3OCOC4)F HTS03237 C1CCC(CC1)C[C@@H](C(=O)O)N SB02002 c1cc(ccc1S(=O)(=O)C2=CC34CCCC3(C2)C=C(C4)S(=O)(=O)c5ccc(cc5)Cl)Cl RJC02964 Cc1c(cn(n1)C(=O)Nc2c(onc2c3c(cccc3Cl)Cl)C)c4ccccc4 CD09350 c1ccc(c(c1)CNC(=O)c2cccc3c2nsn3)Cl HTS13873 Cc1ccccc1N2CCN(CC2)C(=O)c3cccc4c3nsn4 HTS13890 Cc1cc(nc(c1C#N)Sc2c(ncn2C)[N+](=O)[O-])C HTS03867 Cc1ccc(cc1)/N=C/c2c(cnn2c3ccccc3)C(=O)OC SPB05120 c1cc(oc1)c2cc(nc3c2c(c(o3)C(=O)NN)N)c4cccs4 HTS12664 c1ccc(cc1)C(=O)C2=NN(C3(C2c4ccc(cc4)Cl)C(=O)c5ccccc5C3=O)c6ccccc6 HTS13244 CSCCNC(=O)Nc1ccc(cc1)Cl CD06889 c1(c(nc(nc1O)N)N)Br BTB13031 Cc1cc(no1)NC(=O)c2c(onc2c3c(cccc3Cl)F)C CD09161 Cc1ccc(cc1)CNC(=O)c2cccc3c2nsn3 HTS13874 c1cc(c2c(c1)nsn2)C(=O)NCc3ccc(cc3)F HTS13876 c1cc(c2c(c1)nsn2)C(=O)Nc3ccc(cc3)Cl HTS13877 Cc1ccc(cc1)NC(=O)c2cccc3c2nsn3 HTS13878 COc1ccc(cc1)SCCC(=O)NNS(=O)(=O)c2cccs2 HTS05853 CC(C)(C)OC(=O)NCc1nnc(n1C)SCc2ccc(cc2)Cl KM10584 c1coc(c1)/C=N/CC2CCC(CC2)C/N=C/c3occc3 S01517 c1ccc(cc1)c2cc(cc(n2)c3cccc(c3)[N+](=O)[O-])c4cccs4 RB00120 c1cc(c(cc1[N+](=O)[O-])Cl)CSc2c(cncc2Cl)Cl RF03615 Cc1ccc(cc1)S(=NC(=O)NS(=O)(=O)Oc2ccc(cc2Cl)Cl)(=O)C KM03066 c1cc(ccc1S(=O)(=O)/C(=C/c2c[nH]cn2)/C#N)Cl KM08309 Cc1c(cc2c(c1N)C(CC2(C)C)(C)C)NC(=S)Nc3ccc(c(c3)Cl)Cl CD03881 C/C(=N\NC(=S)N)/c1cccs1 BTB13750 c1cc(cc(c1)NC(=O)c2cccc3c2nsn3)c4cccs4 HTS13861 COc1cc(cc(c1OC)OC)C(CC(=O)CNc2ccc3c(c2)OCCCO3)CC(=O)O HTS00131 c1ccc2c(c1)CCN2/C=C(\C#N)/C(=O)c3cccc(c3)C(F)(F)F KM05387 c1ccc(cc1)c2c3ccc(cc3[nH]c2NC(=O)c4cccs4)[N+](=O)[O-] HTS02308 c1ccc2c(c1)nnn2Cc3n[nH]c(=S)n3c4cccc(c4)C(F)(F)F HTS12624 c1cc(c(c(c1)Cl)Oc2ccc(cc2Cl)[N+](=O)[O-])Cl BTB03905 Cc1cc(c(c(c1)C)S(=O)(=O)O)C.CS(=N)c1c(cc(cn1)Cl)C(F)(F)F KM05698 c1cc(cc(c1)Cl)CC(=O)c2cccc(c2)C#N MO00231 c1cc-2c(cc1[N+](=O)[O-])C(=O)c3c2c(cc(c3)[N+](=O)[O-])O BTB10911 c1cc(nc(c1)N2CCCCC2)CNC(=O)c3cccc4c3nsn4 HTS13848 Cc1nc(no1)c2cccc(c2)NC(=O)c3cccc4c3nsn4 HTS13849 c1cc(cc(c1)NC(=O)c2cccc3c2nsn3)c4cncnc4 HTS13851 Cn1cnnc1c2ccc(cc2)NC(=O)c3cccc4c3nsn4 HTS13865 Cn1c(c(cn1)Br)NC(=O)Nc2ccc(cc2)F GK03416 COc1ccc(cc1Br)C2C3C(=NN2)C4CCN3CC4 DSHS00404 c1cc(sc1)S(=O)(=O)CCS(=O)(=O)c2ccc(cc2)Cl KM02413 Cc1ccc(cc1)S(=O)(=O)N=S2(=O)CCCS(=O)(=O)C2 KM03022 c1cc(oc1)Cn2c(nnc2SCc3ccncc3)c4ccc(cc4)C(F)(F)F HTS11114 Cc1ccc(cc1)C(=O)Nc2ccc(nc2N3CCOCC3)N4CCOCC4 SEW05599 CC(C)(C)c1ccc(cc1)NC(=O)/C=C/c2ccc(s2)c3cccs3 SEW02638 CC(=O)OC(C)(C)/C=C/C(=O)C(C)(C1[C@@H](C[C@@]2([C@@]1(CC(=O)[C@@]3(C2CC=C4C3CC[C@H](C4(C)C)O)CO)C)C)O)O BTB13120 c1ccc(cc1)C(=O)NC2CCN(CC2)CC(=O)N(c3ccccc3)C4CCCCC4 BTB14620 c1ccc(c(c1)CSc2ccc(cc2)Cl)OCC(=O)N/N=C/c3ccccc3Cl KM04700 c1ccc(cc1)S(=O)(=O)Nc2ccccc2C(=O)NC3CCSC3 CD10389 COc1cccc2c1c(no2)NS(=O)(=O)c3ccc4ccccc4c3 HTS13807 Cc1cc(cc(c1Cl)C)Oc2c(cccn2)[N+](=O)[O-] BTB09566 CC(=O)Nc1ccc(cc1F)Br BTB07539 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)c3nnc(o3)S SPB08172 Cn1c(nnc1S)CC2C(=O)Nc3ccccc3S2 KM07420 c1ccc(c(c1)CNC(=O)c2cccc3c2nsn3)N4CCCC4 HTS13852 c1cc(cc(c1)Cl)S(=O)(=O)N2CCN=C(C=C2)C(F)(F)F HTS00229 CC1(C2CCC1(C(=O)C2)CS(=O)(=O)N3CCCN(CC3)c4nc5ccc(cc5s4)Cl)C AW01081 COC(=O)c1cc(=O)n2c(nnc2s1)c3cccs3 SPB05639 CCCCCc1c(c2ccc(cc2oc1=O)O)COC RJF01950 COc1ccc(cc1)Oc2cc(ccn2)C(F)(F)F SEW05710 c1cnn(c1)c2ccc(cc2)S(=O)(=O)Nc3ccc4c(c3)nsn4 HTS13792 Cc1nc(cs1)c2ccc(cc2)S(=O)(=O)Nc3ccc4c(c3)nsn4 HTS13794 Cc1c(c(n(n1)c2ccccc2)C)S(=O)(=O)Nc3ccc4c(c3)nsn4 HTS13795 c1ccc(cc1)C2=NCCN=C2c3ccccc3 S12965 c1ccc2c(c1)N(c3ccccc3S2)C(=O)CSc4[nH]cnn4 HTS10348 COc1ccc(cc1)C(=O)N2CCN(CC2)CCCc3c[nH]c4c3cc(cc4)F HTS01688 c1ccc(cc1)C23c4ccccc4C(=O)N2CCN3C(=O)C(Cl)(Cl)Cl DSHS01065 CCn1c(c(c(n1)C)NS(=O)(=O)c2ccc(cc2)Cl)C(=O)OC SPB01862 CN1CCN(CC1)c2ccc(cc2)CNC(=O)c3cccc4c3nsn4 HTS13836 c1ccc(cc1)Oc2ccc(cn2)NC(=O)c3cccc4c3nsn4 HTS13837 c1ccc(c(c1)CNC(=O)c2cccc3c2nsn3)n4cccn4 HTS13838 c1cc(c2c(c1)nsn2)C(=O)Nc3cccnc3N4CCOCC4 HTS13839 c1cc(c2c(c1)nsn2)C(=O)NCc3ccc4c(c3)ccs4 HTS13840 c1cc(c2c(c1)nsn2)C(=O)Nc3ccc4c(c3)ccs4 HTS13841 c1ccc(cc1)CN2C(=O)C3C4c5ccccc5C(C3C2=O)c6c4cccc6 JFD00490 Cc1c(c(n(n1)S(=O)(=O)c2ccc(cc2)Cl)C)Sc3ncccn3 SPB04375 Cc1c(ccc(c1O)C(=O)/C=C/N(C)C)OCc2ccc(c(c2)Cl)Cl RH00452 CN(CCOC(=O)Nc1ccc(cc1)Cl)c2c(cc(cn2)C(F)(F)F)Cl SPB06274 C1CCC\2C(C1)CC/C2=N/O JFD00553 Cc1nc(nc(n1)SC)N/C=C/2\C(=O)c3ccccc3N(S2(=O)=O)C KM01412 COc1ccccc1C2CCN(CC2)Cc3c[nH]c4c3cccc4 HTS04089 c1ccnc(c1)Sc2ccc(cc2[N+](=O)[O-])S(=O)(=O)N DSHS00894 Cc1c(cc(n1c2ccccc2)C(C)(C)C)C(=O)Nc3cccc(c3)OC SP00313 c1cc(ccc1COc2ccc(cc2)C(=O)CSCc3ccc(c(c3)Cl)Cl)[N+](=O)[O-] BTB09557 Cc1c(c(on1)C)NC(=O)c2cccc3c2nsn3 HTS13823 c1cc(c2c(c1)OCCO2)CNC(=O)c3cccc4c3nsn4 HTS13825 c1ccnc(c1)c2ccc(s2)CNC(=O)c3cccc4c3nsn4 HTS13826 Cc1c(c(c(c(c1C)C)S(=O)(=O)Nc2cccnc2)C)C CD06578 CC1(Cc2cccc(c2O1)C(=O)N3CCC(CC3)c4c[nH]c5c4cccc5)C SCR00498 c1ccnc(c1)CCNC(=S)NN2C3CSC2CS3 JM00039 Cc1ccc(cc1)S(=O)(=O)N(Cc2ccc(cc2)OC)Cc3cccn3C HTS00763 c1ccc(c(c1)NC(=O)/C=C\C(=O)O)SCC(Cn2ccc(n2)C(F)(F)F)O HAN00305 CCOC(=O)C(C(F)(F)F)(Nc1ccc(cc1F)F)NC(=O)c2ccccc2 RJC01582 c1cc(ccc1C(=O)CSc2nc(cc(n2)O)C(F)(F)F)Cl RJF00253 CN1CCN(CC1)c2ccc(cc2)NC(=O)c3cccc4c3nsn4 HTS13884 c1cc(c2c(c1)nsn2)C(=O)Nc3ccc4c(c3)scn4 HTS13828 c1cc(c2c(c1)OCCO2)C(=O)N3CCN(CC3)c4ncccn4 HTS13919 c1ccc(cc1)NC(=O)c2ccc(cc2)n3cccc3 HTS13920 c1ccn(c1)c2ccc(cc2)C(=O)NCCN3CCCC3 HTS13921 c1ccc(cc1)CCNC(=O)c2ccc(cc2)n3cccc3 HTS13923 CC(C)(C)c1cc(n(n1)C)NC(=O)Nc2ccc(cc2)OC(F)(F)F KM08493 c1ccc(cc1)c2c(csc2C(F)(F)F)NC(=S)Nc3cccc(c3)C(F)(F)F SEW03236 CS(=O)CC(c1ccc(cc1)Cl)(c2ccc(cc2)Cl)O RDR03943 COc1ccc(c(c1)OC)Nc2cc(nc3n2ncn3)c4ccccc4 HTS11993 Cc1ccccc1N2C(C3C(O2)C(=O)N(C3=O)c4ccccc4)c5ccc(cc5)N(C)C RJC02533 CCCCCCCCCCNS(=O)(=O)c1cc2c(c(c1)[N+](=O)[O-])-c3c(cc(cc3[N+](=O)[O-])S(=O)(=O)NCCCCCCCCCC)C2=O JFD01206 c1cc(c2c(c1)nsn2)C(=O)N3CCN(CC3)c4ccc(cc4)F HTS13892 