| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 830 | 25 | 13 | 8 |
| Functional ≤ 10μM | 2 | 0 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GBRA5_HUMAN | P31644 | CHEMBL5112 | GABA Receptor Alpha-5 Subunit, Human | 957 | 69 | 31 | 18 |
| GBRA5_MOUSE | Q8BHJ7 | CHEMBL2304 | GABA Receptor Alpha-5 Subunit, Mouse | 37 | 3 | 2 | 2 |
| GBRA5_RAT | P19969 | CHEMBL300 | GABA Receptor Alpha-5 Subunit, Rat | 189 | 15 | 11 | 7 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| GBRA5-2-E | GABA Receptor Alpha-5 Subunit (cluster #2 Of 8), Eukaryotic | 24 | 4 | 4 | 3 |
| GBRA5-3-E | GABA Receptor Alpha-5 Subunit (cluster #3 Of 8), Eukaryotic | 154 | 16 | 7 | 2 |
| GBRA5-4-E | GABA Receptor Alpha-5 Subunit (cluster #4 Of 8), Eukaryotic | 3 | 0 | 0 | 0 |
| GBRA5-5-E | GABA Receptor Alpha-5 Subunit (cluster #5 Of 8), Eukaryotic | 4 | 4 | 1 | 1 |
| GBRA5-6-E | GABA Receptor Alpha-5 Subunit (cluster #6 Of 8), Eukaryotic | 134 | 30 | 16 | 10 |
| GBRA5-7-E | GABA Receptor Alpha-5 Subunit (cluster #7 Of 8), Eukaryotic | 30 | 0 | 0 | 0 |
| GBRA5-8-E | GABA Receptor Alpha-5 Subunit (cluster #8 Of 8), Eukaryotic | 4 | 4 | 1 | 1 |
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