UCSF

Voltage-gated Calcium Channel Alpha2/delta Subunit 1, Rat (22 Compounds)

Swissprot:
CA2D1_RAT
Stitch:
CA2D1_RAT
UniProt:
P54290
ChEMBL:
CHEMBL3420
PDB:
Cacna2d1

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 22 7 5 4
Binding ≤ 1μM 19 7 5 4
Functional ≤ 10μM 2 1 1 1

Reactome Network (0)

UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
CA2D1_HUMAN P54289 CHEMBL1919 Voltage-gated Calcium Channel Alpha2/delta Subunit 1, Human 295 44 3 2
CA2D1_MOUSE O08532 CHEMBL4676 Voltage-gated Calcium Channel Alpha2/delta Subunit 1, Mouse 84 72 10 4
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
CA2D2_RAT Q8CFG6 CHEMBL3914 Voltage-gated Calcium Channel Alpha2/delta Subunit 2, Rat 4 3 3 2
CA2D3_RAT Q8CFG5 CHEMBL3281 Voltage-gated Calcium Channel Alpha2/delta Subunit 3, Rat 4 3 3 2

Clustered By Gene (0)

Clustered By Organism (3)

Code Description Substances Purchasable Natural In Man
CA2D1-1-E Voltage-gated Calcium Channel Alpha2/delta Subunit 1 (cluster #1 Of 4), Eukaryotic 81 59 9 4
CA2D1-2-E Voltage-gated Calcium Channel Alpha2/delta Subunit 1 (cluster #2 Of 4), Eukaryotic 185 8 0 0
CA2D1-3-E Voltage-gated Calcium Channel Alpha2/delta Subunit 1 (cluster #3 Of 4), Eukaryotic 52 0 0 0
CA2D1-4-E Voltage-gated Calcium Channel Alpha2/delta Subunit 1 (cluster #4 Of 4), Eukaryotic 86 54 7 4
Uniprot Swissprot Chembl Description Number Shared
CAC1B_RAT Q02294 CHEMBL5107 Voltage-gated N-type Calcium Channel Alpha-1B Subunit, Rat 18
CACB1_RAT P54283 CHEMBL1075136 Voltage-dependent L-type Calcium Channel Subunit Beta-1, Rat 18
CA2D1_HUMAN P54289 CHEMBL1919 Voltage-gated Calcium Channel Alpha2/delta Subunit 1, Human 4
CA2D2_HUMAN Q9NY47 CHEMBL3896 Voltage-gated Calcium Channel Alpha2/delta Subunit 2, Human 4
CA2D2_RAT Q8CFG6 CHEMBL3914 Voltage-gated Calcium Channel Alpha2/delta Subunit 2, Rat 4
CA2D3_RAT Q8CFG5 CHEMBL3281 Voltage-gated Calcium Channel Alpha2/delta Subunit 3, Rat 4
CA2D3_HUMAN Q8IZS8 CHEMBL3763 Voltage-gated Calcium Channel Alpha2/delta Subunit 3, Human 3
CA2D4_HUMAN Q7Z3S7 CHEMBL5376 Voltage-gated Calcium Channel Alpha2/delta-4 Subunit, Human 3
CAC1B_HUMAN Q00975 CHEMBL4478 Voltage-gated N-type Calcium Channel Alpha-1B Subunit, Human 2
O77773_PIG O77773 CHEMBL3985 Voltage-dependent Calcium Channel Alpha2delta Subunit, Pig 2
P97706_RAT P97706 CHEMBL4957 Sodium Channel Protein Type VI Alpha Subunit, Rat 2
SCN5A_RAT P15389 CHEMBL3866 Sodium Channel Protein Type V Alpha Subunit, Rat 2
CA2D1_MOUSE O08532 CHEMBL4676 Voltage-gated Calcium Channel Alpha2/delta Subunit 1, Mouse 1
CAC1G_HUMAN O43497 CHEMBL4641 Voltage-gated T-type Calcium Channel Alpha-1G Subunit, Human 1
CAC1H_HUMAN O95180 CHEMBL1859 Voltage-gated T-type Calcium Channel Alpha-1H Subunit, Human 1
CAC1I_HUMAN Q9P0X4 CHEMBL5558 Voltage-gated T-type Calcium Channel Alpha-1I Subunit, Human 1
DRD2_RAT P61169 CHEMBL339 Dopamine D2 Receptor, Rat 1
OPRD_HUMAN P41143 CHEMBL236 Delta Opioid Receptor, Human 1
OPRK_HUMAN P41145 CHEMBL237 Kappa Opioid Receptor, Human 1
OPRM_HUMAN P35372 CHEMBL233 Mu Opioid Receptor, Human 1
SCN1A_HUMAN P35498 CHEMBL1845 Sodium Channel Protein Type I Alpha Subunit, Human 1
SCN1A_RAT P04774 CHEMBL4906 Sodium Channel Protein Type I Alpha Subunit, Rat 1
SCN2A_HUMAN Q99250 CHEMBL4187 Sodium Channel Protein Type II Alpha Subunit, Human 1
SCN2A_RAT P04775 CHEMBL3399 Sodium Channel Protein Type II Alpha Subunit, Rat 1
SCN3A_HUMAN Q9NY46 CHEMBL5163 Sodium Channel Protein Type III Alpha Subunit, Human 1
SCN3A_RAT P08104 CHEMBL4966 Sodium Channel Protein Type III Alpha Subunit, Rat 1
SCN8A_HUMAN Q9UQD0 CHEMBL5202 Sodium Channel Protein Type VIII Alpha Subunit, Human 1
SCN8A_RAT O88420 CHEMBL2752 Sodium Channel Protein Type VIII Alpha Subunit, Rat 1