| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 1,615 | 22 | 3 | 9 |
| Functional ≤ 10μM | 191 | 7 | 2 | 2 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| EDNRA_HUMAN | P25101 | CHEMBL252 | Endothelin Receptor ET-A, Human | 1,225 | 26 | 7 | 11 |
| EDNRA_MOUSE | Q61614 | CHEMBL2286 | Endothelin Receptor ET-A, Mouse | 16 | 2 | 0 | 0 |
| EDNRA_PIG | Q29010 | CHEMBL4130 | Endothelin Receptor ET-A, Pig | 264 | 2 | 1 | 1 |
| EDNRA_RAT | P26684 | CHEMBL4566 | Endothelin Receptor ET-A, Rat | 905 | 11 | 6 | 10 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| EDNRA-2-E | Endothelin Receptor ET-A (cluster #2 Of 3), Eukaryotic | 10 | 0 | 0 | 0 |
| EDNRA-3-E | Endothelin Receptor ET-A (cluster #3 Of 3), Eukaryotic | 711 | 8 | 7 | 9 |
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