| Annotation Type | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|
| Binding ≤ 10μM | 827 | 43 | 30 | 14 |
| Binding ≤ 1μM | 577 | 34 | 17 | 12 |
| UniProt | Swissprot | ChEMBL | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|---|---|
| ACES_BOVIN | P23795 | CHEMBL4768 | Acetylcholinesterase, Bovin | 332 | 18 | 13 | 14 |
| ACES_HUMAN | P22303 | CHEMBL220 | Acetylcholinesterase, Human | 1,893 | 166 | 81 | 42 |
| ACES_MOUSE | P21836 | CHEMBL3198 | Acetylcholinesterase, Mouse | 174 | 27 | 11 | 14 |
| ACES_RAT | P37136 | CHEMBL3199 | Acetylcholinesterase, Rat | 712 | 37 | 13 | 17 |
| ACES_TORCA | P04058 | CHEMBL4780 | Acetylcholinesterase, Torca | 144 | 38 | 13 | 18 |
| Code | Description | Substances | Purchasable | Natural | In Man |
|---|---|---|---|---|---|
| ACES-1-E | Acetylcholinesterase (cluster #1 Of 12), Eukaryotic | 1,833 | 54 | 43 | 24 |
| ACES-10-E | Acetylcholinesterase (cluster #10 Of 12), Eukaryotic | 750 | 87 | 33 | 18 |
| ACES-11-E | Acetylcholinesterase (cluster #11 Of 12), Eukaryotic | 0 | 0 | 0 | 0 |
| ACES-12-E | Acetylcholinesterase (cluster #12 Of 12), Eukaryotic | 4 | 3 | 2 | 0 |
| ACES-2-E | Acetylcholinesterase (cluster #2 Of 12), Eukaryotic | 427 | 36 | 9 | 6 |
| ACES-3-E | Acetylcholinesterase (cluster #3 Of 12), Eukaryotic | 24 | 1 | 4 | 0 |
| ACES-4-E | Acetylcholinesterase (cluster #4 Of 12), Eukaryotic | 9 | 3 | 5 | 1 |
| ACES-5-E | Acetylcholinesterase (cluster #5 Of 12), Eukaryotic | 336 | 29 | 9 | 8 |
| ACES-6-E | Acetylcholinesterase (cluster #6 Of 12), Eukaryotic | 62 | 1 | 1 | 1 |
| ACES-7-E | Acetylcholinesterase (cluster #7 Of 12), Eukaryotic | 1 | 1 | 0 | 0 |
| ACES-8-E | Acetylcholinesterase (cluster #8 Of 12), Eukaryotic | 36 | 5 | 3 | 1 |
| ACES-9-E | Acetylcholinesterase (cluster #9 Of 12), Eukaryotic | 18 | 10 | 3 | 4 |
| Uniprot | Swissprot | Chembl | Description | Number Shared |
|---|---|---|---|---|
| CHLE_HORSE | P81908 | CHEMBL5763 | Cholinesterase, Horse | 250 |
| ACES_HUMAN | P22303 | CHEMBL220 | Acetylcholinesterase, Human | 187 |
| Q9N1N9_HORSE | Q9N1N9 | CHEMBL5077 | Butyrylcholinesterase, Horse | 129 |
| CHLE_HUMAN | P06276 | CHEMBL1914 | Butyrylcholinesterase, Human | 77 |
| ACES_RAT | P37136 | CHEMBL3199 | Acetylcholinesterase, Rat | 39 |
| ACES_BOVIN | P23795 | CHEMBL4768 | Acetylcholinesterase, Bovin | 37 |
| ACES_TORCA | P04058 | CHEMBL4780 | Acetylcholinesterase, Torca | 36 |
| Q9JKC1_RAT | Q9JKC1 | CHEMBL3403 | Butyrylcholinesterase, Rat | 10 |
| ACES_MOUSE | P21836 | CHEMBL3198 | Acetylcholinesterase, Mouse | 9 |
| Z104298 | Z104298 | CHEMBL1907604 | Glutamate NMDA Receptor; GRIN1/GRIN2A | 9 |
| ACM2_PIG | P06199 | CHEMBL4781 | Muscarinic Acetylcholine Receptor M2, Pig | 7 |
| Z104297 | Z104297 | CHEMBL1907603 | Glutamate NMDA Receptor; GRIN1/GRIN2B | 6 |
| CLAT_RAT | P32738 | CHEMBL3945 | Choline Acetylase, Rat | 4 |
| AGTRB_RAT | P29089 | CHEMBL263 | Angiotensin II Type 1b (AT-1b) Receptor, Rat | 3 |
| CHLE_MOUSE | Q03311 | CHEMBL2528 | Butyrylcholinesterase, Mouse | 3 |
| HRH3_HUMAN | Q9Y5N1 | CHEMBL264 | Histamine H3 Receptor, Human | 2 |
| KCNH2_HUMAN | Q12809 | CHEMBL240 | HERG, Human | 2 |
| ACHE_HUMAN | Q04844 | CHEMBL2484 | Acetylcholine Receptor Protein Epsilon Chain, Human | 1 |
| ACM1_MOUSE | P12657 | CHEMBL3733 | Muscarinic Acetylcholine Receptor M1, Mouse | 1 |
| ACM2_MOUSE | Q9ERZ4 | CHEMBL3197 | Muscarinic Acetylcholine Receptor M2, Mouse | 1 |
| ACM2_RAT | P10980 | CHEMBL309 | Muscarinic Acetylcholine Receptor M2, Rat | 1 |
| BACE1_HUMAN | P56817 | CHEMBL4822 | Beta-secretase 1, Human | 1 |
| HNMT_RAT | Q01984 | CHEMBL3241 | Histamine N-methyltransferase, Rat | 1 |
| LOX1_SOYBN | P08170 | CHEMBL4586 | Seed Lipoxygenase-1, Soybn | 1 |
| OPRD_RAT | P33533 | CHEMBL269 | Delta Opioid Receptor, Rat | 1 |
| OPRK_CAVPO | P41144 | CHEMBL3952 | Kappa Opioid Receptor, Guinea Pig | 1 |
| OPRM_RAT | P33535 | CHEMBL270 | Mu Opioid Receptor, Rat | 1 |
| PLCG1_BOVIN | P08487 | CHEMBL5566 | 1-phosphatidylinositol-4,5-bisphosphate Phosphodiesterase Gamma-1, Bovin | 1 |
| Z104302 | Z104302 | CHEMBL1907608 | Glutamate NMDA Receptor | 1 |
| Z104303 | Z104303 | CHEMBL1907609 | Muscarinic Acetylcholine Receptor | 1 |
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