UCSF

Urotensin II Receptor, Human (219 Compounds)

Swissprot:
UR2R_HUMAN
Stitch:
UR2R_HUMAN
UniProt:
Q9UKP6
ChEMBL:
CHEMBL3764
Reactome:
REACT_18283
REACT_14819
PDB:
UTS2R

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 219 1 0 1
Binding ≤ 1μM 202 0 0 1
Functional ≤ 10μM 49 2 0 1

Reactome Network (2)

Uniprot Swissprot Chembl Description Number Shared
5HT2B_HUMAN P41595 CHEMBL1833 Serotonin 2b (5-HT2b) Receptor, Human 1
5HT2C_HUMAN P28335 CHEMBL225 Serotonin 2c (5-HT2c) Receptor, Human 1
UTS2_HUMAN O95399 CHEMBL6165 Urotensin-2, Human 1

Peptide ligand-binding receptors

Uniprot Swissprot Chembl Description Number Shared
OPRD_HUMAN P41143 CHEMBL236 Delta Opioid Receptor, Human 1
OPRK_HUMAN P41145 CHEMBL237 Kappa Opioid Receptor, Human 74
OPRM_HUMAN P35372 CHEMBL233 Mu Opioid Receptor, Human 1
UTS2_HUMAN O95399 CHEMBL6165 Urotensin-2, Human 1
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
UR2R_RAT P49684 CHEMBL4921 Urotensin II Receptor, Rat 3 0 0 0

Clustered By Gene (0)

Uniprot Swissprot Chembl Description Number Shared
UR2R_RAT P49684 CHEMBL4921 Urotensin II Receptor, Rat 32
Q533H1_FELCA Q533H1 CHEMBL5226 Urotensin II Receptor, Felca 10
5HT1A_HUMAN P08908 CHEMBL214 Serotonin 1a (5-HT1a) Receptor, Human 1
5HT1D_HUMAN P28221 CHEMBL1983 Serotonin 1d (5-HT1d) Receptor, Human 1
5HT1F_HUMAN P30939 CHEMBL1805 Serotonin 1f (5-HT1f) Receptor, Human 1
5HT2B_HUMAN P41595 CHEMBL1833 Serotonin 2b (5-HT2b) Receptor, Human 1
5HT2C_HUMAN P28335 CHEMBL225 Serotonin 2c (5-HT2c) Receptor, Human 1
5HT6R_HUMAN P50406 CHEMBL3371 Serotonin 6 (5-HT6) Receptor, Human 1
DRD2_HUMAN P14416 CHEMBL217 Dopamine D2 Receptor, Human 1
KCNH2_HUMAN Q12809 CHEMBL240 HERG, Human 1
OPRD_HUMAN P41143 CHEMBL236 Delta Opioid Receptor, Human 1
OPRK_CAVPO P41144 CHEMBL3952 Kappa Opioid Receptor, Guinea Pig 1
OPRK_HUMAN P41145 CHEMBL237 Kappa Opioid Receptor, Human 1
OPRK_MOUSE P33534 CHEMBL4329 Kappa Opioid Receptor, Mouse 1
OPRM_CAVPO P97266 CHEMBL4354 Mu Opioid Receptor, Guinea Pig 1
OPRM_HUMAN P35372 CHEMBL233 Mu Opioid Receptor, Human 1
UTS2_HUMAN O95399 CHEMBL6165 Urotensin-2, Human 1
UTS2_MACMU Q8HYC2 CHEMBL1163107 Urotensin-2, Macmu 1