| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 12 | 3 | 2 | 3 |
| Binding ≤ 1μM | 11 | 3 | 2 | 3 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_160254 | Constitutive Signaling by NOTCH1 HD+PEST Domain Mutants | Homo sapiens |
| REACT_160243 | Constitutive Signaling by NOTCH1 PEST Domain Mutants | Homo sapiens |
| REACT_121111 | Downregulation of SMAD2/3:SMAD4 transcriptional activity | Homo sapiens |
| REACT_228222 | HDACs deacetylate histones | Homo sapiens |
| REACT_118780 | NOTCH1 Intracellular Domain Regulates Transcription | Homo sapiens |
| REACT_19241 | Regulation of lipid metabolism by Peroxisome proliferator-activated receptor alp | Homo sapiens |
| REACT_27161 | Transcriptional regulation of white adipocyte differentiation | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDA10_HUMAN | Q969S8 | CHEMBL5103 | Histone Deacetylase 10, Human | 3 |
| HDA11_HUMAN | Q96DB2 | CHEMBL3310 | Histone Deacetylase 11, Human | 3 |
| HDAC1_HUMAN | Q13547 | CHEMBL325 | Histone Deacetylase 1, Human | 9 |
| HDAC2_HUMAN | Q92769 | CHEMBL1937 | Histone Deacetylase 2, Human | 10 |
| HDAC3_HUMAN | O15379 | CHEMBL1829 | Histone Deacetylase 3, Human | 12 |
| HDAC4_HUMAN | P56524 | CHEMBL3524 | Histone Deacetylase 4, Human | 5 |
| HDAC5_HUMAN | Q9UQL6 | CHEMBL2563 | Histone Deacetylase 5, Human | 4 |
| HDAC6_HUMAN | Q9UBN7 | CHEMBL1865 | Histone Deacetylase 6, Human | 9 |
| HDAC7_HUMAN | Q8WUI4 | CHEMBL2716 | Histone Deacetylase 7, Human | 5 |
| HDAC8_HUMAN | Q9BY41 | CHEMBL3192 | Histone Deacetylase 8, Human | 9 |
| HDAC9_HUMAN | Q9UKV0 | CHEMBL4145 | Histone Deacetylase 9, Human | 4 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDA10_HUMAN | Q969S8 | CHEMBL5103 | Histone Deacetylase 10, Human | 3 |
| HDA11_HUMAN | Q96DB2 | CHEMBL3310 | Histone Deacetylase 11, Human | 3 |
| HDAC1_HUMAN | Q13547 | CHEMBL325 | Histone Deacetylase 1, Human | 9 |
| HDAC2_HUMAN | Q92769 | CHEMBL1937 | Histone Deacetylase 2, Human | 10 |
| HDAC3_HUMAN | O15379 | CHEMBL1829 | Histone Deacetylase 3, Human | 12 |
| HDAC4_HUMAN | P56524 | CHEMBL3524 | Histone Deacetylase 4, Human | 5 |
| HDAC5_HUMAN | Q9UQL6 | CHEMBL2563 | Histone Deacetylase 5, Human | 4 |
| HDAC6_HUMAN | Q9UBN7 | CHEMBL1865 | Histone Deacetylase 6, Human | 9 |
| HDAC7_HUMAN | Q8WUI4 | CHEMBL2716 | Histone Deacetylase 7, Human | 5 |
| HDAC8_HUMAN | Q9BY41 | CHEMBL3192 | Histone Deacetylase 8, Human | 9 |
| HDAC9_HUMAN | Q9UKV0 | CHEMBL4145 | Histone Deacetylase 9, Human | 4 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDAC1_HUMAN | Q13547 | CHEMBL325 | Histone Deacetylase 1, Human | 9 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDA10_HUMAN | Q969S8 | CHEMBL5103 | Histone Deacetylase 10, Human | 3 |
| HDAC1_HUMAN | Q13547 | CHEMBL325 | Histone Deacetylase 1, Human | 9 |
| HDAC2_HUMAN | Q92769 | CHEMBL1937 | Histone Deacetylase 2, Human | 10 |
| HDAC3_HUMAN | O15379 | CHEMBL1829 | Histone Deacetylase 3, Human | 12 |
| HDAC8_HUMAN | Q9BY41 | CHEMBL3192 | Histone Deacetylase 8, Human | 9 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDA10_HUMAN | Q969S8 | CHEMBL5103 | Histone Deacetylase 10, Human | 3 |
| HDA11_HUMAN | Q96DB2 | CHEMBL3310 | Histone Deacetylase 11, Human | 3 |
| HDAC1_HUMAN | Q13547 | CHEMBL325 | Histone Deacetylase 1, Human | 9 |
| HDAC2_HUMAN | Q92769 | CHEMBL1937 | Histone Deacetylase 2, Human | 10 |
| HDAC3_HUMAN | O15379 | CHEMBL1829 | Histone Deacetylase 3, Human | 12 |
| HDAC4_HUMAN | P56524 | CHEMBL3524 | Histone Deacetylase 4, Human | 5 |
| HDAC5_HUMAN | Q9UQL6 | CHEMBL2563 | Histone Deacetylase 5, Human | 4 |
| HDAC6_HUMAN | Q9UBN7 | CHEMBL1865 | Histone Deacetylase 6, Human | 9 |
