UCSF

G-protein Coupled Estrogen Receptor 1, Human (3 Compounds)

Swissprot:
GPER_HUMAN
Stitch:
GPER_HUMAN
UniProt:
Q99527
ChEMBL:
CHEMBL5872
Reactome:
REACT_19231
REACT_14819
PDB:
GPER

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 3 3 1 1
Binding ≤ 1μM 3 3 1 1
Functional ≤ 10μM 3 3 1 1

Reactome Network (2)

Reactome ID Description Species
REACT_19231 G alpha (i) signalling events Homo sapiens
REACT_14819 Peptide ligand-binding receptors Homo sapiens

Clustered By Gene (0)

Uniprot Swissprot Chembl Description Number Shared
ESR1_MOUSE P19785 CHEMBL3065 Estrogen Receptor Alpha, Mouse 2
ESR2_MOUSE O08537 CHEMBL2995 Estrogen Receptor Beta, Mouse 2
Z80224 Z80224 CHEMBL387 MCF7 (Breast Carcinoma Cells) 2
Z80475 Z80475 CHEMBL613834 SK-BR-3 (Breast Adenocarcinoma) 2
ANDR_HUMAN P10275 CHEMBL1871 Androgen Receptor, Human 1
ERR1_HUMAN P11474 CHEMBL3429 Estrogen-related Receptor Alpha, Human 1
ERR2_HUMAN O95718 CHEMBL3751 Estrogen-related Receptor Beta, Human 1
ESR1_BOVIN P49884 CHEMBL2930 Estrogen Receptor Alpha, Bovin 1
ESR1_HUMAN P03372 CHEMBL206 Estrogen Receptor Alpha, Human 1
ESR1_RAT P06211 CHEMBL2724 Estrogen Receptor Alpha, Rat 1
ESR2_HUMAN Q92731 CHEMBL242 Estrogen Receptor Beta, Human 1
ESR2_RAT Q62986 CHEMBL3021 Estrogen Receptor Beta, Rat 1
SHBG_HUMAN P04278 CHEMBL3305 Testis-specific Androgen-binding Protein, Human 1
Z80226 Z80226 CHEMBL614323 MCF7-2A 1
Z81068 Z81068 CHEMBL614649 Ishikawa (Uterine Carcinoma Cells) 1
Z81247 Z81247 CHEMBL399 HeLa (Cervical Adenocarcinoma Cells) 1