| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 384 | 0 | 0 | 0 |
| Binding ≤ 1μM | 178 | 0 | 0 | 0 |
| Functional ≤ 10μM | 159 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_19327 | G alpha (s) signalling events | Homo sapiens |
| REACT_14819 | Peptide ligand-binding receptors | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| MC4R_HUMAN | P32245 | CHEMBL259 | Melanocortin Receptor 4, Human | 408 |
| MC5R_HUMAN | P33032 | CHEMBL4608 | Melanocortin Receptor 5, Human | 248 |
| MSHR_HUMAN | Q01726 | CHEMBL3795 | Melanocortin Receptor 1, Human | 244 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| GHSR_HUMAN | Q92847 | CHEMBL4616 | Ghrelin Receptor, Human | 6 |
| MC4R_HUMAN | P32245 | CHEMBL259 | Melanocortin Receptor 4, Human | 408 |
| MC5R_HUMAN | P33032 | CHEMBL4608 | Melanocortin Receptor 5, Human | 248 |
| MSHR_HUMAN | Q01726 | CHEMBL3795 | Melanocortin Receptor 1, Human | 244 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| MC3R_MOUSE | P33033 | CHEMBL4774 | Melanocortin Receptor 3, Mouse | 17 | 0 | 0 | 0 |
| MC3R_RAT | P32244 | CHEMBL4023 | Melanocortin Receptor 3, Rat | 3 | 0 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| MC4R_HUMAN | P32245 | CHEMBL259 | Melanocortin Receptor 4, Human | 407 |
| MC5R_HUMAN | P33032 | CHEMBL4608 | Melanocortin Receptor 5, Human | 247 |
| MSHR_HUMAN | Q01726 | CHEMBL3795 | Melanocortin Receptor 1, Human | 244 |
| MSHR_MOUSE | Q01727 | CHEMBL4077 | Melanocortin Receptor 1, Mouse | 26 |
| MC4R_RAT | P70596 | CHEMBL2700 | Melanocortin Receptor 4, Rat | 12 |
| MC4R_MOUSE | P56450 | CHEMBL3719 | Melanocortin Receptor 4, Mouse | 11 |
| GHSR_HUMAN | Q92847 | CHEMBL4616 | Ghrelin Receptor, Human | 5 |
| MC3R_MOUSE | P33033 | CHEMBL4774 | Melanocortin Receptor 3, Mouse | 5 |
| MC3R_RAT | P32244 | CHEMBL4023 | Melanocortin Receptor 3, Rat | 4 |
| Z50594 | Z50594 | CHEMBL375 | Mus Musculus | 2 |
| Z50597 | Z50597 | CHEMBL376 | Rattus Norvegicus | 2 |
| Z80936 | Z80936 | CHEMBL614818 | HEK293 (Embryonic Kidney Fibroblasts) | 2 |
| Z81011 | Z81011 | CHEMBL614840 | Human Cell Lines | 2 |
| MC5R_MOUSE | P41149 | CHEMBL4489 | Melanocortin Receptor 5, Mouse | 1 |
| MC5R_RAT | P35345 | CHEMBL2701 | Melanocortin Receptor 5, Rat | 1 |
| MTR1B_HUMAN | P49286 | CHEMBL1946 | Melatonin Receptor 1B, Human | 1 |
| Z80236 | Z80236 | CHEMBL614332 | MCR (Frog Skin Melanocyte Cells) | 1 |