UCSF

Calcium Sensing Receptor, Human (194 Compounds)

Swissprot:
CASR_HUMAN
Stitch:
CASR_HUMAN
UniProt:
P41180
ChEMBL:
CHEMBL1878
Reactome:
REACT_18319
REACT_19231
REACT_18283
PDB:
CASR

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 194 8 2 2
Binding ≤ 1μM 159 4 2 2
Functional ≤ 10μM 228 2 0 0

Reactome Network (3)

Reactome ID Description Species
REACT_18319 Class C/3 (Metabotropic glutamate/pheromone receptors) Homo sapiens
REACT_19231 G alpha (i) signalling events Homo sapiens
REACT_18283 G alpha (q) signalling events Homo sapiens
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
CASR_BOVIN P35384 CHEMBL1075316 Extracellular Calcium-sensing Receptor, Bovin 1 1 0 0
CASR_RAT P48442 CHEMBL2516 Calcium Sensing Receptor, Rat 1 0 1 1

Clustered By Gene (0)

Uniprot Swissprot Chembl Description Number Shared
KCNH2_HUMAN Q12809 CHEMBL240 HERG, Human 10
SC6A2_HUMAN P23975 CHEMBL222 Norepinephrine Transporter, Human 10
SC6A3_HUMAN Q01959 CHEMBL238 Dopamine Transporter, Human 10
SC6A4_HUMAN P31645 CHEMBL228 Serotonin Transporter, Human 10
ADRB2_HUMAN P07550 CHEMBL210 Beta-2 Adrenergic Receptor, Human 9
CASR_RAT P48442 CHEMBL2516 Calcium Sensing Receptor, Rat 5
ADRB3_HUMAN P13945 CHEMBL246 Beta-3 Adrenergic Receptor, Human 4
ADRB1_HUMAN P08588 CHEMBL213 Beta-1 Adrenergic Receptor, Human 1
CASR_BOVIN P35384 CHEMBL1075316 Extracellular Calcium-sensing Receptor, Bovin 1
Z80936 Z80936 CHEMBL614818 HEK293 (Embryonic Kidney Fibroblasts) 1

Most Common Rings