c1ccc2c(c1)CCN(C2)C(=O)c3cccc4c3nsn4 HTS13893 COc1ccccc1C2CCN(CC2)C(=O)c3cccc4c3nsn4 HTS13894 Cc1c(c(no1)c2ccccc2)CN(C)C(=O)c3cccc4c3nsn4 HTS13895 CC(C)(C)C1CCN(CC1)C(=O)c2cccc3c2nsn3 HTS13909 CN(Cc1ccncc1)C(=O)c2ccc(cc2)n3cccc3 HTS13925 c1ccc(cc1)S(=O)(=O)NNC(=O)c2csc3c2cc(cc3)Cl MWP00301 Cc1c(c(no1)c2ccccc2Cl)C(=O)N3c4ccccc4NC(=O)CC3C BTB00660 Cc1ccc(cc1)Cn2c(=O)ccc(n2)C BTB06990 c1ccc2c(c1)nc(s2)/C(=C/c3c(cccc3Cl)F)/C#N GK00311 c1cc(c2c(c1)nsn2)C(=O)NCCc3ccc(cc3)Cl HTS13871 c1cc(cc(c1)NC(=O)c2cccc3c2nsn3)c4cnco4 HTS13882 c1ccc(c(c1)N2CCN(CC2)C(=O)c3cccc4c3nsn4)Cl HTS13908 c1cc(ccc1C(=O)Nc2nc3ccc(cc3s2)Cl)C(F)(F)F HTS08907 Cc1cc(c2ccccc2n1)N3CCN(CC3)C(=O)c4cccc5c4nsn5 HTS13912 c1ccc(cc1)C(=O)C2CCN(CC2)C(=O)c3cccc4c3nsn4 HTS13913 Cc1cc(c2cc(ccc2n1)F)OCc3c(c(c(c(c3C)C)C)C)C BTB01285 c1cscc1S(=O)(=O)CC#N SEW03663 CNC(=O)c1cnn(c1COC)c2c(cc(cc2Cl)Cl)Cl CD10620 c1ccc(cc1)OCCNC(=O)c2cccc3c2nsn3 HTS13866 COc1c(cccn1)NC(=O)c2cccc3c2nsn3 HTS13883 CCCCCC1C(CC(N(C1c2ccccc2)C)c3ccccc3)O RJC03605 c1cc(cnc1)c2nc(cs2)c3cc(n(n3)c4ccc(cc4)Cl)N MWP00715 COc1ccccc1NC(=O)N=S2CCN(CC2)C(=O)c3ccc(cc3)Cl KM06141 CSc1nnc(s1)SCc2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl SPB02574 c1cc(ccc1/C=N/NC(=O)CSCC(=O)Nc2ccc(cc2)OC(F)(F)F)Cl KM09125 CN(/C=C/C=C/1\c2ccccc2C(=C1c3ccccc3)c4ccccc4)c5ccccc5 BTB11084 c1ccc(c(c1)C(F)(F)F)NC(=O)/C=C/C(=O)Nc2ccccc2C(F)(F)F CD07699 c1ccc(c(c1)S(=O)(=O)NC23CC4CC(C2)CC(C4)C3)I NRB00633 C1CN(CCN1C(=S)NC2CC3CC2C=C3)C(=S)NC4CC5CC4C=C5 CD04675 c1ccc(cc1)CCNC(=O)c2cccc3c2nsn3 HTS13870 CCOC(=O)Cn1c2c(cc(s2)c3ccccc3)c(=O)n(c1=O)c4ccc(cc4)Cl HTS13126 C[C@H](C(=O)N1CCC(CC1)c2ccccc2OC)N3CCN(CC3)c4ccc(cn4)C(F)(F)F HTS00011 c1cc(ccc1c2cc(cs2)C(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F)Cl MBE00082 c1cc2c(cc1CN3CCN(CC3)C(=O)c4c(ccs4)Cl)OCO2 HTS03251 Cc1c(cccc1Cl)NC(=S)N/N=C/c2ccc(cc2)N(C)C RDR00321 Cc1c(c(c(o1)C)S(=O)(=O)NCc2cccs2)C(=O)O SP01427 COC(=O)c1cscc1Sc2ccc(cc2)Cl KM04847 c1cc(ccc1C(=O)c2cc3c(cc2Br)OCCO3)Cl BTB12948 Cc1ccc(cc1)C(=O)c2cc3c(cc2Br)OCCO3 BTB12951 CC1CN=C(S1)Nc2ccc(cc2)F BTB13009 CCCCCc1ccc(cc1)c2[nH]c(nn2)Sc3ccc(cc3[N+](=O)[O-])C(F)(F)F SPB01209 Cc1nc2ccc(cc2s1)NC(=O)c3cccc4c3nsn4 HTS13854 Cc1c(c(n(n1)C)C)NC(=O)c2cccc3c2nsn3 HTS13856 Cn1ccc(n1)NC(=O)c2cccc3c2nsn3 HTS13857 CCCCc1ccc(c(c1)C)NC(=O)N2CCN(CC2)c3cc(nc4c3cccc4)C HTS01454 CC(C)(C)OC(=O)N1CCCN(CC1)S(=O)(=O)c2ccc3c(c2)CCO3 HTS10678 c1ccc(cc1)CN2CCC(CC2)NC(=O)c3ccccc3 RH01186 Cc1c(c(nc(n1)c2ccccn2)N(C)C)Cl RDR03818 Cc1cc(ccc1NC(=O)c2ccccc2[N+](=O)[O-])Cl PD00342 COc1ccc(cc1)C(=O)NNc2c(cc(cc2[N+](=O)[O-])C(F)(F)F)[N+](=O)[O-] CD03563 c1cc(ccc1C(F)(F)F)S(=O)(=O)Nc2ccc3c(c2)nsn3 HTS13798 COc1cccc2c1c(no2)NC(=O)c3cccc(c3)Cl HTS13799 COc1cc(cc(c1OC)OC)C(=O)OC(Cc2ccccc2)C(F)(F)F SEW03677 Cc1c(c(n(n1)c2ccccc2)N3CCOCC3)[N+](=O)[O-] BTB13490 c1cc(c2c(c1)nsn2)C(=O)Nc3ccc(cc3)n4cccn4 HTS13835 Cc1c(nc(o1)c2ccccc2)CNC(=O)c3cccc4c3nsn4 HTS13842 c1cc(cc(c1)N2CCOCC2)NC(=O)c3cccc4c3nsn4 HTS13846 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)Nc2ccccc2)C CD03114 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)N2CCOCC2)C CD04588 CSc1c(c([nH]n1)NC(=O)c2ccccc2Cl)S(=O)(=O)c3ccc(cc3)Cl KM01223 c1ccc(cc1)NN2C(NN=C2c3cc(cc(c3O)Cl)Cl)NS(=O)(=O)c4ccccc4 CD03630 c1ccc2c(c1)n(c(=O)o2)CCC(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F SPB02699 Cc1c(snn1)c2nc(cs2)/C(=N/OC(=O)c3ccc(cc3)C(F)(F)F)/C SPB03851 c1cc(cc(c1)C#N)COc2ccc(cc2)Cl KM01628 CN(C)n1cccc1/C=C(\C#N)/C(=O)c2cccc(c2)C(F)(F)F KM04616 COc1ccc(cc1)C(=O)Nc2c3c(cccc3OC)on2 HTS13800 Cc1cccc(c1)C(=O)Nc2c3c(cccc3OC)on2 HTS13801 COC(=O)c1cnc(cc1C(F)(F)F)Oc2ccc(cc2)NC(=O)NC(=O)c3ccccc3Cl RF04741 c1cc2c(cc1Br)/C(=N/N)/C(=O)N2 CD00914 c1ccc2c(c1)nc(s2)CNC(=O)c3cccc4c3nsn4 HTS13829 c1cc(c(cc1C(=O)O)OC(F)(F)F)C(=O)O TL00678 Cc1nn(c(=O)o1)c2ccc(cn2)C(F)(F)F RF04815 c1ccc(cc1)COc2ccc(c(c2OCc3ccccc3)CCC#N)Br BTB10144 Cc1nc(cs1)C(=N)NC(=O)c2ccc(cc2)OC(F)(F)F SPB06506 CCCCc1ccc(c(c1)C)N/C=C(\C#N)/C(=O)OC RH00558 Cc1c(nc(s1)c2cnccn2)CC(=O)O HTS05437 Cc1c(c(no1)c2ccc(cc2Cl)Cl)c3csc(n3)Nc4c(cccc4Cl)Cl SPB06642 Cc1c(c(no1)c2ccccc2Cl)C(=O)NC3CCCCC3NC(=O)c4c(onc4c5ccccc5Cl)C DSHS00203 CN(Cc1cc2cccnc2s1)C(=O)c3cccc4c3nsn4 HTS13897 C/C(=N\OCC(=O)Nc1ccc(cc1)Cl)/c2ccc(cc2)Cl KM05929 c1cc(c2c(c1)nsn2)C(=O)NCc3ccc(cc3)c4cccs4 HTS13831 Cc1cc(n(n1)C)CNC(=O)c2cccc3c2nsn3 HTS13832 Cc1c(c(n(n1)C)C)CNC(=O)c2cccc3c2nsn3 HTS13834 CC(C)(C)C1CCN(CC1)C(=O)c2ccc(cc2)n3cccc3 HTS13926 CCOC(=O)C1CCN(CC1)C(=O)c2c(ccs2)Cl HTS06478 c1cc(cc(c1)NC(=O)CCn2cc(ccc2=O)C(F)(F)F)C(F)(F)F SPB06413 c1ccc(cc1)C(=O)CSc2nc3ccccc3c(=O)n2c4ccc(c(c4)Cl)F CD06738 Cc1c(cc(o1)c2cccs2)C(=O)NCCNc3nccc(n3)C(F)(F)F AW00870 c1ccc(cc1)NC(=O)OC2CC3CC4C2C4C3 NRB01900 CN(Cc1cc2ccccc2s1)C(=O)c3cccc4c3nsn4 HTS13898 Cc1c(n2ccccc2n1)CN(C)C(=O)c3cccc4c3nsn4 HTS13899 CN(Cc1cc(on1)c2ccccc2)C(=O)c3cccc4c3nsn4 HTS13900 Cc1nc(no1)c2ccc(cc2)CN(C)C(=O)c3cccc4c3nsn4 HTS13901 Cc1nc(no1)c2cccc(c2)CN(C)C(=O)c3cccc4c3nsn4 HTS13902 Cc1c(nnc(n1)c2ccc(cn2)C(F)(F)F)C SPB06962 c1c(cc(cc1C(F)(F)F)NC(=S)NCCCN2CCOCC2)C(F)(F)F BTB12683 c1cc(c2c(c1)nsn2)C(=O)N3CCN(CC3)c4ccc(cc4)Cl HTS13886 c1cc(cc(c1)Cl)N2CCN(CC2)C(=O)c3cccc4c3nsn4 HTS13888 c1ccc(cc1)C2C(=O)NCCS2 KM03386 c1ccc(cc1)n2cc(c(n2)c3ccc(cc3)Cl)/C=N/NC(=O)CSc4nnc(n4c5ccccc5)c6ccncc6 HTS11951 c1ccc(c(c1)C(=O)Nc2ccsc2C(=O)NN)Cl GK02723 c1c(cc(c2c1COCO2)CSC(=S)N3CCSCC3)Cl CD08190 c1cc(c2c(c1)OCCO2)C(=O)NCC3CCOCC3 HTS13917 c1cc(cc(c1)NC(=O)c2cccc3c2OCCO3)c4cncnc4 HTS13918 CCC(c1ccccc1)C(=O)Nc2ccc(cc2)C(F)(F)F BTB02050 c1ccc(cc1)C(c2ccccc2)C(=O)NNc3c(cncc3Cl)Cl RF01363 C/C(=N\NC(=O)N)/c1cc(cc(c1O)Cl)Cl CD03825 CC(C)(C)OC(=O)N1CCCN(CC1)C(=S)Nc2ccc(cc2Cl)Cl AW00371 c1cc(c(c(c1)Cl)CNC(=O)COCC(=O)O)F PD00484 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3cccc4c3nsn4 