| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 4,969 | 188 | 36 | 30 |
| Functional ≤ 10μM | 632 | 49 | 10 | 6 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| AA2AR_CAVPO | P46616 | CHEMBL2605 | Adenosine A2a Receptor, Guinea Pig | 18 | 9 | 3 | 3 |
| AA2AR_HUMAN | P29274 | CHEMBL251 | Adenosine A2a Receptor, Human | 2,605 | 153 | 29 | 23 |
| AA2AR_MOUSE | Q60613 | CHEMBL2115 | Adenosine A2a Receptor, Mouse | 5 | 2 | 0 | 1 |
| AA2AR_RAT | P30543 | CHEMBL302 | Adenosine A2a Receptor, Rat | 2,846 | 130 | 40 | 27 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| AA2AR-2-E | Adenosine A2a Receptor (cluster #2 Of 4), Eukaryotic | 59 | 29 | 5 | 4 |
| AA2AR-3-E | Adenosine A2a Receptor (cluster #3 Of 4), Eukaryotic | 121 | 25 | 12 | 4 |
| AA2AR-4-E | Adenosine A2a Receptor (cluster #4 Of 4), Eukaryotic | 33 | 7 | 3 | 3 |
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