 
| Annotation Type | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|
| Binding ≤ 10μM | 65 | 2 | 2 | 2 | 
| Binding ≤ 1μM | 61 | 2 | 2 | 2 | 
| Functional ≤ 10μM | 116 | 1 | 1 | 1 | 
| Reactome ID | Description | Species | 
|---|---|---|
| REACT_15525 | Nuclear Receptor transcription pathway | Homo sapiens | 
| Uniprot | Swissprot | Chembl | Description | Number Shared | 
|---|---|---|---|---|
| ANDR_HUMAN | P10275 | CHEMBL1871 | Androgen Receptor, Human | 6 | 
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|---|---|---|
| VDR_BOVIN | Q28037 | CHEMBL3452 | Vitamin D Receptor, Bovin | 15 | 1 | 1 | 1 | 
| VDR_CHICK | O42392 | CHEMBL2353 | Vitamin D Receptor, Chick | 14 | 1 | 1 | 1 | 
| VDR_MOUSE | P48281 | CHEMBL5601 | Vitamin D Receptor, Mouse | 8 | 0 | 0 | 0 | 
| VDR_RAT | P13053 | CHEMBL3150 | Vitamin D Receptor, Rat | 49 | 1 | 1 | 1 | 
| Code | Description | Substances | Purchasable | Natural | In Man | 
|---|---|---|---|---|---|
| VDR-1-E | Vitamin D Receptor (cluster #1 Of 2), Eukaryotic | 125 | 2 | 2 | 2 | 
| VDR-2-E | Vitamin D Receptor (cluster #2 Of 2), Eukaryotic | 16 | 0 | 0 | 0 | 
| Uniprot | Swissprot | Chembl | Description | Number Shared | 
|---|---|---|---|---|
| Z80156 | Z80156 | CHEMBL383 | HL-60 (Promyeloblast Leukemia Cells) | 97 | 
| ANDR_MOUSE | P19091 | CHEMBL3056 | Androgen Receptor, Mouse | 10 | 
| VDR_BOVIN | Q28037 | CHEMBL3452 | Vitamin D Receptor, Bovin | 7 | 
| ANDR_HUMAN | P10275 | CHEMBL1871 | Androgen Receptor, Human | 6 | 
| HDAC6_HUMAN | Q9UBN7 | CHEMBL1865 | Histone Deacetylase 6, Human | 3 | 
| VDR_CHICK | O42392 | CHEMBL2353 | Vitamin D Receptor, Chick | 1 | 
| VDR_RAT | P13053 | CHEMBL3150 | Vitamin D Receptor, Rat | 1 | 
| Z100081 | Z100081 | CHEMBL613107 | PBMC (Peripheral Blood Mononuclear Cells) | 1 | 
| Z50587 | Z50587 | CHEMBL372 | Homo Sapiens | 1 | 
| Z80224 | Z80224 | CHEMBL387 | MCF7 (Breast Carcinoma Cells) | 1 | 
| Z80437 | Z80437 | CHEMBL614885 | RWLeu4 | 1 | 
| Z80566 | Z80566 | CHEMBL612794 | U-937 (Histiocytic Lymphoma Cells) | 1 | 
| Z81117 | Z81117 | CHEMBL613995 | Keratinocytes (Keratinocytes) | 1 | 
| Z81298 | Z81298 | CHEMBL614846 | PE Cell Line | 1 | 
| Z81338 | Z81338 | CHEMBL614309 | T-cells | 1 |