| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 33 | 4 | 2 | 1 |
| Binding ≤ 1μM | 22 | 1 | 1 | 0 |
| Functional ≤ 10μM | 1 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_75770 | Voltage gated Potassium channels | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| KCND3_HUMAN | Q9UK17 | CHEMBL1964 | Voltage-gated Potassium Channel Subunit Kv4.3, Human | 1 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| KCNQ1_CAVPO | O70344 | CHEMBL5135 | Voltage-gated Potassium Channel Subunit Kv7.1, Guinea Pig | 74 | 3 | 4 | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| KCNQ2_HUMAN | O43526 | CHEMBL2476 | Voltage-gated Potassium Channel Subunit Kv7.2, Human | 20 | 4 | 1 | 1 |
| KCNQ3_HUMAN | O43525 | CHEMBL2684 | Voltage-gated Potassium Channel Subunit Kv7.3, Human | 18 | 4 | 1 | 1 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| KCNQ1-1-E | Voltage-gated Potassium Channel Subunit Kv7.1 (cluster #1 Of 2), Eukaryotic | 109 | 7 | 5 | 1 |
| KCNQ1-2-E | Voltage-gated Potassium Channel Subunit Kv7.1 (cluster #2 Of 2), Eukaryotic | 2 | 1 | 2 | 1 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| KCNE1_HUMAN | P15382 | CHEMBL4872 | Voltage-gated Potassium Channel Beta Subunit Mink, Human | 32 |
| KCNQ1_CAVPO | O70344 | CHEMBL5135 | Voltage-gated Potassium Channel Subunit Kv7.1, Guinea Pig | 3 |
| KCNN4_HUMAN | O15554 | CHEMBL4305 | Intermediate Conductance Calcium-activated Potassium Channel Protein 4, Human | 2 |
| 5HT2A_HUMAN | P28223 | CHEMBL224 | Serotonin 2a (5-HT2a) Receptor, Human | 1 |
| 5HT2A_RAT | P14842 | CHEMBL322 | Serotonin 2a (5-HT2a) Receptor, Rat | 1 |
| 5HT2C_HUMAN | P28335 | CHEMBL225 | Serotonin 2c (5-HT2c) Receptor, Human | 1 |
| DRD2_HUMAN | P14416 | CHEMBL217 | Dopamine D2 Receptor, Human | 1 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 1 |
| Z104304 | Z104304 | CHEMBL1907610 | Adrenergic Receptor Alpha-1 | 1 |