| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 79 | 2 | 0 | 0 |
| Binding ≤ 1μM | 69 | 2 | 0 | 0 |
| Functional ≤ 10μM | 267 | 7 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_18283 | G alpha (q) signalling events | Homo sapiens |
| REACT_14819 | Peptide ligand-binding receptors | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| GRPR_HUMAN | P30550 | CHEMBL4959 | Gastrin Releasing Peptide Receptor, Human | 1 |
| NMBR_HUMAN | P28336 | CHEMBL3636 | Neuromedin B Receptor, Human | 1 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| GRPR_HUMAN | P30550 | CHEMBL4959 | Gastrin Releasing Peptide Receptor, Human | 1 |
| NMBR_HUMAN | P28336 | CHEMBL3636 | Neuromedin B Receptor, Human | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| BRS3_MOUSE | O54798 | CHEMBL1075140 | Bombesin Receptor Subtype-3, Mouse | 2 | 0 | 0 | 0 |
| BRS3_RAT | Q8K418 | CHEMBL1075111 | Bombesin Receptor Subtype-3, Rat | 2 | 0 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| BRSK1_HUMAN | Q8TDC3 | CHEMBL5650 | BR Serine/threonine-protein Kinase 1, Human | 5 | 5 | 2 | 2 |
| BRSK2_HUMAN | Q8IWQ3 | CHEMBL4574 | BR Serine/threonine-protein Kinase 2, Human | 9 | 6 | 2 | 2 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| BRS3-1-E | Bombesin Receptor Subtype-3 (cluster #1 Of 2), Eukaryotic | 53 | 0 | 0 | 0 |
| BRS3-2-E | Bombesin Receptor Subtype-3 (cluster #2 Of 2), Eukaryotic | 28 | 4 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| BRS3_MOUSE | O54798 | CHEMBL1075140 | Bombesin Receptor Subtype-3, Mouse | 110 |
| BRS3_RAT | Q8K418 | CHEMBL1075111 | Bombesin Receptor Subtype-3, Rat | 38 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 5 |
| GRPR_HUMAN | P30550 | CHEMBL4959 | Gastrin Releasing Peptide Receptor, Human | 1 |
| NMBR_HUMAN | P28336 | CHEMBL3636 | Neuromedin B Receptor, Human | 1 |
| NR1I2_HUMAN | O75469 | CHEMBL3401 | Pregnane X Receptor, Human | 1 |
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