ZINC 12

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Quick Search ZINC ID or SMILES

Names
Compounds (541)
Reactome (0)
Related By:
Pathway (0)
Organism (2)
Gene (0)
Org. Clust. (0)
ChEMBL (81)
Rings (5)

Peripheral-type Benzodiazepine Receptor, Rat (541 Compounds)

Swissprot:: TSPO_RAT
Stitch:: TSPO_RAT
UniProt:: P16257
ChEMBL:: CHEMBL4552
PDB:: Tspo

Compound Summary

Annotation Type	Substances	Purchasable	Natural	In Man
Binding ≤ 10μM	541	32	6	6
Binding ≤ 1μM	471	28	5	5

UniProt	Swissprot	ChEMBL	Description	Substances	Purchasable	Natural	In Man
TSPO_BOVIN	P30535	CHEMBL2419	Peripheral-type Benzodiazepine Receptor, Bovin	18	0	0	0
TSPO_MOUSE	P50637	CHEMBL2149	Peripheral-type Benzodiazepine Receptor, Mouse	2	2	0	0

Clustered By Gene (0)

Uniprot	Swissprot	Chembl	Description	Number Shared
Z104301	Z104301	CHEMBL1907607	GABA-A Receptor; Anion Channel	60
CAC1C_RAT	P22002	CHEMBL3762	Voltage-gated L-type Calcium Channel Alpha-1C Subunit, Rat	14
CAC1D_RAT	P27732	CHEMBL4132	Voltage-gated L-type Calcium Channel Alpha-1D Subunit, Rat	13
CNR1_HUMAN	P21554	CHEMBL218	Cannabinoid CB1 Receptor, Human	10
CNR2_HUMAN	P34972	CHEMBL253	Cannabinoid CB2 Receptor, Human	9
TSPOA_HUMAN	P30536	CHEMBL5742	Translocator Protein, Human	9
GBRA2_RAT	P23576	CHEMBL341	GABA Receptor Alpha-2 Subunit, Rat	8
TSPOB_HUMAN	B1AH88	CHEMBL5139	Peripheral-type Benzodiazepine Receptor, Human	5
GBRA1_HUMAN	P14867	CHEMBL1962	GABA Receptor Alpha-1 Subunit, Human	3
GBRA2_HUMAN	P47869	CHEMBL4956	GABA Receptor Alpha-2 Subunit, Human	3
GBRA3_HUMAN	P34903	CHEMBL3026	GABA Receptor Alpha-3 Subunit, Human	3
GBRB3_HUMAN	P28472	CHEMBL1847	GABA Receptor Beta-3 Subunit, Human	3
GBRG2_HUMAN	P18507	CHEMBL1788	GABA Receptor Gamma-2 Subunit, Human	3
OPRK_HUMAN	P41145	CHEMBL237	Kappa Opioid Receptor, Human	3
5HT2A_HUMAN	P28223	CHEMBL224	Serotonin 2a (5-HT2a) Receptor, Human	2
GBRA1_BOVIN	P08219	CHEMBL3627	GABA Receptor Alpha-1 Subunit, Bovin	2
GBRA1_RAT	P62813	CHEMBL343	GABA Receptor Alpha-1 Subunit, Rat	2
GBRA2_BOVIN	P10063	CHEMBL2321	GABA Receptor Alpha-2 Subunit, Bovin	2
GBRA3_BOVIN	P10064	CHEMBL3628	GABA Receptor Alpha-3 Subunit, Bovin	2
GBRA3_RAT	P20236	CHEMBL328	GABA Receptor Alpha-3 Subunit, Rat	2
GBRA4_BOVIN	P20237	CHEMBL3140	GABA Receptor Alpha-4 Subunit, Bovin	2
GBRA4_RAT	P28471	CHEMBL292	GABA Receptor Alpha-4 Subunit, Rat	2
GBRA5_HUMAN	P31644	CHEMBL5112	GABA Receptor Alpha-5 Subunit, Human	2
GBRA5_RAT	P19969	CHEMBL300	GABA Receptor Alpha-5 Subunit, Rat	2
GBRA6_RAT	P30191	CHEMBL293	GABA Receptor Alpha-6 Subunit, Rat	2
GBRB1_BOVIN	P08220	CHEMBL2848	GABA Receptor Beta-1 Subunit, Bovin	2
GBRB2_HUMAN	P47870	CHEMBL1920	GABA Receptor Beta-2 Subunit, Human	2
GBRB2_RAT	P63138	CHEMBL295	GABA Receptor Beta-2 Subunit, Rat	2
GBRB3_RAT	P63079	CHEMBL316	GABA Receptor Beta-3 Subunit, Rat	2
GBRG2_BOVIN	P22300	CHEMBL5138	GABA Receptor Gamma-2 Subunit, Bovin	2
GBRG2_RAT	P18508	CHEMBL297	GABA Receptor Gamma-2 Subunit, Rat	2
GBRG3_RAT	P28473	CHEMBL336	GABA Receptor Gamma-3 Subunit, Rat	2
TSPO_MOUSE	P50637	CHEMBL2149	Peripheral-type Benzodiazepine Receptor, Mouse	2
5HT1B_HUMAN	P28222	CHEMBL1898	Serotonin 1b (5-HT1b) Receptor, Human	1
5HT2B_HUMAN	P41595	CHEMBL1833	Serotonin 2b (5-HT2b) Receptor, Human	1