KM09924 CCCCCc1ccc(cc1)/C(=N/O)/N BR00034 Cc1ccc(cc1)C(=O)Nc2ccccc2Sc3ccc(cc3[N+](=O)[O-])Cl DSHS00741 CCOC(=O)C1CCCN(C1)C(=O)Nc2c(onc2c3ccccc3)C HTS06915 c1cc(oc1)c2nnc(n2c3ccc4c(c3)OCCO4)SCc5ccc(cc5Cl)Cl SPB08064 c1ccc(c(c1)C(F)(F)F)NC(=S)Nc2ccc(cc2)c3csnn3 SEW00803 CCOC(=O)C1CCCN(C1)S(=O)(=O)c2cccc3c2nsn3 HTS06913 c1cc(cc(c1)C(F)(F)F)C(=O)N2CCN(CC2)c3c(cncc3Cl)Cl SPB06845 c1cc(c(c(c1)Cl)CC(=N)N)Cl.Cl SPB00311 Cc1ccc(c(c1)C)NC(=O)/C(=C/c2ccc[nH]2)/C#N CD01685 CS(=NS(=O)(=O)c1cccc2c1nsn2)(=O)c3ccc(cc3)Cl KM06387 CCO.C/C(=N\OC(=O)Nc1ccc(cc1)Cl)/c2ccc3c(c2)CCO3 KM06623 C/C(=N\O)/c1ccc(c(c1)OC)OC KM06669 Cc1ccc(cc1)S(=O)(=O)N/N=C/c2ccc(cc2)[N+](=O)[O-] BTB02168 CCOC(=O)c1c(nn(c1C)c2ccc(cc2)NC(=O)c3ccccc3C(=O)O)C SEW04180 c1cc(sc1c2cc(on2)C(F)(F)F)S(=O)(=O)N3CCN(CC3)c4c(cc(cn4)C(F)(F)F)Cl SP01062 CCOC(=O)Cc1c2ccccc2c(=O)n(n1)Cc3nc(cs3)C(=O)OCC KM07148 COc1ccc(cc1OC)S(=O)(=O)Nc2ccc(cc2)S(=O)(=O)Nc3ccccc3Oc4ccc(cc4Cl)Cl RJF01717 C1CC1Cn2nc(nn2)N3CCOCC3 RJF01779 CCCNC(=O)NNC(=O)C(C)n1nc(nn1)N2CCOCC2 RJF01832 CCNc1c2c3c(sc2nc(n1)SCc4ccc(cc4)[N+](=O)[O-])CN(CC3)C HTS13525 c1cc(ccc1NC(=O)CN2CCCC2)S(=O)(=O)N HTS13517 COc1cc(cc(c1OC)OC)c2[nH]c(c(n2)c3ccccc3)c4ccccc4 HTS13443 c1ccc(c(c1)C(F)(F)F)NC(=O)/C=C/C(=O)O S07824 Cc1c(c(no1)c2ccccc2Cl)C(=O)O/N=C/3\CCCCN3 CD03092 c1ccc(cc1)Oc2c(cccn2)c3nnc(n3c4cc(cc(c4)C(F)(F)F)C(F)(F)F)S BTB03072 COc1ccc(cc1)C(=O)N/N=C/c2cccn2c3ccc(cc3)Cl SEW05652 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NN(C)c3ccc(cn3)[N+](=O)[O-] CD06958 c1ccc(c(c1)Cn2c3c(c(ncn3)SCc4ccc(cc4)[N+](=O)[O-])nn2)Cl HTS12155 CC(C(=O)NNC(=O)C1CC1)n2nc(nn2)N3CCOCC3 RJF01848 COc1cc(ccc1OCc2ccccc2)/C=N/C3CCCCCCCCCCC3 S00616 COC(=O)c1cc(c(nc1)Sc2nnc(n2c3cccc(c3)C(F)(F)F)O)[N+](=O)[O-] SPB07446 CC(=O)N/C(=C\c1ccc(cc1)OC(F)F)/C(=O)O SPB08023 CC(=O)N[C@@H](Cc1cccc(c1OC)OCC2CCCC2)C(=O)O SPB08031 CC(C)(C)c1ccc(cc1)C(=O)N/N=C/c2cc(cc(c2O)Cl)Cl BTB03791 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)Oc3c(cc(cc3Cl)Cl)C(=O)C BTB04936 c1ccc2c(c1)c\3c([nH]2)CCC/C3=N\OC(=O)c4c(cccc4Cl)Cl BTB13760 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)NNC(=S)Nc2cccc(c2)OC CD01990 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)Nc3ccc(cc3)Cl)Cl GK03154 Cn1c(=O)cc(c2c1n(c(=O)n(c2=O)C)C)N3CCOCC3 RJC03102 COc1ccc(cc1)S(=O)(=O)C2CS(=O)(=O)CC2O SEW03550 CCOC(=O)N/N=C/c1csnn1 SEW05521 CCOC(=O)c1c(nc(s1)c2csc(n2)C)C SPB03494 CC(=O)/C(=N/Nc1ccc(cc1)Cl)/C(=O)c2ccccc2 SPB04009 c1cc2cc([nH]c2c(c1)[N+](=O)[O-])C(=O)O KM09181 CCOC(=O)CCc1nc(no1)c2ccc(cc2)Cl BTB02283 c1ccc(cc1)CCNC(=S)NNC(=O)CCc2nc(no2)c3ccc(cc3)Cl BTB02323 c1ccc(cc1)n2c(c(c(n2)/C(=C/c3ccc4c(c3)OCO4)/C#N)C#N)n5cccc5 BTB02390 CC1N=C(NO1)c2ccc(cc2)Cl BTB02406 C/C(=C\C(=O)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F)/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F BTB03190 CC(=O)Nc1ccccc1OCCN(Cc2ccccc2)C(=O)c3ccc(cc3)Cl S14200 c1ccc-2c(c1)Cc3c2c(ccc3)C(=O)Nc4nccs4 RJC03563 c1cc(ccc1CSc2[nH]c3cc(c(cc3n2)Cl)Cl)OC(F)(F)F HTS08202 CC(C)(C)c1ccc(cc1)C(=O)Oc2c(c(sc2C(=O)OC)Br)Br GK01954 Cn1c(nnc1S)CCN(Cc2ccco2)S(=O)(=O)c3ccc(cc3)Cl KM09435 CSC1=N/C(=C\Nc2cccc(c2)Cl)/C(=O)N1Cc3cccc(c3)Cl RF03496 CCOC(=O)/C(=C/NCCc1c[nH]c2c1cccc2)/C#N BTB03644 c1cc2c(c(c1)F)c(=O)oc(n2)c3ccco3 BTB04367 COc1ccc(cc1)/C=C(\C#N)/c2ccccn2 PD00097 Cc1c(sc(n1)c2cccs2)c3ccnc(n3)SCC(=O)Nc4ccc(cc4)C(C)C SPB02652 CN(Cc1ccnc(c1)N2CCOCC2)C(=O)c3cccc4c3nsn4 HTS13903 CC(C)(C)C(=O)NC(=S)Nc1cc(cc(c1)C(F)(F)F)C(F)(F)F NH00479 Cc1ccc(cc1)NC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F SP00941 CC(=O)Nc1ccc(cc1Cl)S(=O)(=O)NCCN2CCNC2=O HTS02490 CCOC(=O)/C(=C/c1cn(nc1C)c2ccccc2)/C#N HTS09958 CCOC(=O)C(Cc1cc(cc2c1OCOC2)F)(C(=O)OCC)NC(=O)C HTS11147 Cc1ccc(cc1C)NC(=S)NNC(=O)CSc2nnc(n2c3ccccc3)c4ccccc4OC RH01157 c1ccc2c(c1)c(c(s2)C(=O)N(CCC#N)Cc3ccncc3)Cl BTB00316 c1ccc(cc1)C(=O)NC2CCN(CC2)C(=O)c3cc(oc3C(F)(F)F)c4ccc(cc4)Cl HTS02394 CN1CCN(CC1)c2ccc(cc2)CNC(=O)c3csc4c3cccc4 SCR00779 CN(Cc1ccc(cc1)c2ccsc2)C(=O)c3cccc4c3nsn4 HTS13905 c1ccc(cc1)c2nc(sn2)N3CCN(CC3)C(=O)c4cccc5c4nsn5 HTS13906 Cc1cc(n(c(=O)c1C#N)/N=c\2/n(cc(s2)c3ccccc3)C4CC5CC4C=C5)C SCR00168 c1cc(ncc1C(F)(F)F)N2CCCN(CC2)C(=O)CCN3CCN(CC3)c4nccc(n4)C(F)(F)F AW00936 CC(C)(C(=O)Nc1ccc2c(c1)nccn2)Oc3ccc(cc3)Cl SCR01274 Cn1c(nnc1SCc2nc(no2)c3ccc(cc3)OC)C(F)(F)F SPB00249 c1c(cc(c2c1nc(cc2N3CCCCCCC3)C(F)(F)F)Cl)Cl KM10695 Cc1cc(cc(c1)n2c(c(c(n2)c3cc(oc3C)C(C)(C)C)C#N)SC)C SP00989 CN1CCN(CC1)S(=O)(=O)c2ccc(s2)c3cc(on3)C(F)(F)F SP01083 Cc1cccc(c1)Cn2c(cc(n2)C(C)(C)C)C(=O)O SPB08112 c1cc(c(c(c1)Cl)CS(=O)(=O)c2cccs2)Cl KM02863 CC(C)S(=O)(=O)c1csc(c1Cl)C(=O)NNC(=O)Nc2ccccc2 KM02438 c1ccc2c(c1)cccc2CSCc3nnc(n3C4CCCCC4)S RH01679 Cc1cccc(c1)NC(=O)c2cc(n(n2)Cc3c(cccc3Cl)Cl)C SPB07782 c1ccc2c(c1)c3c(c(=O)o2)C(C(=C(O3)N)C#N)c4cccs4 HTS09876 Cc1ccc(cc1)c2cc(cc(c2C(=O)c3ccccc3)C)c4ccccc4 NRB03292 COc1ccccc1C2CCN(CC2)C(=O)CSCc3cccc4c3cccc4 RH01613 c1ccc2c(c1)c(cn(c2=O)Nc3ccc(cc3)Br)Br NRB04060 Cc1cccc(c1)c2nc(on2)c3c(noc3C)C SP00839 CC1(CCC(=O)/C(=C\c2ccc(s2)Cl)/C1=O)C SEW04031 Cc1ccc(cc1)S(=O)(=O)NC(=O)N2CCN(CC2)Cc3ccccc3 HTS02786 c1cc(ccc1C(F)(F)F)S(=O)(=O)NCCNC(=O)N2CCOCC2 RDR03015 CC(=O)Nc1ccc(cc1Br)F BTB04571 CC(C)(C)c1ccc(cc1)NC(=S)Nc2ccccn2 BTB04723 Cc1cc2nnc(c(n2n1)C)C(=O)NN KM01117 Cc1c(c(n(n1)CC(=O)NNC(=S)NC)C)Br KM02936 CCOC(=O)c1c(nsc1NC(=O)Oc2ccccc2)C KM04199 Cc1ccc(cc1)S(=O)(=O)/C(=C/c2c([nH]c(c2C(=O)OC)C)C)/C#N KM08864 c1c(cc(c-2c1C(=O)c3c2c(cc(c3)[N+](=O)[O-])[N+](=O)[O-])[N+](=O)[O-])[N+](=O)[O-] JFD03647 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)NC(C)(C)CO CD06800 c1cc(cc(c1)NC(=S)C(C#N)C(=O)N2CCCC2)C(F)(F)F DP00468 c1ccc2c(c1)CC(C2)NCC(COc3ccc(cc3)F)O HTS00716 Cn1c2ccccc2c(n1)NC(=O)C3CCC3C(=O)O HTS00765 