UCSF

Glucocorticoid Receptor, Rat (136 Compounds)

Swissprot:
GCR_RAT
Stitch:
GCR_RAT
UniProt:
P06536
ChEMBL:
CHEMBL3368
PDB:
1GDC (DOCK)
1GLU (DOCK)
1LAT (DOCK)
1R4O (DOCK)
1R4R (DOCK)
1RGD (DOCK)
2GDA (DOCK)
3FYL (DOCK)
3G6P (DOCK)
3G6Q (DOCK)
3G6R (DOCK)
3G6T (DOCK)
3G6U (DOCK)
3G8U (DOCK)
3G8X (DOCK)
3G97 (DOCK)
3G99 (DOCK)
3G9I (DOCK)
3G9J (DOCK)
3G9M (DOCK)
3G9O (DOCK)
3G9P (DOCK)
Nr3c1

Compound Summary

Annotation Type Substances Purchasable Natural In Man
Binding ≤ 10μM 136 8 7 6
Binding ≤ 1μM 134 8 7 6
Functional ≤ 10μM 48 3 1 2

Reactome Network (0)

UniProt Swissprot ChEMBL Description Substances Purchasable Natural In Man
GCR_HUMAN P04150 CHEMBL2034 Glucocorticoid Receptor, Human 1,714 39 22 10
GCR_MOUSE P06537 CHEMBL3144 Glucocorticoid Receptor, Mouse 15 1 1 1

Clustered By Gene (0)

Clustered By Organism (1)

Code Description Substances Purchasable Natural In Man
GCR-1-E Glucocorticoid Receptor (cluster #1 Of 2), Eukaryotic 1,603 10 7 1
GCR-2-E Glucocorticoid Receptor (cluster #2 Of 2), Eukaryotic 266 38 25 15
Uniprot Swissprot Chembl Description Number Shared
GCR_HUMAN P04150 CHEMBL2034 Glucocorticoid Receptor, Human 37
Z80110 Z80110 CHEMBL613507 CV-1 (Kidney Cells) 12
Z100081 Z100081 CHEMBL613107 PBMC (Peripheral Blood Mononuclear Cells) 11
PRGR_HUMAN P06401 CHEMBL208 Progesterone Receptor, Human 8
Z50594 Z50594 CHEMBL375 Mus Musculus 8
Z80682 Z80682 CHEMBL392 A549 (Lung Carcinoma Cells) 8
MCR_HUMAN P08235 CHEMBL1994 Mineralocorticoid Receptor, Human 7
ANDR_HUMAN P10275 CHEMBL1871 Androgen Receptor, Human 5
GCR_MOUSE P06537 CHEMBL3144 Glucocorticoid Receptor, Mouse 4
Z81011 Z81011 CHEMBL614840 Human Cell Lines 3
ESR1_HUMAN P03372 CHEMBL206 Estrogen Receptor Alpha, Human 1
ESR2_HUMAN Q92731 CHEMBL242 Estrogen Receptor Beta, Human 1
PRGR_CHICK P07812 CHEMBL3304 Progesterone Receptor, Chick 1
PRGR_RAT Q63449 CHEMBL2596 Progesterone Receptor, Rat 1
VP16_HHV11 P06492 CHEMBL4218 Alpha Trans-inducing Protein (VP16), Hhv11 1
Z50425 Z50425 CHEMBL364 Plasmodium Falciparum 1
Z80156 Z80156 CHEMBL383 HL-60 (Promyeloblast Leukemia Cells) 1
Z80491 Z80491 CHEMBL614163 SK-N-MC (Neuroepithelioma Cells) 1
Z80951 Z80951 CHEMBL614822 NIH3T3 (Fibroblasts) 1
Z80954 Z80954 CHEMBL614071 HFF (Foreskin Fibroblasts) 1
Z81247 Z81247 CHEMBL399 HeLa (Cervical Adenocarcinoma Cells) 1