UCSF

Cholecystokinin A Receptor, Human (524 Compounds)

Swissprot:
CCKAR_HUMAN
Stitch:
CCKAR_HUMAN
UniProt:
P32238
ChEMBL:
CHEMBL1901
Reactome:
REACT_18283
REACT_14819
PDB:
1D6G (DOCK)
1HZN (DOCK)
1PB2 (DOCK)
CCKAR

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 524 9 8 5
Binding ≤ 1μM 313 6 5 4
Functional ≤ 10μM 120 1 2 1

Reactome Network (2)

Reactome ID Description Species
REACT_18283 G alpha (q) signalling events Homo sapiens
REACT_14819 Peptide ligand-binding receptors Homo sapiens
Uniprot Swissprot Chembl Description Number Shared
GASR_HUMAN P32239 CHEMBL298 Cholecystokinin B Receptor, Human 328

Peptide ligand-binding receptors

Uniprot Swissprot Chembl Description Number Shared
GASR_HUMAN P32239 CHEMBL298 Cholecystokinin B Receptor, Human 328
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
CCKAR_CAVPO Q63931 CHEMBL3501 Cholecystokinin A Receptor, Guinea Pig 41 0 0 0
CCKAR_MOUSE O08786 CHEMBL2798 Cholecystokinin A Receptor, Mouse 46 1 1 1
CCKAR_RAT P30551 CHEMBL2871 Cholecystokinin A Receptor, Rat 1,390 29 10 10

Clustered By Gene (0)

Uniprot Swissprot Chembl Description Number Shared
GASR_HUMAN P32239 CHEMBL298 Cholecystokinin B Receptor, Human 328
CCKAR_RAT P30551 CHEMBL2871 Cholecystokinin A Receptor, Rat 119
GASR_RAT P30553 CHEMBL3508 Cholecystokinin B Receptor, Rat 59
GASR_MOUSE P56481 CHEMBL2854 Cholecystokinin B Receptor, Mouse 19
CCKAR_MOUSE O08786 CHEMBL2798 Cholecystokinin A Receptor, Mouse 10
Z50597 Z50597 CHEMBL376 Rattus Norvegicus 4
CNR2_HUMAN P34972 CHEMBL253 Cannabinoid CB2 Receptor, Human 2
COX1_HUMAN P00395 CHEMBL6173 Cytochrome C Oxidase Subunit 1, Human 2
5HT1A_HUMAN P08908 CHEMBL214 Serotonin 1a (5-HT1a) Receptor, Human 1
5HT5A_HUMAN P47898 CHEMBL3426 Serotonin 5a (5-HT5a) Receptor, Human 1
AA3R_HUMAN P33765 CHEMBL256 Adenosine A3 Receptor, Human 1
CCKAR_CAVPO Q63931 CHEMBL3501 Cholecystokinin A Receptor, Guinea Pig 1
CNR2_MOUSE P47936 CHEMBL5373 Cannabinoid CB2 Receptor, Mouse 1
FAAH1_MOUSE O08914 CHEMBL3455 Anandamide Amidohydrolase, Mouse 1
GPR44_HUMAN Q9Y5Y4 CHEMBL5071 G Protein-coupled Receptor 44, Human 1
GPR44_MOUSE Q9Z2J6 CHEMBL2291 G Protein-coupled Receptor 44, Mouse 1
KCNH2_HUMAN Q12809 CHEMBL240 HERG, Human 1
OPRD_RAT P33533 CHEMBL269 Delta Opioid Receptor, Rat 1
OPRK_RAT P34975 CHEMBL3614 Kappa Opioid Receptor, Rat 1
OPRM_RAT P33535 CHEMBL270 Mu Opioid Receptor, Rat 1
SGMR1_RAT Q9R0C9 CHEMBL3602 Sigma Opioid Receptor, Rat 1

Most Common Rings