 
| Annotation Type | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|
| Binding ≤ 10μM | 6,188 | 278 | 58 | 40 | 
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|---|---|---|
| AA1R_BOVIN | P28190 | CHEMBL4975 | Adenosine A1 Receptor, Bovin | 714 | 56 | 10 | 8 | 
| AA1R_CHICK | P49892 | CHEMBL2114 | Adenosine A1 Receptor, Chick | 24 | 3 | 0 | 1 | 
| AA1R_HUMAN | P30542 | CHEMBL226 | Adenosine A1 Receptor, Human | 2,632 | 98 | 19 | 17 | 
| AA1R_MOUSE | Q60612 | CHEMBL3688 | Adenosine A1 Receptor, Mouse | 25 | 3 | 1 | 2 | 
| AA1R_RAT | P25099 | CHEMBL318 | Adenosine A1 Receptor, Rat | 3,254 | 205 | 59 | 36 | 
| Code | Description | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|---|
| AA1R-1-E | Adenosine A1 Receptor (cluster #1 Of 4), Eukaryotic | 101 | 19 | 9 | 5 | 
| AA1R-3-E | Adenosine A1 Receptor (cluster #3 Of 4), Eukaryotic | 12 | 6 | 4 | 1 | 
| AA1R-4-E | Adenosine A1 Receptor (cluster #4 Of 4), Eukaryotic | 4 | 0 | 0 | 0 | 
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