| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 281 | 4 | 2 | 2 |
| Functional ≤ 10μM | 50 | 0 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| HCAR2_HUMAN | Q8TDS4 | CHEMBL3785 | Nicotinic Acid Receptor 1, Human | 365 | 20 | 5 | 3 |
| HCAR2_MOUSE | Q9EP66 | CHEMBL4420 | HM74 Nicotinic Acid GPCR, Mouse | 70 | 1 | 1 | 1 |
| HCAR2_RAT | Q80Z39 | CHEMBL4731 | HM74 Nicotinic Acid GPCR, Rat | 19 | 8 | 3 | 1 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| HCAR2-2-E | HM74 Nicotinic Acid GPCR (cluster #2 Of 4), Eukaryotic | 50 | 11 | 3 | 1 |
| HCAR2-3-E | HM74 Nicotinic Acid GPCR (cluster #3 Of 4), Eukaryotic | 31 | 1 | 1 | 0 |
| HCAR2-4-E | HM74 Nicotinic Acid GPCR (cluster #4 Of 4), Eukaryotic | 16 | 9 | 1 | 0 |