| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 29 | 2 | 1 | 1 |
| Binding ≤ 1μM | 29 | 2 | 1 | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| ESR1_HUMAN | P03372 | CHEMBL206 | Estrogen Receptor Alpha, Human | 1,669 | 74 | 54 | 67 |
| ESR1_MOUSE | P19785 | CHEMBL3065 | Estrogen Receptor Alpha, Mouse | 10 | 5 | 2 | 2 |
| ESR1_RAT | P06211 | CHEMBL2724 | Estrogen Receptor Alpha, Rat | 84 | 14 | 11 | 11 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| ESR1-1-E | Estrogen Receptor Alpha (cluster #1 Of 5), Eukaryotic | 1,489 | 63 | 46 | 66 |
| ESR1-2-E | Estrogen Receptor Alpha (cluster #2 Of 5), Eukaryotic | 118 | 14 | 11 | 7 |
| ESR1-3-E | Estrogen Receptor Alpha (cluster #3 Of 5), Eukaryotic | 39 | 3 | 1 | 1 |
| ESR1-4-E | Estrogen Receptor Alpha (cluster #4 Of 5), Eukaryotic | 17 | 0 | 0 | 0 |
| ESR1-5-E | Estrogen Receptor Alpha (cluster #5 Of 5), Eukaryotic | 84 | 5 | 5 | 5 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| ESR1_HUMAN | P03372 | CHEMBL206 | Estrogen Receptor Alpha, Human | 29 |
| ESR2_HUMAN | Q92731 | CHEMBL242 | Estrogen Receptor Beta, Human | 29 |
| ESR2_MOUSE | O08537 | CHEMBL2995 | Estrogen Receptor Beta, Mouse | 29 |
| ANDR_HUMAN | P10275 | CHEMBL1871 | Androgen Receptor, Human | 1 |
| ERR1_HUMAN | P11474 | CHEMBL3429 | Estrogen-related Receptor Alpha, Human | 1 |
| ERR2_HUMAN | O95718 | CHEMBL3751 | Estrogen-related Receptor Beta, Human | 1 |
| ESR1_MOUSE | P19785 | CHEMBL3065 | Estrogen Receptor Alpha, Mouse | 1 |
| ESR1_RAT | P06211 | CHEMBL2724 | Estrogen Receptor Alpha, Rat | 1 |
| ESR2_RAT | Q62986 | CHEMBL3021 | Estrogen Receptor Beta, Rat | 1 |
| GPER_HUMAN | Q99527 | CHEMBL5872 | G-protein Coupled Estrogen Receptor 1, Human | 1 |
| SHBG_HUMAN | P04278 | CHEMBL3305 | Testis-specific Androgen-binding Protein, Human | 1 |