COC(=O)/C=C(\C(=O)OC)/Nc1ccc(c(c1)Cl)Cl BTB05400 Cc1ccc(cc1)C(=O)/C=C/Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F NRB05044 c1ccc2c(c1)CC(C2)NS(=O)(=O)c3ccc(cc3)c4csnn4 HTS08628 CC1C2=C(CC(CC2=O)(C)C)OC3=C1C(=O)CC(C3)(C)C RJC02776 Cc1cc(ccc1/N=C/c2ccc(cc2)c3ccccc3)Br S00608 CC1=C(C(C2=C(N1)CC(CC2=O)c3ccc(cc3)F)c4c[nH]nc4c5ccccc5)C(=O)OC HTS05053 Cc1ccc(cc1)c2c(cn(n2)c3ccccc3)/C=N/n4c(n[nH]c4=S)c5ccncc5 HTS11972 CC1=N/C(=C/c2ccc(c(c2)Br)OC)/C(=O)O1 PHG00467 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NC(=S)Nc3ccccc3F RJF01490 Cc1cc(c(cc1C)Nc2nnc(s2)SCC(=O)c3ccccc3)C S05129 Cc1c(=O)nc2n(n1)c(=O)/c(=C/c3ccc(cc3)OCc4ccccc4)/s2 HTS13411 Cc1c(c(on1)C)S(=O)(=O)Nc2ccc(cc2)c3cn4c(n3)SCC4 HTS05747 Cc1c(c(nn1C)/C=C/N(C)C)[N+](=O)[O-] CD09679 CCOC(=O)C1=C(OCC1=O)Nc2ccc(cc2)OC(F)(F)F KM08749 CCc1cc2c(cc1c3csc(n3)C)C(CCC2(C)C)(C)C SEW06176 c1ccc(cc1)S(=O)(=O)c2cc(sc2)S(=O)(=O)N3CCN(CC3)C(=O)C4CCCO4 HTS10892 COC(=O)c1ccc2c(c1)nsn2 RDP00063 c1cc(cc(c1)Cl)NC(=O)c2c(c3c(c4c(nc3s2)CCC4)c5cccnc5)N SPB07098 CC(C)c1ccc(cc1)NC(=S)N(Cc2ccccc2)C(C)C S06126 Cc1ccc(cc1)S(=O)(=O)Nc2ccc3c(cc(=O)oc3c2)COC RJF01162 c1cc(cnc1)NC(=S)N2CCCN(CC2)c3c(cc(cn3)C(F)(F)F)Cl AW00192 c1ccc2c(c1)cnn(c2=O)CCOC(=O)c3ccc4c(c3)CCO4 HTS03026 CC1CCN(CC1)C(=O)CN2C(=O)c3ccccc3C2=O SCR00939 CCn1c(nnc1SCC(=O)Nc2ccc(cc2)S(=O)(=O)N)c3ccco3 HTS13512 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC)OC(=O)C)OC(=O)C)O[C@@H]2[C@@H]([C@H]([C@@H]([C@H](O2)COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD00303 Cc1cc(n(n1)C)N2C(=O)c3ccccc3C2=O HTS04718 c1cc(oc1)c2cc([nH]c(=O)c2C#N)c3ccco3 HTS10308 Cc1csc2c1c(c(s2)/C=N/C(=C(/C#N)\N)/C#N)C KM04716 Cc1cccc(c1NC(=O)N2CCCN(CC2)c3nc4ccc(cc4s3)Cl)Cl AW00332 c1cc(c(c(c1)Cl)CSc2nnc(o2)c3ccco3)F AW00540 c1c(cnc(c1Cl)NCCCN2C(=O)CC3(C2=O)CCCC3)C(F)(F)F AW00906 c1ccc2c(c1)cccc2CN3CCCN(CC3)C(=O)c4cccs4 AW00976 c1ccc(cc1)S(=O)(=O)/C(=N/O)/C#N KM01354 COC(=O)C(Cc1c[nH]c2c1cccc2)NS(=O)(=O)c3ccccc3C(F)(F)F RH01618 c1cc(ccc1c2nnco2)Oc3ccc(cc3[N+](=O)[O-])C(F)(F)F SEW04607 Cc1c(sc(n1)c2cccc(c2)n3cccc3)C(=O)NN SPB02296 Cn1c(nnc1SCC(=O)Nc2cccc(c2)Cl)c3ccc(nc3)OCC(F)(F)F SPB06609 Cc1cc(c(cc1Cl)Cl)S(=O)(=O)NCc2c(cccc2N(C)C)N(C)C CD09727 c1ccc(cc1)c2c(n3ccsc3n2)Sc4ccccc4 RJC03562 Cc1c2c(n(n1)c3ccccc3)NC4=C(C2c5ccc(cc5)OCc6ccccc6)C(=O)CC(C4)(C)C HTS12051 CCOC(=O)c1c-2c(c(s1)SC(C)C)S(=O)(=O)N(c3c2cccc3)C KM03303 Cc1cc(c(o1)C)S(=O)(=O)NCC2CCN(CC2)C(=O)OC(C)(C)C SCR01340 CN(C)/C=C/C(=N)SCc1c(cccc1Cl)F.Cl CD11190 CS(=NC(=O)c1ccc(cc1)C(F)(F)F)(=O)c2ccccc2 KM02838 Cc1cc(ccc1Br)NCn2c(=O)c3ccccc3cn2 PD00563 CC(=O)N1c2ccccc2CC1S(=O)(=O)[O-].[Na+] RH00719 CN([C@H]1CCN2CCc3ccccc3C2C1)S(=O)(=O)C RH01707 c1ccc(cc1)C(=O)C2=NNCC2c3cccc4c3cccc4 RJC01653 c1ccc(cc1)c2nc3ccccc3c(=O)n2c4cc(cc(c4)C(F)(F)F)C(F)(F)F DP01611 c1ccc2c(c1)C/C(=N\OC(=O)c3cccs3)/C2=O PD00173 COc1ccccc1CCNC(=O)c2c(nccn2)C(=O)O HTS03734 c1ccc(cc1)c2csc3c2c(ncn3)NCCNC(=O)c4cccs4 AW01019 c1ccc(c(c1)NC(=S)N(Cc2ccc3c(c2)OCO3)c4ccc(cc4)F)Cl BTB01040 COc1cc(cc(c1OC)OC)C(=O)Nc2ccc(cc2)F BTB01248 c1cc2c(cc1CCC(=O)O)OCO2 BTB02068 CN(C)c1ccc(cc1)CC(C#N)c2ccc(cc2)NC(=O)c3c(cccc3OC)OC BTB02179 c1cc(ccc1C(=O)Cn2ccc(n2)C(F)(F)F)Cl HAN00222 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])N2CCCCCC2 S05655 c1ccc(cc1)C/N=C(\c2ccco2)/n3c(=S)nc(n(c3=S)Cc4ccccc4)c5ccco5 BTB14967 CCNc1c(nc2cc(ccc2n1)Cl)NCC RH01327 c1cnc(nc1C(F)(F)F)N2CCCN(CC2)C(=O)CSCC(=O)O HTS02699 CS/C(=C(/C#N)\C(=O)c1cc(c(s1)C(F)(F)F)c2ccccc2)/Nc3ccc(cc3)Cl SEW03446 Cc1ccc(cc1)Sc2ccc(cn2)NC(=O)Nc3ccc(cc3)OC(F)(F)F BTB08354 Cn1c2c3cccc(c3nc(c2c(=O)n1Cc4ccccc4Cl)SC)Cl KM08965 c1ccc(cc1)N\2C(=CS/C2=C(/C#N)\c3[nH]c4ccccc4n3)c5ccc(cc5)Cl HTS07517 CC(=O)Nc1cccc(c1)n2nc(nn2)SCC(=O)Nc3ccc(c(c3)Cl)F HTS02142 c1cc2c(cc(nc2c(c1)Br)C(F)(F)F)Oc3ccc(cc3Cl)F KM07486 c1cc(cnc1)c2c(non2)/N=C\NO SPB04559 Cc1cccc(c1)NC(=S)N2CCC(CC2)c3ccccc3OC RH01414 Cc1ccc(cc1)Sc2ccccc2/N=C/c3c(cccc3Cl)F S06343 c1cc(ccc1Oc2ccc(cn2)C(=O)NN)Cl SPB03944 CC(C(=O)Nc1nccs1)Oc2ccc(cc2Cl)Cl RDR02227 CCC1C(NC(C(C1=O)CC)c2ccccc2)c3ccccc3 RJC03633 Cc1ccc(c(c1)C)N2C(=O)CC(C2=O)N3CCSCC3 S12380 Cc1c(nn(n1)c2ccccc2)CNC(=O)C3CC3 SCR01448 CC1(C/C(=N\Nc2cc(cc(c2)C(F)(F)F)C(F)(F)F)/c3cc(c(c(c3O1)O)O)C(C)(C)C)C SEW02683 CCOC(=O)c1c(nc(s1)c2c(ccs2)CSc3ccc(cc3)Cl)C SEW01704 C/C(=N\Nc1ccc(cc1F)F)/c2ccc(o2)c3ccsc3C(=O)OC SEW01859 CN(C)c1c(cc(cc1F)C(=O)NC(=O)Nc2nnc(s2)C(F)(F)F)F SEW01894 c1cc(ccc1/C=C\2/CSc3c(ccs3)C2=O)C(F)(F)F SEW02095 CCOC(=O)c1c[nH]c(n1)SCc2ccccc2 HTS13933 CC(=O)C(C#N)c1nc(cs1)c2ccc(cc2)F CD09157 CCc1cnc(nc1c2c(cccc2F)F)NS(=O)(=O)c3cc(sc3Cl)Cl CD09844 CC(=O)N1CCC(CC1)C(=O)O CD09938 Cc1csc2c1c(ncn2)Sc3ccc(cc3)Cl GK01666 COC(=O)c1c(cc(s1)c2cccs2)NS(=O)(=O)c3ccc(cc3)Cl GK03703 COC(=O)c1c(c(cs1)S(=O)(=O)Cc2ccco2)N KM03329 Cc1c(c(sc1c2nc(cs2)c3ccc(cc3)Cl)SC)C(=O)C KM04586 c1cc(ccc1c2cc(n(n2)c3ccc(cc3)Cl)N)OC(F)(F)F KM04940 Cc1c(c(no1)c2ccccc2)C(=O)NC3CCS(=O)(=O)C3 HTS02850 CCOC(=O)C(Cc1cc(c(c(c1)I)Oc2ccc(cc2)OC)I)NC(=O)C KM08406 c1ccc(cc1)S(=O)(=O)CCN2CCC(CC2)n3cccc3 KM08638 c1ccc(cc1)C(=O)OCC#Cc2ccc(cc2)C#N KM09059 c1cc(oc1)C(=O)NNC(=O)c2cc3cc(ccc3[nH]2)OC(F)(F)F KM09385 c1cc(cc(c1)NC(=O)Nc2ccc3c(c2)non3)C(F)(F)F KM09750 CC1(Cc2cccc(c2O1)C(=O)NCC3COc4ccccc4O3)C SCR00517 Cc1c(nn(n1)c2ccccc2)CNC(=O)c3cc(cc4c3OCOC4)F SCR00560 Cc1csc2c1ncnc2SCC(C(F)(F)F)O SCR00932 CCOC(=O)c1c[nH]c(n1)SCc2ccccc2Cl HTS13934 CC(C)(C)c1cc(n(n1)S(=O)(=O)c2ccc(cc2)Cl)SC CD10660 CC(C)NC(=S)Nc1cccc(c1)C(=O)OC DFP00328 c1cc(ccc1CSC2=NCCCN2C3CCCCC3)C#N.Br DP01449 c1ccc(cc1)N2C(=O)C(=Cc3ccco3)C(=O)N(C2=S)c4ccccc4 JFD01809 COCn1c2ccccc2nn1 JFD02338 CC1(C2CCC1(C(=O)NC2=O)C)C JFD02360 c1ccc(cc1)Oc2ccsc2/C=C(\C#N)/C(=O)c3cccs3 KM05515 c1ccc(cc1)CN2CCC(CC2)NC(=O)C3CCCCC3 RJC03035 