UCSF

Calcitonin Gene-related Peptide Type 1 Receptor, Human (377 Compounds)

Swissprot:
CALRL_HUMAN
Stitch:
CALRL_HUMAN
UniProt:
Q16602
ChEMBL:
CHEMBL3798
Reactome:
REACT_18290
REACT_19327
PDB:
3AQF (DOCK)
3N7P (DOCK)
3N7R (DOCK)
3N7S (DOCK)
CALCRL

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 377 0 1 1
Binding ≤ 1μM 324 0 1 1
Functional ≤ 10μM 314 0 1 1

Reactome Network (2)

Uniprot Swissprot Chembl Description Number Shared
RAMP1_HUMAN O60894 CHEMBL3316 Receptor Activity-modifying Protein 1, Human 35

G alpha (s) signalling events

Uniprot Swissprot Chembl Description Number Shared
RAMP1_HUMAN O60894 CHEMBL3316 Receptor Activity-modifying Protein 1, Human 35
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
CALRL_RAT Q63118 CHEMBL4755 Calcitonin Gene-related Peptide Type 1 Receptor, Rat 0 0 0 0

Clustered By Gene (0)

Uniprot Swissprot Chembl Description Number Shared
RAMP1_HUMAN O60894 CHEMBL3316 Receptor Activity-modifying Protein 1, Human 35
MP2K2_HUMAN P36507 CHEMBL2964 Dual Specificity Mitogen-activated Protein Kinase Kinase 2, Human 18
Z50797 Z50797 CHEMBL614875 Rhesus Monkey 5
KCNH2_HUMAN Q12809 CHEMBL240 HERG, Human 1