| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 36 | 3 | 2 | 3 |
| Functional ≤ 10μM | 6 | 0 | 0 | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| PDK1_HUMAN | Q15118 | CHEMBL4766 | Pyruvate Dehydrogenase Kinase Isoform 1, Human | 134 | 4 | 3 | 4 |
| PDK1_RAT | Q63065 | CHEMBL2416 | Pyruvate Dehydrogenase Kinase Isoform 1, Rat | 48 | 2 | 0 | 1 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| PDK1-2-E | Pyruvate Dehydrogenase Kinase Isoform 1 (cluster #2 Of 3), Eukaryotic | 5 | 1 | 1 | 0 |
| PDK1-3-E | Pyruvate Dehydrogenase Kinase Isoform 1 (cluster #3 Of 3), Eukaryotic | 141 | 2 | 0 | 1 |
![4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline](http://zinc12.docking.org/img/rings/38782.gif)
![4,5-dihydro-1H-pyrazolo[4,3-h]quinazolin-8-yl(phenyl)amine](http://zinc12.docking.org/img/rings/38783.gif)
![Phenyl-[1-(4-piperidylmethyl)-4,5-dihydropyrazolo[4,3-h]quinazolin-8-yl]amine](http://zinc12.docking.org/img/rings/38781.gif)