c1ccc(cc1)CN2CCN(CC2)S(=O)(=O)c3cc(cc(c3)C(F)(F)F)C(F)(F)F RJC03074 CC(c1ccccc1)NC2CCCCC2.Cl RJC04065 Cc1c(c([nH]n1)N/N=C/c2ccccc2Cl)C(=O)O RJC04088 c1cc(cnc1)C2N(C(=O)CS2)c3ccc(cc3)Cl S06685 Cc1cc(ccc1NC(=O)c2ccc(cc2)C(C)(C)C)F S06992 c1ccc2c(c1)cc3ccccc3c2/C=C/[N+](=O)[O-] S09756 c1cc(cnc1)C2N(C(=O)CS2)c3ccc(cc3)C(F)(F)F S11740 Cc1ccccc1/C=C(\C#N)/C(=O)OC S12945 c1ccc2c(c1)C(=O)C(=Cc3ccc(cc3)C(F)(F)F)C2=O S12972 c1cc(cc(c1)Cl)NC(=O)C(Cl)Cl CD04825 c1ccc2c(c1)/C(=C\c3ccc(o3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F)/C(=O)N2 CD04872 c1ccc2c(c1)c(nc3n2nnc3c4ccc(cc4)[N+](=O)[O-])N CD05127 Cc1c(nnn1c2cc(cc(c2)C(F)(F)F)C(F)(F)F)C(=O)C CD05142 c1cc(c(c(c1)Cl)CSc2nnc(s2)SCc3c(cccc3Cl)F)F CD05576 c1ccc2c(c1)cccc2CC3=NCCN3.Cl JFD03925 Cc1ccc(cc1)c2cncnc2NC(=O)c3ccccc3 JM00055 CC(C)(C)C(=O)Nc1ccccc1Sc2ccc(cc2[N+](=O)[O-])C(F)(F)F JP00517 COc1cccc(c1)/C=C\2/C(Oc3ccccc3C2=O)c4ccccc4 RJC00157 c1ccc(cc1)C2CC(=Nc3ccccc3N2)c4ccc(cc4)OCC(=O)N RJC00377 c1ccc(c(c1)COC(=O)c2cc(cc(c2)[N+](=O)[O-])[N+](=O)[O-])Br RJC00417 c1cc(cc(c1)Cl)Nc2ncnc(n2)N RJF00707 COC(=O)c1cc(ccc1SCc2ccc(cc2)Cl)[N+](=O)[O-] RJF01608 Cc1c(sc2n1nc(n2)c3ccc(cc3)Cl)C(=O)N4CCCCC4 SPB05505 CC(C)(C)NC(=S)N/N=C/c1c(cc(cn1)C(F)(F)F)Sc2ccc(cc2)Cl SPB06009 c1cc(c(cc1Cl)Cl)C(=O)Cn2cc(ccc2=O)C(F)(F)F SPB06467 COc1cc(cc(c1OC)OC)c2cc3c4ccccc4oc(=O)c3c(c2C#N)N HTS13321 Cc1cc(nc2c1c3c(s2)C(=O)N(CC(=O)N3)c4ccc(cc4)Cl)C HTS13364 c1ccc(cc1)C(=O)CSc2c3c4c(sc3nc(n2)SCC(=O)c5ccccc5)CCC4 HTS13502 C([C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)NC(=O)N)O)O)O)O JFD00295 CN(C)C(=O)Sc1c(n[nH]c1SC)c2ccc(cc2)Cl RF04998 CC(C)CCNC(=O)c1cc(cc2c1-c3ccc(cc3C2=O)[N+](=O)[O-])[N+](=O)[O-] RJC01706 Cc1c(sc(n1)c2ccc(cc2)C(F)(F)F)C(=O)Sc3ccc(cc3)C(F)(F)F SPB03049 CC(=O)c1csc(n1)CS(=O)(=O)c2ccc(cc2)Cl SPB03549 c1cc(c(nc1)SC(=O)c2ccc(cc2)Cl)C(F)(F)F SPB03691 CC(C)(C)C(=O)N1CCN(CC1)Cc2ccc3c(c2)OCO3 SPB07284 CCOC(=O)c1c[nH]c(n1)SCc2ccc(cc2)C HTS13931 CCOC(=O)C(C(F)(F)F)(Nc1ccccc1C)NC(=O)c2cccc(c2)Cl BTB13578 CC(C)(C)NC(=O)NCC1CCCC1NC(=O)NC(C)(C)C CD00718 c1ccc(cc1)C(C[N+](=O)[O-])C2c3ccccc3NC2=O HTS10086 CC(C)(CC(=O)N1CCN(CC1)c2ncccn2)CC(=O)O HTS10742 c1ccc(cc1)C2=NOC(C2)CNC(=S)NCc3ccco3 HTS11170 c1ccc2c(c1)/C(=N/c3cccc(c3)C(F)(F)F)/C(=O)N2 HTS12040 Cc1cc(ccc1NC(=S)Nc2cccc(c2)NC(=O)c3ccccc3O)Br RDR01513 CCOC(=O)C1=C(N(C(=O)C1)c2ccccc2)C RH00187 c1ccc2c(c1)-c3c4c(cccc4n[nH]3)C2=O RH00237 c1ccc(cc1)n2c3ccccc3c4c(c2=O)c(cc(=O)o4)O RH00499 CCCCc1ccc(c(c1)C)NC(=O)CSc2nnc(s2)NC(=O)c3cccs3 RH00565 c1cc(c(cc1Cl)Cl)OCC(=O)N SPB00368 CC(/C(=N/OC(=O)c1ccc(cc1)C(C)(C)C)/N)Oc2ccc(cc2Cl)Cl SPB00395 c1cc(c(c(c1)Cl)CS(=O)(=O)c2ccc(cn2)C(F)(F)F)Cl SPB03863 c1ccc(cc1)C(=O)c2c(=O)ccn(n2)c3ccc(cc3)C(F)(F)F SPB04030 c1ccc2c(c1)n(c(=O)o2)CCC(=O)NCCN3CCCCC3 SPB08417 CCOC(=O)/C(=C/Nc1ccc(nc1)Oc2cc(cnc2)Cl)/C#N BTB07786 c1ccnc(c1)NC(C(F)(F)F)(C(F)(F)F)NC(=O)c2cccnc2 BTB14289 CN1CCN(C(C1)CN(C)S(=O)(=O)c2ccc(cc2)Cl)C MO08512 COC(=O)CNC(=O)c1cccnc1SC BTB08721 Cc1ccc(cc1)S(=O)(=O)N(CC=C)c2ccccc2C3=N/C(=C\c4ccccc4Cl)/C(=O)O3 BTB08799 COC(=O)C(=C(SC)SC)C(=O)OC BTB08894 Cc1nc(c(c(n1)SC)C#N)Nc2cccc(c2)C(F)(F)F BTB08946 c1ccc(cc1)C2=NN(C(C2)c3cccc4c3cccc4)c5ccccc5 BTB13679 CN1C2C[C@@H](CC1CC2)NC(=O)CSc3ccc(cc3)Cl BTB14843 CSC(=S)OCC12CC3CC(C1)CC(C3)C2 BTB15001 c1ccc(cc1)c2cc3[nH]c4c(c(=O)n3n2)CN(C4=O)Cc5ccco5 HTS08101 CCc1cc(c(s1)NC(=O)COc2ccc(cc2Cl)Cl)C(=O)c3ccc(cc3)OC HTS08124 CC1(CC2=C(C(c3c(=O)[nH]c(nc3N2)SC)c4ccc(cc4)OCc5ccccc5)C(=O)C1)C HTS12055 COc1cc(c(cc1Cl)OC)n2c(=O)c3ccccc3nc2SCC(=O)c4ccc(cc4)Cl RDR01736 CCOC(=O)c1ccc(cc1)OS(=O)(=O)c2ccc(cc2)NC(=O)C RDR02595 c1cc(ccc1CC(=O)Nc2ccc(cc2)[N+](=O)[O-])[N+](=O)[O-] RF00492 CCOC(=O)C1=C(NC(=O)NC1c2ccc(o2)c3cccc(c3)[N+](=O)[O-])C RF00629 Cc1cc(nn1C)C(=O)NNC(=O)COc2ccc(cc2Cl)Cl SPB00658 C#CCSc1nnc(n1c2cccc(c2)C(F)(F)F)O SPB00733 c1ccnc(c1)SCc2cc(=O)[nH]c(=O)[nH]2 SPB01211 COc1cc2c(c(c1OC)OC)nc(oc2=O)c3cccs3 BTB05478 c1ccn(c1)Cc2c(cccc2Cl)Sc3ccc(cc3)Cl HTS05272 CN1CCN(CC1)Cc2c[nH]nc2c3ccccc3 HTS05673 COc1ccc(cc1)c2c(c[nH]n2)CN3CCN(CC3)c4cc(ccn4)C(F)(F)F HTS05693 c1ccc(c(c1)NC(=O)CSCC(=O)O)SCCS(=O)(=O)c2ccc(cc2)Cl HTS05791 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)c3c(nccn3)C(=O)O)C(F)(F)F HTS08391 c1cc(cc(c1)Oc2ccc(cn2)NC(=O)Nc3ccc(cc3)F)C(F)(F)F HTS08495 c1ccc2c(c1)c(cc(n2)c3cccs3)C(=O)O NRB03637 CC12CCC3C(C1CCC2=O)CCC4=CC(=O)CCC34 NRB03818 CCCCCCCCCCCCSC1CC(=O)N(C1=O)c2cccc(c2)C#C PD00249 COC(=O)c1ccc(cc1)CC(=S)C(c2ccccc2)(c3ccccc3)c4ccccc4 SEW05884 c1cc(ncc1C(F)(F)F)N2CCN(CC2)c3ccc(cn3)[N+](=O)[O-] SEW05961 CC(C)Cc1ccc(cc1)C(C)C(=O)Nc2ccc3c(c2)OCCO3 SEW06240 c1cc(ccc1N2CC(CC2=O)C(=O)O)OC(F)(F)F SEW06291 c1cc(sc1)c2nc(on2)/C=C/c3ccc(cc3)OC(F)(F)F SEW06325 Cc1cc(ccc1Cl)c2cc(nc(n2)N)c3cc(cs3)Br BTB06203 COc1ccc(c(c1)c2nnc(o2)c3ccccc3NS(=O)(=O)c4ccc(cc4)Cl)Br BTB06959 C/C(=N\OC(=O)c1ccc(cc1)Cl)/c2cc[nH]c2 BTB07178 Cc1ccc(c(n1)[N+](=O)[O-])Oc2ccc(cn2)[N+](=O)[O-] BTB07276 Cc1nc(cs1)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3)Cl)NC(=O)C HTS03130 c1cc(ccc1NC(=S)NCCN2CCNC2=O)OC(F)(F)F HTS03380 C1CCNC(=O)C(C1)NC(=O)CCC(=O)O HTS06535 Cc1csc2c1cc(cc2)Cl MWP00002 Cc1c2cc(ccc2sc1c3csc(n3)c4ccc(cc4)Cl)Cl MWP00223 c1cc(cc(c1)[N+](=O)[O-])NC(=O)C(=S)NCc2ccco2 NRB00111 c1cc2c(cc1NCC(=O)NN)OCO2 NRB00206 c1ccc(cc1)c2c(cnn2c3ccccc3)c4nnnn4c5ccc(cc5)Br NRB05137 c1cc(c(cc1F)F)CNS(=O)(=O)c2ccc(s2)c3ccno3 SEW02297 c1cc(sc1)c2ccc(s2)/C=C/C(=O)Oc3ccc(cc3)Cl SEW02644 CSc1ccc(s1)/C=C(\C#N)/S(=O)(=O)c2ccc(cc2Cl)Cl SEW03580 CSc1c(c(nc(n1)c2ccc(cc2)Cl)N)c3ccccc3 EN00095 Cc1cc(nn1C(C)(C)C)C(=O)NNC(=O)c2cc(on2)C HTS00017 COc1ccccc1C2CCN(CC2)C(=O)CSc3nnc(s3)NC(=O)c4ccccc4 HTS00036 Cc1ccc(cc1)C(=O)Cn2cc(nc2C)[N+](=O)[O-] HTS00290 c1ccc2c(c1)CCN(C2)S(=O)(=O)c3cccc4c3nccc4 HTS00639 