| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 16 | 1 | 1 | 1 |
| Binding ≤ 1μM | 10 | 1 | 1 | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 2,874 | 203 | 156 | 161 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| KCNH2-1-E | HERG (cluster #1 Of 5), Eukaryotic | 1,730 | 79 | 64 | 65 |
| KCNH2-2-E | HERG (cluster #2 Of 5), Eukaryotic | 112 | 19 | 10 | 13 |
| KCNH2-3-E | HERG (cluster #3 Of 5), Eukaryotic | 141 | 7 | 6 | 6 |
| KCNH2-4-E | HERG (cluster #4 Of 5), Eukaryotic | 136 | 7 | 4 | 4 |
| KCNH2-5-E | HERG (cluster #5 Of 5), Eukaryotic | 807 | 98 | 78 | 79 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| KCNQ1_CAVPO | O70344 | CHEMBL5135 | Voltage-gated Potassium Channel Subunit Kv7.1, Guinea Pig | 13 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 1 |