UCSF

A-427 (Lung Carcinoma Cells) (119 Compounds)

Swissprot:
Z80019
Stitch:
Z80019
UniProt:
Z80019
ChEMBL:
CHEMBL614515

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Functional ≤ 10μM 119 13 10 6

Reactome Network (0)

Clustered By Gene (0)

Uniprot Swissprot Chembl Description Number Shared
Z80224 Z80224 CHEMBL387 MCF7 (Breast Carcinoma Cells) 107
Z80390 Z80390 CHEMBL390 PC-3 (Prostate Carcinoma Cells) 107
Z80682 Z80682 CHEMBL392 A549 (Lung Carcinoma Cells) 96
Z80712 Z80712 CHEMBL614361 T47D (Breast Carcinoma Cells) 91
Z80211 Z80211 CHEMBL614721 LoVo (Colon Adenocarcinoma Cells) 90
Z81335 Z81335 CHEMBL612263 HCT-15 (Colon Adenocarcinoma Cells) 90
Z80563 Z80563 CHEMBL615025 U-373 MG ( Glioblastoma Cells) 87
Z80565 Z80565 CHEMBL614247 U-87 MG (Glioblastoma Cells) 87
Z80179 Z80179 CHEMBL614586 J82 (Bladder Carcinoma Cells) 86
Z80532 Z80532 CHEMBL614774 T-24 (Bladder Carcinoma Cells) 70
Z80012 Z80012 CHEMBL614512 A 172 (Glioblastoma Cells) 31
Z80186 Z80186 CHEMBL385 K562 (Erythroleukemia Cells) 21
Z80522 Z80522 CHEMBL614243 SW1088 (Astrocytoma Cells) 17
Z80166 Z80166 CHEMBL384 HT-29 (Colon Adenocarcinoma Cells) 8
Z81017 Z81017 CHEMBL614647 WiDr (Colon Adenocarcinoma Cells) 7
Z80193 Z80193 CHEMBL386 L1210 (Lymphocytic Leukemia Cells) 6
Z80125 Z80125 CHEMBL613508 DU-145 (Prostate Carcinoma) 5
Z81170 Z81170 CHEMBL612518 LNCaP (Prostate Carcinoma) 5
Z81252 Z81252 CHEMBL400 MDA-MB-231 (Breast Adenocarcinoma Cells) 5
Z80056 Z80056 CHEMBL613852 CAKI-2 (Renal Carcinoma Cells) 4
Z80120 Z80120 CHEMBL614285 DLD-1 (Colon Adenocarcinoma Cells) 4
Z80164 Z80164 CHEMBL614580 HT-1080 (Fibrosarcoma Cells) 4
Z80354 Z80354 CHEMBL614213 OVCAR-3 (Ovarian Adenocarcinoma Cells) 4
Z80362 Z80362 CHEMBL389 P388 (Lymphoma Cells) 4
Z80485 Z80485 CHEMBL614919 SK-MEL-28 (Melanoma Cells) 4
Z80928 Z80928 CHEMBL394 HCT-116 (Colon Carcinoma Cells) 4
Z81248 Z81248 CHEMBL614021 Malme-3M (Melanoma Cells) 4
Z80014 Z80014 CHEMBL614514 A204 (Rhabdomyosarcoma Cells) 3
Z80021 Z80021 CHEMBL614516 A498 (Renal Carcinoma Cells) 3
Z80025 Z80025 CHEMBL614519 ACHN (Renal Adenocarcinoma Cells) 3
Z80045 Z80045 CHEMBL613870 BT-20 (Breast Carcinoma Cells) 3
Z80048 Z80048 CHEMBL614530 BXPC-3 (Pancreatic Adenocarcinoma Cells) 3
Z80064 Z80064 CHEMBL382 CCRF-CEM (T-cell Leukemia) 3
Z80086 Z80086 CHEMBL613506 CFPAC-1 (Pancreatic Carcinoma Cells) 3
Z80156 Z80156 CHEMBL383 HL-60 (Promyeloblast Leukemia Cells) 3
Z80254 Z80254 CHEMBL614343 MES-SA (Uterine Sarcoma Cells) 3