c1ccc(cc1)COC(=O)N2CCC(CC2)C(=O)Nc3ccc(cc3Cl)N4CCOCC4 HTS03153 CC(C)(C)c1c(c(n(n1)C)C(C)(C)C)NC(=O)c2cccnc2 HTS03453 CCOC(=O)C1CCN(CC1)c2cc(nc3c2cccc3)C(F)(F)F KM09897 C=CCNC(=S)NNC(=O)c1ccc2c(c1)cccn2 KM10575 CSc1nccc(n1)c2ccc(s2)S(=O)(=O)Nc3cc(cc(c3)C(F)(F)F)C(F)(F)F KM10677 c1ccc2c(c1)cc(s2)CNC(=O)CN3C(=O)c4ccccc4C3=O SCR00956 CC(C)NC(=O)c1c(nsc1SC)SC SEW00244 c1cc(ccc1c2cnco2)NC(=O)C3C4CC(C3C(=O)O)C=C4 SEW01188 C/C(=N\Nc1ccccc1)/COc2ccc(cc2)c3csnn3 SEW01198 CC(=O)C(C(=O)C)/N=N/c1ccc2c(c1)COCO2 SEW03675 CCOC(=O)c1c[nH]c(n1)SCc2ccc(cc2)F HTS13935 c1cc(ccc1C(=O)N)C(=N)NS(=O)(=O)c2cc(cc(c2)C(F)(F)F)C(F)(F)F CD09001 CNc1ccccc1C(=O)NNC(=O)c2ccccc2Cl DP01966 COc1cc(cc(c1OC)OC)C2C3C(=NN2)C4CCN3CC4 DSHS00388 c1cc(c(cc1/C=C/2\C(=O)C3CCN2CC3)Cl)Cl DSHS00405 c1ccc2c(c1)c(=O)n(c(n2)SCC(=O)N3CCOCC3)c4ccc(c(c4)Cl)Cl HTS00684 Cc1ccc(cc1Cl)c2c(sc(n2)NC(=O)C3CC3)C HTS00995 c1cc2c(cc1C(=O)CN3CCN(CC3)c4ccc(cn4)C(F)(F)F)OCCO2 HTS01190 Cn1c(ccc1S(=O)(=O)NCCNc2cccc(n2)C(F)(F)F)C(=O)OC HTS01545 CC(c1ccn(n1)S(=O)(=O)c2ccc(cc2)Cl)SC KM07768 CCc1ccc2c(c1)cc([nH]2)C(=O)Nc3ccccc3C(C)CC KM11023 c1cc(c(cc1F)F)C(=O)NC(=S)N2CCCCC2 MGH00239 c1ccc(cc1)COc2ccc(cc2)NC(=O)/C=C/C(=O)O S14365 c1ccc(cc1)C2=N/C(=C/c3ccc(cc3)C(F)(F)F)/C(=O)S2 S14999 c1ccc(c(c1)N)Sc2cc(cc(c2Sc3ccccc3N)[N+](=O)[O-])C(F)(F)F CD04390 CC1(OC(=O)C(=Cc2c[nH]c3c2cccc3)C(=O)O1)C CD06278 CN(c1cccc(c1C#N)F)NS(=O)(=O)c2ccc(c(c2)Cl)Cl CD07021 CC(C)(C)C(=N)NS(=O)(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F CD07487 COc1ccccc1NC(=S)NCc2ccncc2 DSHS01218 Cc1cc(n(n1)C)NC(=O)c2ccccc2 KM00005 c1cc(c(cc1/N=N/c2c(n[nH]c2N)C3CC3)Cl)Cl KM00400 c1cc(ccc1C2SCCS2)NC(=O)Nc3ccc(cc3)Cl KM00781 c1ccc(c(c1)NS(=O)(=O)c2cccs2)SCCS(=O)(=O)c3ccc(cc3)Cl KM02008 COc1cc(nc2c1cc(cc2)C#CCOC(=O)Nc3ccc(cc3)OC(F)(F)F)C(F)(F)F KM08022 c1ccc(cc1)C#Cc2cc(sc2)/C=N/Nc3c(cc(cc3Cl)Cl)Cl KM08145 COc1ccc(cc1)C(=O)/C(=C/c2ccc(s2)C#Cc3ccccc3)/C#N KM08198 CC(C)(C)S(=O)(=O)/C(=C/N1CCN(CC1)C(c2ccccc2)c3ccccc3)/C#N KM08216 CCCN1CN(C(=S)SC1)CCC S01958 c1ccnc(c1)c2ccccn2 SB01187 c1cc2c(cc1S(=O)(=O)[O-])nc([nH]2)S.[Na+] SB01380 c1cc(cnc1)CN(CCC#N)C(=S)NC2CC3CC2C=C3 CD01839 CCCc1c(ccc(c1O)C(=O)C)OCCCOc2ccc3c(c2)occ(c3=O)c4ccccc4 JFD00308 c1ccc2c(c1)c(c[nH]2)C(c3ccncc3)O JFD00791 CC(=O)NC(C(F)(F)F)(C(F)(F)F)NCc1ccccc1 JFD01037 Cc1c(cccc1Cl)Nc2ccccc2C(=O)O JFD01579 c1cc(ccc1C(CC(=O)O)CC(=O)O)Cl RH00811 C[C@@]1\2CCC(C1)C(/C2=N\OC(=O)c3cccc(c3)C(F)(F)F)(C)C RJC01963 c1ccc(cc1)NC2CS(=O)(=O)C=C2 RJC02397 CCOC(=O)NC(C(F)(F)F)(C(F)(F)F)Nc1ccc(cc1)C(=O)C RJC02602 COc1ccc(cc1)C(=O)NC(C(F)(F)F)(C(F)(F)F)Nc2ccc(c(c2)Cl)Cl RJC02688 c1ccc2c(c1)C3c4ccccc4C2C5C3C(=O)C=CC5=O RJC02958 CC(C)c1cccc(c1NC(=S)Nc2cccc(c2)C(F)(F)F)C(C)C S04430 Cc1cc(ccc1F)NC(=S)NNC S05503 c1ccc(cc1)C(=O)CCCCCCCC(=O)O XBX00047 CON1C(=O)c2ccccc2C1=O XBX00238 Cc1c(c(c(c(c1C)C)CSc2nc3ccccc3s2)C)C CD02173 CC(=O)c1ccccc1OC(=O)C CD02515 COc1cccc(c1C(=O)Nc2ccccc2NC(=O)c3c(cccc3OC)OC)OC CD03969 CCOC(=O)N1CCc2c(sc(c2C#N)NC(=O)CN3CCOCC3)C1 HTS12784 COc1cccc(c1)n2cc([nH]c2=S)c3ccc(cc3)F HTS13082 CCC1c2c(c3ccccc3[nH]2)CCN1C(=O)c4ccc(cc4)Cl RH01287 C/C(=N\O)/CCc1ccc(c(c1)OC)OCc2ccc(c(c2)Cl)Cl RH01446 Cc1ccc(cc1)Sc2c(cccn2)n3cccc3 RH02119 c1ccc(cc1)c2csc(n2)CS(=O)(=O)c3ccc(cc3)Cl SPB01728 COC(c1ccc(c(n1)S)C#N)OC SPB04265 CCOC(=O)c1c(sc(n1)c2ccccc2)C(=O)/C=C/N(C)C SPB04631 CC(C)c1ccc(cc1)NC(=O)CSc2nccc(n2)c3cc(no3)c4ccc(cc4Cl)Cl SPB05073 Cc1cc(nc(c1[N+](=O)[O-])C)C XBX00240 Cc1cc(c(c(c1)/N=N\c2ccc(cc2[N+](=O)[O-])Cl)O)C XBX00328 CCOC(=O)/C(=C/C(=O)c1ccc2cc3ccccc3cc2c1)/O BTB12161 CCOC(=O)C12CCC(CC1)NC2=O BTBG00041 c1ccc(cc1)Oc2ccc(cn2)C(=O)O CC19601 Cc1c(snn1)c2nnc(o2)c3ccccc3C(F)(F)F HTS08717 CCN(CC)CC(=O)Nc1c(cc(s1)c2ccccc2)C(=O)OCC HTS13141 c1ccc(cc1)C(=O)N/C(=C\c2ccco2)/C(=O)N/N=C/c3ccc(cc3)F HTS13207 c1cc(sc1)c2[nH]c(nn2)SCC(=O)O HTS13296 CC(C)(C)c1cc(nn1c2ccccc2)C(=O)O RF01159 Cc1c(c(no1)c2c(cccc2Cl)Cl)NC(=O)O/N=C/c3cccc(c3)[N+](=O)[O-] RF01313 CC(C)(C)c1ccc(cc1)OCC(=S)N SPB02074 CSc1nnc(s1)SCc2nc(cs2)c3ccc(cc3)Cl SPB02227 Cc1cc(n2c(n1)nc(n2)SCC(=O)Nc3ccc(cc3)Cl)C SPB02423 CC1(CCc2c1cc(cc2C3=NNC(C3)(C(F)(F)F)O)C(C)(C)C)C KM10714 Cc1cccc(c1)C(=O)c2ccccc2C(=O)O BTB10830 CCCCCCCCCCCOC(=O)c1cc(cc2c1-c3ccc(cc3C2=C(C#N)C#N)[N+](=O)[O-])[N+](=O)[O-] BTB10890 c1cc(ccc1N/N=C(\C#N)/C(=O)N)Cl HTS09025 CC1CC(=O)Nc2ccccc2N1S(=O)(=O)c3ccc(cc3F)F HTS09694 CC1CC(=O)Nc2ccccc2N1C(=O)c3cccs3 HTS09698 Cc1cc(no1)C(=O)Nc2cc(nn2C)c3ccccc3 HTS09747 c1ccc(cc1)c2ccc(cc2)NC(=O)c3ccccc3C(=O)O PD00478 c1ccc(c(c1)/C=C(\C#N)/c2ccc(cc2)[N+](=O)[O-])Cl PHG00044 Cc1cc(nc(n1)N/C=C\2/C(=O)N(C(=N2)SC)Cc3cccc(c3)Cl)C RF03497 CC(C)Nc1cc(c(cn1)C(=O)Nc2ccc(cc2Cl)Cl)C(F)(F)F RF04426 CC(C)(C)NC(=S)N/N=C/c1cc(n(c1)C)C(=O)OC SEW06442 CC(C)Cc1ccc(cc1)C(C)/C(=N/O)/N SEW06537 CCOC(=O)c1cc(n(c1C)CCCN2CCOCC2)C(C)(C)C SP00318 c1ccc(c(c1)OCc2nc(cs2)c3ccc(cc3)C(F)(F)F)Cl SP00652 Cc1c(c(nc(n1)c2ccccn2)N3CCCCC3)Cl HTS13927 Cc1c(c(nc(n1)c2ccccn2)NCc3ccco3)Cl HTS13929 Cc1c(c(nc(n1)c2ccccn2)N3CCc4ccccc4C3)Cl HTS13930 CC(C)(C)c1csc(n1)Cc2ccc(cc2)[N+](=O)[O-].Br BTB05043 c1ccn(c1)c2cc(c(cc2Cl)NS(=O)(=O)c3ccc(cc3)Cl)Oc4ccc(cc4)Cl BTB07559 c1cc(cc(c1)Cl)c2nnc(o2)c3cc(ccc3Oc4cc(cnc4)Cl)[N+](=O)[O-] BTB08053 c1ccc(c(c1)NC(=O)c2ccc(cc2)C#N)Sc3nc4ccc(cc4s3)Cl HTS03934 c1cc(sc1)CN(CCC#N)C(=O)c2c(nccn2)C(=O)O HTS06543 CCN(CC)S(=O)(=O)c1ccc(cc1)c2cc(sc2C(F)(F)F)C(=O)OC HTS07172 Cc1c2c([nH]n1)OC(=C(C2c3ccc(cc3)Cl)C#N)N HTS07493 CCOC(=O)Cn1cnc2c(c1=O)c3c(s2)CC(CC3)C HTS07661 Cc1c(c(ncn1)OCC(=O)Nc2ccc(cc2)F)CC(=O)OC HTS07758 c1cocc1C=C2C(=O)OC3(CCCCC3)OC2=O NRB00396 COc1cc(cc(c1OC)OC)C2=N/C(=C/C=C/c3ccccc3)/C(=O)O2 PHG00776 CCOc1c(c(=O)c1=O)N2CCCCC2 RDP00188 CS(=O)(=O)/C(=C\c1ccc(s1)Cl)/C#N SEW03829 CN(C)/C=C/C(=O)c1ccncc1 SEW04051 Cc1ccc(cc1)S(=O)(=O)NC(=O)NNc2c(cc(cc2Cl)Cl)C(F)(F)F