| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 3,810 | 186 | 15 | 14 |
| Functional ≤ 10μM | 225 | 24 | 8 | 6 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| CNR1_HUMAN | P21554 | CHEMBL218 | Cannabinoid CB1 Receptor, Human | 2,791 | 161 | 19 | 12 |
| CNR1_MOUSE | P47746 | CHEMBL3037 | Cannabinoid CB1 Receptor, Mouse | 103 | 19 | 5 | 3 |
| CNR1_RAT | P20272 | CHEMBL3571 | Cannabinoid CB1 Receptor, Rat | 1,424 | 89 | 26 | 10 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| CNR1-2-E | Cannabinoid CB1 Receptor (cluster #2 Of 5), Eukaryotic | 68 | 14 | 9 | 3 |
| CNR1-3-E | Cannabinoid CB1 Receptor (cluster #3 Of 5), Eukaryotic | 290 | 38 | 12 | 1 |
| CNR1-4-E | Cannabinoid CB1 Receptor (cluster #4 Of 5), Eukaryotic | 3 | 0 | 0 | 0 |
| CNR1-5-E | Cannabinoid CB1 Receptor (cluster #5 Of 5), Eukaryotic | 18 | 3 | 1 | 1 |
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