| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 604 | 15 | 0 | 0 |
| Binding ≤ 1μM | 502 | 10 | 0 | 0 |
| Functional ≤ 10μM | 35 | 0 | 0 | 0 |
| Reactome ID | Description | Species |
|---|---|---|
| REACT_20506 | Na+/Cl- dependent neurotransmitter transporters | Homo sapiens |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| SC6A5_HUMAN | Q9Y345 | CHEMBL3060 | Glycine Transporter 2, Human | 63 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| SC6A9_MOUSE | P28571 | CHEMBL1075303 | Sodium- And Chloride-dependent Glycine Transporter 1, Mouse | 6 | 0 | 0 | 0 |
| SC6A9_RAT | P28572 | CHEMBL4556 | Glycine Transporter 1, Rat | 27 | 2 | 0 | 0 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| SC6A1_HUMAN | P30531 | CHEMBL1903 | GABA Transporter 1, Human | 84 | 7 | 4 | 2 |
| SC6A2_HUMAN | P23975 | CHEMBL222 | Norepinephrine Transporter, Human | 2,711 | 158 | 43 | 54 |
| SC6A3_HUMAN | Q01959 | CHEMBL238 | Dopamine Transporter, Human | 2,208 | 143 | 41 | 50 |
| SC6A4_HUMAN | P31645 | CHEMBL228 | Serotonin Transporter, Human | 4,112 | 205 | 45 | 56 |
| SC6A5_HUMAN | Q9Y345 | CHEMBL3060 | Glycine Transporter 2, Human | 116 | 8 | 0 | 0 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| SC6A5_HUMAN | Q9Y345 | CHEMBL3060 | Glycine Transporter 2, Human | 63 |
| OPRM_HUMAN | P35372 | CHEMBL233 | Mu Opioid Receptor, Human | 55 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 50 |
| OPRX_HUMAN | P41146 | CHEMBL2014 | Nociceptin Receptor, Human | 16 |
| 5HT1B_HUMAN | P28222 | CHEMBL1898 | Serotonin 1b (5-HT1b) Receptor, Human | 8 |
| SC6A9_MOUSE | P28571 | CHEMBL1075303 | Sodium- And Chloride-dependent Glycine Transporter 1, Mouse | 6 |
| SC6A9_RAT | P28572 | CHEMBL4556 | Glycine Transporter 1, Rat | 6 |
| GALR1_RAT | Q62805 | CHEMBL5504 | Galanin Receptor Type 1, Rat | 1 |
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