| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 1,249 | 78 | 38 | 23 |
| Functional ≤ 10μM | 43 | 5 | 2 | 1 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| GBRA1_BOVIN | P08219 | CHEMBL3627 | GABA Receptor Alpha-1 Subunit, Bovin | 302 | 43 | 17 | 5 |
| GBRA1_HUMAN | P14867 | CHEMBL1962 | GABA Receptor Alpha-1 Subunit, Human | 959 | 77 | 35 | 22 |
| GBRA1_MOUSE | P62812 | CHEMBL3139 | GABA Receptor Alpha-1 Subunit, Mouse | 45 | 6 | 5 | 2 |
| GBRA1_RAT | P62813 | CHEMBL343 | GABA Receptor Alpha-1 Subunit, Rat | 207 | 16 | 9 | 6 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| GBRA1-2-E | GABA Receptor Alpha-1 Subunit (cluster #2 Of 8), Eukaryotic | 28 | 2 | 2 | 0 |
| GBRA1-3-E | GABA Receptor Alpha-1 Subunit (cluster #3 Of 8), Eukaryotic | 33 | 2 | 1 | 1 |
| GBRA1-4-E | GABA Receptor Alpha-1 Subunit (cluster #4 Of 8), Eukaryotic | 14 | 0 | 0 | 0 |
| GBRA1-5-E | GABA Receptor Alpha-1 Subunit (cluster #5 Of 8), Eukaryotic | 12 | 4 | 1 | 1 |
| GBRA1-6-E | GABA Receptor Alpha-1 Subunit (cluster #6 Of 8), Eukaryotic | 134 | 30 | 10 | 0 |
| GBRA1-7-E | GABA Receptor Alpha-1 Subunit (cluster #7 Of 8), Eukaryotic | 4 | 4 | 1 | 1 |
| GBRA1-8-E | GABA Receptor Alpha-1 Subunit (cluster #8 Of 8), Eukaryotic | 3 | 0 | 0 | 0 |
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