| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Functional ≤ 10μM | 11 | 1 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_18319 | Class C/3 (Metabotropic glutamate/pheromone receptors) | Homo sapiens |
| REACT_19231 | G alpha (i) signalling events | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| GRM1_HUMAN | Q13255 | CHEMBL3772 | Metabotropic Glutamate Receptor 1, Human | 3 |
| GRM2_HUMAN | Q14416 | CHEMBL5137 | Metabotropic Glutamate Receptor 2, Human | 1 |
| GRM3_HUMAN | Q14832 | CHEMBL2888 | Metabotropic Glutamate Receptor 3, Human | 1 |
| GRM4_HUMAN | Q14833 | CHEMBL2736 | Metabotropic Glutamate Receptor 4, Human | 4 |
| GRM5_HUMAN | P41594 | CHEMBL3227 | Metabotropic Glutamate Receptor 5, Human | 3 |
| GRM8_HUMAN | O00222 | CHEMBL3228 | Metabotropic Glutamate Receptor 8, Human | 11 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| GRM2_HUMAN | Q14416 | CHEMBL5137 | Metabotropic Glutamate Receptor 2, Human | 1 |
| GRM3_HUMAN | Q14832 | CHEMBL2888 | Metabotropic Glutamate Receptor 3, Human | 1 |
| GRM4_HUMAN | Q14833 | CHEMBL2736 | Metabotropic Glutamate Receptor 4, Human | 4 |
| GRM8_HUMAN | O00222 | CHEMBL3228 | Metabotropic Glutamate Receptor 8, Human | 11 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GRM7_MOUSE | Q68ED2 | CHEMBL3966 | Metabotropic Glutamate Receptor 7, Mouse | 5 | 3 | 1 | 1 |
| GRM7_RAT | P35400 | CHEMBL3879 | Metabotropic Glutamate Receptor 7, Rat | 5 | 2 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GRM1_HUMAN | Q13255 | CHEMBL3772 | Metabotropic Glutamate Receptor 1, Human | 51 | 12 | 6 | 4 |
| GRM2_HUMAN | Q14416 | CHEMBL5137 | Metabotropic Glutamate Receptor 2, Human | 293 | 14 | 4 | 3 |
| GRM3_HUMAN | Q14832 | CHEMBL2888 | Metabotropic Glutamate Receptor 3, Human | 14 | 5 | 2 | 2 |
| GRM4_HUMAN | Q14833 | CHEMBL2736 | Metabotropic Glutamate Receptor 4, Human | 137 | 45 | 3 | 3 |
| GRM5_HUMAN | P41594 | CHEMBL3227 | Metabotropic Glutamate Receptor 5, Human | 523 | 45 | 4 | 4 |
| GRM6_HUMAN | O15303 | CHEMBL4573 | Metabotropic Glutamate Receptor 6, Human | 4 | 3 | 1 | 1 |
| GRM8_HUMAN | O00222 | CHEMBL3228 | Metabotropic Glutamate Receptor 8, Human | 5 | 3 | 1 | 1 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| GRM8_HUMAN | O00222 | CHEMBL3228 | Metabotropic Glutamate Receptor 8, Human | 11 |
| GRM2_RAT | P31421 | CHEMBL2851 | Metabotropic Glutamate Receptor 2, Rat | 9 |
| GRM3_RAT | P31422 | CHEMBL3067 | Metabotropic Glutamate Receptor 3, Rat | 9 |
| GRM4_HUMAN | Q14833 | CHEMBL2736 | Metabotropic Glutamate Receptor 4, Human | 4 |
| GRM1_HUMAN | Q13255 | CHEMBL3772 | Metabotropic Glutamate Receptor 1, Human | 3 |
| GRM5_HUMAN | P41594 | CHEMBL3227 | Metabotropic Glutamate Receptor 5, Human | 3 |
| GRM2_HUMAN | Q14416 | CHEMBL5137 | Metabotropic Glutamate Receptor 2, Human | 1 |
| GRM3_HUMAN | Q14832 | CHEMBL2888 | Metabotropic Glutamate Receptor 3, Human | 1 |