SEW04437 Cn1c2cccc(c2c(n1)NC(=O)c3ccc(o3)CSc4ccc(cc4)Cl)F SP01323 c1cc(cc(c1)O)Nc2ccc(nn2)Nc3cccc(c3)O MO08553 c1cc2c(cc1Cl)c(cs2)CO CC00123 Cn1c(nnc1SCC(=O)Nc2ccc(cc2)S(=O)(=O)N)c3ccncc3 HTS13507 CCNc1c2c3c(sc2[nH]c(=S)n1)CN(CC3)C HTS13522 Cc1c(sc(n1)COc2cccc(c2)Cl)c3ccnn3C(=O)C4CC4 SPB02584 CCOC(=O)c1cc2c(ccnc2N(C)C)nc1C(F)(F)F SPB04552 Cc1ccc(cc1)SCc2ccccc2c3[nH]c4ccccc4n3 BTB03603 c1ccc(c(c1)C(=O)OCc2ccc(cc2Cl)Cl)Cl BTB04172 c1ccc(cc1)CS(=O)(=O)CC(=O)Nc2ccc(c(c2)Cl)F BTB04192 COC(=O)C1=C(CSC1)Nc2ccccc2NC(=O)c3c(cccc3Cl)Cl HTS04267 Cc1csc(c1c2nc3ccccc3s2)NC(=O)Nc4ccc(cc4)OCc5ccccc5 HTS04320 CC(C)c1ccc(cc1)NC(=O)CSc2ncccn2 HTS04454 c1cc(c(nc1)NNC(=O)COCC(=O)O)C#N HTS04935 c1cc(cc(c1)Cl)NC(=S)NNC(=O)c2ccncc2 ML00381 CCOC(=O)NN=C1CCCC1 ML00453 Cc1ccc(cc1)Nc2ccc(cc2[N+](=O)[O-])[N+](=O)[O-] NRB00609 c1ccc2c(c1)c(=O)cc(o2)c3ccc(cc3)Cl NRB02678 c1ccc2c(c1)C=CC(=O)C2=NNc3ccc(cc3)Br NRB02969 c1cc(ccc1n2c(nnn2)/C=C/N3CCOCC3)Br NRB03126 CC(C)(C)C(=O)Nc1cccc(c1)c2ncon2 SEW01243 CC(C)(C)c1ccc(cc1)C(=O)c2ccc3c(c2)CCC3 SEW04499 Cc1c(c(nc(n1)c2ccccn2)N3CCN(CC3)C)Cl HTS13928 c1cc(ccc1C(=O)N2CCSC2COc3ccc(cc3)[N+](=O)[O-])Cl FM00280 CCOC(=O)CC(=O)Nc1ccsc1C(=O)N GK00478 Cc1cc(c2cc(ccc2n1)F)Oc3c(cccn3)[N+](=O)[O-] BTB04495 Cc1ccc2c(c1)sc(n2)N BTB04798 CCCc1ccc(cc1)S(=O)(=O)Nc2ccc3c(c2)OCCO3 HTS01872 CC(C)(C)c1ccc(cc1)c2nnc(n2c3ccc4c(c3)OCO4)SCc5cccc(c5)C(=O)N HTS02049 Cc1c(cnn1c2ccc(cc2)Cl)C(=O)NCCSCc3c(cccc3Cl)F HTS02285 Cc1c(c(no1)c2ccccc2)CNC(=O)Nc3ccccc3 SCR00083 Cc1c(sc(n1)c2ccc(s2)c3ccc(s3)C(=O)C)C(=O)C HTS13968 CCOC(=O)CSc1[nH]cc(n1)C(=O)OCC HTS13936 CCOC(=O)c1cc(nc(n1)O)C SPB04779 CC1(C=Cc2cc(c(cc2O1)OCc3ccc(cc3)[N+](=O)[O-])OCc4ccc(cc4)[N+](=O)[O-])C JFD00323 CC(CNc1ccccc1)/C(=N/c2ccccc2)/Nc3ccccc3.Cl RJC01315 C1CCC(=NN=C(N)N)CC1.Cl RJC01501 CO[C@H]1[C@@H]([C@@H]([C@H]2[C@H](O1)COC(O2)c3ccccc3)F)O RJC03737 Cc1ccc(cc1)C(=O)N2CCN(CC2)c3c(cccn3)C(F)(F)F SEW05958 Cc1ccc(cc1)C(=O)Nc2cc(sc2C(=O)N)c3ccccc3 GK03724 CC(=O)c1cc(ccc1SC)[N+](=O)[O-] KM03208 COc1ccc(cc1)/C(=C\c2nccn2C(=O)c3ccc(cc3)OC)/OC(=O)c4ccc(cc4)OC KM09945 CC(=O)Nc1ccc(cc1)S(=O)(=O)Nc2nc(cc(n2)c3ccc(cc3)OC)c4ccc(cc4)OC NRB00358 Cc1ccc(cc1)C(=O)CSc2nnnn2c3cccc(c3)Cl S03378 c1c(ccc(c1)/C=N/c2cc(cc(c2)C(F)(F)F)C(F)(F)F)/C=N/c3cc(cc(c3)C(F)(F)F)C(F)(F)F S06056 c1cc(cc(c1)[N+](=O)[O-])C(=O)Cn2c3c(cccn3)oc2=O SPB06637 c1ccc(c(c1)CSc2nnc(o2)c3ccc(nc3)OCC(F)(F)F)C(F)(F)F SPB06670 Cc1cc(c(c(c1CSC2=NCCN2)C)CSC3=NCCN3)C.Cl.Cl DP01468 CCOC(=O)COc1ccccc1/C=C(/C#N)\S(=O)(=O)c2cccs2 KM05799 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)n2cccc2C=C(C#N)C#N SEW04518 Cc1ccc(cc1)S(=O)(=O)NC(=O)NCc2csc3c2cc(cc3)Cl HTS04216 COc1ccc(cc1)C(=O)Nc2ccc(nc2)Oc3c4ccc(cc4ncn3)Cl HTS07322 COc1ccc(c(c1)S(=O)(=O)NCc2ccc(cc2)S(=O)(=O)N)OC SCR01168 Cn1cnnc1Sc2cc(c(cc2Sc3nncn3C)C#N)C#N JFD02050 Cc1ccc(cc1)c2c(nc(s2)Nc3c(cccc3Cl)Cl)c4ccc(cc4)Cl.Br DP00555 Cc1c2cc(sc2n(n1)C)C(=O)Nc3ccc4c(c3)nccn4 SCR01275 c1ccc(cc1)S(=O)(=O)c2cscc2N KM01765 c1cc(cnc1)c2csc(n2)c3cccnc3 RDR03964 c1cc(sc1)CNc2n[nH]c(=S)s2 S07673 CC(=O)CC(=O)Nc1ccccc1Cl BTB13411 CC(C)(C)SCCNC(=O)c1ccco1 CD08271 COc1ccc(cc1)C(=O)CSc2nnc(n2c3cccc(c3)C(F)(F)F)c4cc(c(c(c4)OC)OC)OC.Br ML00371 CC(C)Nc1nc(cs1)c2c(cccc2Cl)F.Br RF02510 c1cc(cnc1)CNCc2ccc(cc2)Cl.Cl.Cl RF03319 c1cc(ccc1C(F)(F)F)S(=O)(=O)O/N=C(/C2CSCCS2)\N.Cl GK02370 CN(C)c1ccc(cc1)C(=O)C(F)(F)F NRB01008 Cc1cc(c(cc1C)NC(=O)CC#N)C DP00098 Cc1cc(c(cc1C)NC(=O)N)C PHG00002 CCOC(=O)CC1C(=S)Nc2ccccc2S1 KM06801 c1ccc2c(c1)NC3(S2)CC(SC3)c4cccs4 HTS09423 CC(C)(c1cc(cc(c1)OC)OC)OC(=O)NCC(=O)O.C1CCC(CC1)N RJC02215 c1cc[n+](cc1)C[n+]2ccccc2.[I-].[I-] RJC02411 CCOC(=O)c1cc([nH]n1)c2cccs2 SPB04031 CCOC(=O)C1=C(NC(=O)NC1c2ccc(cc2)F)C HTS13448 c1cc(c(c(c1)F)C#N)NC(=O)C2CCCCC2 HTS09359 COc1cc(c(cc1OC)NC(=O)Nc2ccc(cc2)OC(F)(F)F)C(=O)OC GK03121 c1cc(c(cc1Cl)Cl)S(=O)(=O)CC#N KM06455 c1cc(sc1)C(=O)Nc2ccc(cc2)N3CCCCC3 HTS08408 Cc1c(c2ccccc2[nH]1)CCC#N BTB13429 c1ccc2c(c1)-c3c(cccc3C2=O)C#N BTB10894 c1cc(ccc1c2cc(=S)ss2)Cl EN00275 c1ccc(cc1)CNC(=O)Nc2ccccc2 KM09658 CN(CCC#N)c1ccc(cc1)C2Nc3ccccc3O2 DP01286 COc1cccc2c1nc(s2)N AC16035 CC(C)(C)OC(=O)N1CCCN(CC1)C(=S)Nc2ccccc2N3CCOCC3 AW00380 c1ccc(cc1)C2CC(=Nc3ccccc3S2)c4ccc(cc4)OCC(=O)Nc5ccccc5 RJC00348 c1ccc2c(c1)cccc2/C=N/NC(=S)Nc3cccc(c3)C(F)(F)F S03263 c1cc(c(c(c1)Cl)Cl)c2nnn(n2)CCC(=O)NNC(=S)Nc3ccc(c(c3)Cl)Cl RJF02209 Cc1ccc(cc1)CSc2nnc(n2CCCOC)c3ccc(cc3)C(C)(C)C SPB00458 COc1ccc(cc1)C(=O)/C=C/Nc2ccccc2C#N BTB12037 Cc1ccc(cc1)c2csc(n2)c3cccnc3.Br ML00066 c1ccc(c(c1)Nc2nc(cs2)c3ccc(cc3)[N+](=O)[O-])Cl.Br ML00085 c1cc2cccc3c2c(c1)NC(=N3)N.Br AC21366 c1ccc(cc1)NC2=CC(N(C2=O)c3ccccc3)c4ccccc4F BTB12155 CC1(CN=C(S1)N(c2cccc(c2)C(F)(F)F)C(=O)Nc3ccccc3)C BTB13191 CSc1nc2ccc(cc2s1)NS(=O)(=O)c3ccccc3C(F)(F)F KM07547 C=CCN/C=C(\C#N)/S(=O)(=O)c1ccc(cc1)Cl KM00757 CN(C)/C=C/C(=O)c1ccc(s1)C#Cc2ccccc2 KM08044 c1cc(sc1)c2nnc3n2N=C(CS3)c4ccc5c(c4)OCCO5.Br HTS09251 c1cc(ccc1c2csc(n2)NNC(=O)c3ccncc3)Br HTS13463 Cc1ccc(cc1)c2cc(c3c(ncnc3n2)N)c4ccccc4 HTS13546 Cc1nc(cs1)c2ccc(cc2)NC(=O)c3cccc4c3nsn4 HTS13816 CC(C)Sc1c(cccc1Cl)NC(=O)Nc2cccc(c2)[N+](=O)[O-] KM10153 CCCCc1ccc(cc1)C(=O)N=S2CCN(CC2)C(=O)c3ccc(cc3)Cl KM06239 COc1cc2c(cc1OC)[nH]c(=O)n(c2=O)CCO PD00491 COc1cc(cc(c1OC)OC)c2nnc(n2c3cccc(c3)C(F)(F)F)SCC(=O)c4ccc(cc4)F.Br ML00373 CC(=O)OC[C@@H]1[C@H]([C@@H]([C@H]([C@@H](O1)OC(=O)C)N2C(=O)c3ccccc3C2=O)OC(=O)C)OC(=O)C RJC01343 c1cc(c(cc1Cl)NC(=N)NC#N)Cl NRB04579 CSC(=O)NC(=O)c1cccc(=O)o1 SEW01645 c1ccc2c(c1)cc(c(=O)o2)c3ccc(cc3)[N+](=O)[O-] PHG00097 COC(=O)c1c(ccs1)Oc2ccc(cc2NC(=O)Nc3ccccc3)C(F)(F)F GK03084 COc1cc(cc(c1OC)OC)C(=O)Nc2ccc(c(c2)Cl)Cl JFD02698 COc1cc(ccc1O)/C=N/CCNc2c3c(csc3ncn2)c4ccccc4 AW00997 Cc1cc(nc(n1)NS(=O)(=O)c2ccc(cc2)NC(=O)Nc3ccc(cc3Cl)Cl)C