| HDAC7_HUMAN | Q8WUI4 | CHEMBL2716 | Histone Deacetylase 7, Human | 5 |
| HDAC8_HUMAN | Q9BY41 | CHEMBL3192 | Histone Deacetylase 8, Human | 9 |
| HDAC9_HUMAN | Q9UKV0 | CHEMBL4145 | Histone Deacetylase 9, Human | 4 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDAC3_HUMAN | O15379 | CHEMBL1829 | Histone Deacetylase 3, Human | 12 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDAC3_HUMAN | O15379 | CHEMBL1829 | Histone Deacetylase 3, Human | 12 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| NCOR2-1-E | Nuclear Receptor Corepressor 2 (cluster #1 Of 2), Eukaryotic | 8 | 2 | 2 | 2 |
| NCOR2-2-E | Nuclear Receptor Corepressor 2 (cluster #2 Of 2), Eukaryotic | 4 | 1 | 0 | 1 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| HDAC3_HUMAN | O15379 | CHEMBL1829 | Histone Deacetylase 3, Human | 12 |
| HDAC2_HUMAN | Q92769 | CHEMBL1937 | Histone Deacetylase 2, Human | 10 |
| HDAC1_HUMAN | Q13547 | CHEMBL325 | Histone Deacetylase 1, Human | 9 |
| HDAC6_HUMAN | Q9UBN7 | CHEMBL1865 | Histone Deacetylase 6, Human | 9 |
| HDAC8_HUMAN | Q9BY41 | CHEMBL3192 | Histone Deacetylase 8, Human | 9 |
| HDAC4_HUMAN | P56524 | CHEMBL3524 | Histone Deacetylase 4, Human | 5 |
| HDAC7_HUMAN | Q8WUI4 | CHEMBL2716 | Histone Deacetylase 7, Human | 5 |
| HDAC5_HUMAN | Q9UQL6 | CHEMBL2563 | Histone Deacetylase 5, Human | 4 |
| HDAC9_HUMAN | Q9UKV0 | CHEMBL4145 | Histone Deacetylase 9, Human | 4 |
| HDA10_HUMAN | Q969S8 | CHEMBL5103 | Histone Deacetylase 10, Human | 3 |
| HDA11_HUMAN | Q96DB2 | CHEMBL3310 | Histone Deacetylase 11, Human | 3 |
| HDAH_ALCSD | Q70I53 | CHEMBL6017 | Histone Deacetylase-like Amidohydrolase, Alcsd | 3 |
| Q9XYC7_PLAFA | Q9XYC7 | CHEMBL5541 | Histone Deacetylase, Plafa | 3 |
| B1WBY8_RAT | B1WBY8 | CHEMBL4705 | Histone Deacetylase 2, Rat | 2 |
| HDAC1_MOUSE | O09106 | CHEMBL4001 | Histone Deacetylase 1, Mouse | 2 |
| HDAC1_RAT | Q4QQW4 | CHEMBL2915 | Histone Deacetylase 1, Rat | 2 |
| HDAC3_RAT | Q6P6W3 | CHEMBL2628 | Histone Deacetylase 3, Rat | 2 |
| HDAC4_RAT | Q99P99 | CHEMBL2874 | Histone Deacetylase 4, Rat | 2 |
| HDAC7_RAT | Q99P96 | CHEMBL2914 | Histone Deacetylase 7, Rat | 2 |
| Q5RJZ2_RAT | Q5RJZ2 | CHEMBL4025 | Histone Deacetylase 5, Rat | 2 |
| Q94F81_MAIZE | Q94F81 | CHEMBL4919 | Histone Deacetylase HD2, Maize | 2 |
| Q99P97_RAT | Q99P97 | CHEMBL3101 | Histone Deacetylase 6, Rat | 2 |
| Q9ZTP8_MAIZE | Q9ZTP8 | CHEMBL3541 | Histone Deacetylase HD1B, Maize | 2 |
| TF_HUMAN | P13726 | CHEMBL4081 | Coagulation Factor III, Human | 2 |
| HDA11_MOUSE | Q91WA3 | CHEMBL5143 | Histone Deacetylase 11, Mouse | 1 |
| HDAC1_CHICK | P56517 | CHEMBL4582 | Histone Deacetylase 1, Chick | 1 |
| HDAC2_CHICK | P56519 | CHEMBL4583 | Histone Deacetylase 2, Chick | 1 |
| HDAC2_MOUSE | P70288 | CHEMBL4238 | Histone Deacetylase 2, Mouse | 1 |
| HDAC3_CHICK | P56520 | CHEMBL4584 | Histone Deacetylase 3, Chick | 1 |
| HDAC3_MOUSE | O88895 | CHEMBL5142 | Histone Deacetylase 3, Mouse | 1 |
| HDAC4_CHICK | P83038 | CHEMBL5599 | Histone Deacetylase 4, Chick | 1 |
| HDAC5_MOUSE | Q9Z2V6 | CHEMBL2768 | Histone Deacetylase 5, Mouse | 1 |
| HDAC6_MOUSE | Q9Z2V5 | CHEMBL2878 | Histone Deacetylase 6, Mouse | 1 |
| HDAC7_MOUSE | Q8C2B3 | CHEMBL4219 | Histone Deacetylase 7, Mouse | 1 |
| HDAC8_MOUSE | Q8VH37 | CHEMBL2347 | Histone Deacetylase 8, Mouse | 1 |
| HDAC9_MOUSE | Q99N13 | CHEMBL5204 | Histone Deacetylase 9, Mouse | 1 |
| Q7K6A1_PLAF7 | Q7K6A1 | CHEMBL1293190 | Histone Deacetylase, Plaf7 | 1 |
| Q7YY07_CRYPV | Q7YY07 | CHEMBL4740 | Histone Deacetylase, Crypv | 1 |
| Q7YY76_CRYPV | Q7YY76 | CHEMBL3626 | Histone Deacetylase, Crypv | 1 |
| SF3B3_HUMAN | Q15393 | CHEMBL1250378 | Splicing Factor 3B Subunit 3, Human | 1 |