| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 714 | 56 | 10 | 8 |
| Binding ≤ 1μM | 580 | 48 | 8 | 6 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_217608 | Adenosine P1 receptors | Bos taurus |
| REACT_210568 | G alpha (i) signalling events | Bos taurus |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| AA1R_CHICK | P49892 | CHEMBL2114 | Adenosine A1 Receptor, Chick | 24 | 3 | 0 | 1 |
| AA1R_HUMAN | P30542 | CHEMBL226 | Adenosine A1 Receptor, Human | 2,632 | 98 | 19 | 17 |
| AA1R_MOUSE | Q60612 | CHEMBL3688 | Adenosine A1 Receptor, Mouse | 25 | 3 | 1 | 2 |
| AA1R_RAT | P25099 | CHEMBL318 | Adenosine A1 Receptor, Rat | 3,254 | 205 | 59 | 36 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| AA1R-1-E | Adenosine A1 Receptor (cluster #1 Of 4), Eukaryotic | 101 | 19 | 9 | 5 |
| AA1R-2-E | Adenosine A1 Receptor (cluster #2 Of 4), Eukaryotic | 6,188 | 278 | 58 | 40 |
| AA1R-3-E | Adenosine A1 Receptor (cluster #3 Of 4), Eukaryotic | 12 | 6 | 4 | 1 |
| AA1R-4-E | Adenosine A1 Receptor (cluster #4 Of 4), Eukaryotic | 4 | 0 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| AA2AR_HUMAN | P29274 | CHEMBL251 | Adenosine A2a Receptor, Human | 209 |
| AA3R_HUMAN | P33765 | CHEMBL256 | Adenosine A3 Receptor, Human | 187 |
| AA1R_HUMAN | P30542 | CHEMBL226 | Adenosine A1 Receptor, Human | 122 |
| AA1R_RAT | P25099 | CHEMBL318 | Adenosine A1 Receptor, Rat | 121 |
| AA2AR_RAT | P30543 | CHEMBL302 | Adenosine A2a Receptor, Rat | 60 |
| AA3R_RAT | P28647 | CHEMBL3360 | Adenosine A3 Receptor, Rat | 46 |
| AA2BR_RAT | P29276 | CHEMBL2592 | Adenosine A2b Receptor, Rat | 44 |
| AA2BR_HUMAN | P29275 | CHEMBL255 | Adenosine A2b Receptor, Human | 38 |
| Q4VQ11_PIG | Q4VQ11 | CHEMBL1075029 | A1 Adenosine Receptor, Pig | 31 |
| ADCY2_RAT | P26769 | CHEMBL2958 | Adenylate Cyclase Type II, Rat | 16 |
| GBRA1_BOVIN | P08219 | CHEMBL3627 | GABA Receptor Alpha-1 Subunit, Bovin | 13 |
| GBRA2_BOVIN | P10063 | CHEMBL2321 | GABA Receptor Alpha-2 Subunit, Bovin | 13 |
| GBRA3_BOVIN | P10064 | CHEMBL3628 | GABA Receptor Alpha-3 Subunit, Bovin | 13 |
| GBRA4_BOVIN | P20237 | CHEMBL3140 | GABA Receptor Alpha-4 Subunit, Bovin | 13 |
| GBRB1_BOVIN | P08220 | CHEMBL2848 | GABA Receptor Beta-1 Subunit, Bovin | 13 |
| GBRG2_BOVIN | P22300 | CHEMBL5138 | GABA Receptor Gamma-2 Subunit, Bovin | 13 |
| AA2AR_CAVPO | P46616 | CHEMBL2605 | Adenosine A2a Receptor, Guinea Pig | 10 |
| Z50597 | Z50597 | CHEMBL376 | Rattus Norvegicus | 10 |
| ADCY3_RAT | P21932 | CHEMBL4864 | Adenylate Cyclase Type III, Rat | 6 |
| ADCY4_RAT | P26770 | CHEMBL2879 | Adenylate Cyclase Type IV, Rat | 6 |
| ADCY5_RAT | Q04400 | CHEMBL2880 | Adenylate Cyclase Type V, Rat | 6 |
| ADCY6_RAT | Q03343 | CHEMBL2975 | Adenylate Cyclase Type VI, Rat | 6 |
| ADCY8_RAT | P40146 | CHEMBL3082 | Adenylate Cyclase Type VIII, Rat | 6 |
| AA1R_MOUSE | Q60612 | CHEMBL3688 | Adenosine A1 Receptor, Mouse | 4 |
| AA1R_CHICK | P49892 | CHEMBL2114 | Adenosine A1 Receptor, Chick | 3 |
| AA2AR_MOUSE | Q60613 | CHEMBL2115 | Adenosine A2a Receptor, Mouse | 2 |
| AA3R_MOUSE | Q61618 | CHEMBL1075269 | Adenosine Receptor A3, Mouse | 2 |
| OXGR1_RAT | Q6Y1R5 | CHEMBL2325 | G Protein-coupled Receptor 80, Rat | 1 |
| PDE1A_BOVIN | P14100 | CHEMBL3774 | Phosphodiesterase 1A, Bovin | 1 |
| PDE1A_HUMAN | P54750 | CHEMBL3421 | Phosphodiesterase 1A, Human | 1 |
| PDE1B_BOVIN | Q01061 | CHEMBL2650 | Phosphodiesterase 1B, Bovin | 1 |
| PDE1B_HUMAN | Q01064 | CHEMBL4425 | Phosphodiesterase 1B, Human | 1 |
| PDE1C_HUMAN | Q14123 | CHEMBL4619 | Phosphodiesterase 1C, Human | 1 |
| PDE3A_HUMAN | Q14432 | CHEMBL241 | Phosphodiesterase 3A, Human | 1 |
| PDE3B_HUMAN | Q13370 | CHEMBL290 | Phosphodiesterase 3B, Human | 1 |
| PDE4A_HUMAN | P27815 | CHEMBL254 | Phosphodiesterase 4A, Human | 1 |
| PDE4B_HUMAN | Q07343 | CHEMBL275 | Phosphodiesterase 4B, Human | 1 |
| PDE4C_HUMAN | Q08493 | CHEMBL291 | Phosphodiesterase 4C, Human | 1 |
| PDE4D_HUMAN | Q08499 | CHEMBL288 | Phosphodiesterase 4D, Human | 1 |
| PDE5A_HUMAN | O76074 | CHEMBL1827 | Phosphodiesterase 5A, Human | 1 |
| PDE7A_HUMAN | Q13946 | CHEMBL3012 | Phosphodiesterase 7A, Human | 1 |
| PDE7B_HUMAN | Q9NP56 | CHEMBL4716 | Phosphodiesterase 7B, Human | 1 |
| S29A1_HUMAN | Q99808 | CHEMBL1997 | Equilibrative Nucleoside Transporter 1, Human | 1 |
| SCN1A_HUMAN | P35498 | CHEMBL1845 | Sodium Channel Protein Type I Alpha Subunit, Human | 1 |
| SCN2A_HUMAN | Q99250 | CHEMBL4187 | Sodium Channel Protein Type II Alpha Subunit, Human | 1 |
| SCN3A_HUMAN | Q9NY46 | CHEMBL5163 | Sodium Channel Protein Type III Alpha Subunit, Human | 1 |
| SCN8A_HUMAN | Q9UQD0 | CHEMBL5202 | Sodium Channel Protein Type VIII Alpha Subunit, Human | 1 |
| Z100273 | Z100273 | CHEMBL612413 | P3 Purinoceptor | 1 |
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse
Browse