UCSF

Bradykinin B1 Receptor, Human (443 Compounds)

Swissprot:
BKRB1_HUMAN
Stitch:
BKRB1_HUMAN
UniProt:
P46663
ChEMBL:
CHEMBL4308
Reactome:
REACT_19231
REACT_18283
REACT_14819
PDB:
BDKRB1

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 443 3 0 0
Binding ≤ 1μM 416 3 0 0
Functional ≤ 10μM 321 1 0 0

Reactome Network (3)

Reactome ID Description Species
REACT_19231 G alpha (i) signalling events Homo sapiens
REACT_18283 G alpha (q) signalling events Homo sapiens
REACT_14819 Peptide ligand-binding receptors Homo sapiens
Uniprot Swissprot Chembl Description Number Shared
BKRB2_HUMAN P30411 CHEMBL3157 Bradykinin B2 Receptor, Human 17
CNR1_HUMAN P21554 CHEMBL218 Cannabinoid CB1 Receptor, Human 1

G alpha (q) signalling events

Uniprot Swissprot Chembl Description Number Shared
BKRB2_HUMAN P30411 CHEMBL3157 Bradykinin B2 Receptor, Human 17
NK1R_HUMAN P25103 CHEMBL249 Neurokinin 1 Receptor, Human 11

Peptide ligand-binding receptors

Uniprot Swissprot Chembl Description Number Shared
BKRB2_HUMAN P30411 CHEMBL3157 Bradykinin B2 Receptor, Human 17
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
BKRB1_CANFA Q9BDQ5 CHEMBL4724 Bradykinin B1 Receptor, Canine 2 0 0 0
BKRB1_MACMU Q8HZP2 CHEMBL1250405 B1 Bradykinin Receptor, Macmu 1 0 0 0
BKRB1_MOUSE Q61125 CHEMBL1250407 B1 Bradykinin Receptor, Mouse 1 0 0 0
BKRB1_RABIT P48748 CHEMBL4087 Bradykinin B1 Receptor, Rabit 18 0 0 0
BKRB1_RAT P97583 CHEMBL4613 Bradykinin B1 Receptor, Rat 15 0 0 0
UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
BKRB2_HUMAN P30411 CHEMBL3157 Bradykinin B2 Receptor, Human 400 0 0 0

Clustered By Gene (0)

Uniprot Swissprot Chembl Description Number Shared
BKRB1_RABIT P48748 CHEMBL4087 Bradykinin B1 Receptor, Rabit 20
BKRB1_RAT P97583 CHEMBL4613 Bradykinin B1 Receptor, Rat 19
BKRB2_HUMAN P30411 CHEMBL3157 Bradykinin B2 Receptor, Human 17
NK1R_HUMAN P25103 CHEMBL249 Neurokinin 1 Receptor, Human 11
Z50592 Z50592 CHEMBL374 Oryctolagus Cuniculus 5
BKRB1_CANFA Q9BDQ5 CHEMBL4724 Bradykinin B1 Receptor, Canine 3
KCNH2_HUMAN Q12809 CHEMBL240 HERG, Human 3
BKRB1_MACMU Q8HZP2 CHEMBL1250405 B1 Bradykinin Receptor, Macmu 1
BKRB1_MOUSE Q61125 CHEMBL1250407 B1 Bradykinin Receptor, Mouse 1
CNR1_HUMAN P21554 CHEMBL218 Cannabinoid CB1 Receptor, Human 1

Most Common Rings