| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 99 | 1 | 0 | 0 |
| Binding ≤ 1μM | 83 | 0 | 0 | 0 |
| Functional ≤ 10μM | 17 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_250376 | G alpha (i) signalling events | Mus musculus |
| REACT_207651 | G alpha (q) signalling events | Mus musculus |
| REACT_235286 | Peptide ligand-binding receptors | Mus musculus |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| MCHR1_HUMAN | Q99705 | CHEMBL344 | Melanin-concentrating Hormone Receptor 1, Human | 2,286 | 34 | 0 | 0 |
| MCHR1_RAT | P97639 | CHEMBL1075228 | Melanin-concentrating Hormone Receptor 1, Rat | 52 | 0 | 0 | 0 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| MCHR1-1-E | Melanin-concentrating Hormone Receptor 1 (cluster #1 Of 2), Eukaryotic | 1,937 | 18 | 0 | 0 |
| MCHR1-2-E | Melanin-concentrating Hormone Receptor 1 (cluster #2 Of 2), Eukaryotic | 441 | 17 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| MCHR1_HUMAN | Q99705 | CHEMBL344 | Melanin-concentrating Hormone Receptor 1, Human | 34 |
| 5HT2B_HUMAN | P41595 | CHEMBL1833 | Serotonin 2b (5-HT2b) Receptor, Human | 4 |
| 5HT2A_HUMAN | P28223 | CHEMBL224 | Serotonin 2a (5-HT2a) Receptor, Human | 1 |
| 5HT2C_HUMAN | P28335 | CHEMBL225 | Serotonin 2c (5-HT2c) Receptor, Human | 1 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 1 |
| MCHR1_RAT | P97639 | CHEMBL1075228 | Melanin-concentrating Hormone Receptor 1, Rat | 1 |