| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 21 | 8 | 9 | 7 |
| Functional ≤ 10μM | 6 | 1 | 1 | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| TRFR_HUMAN | P34981 | CHEMBL1810 | Thyrotropin-releasing Hormone Receptor, Human | 6 | 1 | 1 | 1 |
| TRFR_MOUSE | P21761 | CHEMBL2467 | Thyrotropin-releasing Hormone Receptor, Mouse | 9 | 3 | 4 | 2 |
| TRFR_RAT | Q01717 | CHEMBL4553 | Thyrotropin-releasing Hormone Receptor, Rat | 6 | 4 | 4 | 4 |