ZINC 12

User Information

Not Authenticated — sign in

Active cart: Temporary Cart (0 items)

Navigation

About
- ZINC
- BCIRC
- Irwin Lab
- Shoichet Lab
- UCSF
- Acknowledgements
- Facts
- Usage
Search
- By:
- Text
- Structure
- Properties
- Catalogs
- ZINC
- Targets
- Rings
- Combination
Subsets
- By:
- Catalog
- Property
- Target
- Ring
- Cart
Help
- Introduction
- FAQ
- Scripting/API
- Quick Search
- Problems
- Filtering
- History
Social
- ZINC Fans
- Decoy Club
- DOCK Fans
- Facebook
- Twitter
- Blog
- Linkedin
Quick Search ZINC ID or SMILES

Names
Compounds (1,390)
Reactome (0)
Related By:
Pathway (0)
Organism (3)
Gene (0)
Org. Clust. (0)
ChEMBL (42)
Rings (10)

Cholecystokinin A Receptor, Rat (1,390 Compounds)

Swissprot:: CCKAR_RAT
Stitch:: CCKAR_RAT
UniProt:: P30551
ChEMBL:: CHEMBL2871
PDB:: Cckar

Compound Summary

Annotation Type	Substances	Purchasable	Natural	In Man
Binding ≤ 10μM	1,390	29	10	10
Binding ≤ 1μM	859	27	8	8
Functional ≤ 10μM	9	0	0	0

UniProt	Swissprot	ChEMBL	Description	Substances	Purchasable	Natural	In Man
CCKAR_CAVPO	Q63931	CHEMBL3501	Cholecystokinin A Receptor, Guinea Pig	41	0	0	0
CCKAR_HUMAN	P32238	CHEMBL1901	Cholecystokinin A Receptor, Human	524	9	8	5
CCKAR_MOUSE	O08786	CHEMBL2798	Cholecystokinin A Receptor, Mouse	46	1	1	1

Clustered By Gene (0)

Uniprot	Swissprot	Chembl	Description	Number Shared
GASR_HUMAN	P32239	CHEMBL298	Cholecystokinin B Receptor, Human	435
GASR_MOUSE	P56481	CHEMBL2854	Cholecystokinin B Receptor, Mouse	345
GASR_RAT	P30553	CHEMBL3508	Cholecystokinin B Receptor, Rat	253
CCKAR_HUMAN	P32238	CHEMBL1901	Cholecystokinin A Receptor, Human	119
OPRD_RAT	P33533	CHEMBL269	Delta Opioid Receptor, Rat	25
OPRK_RAT	P34975	CHEMBL3614	Kappa Opioid Receptor, Rat	25
OPRM_RAT	P33535	CHEMBL270	Mu Opioid Receptor, Rat	25
SGMR1_RAT	Q9R0C9	CHEMBL3602	Sigma Opioid Receptor, Rat	25
CCKAR_CAVPO	Q63931	CHEMBL3501	Cholecystokinin A Receptor, Guinea Pig	17
CCKAR_MOUSE	O08786	CHEMBL2798	Cholecystokinin A Receptor, Mouse	3
5HT2A_BOVIN	Q75Z89	CHEMBL3446	Serotonin 2a (5-HT2a) Receptor, Bovin	2
5HT2A_HUMAN	P28223	CHEMBL224	Serotonin 2a (5-HT2a) Receptor, Human	2
5HT2C_HUMAN	P28335	CHEMBL225	Serotonin 2c (5-HT2c) Receptor, Human	2
5HT2C_RAT	P08909	CHEMBL324	Serotonin 2c (5-HT2c) Receptor, Rat	2
HRH2_HUMAN	P25021	CHEMBL1941	Histamine H2 Receptor, Human	2
MCHR1_HUMAN	Q99705	CHEMBL344	Melanin-concentrating Hormone Receptor 1, Human	2
OPRD_HUMAN	P41143	CHEMBL236	Delta Opioid Receptor, Human	2
OPRK_HUMAN	P41145	CHEMBL237	Kappa Opioid Receptor, Human	2
OPRM_HUMAN	P35372	CHEMBL233	Mu Opioid Receptor, Human	2
SC6A3_BOVIN	P27922	CHEMBL2986	Dopamine Transporter, Bovin	2
SC6A3_HUMAN	Q01959	CHEMBL238	Dopamine Transporter, Human	2
GBRA1_HUMAN	P14867	CHEMBL1962	GABA Receptor Alpha-1 Subunit, Human	1
GBRA2_HUMAN	P47869	CHEMBL4956	GABA Receptor Alpha-2 Subunit, Human	1
GBRA3_HUMAN	P34903	CHEMBL3026	GABA Receptor Alpha-3 Subunit, Human	1
GBRA4_HUMAN	P48169	CHEMBL2472	GABA Receptor Alpha-4 Subunit, Human	1
GBRA5_HUMAN	P31644	CHEMBL5112	GABA Receptor Alpha-5 Subunit, Human	1
GBRA6_HUMAN	Q16445	CHEMBL2579	GABA Receptor Alpha-6 Subunit, Human	1
GBRB1_HUMAN	P18505	CHEMBL4558	GABA Receptor Beta-1 Subunit, Human	1
GBRB2_HUMAN	P47870	CHEMBL1920	GABA Receptor Beta-2 Subunit, Human	1
GBRB3_HUMAN	P28472	CHEMBL1847	GABA Receptor Beta-3 Subunit, Human	1
GBRD_HUMAN	O14764	CHEMBL3591	GABA Receptor Delta Subunit, Human	1
GBRE_HUMAN	P78334	CHEMBL4635	GABA Receptor Epsilon Subunit, Human	1
GBRG1_HUMAN	Q8N1C3	CHEMBL4044	GABA Receptor Gamma-1 Subunit, Human	1
GBRG2_HUMAN	P18507	CHEMBL1788	GABA Receptor Gamma-2 Subunit, Human	1
GBRG3_HUMAN	Q99928	CHEMBL2739	GABA Receptor Gamma-3 Subunit, Human	1
GBRP_HUMAN	O00591	CHEMBL3506	GABA Receptor Pi Subunit, Human	1
GBRT_HUMAN	Q9UN88	CHEMBL2843	GABA Receptor Theta Subunit, Human	1
KCNH2_HUMAN	Q12809	CHEMBL240	HERG, Human	1
NMBR_HUMAN	P28336	CHEMBL3636	Neuromedin B Receptor, Human	1
SCN9A_HUMAN	Q15858	CHEMBL4296	Sodium Channel Protein Type IX Alpha Subunit, Human	1
Z104301	Z104301	CHEMBL1907607	GABA-A Receptor; Anion Channel	1
Z50597	Z50597	CHEMBL376	Rattus Norvegicus	1