| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 106 | 22 | 6 | 4 |
| Functional ≤ 10μM | 3 | 3 | 1 | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GABR1_HUMAN | Q9UBS5 | CHEMBL2064 | GABA-B Receptor 1, Human | 32 | 5 | 3 | 3 |
| GABR1_RAT | Q9Z0U4 | CHEMBL2753 | GABA-B Receptor 1, Rat | 104 | 29 | 6 | 4 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| GABR1-2-E | GABA-B Receptor 1 (cluster #2 Of 3), Eukaryotic | 14 | 8 | 1 | 1 |
| GABR1-3-E | GABA-B Receptor 1 (cluster #3 Of 3), Eukaryotic | 5 | 1 | 1 | 1 |