ZINC 12

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Quick Search ZINC ID or SMILES

Names
Compounds (81)
Reactome (0)
Related By:
Pathway (0)
Organism (5)
Gene (0)
Org. Clust. (2)
ChEMBL (73)
Rings (21)

Serotonin 2a (5-HT2a) Receptor, Pig (81 Compounds)

Swissprot:: 5HT2A_PIG
Stitch:: 5HT2A_PIG
UniProt:: P50129
ChEMBL:: CHEMBL2490
PDB:: HTR2A

Compound Summary

Annotation Type	Substances	Purchasable	Natural	In Man
Binding ≤ 10μM	81	6	1	1
Binding ≤ 1μM	48	3	1	1

UniProt	Swissprot	ChEMBL	Description	Substances	Purchasable	Natural	In Man
5HT2A_BOVIN	Q75Z89	CHEMBL3446	Serotonin 2a (5-HT2a) Receptor, Bovin	134	13	9	11
5HT2A_CANFA	O46635	CHEMBL5781	5-hydroxytryptamine Receptor 2A, Canine	1	0	0	0
5HT2A_HUMAN	P28223	CHEMBL224	Serotonin 2a (5-HT2a) Receptor, Human	2,122	202	55	44
5HT2A_MOUSE	P35363	CHEMBL5377	Serotonin 2a (5-HT2a) Receptor, Mouse	169	9	6	6
5HT2A_RAT	P14842	CHEMBL322	Serotonin 2a (5-HT2a) Receptor, Rat	2,538	306	92	100

Clustered By Gene (0)

Clustered By Organism (2)

Code	Description	Substances	Purchasable	Natural	In Man
5HT2A-1-E	Serotonin 2a (5-HT2a) Receptor (cluster #1 Of 3), Eukaryotic	4,353	322	100	96
5HT2A-2-E	Serotonin 2a (5-HT2a) Receptor (cluster #2 Of 3), Eukaryotic	530	142	16	25
5HT2A-3-E	Serotonin 2a (5-HT2a) Receptor (cluster #3 Of 3), Eukaryotic	18	2	1	1

