UCSF

Peroxisome Proliferator-activated Receptor Delta, Human (656 Compounds)

Swissprot:
PPARD_HUMAN
Stitch:
PPARD_HUMAN
UniProt:
Q03181
ChEMBL:
CHEMBL3979
Reactome:
REACT_11082
REACT_15525
REACT_12528
PDB:
1GWX (DOCK)
1Y0S (DOCK)
2AWH (DOCK)
2B50 (DOCK)
2BAW (DOCK)
2ENV (DOCK)
2GWX (DOCK)
2J14 (DOCK)
2Q5G (DOCK)
2XYJ (DOCK)
2XYW (DOCK)
2XYX (DOCK)
2ZNP (DOCK)
2ZNQ (DOCK)
3D5F (DOCK)
3DY6 (DOCK)
3ET2 (DOCK)
3GWX (DOCK)
3GZ9 (DOCK)
3OZ0 (DOCK)
3PEQ (DOCK)
3SP9 (DOCK)
PPARD

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 656 13 6 12
Binding ≤ 1μM 482 6 1 5
Functional ≤ 10μM 753 7 3 8
Uniprot Swissprot Chembl Description Number Shared
NR1H2_HUMAN P55055 CHEMBL4093 LXR-beta, Human 21
PPARA_HUMAN Q07869 CHEMBL239 Peroxisome Proliferator-activated Receptor Alpha, Human 902
PPARG_HUMAN P37231 CHEMBL235 Peroxisome Proliferator-activated Receptor Gamma, Human 700
RARG_HUMAN P13631 CHEMBL2003 Retinoic Acid Receptor Gamma, Human 2
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
PPARD_MOUSE P35396 CHEMBL2458 Peroxisome Proliferator-activated Receptor Delta, Mouse 7 3 3 1

Clustered By Gene (0)

Clustered By Organism (1)

Code Description Substances Purchasable Natural In Man
PPARD-1-E Peroxisome Proliferator-activated Receptor Delta (cluster #1 Of 2), Eukaryotic 96 2 3 2
PPARD-2-E Peroxisome Proliferator-activated Receptor Delta (cluster #2 Of 2), Eukaryotic 565 11 4 10
Uniprot Swissprot Chembl Description Number Shared
PPARA_HUMAN Q07869 CHEMBL239 Peroxisome Proliferator-activated Receptor Alpha, Human 902
PPARG_HUMAN P37231 CHEMBL235 Peroxisome Proliferator-activated Receptor Gamma, Human 695
PPARG_MOUSE P37238 CHEMBL2459 Peroxisome Proliferator-activated Receptor Gamma, Mouse 122
PPARG_RAT O88275 CHEMBL4797 Peroxisome Proliferator-activated Receptor Gamma, Rat 56
PPARD_MOUSE P35396 CHEMBL2458 Peroxisome Proliferator-activated Receptor Delta, Mouse 29
PPARA_MOUSE P23204 CHEMBL2128 Peroxisome Proliferator-activated Receptor Alpha, Mouse 24
NR1H2_HUMAN P55055 CHEMBL4093 LXR-beta, Human 21
NR1H3_HUMAN Q13133 CHEMBL2808 LXR-alpha, Human 21
Z80169 Z80169 CHEMBL614039 Huh-7 (Hepatocellular Carcinoma) 10
PPARA_CANFA Q95N78 CHEMBL2847 Peroxisome Proliferator-activated Receptor Alpha, Canine 8
PPARA_RAT P37230 CHEMBL2129 Peroxisome Proliferator-activated Receptor Alpha, Rat 8
Z80548 Z80548 CHEMBL614245 THP-1 (Acute Monocytic Leukemia Cells) 4
AOFB_HUMAN P27338 CHEMBL2039 Monoamine Oxidase B, Human 2
RARG_HUMAN P13631 CHEMBL2003 Retinoic Acid Receptor Gamma, Human 2
RXRA_RAT Q05343 CHEMBL4431 Retinoid X Receptor Alpha, Rat 2
Z80178 Z80178 CHEMBL614040 J774.A1 (Macrophage Cells) 1
Z81020 Z81020 CHEMBL395 HepG2 (Hepatoblastoma Cells) 1
Z81135 Z81135 CHEMBL614793 L6 (Skeletal Muscle Myoblast Cells) 1
Z81244 Z81244 CHEMBL614123 J774 (Macrophage Cells) 1