A2AMW3_MOUSE	A2AMW3	CHEMBL3121	GABA Receptor Epsilon Subunit, Mouse	1
AA3R_HUMAN	P33765	CHEMBL256	Adenosine A3 Receptor, Human	1
CAC1C_HUMAN	Q13936	CHEMBL1940	Voltage-gated L-type Calcium Channel Alpha-1C Subunit, Human	1
CAC1C_RABIT	P15381	CHEMBL2830	Voltage-gated L-type Calcium Channel Alpha-1C Subunit, Rabit	1
CAC1D_HUMAN	Q01668	CHEMBL4138	Voltage-gated L-type Calcium Channel Alpha-1D Subunit, Human	1
CAC1S_RAT	Q02485	CHEMBL4108	Voltage-gated L-type Calcium Channel Alpha-1S Subunit, Rat	1
FABPL_RAT	P02692	CHEMBL5738	Fatty Acid-binding Protein, Liver, Rat	1
GBRA1_MOUSE	P62812	CHEMBL3139	GABA Receptor Alpha-1 Subunit, Mouse	1
GBRA2_MOUSE	P26048	CHEMBL2705	GABA Receptor Alpha-2 Subunit, Mouse	1
GBRA3_MOUSE	P26049	CHEMBL3387	GABA Receptor Alpha-3 Subunit, Mouse	1
GBRA4_HUMAN	P48169	CHEMBL2472	GABA Receptor Alpha-4 Subunit, Human	1
GBRA4_MOUSE	Q9D6F4	CHEMBL4182	GABA Receptor Alpha-4 Subunit, Mouse	1
GBRA5_MOUSE	Q8BHJ7	CHEMBL2304	GABA Receptor Alpha-5 Subunit, Mouse	1
GBRA6_HUMAN	Q16445	CHEMBL2579	GABA Receptor Alpha-6 Subunit, Human	1
GBRA6_MOUSE	P16305	CHEMBL4710	GABA Receptor Alpha-6 Subunit, Mouse	1
GBRB1_HUMAN	P18505	CHEMBL4558	GABA Receptor Beta-1 Subunit, Human	1
GBRB1_MOUSE	P50571	CHEMBL2839	GABA Receptor Beta-1 Subunit, Mouse	1
GBRB1_RAT	P15431	CHEMBL334	GABA Receptor Beta-1 Subunit, Rat	1
GBRB3_MOUSE	P63080	CHEMBL4231	GABA Receptor Beta-3 Subunit, Mouse	1
GBRD_HUMAN	O14764	CHEMBL3591	GABA Receptor Delta Subunit, Human	1
GBRD_MOUSE	P22933	CHEMBL3907	GABA Receptor Delta Subunit, Mouse	1
GBRD_RAT	P18506	CHEMBL337	GABA Receptor Delta Subunit, Rat	1
GBRE_HUMAN	P78334	CHEMBL4635	GABA Receptor Epsilon Subunit, Human	1
GBRE_RAT	Q9ES14	CHEMBL306	GABA Receptor Epsilon Subunit, Rat	1
GBRG1_HUMAN	Q8N1C3	CHEMBL4044	GABA Receptor Gamma-1 Subunit, Human	1
GBRG1_MOUSE	Q9R0Y8	CHEMBL2891	GABA Receptor Gamma-1 Subunit, Mouse	1
GBRG1_RAT	P23574	CHEMBL296	GABA Receptor Gamma-1 Subunit, Rat	1
GBRG2_MOUSE	P22723	CHEMBL2941	GABA Receptor Gamma-2 Subunit, Mouse	1
GBRG3_HUMAN	Q99928	CHEMBL2739	GABA Receptor Gamma-3 Subunit, Human	1
GBRG3_MOUSE	P27681	CHEMBL4236	GABA Receptor Gamma-3 Subunit, Mouse	1
GBRP_HUMAN	O00591	CHEMBL3506	GABA Receptor Pi Subunit, Human	1
GBRP_MOUSE	Q8QZW7	CHEMBL2746	GABA Receptor Pi Subunit, Mouse	1
GBRR1_RAT	P50572	CHEMBL3588	GABA Receptor Rho-1 Subunit, Rat	1
GBRT_HUMAN	Q9UN88	CHEMBL2843	GABA Receptor Theta Subunit, Human	1
GBRT_MOUSE	Q9JLF1	CHEMBL3249	GABA Receptor Theta Subunit, Mouse	1
KCNH2_HUMAN	Q12809	CHEMBL240	HERG, Human	1
MDR1_HUMAN	P08183	CHEMBL4302	P-glycoprotein 1, Human	1
MRP1_HUMAN	P33527	CHEMBL3004	Multidrug Resistance-associated Protein 1, Human	1
P97706_RAT	P97706	CHEMBL4957	Sodium Channel Protein Type VI Alpha Subunit, Rat	1
Q91ZM7_RAT	Q91ZM7	CHEMBL305	GABA Receptor Theta Subunit, Rat	1
S22A1_HUMAN	O15245	CHEMBL5685	Solute Carrier Family 22 Member 1, Human	1
SCN1A_HUMAN	P35498	CHEMBL1845	Sodium Channel Protein Type I Alpha Subunit, Human	1
SCN2A_HUMAN	Q99250	CHEMBL4187	Sodium Channel Protein Type II Alpha Subunit, Human	1
SCN3A_HUMAN	Q9NY46	CHEMBL5163	Sodium Channel Protein Type III Alpha Subunit, Human	1
SCN5A_RAT	P15389	CHEMBL3866	Sodium Channel Protein Type V Alpha Subunit, Rat	1
SCN8A_HUMAN	Q9UQD0	CHEMBL5202	Sodium Channel Protein Type VIII Alpha Subunit, Human	1