HTS07243 c1ccc(cc1)S(=O)(=O)c2cscc2NC(=O)Nc3ccc(cc3)Cl KM01825 CC1=Nc2ccccc2NC(C1)(C)C RJC00373 c1ccc(cc1)n2c(c(sc2=S)C(=O)N/N=C/c3ccc(cc3)Cl)N HTS07570 Cc1c(c(no1)c2c(cccc2Cl)Cl)C(=O)O/N=C(/c3ccco3)\O CD05022 c1cc(cnc1)C2CCCN2S(=O)(=O)c3ccc(cc3Cl)Cl CD10450 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)NS(=O)(=O)c3ccc(c(c3)OC)OC RJF01031 c1cc(ccc1C(c2ccc(cc2)F)N3CCNCC3)F AC10018 c1cc(c(cc1c2cnc3cc(cc(c3n2)Cl)C(F)(F)F)Cl)Cl BTB05383 c1cc(cc(c1)F)CSC2=NCN(CN2)C3CC3.Cl BTB04277 CCc1ccccc1NC(=N)NC(=N)N.Cl RDR01691 CCOC(=O)c1c(c(n(c1NC(=O)c2ccc(cc2)Cl)CC3CC3)C)C SPB01921 Cc1c(c(n(n1)c2ccccc2)C)c3nnc(o3)c4c(nn(c4C)c5ccccc5)C SEW04236 COc1ccccc1C2=NOC(C2)COC(=O)c3ccc(cc3)[N+](=O)[O-] HTS11171 Cc1cc(nc2c1c3c(s2)c(=O)n(cn3)/N=C/c4cccc(c4)OC)C HTS12657 Cc1c(cc(o1)c2cccs2)C(=O)O AW00850 Cc1c(nn(n1)c2ccccc2)CNC(=O)Cc3ccccc3OC SCR01437 c1cc(cc(c1)NC(=O)c2cccc3c2nsn3)Cn4cccn4 HTS13855 c1cc(ccc1C(=O)/C=C/Sc2ccc(cn2)C(F)(F)F)Cl NRB04305 CCOc1ccc(cc1)NC(=O)/C=C/c2ccc(c(c2)[N+](=O)[O-])N3CCC(CC3)c4ccccc4OC RH01696 CC(C)(C)c1ccc(cc1)c2n[nH]nn2 SPB01120 c1cc[n+](cc1)CC(=O)N2CCN(CC2)c3ccc(cc3[N+](=O)[O-])C(F)(F)F.[Cl-] BTB04708 c1ccc(cc1)c2c(c(nnc2c3ccccc3)N/N=C(\c4ccccc4)/C(c5ccccc5)O)c6ccccc6 BTB13525 c1cc(c(cc1[N+](=O)[O-])[N+](=O)[O-])ONS(=O)(=O)c2cc(c(s2)Br)Br BTB09585 Cc1ccc(c(c1)C(=O)O)NC(=O)C HTS13970 CC12CCC(CC1)(CC2=O)O BTB14472 c1ccc(cc1)CN(Cc2ccccc2)CC(=O)O HTS11212 Cc1cc(c(cc1C)NC(=N)NN)C.I RDR02117 c1ccc(cc1)S(=O)(=O)Oc2ccc(cc2)c3csnn3 SEW01164 COCc1cc(nc(n1)NC(=N)Nc2ccccc2SC)O RJF00569 COC(=O)C/C(=N/Nc1ccc(cc1)C(F)(F)F)/C(=O)OC SEW03479 Cc1cc(nn1C)C(=O)NNc2ccc(cc2F)F SPB00660 Cc1cc(no1)NS(=O)(=O)c2ccc(cc2)N RJF01028 CC(CN1CCN(CC1)Cc2ccccc2)N(c3ccccn3)C(=O)c4cccc(c4)[N+](=O)[O-].Cl.Cl.Cl BTB15236 COC(=O)c1cnn(c1C=C(C#N)C#N)c2ccccc2 SPB05268 c1ccc2c(c1)[nH]c(n2)N3C(=O)c4cccc5c4c(ccc5)C3=O BTB11694 Cc1c(c(c(c(c1C)C)CN2CCCC(C2)C)C)C CD00074 c1cc(ccc1C(=O)N(CCC#N)CCC#N)Cl CD02217 COC(=O)c1c(ccs1)N2C(=O)c3ccccc3C2=O GK01178 CCOC(=O)c1c(nc(s1)c2ccccc2)O SPB01861 Cc1c(ccc(n1)C(F)(F)F)C(=O)NCC=C AW00742 CC(C)(C)OC(=O)N1CCCC[C@@H]1C(=O)O AC39925 c1ccc(cc1)C(=O)O[C@H]([C@H](C(=O)O)OC(=O)c2ccccc2)C(=O)O SCR01521 CC(=O)N[C@H](CC(=O)N)C(=O)O NRB05180 Cc1cn2c(nc1=O)O[C@@H]3C[C@H]2O[C@@H]3CO BTB14109 CC(C)(C)OC(=O)N1CCCC[C@H]1C(=O)O AC39783 CCOC(=O)CSc1nc(cn1c2ccc(cc2OC)OC)c3ccccc3 HTS13232 CCCN(CCC)S(=O)(=O)c1ccc(cc1)C(=O)O/N=C(/c2ccc3c(c2)OCO3)\N CD02624 c1ccc2c(c1)n(c(=O)o2)CCC(=O)Sc3ccc(cc3)C(F)(F)F SPB02722 CCn1c(cc(n1)C)C(=O)NNC(=S)NC SPB02530 Cc1cc(c(c(c1)CC(C)(C)C(=O)O)C(=O)O)C CD01061 c1cc(oc1C(=O)NC2=NCCS2)[N+](=O)[O-] BR00042 c1ccc(cc1)CC2CCN(CC2)S(=O)(=O)c3cc(c(s3)Cl)Br HTS00832 CCCCNC(=O)O/N=C(/CS(=O)(=O)C(C)(C)C)\N KM02275 c1ccc(cc1)OCCN2CCN(CC2)C(=O)c3ccc(cc3)Cl TB00007 c1cc(cc(c1)NC(=O)c2ccc(c(c2OCC(F)(F)F)C#N)OCC(F)(F)F)C(F)(F)F MWP01212 c1cc(ccc1CC(=O)Nc2nccs2)[N+](=O)[O-] RF00491 Cc1c(c(sc1C(=O)OC)S(=O)C)c2ccno2 KM05174 Cc1c(cc(n1CCSC)c2ccccc2)C(=O)N3CCCCC3 SP00873 COc1cccc(c1O)/C=N/c2cc(cc(c2)C(F)(F)F)C(F)(F)F GK03596 CC(C)(C)C(=O)NCC1COc2ccccc2O1 KM07136 Cc1ccc(cc1C)OCC(CNc2ccc(c(c2)C(F)(F)F)Br)O HTS01930 c1cc(c(nc1)SCC(=O)Nc2cc(cc(c2)Cl)Cl)C(=O)O RH00878 Cc1cc(c2ccccc2n1)N3CCN(CC3)C(=O)c4cc5cc(c(cc5oc4=O)OC)OC HTS10627 CC(C)c1ccc(cc1)NC2(CCCCC2)C#N DSHS00049 Cc1nc(cn1C)S(=O)(=O)N2CCN(CC2)C3c4ccccc4-c5c3cccc5 HTS08761 CSc1c(c(nc(n1)SC)c2ccco2)C#N KM01064 c1cc(c(cc1C=C2C(=O)NC(=O)NC2=O)O)O CD00393 CC1c2cc(c(cc2CCN1C(=S)Nc3cc(c(c(c3)OC)OC)OC)OC)OC BTB04348 COc1ccc(cc1)c2c(c[nH]n2)/C=N/Nc3c(cc(cn3)C(F)(F)F)Cl SEW06357 C/S(=N\S(=O)(=O)c1cccc2c1nsn2)/c3c(cc(cn3)Cl)C(F)(F)F KM08416 Cc1cn(nc1C(=O)Nc2c3ccccc3n(n2)C)c4ccccc4 HTS02208 COC(=O)c1cc(cn1c2ccc(cc2)Cl)/C=C(\C#N)/S(=O)(=O)C SEW06675 Cc1c2c(cc(s2)C(C)(C)C)sc1c3nc(no3)c4cc(cc(c4)C(F)(F)F)C(F)(F)F GK03109 COc1ccc(cc1OC)c2nc(no2)CS(=O)(=O)c3ccsc3 SP00786 c1cc2cccc3c2c(c1)c(=O)c4cccc5c4c(s3)ccc5 NRB00685 c1ccc2c(c1)ncc(n2)NCCNc3c(cc(cn3)C(F)(F)F)Cl RDR04080 CN1CC2C(N(N=C2/C(=C/c3ccc(cc3)C(F)(F)F)/C1)C)c4ccc(cc4)C(F)(F)F S13506 COc1cc(cc(c1OC)OC)c2n[nH]c(=S)n2c3cccc(c3)C(F)(F)F ML00370 c1cc(ccc1NC=C(C#N)C#N)S(=O)(=O)c2ccc(cc2)NC=C(C#N)C#N BTB06667 Cc1nc(cn1CC(=O)c2ccc(s2)c3cccnc3)[N+](=O)[O-] HTS04156 c1ccc(cc1)C(=O)OC(C#N)c2cccc(c2)[N+](=O)[O-] XBX00116 c1ccc(cc1)Oc2ccc(cc2)OS(=O)(=O)c3ccc(cc3)C#N BTB14633 Cc1c2c(nc(nc2sc1c3ccc(c(c3)OC)OC)c4cc(cc(c4)OC)OC)N CD02075 c1ccc2c(c1)C(=O)N(C2=O)C(CCC(=O)Nc3ccc4c(c3)COCO4)C(=O)O BTB07136 COc1ccc(cc1)n2c(n[nH]c2=S)c3ccncc3 ML00390 CCSC([C@H]([C@@H]([C@@H]([C@H](COC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C)OC(=O)C JFD01223 c1ccc(cc1)C/N=C\2/C3=C(CCCC3)/C(=N\c4ccccc4)/S2 HTS07414 CC(C)n1c2ccc(cc2nc1SCC(=O)c3ccccc3)Cl HTS02666 c1ccc(cc1)CN2CCN(CC2)/C=C(\C#N)/S(=O)(=O)c3ccc(cc3)Cl KM09014 Cc1c(c(no1)c2ccccc2Cl)NC(=O)N3c4ccc(cc4CCC3C)F BTB03394 c1ccc(c(c1)NC(=O)c2c(cccc2F)F)SCc3nc(on3)c4cccs4 SEW06394 Cc1c(snn1)C(=O)N2CCc3cc(c(cc3C2C)OC)OC HTS04859 Cc1cc(ccc1O)C(C)(C)c2ccc(c(c2)C)O BTB14075 CC(C)(C)S(=O)(=O)Cc1nc(cs1)c2ccc(cc2)C(F)(F)F SP00571 Cc1ccc(cc1NS(=O)(=O)c2cccc(c2)C(F)(F)F)S(=O)(=O)N(C)C HTS05504 c1cc(ncc1S(=O)(=O)N2CCN(CC2)c3c(cncc3Cl)Cl)N4CCOCC4 SCR01192 Cc1cc2ccccc2c(c1C#N)/N=C/c3cc(cc(c3O)Br)Br DSHS00330 c1ccc(cc1)C(=O)/C(=C/c2ccc3c(c2)CCO3)/C#N KM06426 Cn1c(ccc1S(=O)(=O)N2CCCN(CC2)c3ccc(cn3)C(F)(F)F)C(=O)OC HTS01549 CC1CCC(OC1)C2C(C3C(O2)CC4C3(CC=C5C4CCC6C5(CCC(C6)O)C)C)C NRB03658 CC(C)(C)c1ccc(c(c1)C(C)(C)C)OC(=O)NC(=O)c2ccccc2Cl BTB04120 c1ccc2c(c1)c(=O)n(c(=O)n2Cc3ccc(cc3)Cl)Cc4ccc(cc4)Cl HTS11468 CCCCc1ccc(cc1)n2c(coc2=O)c3ccc(cc3)F HTS02872 c1ccc(c(c1)[N+](=O)[O-])S(=O)(=O)CC(=O)O BTB13851 COC(=S)NC(=O)/C=C/c1ccccc1 PD00687 c1ccc2c(c1)c3c(c(=O)o2)Sc4ccccc4N3 MGH00118 c1ccc(cc1)CN2C3CCCC2CC(=O)C3 KM08807