Uniprot	Swissprot	Chembl	Description	Number Shared
DRD3_HUMAN	P35462	CHEMBL234	Dopamine D3 Receptor, Human	79
DRD2_HUMAN	P14416	CHEMBL217	Dopamine D2 Receptor, Human	76
DRD1_PIG	P50130	CHEMBL5067	Dopamine D1 Receptor, Pig	72
DRD4_HUMAN	P21917	CHEMBL219	Dopamine D4 Receptor, Human	37
5HT1A_HUMAN	P08908	CHEMBL214	Serotonin 1a (5-HT1a) Receptor, Human	36
ADA1A_HUMAN	P35348	CHEMBL229	Alpha-1a Adrenergic Receptor, Human	26
ADA1B_HUMAN	P35368	CHEMBL232	Alpha-1b Adrenergic Receptor, Human	26
ADA1D_HUMAN	P25100	CHEMBL223	Alpha-1d Adrenergic Receptor, Human	26
5HT2C_HUMAN	P28335	CHEMBL225	Serotonin 2c (5-HT2c) Receptor, Human	24
5HT2B_HUMAN	P41595	CHEMBL1833	Serotonin 2b (5-HT2b) Receptor, Human	20
DRD1_BOVIN	Q95136	CHEMBL2967	Dopamine D1 Receptor, Bovin	7
DRD1_HUMAN	P21728	CHEMBL2056	Dopamine D1 Receptor, Human	7
5HT2A_HUMAN	P28223	CHEMBL224	Serotonin 2a (5-HT2a) Receptor, Human	5
DRD2_RAT	P61169	CHEMBL339	Dopamine D2 Receptor, Rat	3
DRD3_RAT	P19020	CHEMBL3138	Dopamine D3 Receptor, Rat	3
DRD2_BOVIN	P20288	CHEMBL3998	Dopamine D2 Receptor, Bovin	2
HRH1_HUMAN	P35367	CHEMBL231	Histamine H1 Receptor, Human	2
KCNH2_HUMAN	Q12809	CHEMBL240	HERG, Human	2
5HT1A_RAT	P19327	CHEMBL273	Serotonin 1a (5-HT1a) Receptor, Rat	1
5HT1B_RAT	P28564	CHEMBL3459	Serotonin 1b (5-HT1b) Receptor, Rat	1
5HT1D_RAT	P28565	CHEMBL5450	Serotonin 1d (5-HT1d) Receptor, Rat	1
5HT1E_HUMAN	P28566	CHEMBL2182	Serotonin 1e (5-HT1e) Receptor, Human	1
5HT1F_RAT	P30940	CHEMBL4646	Serotonin 1f (5-HT1f) Receptor, Rat	1
5HT2A_BOVIN	Q75Z89	CHEMBL3446	Serotonin 2a (5-HT2a) Receptor, Bovin	1
5HT2A_MOUSE	P35363	CHEMBL5377	Serotonin 2a (5-HT2a) Receptor, Mouse	1
5HT2A_RAT	P14842	CHEMBL322	Serotonin 2a (5-HT2a) Receptor, Rat	1
5HT2B_MOUSE	Q02152	CHEMBL2583	Serotonin 2b (5-HT2b) Receptor, Mouse	1
5HT2B_RAT	P30994	CHEMBL323	Serotonin 2b (5-HT2b) Receptor, Rat	1
5HT2C_MOUSE	P34968	CHEMBL3006	Serotonin 2c (5-HT2c) Receptor, Mouse	1
5HT2C_RAT	P08909	CHEMBL324	Serotonin 2c (5-HT2c) Receptor, Rat	1
5HT6R_HUMAN	P50406	CHEMBL3371	Serotonin 6 (5-HT6) Receptor, Human	1
5HT7R_RAT	P32305	CHEMBL3223	Serotonin 7 (5-HT7) Receptor, Rat	1
ACM1_HUMAN	P11229	CHEMBL216	Muscarinic Acetylcholine Receptor M1, Human	1
ACM1_RAT	P08482	CHEMBL276	Muscarinic Acetylcholine Receptor M1, Rat	1
ACM2_HUMAN	P08172	CHEMBL211	Muscarinic Acetylcholine Receptor M2, Human	1
ACM2_RAT	P10980	CHEMBL309	Muscarinic Acetylcholine Receptor M2, Rat	1
ACM3_HUMAN	P20309	CHEMBL245	Muscarinic Acetylcholine Receptor M3, Human	1
ACM4_HUMAN	P08173	CHEMBL1821	Muscarinic Acetylcholine Receptor M4, Human	1
ACM5_HUMAN	P08912	CHEMBL2035	Muscarinic Acetylcholine Receptor M5, Human	1
ADA1A_BOVIN	P18130	CHEMBL4892	Alpha-1a Adrenergic Receptor, Bovin	1
ADA1A_RAT	P43140	CHEMBL319	Alpha-1a Adrenergic Receptor, Rat	1
ADA1B_RAT	P15823	CHEMBL315	Alpha-1b Adrenergic Receptor, Rat	1
ADA1D_RAT	P23944	CHEMBL326	Alpha-1d Adrenergic Receptor, Rat	1
ADA2A_RAT	P22909	CHEMBL327	Alpha-2a Adrenergic Receptor, Rat	1
ADA2B_RAT	P19328	CHEMBL266	Alpha-2b Adrenergic Receptor, Rat	1
ADA2C_RAT	P22086	CHEMBL314	Alpha-2c Adrenergic Receptor, Rat	1
AP2S1_RAT	P62744	CHEMBL1697667	AP-2 Complex Subunit Sigma, Rat	1
DRD1_RAT	P18901	CHEMBL265	Dopamine D1 Receptor, Rat	1
DRD2_CHLAE	P52702	CHEMBL5456	Dopamine D2 Receptor, Chlae	1
DRD4_RAT	P30729	CHEMBL3361	Dopamine D4 Receptor, Rat	1
DRD5_HUMAN	P21918	CHEMBL1850	Dopamine D5 Receptor, Human	1
DRD5_RAT	P25115	CHEMBL2281	Dopamine D5 Receptor, Rat	1
EBP_HUMAN	Q15125	CHEMBL4931	3-beta-hydroxysteroid-delta(8),delta(7)-isomerase, Human	1
ERG2_YEAST	P32352	CHEMBL3224	C-8 Sterol Isomerase, Yeast	1
HRH1_RAT	P31390	CHEMBL4701	Histamine H1 Receptor, Rat	1
MDR1_HUMAN	P08183	CHEMBL4302	P-glycoprotein 1, Human	1
OPRD_RAT	P33533	CHEMBL269	Delta Opioid Receptor, Rat	1
OPRK_RAT	P34975	CHEMBL3614	Kappa Opioid Receptor, Rat	1
OPRM_RAT	P33535	CHEMBL270	Mu Opioid Receptor, Rat	1
Q4U254_9ENTO	Q4U254	CHEMBL2857	Human Rhinovirus A Protease, 9ento	1
Q63380_RAT	Q63380	CHEMBL6184	Transporter, Rat	1
Q72874_9HIV1	Q72874	CHEMBL243	Human Immunodeficiency Virus Type 1 Protease, 9hiv1	1
SC6A4_HUMAN	P31645	CHEMBL228	Serotonin Transporter, Human	1
SCN1A_HUMAN	P35498	CHEMBL1845	Sodium Channel Protein Type I Alpha Subunit, Human	1
SCN2A_HUMAN	Q99250	CHEMBL4187	Sodium Channel Protein Type II Alpha Subunit, Human	1
SCN3A_HUMAN	Q9NY46	CHEMBL5163	Sodium Channel Protein Type III Alpha Subunit, Human	1
SCN8A_HUMAN	Q9UQD0	CHEMBL5202	Sodium Channel Protein Type VIII Alpha Subunit, Human	1
SGMR1_CAVPO	Q60492	CHEMBL4153	Sigma-1 Receptor, Guinea Pig	1
SGMR1_HUMAN	Q99720	CHEMBL287	Sigma Opioid Receptor, Human	1
SGMR1_RAT	Q9R0C9	CHEMBL3602	Sigma Opioid Receptor, Rat	1
Z100491	Z100491	CHEMBL613288	Sigma 2 Receptor	1
Z104303	Z104303	CHEMBL1907609	Muscarinic Acetylcholine Receptor	1
Z104304	Z104304	CHEMBL1907610	Adrenergic Receptor Alpha-1	1