| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 4 | 4 | 4 | 2 |
| Binding ≤ 1μM | 1 | 1 | 1 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_15480 | ABC-family proteins mediated transport | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| MDR1_HUMAN | P08183 | CHEMBL4302 | P-glycoprotein 1, Human | 1 |
| MRP1_HUMAN | P33527 | CHEMBL3004 | Multidrug Resistance-associated Protein 1, Human | 3 |
| MRP3_HUMAN | O15438 | CHEMBL5918 | Canalicular Multispecific Organic Anion Transporter 2, Human | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| MRP1_HUMAN | P33527 | CHEMBL3004 | Multidrug Resistance-associated Protein 1, Human | 127 | 20 | 18 | 10 |
| MRP3_HUMAN | O15438 | CHEMBL5918 | Canalicular Multispecific Organic Anion Transporter 2, Human | 1 | 1 | 1 | 1 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| MRP1_HUMAN | P33527 | CHEMBL3004 | Multidrug Resistance-associated Protein 1, Human | 3 |
| CLTR1_HUMAN | Q9Y271 | CHEMBL1798 | Cysteinyl Leukotriene Receptor 1, Human | 2 |
| CLTR2_HUMAN | Q9NS75 | CHEMBL4330 | Cysteinyl Leukotriene Receptor 2, Human | 2 |
| ABCG2_HUMAN | Q9UNQ0 | CHEMBL5393 | ATP-binding Cassette Sub-family G Member 2, Human | 1 |
| CYSP_TRYCR | P25779 | CHEMBL3563 | Cruzipain, Trycr | 1 |
| MDR1_HUMAN | P08183 | CHEMBL4302 | P-glycoprotein 1, Human | 1 |
| MRP3_HUMAN | O15438 | CHEMBL5918 | Canalicular Multispecific Organic Anion Transporter 2, Human | 1 |