| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 8 | 1 | 1 | 1 |
| Binding ≤ 1μM | 5 | 0 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| PCSK4_HUMAN | Q6UW60 | CHEMBL4861 | Subtilisin/kexin Type 4, Human | 0 | 0 | 0 | 0 |
| PCSK5_HUMAN | Q92824 | CHEMBL2826 | Subtilisin/kexin Type 5, Human | 5 | 0 | 0 | 0 |
| PCSK6_HUMAN | P29122 | CHEMBL2951 | Subtilisin/kexin Type 6, Human | 5 | 0 | 0 | 0 |
| PCSK9_HUMAN | Q8NBP7 | CHEMBL2929 | Subtilisin/kexin Type 9, Human | 0 | 0 | 0 | 0 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| PCSK7-1-E | Subtilisin/kexin Type 7 (cluster #1 Of 3), Eukaryotic | 1 | 1 | 1 | 1 |
| PCSK7-2-E | Subtilisin/kexin Type 7 (cluster #2 Of 3), Eukaryotic | 4 | 0 | 0 | 0 |
| PCSK7-3-E | Subtilisin/kexin Type 7 (cluster #3 Of 3), Eukaryotic | 3 | 0 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| FURIN_HUMAN | P09958 | CHEMBL2611 | Furin, Human | 3 |
| NEC1_HUMAN | P29120 | CHEMBL3182 | Prohormone Convertase 1, Human | 3 |
| NEC2_HUMAN | P16519 | CHEMBL2433 | Prohormone Convertase 2, Human | 3 |
| PCSK5_HUMAN | Q92824 | CHEMBL2826 | Subtilisin/kexin Type 5, Human | 3 |
| PCSK6_HUMAN | P29122 | CHEMBL2951 | Subtilisin/kexin Type 6, Human | 3 |
| NQO1_HUMAN | P15559 | CHEMBL3623 | Quinone Reductase 1), Human | 1 |
| PLMN_HUMAN | P00747 | CHEMBL1801 | Plasminogen, Human | 1 |