Z80269 Z80269 CHEMBL614354 MKN-45 (Gastric Adenocarcinoma Cells) 3
Z80316 Z80316 CHEMBL614771 NCI-H128 3
Z80381 Z80381 CHEMBL614139 PANC-1 (Pancreatic Carcinoma Cells) 3
Z80475 Z80475 CHEMBL613834 SK-BR-3 (Breast Adenocarcinoma) 3
Z80493 Z80493 CHEMBL614925 SK-OV-3 (Ovarian Carcinoma Cells) 3
Z80539 Z80539 CHEMBL614775 T98G (Glioblastoma Cells) 3
Z80608 Z80608 CHEMBL614393 ZR-75-1 (Breast Carcinoma Cells) 3
Z80640 Z80640 CHEMBL613102 786-0 (Renal Carcinoma Cells) 3
Z80661 Z80661 CHEMBL614567 A704 (Renal Carcinoma Cells) 3
Z80697 Z80697 CHEMBL614279 Bel-7402 (Hepatoma Cells) 3
Z80800 Z80800 CHEMBL614725 MIA PaCa-2 (Pancreatic Carcinoma Cells) 3
Z80847 Z80847 CHEMBL612250 FaDu (Pharyngeal Carcinoma Cells) 3
Z80891 Z80891 CHEMBL614804 H4 (Hepatoma Cells) 3
Z80991 Z80991 CHEMBL614645 Hs-578T (Breast Carcinoma Cells) 3
Z80996 Z80996 CHEMBL614836 HT1197 (Bladder Carcinoma Cells) 3
Z81024 Z81024 CHEMBL396 NCI-H460 (Non-small Cell Lung Carcinoma) 3
Z81184 Z81184 CHEMBL614096 LOX IMVI (Melanoma Cells) 3
Z81247 Z81247 CHEMBL399 HeLa (Cervical Adenocarcinoma Cells) 3
Z80026 Z80026 CHEMBL613860 AGS (Gastric Adenocarcinoma Cells) 2
Z80088 Z80088 CHEMBL613853 CHO (Ovarian Cells) 2
Z80119 Z80119 CHEMBL614059 Detroit 98 2
Z80145 Z80145 CHEMBL614045 H69 2
Z80152 Z80152 CHEMBL613510 HCT-8 (Ileocecal Adenocarcinoma) 2
Z80188 Z80188 CHEMBL614590 KB 3-1 (Cervical Epithelial Carcinoma Cells) 2
Z80285 Z80285 CHEMBL614177 MOLT-4 (Acute T-lymphoblastic Leukemia Cells) 2
Z80482 Z80482 CHEMBL614917 SK-MEL-2 (Melanoma Cells) 2
Z80495 Z80495 CHEMBL614927 SK-VLB 2
Z80526 Z80526 CHEMBL612544 SW480 (Colon Adenocarcinoma Cells) 2
Z80548 Z80548 CHEMBL614245 THP-1 (Acute Monocytic Leukemia Cells) 2
Z80623 Z80623 CHEMBL612911 Panel (56 Tumour Cell Lines) 2
Z80799 Z80799 CHEMBL612517 RPMI 8402 (Pre-T-lymphoblastoid Cells) 2
Z81020 Z81020 CHEMBL395 HepG2 (Hepatoblastoma Cells) 2
Z81034 Z81034 CHEMBL614004 A2780 (Ovarian Carcinoma Cells) 2
Z81084 Z81084 CHEMBL613992 KB VCR R 2
Z81115 Z81115 CHEMBL398 KB (Squamous Cell Carcinoma) 2
Z81131 Z81131 CHEMBL612266 L Cells (Fibroblasts) 2
Z81245 Z81245 CHEMBL614697 MDA-MB-435 (Breast Carcinoma Cells) 2
Z81331 Z81331 CHEMBL612262 SW-620 (Colon Adenocarcinoma Cells) 2
CHK1_HUMAN O14757 CHEMBL4630 Serine/threonine-protein Kinase Chk1, Human 1
SSR1_HUMAN P30872 CHEMBL1917 Somatostatin Receptor 1, Human 1
SSR2_HUMAN P30874 CHEMBL1804 Somatostatin Receptor 2, Human 1
