| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 1 | 1 | 0 | 0 |
| Binding ≤ 1μM | 1 | 1 | 0 | 0 |
| Functional ≤ 10μM | 6 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_22303 | Highly calcium permeable postsynaptic nicotinic acetylcholine receptors | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| ACHA2_HUMAN | Q15822 | CHEMBL1794 | Neuronal Acetylcholine Receptor Protein Alpha-2 Subunit, Human | 1 |
| ACHA3_HUMAN | P32297 | CHEMBL3068 | Neuronal Acetylcholine Receptor Protein Alpha-3 Subunit, Human | 1 |
| ACHA4_HUMAN | P43681 | CHEMBL1882 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Human | 1 |
| ACHA5_HUMAN | P30532 | CHEMBL2454 | Neuronal Acetylcholine Receptor Protein Alpha-5 Subunit, Human | 1 |
| ACHA6_HUMAN | Q15825 | CHEMBL2356 | Neuronal Acetylcholine Receptor Protein Alpha-6 Subunit, Human | 1 |
| ACHA7_HUMAN | P36544 | CHEMBL2492 | Neuronal Acetylcholine Receptor Protein Alpha-7 Subunit, Human | 7 |
| ACHA_HUMAN | P02708 | CHEMBL4808 | Acetylcholine Receptor Protein Alpha Chain, Human | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| ACHA9_RAT | P43144 | CHEMBL2585 | Neuronal Acetylcholine Receptor Protein Alpha-9 Subunit, Rat | 300 | 51 | 14 | 3 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| ACHA2_HUMAN | Q15822 | CHEMBL1794 | Neuronal Acetylcholine Receptor Protein Alpha-2 Subunit, Human | 24 | 6 | 4 | 4 |
| ACHA3_HUMAN | P32297 | CHEMBL3068 | Neuronal Acetylcholine Receptor Protein Alpha-3 Subunit, Human | 84 | 15 | 7 | 7 |
| ACHA4_HUMAN | P43681 | CHEMBL1882 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Human | 140 | 21 | 4 | 4 |
| ACHA5_HUMAN | P30532 | CHEMBL2454 | Neuronal Acetylcholine Receptor Protein Alpha-5 Subunit, Human | 5 | 3 | 1 | 0 |
| ACHA6_HUMAN | Q15825 | CHEMBL2356 | Neuronal Acetylcholine Receptor Protein Alpha-6 Subunit, Human | 5 | 3 | 1 | 0 |
| ACHA7_HUMAN | P36544 | CHEMBL2492 | Neuronal Acetylcholine Receptor Protein Alpha-7 Subunit, Human | 142 | 31 | 15 | 10 |
| ACHA_HUMAN | P02708 | CHEMBL4808 | Acetylcholine Receptor Protein Alpha Chain, Human | 8 | 3 | 1 | 0 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| ACHA9-1-E | Neuronal Acetylcholine Receptor Protein Alpha-9 Subunit (cluster #1 Of 4), Eukaryotic | 67 | 13 | 0 | 0 |
| ACHA9-2-E | Neuronal Acetylcholine Receptor Protein Alpha-9 Subunit (cluster #2 Of 4), Eukaryotic | 75 | 7 | 0 | 0 |
| ACHA9-3-E | Neuronal Acetylcholine Receptor Protein Alpha-9 Subunit (cluster #3 Of 4), Eukaryotic | 50 | 11 | 9 | 1 |
| ACHA9-4-E | Neuronal Acetylcholine Receptor Protein Alpha-9 Subunit (cluster #4 Of 4), Eukaryotic | 109 | 21 | 5 | 2 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| ACH10_HUMAN | Q9GZZ6 | CHEMBL2551 | Neuronal Acetylcholine Receptor Protein Alpha-10 Subunit, Human | 7 |
| ACHA7_HUMAN | P36544 | CHEMBL2492 | Neuronal Acetylcholine Receptor Protein Alpha-7 Subunit, Human | 7 |
| ACHA2_HUMAN | Q15822 | CHEMBL1794 | Neuronal Acetylcholine Receptor Protein Alpha-2 Subunit, Human | 1 |
| ACHA2_RAT | P12389 | CHEMBL2584 | Neuronal Acetylcholine Receptor Protein Alpha-2 Subunit, Rat | 1 |
| ACHA3_HUMAN | P32297 | CHEMBL3068 | Neuronal Acetylcholine Receptor Protein Alpha-3 Subunit, Human | 1 |
| ACHA3_RAT | P04757 | CHEMBL3818 | Neuronal Acetylcholine Receptor Protein Alpha-3 Subunit, Rat | 1 |
| ACHA4_HUMAN | P43681 | CHEMBL1882 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Human | 1 |
| ACHA4_RAT | P09483 | CHEMBL307 | Neuronal Acetylcholine Receptor Protein Alpha-4 Subunit, Rat | 1 |
| ACHA5_HUMAN | P30532 | CHEMBL2454 | Neuronal Acetylcholine Receptor Protein Alpha-5 Subunit, Human | 1 |
| ACHA6_HUMAN | Q15825 | CHEMBL2356 | Neuronal Acetylcholine Receptor Protein Alpha-6 Subunit, Human | 1 |
| ACHA_HUMAN | P02708 | CHEMBL4808 | Acetylcholine Receptor Protein Alpha Chain, Human | 1 |
| ACHD_TORCA | P02718 | CHEMBL3916 | Acetylcholine Receptor Protein Delta Chain, Torca | 1 |
| Z104290 | Z104290 | CHEMBL1907596 | Neuronal Acetylcholine Receptor; Alpha4/beta2 | 1 |