| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 369 | 32 | 18 | 11 |
| Functional ≤ 10μM | 142 | 6 | 3 | 6 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| TOP1_HUMAN | P11387 | CHEMBL1781 | DNA Topoisomerase I, Human | 358 | 28 | 14 | 10 |
| TOP1_MOUSE | Q04750 | CHEMBL2814 | DNA Topoisomerase I, Mouse | 29 | 1 | 2 | 1 |
| TOP1_RAT | Q9WUL0 | CHEMBL1075164 | DNA Topoisomerase 1, Rat | 1 | 1 | 1 | 0 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| TOP1-2-E | DNA Topoisomerase 1 (cluster #2 Of 2), Eukaryotic | 1 | 0 | 0 | 0 |