SSR3_HUMAN P32745 CHEMBL2028 Somatostatin Receptor 3, Human 1
SSR4_HUMAN P31391 CHEMBL1853 Somatostatin Receptor 4, Human 1
SSR5_HUMAN P35346 CHEMBL1792 Somatostatin Receptor 5, Human 1
TOP1_HUMAN P11387 CHEMBL1781 DNA Topoisomerase I, Human 1
TOP1_MOUSE Q04750 CHEMBL2814 DNA Topoisomerase I, Mouse 1
TOP2A_HUMAN P11388 CHEMBL1806 DNA Topoisomerase II Alpha, Human 1
TOP2A_MOUSE Q01320 CHEMBL3586 DNA Topoisomerase II Alpha, Mouse 1
TOP2B_HUMAN Q02880 CHEMBL3396 DNA Topoisomerase II Beta, Human 1
TOP2B_MOUSE Q64511 CHEMBL5564 DNA Topoisomerase II Beta, Mouse 1
Z100501 Z100501 CHEMBL613290 Lu1 (Lung Carcinoma Cells) 1
Z100519 Z100519 CHEMBL614637 KETR3 (Renal Carcinoma Cells) 1
Z100733 Z100733 CHEMBL613866 CT26 (Colon Carcinoma Cells) 1
Z100752 Z100752 CHEMBL612568 Renca (Renal Carcinoma Cells) 1
Z103203 Z103203 CHEMBL1075388 A375 1
Z103205 Z103205 CHEMBL1075390 A431 1
Z103408 Z103408 CHEMBL1075593 SW626 1
Z103413 Z103413 CHEMBL1075598 SW948 1
Z50425 Z50425 CHEMBL364 Plasmodium Falciparum 1
Z80039 Z80039 CHEMBL614526 BGC-823 (Stomach Adenocarcinoma Cells) 1
Z80054 Z80054 CHEMBL614058 Caco-2 (Colon Adenocarcinoma Cells) 1
Z80068 Z80068 CHEMBL614542 CCRF-SB (Lymphoblastic Leukemia Cells) 1
Z80099 Z80099 CHEMBL614561 COLO 205 (Colon Adenocarcinoma Cells) 1
Z80105 Z80105 CHEMBL613854 COR-L23 (Lung Carcinoma Cells) 1
Z80115 Z80115 CHEMBL612702 DC3F 1
Z80295 Z80295 CHEMBL388 MT4 (Lymphocytes) 1
Z80372 Z80372 CHEMBL614224 P388CPT5 1
Z80414 Z80414 CHEMBL614628 Raji (B-lymphoblastic Cells) 1
Z80466 Z80466 CHEMBL614907 SF268 1
Z80559 Z80559 CHEMBL615021 U251 1
Z80596 Z80596 CHEMBL612811 WISH (Amniotic Epithelial Cells) 1
Z80647 Z80647 CHEMBL613103 833K Cell Line 1
Z80742 Z80742 CHEMBL614657 C6 (Glioma Cells) 1
Z80751 Z80751 CHEMBL614379 Caov-3 Cell Line 1
Z80784 Z80784 CHEMBL614462 Col2 (Colon Carcinoma Cells) 1
Z80874 Z80874 CHEMBL393 CEM (T-cell Leukemia) 1
Z80876 Z80876 CHEMBL614159 NCI-H125 1
Z80898 Z80898 CHEMBL614785 NCI-H928 1
Z80930 Z80930 CHEMBL614817 HEC-1B Cell Line 1
Z81054 Z81054 CHEMBL613977 SF-268 (Glioblastoma Cells) 1
Z81072 Z81072 CHEMBL397 Jurkat (Acute Leukemic T-cells) 1
Z81080 Z81080 CHEMBL613991 KATO-III Cell Line 1
Z81134 Z81134 CHEMBL614650 L2987 (Lung Adenocarcinoma Cells) 1
Z81160 Z81160 CHEMBL614088 Lewis Lung Carcinoma Cell Line 1
Z81164 Z81164 CHEMBL614091 LL Cell Line 1
Z81281 Z81281 CHEMBL614997 NCI-H23 (Non-small Cell Lung Carcinoma Cells) 1
Z81342 Z81342 CHEMBL614703 Tumour Cell Lines 1